geroprotector

Any compound that supports healthy aging, slows the biological aging process, or extends lifespan.

ChEBI ID: 176497

Members (175)

Member	Definition	Class
1-(2-(4-aminophenyl)ethyl)-4-(3-trifluoromethylphenyl)piperazine	A N-arylpiperazine that is piperazine substituted by 2-(4-aminophenyl)ethyl and 3-(trifluoromethyl)phenyl groups at positions 1 and 4, respectively. It is a selective 5-HT1A serotonin receptor agonist and 5-HT1D serotonin receptor antagonist.	LY-165163
1,2,3,4,6-pentakis-O-galloyl-beta-D-glucose	A galloyl-beta-D-glucose compound having five galloyl groups in the 1-, 2-, 3-, 4- and 6-positions.	1,2,3,4,6-pentakis-O-galloyl-beta-D-glucose
10-hydroxy-2-decenoic acid	An omega-hydroxy amino acid that is 2-decenoic acid in which one of the hydrogens attached to the terminal carbon is replaced by a hydroxy group and in which the C=C double bond has E configuration. It is a component of royal jelly.	(E)-10-hydroxydec-2-enoic acid
2-(1H-benzimidazol-2-yl)aniline	A member of the class of benzimidazoles that is 1H-benzimidazole substituted by a 2-aminophenyl group at position 2.	2-(1H-benzimidazol-2-yl)aniline
2-(2-hydroxyphenyl)benzothiazole	A member of the class of benzothiazoles that is 1,3-benzothiazole substituted by a 2-hydroxyphenyl group at position 2.	2-(1,3-benzothiazol-2-yl)phenol
2-(2'-hydroxyphenyl)benzoxazole	A member of the class of 1,3-benzoxazoles that is 1,3-benzoxazole substituted by a 2-hydroxyphenyl group at position 2.	2-(1,3-benzoxazol-2-yl)phenol
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-one	A chromone substituted with a phenyl group at position 8 and a morpholine group at position 2.	LY294002
2,4-dinitrophenol	A dinitrophenol having the nitro groups at the 2- and 4-positions.	2,4-dinitrophenol
3-(n,n-dimethylsulfonamido)-4-methyl-nitrobenzene	A C-nitro compound that is benzene substituted by N,N-dimethylaminosulfonyl, methyl and nitro groups at positions 1, 2 and 5, respectively. It is a phosphodiesterase inhibitor selective for the PDE7 subtype (Ki = 180 nM).	BRL-50481
3,3-diethyl-2-pyrrolidinone	A pyrrolidin-2-one substituted by two ethyl groups at position 3.	3,3-diethyl-2-pyrrolidinone
3,3',4,5'-tetrahydroxystilbene	A stilbenol that is trans-stilbene in which one of the phenyl groups is substituted by hydroxy groups at positions 3 and 4, while the other phenyl group is substituted by hydroxy groups at positions 3 and 5.	piceatannol
3,4-dichloroisocoumarin	A member of the class of isocoumarins that is isocoumarin substituted by chloro groups at positions 3 and 4. It is a serine protease inhibitor.	3,4-dichloroisocoumarin
3,8-dihydroxy-6h-dibenzo(b,d)pyran-6-one		Urolithin A
4-(1-((5-((2,6-dimethylphenoxy)methyl)-3-isoxazolyl)carbonyl)-4-piperidinyl)pyridine	An N-acylpiperidine obtained by formal condensation of the carboxy group of 5-[(2,6-dimethylphenoxy)methyl]-1,2-oxazole-3-carboxylic acid with the secondary amino group of 4-(pyridin-4-yl)piperidine.	dafadine A
4-hydroxyphenylethanol	A phenol substituted at position 4 by a 2-hydroxyethyl group.	2-(4-hydroxyphenyl)ethanol
4-phenyl-3-furoxancarbonitrile	A 1,2,5-oxadiazole substituted by an oxido, cyano and phenyl groups at positions 2, 3 and 4, respectively. It is a vasodilator and inhibitor of platelet aggregation.	4-phenyl-3-furoxancarbonitrile
4-phenylbutyric acid, sodium salt	The organic sodium salt of 4-phenylbutyric acid. A prodrug for phenylacetate, it is used to treat urea cycle disorders.	sodium phenylbutyrate
5-(4-phenylbutoxy)psoralen	A member of the class of psoralens that is psoralen substituted by a 4-phenylbutoxy group at position 5. It is a potent inhibitor of the voltage-gated potassium channel Kv1.3 (EC50 = 3 nM).	psora 4
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol	A carbotetracyclic compound that is 5,6,11,12-tetrahydrochrysene substituted by hydroxy groups at positions 2 and 8 and by ethyl groups at positions 5 and 11 (the 5R,11R-stereoisomer). It is an agonist of ER-alpha and antagonist of ER-beta receptors.	(R,R)-5,11-diethyl-5,6,11,12-tetrahydro-2,8-chrysenediol
acarbose	A tetrasaccharide derivative consisting of a dideoxy-4-{[4,5,6-trihydroxy-3-(hydroxymethyl)cyclohex-2-en-1-yl C7 cyclitol moiety [called valienol (or valienamine)] linked via nitrogen to isomaltotriose.	acarbose
acetaminophen	A member of the class of phenols that is 4-aminophenol in which one of the hydrogens attached to the amino group has been replaced by an acetyl group.	paracetamol
acetylcysteine	An N-acetyl-L-amino acid that is the N-acetylated derivative of the natural amino acid L-cysteine.	N-acetyl-L-cysteine
ag 1295		6,7-dimethyl-2-phenylquinoxaline
ag 1879	A member of the class of pyrazolopyrimidine that is pyrazolo[3,4-d]pyrimidin-4-amine bearing additional tert-butyl and 4-chlorophenyl substituents at positions 1 and 3 respectively. It is a potent ATP-competitive inhibitor of the Src family of protein tyrosine kinases.	PP2
ag-490	A monocarboxylic acid amide obtained by formal condensation of the carboxy group of (2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enoic acid with the amino group of benzylamine.	tyrphostin B42
alfatradiol	An estradiol that is estra-1,3,5(10)-triene substituted by hydroxy groups at positions 3 and 17 (the 17alpha stereoisomer).	17alpha-estradiol
amoxapine	A dibenzooxazepine compound having a chloro substituent at the 2-position and a piperazin-1-yl group at the 11-position.	amoxapine
amperozide	A member of the class of ureas that is urea in which three of the four hydrogens are replaced by ethyl and 4-[4,4-bis(4-fluorophenyl)butyl]piperazin-1-yl groups. An atypical antipsychotic which was in clinical development for the treatment of schizophrenia and substance-related disorders. It is a potent 5-HT2A antagonist and used in veterinary medicine because of its sedative effect on pigs.	amperozide
amperozide hydrochloride	The hydrochloride salt of amperozide.	amperozide hydrochloride
ascorbic acid	The L-enantiomer of ascorbic acid and conjugate acid of L-ascorbate.	L-ascorbic acid
aspirin	A member of the class of benzoic acids that is salicylic acid in which the hydrogen that is attached to the phenolic hydroxy group has been replaced by an acetoxy group. A non-steroidal anti-inflammatory drug with cyclooxygenase inhibitor activity.	acetylsalicylic acid
b 43	A member of the class of pyrrolopyrimidines that is 7H-pyrrolo[2,3-d]pyrimidine substituted by amino, 4-phenoxyphenyl, and cyclopentyl groups at positions 4, 5 and 7, respectively. It is a potent inhibitor of Lck that inhibits Lck (64-509) and LckCD isoforms (IC50 of less than 1 and 2 nM, respectively).	RK-24466
baicalein	A trihydroxyflavone with the hydroxy groups at positions C-5, -6 and -7.	baicalein
berberine		berberine
bezafibrate	A monocarboxylic acid amide obtained by the formal condensation of the carboxy group of 4-chlorobenzoic acid with the amino group of 2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic acid. Benafibrate is used for the treatment of hyperlipidaemia.	bezafibrate
brl 15572	An N-alkylpiperazine that is 1-(3-chlorophenyl)piperazine carrying a 3,3-diphenyl-2-hydroxyprop-1-yl group at position 4. A selective h5-HT1D antagonist, displaying 60-fold selectivity over h5-HT1B, and exhibiting little or no affinity for a range of other receptor types.	3-[4-(3-chlorophenyl)piperazin-1-yl]-1,1-diphenylpropan-2-ol
buformin	A member of the class of biguanides that is biguanide substituted by a butyl group at position 1. It is an antidiabetic drug with potential antitumor effect.	buformin
butein	A chalcone that is (E)-chalcone bearing four additional hydroxy substituents at positions 2', 3, 4 and 4'.	butein
butylated hydroxytoluene	A member of the class of phenols that is 4-methylphenol substituted by tert-butyl groups at positions 2 and 6.	2,6-di-tert-butyl-4-methylphenol
caffeic acid	The trans-isomer of caffeic acid.	trans-caffeic acid
caffeine	A trimethylxanthine in which the three methyl groups are located at positions 1, 3, and 7. A purine alkaloid that occurs naturally in tea and coffee.	caffeine
carbonyl cyanide m-chlorophenyl hydrazone	A member of the class of monochlorobenzenes that is benzene substituted by 2-(1,3-dinitrilopropan-2-ylidene)hydrazinyl and chloro groups at positions 1 and 3, respectively. It is a mitochondrial depolarizing agent that induces reactive oxygen species mediated cell death.	CCCP
carbonyl cyanide p-trifluoromethoxyphenylhydrazone	A hydrazone that is hydrazonomalononitrile in which one of the hydrazine hydrogens is substituted by a p-trifluoromethoxyphenyl group.	carbonyl cyanide p-trifluoromethoxyphenylhydrazone
carnosine	A dipeptide that is the N-(beta-alanyl) derivative of L-histidine.	carnosine zwitterion; carnosine
catechin	The monohydrate of (+)-catechin.	(+)-catechin monohydrate
celecoxib	A member of the class of pyrazoles that is 1H-pyrazole which is substituted at positions 1, 3 and 5 by 4-sulfamoylphenyl, trifluoromethyl and p-tolyl groups, respectively. A cyclooxygenase-2 inhibitor, it is used in the treatment of arthritis.	celecoxib
cgp 52411	Phthalimide substituted at the 4- and 5-positions by anilino groups.	4,5-dianilinophthalimide
chicoric acid		chicoric acid
chloramphenicol	An organochlorine compound that is dichloro-substituted acetamide containing a nitrobenzene ring, an amide bond and two alcohol functions.	chloramphenicol
cholecalciferol	A hydroxy seco-steroid that is (5Z,7E)-9,10-secocholesta-5,7,10(19)-triene in which the pro-S hydrogen at position 3 has been replaced by a hydroxy group. It is the inactive form of vitamin D3, being hydroxylated in the liver to calcidiol (25-hydroxyvitamin D3), which is then further hydroxylated in the kidney to give calcitriol (1,25-dihydroxyvitamin D3), the active hormone.	calciol
chromium tripicolinate		tris(picolinato)chromium
cinnarizine		cinnarizine
cis-flupenthixol dihydrochloride	The dihydrochloride salt of cis-flupenthixol.	cis-flupenthixol dihydrochloride
clofibrate	The ethyl ester of clofibric acid.	clofibrate
creatine	A glycine derivative having methyl and amidino groups attached to the nitrogen.	creatine zwitterion; creatine
curcumin	A beta-diketone that is methane in which two of the hydrogens are substituted by feruloyl groups. A natural dyestuff found in the root of Curcuma longa.	curcumin
cyclosporine	A cyclic nonribosomal peptide of eleven amino acids; an immunosuppressant drug widely used in post-allogeneic organ transplant to reduce the activity of the patient's immune system, and therefore the risk of organ rejection. Also causes reversible inhibition of immunocompetent lymphocytes in the G0- and G1-phase of the cell cycle.	cyclosporin A
cyproterone acetate	A steroid ester resulting from the formal condensation of the carboxy group of acetic acid with the 17-hydroxy group of cyproterone. It is an antiandrogenic drug which has recently been recognized to promote the occurrence and growth of intracranial meningiomas.	cyproterone acetate
cysteamine	An amine that consists of an ethane skeleton substituted with a thiol group at C-1 and an amino group at C-2.	cysteamine
danazol		danazol
dibromoacetic acid	A monocarboxylic acid that is acetic acid in which two of the methyl hydrogens are replaced by bromo groups.	dibromoacetic acid
didanosine	A purine 2',3'-dideoxyribonucleoside that is inosine in which the hydroxy groups at both the 2' and the 3' positions on the sugar moiety have been replaced by hydrogen. An antiviral drug, it is used as a medication to treat HIV/AIDS.	didanosine
dihydroergocristine monomesylate	The methanesulfonic acid salt of dihydroergocristine. It has been used as the for the symptomatic treatment of mental deterioration associated with cerebrovascular insufficiency and in peripheral vascular disease. It is also a component of ergoloid mesylate (codergocrine mesilate), a mixture of ergot alkaloid derivatives that is used as a vasodilator and has shown mild benefits in the treatment of vascular dementia.	dihydroergocristine mesylate
dimethyl sulfoxide	A 2-carbon sulfoxide in which the sulfur atom has two methyl substituents.	dimethyl sulfoxide
dimethylformamide	A member of the class of formamides that is formamide in which the amino hydrogens are replaced by methyl groups.	N,N-dimethylformamide
dimethylnitrosamine		N-nitrosodimethylamine
dipropylacetamide	A fatty amide derived from valproic acid.	valpromide
doxazosin mesylate		doxazosin mesylate
edetic acid		ethylenediaminetetraacetic acid
ellagic acid	An organic heterotetracyclic compound resulting from the formal dimerisation of gallic acid by oxidative aromatic coupling with intramolecular lactonisation of both carboxylic acid groups of the resulting biaryl. It is found in many fruits and vegetables, including raspberries, strawberries, cranberries, and pomegranates.	ellagic acid
enalapril	A dicarboxylic acid monoester that is ethyl 4-phenylbutanoate in which a hydrogen alpha to the carboxy group is substituted by the amino group of L-alanyl-L-proline (S-configuration).	enalapril
epigallocatechin gallate	A gallate ester obtained by the formal condensation of gallic acid with the (3R)-hydroxy group of (-)-epigallocatechin.	(-)-epigallocatechin 3-gallate
ethidium bromide	The organic bromide salt of ethidium.	ethidium bromide
ethosuximide	A dicarboximide that is pyrrolidine-2,5-dione in which the hydrogens at position 3 are substituted by one methyl and one ethyl group. An antiepileptic, it is used in the treatment of absence seizures and may be used for myoclonic seizures, but is ineffective against tonic-clonic seizures.	ethosuximide
ethoxyquin	A quinoline that is 1,2-dihydroquinoline bearing three methyl substituents at position 2, 2 and 4 as well as an ethoxy substituent at position 6.	ethoxyquin
everolimus	A macrocyclic lactone that is rapamycin in which the hydroxy group attached to the cyclohexyl moiety has been converted into the corresponding 2-hydroxyethyl ether. It is an immunosuppressant and antineoplastic agent.	everolimus
fasudil	An isoquinoline substituted by a (1,4-diazepan-1-yl)sulfonyl group at position 5. It is a Rho-kinase inhibitor and its hydrochloride hydrate form is approved for the treatment of cerebral vasospasm and cerebral ischemia.	fasudil
fenofibrate	A chlorobenzophenone that is (4-chlorophenyl)(phenyl)methanone substituted by a [2-methyl-1-oxo-1-(propan-2-yloxy)propan-2-yl]oxy group at position 1 on the phenyl ring.	fenofibrate
fisetin	A 7-hydroxyflavonol with additional hydroxy groups at positions 3, 3' and 4'.	fisetin
foscarnet	Phosphoric acid in which one of the hydroxy groups is replaced by a carboxylic acid group. It is used as the trisodium salt as an antiviral agent in the treatment of cytomegalovirus retinitis (CMV retinitis, an inflamation of the retina that can lead to blindness) and as an alternative to ganciclovir for AIDS patients who require concurrent antiretroviral therapy but are unable to tolerate ganciclovir due to haematological toxicity.	phosphonoformic acid
fullerene c60		C60 fullerene
fumaric acid	A butenedioic acid in which the C=C double bond has E geometry. It is an intermediate metabolite in the citric acid cycle.	fumaric acid
gallic acid	A trihydroxybenzoic acid in which the hydroxy groups are at positions 3, 4, and 5.	gallic acid
genistein	A 7-hydroxyisoflavone with additional hydroxy groups at positions 5 and 4'. It is a phytoestrogenic isoflavone with antioxidant properties.	genistein
glaucarubinone	A quassinoid with formula C25H34O10. It is a natural product isolated from several plant species and exhibits anti-cancer and anti-malarial properties.	glaucarubinone
glucosamine	A D-glucosamine whose structure comprises D-glucopyranose having an amino substituent at position 2.	2-amino-2-deoxy-D-glucopyranose
glycerol	A triol with a structure of propane substituted at positions 1, 2 and 3 by hydroxy groups.	glycerol
guanabenz acetate		Guanabenz acetate
guanfacine hydrochloride		Guanfacine hydrochloride
ibuprofen	A monocarboxylic acid that is propionic acid in which one of the hydrogens at position 2 is substituted by a 4-(2-methylpropyl)phenyl group.	ibuprofen
isoliquiritigenin	A member of the class of chalcones that is trans-chalcone hydroxylated at C-2', -4 and -4'.	isoliquiritigenin
juglone	A hydroxy-1,4-naphthoquinone that is 1,4-naphthoquinone in which the hydrogen at position 5 has been replaced by a hydroxy group. A plant-derived 1,4-naphthoquinone with confirmed antibacterial and antitumor activities.	juglone
kaempferol	A tetrahydroxyflavone in which the four hydroxy groups are located at positions 3, 5, 7 and 4'. Acting as an antioxidant by reducing oxidative stress, it is currently under consideration as a possible cancer treatment.	kaempferol
kanamycin sulfate		kanamycin A sulfate
kinetin	A member of the class of 6-aminopurines that is adenine carrying a (furan-2-ylmethyl) substituent at the exocyclic amino group.	kinetin
kn 93	A sulfonamide resulting from the formal condensation of p-methoxybenzenesulfonic acid with the anilino nitrogen of 2-(aminomethyl)-N-(2-hydroxyethyl)aniline in which the hydrogens of the primary amino group have been replaced by methyl and p-chlorocinnamyl groups. KN-93 is a selective inhibitor of Ca(2+)/calmodulin-dependent protein kinase II.	KN-93
l 744832	A secondary carboxamide resulting from the formal condensation of the carboxy group of 2-{[(2S,3S)-2-{[(2R)-2-amino-3-sulfanylpropyl]amino}-3-methylpentyl]oxy}-3-phenylpropanoic acid with the amino group of propan-2-yl (2S)-2-amino-4-(methylsulfonyl)butanoate. It is a farnesyltransferase inhibitor that exhibits anticancer properties.	L-744,832
lamotrigine	A member of the class of 1,2,4-triazines in which the triazene skeleton is substituted by amino groups at positions 3 and 5, and by a 2,3-dichlorophenyl group at position 6.	lamotrigine
latrepirdine		latrepirdine
lfm a13	An enamide obtained by formal condensation of the carboxy group of (2Z)-2-cyano-3-hydroxybut-2-enoic acid with the amino group of 2,5-dibromoaniline. It is a dual-function inhibitor of Bruton's tyrosine kinase (BTK) and Polo-like kinases (PLK) that exhibits anticancer properties.	LFM-A13
lithium chloride	A metal chloride salt with a Li(+) counterion.	lithium chloride
lithocholic acid	A monohydroxy-5beta-cholanic acid with a alpha-hydroxy substituent at position 3. It is a bile acid obtained from chenodeoxycholic acid by bacterial action.	lithocholic acid
lonidamine	A member of the class of indazoles that is 1H-indazole that is substituted at positions 1 and 3 by 2,4-dichlorobenzyl and carboxy groups, respectively.	lonidamine
loratadine	A benzocycloheptapyridine that is 6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridine substituted by a chloro group at position 8 and a 1-(ethoxycarbonyl)piperidin-4-ylidene group at position 11. It is a H1-receptor antagonist commonly employed in the treatment of allergic disorders.	loratadine
loxapine succinate		loxapine succinate
ly 367265	A fluoroindole that is 1H-indole in which the hydrogens at positions 3 and 6 are replaced by 1-[2-(2,2-dioxo-5,6-dihydro-4H-2lambda(6)-[1,2,5]thiadiazolo[4,3,2-ij]quinolin-1(2H)-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl and fluoro groups, respectively. It is an inhibitor of the 5-hydroxytryptamine transporter (Ki = 2.3 nM) and an antagonist of 5-hydroxytryptamine(2A) receptor (Ki = 0.81 nM).	LY-367,265
masoprocol	A tetrol that is butane which is substituted at positions 2 and 3 by 3,4-dihydroxybenzyl groups. Masoprocol, the meso-form found in the leaves of the creosote bush (Larrea divaricata), is a potent lipoxygenase inhibitor.	nordihydroguaiaretic acid
melatonin	A member of the class of acetamides that is acetamide in which one of the hydrogens attached to the nitrogen atom is replaced by a 2-(5-methoxy-1H-indol-3-yl)ethyl group. It is a hormone secreted by the pineal gland in humans.	melatonin
mercaptoethanol		mercaptoethanol
metergoline	An ergoline alkaloid that is the N-benzyloxycarbonyl derivative of lysergamine. A 5-HT2 antagonist. Also 5-HT1 antagonist and 5-HT1D ligand. Has moderate affinity for 5-HT6 and high affinity for 5-HT7.	metergoline
metformin	A member of the class of guanidines that is biguanide the carrying two methyl substituents at position 1.	metformin
methionine sulfoximine	A methionine sulfoximine in which the amino group has S-stereochemistry.	L-methionine sulfoximine zwitterion; L-methionine sulfoximine
methiothepin	A dibenzothiepine that is 10,11-dihydrodibenzo[b,f]thiepine bearing additional methylthio and 4-methylpiperazin-1-yl substituents at positions 8 and 10 respectively. Potent 5-HT2 antagonist, also active as 5-HT1 antagonist. Differentiates 5-HT1D sub-types. Also displays affinity for rodent 5-HT5B, 5-HT5A, 5-HT7 and 5-HT6 receptors (pK1 values are 6.6, 7.0, 8.4 and 8.7 respectively).	methiothepin
methyl 2,5-dihydroxycinnamate	A cinnamate ester that is the methyl ester of 2,5-dihydroxycinnamic acid.	2,5-dihydroxycinnamic acid methyl ester
methylergonovine maleate		Methylergonovine Maleate
metoprolol	A propanolamine that is 1-(propan-2-ylamino)propan-2-ol substituted by a 4-(2-methoxyethyl)phenoxy group at position 1.	metoprolol
mianserin	A dibenzoazepine (specifically 1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino[1,2-a]azepine) methyl-substituted on N-2. Closely related to (and now mostly superseded by) the tetracyclic antidepressant mirtazapinean, it is an atypical antidepressant used in the treatment of depression throughout Europe and elsewhere.	mianserin
mianserin hydrochloride	The hydrochloride salt of mianserin, a tetracyclic compound with antidepressant effects.	mianserin hydrochloride
morphine	A morphinane alkaloid that is a highly potent opiate analgesic psychoactive drug. Morphine acts directly on the central nervous system (CNS) to relieve pain but has a high potential for addiction, with tolerance and both physical and psychological dependence developing rapidly. Morphine is the most abundant opiate found in Papaver somniferum (the opium poppy).	morphine
myricetin	A hexahydroxyflavone that is flavone substituted by hydroxy groups at positions 3, 3', 4', 5, 5' and 7. It has been isolated from the leaves of Myrica rubra and other plants.	myricetin
n-(3-(aminomethyl)benzyl)acetamidine	An aralkylamine that is Nbenzylacetamidine substituted at position 3 on the benzene ring by an aminomethyl group. An inhibitor of nitric oxide synthase.	N-[3-(aminomethyl)benzyl]acetamidine
n-oleoylethanolamine	An N-(long-chain-acyl)ethanolamine that is the ethanolamide of oleic acid. The monounsaturated analogue of the endocannabinoid anandamide.	oleoyl ethanolamide
n,n'-dibenzhydrylethane-1,2-diamine dihydrochloride	A hydrochloride obtained by combining N,N'-bis(diphenylmethyl)ethane-1,2-diamine with two molar equivalent of hydrochloric acid.	AMN082 dihydrochloride
nad		NAD zwitterion
naphthazarin	A naphthoquinone that is 1,4-naphthoquinone in which the hydrogens at positions 5 and 8 are replaced by hydroxy groups.	naphthazarin
niacinamide	A pyridinecarboxamide that is pyridine in which the hydrogen at position 3 is replaced by a carboxamide group.	nicotinamide
nicardipine hydrochloride		nicardipine hydrochloride
nicotinamide-beta-riboside	A pyridine nucleoside consisting of nicotinamide with a beta-D-ribofuranosyl moiety at the 1-position.	N-ribosylnicotinamide
nitrendipine	A dihydropyridine that is 1,4-dihydropyridine substituted by methyl groups at positions 2 and 6, a 3-nitrophenyl group at position 4, a ethoxycarbonyl group at position 3 and a methoxycarbonyl group at position 5. It is a calcium-channel blocker used in the treatment of hypertension.	nitrendipine
nitroflurbiprofen	A carboxylic ester obtained by formal condensation of the carboxy group of flurbiprofen with the free hydroxy group of 4-(nitrooxy)butanol. It is a non-steroidal anti-inflammatory agent showing inhibitory effects against the cyclooxygenases COX1 and COX2.	nitroflurbiprofen
nortriptyline hydrochloride		Nortriptyline hydrochloride
nsc 664704	An indolobenzazepine that is paullone in which the hydrogen at position 9 is replaced by a bromo substituent. It is an ATP-competitive inhibitor of cyclin-dependent kinases (CDKs) and glycogen synthase kinase 3beta (GSK3beta).	kenpaullone
oxaloacetic acid	An oxodicarboxylic acid that is succinic acid bearing a single oxo group.	oxaloacetic acid
oxatomide	A member of the class of benzimidazoles that is 1,3-dihydro-2H-benzimidazol-2-one substituted by a 3-[4-(diphenylmethyl)piperazin-1-yl]propyl group at position 1. It is an anti-allergic drug.	oxatomide
oxoline	A member of the class of tetralins that is tetralin in which oxo groups replace the hydrogens at positions 1, 2, 3, and 4.	naphthalene-1,2,3,4-tetrone
pantothenic acid	A pantothenic acid having R-configuration.	(R)-pantothenic acid
paraquat	An organic cation that consists of 4,4'-bipyridine bearing two N-methyl substituents loctated at the 1- and 1'-positions.	paraquat
paxilline	An indole diterpene alkaloid with formula C27H33NO4 isolated from Penicillium paxilli. It is a potent inhibitor of large conductance Ca2(+)- and voltage-activated K(+) (BK)-type channels.	paxilline
pd 98059	A member of the class of monomethoxyflavones that is 3'-methoxyflavone bearing an additional amino substituent at position 2'.	2-(2-amino-3-methoxyphenyl)chromen-4-one
pergolide mesylate	A methanesulfonate salt obtained from pergolide by mixing eqimolar amount of pergolide and methanesulfonic acid. A dopamine D2 receptor agonist which also has D1 and D2 agonist properties, it is used in the management of Parkinson's disease, although it was withdrawn from the U.S. and Canadian markets in 2007 due to an increased risk of cardiac valve dysfunction.	pergolide mesylate
phenformin	A member of the class of biguanides that is biguanide in which one of the terminal nitrogen atoms is substituted by a 2-phenylethyl group. It was used as an anti-diabetic drug but was later withdrawn from the market due to potential risk of lactic acidosis.	phenformin
pioglitazone	A member of the class of thiazolidenediones that is 1,3-thiazolidine-2,4-dione substituted by a benzyl group at position 5 which in turn is substituted by a 2-(5-ethylpyridin-2-yl)ethoxy group at position 4 of the phenyl ring. It exhibits hypoglycemic activity.	pioglitazone
polydatin	A stilbenoid that is trans-resveratrol substituted at position 3 by a beta-D-glucosyl residue.	trans-piceid
promethazine hydrochloride	The hydrochloride salt of promethazine.	promethazine hydrochloride
pyrazolanthrone	A member of the class of anthrapyrazoles that is anthra[1,9-cd]pyrazole substituted at position 6 by an oxo group. An inhibitor of c-Jun N-terminal kinase.	anthra[1,9-cd]pyrazol-6(2H)-one
pyrrolidine dithiocarbamate	A member of the class of dithiocarbamic acids that is the N-dithiocarboxy derivative of pyrrolidine.	pyrrolidine dithiocarbamate
quercetin	A pentahydroxyflavone having the five hydroxy groups placed at the 3-, 3'-, 4'-, 5- and 7-positions. It is one of the most abundant flavonoids in edible vegetables, fruit and wine.	quercetin
quercetin 3-o-glucopyranoside	A quercetin O-glucoside that is quercetin with a beta-D-glucosyl residue attached at position 3. Isolated from Lepisorus contortus, it exhibits antineoplastic activityand has been found to decrease the rate of polymerization and sickling of red blood cells	quercetin 3-O-beta-D-glucopyranoside
resveratrol	A stilbenol that is stilbene in which the phenyl groups are substituted at positions 3, 5, and 4' by hydroxy groups.	resveratrol
rifampin	A member of the class of rifamycins that is a a semisynthetic antibiotic derived from Amycolatopsis rifamycinica (previously known as Amycolatopsis mediterranei and Streptomyces mediterranei).	rifampicin zwitterion; rifampicin
rosmarinic acid	A stereoisomer of rosmarinic acid having (R)-configuration.	(R)-rosmarinic acid
rtki cpd	A member of the class of quinazolines that is quinazoline substituted by methoxy groups at positions 6 and 7 and a (3-chlorophenyl)nitrilo group at position 4. It acts as an epidermal growth factor receptor antagonist.	tyrphostin AG 1478
sb 203580	A member of the class of imidazoles carrying 4-methylsulfinylphenyl, 4-pyridyl and 4-fluorophenyl substituents at positions 2, 4 and 5 respectively. An inhibitor of mitogen-activated protein kinase.	SB 203580
selegiline		(-)-selegiline
simvastatin	A member of the class of hexahydronaphthalenes that is lovastatin in which the 2-methylbutyrate ester moiety has been replaced by a 2,2-dimethylbutyrate ester group. It is used as a cholesterol-lowering and anti-cardiovascular disease drug.	simvastatin
sirolimus	A macrolide lactam isolated from Streptomyces hygroscopicus consisting of a 29-membered ring containing 4 trans double bonds, three of which are conjugated. It is an antibiotic, immunosupressive and antineoplastic agent.	sirolimus
sodium butyrate	An organic sodium salt resulting from the replacement of the proton from the carboxy group of butyric acid by a sodium ion.	sodium butyrate
spermidine	A triamine that is the 1,5,10-triaza derivative of decane.	spermidine
staurosporine		staurosporine
theanine	A N(5)-alkylglutamine where the alkyl group is ethyl. It has been isolated from green tea.	N(5)-ethyl-L-glutamine zwitterion; N(5)-ethyl-L-glutamine
thiazolidine-4-carboxylic acid, (r)-isomer	An optically active version of thioproline having L-configuration.	L-thioproline
thioctic acid	A heterocyclic thia fatty acid comprising pentanoic acid with a 1,2-dithiolan-3-yl group at the 5-position.	lipoic acid
thioflavin t	An organic chloride salt having 2-[4-(dimethylamino)phenyl]-3,6-dimethyl-1,3-benzothiazol-3-ium as the counterion. It is widely used to visualise and quantify the presence of amyloids, both in vitro and in vivo.	thioflavine T
thioridazine hydrochloride		thioridazine hydrochloride
trametinib	A pyridopyrimidine that is used (as its dimethyl sulfoxide addition compound) for the treatment of patients with unresectable or metastatic melanoma with BRAF V600E or V600K mutations, and who have not received prior BRAF inhibitor treatment.	trametinib
trehalose	A trehalose in which both glucose residues have alpha-configuration at the anomeric carbon.	alpha,alpha-trehalose
trichostatin a		trichostatin A
trimethadione	An oxazolidinone that is 1,3-oxazolidine-2,4-dione substituted by methyl groups at positions 3, 5 and 5. It is an antiepileptic agent.	trimethadione
tyrphostin a1		tyrphostin 1
tyrphostin a9		Malonoben
ursolic acid	A pentacyclic triterpenoid that is urs-12-en-28-oic acid substituted by a beta-hydroxy group at position 3.	ursolic acid
valproate sodium	The sodium salt of valproic acid.	sodium valproate
vincristine sulfate	An organic sulfate salt containing equimolar amounts of vincristine(2+) and sulfate. Used for the treatment of a variety of cancers.	vincristine sulfate
vinpocetine		Vinpocetine
wortmannin		wortmannin

Research

Studies (579,535)

Timeframe	Studies, Drugs with This Role(%)	All Drugs %
pre-1990	156,290 (26.97)	18.7374
1990's	78,260 (13.50)	18.2507
2000's	125,736 (21.70)	29.6817
2010's	162,726 (28.08)	24.3611
2020's	56,523 (9.75)	2.80

Study Types

Publication Type	Studies, Drugs with this Role (%)	All Drugs (%)
Trials	53,176 (8.14%)	5.53%
Reviews	46,242 (7.08%)	6.00%
Case Studies	26,584 (4.07%)	4.05%
Observational	2,121 (0.32%)	0.25%
Other	525,022 (80.38%)	84.16%

Protein Targets (2,073)

Potency Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1	Homo sapiens (human)	Potency	22.1127	1	59
15-lipoxygenase, partial	Homo sapiens (human)	Potency	15.0629	1	39
2,3-bisphosphoglycerate-independent phosphoglycerate mutase	Leishmania major strain Friedlin	Potency	29.6322	1	2
67.9K protein	Vaccinia virus	Potency	17.0516	2	48
acetylcholinesterase	Homo sapiens (human)	Potency	46.1465	4	51
acid sphingomyelinase	Homo sapiens (human)	Potency	91.1129	1	8
activating transcription factor 6	Homo sapiens (human)	Potency	29.6342	2	35
Adenosine receptor A1	Rattus norvegicus (Norway rat)	Potency	10.0000	1	1
aldehyde dehydrogenase 1 family, member A1	Homo sapiens (human)	Potency	24.7626	2	111
alpha-galactosidase	Homo sapiens (human)	Potency	37.9921	4	16
Alpha-synuclein	Homo sapiens (human)	Potency	11.5257	1	15
Amyloid-beta precursor protein	Homo sapiens (human)	Potency	20.0496	1	5
apical membrane antigen 1, AMA1	Plasmodium falciparum 3D7	Potency	20.5010	1	14
AR protein	Homo sapiens (human)	Potency	26.8373	12	397
aryl hydrocarbon receptor	Homo sapiens (human)	Potency	31.7592	3	61
arylsulfatase A	Homo sapiens (human)	Potency	9.4895	1	23
ATAD5 protein, partial	Homo sapiens (human)	Potency	15.2988	13	79
Ataxin-2	Homo sapiens (human)	Potency	23.8237	2	47
ATP-dependent phosphofructokinase	Trypanosoma brucei brucei TREU927	Potency	14.2404	5	39
ATPase family AAA domain-containing protein 5	Homo sapiens (human)	Potency	30.0903	2	40
atrial natriuretic peptide receptor 1 precursor	Homo sapiens (human)	Potency	18.4691	1	13
atrial natriuretic peptide receptor 2 precursor	Homo sapiens (human)	Potency	16.1047	1	9
beta-2 adrenergic receptor	Homo sapiens (human)	Potency	9.4360	2	2
Bloom syndrome protein isoform 1	Homo sapiens (human)	Potency	23.2198	2	98
BRCA1	Homo sapiens (human)	Potency	12.8250	1	7
bromodomain adjacent to zinc finger domain 2B	Homo sapiens (human)	Potency	41.6228	1	32
caspase 7, apoptosis-related cysteine protease	Homo sapiens (human)	Potency	48.4961	1	14
caspase-1 isoform alpha precursor	Homo sapiens (human)	Potency	15.6660	1	8
caspase-3	Cricetulus griseus (Chinese hamster)	Potency	60.4918	1	8
caspase-3	Homo sapiens (human)	Potency	48.4961	1	14
Caspase-7	Cricetulus griseus (Chinese hamster)	Potency	60.4918	1	8
Caspase-7	Homo sapiens (human)	Potency	10.2074	1	7
Cellular tumor antigen p53	Homo sapiens (human)	Potency	33.8775	3	96
cellular tumor antigen p53 isoform a	Homo sapiens (human)	Potency	14.4382	2	53
Chain A, 2-oxoglutarate Oxygenase	Homo sapiens (human)	Potency	19.8698	1	65
Chain A, ATP-DEPENDENT DNA HELICASE Q1	Homo sapiens (human)	Potency	9.7145	3	37
Chain A, Beta-lactamase	Escherichia coli K-12	Potency	44.5357	2	34
Chain A, Breast cancer type 1 susceptibility protein	Homo sapiens (human)	Potency	16.2952	2	8
Chain A, Cruzipain	Trypanosoma cruzi	Potency	25.0158	3	35
Chain A, Ferritin light chain	Equus caballus (horse)	Potency	29.3607	2	45
Chain A, HADH2 protein	Homo sapiens (human)	Potency	17.5664	2	66
Chain A, JmjC domain-containing histone demethylation protein 3A	Homo sapiens (human)	Potency	54.2204	1	27
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE	Homo sapiens (human)	Potency	270.4433	4	98
Chain A, PAPAIN	Carica papaya (papaya)	Potency	28.1838	1	1
Chain A, Putative fructose-1,6-bisphosphate aldolase	Giardia intestinalis	Potency	13.0689	2	33
Chain A, TYROSYL-DNA PHOSPHODIESTERASE	Homo sapiens (human)	Potency	18.8110	2	66
Chain B, HADH2 protein	Homo sapiens (human)	Potency	17.5664	2	66
chaperonin-containing TCP-1 beta subunit homolog	Homo sapiens (human)	Potency	57.9244	1	2
Cholecystokinin receptor type A	Rattus norvegicus (Norway rat)	Potency	710.0000	1	1
chromobox protein homolog 1	Homo sapiens (human)	Potency	42.7400	2	54
ClpP	Bacillus subtilis	Potency	19.4543	1	3
core-binding factor subunit beta isoform 2	Homo sapiens (human)	Potency	10.6863	3	8
CREB-binding protein	Homo sapiens (human)	Potency	17.0453	2	4
cytochrome P450 2C19 precursor	Homo sapiens (human)	Potency	12.5590	1	31
cytochrome P450 2C9 precursor	Homo sapiens (human)	Potency	15.7449	1	38
cytochrome P450 2C9, partial	Homo sapiens (human)	Potency	15.7655	1	20
cytochrome P450 2D6	Homo sapiens (human)	Potency	13.3556	1	29
cytochrome P450 2D6 isoform 1	Homo sapiens (human)	Potency	17.8775	1	34
cytochrome P450 3A4 isoform 1	Homo sapiens (human)	Potency	13.4494	2	152
cytochrome P450 family 3 subfamily A polypeptide 4	Homo sapiens (human)	Potency	8.7436	2	38
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a	Homo sapiens (human)	Potency	32.4156	1	48
D(1A) dopamine receptor	Homo sapiens (human)	Potency	4.8851	3	40
D(1A) dopamine receptor	Sus scrofa (pig)	Potency	13.9100	1	7
D(3) dopamine receptor isoform e	Homo sapiens (human)	Potency	0.0163	1	2
Disintegrin and metalloproteinase domain-containing protein 17	Homo sapiens (human)	Potency	13.7590	1	8
DNA dC->dU-editing enzyme APOBEC-3F isoform a	Homo sapiens (human)	Potency	29.8304	1	3
DNA dC->dU-editing enzyme APOBEC-3G isoform 1	Homo sapiens (human)	Potency	23.1805	2	7
DNA polymerase beta	Homo sapiens (human)	Potency	27.9540	1	20
DNA polymerase eta isoform 1	Homo sapiens (human)	Potency	22.1925	2	17
DNA polymerase III, partial	Bacillus subtilis	Potency	19.7373	1	3
DNA polymerase iota isoform a (long)	Homo sapiens (human)	Potency	43.9004	2	44
DNA polymerase kappa isoform 1	Homo sapiens (human)	Potency	18.1255	2	69
dopamine D1 receptor	Homo sapiens (human)	Potency	7.7177	1	3
dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	Potency	0.1000	1	1
endonuclease IV	Escherichia coli	Potency	12.8206	2	30
epidermal growth factor receptor isoform a precursor	Homo sapiens (human)	Potency	0.1996	4	4
estrogen nuclear receptor alpha	Homo sapiens (human)	Potency	29.6903	12	413
estrogen receptor 2 (ER beta)	Homo sapiens (human)	Potency	28.0189	3	67
estrogen-related nuclear receptor alpha	Homo sapiens (human)	Potency	26.3434	10	367
euchromatic histone-lysine N-methyltransferase 2	Homo sapiens (human)	Potency	18.0716	2	139
EWS/FLI fusion protein	Homo sapiens (human)	Potency	18.5727	4	122
eyes absent homolog 2 isoform a	Homo sapiens (human)	Potency	108.6544	1	2
farnesoid X nuclear receptor	Homo sapiens (human)	Potency	30.2774	5	73
Fatty-acid amide hydrolase 1	Rattus norvegicus (Norway rat)	Potency	19.9526	1	1
flap endonuclease 1	Homo sapiens (human)	Potency	19.0583	3	45
fructose-bisphosphate aldolase A	Oryctolagus cuniculus (rabbit)	Potency	41.5242	1	2
Fumarate hydratase	Homo sapiens (human)	Potency	26.5114	1	17
G	Vesicular stomatitis virus	Potency	15.7655	1	20
GABA theta subunit	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
galactokinase	Homo sapiens (human)	Potency	26.0642	2	2
GALC protein	Homo sapiens (human)	Potency	17.1782	1	3
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	Potency	13.7878	1	77
Gastrin/cholecystokinin type B receptor	Rattus norvegicus (Norway rat)	Potency	710.0000	1	1
geminin	Homo sapiens (human)	Potency	14.1116	5	140
GLI family zinc finger 3	Homo sapiens (human)	Potency	21.9531	3	132
glp-1 receptor, partial	Homo sapiens (human)	Potency	13.3430	2	23
GLS protein	Homo sapiens (human)	Potency	12.9969	2	45
glucocerebrosidase	Homo sapiens (human)	Potency	20.1704	6	45
glucocorticoid receptor [Homo sapiens]	Homo sapiens (human)	Potency	24.3742	5	124
glucokinase regulatory protein	Homo sapiens (human)	Potency	28.9342	1	2
Glutamate receptor 1	Rattus norvegicus (Norway rat)	Potency	6.9037	1	8
Glutamate receptor 2	Rattus norvegicus (Norway rat)	Potency	30.8670	2	38
Glutamate receptor 3	Rattus norvegicus (Norway rat)	Potency	6.9037	1	8
Glutamate receptor 4	Rattus norvegicus (Norway rat)	Potency	6.9037	1	8
glyceraldehyde-3-phosphate dehydrogenase isoform 1	Homo sapiens (human)	Potency	52.2758	1	2
Glycoprotein hormones alpha chain	Homo sapiens (human)	Potency	6.7294	1	2
GTP-binding nuclear protein Ran isoform 1	Homo sapiens (human)	Potency	22.9516	1	8
Guanine nucleotide-binding protein G	Homo sapiens (human)	Potency	34.3829	2	9
guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1	Homo sapiens (human)	Potency	16.5563	1	6
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)	Homo sapiens (human)	Potency	21.1388	2	21
heat shock protein beta-1	Homo sapiens (human)	Potency	42.9042	2	43
hemoglobin subunit beta	Homo sapiens (human)	Potency	28.2641	2	4
hexokinase-4 isoform 1	Homo sapiens (human)	Potency	28.9342	1	2
Histamine H2 receptor	Cavia porcellus (domestic guinea pig)	Potency	14.6300	2	204
histone acetyltransferase KAT2A isoform 1	Homo sapiens (human)	Potency	23.0434	1	26
histone deacetylase 9 isoform 3	Homo sapiens (human)	Potency	26.6394	2	25
Histone H2A.x	Cricetulus griseus (Chinese hamster)	Potency	64.4240	2	51
histone-lysine N-methyltransferase 2A isoform 2 precursor	Homo sapiens (human)	Potency	40.8152	1	14
HLA class I histocompatibility antigen, B alpha chain	Homo sapiens (human)	Potency	15.7655	1	20
huntingtin isoform 2	Homo sapiens (human)	Potency	18.3915	3	10
hypothetical protein, conserved	Trypanosoma brucei	Potency	23.9641	4	15
hypoxia-inducible factor 1 alpha subunit	Homo sapiens (human)	Potency	38.7935	2	40
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)	Homo sapiens (human)	Potency	13.0751	3	62
IDH1	Homo sapiens (human)	Potency	15.5710	1	29
importin subunit beta-1 isoform 1	Homo sapiens (human)	Potency	47.2153	2	16
Inositol hexakisphosphate kinase 1	Homo sapiens (human)	Potency	15.7655	1	40
Inositol monophosphatase 1	Rattus norvegicus (Norway rat)	Potency	49.3301	4	34
Integrin alpha-IIb	Homo sapiens (human)	Potency	15.1188	1	26
Integrin beta-3	Homo sapiens (human)	Potency	15.1188	1	26
Interferon beta	Homo sapiens (human)	Potency	15.7130	3	63
interleukin 8	Homo sapiens (human)	Potency	71.0705	1	11
isocitrate dehydrogenase 1, partial	Homo sapiens (human)	Potency	50.1187	1	3
lamin isoform A-delta10	Homo sapiens (human)	Potency	11.7320	2	88
lethal factor (plasmid)	Bacillus anthracis str. A2012	Potency	11.2500	1	36
lethal(3)malignant brain tumor-like protein 1 isoform I	Homo sapiens (human)	Potency	9.6729	2	7
Luciferase	Photinus pyralis (common eastern firefly)	Potency	30.4732	4	52
luciferase	Photuris pensylvanica (Pennsylania firefly)	Potency	14.2191	1	2
lysosomal alpha-glucosidase preproprotein	Homo sapiens (human)	Potency	22.2013	5	23
M-phase phosphoprotein 8	Homo sapiens (human)	Potency	32.2546	1	47
Microtubule-associated protein tau	Homo sapiens (human)	Potency	16.6416	2	147
mitogen-activated protein kinase 1	Homo sapiens (human)	Potency	20.2710	4	58
muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	Potency	7.6779	2	47
muscleblind-like protein 1 isoform 1	Homo sapiens (human)	Potency	23.2153	3	19
Neuronal acetylcholine receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	26.8238	1	5
Neuronal acetylcholine receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	26.8238	1	5
neuropeptide S receptor isoform A	Homo sapiens (human)	Potency	12.0896	5	37
NFKB1 protein, partial	Homo sapiens (human)	Potency	6.0766	2	44
nonstructural protein 1	Influenza A virus (A/WSN/1933(H1N1))	Potency	17.2810	1	26
NPC intracellular cholesterol transporter 1 precursor	Homo sapiens (human)	Potency	29.8139	1	16
Nrf2	Homo sapiens (human)	Potency	21.7152	2	9
nuclear factor erythroid 2-related factor 2 isoform 1	Homo sapiens (human)	Potency	28.8715	4	154
nuclear factor erythroid 2-related factor 2 isoform 2	Homo sapiens (human)	Potency	18.3585	2	28
nuclear factor NF-kappa-B p105 subunit isoform 1	Homo sapiens (human)	Potency	34.9731	1	7
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a	Homo sapiens (human)	Potency	35.8133	2	32
Nuclear receptor ROR-gamma	Homo sapiens (human)	Potency	37.4099	1	15
nuclear receptor ROR-gamma isoform 1	Mus musculus (house mouse)	Potency	17.8457	4	79
nuclear receptor subfamily 1, group I, member 2	Rattus norvegicus (Norway rat)	Potency	12.7219	1	4
nuclear receptor subfamily 1, group I, member 3	Homo sapiens (human)	Potency	32.2263	3	101
Ornithine decarboxylase	Rattus norvegicus (Norway rat)	Potency	8.8323	1	5
P53	Homo sapiens (human)	Potency	20.8248	1	7
parathyroid hormone/parathyroid hormone-related peptide receptor precursor	Homo sapiens (human)	Potency	53.4323	1	18
Parkin	Homo sapiens (human)	Potency	18.1055	3	24
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1	Homo sapiens (human)	Potency	39.8069	2	27
peripheral myelin protein 22	Rattus norvegicus (Norway rat)	Potency	15.5415	2	25
peripheral myelin protein 22 isoform 1	Homo sapiens (human)	Potency	51.9697	1	44
peroxisome proliferator activated receptor gamma	Homo sapiens (human)	Potency	29.7902	5	111
Peroxisome proliferator-activated receptor alpha	Homo sapiens (human)	Potency	39.8107	1	1
peroxisome proliferator-activated receptor delta	Homo sapiens (human)	Potency	33.4402	5	91
phosphoglycerate kinase	Trypanosoma brucei brucei TREU927	Potency	8.7081	3	7
phosphopantetheinyl transferase	Bacillus subtilis	Potency	47.0928	3	57
PINK1	Homo sapiens (human)	Potency	32.1368	1	6
plasminogen precursor	Mus musculus (house mouse)	Potency	8.4490	2	15
Platelet-activating factor receptor	Homo sapiens (human)	Potency	25.6841	1	4
polyprotein	Zika virus	Potency	26.5114	1	17
polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	Potency	11.1713	1	12
Polyunsaturated fatty acid lipoxygenase ALOX15B	Homo sapiens (human)	Potency	13.2177	1	45
potassium voltage-gated channel subfamily H member 2 isoform d	Homo sapiens (human)	Potency	12.6391	1	52
PPM1D protein	Homo sapiens (human)	Potency	14.1958	1	24
pregnane X nuclear receptor	Homo sapiens (human)	Potency	31.8924	3	67
pregnane X receptor	Rattus norvegicus (Norway rat)	Potency	45.2385	1	11
progesterone receptor	Homo sapiens (human)	Potency	23.6844	3	69
putative alpha-glucosidase	Oryza sativa Japonica Group (Japanese rice)	Potency	39.8107	1	1
pyruvate kinase	Leishmania mexicana mexicana	Potency	9.2146	2	10
pyruvate kinase PKM isoform a	Homo sapiens (human)	Potency	11.0550	2	6
pyruvate kinase PKM isoform b	Homo sapiens (human)	Potency	8.8323	2	10
RAF proto-oncogene serine/threonine-protein kinase isoform b	Homo sapiens (human)	Potency	12.0891	1	3
Rap guanine nucleotide exchange factor 3	Homo sapiens (human)	Potency	31.5636	2	8
Rap guanine nucleotide exchange factor 4	Homo sapiens (human)	Potency	42.7410	1	9
RAR-related orphan receptor gamma	Mus musculus (house mouse)	Potency	25.3740	2	111
ras-related protein Rab-9A	Homo sapiens (human)	Potency	51.1270	1	20
regulator of G-protein signaling 4	Homo sapiens (human)	Potency	19.5852	1	37
retinoic acid nuclear receptor alpha variant 1	Homo sapiens (human)	Potency	34.6361	3	147
retinoid X nuclear receptor alpha	Homo sapiens (human)	Potency	192.7276	4	117
RGS12	Homo sapiens (human)	Potency	16.5563	1	6
runt-related transcription factor 1 isoform AML1b	Homo sapiens (human)	Potency	10.6863	3	8
serine-protein kinase ATM isoform a	Homo sapiens (human)	Potency	32.3105	1	2
serine/threonine-protein kinase mTOR isoform 1	Homo sapiens (human)	Potency	18.1002	4	38
serine/threonine-protein kinase PLK1	Homo sapiens (human)	Potency	16.0076	1	6
signal transducer and activator of transcription 6, interleukin-4 induced	Homo sapiens (human)	Potency	19.0145	3	5
Single-stranded DNA cytosine deaminase	Homo sapiens (human)	Potency	72.9542	2	4
SMAD family member 2	Homo sapiens (human)	Potency	29.6424	3	44
SMAD family member 3	Homo sapiens (human)	Potency	29.6424	3	44
Smad3	Homo sapiens (human)	Potency	16.4877	3	28
snurportin-1	Homo sapiens (human)	Potency	47.2153	2	16
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	Potency	21.7202	2	18
survival motor neuron protein isoform d	Homo sapiens (human)	Potency	15.6984	2	68
TAR DNA-binding protein 43	Homo sapiens (human)	Potency	16.3251	1	19
TDP1 protein	Homo sapiens (human)	Potency	17.6883	2	287
thioredoxin glutathione reductase	Schistosoma mansoni	Potency	24.2654	1	12
thioredoxin reductase	Rattus norvegicus (Norway rat)	Potency	25.1485	4	113
Thrombopoietin	Homo sapiens (human)	Potency	9.0038	2	40
thyroid hormone receptor beta isoform 2	Rattus norvegicus (Norway rat)	Potency	28.3265	3	153
thyroid hormone receptor beta isoform a	Homo sapiens (human)	Potency	30.2269	4	44
thyroid stimulating hormone receptor	Homo sapiens (human)	Potency	25.6785	6	139
thyrotropin-releasing hormone receptor	Homo sapiens (human)	Potency	30.5358	2	10
transcriptional regulator ERG isoform 3	Homo sapiens (human)	Potency	17.4218	2	8
transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	Potency	20.2698	1	4
tumor necrosis factor	Homo sapiens (human)	Potency	37.5780	1	1
tumor susceptibility gene 101 protein	Homo sapiens (human)	Potency	21.6747	1	3
Type-1A angiotensin II receptor	Rattus norvegicus (Norway rat)	Potency	0.1000	1	1
Type-1B angiotensin II receptor	Rattus norvegicus (Norway rat)	Potency	0.1000	1	1
Type-2 angiotensin II receptor	Rattus norvegicus (Norway rat)	Potency	0.1000	1	1
tyrosine-protein kinase Yes	Homo sapiens (human)	Potency	14.6991	1	4
ubiquitin carboxyl-terminal hydrolase 2 isoform a	Homo sapiens (human)	Potency	13.0783	3	13
urokinase plasminogen activator surface receptor precursor	Mus musculus (house mouse)	Potency	8.4490	2	15
urokinase-type plasminogen activator precursor	Mus musculus (house mouse)	Potency	8.4490	2	15
USP1 protein, partial	Homo sapiens (human)	Potency	47.1765	3	51
v-jun sarcoma virus 17 oncogene homolog (avian)	Homo sapiens (human)	Potency	21.1302	2	74
vitamin D (1,25- dihydroxyvitamin D3) receptor	Homo sapiens (human)	Potency	25.0615	5	84
vitamin D3 receptor isoform VDRA	Homo sapiens (human)	Potency	42.7764	5	58
Voltage-dependent calcium channel gamma-2 subunit	Mus musculus (house mouse)	Potency	37.2572	1	30
Vpr	Human immunodeficiency virus 1	Potency	12.7087	1	6
WRN	Homo sapiens (human)	Potency	15.2443	1	6

Inhibition Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial	Homo sapiens (human)	IC50	0.0005	2	2
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a	Homo sapiens (human)	IC50	9.6995	2	2
1-deoxy-D-xylulose 5-phosphate reductoisomerase	Escherichia coli K-12	IC50	2.2750	1	4
10 kDa chaperonin	Escherichia coli	IC50	36.4450	4	12
10 kDa heat shock protein, mitochondrial	Homo sapiens (human)	IC50	38.6000	2	6
14-3-3 protein gamma	Homo sapiens (human)	IC50	50.0000	1	1
17-beta-hydroxysteroid dehydrogenase type 1	Homo sapiens (human)	IC50	2.8975	2	4
17-beta-hydroxysteroid dehydrogenase type 2	Homo sapiens (human)	IC50	4.5718	2	11
2-5A-dependent ribonuclease	Homo sapiens (human)	IC50	264.0000	1	1
3-hydroxy-3-methylglutaryl-coenzyme A reductase	Homo sapiens (human)	IC50	0.7843	8	8
3-hydroxy-3-methylglutaryl-coenzyme A reductase	Schizosaccharomyces pombe 972h-	IC50	95.2000	1	1
3-hydroxy-3-methylglutaryl-coenzyme A reductase	Homo sapiens (human)	Ki	34.0013	2	2
3-hydroxy-3-methylglutaryl-coenzyme A reductase	Rattus norvegicus (Norway rat)	IC50	0.0112	2	2
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ	Yersinia pseudotuberculosis YPIII	IC50	5.3500	1	2
3-oxoacyl-[acyl-carrier-protein] reductase	Plasmodium falciparum 3D7	IC50	0.3200	1	1
3-oxoacyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	5.5600	1	5
3-phosphoinositide-dependent protein kinase 1	Homo sapiens (human)	IC50	19.2043	5	5
30S ribosomal protein S1	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S10	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S11	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S12	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S13	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S14	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S15	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S16	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S17	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S18	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S19	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S2	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S20	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S21	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S3	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S4	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S5	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S6	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S7	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S8	Escherichia coli K-12	IC50	0.4300	1	1
30S ribosomal protein S9	Escherichia coli K-12	IC50	0.4300	1	1
4-aminobutyrate aminotransferase, mitochondrial	Homo sapiens (human)	IC50	12,800.0000	1	1
4-aminobutyrate aminotransferase, mitochondrial	Rattus norvegicus (Norway rat)	IC50	1.7500	1	4
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT6	Homo sapiens (human)	IC50	38.3662	1	13
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	IC50	0.2668	3	3
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	IC50	1.5831	4	7
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	Ki	0.1483	10	10
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	Ki	1.6026	4	8
5-hydroxytryptamine receptor 1B	Rattus norvegicus (Norway rat)	IC50	1.3924	2	5
5-hydroxytryptamine receptor 1B	Rattus norvegicus (Norway rat)	Ki	0.8384	4	9
5-hydroxytryptamine receptor 1D	Homo sapiens (human)	IC50	0.3802	2	2
5-hydroxytryptamine receptor 1D	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 1D	Rattus norvegicus (Norway rat)	Ki	0.5667	2	3
5-hydroxytryptamine receptor 1F	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 1F	Rattus norvegicus (Norway rat)	Ki	0.5667	2	3
5-hydroxytryptamine receptor 2A	Homo sapiens (human)	IC50	2.2403	3	11
5-hydroxytryptamine receptor 2A	Rattus norvegicus (Norway rat)	IC50	8.0000	2	3
5-hydroxytryptamine receptor 2A	Homo sapiens (human)	Ki	0.2765	16	26
5-hydroxytryptamine receptor 2A	Rattus norvegicus (Norway rat)	Ki	0.4371	7	9
5-hydroxytryptamine receptor 2B	Homo sapiens (human)	IC50	5.3868	1	7
5-hydroxytryptamine receptor 2B	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 2B	Homo sapiens (human)	Ki	3.4280	1	7
5-hydroxytryptamine receptor 2B	Rattus norvegicus (Norway rat)	Ki	0.0028	3	5
5-hydroxytryptamine receptor 2C	Homo sapiens (human)	IC50	2.3169	2	8
5-hydroxytryptamine receptor 2C	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 2C	Homo sapiens (human)	Ki	0.5818	8	17
5-hydroxytryptamine receptor 2C	Rattus norvegicus (Norway rat)	Ki	0.0025	4	6
5-hydroxytryptamine receptor 3A	Cavia porcellus (domestic guinea pig)	IC50	7.6900	1	1
5-hydroxytryptamine receptor 3A	Homo sapiens (human)	IC50	1.4125	2	2
5-hydroxytryptamine receptor 3A	Mus musculus (house mouse)	IC50	1.4125	1	1
5-hydroxytryptamine receptor 3A	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 3A	Mus musculus (house mouse)	Ki	0.2520	1	1
5-hydroxytryptamine receptor 3A	Rattus norvegicus (Norway rat)	Ki	0.0700	1	1
5-hydroxytryptamine receptor 3B	Homo sapiens (human)	IC50	1.4125	2	2
5-hydroxytryptamine receptor 3B	Mus musculus (house mouse)	IC50	1.4125	1	1
5-hydroxytryptamine receptor 3B	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 3B	Mus musculus (house mouse)	Ki	0.2520	1	1
5-hydroxytryptamine receptor 3B	Rattus norvegicus (Norway rat)	Ki	0.0700	1	1
5-hydroxytryptamine receptor 3C	Homo sapiens (human)	IC50	1.4125	2	2
5-hydroxytryptamine receptor 3D	Homo sapiens (human)	IC50	1.4125	2	2
5-hydroxytryptamine receptor 3E	Homo sapiens (human)	IC50	1.4125	2	2
5-hydroxytryptamine receptor 4	Cavia porcellus (domestic guinea pig)	IC50	2.6468	1	7
5-hydroxytryptamine receptor 4	Cavia porcellus (domestic guinea pig)	Ki	1.3858	1	7
5-hydroxytryptamine receptor 4	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 5A	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 5A	Homo sapiens (human)	Ki	0.0334	4	4
5-hydroxytryptamine receptor 5B	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 6	Homo sapiens (human)	IC50	0.2767	9	12
5-hydroxytryptamine receptor 6	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 6	Homo sapiens (human)	Ki	0.0165	16	20
5-hydroxytryptamine receptor 6	Rattus norvegicus (Norway rat)	Ki	0.0807	4	4
5-hydroxytryptamine receptor 7	Cavia porcellus (domestic guinea pig)	IC50	28.0000	1	2
5-hydroxytryptamine receptor 7	Homo sapiens (human)	IC50	50.0218	7	7
5-hydroxytryptamine receptor 7	Homo sapiens (human)	Ki	0.4572	17	19
5-hydroxytryptamine receptor 7	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
5-hydroxytryptamine receptor 7	Rattus norvegicus (Norway rat)	Ki	0.0434	2	4
5-lipoxygenase	Bos taurus (cattle)	IC50	5.3500	3	4
5'-AMP-activated protein kinase subunit beta-1	Homo sapiens (human)	IC50	3.0363	1	5
5'-AMP-activated protein kinase subunit gamma-1	Homo sapiens (human)	IC50	3.0363	1	5
5'-nucleotidase	Homo sapiens (human)	IC50	6.1950	1	2
5'-nucleotidase	Mus musculus (house mouse)	IC50	50.0200	1	2
5'-nucleotidase	Rattus norvegicus (Norway rat)	Ki	0.0453	1	1
50S ribosomal protein L1	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L10	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L11	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L13	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L14	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L15	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L16	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L17	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L18	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L19	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L2	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L20	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L21	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L22	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L23	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L24	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L25	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L27	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L28	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L29	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L3	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L30	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L31	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L31 type B	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L32	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L33	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L34	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L35	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L36	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L36 2	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L4	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L5	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L6	Escherichia coli K-12	IC50	0.4300	1	1
50S ribosomal protein L7/L12	Escherichia coli K-12	IC50	0.4300	1	1
6-phosphogluconate dehydrogenase, decarboxylating	Homo sapiens (human)	IC50	0.7200	1	1
60 kDa chaperonin	Escherichia coli K-12	IC50	250.0000	1	5
60 kDa chaperonin	Escherichia coli	IC50	36.4450	4	12
60 kDa heat shock protein, mitochondrial	Homo sapiens (human)	IC50	38.6000	2	6
7,8-dihydro-8-oxoguanine triphosphatase	Homo sapiens (human)	IC50	24.5000	1	2
72 kDa type IV collagenase	Homo sapiens (human)	IC50	30.2985	5	17
90-kda heat shock protein beta HSP90 beta, partial	Homo sapiens (human)	IC50	27.5411	2	3
acetyl-CoA acetyltransferase/HMG-CoA reductase	Enterococcus faecalis	IC50	1,265.3900	1	1
Acetylcholinesterase	Electrophorus electricus (electric eel)	IC50	128.5040	7	7
Acetylcholinesterase	Homo sapiens (human)	IC50	564.0837	12	15
Acetylcholinesterase	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Acetylcholinesterase	Electrophorus electricus (electric eel)	Ki	109.0000	1	1
Acetylcholinesterase	Homo sapiens (human)	Ki	67.2750	1	4
Acetylcholinesterase	Bos taurus (cattle)	IC50	0.1000	2	3
Acid ceramidase	Homo sapiens (human)	IC50	500.0000	1	1
Acid ceramidase	Homo sapiens (human)	Ki	500.0000	1	1
Acid-sensing ion channel 1	Rattus norvegicus (Norway rat)	IC50	288.0192	5	9
Acid-sensing ion channel 3	Rattus norvegicus (Norway rat)	IC50	512.8610	1	1
Acidic mammalian chitinase	Homo sapiens (human)	IC50	1,000.0000	1	1
Acidic phospholipase A2 EC-I	Echis carinatus (saw-scaled viper)	IC50	2.3000	1	1
Activated CDC42 kinase 1	Homo sapiens (human)	IC50	0.0298	2	2
Activin receptor type-1	Homo sapiens (human)	IC50	4.1977	2	6
Activin receptor type-1B	Homo sapiens (human)	IC50	9.1180	1	1
Acyl-CoA desaturase 1	Mus musculus (house mouse)	IC50	3.4000	1	1
Acyl-CoA desaturase 1	Rattus norvegicus (Norway rat)	Ki	0.2990	1	1
Adenosine receptor A1	Bos taurus (cattle)	IC50	0.1900	1	1
Adenosine receptor A1	Homo sapiens (human)	IC50	11.4270	1	2
Adenosine receptor A1	Rattus norvegicus (Norway rat)	IC50	696.7380	7	9
Adenosine receptor A1	Sus scrofa (pig)	IC50	0.2000	1	1
Adenosine receptor A1	Cavia porcellus (domestic guinea pig)	Ki	100.0000	5	5
Adenosine receptor A1	Homo sapiens (human)	Ki	32.0489	16	17
Adenosine receptor A1	Rattus norvegicus (Norway rat)	Ki	28.7349	35	47
Adenosine receptor A2a	Homo sapiens (human)	IC50	14.6607	1	3
Adenosine receptor A2a	Rattus norvegicus (Norway rat)	IC50	906.4286	2	7
Adenosine receptor A2a	Cavia porcellus (domestic guinea pig)	Ki	50.0000	3	3
Adenosine receptor A2a	Homo sapiens (human)	Ki	19.2976	21	23
Adenosine receptor A2a	Rattus norvegicus (Norway rat)	Ki	114.9027	30	43
Adenosine receptor A2b	Rattus norvegicus (Norway rat)	IC50	63.0000	1	5
Adenosine receptor A2b	Homo sapiens (human)	Ki	26.7211	19	19
Adenosine receptor A2b	Mus musculus (house mouse)	Ki	23.0000	1	1
Adenosine receptor A2b	Rattus norvegicus (Norway rat)	Ki	30.7438	16	23
Adenosine receptor A3	Homo sapiens (human)	IC50	13.8277	1	3
Adenosine receptor A3	Homo sapiens (human)	Ki	28.3205	15	17
Adenosine receptor A3	Rattus norvegicus (Norway rat)	Ki	56.6667	6	6
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1	Homo sapiens (human)	IC50	54.2333	1	3
Albumin	Bos taurus (cattle)	IC50	79.1900	2	2
Albumin	Homo sapiens (human)	Ki	165,959,000,000.0000	1	1
Aldehyde oxidase	Homo sapiens (human)	IC50	0.1149	2	3
Aldehyde oxidase 1	Cavia porcellus (domestic guinea pig)	Ki	4.5300	1	1
Aldo-keto reductase family 1 member A1	Rattus norvegicus (Norway rat)	IC50	2.3200	1	1
Aldo-keto reductase family 1 member A1	Sus scrofa (pig)	IC50	63.7000	2	2
Aldo-keto reductase family 1 member B1	Bos taurus (cattle)	IC50	17.7540	5	5
Aldo-keto reductase family 1 member B1	Homo sapiens (human)	IC50	10.2810	9	15
Aldo-keto reductase family 1 member B1	Rattus norvegicus (Norway rat)	IC50	33.1393	9	17
Aldo-keto reductase family 1 member B1	Sus scrofa (pig)	IC50	33.0500	1	2
Aldo-keto reductase family 1 member B1	Homo sapiens (human)	Ki	25.5000	1	1
Aldo-keto reductase family 1 member B1	Rattus norvegicus (Norway rat)	Ki	5.3534	1	7
Aldo-keto reductase family 1 member B10	Homo sapiens (human)	IC50	47.0000	2	2
Aldo-keto reductase family 1 member B10	Homo sapiens (human)	Ki	3.3200	5	5
Aldo-keto reductase family 1 member C2	Homo sapiens (human)	IC50	6.7100	1	1
Aldo-keto reductase family 1 member C21	Mus musculus (house mouse)	IC50	9.6000	1	2
Aldo-keto reductase family 1 member C21	Mus musculus (house mouse)	Ki	11.0000	1	1
Aldo-keto reductase family 1 member C3	Homo sapiens (human)	IC50	13.2450	4	4
ALK tyrosine kinase receptor	Homo sapiens (human)	IC50	2.2840	18	19
alkaline phosphatase, germ cell type preproprotein	Homo sapiens (human)	IC50	100.0000	1	4
alkaline phosphatase, intestinal	Homo sapiens (human)	IC50	53.5525	2	4
alkaline phosphatase, tissue-nonspecific isozyme isoform 1 preproprotein	Homo sapiens (human)	IC50	46.0750	1	4
Alpha-(1,3)-fucosyltransferase 7	Homo sapiens (human)	IC50	38.3662	1	13
Alpha-1A adrenergic receptor	Bos taurus (cattle)	IC50	0.1087	3	3
Alpha-1A adrenergic receptor	Homo sapiens (human)	IC50	0.4074	2	2
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	5.7868	8	10
Alpha-1A adrenergic receptor	Homo sapiens (human)	Ki	0.0603	1	1
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	2.9691	5	8
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	13.7667	7	10
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	2.9691	5	8
Alpha-1D adrenergic receptor	Homo sapiens (human)	IC50	0.3399	1	5
Alpha-1D adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	3.2768	5	5
Alpha-1D adrenergic receptor	Homo sapiens (human)	Ki	0.1669	1	5
Alpha-1D adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	0.0609	4	5
Alpha-2A adrenergic receptor	Bos taurus (cattle)	IC50	0.1087	3	3
Alpha-2A adrenergic receptor	Homo sapiens (human)	IC50	2.4453	3	9
Alpha-2A adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	0.7050	2	2
Alpha-2A adrenergic receptor	Homo sapiens (human)	Ki	0.9289	3	9
Alpha-2A adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	0.0689	2	2
Alpha-2B adrenergic receptor	Homo sapiens (human)	IC50	3.1034	2	9
Alpha-2B adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	0.7050	2	2
Alpha-2B adrenergic receptor	Homo sapiens (human)	Ki	1.5939	1	8
Alpha-2B adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	0.0620	1	1
Alpha-2C adrenergic receptor	Homo sapiens (human)	IC50	3.1156	4	9
Alpha-2C adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	0.7050	2	2
Alpha-2C adrenergic receptor	Homo sapiens (human)	Ki	0.5807	2	7
Alpha-2C adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	0.0620	1	1
Alpha-amylase	Acarus siro	IC50	3.8000	1	1
Alpha-amylase 1A	Homo sapiens (human)	IC50	171.7496	4	9
Alpha-amylase 1A	Homo sapiens (human)	Ki	2.6000	1	1
Alpha-glucosidase	Blautia obeum	IC50	1,030.0000	1	1
Alpha-glucosidase MAL12	Saccharomyces cerevisiae S288C	IC50	309.9250	3	4
Alpha-glucosidase MAL32	Saccharomyces cerevisiae S288C	IC50	221.7220	4	5
Alpha-ketoglutarate-dependent dioxygenase FTO	Homo sapiens (human)	IC50	150.0000	1	1
Alpha-mannosidase	Canavalia ensiformis (jack bean)	IC50	49.0000	1	1
Alpha-synuclein	Homo sapiens (human)	IC50	20.1831	6	13
Amine oxidase [flavin-containing] A	Homo sapiens (human)	IC50	44.4270	72	78
Amine oxidase [flavin-containing] A	Homo sapiens (human)	Ki	13.5445	8	11
Amine oxidase [flavin-containing] A	Bos taurus (cattle)	IC50	42.7620	4	4
Amine oxidase [flavin-containing] A	Rattus norvegicus (Norway rat)	IC50	7.1306	11	11
Amine oxidase [flavin-containing] A	Bos taurus (cattle)	Ki	9.0283	5	6
Amine oxidase [flavin-containing] A	Rattus norvegicus (Norway rat)	Ki	12.2102	3	4
Amine oxidase [flavin-containing] B	Bos taurus (cattle)	IC50	29.2500	4	4
Amine oxidase [flavin-containing] B	Homo sapiens (human)	IC50	3.1944	107	108
Amine oxidase [flavin-containing] B	Rattus norvegicus (Norway rat)	IC50	2.3258	16	28
Amine oxidase [flavin-containing] B	Bos taurus (cattle)	Ki	1.4417	5	6
Amine oxidase [flavin-containing] B	Homo sapiens (human)	Ki	323.9212	18	23
Amine oxidase [flavin-containing] B	Rattus norvegicus (Norway rat)	Ki	0.6546	4	6
Aminopeptidase N	Homo sapiens (human)	IC50	15.5000	1	1
Aminopeptidase N	Sus scrofa (pig)	IC50	15.5000	1	1
Amyloid-beta precursor protein	Homo sapiens (human)	IC50	25.6725	49	56
Amyloid-beta precursor protein	Homo sapiens (human)	Ki	0.9686	6	7
Androgen receptor	Homo sapiens (human)	IC50	201.2545	6	7
Androgen receptor	Rattus norvegicus (Norway rat)	IC50	29.9436	3	6
Androgen receptor	Homo sapiens (human)	Ki	0.0140	1	1
Androgen receptor	Rattus norvegicus (Norway rat)	Ki	0.0195	1	2
Angiopoietin-1 receptor	Homo sapiens (human)	IC50	5,412.1547	11	11
Angiotensin-converting enzyme	Oryctolagus cuniculus (rabbit)	IC50	104,396.8488	7	7
Angiotensin-converting enzyme	Rattus norvegicus (Norway rat)	IC50	0.1400	1	1
Angiotensin-converting enzyme	Oryctolagus cuniculus (rabbit)	Ki	10.6757	2	3
Angiotensin-converting enzyme	Rattus norvegicus (Norway rat)	Ki	0.5000	1	3
Angiotensin-converting enzyme	Homo sapiens (human)	IC50	1,059.7652	9	12
Angiotensin-converting enzyme 2	Homo sapiens (human)	IC50	5.0700	2	2
Anthrax toxin receptor 2	Homo sapiens (human)	IC50	200.1512	2	6
Apoptosis regulator Bcl-2	Homo sapiens (human)	IC50	0.4500	1	1
Apoptosis regulator Bcl-2	Homo sapiens (human)	Ki	0.3622	2	2
Arachidonate 5-lipoxygenase-activating protein	Homo sapiens (human)	IC50	44.0000	1	1
Arginase	Leishmania amazonensis	IC50	15.7750	1	4
Arginase	Leishmania amazonensis	Ki	1.2000	1	1
Arginase-1	Bos taurus (cattle)	IC50	89.0000	1	2
Arginase-1	Homo sapiens (human)	IC50	622.5000	2	2
Arginase-1	Bos taurus (cattle)	Ki	136.0000	3	3
Aromatase	Homo sapiens (human)	IC50	9.8747	6	7
Aromatase	Homo sapiens (human)	Ki	111.5000	2	2
Aryl hydrocarbon receptor	Homo sapiens (human)	IC50	0.0280	1	1
Arylacetamide deacetylase	Homo sapiens (human)	Ki	300.0000	1	1
ATP-binding cassette sub-family C member 3	Homo sapiens (human)	IC50	121.8947	2	32
ATP-dependent translocase ABCB1	Homo sapiens (human)	IC50	32.7663	52	58
ATP-dependent translocase ABCB1	Mus musculus (house mouse)	IC50	26.3750	4	8
ATP-dependent translocase ABCB1	Homo sapiens (human)	Ki	30.0443	7	7
ATP-dependent translocase ABCB1	Mus musculus (house mouse)	Ki	3.5750	2	2
Aurora kinase A	Homo sapiens (human)	IC50	0.1082	26	26
Aurora kinase B	Homo sapiens (human)	IC50	1.6103	14	21
Aurora kinase C	Homo sapiens (human)	IC50	0.0022	2	2
Autoinducer 2-binding periplasmic protein LuxP	Vibrio harveyi	IC50	50.0000	1	1
B2 bradykinin receptor	Cavia porcellus (domestic guinea pig)	IC50	4.0000	2	2
Basic phospholipase A2 1	Naja melanoleuca (forest cobra)	IC50	2.9000	1	1
Basic phospholipase A2 PLA-A	Protobothrops flavoviridis	IC50	2.5000	1	1
Bcl-2-like protein 1	Homo sapiens (human)	IC50	0.5900	1	1
Bcl-2-like protein 10	Homo sapiens (human)	IC50	0.3600	1	1
Bcl-2-like protein 2	Homo sapiens (human)	IC50	2.3300	1	1
Bcl-2-related protein A1	Homo sapiens (human)	IC50	1.7900	1	1
Bcl2-associated agonist of cell death	Homo sapiens (human)	Ki	0.4900	1	1
BDNF/NT-3 growth factors receptor	Homo sapiens (human)	IC50	0.0004	3	3
Beta lactamase (plasmid)	Pseudomonas aeruginosa	IC50	7.7510	1	1
Beta-1 adrenergic receptor	Homo sapiens (human)	IC50	0.1760	1	1
Beta-1 adrenergic receptor	Homo sapiens (human)	Ki	0.0785	2	2
Beta-1 adrenergic receptor	Mus musculus (house mouse)	Ki	0.0490	1	1
Beta-1 adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	2.2129	5	5
Beta-2 adrenergic receptor	Cavia porcellus (domestic guinea pig)	IC50	0.2500	1	1
Beta-2 adrenergic receptor	Homo sapiens (human)	IC50	2.5730	1	1
Beta-2 adrenergic receptor	Homo sapiens (human)	Ki	0.9945	2	2
Beta-3 adrenergic receptor	Homo sapiens (human)	IC50	40.0992	1	4
Beta-3 adrenergic receptor	Homo sapiens (human)	Ki	30.0745	1	4
Beta-adrenergic receptor kinase 1	Homo sapiens (human)	IC50	1.1595	2	2
Beta-adrenergic receptor kinase 2	Homo sapiens (human)	IC50	0.8560	2	2
Beta-carbonic anhydrase 1	Mycobacterium tuberculosis H37Rv	Ki	5.5686	5	7
Beta-glucuronidase	Homo sapiens (human)	IC50	36.4700	1	1
Beta-glucuronidase	Bos taurus (cattle)	IC50	4.2300	1	1
Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein)	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	2.1550	2	6
Beta-lactamase	Enterobacter cloacae	IC50	269.6667	3	3
Beta-lactamase	Escherichia coli K-12	IC50	58.0000	4	4
Beta-lactamase	Bacillus anthracis	IC50	1,060.0000	1	1
Beta-lactamase	Pseudomonas aeruginosa	IC50	27.9000	1	1
Beta-lactamase VIM-1	Pseudomonas aeruginosa	IC50	9.3000	1	1
Beta-secretase 1	Homo sapiens (human)	IC50	36.1375	11	13
Beta-secretase 1	Homo sapiens (human)	Ki	9.5650	2	2
BH3-interacting domain death agonist	Homo sapiens (human)	IC50	1.0733	6	6
Bifunctional epoxide hydrolase 2	Homo sapiens (human)	IC50	58.6350	4	6
bifunctional UDP-N-acetylglucosamine pyrophosphorylase/glucosamine-1-phosphate N-acetyltransferase	Mycobacterium tuberculosis H37Rv	IC50	44.4250	1	2
Bile acid receptor	Homo sapiens (human)	IC50	1.4661	2	3
Bile salt export pump	Homo sapiens (human)	IC50	171.2618	10	88
Bile salt export pump	Rattus norvegicus (Norway rat)	IC50	286.5333	1	6
Bile salt export pump	Homo sapiens (human)	Ki	9.5000	1	1
Bile salt export pump	Rattus norvegicus (Norway rat)	Ki	6.1000	1	2
BiP isoform A	Glycine max (soybean)	IC50	600.0000	1	1
Bone morphogenetic protein receptor type-1A	Homo sapiens (human)	IC50	4.2880	1	1
Bone morphogenetic protein receptor type-2	Homo sapiens (human)	IC50	1.9400	2	2
Breakpoint cluster region protein	Homo sapiens (human)	IC50	0.0945	4	4
Broad substrate specificity ATP-binding cassette transporter ABCG2	Homo sapiens (human)	IC50	946.7196	10	15
Broad substrate specificity ATP-binding cassette transporter ABCG2	Homo sapiens (human)	Ki	0.5000	1	1
Bromodomain-containing protein 2	Homo sapiens (human)	IC50	10.3000	1	1
Bromodomain-containing protein 3	Homo sapiens (human)	IC50	13.7000	1	1
Bromodomain-containing protein 4	Homo sapiens (human)	IC50	12.4000	1	1
BZLF2	Human herpesvirus 4 type 2 (Epstein-Barr virus type 2)	IC50	2.0300	1	1
C-C chemokine receptor type 2	Homo sapiens (human)	IC50	35.0000	1	1
C-C chemokine receptor type 4	Homo sapiens (human)	IC50	47.2409	3	6
C-C motif chemokine 2	Homo sapiens (human)	IC50	6.9183	1	1
C-X-C chemokine receptor type 1	Homo sapiens (human)	IC50	35.3780	2	4
C-X-C chemokine receptor type 3	Homo sapiens (human)	IC50	67.2500	1	1
Calcineurin subunit B type 1	Homo sapiens (human)	IC50	34.0000	1	1
Calcium dependent protein kinase	Triticum aestivum (bread wheat)	IC50	19.0000	1	1
Calcium-dependent protein kinase 1	Plasmodium falciparum K1	IC50	0.2400	1	1
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A	Homo sapiens (human)	IC50	24.4200	2	2
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A	Homo sapiens (human)	Ki	14.0000	1	1
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A	Bos taurus (cattle)	IC50	500.0000	1	1
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	Bos taurus (cattle)	IC50	500.0000	1	1
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	Homo sapiens (human)	IC50	15.9967	3	3
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	Rattus norvegicus (Norway rat)	IC50	172.5000	2	2
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B	Homo sapiens (human)	Ki	14.0000	1	1
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C	Homo sapiens (human)	IC50	15.9250	2	2
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C	Rattus norvegicus (Norway rat)	IC50	172.5000	2	2
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C	Homo sapiens (human)	Ki	14.0000	1	1
Calcium/calmodulin-dependent protein kinase kinase 1	Homo sapiens (human)	IC50	0.0359	2	2
Calcium/calmodulin-dependent protein kinase kinase 2	Homo sapiens (human)	IC50	0.0246	2	2
Calcium/calmodulin-dependent protein kinase type 1	Homo sapiens (human)	IC50	0.0032	2	2
Calcium/calmodulin-dependent protein kinase type 1B	Homo sapiens (human)	IC50	0.0044	2	2
Calcium/calmodulin-dependent protein kinase type 1D	Homo sapiens (human)	IC50	0.0003	2	2
Calcium/calmodulin-dependent protein kinase type 1G	Homo sapiens (human)	IC50	0.0046	2	2
Calcium/calmodulin-dependent protein kinase type II subunit alpha	Homo sapiens (human)	IC50	0.0022	6	6
Calcium/calmodulin-dependent protein kinase type II subunit alpha	Rattus norvegicus (Norway rat)	IC50	4.2295	2	2
Calcium/calmodulin-dependent protein kinase type II subunit beta	Homo sapiens (human)	IC50	0.3765	8	8
Calcium/calmodulin-dependent protein kinase type II subunit beta	Rattus norvegicus (Norway rat)	IC50	8.4000	1	1
Calcium/calmodulin-dependent protein kinase type II subunit delta	Homo sapiens (human)	IC50	0.0024	5	5
Calcium/calmodulin-dependent protein kinase type II subunit delta	Rattus norvegicus (Norway rat)	IC50	8.4000	1	1
Calcium/calmodulin-dependent protein kinase type II subunit gamma	Homo sapiens (human)	IC50	0.0026	5	5
Calcium/calmodulin-dependent protein kinase type II subunit gamma	Rattus norvegicus (Norway rat)	IC50	8.4000	1	1
Calcium/calmodulin-dependent protein kinase type IV	Homo sapiens (human)	IC50	0.1475	2	2
Calmodulin-1	Homo sapiens (human)	IC50	12.9700	1	1
Calpain-2 catalytic subunit	Homo sapiens (human)	IC50	0.0020	1	1
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A	Homo sapiens (human)	IC50	10.0000	1	1
cAMP-dependent protein kinase	Oryctolagus cuniculus (rabbit)	IC50	500.0000	1	1
cAMP-dependent protein kinase catalytic subunit alpha	Bos taurus (cattle)	IC50	4.2576	6	29
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	IC50	17.2429	17	24
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	Ki	0.4600	1	1
cAMP-dependent protein kinase catalytic subunit alpha	Rattus norvegicus (Norway rat)	IC50	0.0550	3	3
cAMP-dependent protein kinase catalytic subunit alpha	Mus musculus (house mouse)	Ki	0.4950	1	2
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	IC50	3.6786	15	16
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	Ki	0.4600	1	1
cAMP-dependent protein kinase catalytic subunit beta	Bos taurus (cattle)	IC50	100.0000	1	1
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	IC50	3.9221	14	15
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	Ki	0.4600	1	1
cAMP-dependent protein kinase catalytic subunit PRKX	Homo sapiens (human)	IC50	0.0014	2	2
cAMP-dependent protein kinase type II-alpha regulatory subunit	Bos taurus (cattle)	IC50	100.0000	1	1
cAMP-dependent protein kinase type II-beta regulatory subunit	Bos taurus (cattle)	IC50	100.0000	1	1
cAMP-specific 3',5'-cyclic phosphodiesterase 4A	Homo sapiens (human)	IC50	747.0000	1	1
cAMP-specific 3',5'-cyclic phosphodiesterase 4B	Homo sapiens (human)	IC50	117.2667	3	3
cAMP-specific 3',5'-cyclic phosphodiesterase 4D	Homo sapiens (human)	IC50	1.2800	1	1
Canalicular multispecific organic anion transporter 1	Homo sapiens (human)	IC50	101.1579	7	34
Canalicular multispecific organic anion transporter 1	Homo sapiens (human)	Ki	11.2700	3	3
Canalicular multispecific organic anion transporter 1	Rattus norvegicus (Norway rat)	Ki	5.9800	2	2
Cannabinoid receptor 1	Rattus norvegicus (Norway rat)	IC50	25.0050	2	2
Cannabinoid receptor 1	Homo sapiens (human)	Ki	13.4167	5	6
Cannabinoid receptor 1	Rattus norvegicus (Norway rat)	Ki	10.5333	2	3
Cannabinoid receptor 2	Homo sapiens (human)	Ki	14.7800	4	5
Carbonic anhydrase	Candida albicans SC5314	Ki	5.6845	5	6
Carbonic anhydrase	Dicentrarchus labrax (European seabass)	Ki	4.1300	1	1
Carbonic anhydrase	Methanosarcina thermophila	Ki	0.5750	2	2
Carbonic anhydrase	Methanothermobacter thermautotrophicus str. Delta H	Ki	38.5000	1	1
Carbonic anhydrase	Saccharomyces cerevisiae S288C	Ki	0.1080	1	1
Carbonic anhydrase	Stylophora pistillata	Ki	0.6900	1	1
Carbonic anhydrase	Anopheles gambiae (African malaria mosquito)	Ki	0.1730	1	1
Carbonic anhydrase	Astrosclera willeyana	Ki	0.7320	1	1
Carbonic anhydrase	Cryptococcus neoformans var. grubii	Ki	2.0680	2	2
Carbonic anhydrase	Mycobacterium tuberculosis H37Rv	Ki	9.9300	2	2
Carbonic anhydrase	Nakaseomyces glabratus CBS 138	Ki	0.1160	1	1
Carbonic anhydrase	Stylophora pistillata	Ki	0.0342	2	2
Carbonic anhydrase	Sulfurihydrogenibium sp. YO3AOP1	Ki	0.0069	1	1
Carbonic anhydrase 1	Homo sapiens (human)	IC50	5,992.0311	6	10
Carbonic anhydrase 1	Homo sapiens (human)	Ki	187.9229	56	80
Carbonic anhydrase 12	Homo sapiens (human)	Ki	64.8708	17	32
Carbonic anhydrase 13	Homo sapiens (human)	Ki	3.1715	4	4
Carbonic anhydrase 13	Mus musculus (house mouse)	Ki	105.7047	5	19
Carbonic anhydrase 14	Homo sapiens (human)	Ki	89.5090	8	22
Carbonic anhydrase 15	Mus musculus (house mouse)	Ki	3.1470	6	7
Carbonic anhydrase 2	Homo sapiens (human)	IC50	4,855.0558	7	12
Carbonic anhydrase 2	Homo sapiens (human)	Ki	254.7307	67	92
Carbonic anhydrase 2	Mycobacterium tuberculosis H37Rv	Ki	1.7012	3	5
Carbonic anhydrase 3	Bos taurus (cattle)	Ki	6.5260	2	5
Carbonic anhydrase 3	Homo sapiens (human)	Ki	100.3791	8	22
Carbonic anhydrase 4	Bos taurus (cattle)	IC50	16.8152	3	6
Carbonic anhydrase 4	Bos taurus (cattle)	Ki	0.2900	2	2
Carbonic anhydrase 4	Homo sapiens (human)	Ki	88.5568	14	32
Carbonic anhydrase 5A, mitochondrial	Homo sapiens (human)	Ki	2,020.3699	8	22
Carbonic anhydrase 5B, mitochondrial	Homo sapiens (human)	Ki	107.6198	7	21
Carbonic anhydrase 6	Homo sapiens (human)	Ki	104.5752	10	25
Carbonic anhydrase 7	Homo sapiens (human)	Ki	70.7250	13	28
Carbonic anhydrase 9	Homo sapiens (human)	IC50	0.0160	3	3
Carbonic anhydrase 9	Homo sapiens (human)	Ki	114.2355	23	39
Carbonic anhydrase, alpha family	Hydrogenovibrio crunogenus XCL-2	Ki	0.9810	1	1
carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1	Homo sapiens (human)	IC50	7.3780	1	2
Carboxylic ester hydrolase	Equus caballus (horse)	IC50	0.1000	1	1
Carboxylic ester hydrolase	Rattus norvegicus (Norway rat)	IC50	50.0000	1	1
Carnitine O-palmitoyltransferase 1, liver isoform	Homo sapiens (human)	IC50	10.0000	1	1
Carnitine O-palmitoyltransferase 2, mitochondrial	Homo sapiens (human)	IC50	100.0000	1	1
Carnitine O-palmitoyltransferase 2, mitochondrial	Rattus norvegicus (Norway rat)	IC50	100.0000	1	1
Casein kinase I isoform alpha	Homo sapiens (human)	IC50	3.4120	4	4
Casein kinase I isoform alpha	Sus scrofa (pig)	IC50	10.0000	1	1
Casein kinase I isoform alpha-like	Homo sapiens (human)	IC50	1.8400	2	2
Casein kinase I isoform delta	Homo sapiens (human)	IC50	0.5370	5	5
Casein kinase I isoform epsilon	Homo sapiens (human)	IC50	1.2000	2	2
Casein kinase I isoform gamma-1	Homo sapiens (human)	IC50	5.3367	3	3
Casein kinase I isoform gamma-2	Homo sapiens (human)	IC50	1.9467	3	3
Casein kinase I isoform gamma-3	Homo sapiens (human)	IC50	2.6750	2	2
Casein kinase II subunit alpha	Homo sapiens (human)	IC50	7.0264	14	23
Casein kinase II subunit alpha	Homo sapiens (human)	Ki	0.7514	5	7
Casein kinase II subunit alpha	Mus musculus (house mouse)	IC50	10.0000	1	1
Casein kinase II subunit alpha	Rattus norvegicus (Norway rat)	IC50	0.0400	1	1
Casein kinase II subunit alpha 3	Homo sapiens (human)	IC50	2.4400	1	5
Casein kinase II subunit alpha 3	Homo sapiens (human)	Ki	1.1800	1	1
Casein kinase II subunit alpha'	Homo sapiens (human)	IC50	6.3289	13	22
Casein kinase II subunit alpha'	Mus musculus (house mouse)	IC50	10.0000	1	1
Casein kinase II subunit alpha'	Homo sapiens (human)	Ki	0.6750	2	2
Casein kinase II subunit alpha'-interacting protein	Mus musculus (house mouse)	IC50	10.0000	1	1
Casein kinase II subunit beta	Homo sapiens (human)	IC50	6.8975	11	20
Casein kinase II subunit beta	Mus musculus (house mouse)	IC50	10.0000	1	1
Casein kinase II subunit beta	Rattus norvegicus (Norway rat)	IC50	0.0400	1	1
Casein kinase II subunit beta	Homo sapiens (human)	Ki	0.6750	2	2
Caspase-1	Homo sapiens (human)	IC50	17.6865	3	6
Caspase-3	Homo sapiens (human)	IC50	21.9500	1	4
Caspase-4	Homo sapiens (human)	IC50	21.9500	1	4
Caspase-5	Homo sapiens (human)	IC50	21.9500	1	4
Caspase-9	Homo sapiens (human)	IC50	21.9500	1	4
Catechol O-methyltransferase	Mus musculus (house mouse)	IC50	4.5240	2	3
Cathepsin G	Homo sapiens (human)	IC50	93.0000	1	1
Cationic trypsin	Bos taurus (cattle)	IC50	34.0286	2	7
CDGSH iron-sulfur domain-containing protein 1	Homo sapiens (human)	IC50	12.2875	1	4
CDGSH iron-sulfur domain-containing protein 1	Rattus norvegicus (Norway rat)	IC50	1.0000	1	1
CDGSH iron-sulfur domain-containing protein 1	Homo sapiens (human)	Ki	0.5250	1	4
CDGSH iron-sulfur domain-containing protein 2	Homo sapiens (human)	IC50	4.8000	1	1
CDK-activating kinase assembly factor MAT1	Homo sapiens (human)	IC50	0.1216	4	4
Cell division control protein 42 homolog	Homo sapiens (human)	IC50	6.5000	2	2
Cell division cycle 7-related protein kinase	Homo sapiens (human)	IC50	0.0548	2	2
Cereblon isoform 4	Magnetospirillum gryphiswaldense	IC50	20.8000	1	1
Cereblon isoform 4	Magnetospirillum gryphiswaldense	Ki	5,570.2333	3	3
cGMP-dependent 3',5'-cyclic phosphodiesterase	Homo sapiens (human)	IC50	40.0000	1	1
cGMP-dependent 3',5'-cyclic phosphodiesterase	Rattus norvegicus (Norway rat)	IC50	81.3000	1	1
cGMP-dependent protein kinase 1	Homo sapiens (human)	IC50	0.0027	5	5
cGMP-dependent protein kinase 2	Homo sapiens (human)	IC50	0.0161	2	2
cGMP-inhibited 3',5'-cyclic phosphodiesterase A	Homo sapiens (human)	IC50	200.0000	2	2
cGMP-inhibited 3',5'-cyclic phosphodiesterase B	Homo sapiens (human)	IC50	200.0000	2	2
cGMP-specific 3',5'-cyclic phosphodiesterase	Bos taurus (cattle)	IC50	300.0000	1	1
cGMP-specific 3',5'-cyclic phosphodiesterase	Homo sapiens (human)	IC50	39.5225	3	4
Chain A, (3R)-hydroxymyristoyl-acyl carrier protein dehydratase	Helicobacter pylori	Ki	11.2250	1	4
Chain A, APH(2')-Id	Enterococcus casseliflavus	Ki	25.1000	1	1
Chain A, cAMP-dependent protein kinase, alpha-catalytic subunit	Bos taurus (cattle)	IC50	2.2800	1	5
Chain A, Carbonic anhydrase II	Homo sapiens (human)	IC50	0.0210	1	1
Chain A, Casein kinase II subunit alpha	Homo sapiens (human)	Ki	0.0200	1	1
Chain A, Chitinase	Clonostachys rosea	Ki	19,700.0000	1	1
Chain A, Endochitinase	Saccharomyces cerevisiae (brewer's yeast)	Ki	3.2000	1	3
Chain A, Epoxide hydrolase	Aspergillus niger	Ki	250.0000	1	1
Chain A, Erk2	Homo sapiens (human)	Ki	0.0004	1	1
Chain A, Estrogen receptor 1 (alpha)	Homo sapiens (human)	IC50	0.0090	1	1
Chain A, Glycogen Phosphorylase	Oryctolagus cuniculus (rabbit)	Ki	100.0000	1	1
Chain A, Glycogen Synthase Kinase-3 Beta	Homo sapiens (human)	IC50	0.0150	1	2
Chain A, HDLP (HISTONE DEACETYLASE-LIKE PROTEIN)	Aquifex aeolicus	IC50	0.4000	1	1
Chain A, Histone deacetylase 7a	Homo sapiens (human)	IC50	0.3000	1	2
Chain A, Hyaluronidase, phage associated	Streptococcus pyogenes	IC50	1,000.0000	1	1
Chain A, Lck Kinase	Homo sapiens (human)	IC50	0.0200	1	1
Chain A, limonene-1,2-epoxide hydrolase	Rhodococcus erythropolis	Ki	100.0000	1	1
Chain A, Methyltransferase Wbdd	Escherichia coli	IC50	68.0000	1	1
Chain A, Mitogen-activated protein kinase 10	Homo sapiens (human)	IC50	0.1500	1	3
Chain A, NAD-dependent deacetylase	Thermotoga maritima	IC50	1,000.0000	1	1
Chain A, Pancreatic alpha-amylase	Homo sapiens (human)	Ki	110.0000	1	2
Chain A, POLYMERASE PA	Influenza A virus	IC50	1.9000	1	1
Chain A, Polymerase Pa	Influenza A virus (A/California/04/2009(H1N1))	IC50	1.9000	1	4
Chain A, Protein kinase C, theta type	Homo sapiens (human)	Ki	0.0003	1	1
Chain A, Proto-oncogene serine/threonine-protein kinase Pim-1	Homo sapiens (human)	IC50	1.3925	1	8
Chain A, Rho-associated protein kinase 1	Homo sapiens (human)	Ki	0.5300	1	3
Chain A, RNA-directed RNA polymerase NS5	Dengue virus 2 16681-PDK53	IC50	35.0600	1	1
Chain A, Serine/threonine-protein kinase Chk1	Homo sapiens (human)	Ki	0.0078	1	3
Chain A, Serine/threonine-protein kinase TAO2	Rattus norvegicus (Norway rat)	IC50	3.0000	1	1
Chain A, Tyrosine-protein kinase BTK	Homo sapiens (human)	IC50	0.0007	1	1
Chain A, Tyrosine-protein kinase Lyn	Mus musculus (house mouse)	IC50	0.0090	1	2
Chain A, Tyrosine-protein kinase SYK	Homo sapiens (human)	IC50	0.0120	1	1
Chain A, Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	IC50	0.0558	1	1
Chain A, X-ray structure of the sucrose-phosphatase (SPP) from Synechocystis sp.PCC6803 in complex with cellobiose	Synechocystis sp. PCC 6803	Ki	26,000.0000	1	1
Chain A, X-ray structure of the sucrose-phosphatase (SPP) from Synechocystis sp.PCC6803 in complex with maltose	Synechocystis sp. PCC 6803	Ki	26,000.0000	1	1
Chain A, X-ray structure of the sucrose-phosphatase (SPP) from Synechocystis sp.PCC6803 in complex with trehalose	Synechocystis sp. PCC 6803	Ki	26,000.0000	1	1
Chain B, (3R)-hydroxymyristoyl-acyl carrier protein dehydratase	Helicobacter pylori	Ki	11.2250	1	4
Chain B, Cell division protein kinase 6	Homo sapiens (human)	IC50	0.8500	1	1
Chain B, Glycogen Synthase Kinase-3 Beta	Homo sapiens (human)	IC50	0.0150	1	1
Chain B, HDLP (HISTONE DEACETYLASE-LIKE PROTEIN)	Aquifex aeolicus	IC50	0.4000	1	1
Chain B, Rho-associated protein kinase 1	Homo sapiens (human)	Ki	0.5300	1	1
Chain E, Camp-dependent Protein Kinase	Bos taurus (cattle)	Ki	0.0080	1	1
Chain E, cAMP-dependent protein kinase, alpha-catalytic subunit	Mus musculus (house mouse)	Ki	0.5300	1	1
Chain I, cAMP-dependent protein kinase inhibitor alpha	synthetic construct	IC50	2.2800	1	2
Chain I, cAMP-dependent protein kinase inhibitor, alpha form	synthetic construct	Ki	0.5300	1	1
Chain X, Proto-oncogene tyrosine-protein kinase Fyn	Homo sapiens (human)	IC50	0.0048	1	1
Chitotriosidase-1	Homo sapiens (human)	IC50	363.0000	1	2
Cholesteryl ester transfer protein	Homo sapiens (human)	IC50	32.2133	3	3
Choline O-acetyltransferase	Rattus norvegicus (Norway rat)	Ki	25,000.0000	1	1
Cholinesterase	Equus caballus (horse)	IC50	86.4500	4	4
Cholinesterase	Homo sapiens (human)	IC50	853.4535	11	13
Cholinesterase	Homo sapiens (human)	Ki	0.8000	1	1
Chymotrypsin-C	Homo sapiens (human)	IC50	100.0000	1	1
Chymotrypsin-like elastase family member 1	Sus scrofa (pig)	IC50	28.7500	1	4
Chymotrypsinogen A	Bos taurus (cattle)	IC50	196.1667	3	3
Chymotrypsinogen B	Homo sapiens (human)	IC50	100.0000	1	1
Citron Rho-interacting kinase	Homo sapiens (human)	IC50	0.8327	3	3
CMP-N-acetylneuraminate-beta-galactosamide-alpha-2,3-sialyltransferase 1	Homo sapiens (human)	IC50	38.3662	1	13
Coagulation factor VII	Homo sapiens (human)	IC50	0.0340	1	1
Coagulation factor VII	Homo sapiens (human)	Ki	8,000.0000	1	1
Coagulation factor X	Homo sapiens (human)	IC50	0.1700	1	1
Coagulation factor X	Homo sapiens (human)	Ki	0.5700	1	1
Coiled-coil domain-containing protein 6	Homo sapiens (human)	IC50	0.0022	1	1
Collagenase 3	Homo sapiens (human)	IC50	4.2370	2	2
Corticosteroid 11-beta-dehydrogenase isozyme 1	Homo sapiens (human)	IC50	1.9000	1	1
Corticotropin-releasing factor receptor 2	Homo sapiens (human)	Ki	10.0000	1	1
CPG DNA methylase	Spiroplasma monobiae	Ki	0.0280	1	1
CREB-binding protein	Homo sapiens (human)	IC50	33.3333	6	6
Cruzipain	Trypanosoma cruzi	IC50	197.3083	8	12
Cyclin homolog	Herpesvirus saimiri (strain 11)	IC50	20.4358	1	12
Cyclin-A1	Homo sapiens (human)	IC50	0.6936	7	7
Cyclin-A1	Homo sapiens (human)	Ki	0.0040	1	1
Cyclin-A2	Homo sapiens (human)	IC50	3.6633	15	15
Cyclin-A2	Homo sapiens (human)	Ki	0.0026	2	3
Cyclin-C	Homo sapiens (human)	IC50	0.0105	2	2
Cyclin-dependent kinase 1	Homo sapiens (human)	IC50	25.3010	38	43
Cyclin-dependent kinase 1	Oryzias latipes (Japanese medaka)	IC50	13.7653	3	18
Cyclin-dependent kinase 1	Homo sapiens (human)	Ki	0.0020	1	2
Cyclin-dependent kinase 1	Mus musculus (house mouse)	IC50	0.0080	1	1
Cyclin-dependent kinase 12	Homo sapiens (human)	IC50	0.0530	1	1
Cyclin-dependent kinase 13	Homo sapiens (human)	IC50	0.0570	1	1
Cyclin-dependent kinase 14	Homo sapiens (human)	IC50	0.1145	2	2
Cyclin-dependent kinase 16	Homo sapiens (human)	IC50	0.0206	2	2
Cyclin-dependent kinase 17	Homo sapiens (human)	IC50	0.0135	2	2
Cyclin-dependent kinase 18	Homo sapiens (human)	IC50	0.0587	2	2
Cyclin-dependent kinase 2	Homo sapiens (human)	IC50	16.2181	36	37
Cyclin-dependent kinase 2	Homo sapiens (human)	Ki	0.0026	2	3
Cyclin-dependent kinase 3	Homo sapiens (human)	IC50	71.4387	7	7
Cyclin-dependent kinase 4	Homo sapiens (human)	IC50	20.8403	14	15
Cyclin-dependent kinase 4	Homo sapiens (human)	Ki	0.0410	1	1
Cyclin-dependent kinase 5 activator 1	Homo sapiens (human)	IC50	9.3392	18	35
Cyclin-dependent kinase 6	Homo sapiens (human)	IC50	13.3344	9	22
Cyclin-dependent kinase 7	Homo sapiens (human)	IC50	0.2793	5	5
Cyclin-dependent kinase 8	Homo sapiens (human)	IC50	0.0105	2	2
Cyclin-dependent kinase 9	Homo sapiens (human)	IC50	0.0491	10	10
Cyclin-dependent kinase 9	Homo sapiens (human)	Ki	0.0070	1	1
Cyclin-dependent kinase-like 3	Homo sapiens (human)	IC50	1.1000	1	1
Cyclin-dependent-like kinase 5	Homo sapiens (human)	IC50	9.3392	18	35
Cyclin-G-associated kinase	Homo sapiens (human)	IC50	0.3127	4	4
Cyclin-H	Homo sapiens (human)	IC50	0.2793	5	5
Cyclin-K	Homo sapiens (human)	IC50	0.0948	5	5
Cyclin-O	Homo sapiens (human)	IC50	0.0016	4	4
Cyclin-T1	Homo sapiens (human)	IC50	0.0205	6	6
Cyclin-T1	Homo sapiens (human)	Ki	0.0070	1	1
Cyclin-T2	Homo sapiens (human)	IC50	0.0038	1	1
Cyclin-Y	Homo sapiens (human)	IC50	0.0518	8	8
Cyclooxygenase-2	Canis lupus familiaris (dog)	IC50	0.9000	1	1
Cystathionine beta-synthase	Homo sapiens (human)	IC50	18.8000	1	1
Cysteine protease	Trypanosoma brucei rhodesiense	IC50	7.7500	1	1
Cysteine protease ATG4B	Homo sapiens (human)	IC50	4.2500	2	2
Cytochrome c oxidase subunit 1	Ovis aries (sheep)	IC50	19.3500	3	3
Cytochrome c oxidase subunit 2	Homo sapiens (human)	IC50	0.3710	3	3
Cytochrome c oxidase subunit 2	Ovis aries (sheep)	IC50	0.0882	4	4
Cytochrome P450 11B1, mitochondrial	Rattus norvegicus (Norway rat)	IC50	43.3333	1	3
Cytochrome P450 11B2, mitochondrial	Homo sapiens (human)	IC50	0.0110	1	1
Cytochrome P450 1A1	Homo sapiens (human)	IC50	6.6620	6	7
Cytochrome P450 1A1	Homo sapiens (human)	Ki	10.9433	3	6
Cytochrome P450 1A2	Homo sapiens (human)	IC50	12.5251	10	12
Cytochrome P450 1A2	Homo sapiens (human)	Ki	7.1100	2	2
Cytochrome P450 1A2	Rattus norvegicus (Norway rat)	Ki	0.0003	1	1
Cytochrome P450 1B1	Homo sapiens (human)	IC50	1.8525	9	10
Cytochrome P450 1B1	Homo sapiens (human)	Ki	1.8059	4	8
Cytochrome P450 2B1	Rattus norvegicus (Norway rat)	Ki	1.0500	1	1
Cytochrome P450 2C11	Rattus norvegicus (Norway rat)	Ki	0.0003	1	1
Cytochrome P450 2C19	Homo sapiens (human)	IC50	3.4776	4	8
Cytochrome P450 2C8	Homo sapiens (human)	IC50	13.5000	2	2
Cytochrome P450 2C9	Homo sapiens (human)	IC50	15.3306	7	13
Cytochrome P450 2C9	Homo sapiens (human)	Ki	27.6667	2	3
Cytochrome P450 2D26	Rattus norvegicus (Norway rat)	IC50	45.4000	1	1
Cytochrome P450 2D3	Rattus norvegicus (Norway rat)	IC50	1,927.0000	1	1
Cytochrome P450 2D4	Rattus norvegicus (Norway rat)	IC50	833.0000	1	1
Cytochrome P450 2D6	Homo sapiens (human)	IC50	17.1653	13	16
Cytochrome P450 2D6	Homo sapiens (human)	Ki	0.9752	2	2
Cytochrome P450 2J2	Homo sapiens (human)	IC50	14.9996	4	7
Cytochrome P450 2J2	Homo sapiens (human)	Ki	0.0200	1	2
Cytochrome P450 3A4	Homo sapiens (human)	IC50	8.8356	14	17
Cytochrome P450 3A4	Homo sapiens (human)	Ki	6.9640	3	5
Cytochrome P450 3A43	Homo sapiens (human)	IC50	2.0600	1	1
Cytochrome P450 3A43	Homo sapiens (human)	Ki	7.6000	1	2
Cytochrome P450 3A5	Homo sapiens (human)	IC50	21.0300	2	2
Cytochrome P450 3A5	Homo sapiens (human)	Ki	7.6000	1	2
Cytochrome P450 3A7	Homo sapiens (human)	IC50	2.0600	1	1
Cytochrome P450 3A7	Homo sapiens (human)	Ki	7.6000	1	2
Cytoplasmic tyrosine-protein kinase BMX	Homo sapiens (human)	IC50	87.2498	4	4
Cytosol aminopeptidase	Sus scrofa (pig)	IC50	34.3000	1	1
D	Bos taurus (cattle)	IC50	0.0500	1	1
D	Rattus norvegicus (Norway rat)	Ki	0.7110	2	2
D-amino-acid oxidase	Sus scrofa (pig)	IC50	1.0700	2	2
D(1A) dopamine receptor	Homo sapiens (human)	IC50	8.4385	1	6
D(1A) dopamine receptor	Sus scrofa (pig)	IC50	0.0010	1	1
D(1A) dopamine receptor	Homo sapiens (human)	Ki	4.2192	1	6
D(2) dopamine receptor	Bos taurus (cattle)	IC50	0.0500	1	1
D(2) dopamine receptor	Homo sapiens (human)	IC50	2.5332	3	6
D(2) dopamine receptor	Rattus norvegicus (Norway rat)	IC50	7.5053	5	5
D(2) dopamine receptor	Homo sapiens (human)	Ki	0.5292	3	6
D(2) dopamine receptor	Rattus norvegicus (Norway rat)	Ki	0.5664	4	5
D(3) dopamine receptor	Homo sapiens (human)	IC50	21.8212	3	8
D(3) dopamine receptor	Rattus norvegicus (Norway rat)	IC50	2.0000	1	1
D(3) dopamine receptor	Homo sapiens (human)	Ki	7.4435	3	8
D(3) dopamine receptor	Rattus norvegicus (Norway rat)	Ki	1.5240	1	1
D(4) dopamine receptor	Homo sapiens (human)	IC50	3.3113	2	2
D(4) dopamine receptor	Homo sapiens (human)	Ki	3.9400	2	2
Death-associated protein kinase 1	Homo sapiens (human)	IC50	23.6328	7	11
Death-associated protein kinase 2	Homo sapiens (human)	IC50	0.0064	2	2
Death-associated protein kinase 3	Homo sapiens (human)	IC50	0.0026	2	2
Dehydrogenase/reductase SDR family member 9	Rattus norvegicus (Norway rat)	IC50	100.0000	1	1
Delta carbonic anhydrase	Conticribra weissflogii	Ki	0.2650	1	1
Delta-type opioid receptor	Homo sapiens (human)	IC50	0.1166	6	6
Delta-type opioid receptor	Mus musculus (house mouse)	IC50	0.6054	8	12
Delta-type opioid receptor	Rattus norvegicus (Norway rat)	IC50	0.2278	11	16
Delta-type opioid receptor	Homo sapiens (human)	Ki	0.2700	28	35
Delta-type opioid receptor	Mus musculus (house mouse)	Ki	25.0105	2	2
Delta-type opioid receptor	Rattus norvegicus (Norway rat)	Ki	0.1600	14	16
Dihydrofolate reductase	Escherichia coli K-12	IC50	348.9000	1	1
Dihydrofolate reductase	Homo sapiens (human)	IC50	6.2000	1	1
Dihydrofolate reductase	Mus musculus (house mouse)	IC50	6.2000	1	1
Dihydrofolate reductase	Pneumocystis carinii	IC50	6.2000	1	1
Dihydrofolate reductase	Rattus norvegicus (Norway rat)	IC50	6.2000	1	1
Dihydrofolate reductase	Escherichia coli K-12	Ki	15.2400	1	1
Dihydrofolate reductase	Homo sapiens (human)	Ki	6,233.3333	1	3
Dihydroorotate dehydrogenase	Leishmania major	IC50	697.7383	1	6
Dihydroorotate dehydrogenase (quinone), mitochondrial	Homo sapiens (human)	IC50	50.0000	1	1
Dipeptidyl peptidase 3	Homo sapiens (human)	IC50	42.1250	1	4
Dipeptidyl peptidase 4	Homo sapiens (human)	IC50	51.3120	3	10
Dipeptidyl peptidase 4	Rattus norvegicus (Norway rat)	IC50	25.6677	1	3
Discoidin domain-containing receptor 2	Homo sapiens (human)	IC50	0.0008	2	2
Disintegrin and metalloproteinase domain-containing protein 17	Homo sapiens (human)	IC50	110.5000	1	2
DNA (cytosine-5)-methyltransferase 1	Homo sapiens (human)	IC50	15.2500	1	2
DNA (cytosine-5)-methyltransferase 3-like	Homo sapiens (human)	IC50	100.0000	1	1
DNA (cytosine-5)-methyltransferase 3A	Homo sapiens (human)	IC50	100.0000	1	1
DNA dC->dU-editing enzyme APOBEC-3A isoform a	Homo sapiens (human)	IC50	17.5000	1	1
DNA dC->dU-editing enzyme APOBEC-3G isoform 1	Homo sapiens (human)	IC50	3.5033	2	3
DNA gyrase subunit A	Mycobacterium tuberculosis H37Rv	IC50	50.0000	1	1
DNA gyrase subunit B	Mycobacterium tuberculosis H37Rv	IC50	50.0000	1	1
DNA polymerase alpha catalytic subunit	Homo sapiens (human)	IC50	20.0000	1	1
DNA polymerase beta	Homo sapiens (human)	IC50	18.6000	1	1
DNA polymerase beta	Rattus norvegicus (Norway rat)	IC50	6.6500	2	2
DNA polymerase catalytic subunit	Human herpesvirus 3 strain Dumas	IC50	0.2800	1	1
DNA polymerase catalytic subunit	Human herpesvirus 5 strain AD169	IC50	2.5000	2	2
DNA polymerase delta catalytic subunit	Homo sapiens (human)	IC50	20.0000	1	1
DNA polymerase eta	Homo sapiens (human)	IC50	0.0620	1	1
DNA polymerase iota	Homo sapiens (human)	IC50	0.0620	1	1
DNA primase	Mycobacterium tuberculosis CDC1551	IC50	100.0000	1	1
DNA primase TraC	Escherichia coli	IC50	700.0000	1	1
DNA repair protein RAD52 homolog	Homo sapiens (human)	IC50	2.5108	5	5
DNA topoisomerase 1	Homo sapiens (human)	IC50	8.2600	1	1
DNA topoisomerase 2-alpha	Homo sapiens (human)	IC50	1,000.0000	1	1
DNA-(apurinic or apyrimidinic site) endonuclease	Homo sapiens (human)	IC50	0.3200	2	2
DNA-dependent protein kinase catalytic subunit	Homo sapiens (human)	IC50	770.4492	12	13
DNA-dependent protein kinase catalytic subunit	Homo sapiens (human)	Ki	3.6480	5	5
DNA-directed RNA polymerase subunit beta	Escherichia coli O127:H6 str. E2348/69	IC50	511.3333	3	3
DNA-directed RNA polymerase subunit beta	Mycobacterium tuberculosis H37Rv	IC50	0.0100	1	1
Dual serine/threonine and tyrosine protein kinase	Homo sapiens (human)	IC50	0.0552	3	3
Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	IC50	4.0265	19	22
Dual specificity mitogen-activated protein kinase kinase 1	Rattus norvegicus (Norway rat)	IC50	4.2000	1	1
Dual specificity mitogen-activated protein kinase kinase 2	Homo sapiens (human)	IC50	7.6342	8	8
Dual specificity mitogen-activated protein kinase kinase 2	Rattus norvegicus (Norway rat)	IC50	4.2000	1	1
Dual specificity mitogen-activated protein kinase kinase 3	Homo sapiens (human)	IC50	0.0099	2	2
Dual specificity mitogen-activated protein kinase kinase 4	Homo sapiens (human)	IC50	0.7472	4	4
Dual specificity mitogen-activated protein kinase kinase 5	Homo sapiens (human)	IC50	0.0252	2	2
Dual specificity mitogen-activated protein kinase kinase 6	Homo sapiens (human)	IC50	0.0036	3	3
Dual specificity mitogen-activated protein kinase kinase 7	Homo sapiens (human)	IC50	0.9255	2	2
Dual specificity protein kinase CLK1	Homo sapiens (human)	IC50	3.3406	3	3
Dual specificity protein kinase CLK2	Homo sapiens (human)	IC50	1.8994	4	8
Dual specificity protein kinase CLK3	Homo sapiens (human)	IC50	0.9200	2	2
Dual specificity protein kinase CLK4	Homo sapiens (human)	IC50	0.0723	2	2
Dual specificity protein kinase TTK	Homo sapiens (human)	IC50	0.8987	3	3
Dual specificity protein phosphatase 1	Mus musculus (house mouse)	IC50	11.1850	1	2
dual specificity protein phosphatase 3	Homo sapiens (human)	IC50	34.0700	3	3
Dual specificity protein phosphatase 6	Rattus norvegicus (Norway rat)	IC50	19.6000	2	3
Dual specificity testis-specific protein kinase 1	Homo sapiens (human)	IC50	0.1995	2	2
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Homo sapiens (human)	IC50	5.4700	10	10
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Rattus norvegicus (Norway rat)	IC50	3.4473	3	3
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Homo sapiens (human)	IC50	0.0017	3	3
Dual specificity tyrosine-phosphorylation-regulated kinase 2	Homo sapiens (human)	IC50	0.1800	2	2
Dual specificity tyrosine-phosphorylation-regulated kinase 3	Homo sapiens (human)	IC50	0.0231	2	2
E-selectin	Homo sapiens (human)	IC50	500.0000	1	1
E3 ubiquitin-protein ligase XIAP	Homo sapiens (human)	IC50	100.0000	1	1
Ectonucleoside triphosphate diphosphohydrolase 1	Mus musculus (house mouse)	IC50	1.0300	1	2
Egl nine homolog 1	Homo sapiens (human)	IC50	119.5000	2	2
ELAV-like protein 1	Homo sapiens (human)	IC50	1.4000	1	1
ELAV-like protein 3	Homo sapiens (human)	IC50	1.1333	1	3
Endochitinase	Saccharomyces cerevisiae S288C	Ki	3.2000	1	1
Endochitinase A1	Aspergillus fumigatus	IC50	1,000.0000	1	1
Endochitinase B1	Aspergillus fumigatus	IC50	363.0000	1	2
Endothelial PAS domain-containing protein 1	Homo sapiens (human)	IC50	0.4100	2	2
Endothelin receptor type B	Homo sapiens (human)	Ki	0.0347	2	4
Endothelin receptor type B	Rattus norvegicus (Norway rat)	Ki	0.0347	1	2
Endothelin-1 receptor	Homo sapiens (human)	IC50	0.1148	1	1
Enoyl-[acyl-carrier-protein] reductase [NADH]	Mycobacterium tuberculosis H37Rv	IC50	0.0300	1	1
Enoyl-[acyl-carrier-protein] reductase [NADH]	Francisella tularensis subsp. tularensis SCHU S4	IC50	79.0000	1	1
Enoyl-[acyl-carrier-protein] reductase [NADH] FabI	Escherichia coli K-12	IC50	17.5000	2	4
Enoyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	4.0850	3	10
Enoyl-acyl-carrier protein reductase	Plasmodium falciparum (malaria parasite P. falciparum)	Ki	1.1491	3	9
Ephrin type-A receptor 1	Homo sapiens (human)	IC50	0.0947	3	3
Ephrin type-A receptor 2	Homo sapiens (human)	IC50	21.5842	5	5
Ephrin type-A receptor 2	Mus musculus (house mouse)	IC50	68.0000	2	2
Ephrin type-A receptor 3	Homo sapiens (human)	IC50	0.0347	4	4
Ephrin type-A receptor 4	Homo sapiens (human)	IC50	0.0105	2	2
Ephrin type-A receptor 5	Homo sapiens (human)	IC50	0.0159	2	2
Ephrin type-A receptor 6	Homo sapiens (human)	IC50	0.0160	2	2
Ephrin type-A receptor 7	Homo sapiens (human)	IC50	0.0478	2	2
Ephrin type-A receptor 8	Homo sapiens (human)	IC50	0.1061	2	2
Ephrin type-B receptor 1	Homo sapiens (human)	IC50	0.0694	3	3
Ephrin type-B receptor 2	Homo sapiens (human)	IC50	12.0314	4	5
Ephrin type-B receptor 3	Homo sapiens (human)	IC50	1.2855	2	2
Ephrin type-B receptor 4	Homo sapiens (human)	IC50	0.5155	5	5
Epidermal growth factor receptor	Homo sapiens (human)	IC50	57.5290	71	85
Epidermal growth factor receptor	Mus musculus (house mouse)	IC50	5.0500	2	2
Epidermal growth factor receptor	Homo sapiens (human)	Ki	240.0200	5	8
epidermal growth factor receptor isoform a precursor	Homo sapiens (human)	IC50	0.4467	1	1
Epithelial discoidin domain-containing receptor 1	Homo sapiens (human)	IC50	0.9655	3	3
Epoxide hydrolase 1	Homo sapiens (human)	IC50	7.0000	1	1
Estrogen receptor	Homo sapiens (human)	IC50	1.9258	24	28
Estrogen receptor	Homo sapiens (human)	Ki	1.8307	2	3
Estrogen receptor 1	Homo sapiens (human)	IC50	36.0969	1	2
Estrogen receptor beta	Homo sapiens (human)	IC50	1.9202	25	30
Estrogen receptor beta	Homo sapiens (human)	Ki	0.0123	2	2
estrogen receptor beta isoform 1	Homo sapiens (human)	IC50	50.0000	1	1
eukaryotic translation initiation factor 4 gamma 1 isoform 4	Homo sapiens (human)	IC50	32.1157	1	2
eukaryotic translation initiation factor 4E isoform 1	Mus musculus (house mouse)	IC50	32.1157	1	2
Eyes absent homolog 2	Homo sapiens (human)	IC50	386.2500	4	4
Fatty acid synthase	Gallus gallus (chicken)	IC50	55.2800	3	5
Fatty acid synthase	Homo sapiens (human)	IC50	51.9700	1	1
Fatty acid synthase	Rattus norvegicus (Norway rat)	IC50	250.0000	1	1
Fatty acid-binding protein, intestinal	Homo sapiens (human)	Ki	100.8667	2	3
Fatty acid-binding protein, liver	Homo sapiens (human)	Ki	0.0433	1	3
Fatty acid-binding protein, liver	Mus musculus (house mouse)	Ki	0.0430	1	1
Fatty acid-binding protein, liver	Rattus norvegicus (Norway rat)	Ki	425.0435	3	11
Fatty-acid amide hydrolase 1	Homo sapiens (human)	IC50	0.8975	2	2
Fatty-acid amide hydrolase 1	Rattus norvegicus (Norway rat)	IC50	76.3250	3	4
Fatty-acid amide hydrolase 1	Rattus norvegicus (Norway rat)	Ki	10.0000	1	1
Fibroblast growth factor receptor 1	Homo sapiens (human)	IC50	0.0699	7	7
Fibroblast growth factor receptor 2	Homo sapiens (human)	IC50	0.0504	10	10
Fibroblast growth factor receptor 3	Homo sapiens (human)	IC50	0.0554	10	10
Fibroblast growth factor receptor 4	Homo sapiens (human)	IC50	13,900.1457	7	7
fMet-Leu-Phe receptor	Homo sapiens (human)	IC50	10.0000	1	1
Focal adhesion kinase 1	Homo sapiens (human)	IC50	0.4242	11	12
Fructose-1,6-bisphosphatase 1	Homo sapiens (human)	IC50	15.1500	2	2
Fructose-1,6-bisphosphatase 1	Sus scrofa (pig)	IC50	10.0000	1	1
Fructose-1,6-bisphosphatase 1	Rattus norvegicus (Norway rat)	IC50	10.0000	1	1
G protein-coupled receptor kinase 4	Homo sapiens (human)	IC50	0.0914	2	2
G protein-coupled receptor kinase 5	Homo sapiens (human)	IC50	0.0490	2	2
G protein-coupled receptor kinase 6	Homo sapiens (human)	IC50	10.6986	3	4
G-protein coupled receptor	Apis mellifera (honey bee)	IC50	73.0000	1	1
G-protein coupled receptor 35	Homo sapiens (human)	IC50	11.4550	1	4
G-protein coupled receptor 55	Homo sapiens (human)	IC50	1.4652	1	1
G1/S-specific cyclin-D1	Homo sapiens (human)	IC50	19.5345	15	16
G1/S-specific cyclin-D1	Homo sapiens (human)	Ki	0.0410	1	1
G1/S-specific cyclin-D3	Homo sapiens (human)	IC50	0.0550	6	6
G1/S-specific cyclin-E1	Homo sapiens (human)	IC50	0.0108	17	17
G1/S-specific cyclin-E2	Homo sapiens (human)	IC50	0.0110	3	3
G2/mitotic-specific cyclin-B	Marthasterias glacialis (spiny starfish)	IC50	13.7653	3	18
G2/mitotic-specific cyclin-B1	Homo sapiens (human)	IC50	18.9369	26	31
G2/mitotic-specific cyclin-B2	Homo sapiens (human)	IC50	11.2829	12	15
G2/mitotic-specific cyclin-B3	Homo sapiens (human)	IC50	11.2829	12	15
GABA theta subunit	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
GABA theta subunit	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	IC50	2,913.3625	2	4
Gamma-aminobutyric acid receptor subunit alpha-1	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit alpha-2	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit alpha-3	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit alpha-4	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit alpha-5	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit alpha-6	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit beta-1	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit beta-2	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit beta-3	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit delta	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit epsilon	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit gamma-1	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit gamma-2	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit gamma-3	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	IC50	5,810.0000	1	2
Gamma-aminobutyric acid receptor subunit pi	Homo sapiens (human)	Ki	52.8117	2	2
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Gamma-aminobutyric acid receptor subunit theta	Homo sapiens (human)	Ki	52.8117	2	2
Genome polyprotein	Coxsackievirus B3 (strain Nancy)	IC50	1.1000	1	1
Genome polyprotein		IC50	1.6000	1	1
Genome polyprotein	Zika virus	IC50	36.7667	2	3
Genome polyprotein	Zika virus	Ki	0.8000	1	1
Ghrelin O-acyltransferase	Homo sapiens (human)	IC50	100.0000	1	1
Glucocorticoid receptor	Homo sapiens (human)	IC50	7.8463	2	3
Glucocorticoid receptor	Homo sapiens (human)	Ki	1.0315	1	2
Glucose-6-phosphate 1-dehydrogenase	Homo sapiens (human)	IC50	74.5300	1	1
Glucose-6-phosphate 1-dehydrogenase	Saccharomyces cerevisiae S288C	IC50	0.2500	1	1
glucose-6-phosphate 1-dehydrogenase isoform b	Homo sapiens (human)	IC50	80.0000	1	1
glucose-6-phosphate dehydrogenase	Leuconostoc mesenteroides	IC50	25.0000	1	1
glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase	Plasmodium berghei	IC50	50.8333	3	3
Glutamate receptor ionotropic, NMDA 1	Rattus norvegicus (Norway rat)	IC50	41.3950	4	4
Glutamate receptor ionotropic, NMDA 2A	Rattus norvegicus (Norway rat)	IC50	10.2900	2	2
Glutamate receptor ionotropic, NMDA 2B	Rattus norvegicus (Norway rat)	IC50	15.5427	3	3
Glutamate receptor ionotropic, NMDA 2C	Rattus norvegicus (Norway rat)	IC50	50.7900	2	2
Glutamate receptor ionotropic, NMDA 2D	Rattus norvegicus (Norway rat)	IC50	1.5800	1	1
Glutamate receptor ionotropic, NMDA 3A	Rattus norvegicus (Norway rat)	IC50	1.5800	1	1
Glutamate receptor ionotropic, NMDA 3B	Rattus norvegicus (Norway rat)	IC50	1.5800	1	1
Glutaminyl-peptide cyclotransferase	Mus musculus (house mouse)	Ki	1,311.0000	1	2
Glutathione hydrolase 1 proenzyme	Homo sapiens (human)	IC50	36.0000	1	1
Glutathione reductase	Saccharomyces cerevisiae S288C	IC50	48.8000	1	1
Glutathione reductase, mitochondrial	Homo sapiens (human)	IC50	96.9333	3	3
Glutathione S-transferase	Plasmodium falciparum 3D7	IC50	74.4000	1	1
Glutathione S-transferase Mu 1	Mus musculus (house mouse)	IC50	100.0000	1	1
Glutathione S-transferase omega-1	Homo sapiens (human)	IC50	75.0000	1	1
Glutathione S-transferase P	Homo sapiens (human)	IC50	65.3667	2	3
Glyceraldehyde-3-phosphate dehydrogenase, glycosomal	Trypanosoma cruzi	IC50	142.0000	1	1
Glycine receptor subunit alpha-1	Rattus norvegicus (Norway rat)	IC50	2.2695	1	2
Glycine receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Ki	1.0315	1	2
Glycine receptor subunit alpha-2	Rattus norvegicus (Norway rat)	IC50	2.2695	1	2
Glycine receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Ki	1.0315	1	2
Glycine receptor subunit alpha-3	Rattus norvegicus (Norway rat)	IC50	2.2695	1	2
Glycine receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Ki	1.0315	1	2
Glycine receptor subunit beta	Rattus norvegicus (Norway rat)	IC50	2.2695	1	2
Glycine receptor subunit beta	Rattus norvegicus (Norway rat)	Ki	1.0315	1	2
Glycogen phosphorylase, liver form	Homo sapiens (human)	IC50	4.8000	1	1
Glycogen phosphorylase, liver form	Rattus norvegicus (Norway rat)	IC50	648.0000	1	1
Glycogen phosphorylase, muscle form	Oryctolagus cuniculus (rabbit)	IC50	127.9007	14	19
Glycogen phosphorylase, muscle form	Rattus norvegicus (Norway rat)	IC50	182.0000	1	1
Glycogen synthase kinase 3	Plasmodium falciparum 3D7	IC50	10.0000	1	1
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	IC50	0.6772	7	9
Glycogen synthase kinase-3 beta	Homo sapiens (human)	IC50	0.8649	54	56
Glycogen synthase kinase-3 beta	Rattus norvegicus (Norway rat)	IC50	13.0443	4	19
Glycogen synthase kinase-3 beta	Homo sapiens (human)	Ki	0.0220	1	1
Guanine deaminase	Homo sapiens (human)	Ki	10.2000	1	1
HD2 type histone deacetylase HDA106	Zea mays	IC50	19.6974	11	13
HD2 type histone deacetylase HDA106	Zea mays	Ki	0.0044	2	2
heat shock 70kDa protein 1A	Homo sapiens (human)	IC50	66.9200	3	3
heat shock cognate 71 kDa protein isoform 1	Homo sapiens (human)	IC50	99.6000	2	2
heat shock cognate 71 kDa protein isoform 2	Homo sapiens (human)	IC50	99.6000	2	2
Heat shock factor protein 1	Homo sapiens (human)	IC50	50.0000	1	1
heat shock protein HSP 90-alpha isoform 2	Homo sapiens (human)	IC50	27.5411	2	3
Heat shock protein HSP 90-beta	Homo sapiens (human)	IC50	84.2500	2	2
Heme oxygenase 1	Rattus norvegicus (Norway rat)	IC50	14.0000	2	2
Heme oxygenase 2	Rattus norvegicus (Norway rat)	IC50	14.0000	2	2
Hepatocyte growth factor receptor	Homo sapiens (human)	IC50	11.3372	21	22
Hepatocyte growth factor receptor	Homo sapiens (human)	Ki	3.3000	1	1
hexokinase	Trypanosoma brucei brucei TREU927	IC50	11.2894	2	2
Hexokinase-4	Homo sapiens (human)	IC50	0.0006	2	2
High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A	Homo sapiens (human)	IC50	1.2843	7	7
High affinity nerve growth factor receptor	Homo sapiens (human)	IC50	125.2103	8	8
Histamine H1 receptor	Homo sapiens (human)	IC50	0.7499	7	11
Histamine H1 receptor	Rattus norvegicus (Norway rat)	IC50	0.0000	1	2
Histamine H1 receptor	Homo sapiens (human)	Ki	0.1426	5	9
Histamine H2 receptor	Cavia porcellus (domestic guinea pig)	IC50	1.7360	3	5
Histamine H2 receptor	Homo sapiens (human)	IC50	0.9915	1	2
Histamine H2 receptor	Homo sapiens (human)	Ki	0.9755	1	2
Histamine H3 receptor	Rattus norvegicus (Norway rat)	IC50	1.3000	1	2
Histamine H3 receptor	Homo sapiens (human)	Ki	0.0005	1	1
Histamine H4 receptor	Homo sapiens (human)	Ki	7.5060	1	2
Histidine-rich protein PFHRP-II	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	20,000.0000	1	1
Histone acetyltransferase KAT2B	Homo sapiens (human)	IC50	60.0000	2	2
Histone acetyltransferase KAT5	Homo sapiens (human)	IC50	70.0000	2	2
Histone acetyltransferase p300	Homo sapiens (human)	IC50	23.9375	8	8
Histone deacetylase	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	0.0006	1	1
Histone deacetylase	Rattus norvegicus (Norway rat)	IC50	0.1854	8	18
Histone deacetylase	Zea mays	IC50	0.0004	2	2
Histone deacetylase 1	Homo sapiens (human)	IC50	50.0277	120	144
Histone deacetylase 1	Mus musculus (house mouse)	IC50	0.0043	7	7
Histone deacetylase 1	Rattus norvegicus (Norway rat)	IC50	0.1854	8	9
Histone deacetylase 1	Homo sapiens (human)	Ki	39.4069	8	11
Histone deacetylase 1	Mus musculus (house mouse)	Ki	0.0011	1	1
Histone deacetylase 11	Mus musculus (house mouse)	IC50	0.0014	1	1
Histone deacetylase 11	Homo sapiens (human)	IC50	116.7613	45	60
Histone deacetylase 11	Homo sapiens (human)	Ki	76.6170	2	5
Histone deacetylase 2	Homo sapiens (human)	IC50	74.0666	71	95
Histone deacetylase 2	Mus musculus (house mouse)	IC50	0.0014	1	1
Histone deacetylase 2	Homo sapiens (human)	Ki	48.0361	7	10
Histone deacetylase 3	Homo sapiens (human)	IC50	79.5993	64	88
Histone deacetylase 3	Mus musculus (house mouse)	IC50	0.0014	1	1
Histone deacetylase 3	Rattus norvegicus (Norway rat)	IC50	0.1854	8	9
Histone deacetylase 3	Homo sapiens (human)	Ki	42.5207	6	9
Histone deacetylase 4	Homo sapiens (human)	IC50	86.8138	57	81
Histone deacetylase 4	Mus musculus (house mouse)	IC50	0.0014	1	1
Histone deacetylase 4	Rattus norvegicus (Norway rat)	IC50	0.1854	8	9
Histone deacetylase 4	Homo sapiens (human)	Ki	50.0539	5	8
Histone deacetylase 5	Homo sapiens (human)	IC50	107.6855	41	65
Histone deacetylase 5	Mus musculus (house mouse)	IC50	0.0107	2	2
Histone deacetylase 5	Homo sapiens (human)	Ki	55.3320	4	7
Histone deacetylase 6	Homo sapiens (human)	IC50	54.6875	104	128
Histone deacetylase 6	Mus musculus (house mouse)	IC50	0.0387	7	7
Histone deacetylase 6	Homo sapiens (human)	Ki	38.2691	7	10
Histone deacetylase 6	Rattus norvegicus (Norway rat)	IC50	0.1854	8	9
Histone deacetylase 7	Homo sapiens (human)	IC50	109.3349	40	64
Histone deacetylase 7	Mus musculus (house mouse)	IC50	0.0014	1	1
Histone deacetylase 7	Rattus norvegicus (Norway rat)	IC50	0.1854	8	9
Histone deacetylase 7	Homo sapiens (human)	Ki	63.8457	3	6
Histone deacetylase 8	Homo sapiens (human)	IC50	71.7342	75	99
Histone deacetylase 8	Mus musculus (house mouse)	IC50	0.0207	2	2
Histone deacetylase 8	Schistosoma mansoni	IC50	3.6200	1	1
Histone deacetylase 8	Homo sapiens (human)	Ki	40.7403	8	11
Histone deacetylase 9	Homo sapiens (human)	IC50	109.3930	40	64
Histone deacetylase 9	Mus musculus (house mouse)	IC50	0.0014	1	1
Histone deacetylase 9	Homo sapiens (human)	Ki	64.0473	3	6
Histone deacetylase-like amidohydrolase	Alcaligenaceae bacterium FB188	IC50	1.2000	1	1
Histone deacetylase-like amidohydrolase	Alcaligenaceae bacterium FB188	Ki	0.7000	1	1
Histone-lysine N-methyltransferase EHMT1	Homo sapiens (human)	IC50	100.0000	1	1
Histone-lysine N-methyltransferase EHMT2	Homo sapiens (human)	IC50	100.0000	1	1
Histone-lysine N-methyltransferase SETD7	Homo sapiens (human)	IC50	200.0000	1	1
Homeodomain-interacting protein kinase 1	Homo sapiens (human)	IC50	2.6390	1	1
Homeodomain-interacting protein kinase 2	Homo sapiens (human)	IC50	0.3655	2	2
Homeodomain-interacting protein kinase 3	Homo sapiens (human)	IC50	0.4560	2	2
Homeodomain-interacting protein kinase 4	Homo sapiens (human)	IC50	0.2260	2	2
Hyaluronate lyase	Streptococcus pneumoniae TIGR4	IC50	6,000.0000	1	1
Hyaluronidase-1	Homo sapiens (human)	IC50	1,272.5000	1	2
hypothetical protein SA1422	Staphylococcus aureus subsp. aureus N315	IC50	42.9000	2	2
Hypoxia-inducible factor 1-alpha	Homo sapiens (human)	IC50	50.2050	4	4
Hypoxia-inducible factor 1-alpha inhibitor	Homo sapiens (human)	IC50	10.2000	1	1
Ileal sodium/bile acid cotransporter	Homo sapiens (human)	Ki	24.0000	1	1
Inactive tyrosine-protein kinase PEAK1	Homo sapiens (human)	IC50	0.0025	2	2
Indoleamine 2,3-dioxygenase 1	Homo sapiens (human)	IC50	1.0000	2	2
Indoleamine 2,3-dioxygenase 1	Mus musculus (house mouse)	IC50	0.0060	1	2
Induced myeloid leukemia cell differentiation protein Mcl-1	Homo sapiens (human)	IC50	0.9200	1	1
Inhibitor of nuclear factor kappa-B kinase subunit alpha	Homo sapiens (human)	IC50	83.4387	6	6
Inhibitor of nuclear factor kappa-B kinase subunit beta	Homo sapiens (human)	IC50	46.0895	11	11
Inhibitor of nuclear factor kappa-B kinase subunit epsilon	Homo sapiens (human)	IC50	0.0003	2	2
Inositol hexakisphosphate kinase 2	Homo sapiens (human)	IC50	1.3000	1	3
Inositol polyphosphate multikinase	Homo sapiens (human)	IC50	2.6000	1	3
Insulin receptor	Homo sapiens (human)	IC50	12.5954	8	8
Insulin receptor	Mus musculus (house mouse)	IC50	0.2000	1	1
Insulin receptor	Homo sapiens (human)	Ki	2.6000	1	1
Insulin receptor	Rattus norvegicus (Norway rat)	IC50	0.0034	1	1
Insulin receptor-related protein	Homo sapiens (human)	IC50	0.0113	2	2
Insulin-degrading enzyme	Homo sapiens (human)	IC50	100.0000	1	1
Insulin-like growth factor 1 receptor	Homo sapiens (human)	IC50	29.9203	16	17
Integrase	Human immunodeficiency virus 1	IC50	19.1415	26	44
integrase, partial	Human immunodeficiency virus 1	IC50	0.9489	2	2
Integrin alpha-IIb	Homo sapiens (human)	IC50	35.0088	3	3
Integrin beta-3	Homo sapiens (human)	IC50	35.0088	3	3
Interferon-induced, double-stranded RNA-activated protein kinase	Homo sapiens (human)	IC50	4.0500	1	2
Interleukin-1 receptor-associated kinase 1	Homo sapiens (human)	IC50	0.0377	2	2
Interleukin-1 receptor-associated kinase 4	Homo sapiens (human)	IC50	0.0122	4	4
Interleukin-2	Mus musculus (house mouse)	IC50	0.0050	1	1
Interstitial collagenase	Homo sapiens (human)	IC50	2.2193	4	7
intestinal alkaline phosphatase precursor	Mus musculus (house mouse)	IC50	12.0900	1	4
Kappa-type opioid receptor	Cavia porcellus (domestic guinea pig)	IC50	1.3856	7	8
Kappa-type opioid receptor	Homo sapiens (human)	IC50	4.3708	4	4
Kappa-type opioid receptor	Mus musculus (house mouse)	IC50	0.0828	2	4
Kappa-type opioid receptor	Rattus norvegicus (Norway rat)	IC50	0.0545	8	9
Kappa-type opioid receptor	Cavia porcellus (domestic guinea pig)	Ki	4.6570	20	26
Kappa-type opioid receptor	Homo sapiens (human)	Ki	0.3356	27	27
Kappa-type opioid receptor	Mus musculus (house mouse)	Ki	0.9252	2	2
Kappa-type opioid receptor	Rattus norvegicus (Norway rat)	Ki	0.1130	2	2
Kinase suppressor of Ras 1	Homo sapiens (human)	IC50	6.2650	2	2
Kinase suppressor of Ras 2	Homo sapiens (human)	IC50	5.4000	2	2
Kinesin-1 heavy chain	Homo sapiens (human)	IC50	0.0015	1	1
Kynurenine 3-monooxygenase	Rattus norvegicus (Norway rat)	IC50	0.3000	1	1
L-selectin	Homo sapiens (human)	IC50	27.6000	1	1
Lactoperoxidase	Bos taurus (cattle)	IC50	6.1000	1	1
Lactoylglutathione lyase	Homo sapiens (human)	IC50	5.7229	4	7
Lactoylglutathione lyase	Homo sapiens (human)	Ki	9.4411	2	3
Lanosterol 14-alpha demethylase	Homo sapiens (human)	IC50	30.0000	1	1
large T antigen	Betapolyomavirus macacae	IC50	15.5443	1	7
lens epithelium-derived growth factor p75	Homo sapiens (human)	IC50	0.9489	2	2
Lethal factor	Bacillus anthracis	IC50	0.0970	1	1
Leucine-rich repeat serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	0.0076	3	3
Leukocyte tyrosine kinase receptor	Homo sapiens (human)	IC50	0.0173	3	3
Leukotriene A-4 hydrolase	Homo sapiens (human)	IC50	10.0000	2	4
Leukotriene B4 receptor 1	Homo sapiens (human)	IC50	0.0850	1	1
likely tRNA 2'-phosphotransferase	Candida albicans SC5314	IC50	0.2913	2	2
LIM domain kinase 1	Homo sapiens (human)	IC50	0.0026	2	2
LIM domain kinase 2	Homo sapiens (human)	IC50	0.0956	2	2
Linoleate 9S-lipoxygenase-4	Glycine max (soybean)	IC50	590.6667	2	3
Lipoxygenase	Glycine max (soybean)	IC50	23.3460	5	5
Lipoxygenase	Solanum tuberosum (potato)	IC50	5.6667	2	3
Liver carboxylesterase	Sus scrofa (pig)	IC50	250.0000	1	1
Liver carboxylesterase 1	Homo sapiens (human)	IC50	0.1000	1	1
Low molecular weight phosphotyrosine protein phosphatase	Homo sapiens (human)	IC50	9.1500	2	2
Luciferin 4-monooxygenase	Photinus pyralis (common eastern firefly)	IC50	36.7200	5	5
Lymphokine-activated killer T-cell-originated protein kinase	Homo sapiens (human)	IC50	0.0691	2	2
Lysine--tRNA ligase	Homo sapiens (human)	IC50	0.0049	2	2
Lysine-specific demethylase 4E	Homo sapiens (human)	IC50	408.6000	3	4
Lysine-specific demethylase 4E	Homo sapiens (human)	Ki	4.3300	1	1
Lysine-specific histone demethylase 1A	Homo sapiens (human)	IC50	10.4486	6	7
Lysine-specific histone demethylase 1A	Homo sapiens (human)	Ki	1.0000	1	1
Lysosomal alpha-glucosidase	Homo sapiens (human)	IC50	490.2108	13	13
Lysosomal alpha-glucosidase	Mus musculus (house mouse)	IC50	144.4700	1	2
Lysosomal alpha-glucosidase	Rattus norvegicus (Norway rat)	IC50	217.3450	2	2
Lysosomal protective protein	Homo sapiens (human)	IC50	0.6000	1	1
M-phase inducer phosphatase 2	Homo sapiens (human)	IC50	1.4900	1	2
M17 leucyl aminopeptidase	Plasmodium falciparum 3D7	IC50	72.7250	1	2
Macrophage colony-stimulating factor 1 receptor	Homo sapiens (human)	IC50	0.1269	7	9
Macrophage metalloelastase	Homo sapiens (human)	IC50	10.2300	1	1
Macrophage migration inhibitory factor	Homo sapiens (human)	IC50	4.7700	1	1
Macrophage migration inhibitory factor	Homo sapiens (human)	Ki	1.9500	1	1
Macrophage-stimulating protein receptor	Homo sapiens (human)	IC50	0.2195	5	5
Malate dehydrogenase	Thermus thermophilus	IC50	6.0000	1	1
Maltase-glucoamylase, intestinal	Homo sapiens (human)	IC50	319.9231	16	16
Maltase-glucoamylase, intestinal	Homo sapiens (human)	Ki	10.4000	1	1
Mannosyl-oligosaccharide glucosidase	Saccharomyces cerevisiae S288C	IC50	13.3400	1	1
MAP kinase-activated protein kinase 2	Homo sapiens (human)	IC50	0.7350	10	10
MAP kinase-activated protein kinase 3	Homo sapiens (human)	IC50	2.7750	2	2
MAP kinase-activated protein kinase 5	Homo sapiens (human)	IC50	0.4747	3	3
MAP kinase-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	IC50	0.2120	3	3
MAP kinase-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	0.0221	3	3
MAP/microtubule affinity-regulating kinase 3	Homo sapiens (human)	IC50	0.0004	2	2
MAP/microtubule affinity-regulating kinase 4	Homo sapiens (human)	IC50	0.0001	2	2
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	IC50	41.7011	12	12
Maternal embryonic leucine zipper kinase	Homo sapiens (human)	IC50	0.0006	2	2
Matrilysin	Homo sapiens (human)	IC50	34.6845	3	15
Matrix metalloproteinase-14	Homo sapiens (human)	IC50	6.8000	1	1
Matrix metalloproteinase-9	Homo sapiens (human)	IC50	0.3650	5	5
Mcl-1	Homo sapiens (human)	IC50	18.8652	2	3
Megakaryocyte-associated tyrosine-protein kinase	Homo sapiens (human)	IC50	0.4420	2	2
Melatonin receptor type 1A	Homo sapiens (human)	IC50	0.0025	18	18
Melatonin receptor type 1A	Gallus gallus (chicken)	Ki	0.0007	7	8
Melatonin receptor type 1A	Homo sapiens (human)	Ki	0.0003	67	69
Melatonin receptor type 1B	Homo sapiens (human)	IC50	0.0035	12	12
Melatonin receptor type 1B	Gallus gallus (chicken)	Ki	0.0007	8	9
Melatonin receptor type 1B	Homo sapiens (human)	Ki	0.0004	62	64
Melatonin receptor type 1C	Gallus gallus (chicken)	Ki	0.0007	7	8
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	Homo sapiens (human)	IC50	37.3000	4	4
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	Homo sapiens (human)	Ki	16.4885	4	5
Metabotropic glutamate receptor 1	Rattus norvegicus (Norway rat)	IC50	0.0044	4	4
Metallo-beta-lactamase VIM-13	Pseudomonas aeruginosa	IC50	252.6000	1	1
Microtubule-associated protein tau	Homo sapiens (human)	IC50	32.2143	6	7
Misshapen-like kinase 1	Homo sapiens (human)	IC50	0.0004	4	4
Mitogen-activated protein kinase 1	Homo sapiens (human)	IC50	40.9038	13	14
Mitogen-activated protein kinase 1	Rattus norvegicus (Norway rat)	IC50	500.0240	1	2
Mitogen-activated protein kinase 1	Mus musculus (house mouse)	IC50	10.0000	1	1
Mitogen-activated protein kinase 10	Homo sapiens (human)	IC50	9.3601	18	31
Mitogen-activated protein kinase 10	Homo sapiens (human)	Ki	0.0900	1	1
Mitogen-activated protein kinase 11	Homo sapiens (human)	IC50	3.7291	28	29
Mitogen-activated protein kinase 12	Homo sapiens (human)	IC50	4.0953	25	26
Mitogen-activated protein kinase 13	Homo sapiens (human)	IC50	4.0910	25	26
Mitogen-activated protein kinase 14	Homo sapiens (human)	IC50	20.8364	82	98
Mitogen-activated protein kinase 14	Homo sapiens (human)	Ki	0.0375	2	2
Mitogen-activated protein kinase 14	Mus musculus (house mouse)	IC50	0.0560	1	3
Mitogen-activated protein kinase 15	Homo sapiens (human)	IC50	0.0081	3	3
Mitogen-activated protein kinase 2	Pneumocystis carinii	IC50	0.1050	1	1
Mitogen-activated protein kinase 3	Homo sapiens (human)	IC50	9.9602	12	12
Mitogen-activated protein kinase 7	Homo sapiens (human)	IC50	5.9524	4	4
Mitogen-activated protein kinase 8	Homo sapiens (human)	IC50	4.4361	17	18
Mitogen-activated protein kinase 9	Homo sapiens (human)	IC50	1.7016	19	20
Mitogen-activated protein kinase kinase kinase 1	Homo sapiens (human)	IC50	0.4380	2	2
Mitogen-activated protein kinase kinase kinase 10	Homo sapiens (human)	IC50	0.1952	3	3
Mitogen-activated protein kinase kinase kinase 11	Homo sapiens (human)	IC50	0.0160	3	3
Mitogen-activated protein kinase kinase kinase 12	Homo sapiens (human)	IC50	0.0992	2	2
Mitogen-activated protein kinase kinase kinase 14	Homo sapiens (human)	IC50	2.3000	1	1
Mitogen-activated protein kinase kinase kinase 19	Homo sapiens (human)	IC50	0.0087	2	2
Mitogen-activated protein kinase kinase kinase 2	Homo sapiens (human)	IC50	0.0335	2	2
Mitogen-activated protein kinase kinase kinase 21	Homo sapiens (human)	IC50	1.1175	2	2
Mitogen-activated protein kinase kinase kinase 3	Homo sapiens (human)	IC50	0.0092	2	2
Mitogen-activated protein kinase kinase kinase 5	Homo sapiens (human)	IC50	0.2150	5	5
Mitogen-activated protein kinase kinase kinase 6	Homo sapiens (human)	IC50	0.2829	2	2
Mitogen-activated protein kinase kinase kinase 7	Homo sapiens (human)	IC50	0.0565	5	5
Mitogen-activated protein kinase kinase kinase 8	Homo sapiens (human)	IC50	2.3700	1	1
Mitogen-activated protein kinase kinase kinase 9	Homo sapiens (human)	IC50	0.0044	3	3
Mitogen-activated protein kinase kinase kinase kinase 3	Homo sapiens (human)	IC50	0.0001	2	2
Mitogen-activated protein kinase kinase kinase kinase 4	Homo sapiens (human)	IC50	0.0005	2	2
Mitogen-activated protein kinase kinase kinase kinase 5	Homo sapiens (human)	IC50	0.0002	2	2
MO15-related protein kinase Pfmrk	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	112.5714	3	7
Monocarboxylate transporter 1	Rattus norvegicus (Norway rat)	IC50	14.0000	1	1
Monocarboxylate transporter 2	Rattus norvegicus (Norway rat)	IC50	5.0000	1	1
mothers against decapentaplegic homolog 3 isoform 1	Homo sapiens (human)	IC50	0.1420	1	1
Mu-type opioid receptor	Cavia porcellus (domestic guinea pig)	IC50	3.6260	7	8
Mu-type opioid receptor	Homo sapiens (human)	IC50	1.5755	10	13
Mu-type opioid receptor	Mus musculus (house mouse)	IC50	0.3305	7	9
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	IC50	0.0385	11	13
Mu-type opioid receptor	Bos taurus (cattle)	Ki	0.0013	3	3
Mu-type opioid receptor	Cavia porcellus (domestic guinea pig)	Ki	0.0404	16	25
Mu-type opioid receptor	Danio rerio (zebrafish)	Ki	0.1872	2	2
Mu-type opioid receptor	Homo sapiens (human)	Ki	0.2222	33	36
Mu-type opioid receptor	Mus musculus (house mouse)	Ki	0.0801	4	6
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	Ki	1.7961	18	28
Multidrug and toxin extrusion protein 1	Homo sapiens (human)	IC50	375.0000	1	2
Multidrug resistance-associated protein 1	Homo sapiens (human)	IC50	5.0075	11	11
Multidrug resistance-associated protein 1	Homo sapiens (human)	Ki	5.1429	3	7
Multidrug resistance-associated protein 4	Homo sapiens (human)	IC50	113.1710	1	31
Muscarinic acetylcholine receptor M1	Homo sapiens (human)	IC50	3.9485	1	4
Muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	IC50	0.5700	1	4
Muscarinic acetylcholine receptor M1	Homo sapiens (human)	Ki	0.9510	1	4
Muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	Ki	0.0320	2	6
Muscarinic acetylcholine receptor M2	Homo sapiens (human)	IC50	1.8505	1	2
Muscarinic acetylcholine receptor M2	Rattus norvegicus (Norway rat)	IC50	0.5700	1	3
Muscarinic acetylcholine receptor M2	Homo sapiens (human)	Ki	0.6580	1	2
Muscarinic acetylcholine receptor M2	Rattus norvegicus (Norway rat)	Ki	0.0320	2	6
Muscarinic acetylcholine receptor M3	Homo sapiens (human)	IC50	5.4238	1	4
Muscarinic acetylcholine receptor M3	Rattus norvegicus (Norway rat)	IC50	0.5700	1	3
Muscarinic acetylcholine receptor M3	Homo sapiens (human)	Ki	1.1500	1	4
Muscarinic acetylcholine receptor M3	Rattus norvegicus (Norway rat)	Ki	0.0320	2	6
Muscarinic acetylcholine receptor M4	Homo sapiens (human)	IC50	2.4877	1	3
Muscarinic acetylcholine receptor M4	Rattus norvegicus (Norway rat)	IC50	0.5700	1	3
Muscarinic acetylcholine receptor M4	Homo sapiens (human)	Ki	0.3467	1	3
Muscarinic acetylcholine receptor M4	Rattus norvegicus (Norway rat)	Ki	0.0320	2	6
Muscarinic acetylcholine receptor M5	Homo sapiens (human)	IC50	0.6450	1	3
Muscarinic acetylcholine receptor M5	Rattus norvegicus (Norway rat)	IC50	0.9025	2	4
Muscarinic acetylcholine receptor M5	Homo sapiens (human)	Ki	0.4633	1	3
Muscarinic acetylcholine receptor M5	Rattus norvegicus (Norway rat)	Ki	0.0320	2	6
Muscle, skeletal receptor tyrosine-protein kinase	Homo sapiens (human)	IC50	0.1161	3	3
Myeloperoxidase	Homo sapiens (human)	IC50	30.2900	6	7
Myeloperoxidase	Homo sapiens (human)	Ki	0.0900	1	1
Myoglobin	Homo sapiens (human)	IC50	2.3000	1	1
Myosin light chain kinase 2, skeletal/cardiac muscle	Homo sapiens (human)	IC50	0.0147	2	2
Myosin light chain kinase 3	Homo sapiens (human)	IC50	0.1585	2	2
Myosin light chain kinase family member 4	Homo sapiens (human)	IC50	0.0537	2	2
Myosin light chain kinase, smooth muscle	Gallus gallus (chicken)	IC50	5.0300	2	2
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	IC50	5.6405	9	10
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	Ki	18.8500	2	2
Myosin-IIIa	Homo sapiens (human)	IC50	0.0425	2	2
Myosin-IIIb	Homo sapiens (human)	IC50	0.0058	2	2
Myotonin-protein kinase	Homo sapiens (human)	IC50	2.3368	4	4
N-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D	Homo sapiens (human)	IC50	68.0000	1	1
NACHT, LRR and PYD domains-containing protein 3	Homo sapiens (human)	IC50	11.9467	3	3
NAD kinase	Homo sapiens (human)	IC50	0.9600	1	1
NAD kinase	Homo sapiens (human)	Ki	3.2800	1	1
NAD-dependent histone deacetylase SIR2	Saccharomyces cerevisiae S288C	IC50	50.0000	1	1
NAD-dependent protein deacetylase	Schistosoma mansoni	IC50	221.5500	2	2
NAD-dependent protein deacetylase HST2	Saccharomyces cerevisiae S288C	IC50	91.0000	1	1
NAD-dependent protein deacetylase sirtuin-1	Homo sapiens (human)	IC50	130.9500	12	12
NAD-dependent protein deacetylase sirtuin-2	Homo sapiens (human)	IC50	33.0067	14	15
NAD-dependent protein deacetylase sirtuin-3, mitochondrial	Homo sapiens (human)	IC50	78.4571	7	7
NAD-dependent protein deacetylase sirtuin-6	Homo sapiens (human)	IC50	173.3500	4	4
NAD-dependent protein deacetylase sirtuin-6	Homo sapiens (human)	Ki	226.0000	2	2
NAD-dependent protein deacylase sirtuin-5, mitochondrial	Homo sapiens (human)	IC50	58.2000	3	3
NAD(+) hydrolase SARM1	Homo sapiens (human)	IC50	43.8000	1	1
NADPH oxidase 4	Homo sapiens (human)	IC50	0.6503	2	3
Neuraminidase	Influenza A virus (A/Puerto Rico/8/1934(H1N1))	IC50	7.7500	1	1
Neuraminidase	Influenza A virus (A/USSR/90/1977(H1N1))	IC50	174.2333	4	6
Neuraminidase	Influenza A virus (A/Wilson-Smith/1933(H1N1))	IC50	100.0000	1	1
Neuraminidase	Influenza A virus (A/Puerto Rico/8/1934(H1N1))	Ki	14.3000	1	1
Neuraminidase	Influenza A virus (A/RI/5+/1957(H2N2))	IC50	11.9000	1	1
Neuraminidase	Influenza A virus (A/Wilson-Smith/1933(H1N1))	IC50	62.0714	4	14
Neuraminidase	Influenza A virus (A/Wilson-Smith/1933(H1N1))	Ki	12.4500	1	2
Neuronal acetylcholine receptor subunit alpha-4	Rattus norvegicus (Norway rat)	IC50	14.1050	2	2
Neuronal acetylcholine receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Ki	0.0900	1	1
Neuronal acetylcholine receptor subunit beta-2	Rattus norvegicus (Norway rat)	IC50	14.1050	2	2
Neuronal acetylcholine receptor subunit beta-2	Rattus norvegicus (Norway rat)	Ki	0.0900	1	1
Neuronal proto-oncogene tyrosine-protein kinase Src	Mus musculus (house mouse)	IC50	2.2000	1	1
neutrophil cytosol factor 1	Homo sapiens (human)	IC50	50.0000	1	1
Neutrophil elastase	Homo sapiens (human)	IC50	8.8198	6	6
Neutrophil elastase	Homo sapiens (human)	Ki	11.9000	1	1
NF-kappa-B essential modulator	Homo sapiens (human)	IC50	500.0000	1	1
NH(3)-dependent NAD(+) synthetase	Bacillus subtilis subsp. subtilis str. 168	IC50	1.0000	1	1
Nicotinate phosphoribosyltransferase	Homo sapiens (human)	Ki	0.0005	1	1
Nitric oxide synthase, brain	Homo sapiens (human)	IC50	4.8900	2	2
Nitric oxide synthase, brain	Homo sapiens (human)	Ki	7.3000	1	1
Nitric oxide synthase, brain	Rattus norvegicus (Norway rat)	IC50	7.5500	2	2
Nitric oxide synthase, endothelial	Bos taurus (cattle)	IC50	611.3333	3	3
Nitric oxide synthase, endothelial	Homo sapiens (human)	IC50	485.0667	3	3
Nitric oxide synthase, inducible	Homo sapiens (human)	IC50	0.1395	3	3
Nitric oxide synthase, inducible	Mus musculus (house mouse)	IC50	13.3862	5	5
Nociceptin receptor	Cavia porcellus (domestic guinea pig)	Ki	0.0025	1	1
Nociceptin receptor	Mus musculus (house mouse)	Ki	0.0003	1	1
Non-receptor tyrosine-protein kinase TNK1	Homo sapiens (human)	IC50	0.0012	2	2
Non-receptor tyrosine-protein kinase TYK2	Homo sapiens (human)	IC50	0.0137	5	5
NT-3 growth factor receptor	Homo sapiens (human)	IC50	0.0002	2	2
NUAK family SNF1-like kinase 1	Homo sapiens (human)	IC50	0.9353	5	6
NUAK family SNF1-like kinase 2	Homo sapiens (human)	IC50	0.0018	2	2
Nuclear factor NF-kappa-B p100 subunit	Homo sapiens (human)	IC50	35.4250	3	4
Nuclear factor NF-kappa-B p105 subunit	Homo sapiens (human)	IC50	35.4250	3	4
Nuclear receptor corepressor 2	Homo sapiens (human)	IC50	0.0138	7	7
Nuclear receptor corepressor 2	Homo sapiens (human)	Ki	0.0006	2	2
Nuclear receptor ROR-gamma	Homo sapiens (human)	IC50	3.5333	3	3
nuclear receptor subfamily 0 group B member 1	Homo sapiens (human)	IC50	0.8335	1	1
Nuclear receptor subfamily 3 group C member 3	Bos taurus (cattle)	IC50	39.0866	1	1
Nuclear receptor subfamily 3 group C member 3	Bos taurus (cattle)	Ki	32.0228	1	1
Nucleophosmin	Homo sapiens (human)	IC50	40.0000	1	1
Oligo-1,6-glucosidase IMA1	Saccharomyces cerevisiae S288C	IC50	426.3364	10	11
Opioid receptor homologue	Danio rerio (zebrafish)	Ki	0.2230	1	1
Opioid receptor, delta 1b	Danio rerio (zebrafish)	Ki	1.4270	1	1
Ornithine decarboxylase	Homo sapiens (human)	IC50	26.0000	1	1
Oxysterols receptor LXR-alpha	Homo sapiens (human)	IC50	46.0000	3	4
Oxysterols receptor LXR-beta	Homo sapiens (human)	IC50	48.0000	2	3
P-selectin	Homo sapiens (human)	IC50	19.1000	1	1
P2X purinoceptor 7	Homo sapiens (human)	IC50	2.9150	2	2
P2X purinoceptor 7	Rattus norvegicus (Norway rat)	IC50	30.0000	1	1
P2Y purinoceptor 12	Rattus norvegicus (Norway rat)	IC50	0.0400	1	1
Palmitoleoyl-protein carboxylesterase NOTUM	Homo sapiens (human)	IC50	47.0000	2	2
Pancreatic alpha-amylase	Rattus norvegicus (Norway rat)	IC50	26.5000	1	1
Pancreatic alpha-amylase	Sus scrofa (pig)	IC50	11.0238	5	6
Pancreatic alpha-amylase	Rattus norvegicus (Norway rat)	Ki	43.4000	1	1
Pancreatic triacylglycerol lipase	Sus scrofa (pig)	IC50	344.2857	3	7
PAS domain-containing serine/threonine-protein kinase	Homo sapiens (human)	IC50	0.0107	2	2
Peptidyl-prolyl cis-trans isomerase A	Homo sapiens (human)	IC50	0.0252	12	12
Peptidyl-prolyl cis-trans isomerase A	Homo sapiens (human)	Ki	0.0645	8	8
Peptidyl-prolyl cis-trans isomerase B	Homo sapiens (human)	IC50	0.0088	1	1
Peptidyl-prolyl cis-trans isomerase D	Homo sapiens (human)	IC50	0.0036	1	1
Peptidyl-prolyl cis-trans isomerase D	Homo sapiens (human)	Ki	0.0129	4	4
Peptidyl-prolyl cis-trans isomerase FKBP1A	Homo sapiens (human)	IC50	0.0042	6	6
Peptidyl-prolyl cis-trans isomerase FKBP1A	Mus musculus (house mouse)	IC50	0.0010	1	1
Peptidyl-prolyl cis-trans isomerase FKBP1A	Homo sapiens (human)	Ki	1.0844	4	5
Peptidyl-prolyl cis-trans isomerase FKBP1B	Homo sapiens (human)	Ki	0.0060	1	1
Peptidyl-prolyl cis-trans isomerase FKBP4	Homo sapiens (human)	IC50	0.0160	1	1
Peptidyl-prolyl cis-trans isomerase FKBP5	Homo sapiens (human)	Ki	0.0030	1	1
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1	Homo sapiens (human)	IC50	11.2783	6	6
Peptidylglycine alpha-amidating monooxygenase	Rattus norvegicus (Norway rat)	Ki	0.0060	1	1
perilipin-1	Homo sapiens (human)	IC50	9.1670	1	1
perilipin-5	Homo sapiens (human)	IC50	10.2320	1	1
Peroxisome proliferator-activated receptor alpha	Homo sapiens (human)	IC50	5.5000	2	2
Peroxisome proliferator-activated receptor alpha	Mus musculus (house mouse)	IC50	1.1500	1	1
Peroxisome proliferator-activated receptor gamma	Homo sapiens (human)	IC50	5.3628	9	9
Peroxisome proliferator-activated receptor gamma	Mus musculus (house mouse)	IC50	0.7000	1	1
Peroxisome proliferator-activated receptor gamma	Rattus norvegicus (Norway rat)	IC50	0.7000	1	1
Peroxisome proliferator-activated receptor gamma	Homo sapiens (human)	Ki	0.5761	8	8
Phosphatidylinositol 3-kinase regulatory subunit alpha	Homo sapiens (human)	IC50	9,801.4342	7	15
Phosphatidylinositol 4-kinase alpha	Homo sapiens (human)	IC50	0.2800	1	1
Phosphatidylinositol 4-kinase beta	Homo sapiens (human)	IC50	0.4400	1	1
Phosphatidylinositol 4-kinase type 2-alpha	Homo sapiens (human)	IC50	30.0000	1	1
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha	Homo sapiens (human)	IC50	27.0000	1	1
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta	Homo sapiens (human)	IC50	2.1700	6	12
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Bos taurus (cattle)	IC50	3.7533	3	3
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	IC50	2,775.8826	38	53
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	Ki	3.0600	2	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Mus musculus (house mouse)	IC50	0.5000	2	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	IC50	3,870.1808	24	38
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	Homo sapiens (human)	IC50	5,446.1616	19	27
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Homo sapiens (human)	IC50	3,219.2033	24	47
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Mus musculus (house mouse)	IC50	0.5700	1	1
Phosphodiesterase	Bos taurus (cattle)	IC50	300.0000	1	1
Phosphodiesterase	Rattus norvegicus (Norway rat)	IC50	172.5000	2	2
Phosphoenolpyruvate carboxykinase, cytosolic [GTP]	Rattus norvegicus (Norway rat)	Ki	441.0000	1	1
Phosphoglycerate mutase 1	Homo sapiens (human)	IC50	0.4900	2	2
Phosphoinositide 3-kinase regulatory subunit 5	Homo sapiens (human)	IC50	0.8695	1	2
Phospholipase A2	Homo sapiens (human)	IC50	6.5500	2	2
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform	Homo sapiens (human)	IC50	0.0004	5	5
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform	Homo sapiens (human)	IC50	0.0017	3	3
Phosphorylase b kinase regulatory subunit alpha, liver isoform	Homo sapiens (human)	IC50	0.0005	1	1
Phosphorylase b kinase regulatory subunit alpha, skeletal muscle isoform	Homo sapiens (human)	IC50	0.0005	1	1
Phosphorylase b kinase regulatory subunit beta	Homo sapiens (human)	IC50	0.0005	1	1
photoreceptor-specific nuclear receptor	Homo sapiens (human)	IC50	3.6970	1	2
Plasma kallikrein	Homo sapiens (human)	IC50	0.0340	1	1
Plasminogen activator inhibitor 1	Homo sapiens (human)	IC50	3.3455	1	2
Platelet-activating factor receptor	Homo sapiens (human)	IC50	135.0000	1	1
Platelet-activating factor receptor	Cavia porcellus (domestic guinea pig)	Ki	73.3100	1	1
Platelet-derived growth factor receptor alpha	Homo sapiens (human)	IC50	51.0005	10	10
Platelet-derived growth factor receptor alpha	Mus musculus (house mouse)	IC50	26.4505	4	4
Platelet-derived growth factor receptor beta	Homo sapiens (human)	IC50	25.3663	18	22
Platelet-derived growth factor receptor beta	Mus musculus (house mouse)	IC50	22.2404	5	5
Poly [ADP-ribose] polymerase 1	Homo sapiens (human)	IC50	187.0070	6	7
Poly [ADP-ribose] polymerase 2	Mus musculus (house mouse)	IC50	129.5245	1	2
polyadenylate-binding protein 1	Homo sapiens (human)	IC50	50.8075	2	4
Polyamine deacetylase HDAC10	Homo sapiens (human)	IC50	94.4665	50	74
Polyamine deacetylase HDAC10	Mus musculus (house mouse)	IC50	0.0014	1	1
Polyamine deacetylase HDAC10	Homo sapiens (human)	Ki	63.7826	3	6
Polymerase acidic protein	Influenza A virus (A/Puerto Rico/8/1934(H1N1))	IC50	5.8600	1	1
Polypeptide N-acetylgalactosaminyltransferase 2	Homo sapiens (human)	IC50	1.6033	2	3
Polyphenol oxidase 2	Agaricus bisporus	IC50	219.0364	9	11
Polyunsaturated fatty acid 5-lipoxygenase	Homo sapiens (human)	IC50	10.5559	26	30
Polyunsaturated fatty acid 5-lipoxygenase	Mus musculus (house mouse)	IC50	0.4000	1	1
Polyunsaturated fatty acid 5-lipoxygenase	Rattus norvegicus (Norway rat)	IC50	10.0532	13	23
Polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	IC50	14.4117	6	12
Polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	Ki	1.6000	1	1
Polyunsaturated fatty acid lipoxygenase ALOX15	Homo sapiens (human)	IC50	12.8629	8	14
Polyunsaturated fatty acid lipoxygenase ALOX15	Oryctolagus cuniculus (rabbit)	IC50	11.4431	4	7
Polyunsaturated fatty acid lipoxygenase ALOX15	Homo sapiens (human)	Ki	0.6000	1	1
Polyunsaturated fatty acid lipoxygenase ALOX15B	Homo sapiens (human)	IC50	51.8542	4	12
Polyunsaturated fatty acid lipoxygenase ALOX15B	Rattus norvegicus (Norway rat)	IC50	0.2600	1	1
Potassium channel subfamily K member 9	Homo sapiens (human)	IC50	63.4000	1	1
Potassium voltage-gated channel subfamily A member 3	Homo sapiens (human)	IC50	0.7240	1	1
Potassium voltage-gated channel subfamily D member 3	Homo sapiens (human)	IC50	10,000.0000	1	1
Potassium voltage-gated channel subfamily E member 1	Homo sapiens (human)	IC50	129.2445	2	2
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	IC50	848.7223	17	23
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	Ki	28.5708	2	2
Potassium voltage-gated channel subfamily KQT member 1	Homo sapiens (human)	IC50	129.2445	2	2
Potassium-transporting ATPase alpha chain 1	Rattus norvegicus (Norway rat)	IC50	4.5000	1	1
Potassium-transporting ATPase subunit beta	Rattus norvegicus (Norway rat)	IC50	4.5000	1	1
Probable maltase-glucoamylase 2	Homo sapiens (human)	IC50	459.5782	11	11
Procathepsin L	Homo sapiens (human)	IC50	0.5600	1	1
Progesterone receptor	Homo sapiens (human)	IC50	8.0000	2	2
Prolyl 4-hydroxylase	Paramecium bursaria Chlorella virus 1	IC50	1,000.0000	1	2
Prolyl 4-hydroxylase subunit alpha-1	Gallus gallus (chicken)	Ki	26.0000	1	3
Prolyl endopeptidase	Homo sapiens (human)	IC50	107.2000	3	5
Prostaglandin E synthase	Homo sapiens (human)	IC50	1.3608	5	6
Prostaglandin G/H synthase 1	Canis lupus familiaris (dog)	IC50	5.5700	1	1
Prostaglandin G/H synthase 1	Homo sapiens (human)	IC50	56.4029	94	110
Prostaglandin G/H synthase 1	Mus musculus (house mouse)	IC50	3.2601	9	9
Prostaglandin G/H synthase 1	Ovis aries (sheep)	IC50	322.0180	174	242
Prostaglandin G/H synthase 1	Homo sapiens (human)	Ki	62.0000	1	1
Prostaglandin G/H synthase 1	Ovis aries (sheep)	Ki	9.0000	1	1
Prostaglandin G/H synthase 1	Bos taurus (cattle)	IC50	781.6859	10	17
Prostaglandin G/H synthase 1	Rattus norvegicus (Norway rat)	IC50	27.7310	7	10
Prostaglandin G/H synthase 2	Homo sapiens (human)	IC50	106.5275	204	250
Prostaglandin G/H synthase 2	Mus musculus (house mouse)	IC50	10.0878	19	20
Prostaglandin G/H synthase 2	Ovis aries (sheep)	IC50	120.3353	82	112
Prostaglandin G/H synthase 2	Homo sapiens (human)	Ki	17.3336	2	3
Prostaglandin G/H synthase 2	Ovis aries (sheep)	Ki	4.7450	2	2
Prostaglandin G/H synthase 2	Bos taurus (cattle)	IC50	603.0314	4	5
Prostaglandin G/H synthase 2	Rattus norvegicus (Norway rat)	IC50	21.2919	8	11
Prostaglandin-H2 D-isomerase	Mus musculus (house mouse)	IC50	1,500.0000	1	1
Protease	Human immunodeficiency virus 1	IC50	8.0000	1	1
Proteasome subunit beta type-5	Homo sapiens (human)	IC50	484.4817	9	15
Protein cereblon	Homo sapiens (human)	IC50	264.0000	1	1
Protein cereblon	Homo sapiens (human)	Ki	68,568.5000	2	2
Protein DBF4 homolog A	Homo sapiens (human)	IC50	0.0548	2	2
Protein disulfide-isomerase	Homo sapiens (human)	Ki	36.1000	1	1
Protein E6	Human papillomavirus 16	IC50	13.6167	1	3
Protein kinase C alpha type	Homo sapiens (human)	IC50	23.2597	25	32
Protein kinase C alpha type	Rattus norvegicus (Norway rat)	IC50	7.3590	14	14
Protein kinase C beta type	Homo sapiens (human)	IC50	7.2913	25	26
Protein kinase C beta type	Rattus norvegicus (Norway rat)	IC50	6.4402	16	16
Protein kinase C beta type	Rattus norvegicus (Norway rat)	Ki	0.0190	1	1
Protein kinase C delta type	Homo sapiens (human)	IC50	10.5513	18	18
Protein kinase C delta type	Rattus norvegicus (Norway rat)	IC50	8.5845	12	12
Protein kinase C epsilon type	Homo sapiens (human)	IC50	9.2965	21	21
Protein kinase C epsilon type	Rattus norvegicus (Norway rat)	IC50	8.5845	12	12
Protein kinase C eta type	Homo sapiens (human)	IC50	14.5511	13	13
Protein kinase C eta type	Rattus norvegicus (Norway rat)	IC50	8.5845	12	12
Protein kinase C gamma type	Homo sapiens (human)	IC50	9.0524	19	21
Protein kinase C gamma type	Rattus norvegicus (Norway rat)	IC50	6.8690	15	15
Protein kinase C iota type	Homo sapiens (human)	IC50	15.7971	12	12
Protein kinase C theta type	Homo sapiens (human)	IC50	14.5514	12	13
Protein kinase C theta type	Rattus norvegicus (Norway rat)	IC50	8.5845	12	12
Protein kinase C zeta type	Homo sapiens (human)	IC50	11.2815	16	18
Protein kinase C zeta type	Rattus norvegicus (Norway rat)	IC50	8.5845	12	12
Protein mono-ADP-ribosyltransferase PARP15	Homo sapiens (human)	IC50	15.0000	1	1
Protein odd-skipped-related 1	Homo sapiens (human)	IC50	0.0402	2	2
Protein-tyrosine kinase 2-beta	Homo sapiens (human)	IC50	0.0095	2	2
Protein-tyrosine kinase 6	Homo sapiens (human)	IC50	53.7872	5	5
Proteinase-activated receptor 1	Homo sapiens (human)	Ki	0.0022	1	1
Prothrombin	Homo sapiens (human)	IC50	15.7500	2	2
Prothrombin	Bos taurus (cattle)	IC50	19.1933	3	6
Prothrombin	Bos taurus (cattle)	Ki	3.9000	1	1
Proto-oncogene c-Fos	Homo sapiens (human)	IC50	0.0079	1	1
Proto-oncogene tyrosine-protein kinase LCK	Mus musculus (house mouse)	IC50	0.0310	1	1
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	IC50	8.4375	14	14
Proto-oncogene tyrosine-protein kinase ROS	Homo sapiens (human)	IC50	0.0004	6	6
Proto-oncogene tyrosine-protein kinase Src	Gallus gallus (chicken)	IC50	0.0212	2	2
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	IC50	8.3081	43	50
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	Ki	0.5000	2	2
Proton-coupled amino acid transporter 1	Homo sapiens (human)	Ki	5,550.0000	1	2
putative polyprotein		IC50	2.4395	2	2
Pyruvate kinase PKM	Homo sapiens (human)	IC50	43.4367	3	3
Quinolone resistance protein NorA	Staphylococcus aureus	IC50	40.0000	1	1
rac GTPase-activating protein 1 isoform a	Homo sapiens (human)	IC50	44.4900	1	1
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	IC50	2.7906	27	30
RAC-beta serine/threonine-protein kinase	Homo sapiens (human)	IC50	0.4119	8	10
RAC-gamma serine/threonine-protein kinase	Homo sapiens (human)	IC50	0.3701	9	11
RAF proto-oncogene serine/threonine-protein kinase	Homo sapiens (human)	IC50	1.6342	9	10
Receptor tyrosine-protein kinase erbB-2	Homo sapiens (human)	IC50	4.5405	14	14
Receptor tyrosine-protein kinase erbB-3	Homo sapiens (human)	IC50	0.0106	1	1
Receptor tyrosine-protein kinase erbB-4	Homo sapiens (human)	IC50	0.1830	8	8
Receptor-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	0.8198	10	11
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	IC50	2.1559	27	31
Receptor-type tyrosine-protein phosphatase alpha	Homo sapiens (human)	IC50	40.0000	1	1
Receptor-type tyrosine-protein phosphatase epsilon	Homo sapiens (human)	IC50	40.0000	1	1
Receptor-type tyrosine-protein phosphatase F	Homo sapiens (human)	IC50	21.9000	2	2
Receptor-type tyrosine-protein phosphatase S	Homo sapiens (human)	IC50	10.3000	1	1
Regulatory-associated protein of mTOR	Homo sapiens (human)	IC50	0.1500	2	3
Renin	Homo sapiens (human)	IC50	25.4900	2	2
Renin	Homo sapiens (human)	Ki	15.0000	1	1
Replicase polyprotein 1ab	Betacoronavirus England 1	IC50	10.0000	1	7
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	IC50	10.4433	12	24
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	IC50	33.1011	4	9
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	Ki	7.4000	1	1
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	Ki	7.4000	1	1
Retinoblastoma-associated protein	Homo sapiens (human)	IC50	0.0660	1	1
Reverse transcriptase/RNaseH	Human immunodeficiency virus 1	IC50	19.8628	15	16
Rho-associated protein kinase 1	Homo sapiens (human)	IC50	0.6897	15	15
Rho-associated protein kinase 1	Homo sapiens (human)	Ki	0.4300	6	7
Rho-associated protein kinase 2	Bos taurus (cattle)	IC50	0.9613	2	23
Rho-associated protein kinase 2	Homo sapiens (human)	IC50	1.0660	17	17
Rho-associated protein kinase 2	Rattus norvegicus (Norway rat)	IC50	67.3000	2	3
Rho-associated protein kinase 2	Homo sapiens (human)	Ki	0.3300	1	1
Rhodopsin kinase GRK1	Homo sapiens (human)	IC50	0.0680	2	2
Rhodopsin kinase GRK7	Homo sapiens (human)	IC50	0.0053	2	2
Rhomboid protease AarA	Providencia stuartii	IC50	16.8145	1	11
Rhomboid protease GlpG	Escherichia coli K-12	IC50	16.8145	1	11
Rhomboid protease GluP	Bacillus subtilis subsp. subtilis str. 168	IC50	16.8145	1	11
Rhomboid-related protein 1	Mus musculus (house mouse)	IC50	16.8145	1	11
Rhomboid-related protein 3	Mus musculus (house mouse)	IC50	16.8145	1	11
Ribosomal protein S6 kinase alpha-1	Homo sapiens (human)	IC50	0.0004	6	6
Ribosomal protein S6 kinase alpha-2	Homo sapiens (human)	IC50	0.0002	2	2
Ribosomal protein S6 kinase alpha-3	Homo sapiens (human)	IC50	0.0002	3	3
Ribosomal protein S6 kinase alpha-4	Homo sapiens (human)	IC50	0.0071	2	2
Ribosomal protein S6 kinase alpha-5	Homo sapiens (human)	IC50	1.2508	4	4
Ribosomal protein S6 kinase alpha-6	Homo sapiens (human)	IC50	0.0001	2	2
Ribosomal protein S6 kinase beta-1	Homo sapiens (human)	IC50	0.0007	4	4
Ribosomal protein S6 kinase beta-2	Homo sapiens (human)	IC50	0.0015	2	2
Ribosyldihydronicotinamide dehydrogenase [quinone]	Homo sapiens (human)	IC50	7.3161	8	8
Ribosyldihydronicotinamide dehydrogenase [quinone]	Homo sapiens (human)	Ki	0.0422	2	2
RNA polymerase beta subunit (EC 2.7.7.6), partial	Escherichia coli	IC50	18.1060	1	2
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1	Oryctolagus cuniculus (rabbit)	IC50	28.0000	4	6
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1	Oryctolagus cuniculus (rabbit)	Ki	5.8000	1	1
Sarcoplasmic/endoplasmic reticulum calcium ATPase 2	Homo sapiens (human)	IC50	6.0000	1	2
Sarcoplasmic/endoplasmic reticulum calcium ATPase 2	Homo sapiens (human)	Ki	53.0000	1	1
Sarcoplasmic/endoplasmic reticulum calcium ATPase 2	Rattus norvegicus (Norway rat)	Ki	5.8000	1	1
Sarcoplasmic/endoplasmic reticulum calcium ATPase 3	Homo sapiens (human)	IC50	6.0000	1	2
Sarcoplasmic/endoplasmic reticulum calcium ATPase 3	Homo sapiens (human)	Ki	8.6000	1	1
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	IC50	84.1875	11	16
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	Ki	106.7000	1	1
Seed linoleate 9S-lipoxygenase	Glycine max (soybean)	IC50	400.0000	1	1
Sentrin-specific protease 1	Homo sapiens (human)	IC50	1.2932	2	2
Serine-protein kinase ATM	Homo sapiens (human)	IC50	102.5000	4	4
Serine/threonine-protein kinase 10	Homo sapiens (human)	IC50	0.0080	2	2
Serine/threonine-protein kinase 16	Homo sapiens (human)	IC50	0.2385	2	2
Serine/threonine-protein kinase 17A	Homo sapiens (human)	IC50	0.0386	3	3
Serine/threonine-protein kinase 17B	Homo sapiens (human)	IC50	0.0258	1	1
Serine/threonine-protein kinase 24	Homo sapiens (human)	IC50	0.0065	3	3
Serine/threonine-protein kinase 25	Homo sapiens (human)	IC50	0.0029	3	3
Serine/threonine-protein kinase 26	Homo sapiens (human)	IC50	0.0124	2	2
Serine/threonine-protein kinase 3	Homo sapiens (human)	IC50	0.0034	4	4
Serine/threonine-protein kinase 32B	Homo sapiens (human)	IC50	0.0374	2	2
Serine/threonine-protein kinase 32C	Homo sapiens (human)	IC50	0.2320	2	2
Serine/threonine-protein kinase 33	Homo sapiens (human)	IC50	0.0373	2	2
Serine/threonine-protein kinase 36	Homo sapiens (human)	IC50	1.0000	1	1
Serine/threonine-protein kinase 38	Homo sapiens (human)	IC50	0.0037	2	2
Serine/threonine-protein kinase 38-like	Homo sapiens (human)	IC50	0.0012	2	2
Serine/threonine-protein kinase 4	Homo sapiens (human)	IC50	0.0013	2	2
Serine/threonine-protein kinase ATR	Homo sapiens (human)	IC50	327.5000	4	4
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	IC50	0.9236	12	13
Serine/threonine-protein kinase BRSK1	Homo sapiens (human)	IC50	0.0007	2	2
Serine/threonine-protein kinase BRSK2	Homo sapiens (human)	IC50	0.0028	2	2
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	IC50	38.6251	13	13
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	Ki	0.0078	1	1
Serine/threonine-protein kinase Chk2	Homo sapiens (human)	IC50	2.7191	10	10
Serine/threonine-protein kinase D1	Homo sapiens (human)	IC50	17.1962	11	11
Serine/threonine-protein kinase D2	Homo sapiens (human)	IC50	0.0014	2	2
Serine/threonine-protein kinase D3	Homo sapiens (human)	IC50	17.1961	11	11
Serine/threonine-protein kinase DCLK1	Homo sapiens (human)	IC50	0.2670	2	2
Serine/threonine-protein kinase DCLK2	Homo sapiens (human)	IC50	0.0890	2	2
Serine/threonine-protein kinase haspin	Homo sapiens (human)	IC50	0.0422	3	3
Serine/threonine-protein kinase ICK	Homo sapiens (human)	IC50	0.0443	3	3
Serine/threonine-protein kinase LATS1	Homo sapiens (human)	IC50	0.0130	2	2
Serine/threonine-protein kinase LATS2	Homo sapiens (human)	IC50	0.0062	2	2
Serine/threonine-protein kinase LMTK3	Homo sapiens (human)	IC50	0.0000	2	2
Serine/threonine-protein kinase MAK	Homo sapiens (human)	IC50	0.0257	2	2
Serine/threonine-protein kinase MARK1	Homo sapiens (human)	IC50	0.0003	2	2
Serine/threonine-protein kinase MARK2	Homo sapiens (human)	IC50	0.0001	2	2
Serine/threonine-protein kinase MRCK alpha	Homo sapiens (human)	IC50	0.0032	2	2
Serine/threonine-protein kinase MRCK beta	Homo sapiens (human)	IC50	0.0027	2	2
Serine/threonine-protein kinase MRCK gamma	Homo sapiens (human)	IC50	0.0005	2	2
Serine/threonine-protein kinase mTOR	Homo sapiens (human)	IC50	17.6314	24	26
Serine/threonine-protein kinase mTOR	Rattus norvegicus (Norway rat)	IC50	2.5000	1	1
Serine/threonine-protein kinase mTOR	Mus musculus (house mouse)	IC50	0.0000	1	1
Serine/threonine-protein kinase N1	Homo sapiens (human)	IC50	1.2517	5	6
Serine/threonine-protein kinase N2	Homo sapiens (human)	IC50	0.7975	7	7
Serine/threonine-protein kinase N3	Homo sapiens (human)	IC50	0.0105	2	2
Serine/threonine-protein kinase Nek1	Homo sapiens (human)	IC50	0.0122	3	3
Serine/threonine-protein kinase Nek11	Homo sapiens (human)	IC50	0.5210	2	2
Serine/threonine-protein kinase Nek2	Homo sapiens (human)	IC50	2.7588	3	4
Serine/threonine-protein kinase Nek3	Homo sapiens (human)	IC50	43.9500	2	2
Serine/threonine-protein kinase Nek4	Homo sapiens (human)	IC50	0.0851	2	2
Serine/threonine-protein kinase Nek5	Homo sapiens (human)	IC50	0.0864	2	2
Serine/threonine-protein kinase Nek6	Homo sapiens (human)	IC50	7.1150	1	2
Serine/threonine-protein kinase Nek8	Homo sapiens (human)	IC50	0.0263	2	2
Serine/threonine-protein kinase Nek9	Homo sapiens (human)	IC50	0.1010	2	2
Serine/threonine-protein kinase NIM1	Homo sapiens (human)	IC50	0.1102	2	2
Serine/threonine-protein kinase NLK	Homo sapiens (human)	IC50	0.3778	3	3
Serine/threonine-protein kinase PAK 1	Homo sapiens (human)	IC50	4.0003	4	4
Serine/threonine-protein kinase PAK 2	Homo sapiens (human)	IC50	0.0021	4	4
Serine/threonine-protein kinase PAK 3	Homo sapiens (human)	IC50	0.0003	2	2
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	IC50	0.0132	4	4
Serine/threonine-protein kinase PAK 5	Homo sapiens (human)	IC50	0.0039	2	2
Serine/threonine-protein kinase PAK 6	Homo sapiens (human)	IC50	0.0328	2	2
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	IC50	0.8516	21	29
Serine/threonine-protein kinase pim-2	Homo sapiens (human)	IC50	0.0813	5	5
Serine/threonine-protein kinase pim-3	Homo sapiens (human)	IC50	0.3501	4	4
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	IC50	17.9999	16	19
Serine/threonine-protein kinase PLK1	Xenopus laevis (African clawed frog)	IC50	21.4000	2	2
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	Ki	7.6187	1	13
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	IC50	45.3252	7	7
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	Ki	7.6187	1	13
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	IC50	51.5513	16	18
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	Ki	7.6187	1	13
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	IC50	0.9956	3	3
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	Ki	7.6187	1	13
Serine/threonine-protein kinase receptor R3	Homo sapiens (human)	IC50	0.8500	1	1
Serine/threonine-protein kinase SBK1	Homo sapiens (human)	IC50	0.1464	2	2
Serine/threonine-protein kinase Sgk1	Homo sapiens (human)	IC50	0.0100	3	3
Serine/threonine-protein kinase Sgk2	Homo sapiens (human)	IC50	0.0158	2	2
Serine/threonine-protein kinase Sgk3	Homo sapiens (human)	IC50	0.0730	2	2
Serine/threonine-protein kinase SIK1	Homo sapiens (human)	IC50	0.0009	2	2
Serine/threonine-protein kinase SIK2	Homo sapiens (human)	IC50	0.3669	3	3
Serine/threonine-protein kinase SIK3	Homo sapiens (human)	IC50	0.1541	3	3
Serine/threonine-protein kinase STK11	Homo sapiens (human)	IC50	0.0598	2	2
Serine/threonine-protein kinase TAO1	Homo sapiens (human)	IC50	0.0008	2	2
Serine/threonine-protein kinase TAO2	Homo sapiens (human)	IC50	0.0076	2	2
Serine/threonine-protein kinase TAO3	Homo sapiens (human)	IC50	0.0017	2	2
Serine/threonine-protein kinase TBK1	Homo sapiens (human)	IC50	0.0030	2	2
Serine/threonine-protein kinase tousled-like 1	Homo sapiens (human)	IC50	0.0295	3	3
Serine/threonine-protein kinase tousled-like 2	Homo sapiens (human)	IC50	0.0035	2	2
Serine/threonine-protein kinase ULK1	Homo sapiens (human)	IC50	0.0096	2	2
Serine/threonine-protein kinase ULK2	Homo sapiens (human)	IC50	0.0032	2	2
Serine/threonine-protein kinase ULK3	Homo sapiens (human)	IC50	0.0027	2	2
Serine/threonine-protein kinase WNK1	Homo sapiens (human)	IC50	14.8000	2	2
Serine/threonine-protein kinase WNK2	Homo sapiens (human)	IC50	1.4550	2	2
Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens (human)	IC50	0.3231	3	3
Serine/threonine-protein kinase/endoribonuclease IRE2	Homo sapiens (human)	IC50	0.0416	2	2
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform	Homo sapiens (human)	IC50	0.1830	1	1
Short transient receptor potential channel 5	Homo sapiens (human)	IC50	6.8000	1	3
Sialidase	Clostridium perfringens	IC50	9.9500	6	7
Sialidase-2	Homo sapiens (human)	IC50	210.0000	1	5
Sigma intracellular receptor 2	Rattus norvegicus (Norway rat)	IC50	0.0335	2	2
Sigma non-opioid intracellular receptor 1	Cavia porcellus (domestic guinea pig)	IC50	2.5156	4	4
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	IC50	0.0400	1	1
Sigma non-opioid intracellular receptor 1	Rattus norvegicus (Norway rat)	IC50	10.0000	1	1
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	Ki	50.0085	2	2
Signal transducer and activator of transcription 3	Homo sapiens (human)	IC50	24.8000	1	1
SNF-related serine/threonine-protein kinase	Homo sapiens (human)	IC50	0.0059	2	2
Sodium channel protein type 1 subunit alpha	Homo sapiens (human)	IC50	28.0000	2	2
Sodium channel protein type 1 subunit alpha	Rattus norvegicus (Norway rat)	IC50	82.6333	2	3
Sodium channel protein type 10 subunit alpha	Homo sapiens (human)	IC50	76.6667	3	3
Sodium channel protein type 11 subunit alpha	Homo sapiens (human)	IC50	36.0000	1	1
Sodium channel protein type 2 subunit alpha	Homo sapiens (human)	IC50	36.6000	5	5
Sodium channel protein type 2 subunit alpha	Rattus norvegicus (Norway rat)	IC50	63.5800	4	5
Sodium channel protein type 3 subunit alpha	Homo sapiens (human)	IC50	24.3333	3	3
Sodium channel protein type 3 subunit alpha	Rattus norvegicus (Norway rat)	IC50	82.6333	2	3
Sodium channel protein type 4 subunit alpha	Homo sapiens (human)	IC50	36.0000	1	1
Sodium channel protein type 4 subunit alpha	Homo sapiens (human)	Ki	17.0000	1	1
Sodium channel protein type 5 subunit alpha	Homo sapiens (human)	IC50	178.0490	6	6
Sodium channel protein type 7 subunit alpha	Homo sapiens (human)	IC50	36.0000	1	1
Sodium channel protein type 8 subunit alpha	Homo sapiens (human)	IC50	36.0000	1	1
Sodium channel protein type 9 subunit alpha	Homo sapiens (human)	IC50	26.5000	2	2
Sodium- and chloride-dependent betaine transporter	Rattus norvegicus (Norway rat)	IC50	43.3333	1	3
Sodium- and chloride-dependent creatine transporter 1	Homo sapiens (human)	IC50	5.0000	1	1
Sodium- and chloride-dependent GABA transporter 1	Rattus norvegicus (Norway rat)	IC50	43.3333	1	3
Sodium- and chloride-dependent GABA transporter 2	Rattus norvegicus (Norway rat)	IC50	43.3333	1	3
Sodium- and chloride-dependent GABA transporter 3	Rattus norvegicus (Norway rat)	IC50	43.3333	1	3
Sodium-dependent dopamine transporter	Rattus norvegicus (Norway rat)	IC50	10.0140	2	2
Sodium-dependent dopamine transporter	Rattus norvegicus (Norway rat)	Ki	0.1000	1	1
Sodium-dependent dopamine transporter	Homo sapiens (human)	IC50	6.0880	1	6
Sodium-dependent dopamine transporter	Homo sapiens (human)	Ki	4.8370	1	6
Sodium-dependent neutral amino acid transporter B(0)AT2	Homo sapiens (human)	IC50	4.0000	1	1
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	IC50	4.7285	2	8
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	Ki	5.3534	1	7
Sodium-dependent serotonin transporter	Homo sapiens (human)	IC50	4.2463	1	6
Sodium-dependent serotonin transporter	Rattus norvegicus (Norway rat)	IC50	1.1942	5	6
Sodium-dependent serotonin transporter	Homo sapiens (human)	Ki	1.6925	3	8
Sodium-dependent serotonin transporter	Rattus norvegicus (Norway rat)	Ki	3.0009	2	2
Sodium/bile acid cotransporter	Homo sapiens (human)	IC50	1.0000	1	1
Sodium/hydrogen exchanger 1	Rattus norvegicus (Norway rat)	IC50	33.1000	1	1
Solute carrier family 15 member 1	Homo sapiens (human)	IC50	9,750.0000	2	2
Solute carrier family 15 member 1	Rattus norvegicus (Norway rat)	Ki	6,150.0000	2	2
Solute carrier family 15 member 2	Homo sapiens (human)	IC50	28.0000	1	1
Solute carrier family 15 member 2	Rattus norvegicus (Norway rat)	Ki	66.0000	1	1
Solute carrier family 2, facilitated glucose transporter member 1	Homo sapiens (human)	IC50	4.0000	1	1
Solute carrier family 2, facilitated glucose transporter member 1	Homo sapiens (human)	Ki	7.0000	3	3
Solute carrier family 2, facilitated glucose transporter member 2	Homo sapiens (human)	IC50	12.0000	2	4
Solute carrier family 2, facilitated glucose transporter member 4	Mus musculus (house mouse)	IC50	20.0000	1	1
Solute carrier family 2, facilitated glucose transporter member 4	Rattus norvegicus (Norway rat)	Ki	24.7500	1	2
Solute carrier family 22 member 1	Homo sapiens (human)	IC50	669.9580	4	5
Solute carrier family 22 member 2	Homo sapiens (human)	IC50	882.5000	1	2
Solute carrier family 22 member 20	Mus musculus (house mouse)	Ki	10,304.7252	1	6
Solute carrier family 22 member 6	Homo sapiens (human)	IC50	4.1350	2	2
Solute carrier family 22 member 6	Mus musculus (house mouse)	Ki	435.8006	1	6
Solute carrier family 22 member 6	Rattus norvegicus (Norway rat)	Ki	1,132.6250	2	4
Solute carrier family 22 member 8	Homo sapiens (human)	Ki	1,170.0000	1	1
Solute carrier family 23 member 1	Homo sapiens (human)	IC50	156.0000	1	1
Solute carrier organic anion transporter family member 1A1	Rattus norvegicus (Norway rat)	Ki	72.1000	2	2
Solute carrier organic anion transporter family member 1A2	Homo sapiens (human)	Ki	51.0000	1	1
Solute carrier organic anion transporter family member 1A4	Rattus norvegicus (Norway rat)	Ki	810.9533	3	3
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	IC50	4.2449	8	16
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	Ki	3.5769	6	7
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	IC50	4.5430	2	4
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	Ki	2.6400	3	4
Solute carrier organic anion transporter family member 2B1	Homo sapiens (human)	IC50	51.0000	1	2
Solute carrier organic anion transporter family member 2B1	Homo sapiens (human)	Ki	49.5000	1	2
Sorbitol dehydrogenase	Homo sapiens (human)	IC50	106.3000	2	2
Sortase A	Streptococcus mutans	IC50	10.2000	1	1
Splicing factor 3B subunit 3	Homo sapiens (human)	IC50	0.5944	2	2
Squalene monooxygenase	Rattus norvegicus (Norway rat)	IC50	15.3700	3	5
SRSF protein kinase 1	Homo sapiens (human)	IC50	0.0336	2	2
SRSF protein kinase 2	Homo sapiens (human)	IC50	0.2060	2	2
SRSF protein kinase 3	Homo sapiens (human)	IC50	1.7700	2	2
STE20-like serine/threonine-protein kinase	Homo sapiens (human)	IC50	0.0142	3	3
STE20/SPS1-related proline-alanine-rich protein kinase	Homo sapiens (human)	IC50	0.0158	2	2
Steroid hormone receptor ERR1	Homo sapiens (human)	IC50	4.8250	2	2
Steroid hormone receptor ERR2	Homo sapiens (human)	IC50	0.3950	1	1
steroidogenic factor 1	Homo sapiens (human)	IC50	67.5180	1	1
Steryl-sulfatase	Homo sapiens (human)	IC50	0.8000	1	1
Stromelysin-1	Homo sapiens (human)	IC50	2.8255	2	2
Substance-K receptor	Cavia porcellus (domestic guinea pig)	IC50	69.1750	1	4
Substance-K receptor	Homo sapiens (human)	IC50	11.5967	1	3
Substance-K receptor	Homo sapiens (human)	Ki	3.8657	1	3
Substance-P receptor	Cavia porcellus (domestic guinea pig)	IC50	46.7000	2	6
Succinyl-diaminopimelate desuccinylase	Haemophilus influenzae Rd KW20	IC50	1,000.0000	1	1
Sucrase-isomaltase, intestinal	Homo sapiens (human)	IC50	395.5662	13	13
Sucrase-isomaltase, intestinal	Rattus norvegicus (Norway rat)	IC50	303.2750	6	6
Sulfotransferase 1A1	Homo sapiens (human)	Ki	80.0000	1	2
Sulfotransferase 2A1	Homo sapiens (human)	Ki	80.0000	1	2
SUMO-conjugating enzyme UBC9	Homo sapiens (human)	IC50	2.6800	2	2
SUMO1 activating enzyme subunit 1	Homo sapiens (human)	IC50	2.6800	2	2
Target of rapamycin complex subunit LST8	Homo sapiens (human)	IC50	0.1500	2	3
Tat	Human immunodeficiency virus 1	IC50	3.7800	1	2
Telomerase reverse transcriptase	Homo sapiens (human)	IC50	5.0278	23	23
Testis-specific serine/threonine-protein kinase 1	Homo sapiens (human)	IC50	0.0000	2	2
Testis-specific serine/threonine-protein kinase 1	Mus musculus (house mouse)	IC50	0.0003	1	1
Testis-specific serine/threonine-protein kinase 2	Homo sapiens (human)	IC50	0.0038	2	2
Testis-specific serine/threonine-protein kinase 3	Homo sapiens (human)	IC50	0.0051	2	2
Testis-specific serine/threonine-protein kinase 6	Homo sapiens (human)	IC50	0.1525	2	2
Testosterone 17-beta-dehydrogenase 3	Homo sapiens (human)	IC50	71.6840	2	5
TGF-beta receptor type-1	Homo sapiens (human)	IC50	8.5057	5	9
TGF-beta-activated kinase 1 and MAP3K7-binding protein 1	Homo sapiens (human)	IC50	0.0370	2	2
Thioredoxin glutathione reductase	Schistosoma mansoni	IC50	5.6500	2	2
Thioredoxin reductase 1, cytoplasmic	Homo sapiens (human)	IC50	70.7205	7	7
Thioredoxin reductase 1, cytoplasmic	Rattus norvegicus (Norway rat)	IC50	400.0000	1	1
Thioredoxin reductase 2, mitochondrial	Homo sapiens (human)	IC50	82.5000	6	6
Thioredoxin reductase 3	Homo sapiens (human)	IC50	82.5000	6	6
Thiosulfate sulfurtransferase	Homo sapiens (human)	IC50	60.6883	2	6
Thromboxane-A synthase	Homo sapiens (human)	IC50	336.0713	2	3
Tissue alpha-L-fucosidase	Bos taurus (cattle)	IC50	54.0000	1	1
Tissue factor	Homo sapiens (human)	IC50	300.0237	8	10
Tissue factor	Homo sapiens (human)	Ki	8,000.0000	1	1
Tissue-type plasminogen activator	Homo sapiens (human)	IC50	3.3455	1	2
Toll-like receptor 2	Mus musculus (house mouse)	IC50	69.2500	1	1
toll-like receptor 9	Homo sapiens (human)	IC50	8.3620	1	1
TPA: protein transporter TIM10	Saccharomyces cerevisiae S288C	IC50	56.2214	3	7
TPA: protein transporter TIM23	Saccharomyces cerevisiae S288C	IC50	5.0700	1	2
TRAF2 and NCK-interacting protein kinase	Homo sapiens (human)	IC50	0.2083	5	5
transactivating tegument protein VP16 [Human herpesvirus 1]	Human alphaherpesvirus 1 (Herpes simplex virus type 1)	IC50	3.2530	1	2
Transcription factor AP-1	Homo sapiens (human)	IC50	5.4160	3	3
Transcription factor p65	Homo sapiens (human)	IC50	28.3462	4	5
Transient receptor potential cation channel subfamily V member 2	Rattus norvegicus (Norway rat)	IC50	3.6000	2	2
Translin-associated protein X	Homo sapiens (human)	IC50	3.5000	1	1
Transporter	Rattus norvegicus (Norway rat)	IC50	0.0220	1	2
Transporter	Rattus norvegicus (Norway rat)	Ki	0.1010	1	1
Transthyretin	Homo sapiens (human)	IC50	7.8000	1	1
Transthyretin	Homo sapiens (human)	Ki	0.0026	1	1
Trehalose-phosphatase	Brugia malayi	Ki	10,000.0000	1	1
Triosephosphate isomerase	Oryctolagus cuniculus (rabbit)	Ki	123.0000	1	1
Trypsin-1	Homo sapiens (human)	IC50	9.5500	2	2
Trypsin-2	Homo sapiens (human)	IC50	9.5500	2	2
Trypsin-3	Homo sapiens (human)	IC50	9.5500	2	2
Type-1 angiotensin II receptor	Homo sapiens (human)	IC50	0.1246	1	1
Type-1 angiotensin II receptor	Oryctolagus cuniculus (rabbit)	IC50	0.5000	1	1
Type-1 angiotensin II receptor	Sus scrofa (pig)	IC50	0.0480	1	1
Type-2 angiotensin II receptor	Rattus norvegicus (Norway rat)	IC50	0.7050	2	2
Type-2 angiotensin II receptor	Rattus norvegicus (Norway rat)	Ki	0.5000	1	1
Tyrosinase	Homo sapiens (human)	IC50	32.9983	5	6
Tyrosinase	Mus musculus (house mouse)	IC50	250.0170	2	2
Tyrosine-protein kinase ABL1	Homo sapiens (human)	IC50	33.1106	21	28
Tyrosine-protein kinase ABL1	Homo sapiens (human)	Ki	0.5000	1	1
Tyrosine-protein kinase ABL2	Homo sapiens (human)	IC50	8.6181	6	7
Tyrosine-protein kinase Blk	Homo sapiens (human)	IC50	0.0011	2	2
Tyrosine-protein kinase BTK	Homo sapiens (human)	IC50	3.3486	12	12
Tyrosine-protein kinase BTK	Mus musculus (house mouse)	IC50	2.5000	1	1
Tyrosine-protein kinase CSK	Homo sapiens (human)	IC50	30.1085	5	12
Tyrosine-protein kinase Fer	Homo sapiens (human)	IC50	0.0008	3	3
Tyrosine-protein kinase Fes/Fps	Homo sapiens (human)	IC50	0.0039	3	3
Tyrosine-protein kinase Fgr	Homo sapiens (human)	IC50	0.0009	2	2
Tyrosine-protein kinase Fgr	Rattus norvegicus (Norway rat)	IC50	3.5000	1	1
Tyrosine-protein kinase FRK	Homo sapiens (human)	IC50	0.0108	2	2
Tyrosine-protein kinase Fyn	Homo sapiens (human)	IC50	23.5307	15	21
Tyrosine-protein kinase Fyn	Homo sapiens (human)	Ki	8.8500	2	2
Tyrosine-protein kinase HCK	Homo sapiens (human)	IC50	0.0033	3	3
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	IC50	5.3379	3	3
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	Ki	0.0061	1	2
Tyrosine-protein kinase JAK1	Homo sapiens (human)	IC50	0.5666	6	6
Tyrosine-protein kinase JAK2	Homo sapiens (human)	IC50	4,209.1678	12	12
Tyrosine-protein kinase JAK3	Homo sapiens (human)	IC50	4,412,933,333.4466	18	18
Tyrosine-protein kinase Lck	Homo sapiens (human)	IC50	9.1468	28	29
Tyrosine-protein kinase Lck	Homo sapiens (human)	Ki	0.0008	1	1
Tyrosine-protein kinase Lyn	Homo sapiens (human)	IC50	0.0311	14	14
Tyrosine-protein kinase Lyn	Rattus norvegicus (Norway rat)	IC50	7.5000	1	1
Tyrosine-protein kinase Mer	Homo sapiens (human)	IC50	0.0331	3	3
Tyrosine-protein kinase receptor TYRO3	Homo sapiens (human)	IC50	0.0177	3	3
Tyrosine-protein kinase receptor UFO	Homo sapiens (human)	IC50	0.1709	5	6
Tyrosine-protein kinase Srms	Homo sapiens (human)	IC50	6.5000	2	2
Tyrosine-protein kinase SYK	Homo sapiens (human)	IC50	6.7618	15	19
Tyrosine-protein kinase Tec	Homo sapiens (human)	IC50	42.6892	3	3
Tyrosine-protein kinase transforming protein Fps	Fujinami sarcoma virus	Ki	1.8000	1	1
Tyrosine-protein kinase TXK	Homo sapiens (human)	IC50	0.0204	2	2
Tyrosine-protein kinase Yes	Homo sapiens (human)	IC50	83.8853	6	6
Tyrosine-protein kinase Yes	Homo sapiens (human)	Ki	3.6210	1	2
Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	IC50	10,005.0140	10	10
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	IC50	15.2362	45	47
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	Ki	469.9333	3	3
Tyrosine-protein phosphatase non-receptor type 2	Homo sapiens (human)	IC50	7.8000	5	5
Tyrosine-protein phosphatase non-receptor type 6	Homo sapiens (human)	IC50	25.7800	1	1
Tyrosine-protein phosphatase non-receptor type 7	Homo sapiens (human)	IC50	100.0000	1	1
Tyrosine-protein phosphatase YopH	Yersinia enterocolitica	IC50	379.0000	1	1
Tyrosine-protein phosphatase YopH	Yersinia enterocolitica	Ki	40.4000	2	2
Tyrosyl-DNA phosphodiesterase 1	Homo sapiens (human)	IC50	194.0000	2	2
Ubiquitin carboxyl-terminal hydrolase 2	Homo sapiens (human)	IC50	31.5500	2	2
Ubiquitin carboxyl-terminal hydrolase 47	Homo sapiens (human)	IC50	26.0000	1	1
Ubiquitin carboxyl-terminal hydrolase 7	Homo sapiens (human)	IC50	7.0000	1	1
Ubiquitin-like modifier activating enzyme 2	Homo sapiens (human)	IC50	2.6800	2	2
UDP-glucuronosyltransferase 1-6	Homo sapiens (human)	IC50	211.8333	1	6
UDP-glucuronosyltransferase 1A1	Homo sapiens (human)	IC50	160.3000	3	8
UDP-glucuronosyltransferase 1A4	Homo sapiens (human)	IC50	211.8333	1	6
UDP-glucuronosyltransferase 2B10	Homo sapiens (human)	IC50	211.8333	1	6
UDP-glucuronosyltransferase 2B7	Homo sapiens (human)	IC50	211.8333	1	6
unnamed protein product	Aspergillus oryzae RIB40	IC50	52.7195	2	2
Urease	Canavalia ensiformis (jack bean)	IC50	8.5900	1	1
Urease subunit alpha	Helicobacter pylori 26695	IC50	81.1000	3	4
Urease subunit alpha	Helicobacter pylori 26695	Ki	9.3400	1	1
Urease subunit beta	Helicobacter pylori 26695	IC50	81.1000	3	4
Urease subunit beta	Helicobacter pylori 26695	Ki	9.3400	1	1
Urokinase-type plasminogen activator	Homo sapiens (human)	IC50	19.1130	3	7
Urokinase-type plasminogen activator	Mus musculus (house mouse)	IC50	3.3455	1	2
Urotensin-2 receptor	Rattus norvegicus (Norway rat)	IC50	3.9500	1	4
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	IC50	0.0149	7	7
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	IC50	3.5209	40	45
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	Ki	0.0017	1	1
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	IC50	0.1672	10	10
Vasopressin V2 receptor	Homo sapiens (human)	IC50	20.3282	3	6
Vif	Human immunodeficiency virus 1	IC50	4.0600	1	2
Vitamin D3 receptor	Homo sapiens (human)	IC50	15.1185	3	4
Voltage-dependent L-type calcium channel subunit alpha-1C	Cavia porcellus (domestic guinea pig)	IC50	36.0000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1C	Homo sapiens (human)	IC50	571.0501	5	5
Voltage-dependent L-type calcium channel subunit alpha-1C	Mus musculus (house mouse)	IC50	50.0000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1C	Rattus norvegicus (Norway rat)	IC50	50.0006	2	2
Voltage-dependent L-type calcium channel subunit alpha-1C	Homo sapiens (human)	Ki	0.0002	1	1
Voltage-dependent L-type calcium channel subunit alpha-1D	Mus musculus (house mouse)	IC50	50.0000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1D	Rattus norvegicus (Norway rat)	IC50	50.0006	2	2
Voltage-dependent L-type calcium channel subunit alpha-1D	Homo sapiens (human)	IC50	3.8101	3	3
Voltage-dependent L-type calcium channel subunit alpha-1F	Homo sapiens (human)	IC50	3.8101	3	3
Voltage-dependent L-type calcium channel subunit alpha-1F	Mus musculus (house mouse)	IC50	50.0000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1S	Homo sapiens (human)	IC50	3.8101	3	3
Voltage-dependent L-type calcium channel subunit alpha-1S	Mus musculus (house mouse)	IC50	50.0000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1S	Rattus norvegicus (Norway rat)	IC50	50.0006	2	2
Voltage-dependent N-type calcium channel subunit alpha-1B	Homo sapiens (human)	IC50	27.0000	1	1
Voltage-dependent T-type calcium channel subunit alpha-1I	Homo sapiens (human)	IC50	5,000.0000	1	1
Xanthine dehydrogenase/oxidase	Bos taurus (cattle)	IC50	22.8900	6	7
Xanthine dehydrogenase/oxidase	Homo sapiens (human)	IC50	110.8408	6	12
Xanthine dehydrogenase/oxidase	Bos taurus (cattle)	Ki	1.2000	1	1
Xanthine dehydrogenase/oxidase	Homo sapiens (human)	Ki	0.2800	1	1

Activation Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
2-dehydropantoate 2-reductase	Escherichia coli K-12	Kd	6,900.0000	1	1
26S proteasome regulatory subunit 6B	Homo sapiens (human)	Kd	30.0000	1	5
3-phosphoinositide-dependent protein kinase 1	Homo sapiens (human)	Kd	4.2507	3	5
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	EC50	50.0019	2	4
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	Kd	0.3981	1	1
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	Kd	0.1622	1	2
5-hydroxytryptamine receptor 2A	Mus musculus (house mouse)	EC50	16.8059	1	2
5-hydroxytryptamine receptor 2C	Homo sapiens (human)	EC50	0.0004	1	1
5-hydroxytryptamine receptor 4	Cavia porcellus (domestic guinea pig)	EC50	45.0000	1	3
5-hydroxytryptamine receptor 4	Homo sapiens (human)	EC50	10.0000	1	1
5-hydroxytryptamine receptor 7	Homo sapiens (human)	EC50	0.0006	1	1
5'-AMP-activated protein kinase catalytic subunit alpha-1	Homo sapiens (human)	Kd	17.0016	4	10
5'-AMP-activated protein kinase catalytic subunit alpha-2	Homo sapiens (human)	Kd	5.0060	2	4
5'-AMP-activated protein kinase subunit gamma-1	Homo sapiens (human)	Kd	30.0000	1	4
5'-AMP-activated protein kinase subunit gamma-2	Homo sapiens (human)	Kd	30.0000	1	4
AarF domain-containing protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	4
Actin-related protein 2	Homo sapiens (human)	Kd	30.0000	1	4
Actin-related protein 3	Homo sapiens (human)	Kd	30.0000	1	4
Activated CDC42 kinase 1	Homo sapiens (human)	Kd	17.0049	4	10
Activin receptor type-1	Homo sapiens (human)	Kd	17.6175	3	8
Activin receptor type-1B	Homo sapiens (human)	Kd	15.9200	3	8
Activin receptor type-2A	Homo sapiens (human)	Kd	9.7250	2	4
Activin receptor type-2B	Homo sapiens (human)	Kd	18.6500	3	8
Acyl-CoA dehydrogenase family member 10	Homo sapiens (human)	Kd	30.0000	1	4
Acyl-CoA dehydrogenase family member 11	Homo sapiens (human)	Kd	30.0000	1	4
Adenine phosphoribosyltransferase	Homo sapiens (human)	Kd	30.0000	1	4
Adenosine kinase	Homo sapiens (human)	Kd	30.0000	1	5
Adenosine receptor A1	Homo sapiens (human)	Kd	45.0000	1	1
Adenosine receptor A2a	Homo sapiens (human)	Kd	15.3144	2	2
Adenylate kinase 2, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	4
ADP/ATP translocase 2	Homo sapiens (human)	Kd	30.0000	1	4
ADP/ATP translocase 3	Homo sapiens (human)	Kd	30.0000	1	4
Albumin	Homo sapiens (human)	Kd	43.0000	3	3
Albumin	Rattus norvegicus (Norway rat)	Kd	1.4700	1	1
ALK tyrosine kinase receptor	Homo sapiens (human)	Kd	5.0160	2	4
alkaline phosphatase, germ cell type preproprotein	Homo sapiens (human)	EC50	32.3000	1	1
alkaline phosphatase, intestinal	Homo sapiens (human)	EC50	100.0000	1	1
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	1.9740	2	2
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	1.9740	2	2
Alpha-1D adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	1.9740	2	2
Alpha-2A adrenergic receptor	Homo sapiens (human)	EC50	0.0030	1	1
Alpha-2A adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	1.0958	2	2
Alpha-2B adrenergic receptor	Homo sapiens (human)	EC50	0.0005	1	1
Alpha-2B adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	1.0958	2	2
Alpha-2C adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	1.0958	2	2
Alpha-synuclein	Homo sapiens (human)	Kd	3.5000	4	4
Amine oxidase [flavin-containing] A	Homo sapiens (human)	EC50	1.6000	1	1
Amine oxidase [flavin-containing] B	Homo sapiens (human)	Kd	0.0589	1	1
amino acid transporter AGP1	Saccharomyces cerevisiae S288C	EC50	10.8000	1	1
Amyloid-beta precursor protein	Homo sapiens (human)	EC50	5,072.3200	4	5
Angiopoietin-1 receptor	Homo sapiens (human)	Kd	4.1040	3	5
Angiotensin-converting enzyme 2	Homo sapiens (human)	EC50	83.4000	1	1
Ankyrin repeat and protein kinase domain-containing protein 1	Homo sapiens (human)	Kd	5.1350	2	4
AP2-associated protein kinase 1	Homo sapiens (human)	Kd	14.0039	4	10
ATP-dependent 6-phosphofructokinase, platelet type	Homo sapiens (human)	Kd	30.0000	1	4
ATP-dependent RNA helicase DDX1	Homo sapiens (human)	Kd	30.0000	1	5
ATP-dependent RNA helicase DDX3X	Homo sapiens (human)	Kd	30.0000	1	4
ATP-dependent RNA helicase DDX42	Homo sapiens (human)	Kd	30.0000	1	3
ATP-dependent RNA helicase DHX30	Homo sapiens (human)	Kd	30.0000	1	6
ATP-dependent translocase ABCB1	Homo sapiens (human)	EC50	30.6486	10	10
ATP-dependent translocase ABCB1	Homo sapiens (human)	Kd	13.3810	1	3
ATP-dependent translocase ABCB1	Mus musculus (house mouse)	Kd	6.7000	1	1
Atypical kinase COQ8A, mitochondrial	Homo sapiens (human)	Kd	20.0000	3	8
Atypical kinase COQ8B, mitochondrial	Homo sapiens (human)	Kd	6.5500	2	4
Aurora kinase A	Homo sapiens (human)	Kd	14.1123	4	10
Aurora kinase B	Homo sapiens (human)	Kd	17.5048	3	8
Aurora kinase C	Homo sapiens (human)	Kd	4.2262	3	6
bcl-2-like protein 11 isoform 1	Homo sapiens (human)	EC50	350.0000	1	1
BDNF/NT-3 growth factors receptor	Homo sapiens (human)	Kd	5.0019	2	4
Beta-1 adrenergic receptor	Homo sapiens (human)	Kd	1.7790	2	4
Beta-1 adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	0.0229	3	3
Beta-1 adrenergic receptor	Cavia porcellus (domestic guinea pig)	Kd	0.2513	3	3
Beta-2 adrenergic receptor	Cavia porcellus (domestic guinea pig)	Kd	0.1622	3	4
Beta-2 adrenergic receptor	Homo sapiens (human)	Kd	4.5460	3	5
Beta-3 adrenergic receptor	Homo sapiens (human)	Kd	2.3667	1	3
Beta-adrenergic receptor kinase 1	Homo sapiens (human)	Kd	30.0000	1	5
Bile acid receptor	Homo sapiens (human)	EC50	42.2333	3	3
BMP-2-inducible protein kinase	Homo sapiens (human)	Kd	14.3828	4	10
Bone morphogenetic protein receptor type-1A	Homo sapiens (human)	Kd	18.4250	3	8
Bone morphogenetic protein receptor type-1B	Homo sapiens (human)	Kd	20.5783	2	6
Bone morphogenetic protein receptor type-2	Homo sapiens (human)	Kd	19.0375	3	8
Breakpoint cluster region protein	Homo sapiens (human)	Kd	30.0000	1	4
Broad substrate specificity ATP-binding cassette transporter ABCG2	Homo sapiens (human)	EC50	0.5840	4	4
C-terminal-binding protein 1	Homo sapiens (human)	Kd	2.2129	1	7
Calcium-dependent protein kinase 1	Plasmodium falciparum 3D7	Kd	0.4251	1	2
Calcium/calmodulin-dependent protein kinase kinase 1	Homo sapiens (human)	Kd	4.0000	3	5
Calcium/calmodulin-dependent protein kinase kinase 2	Homo sapiens (human)	Kd	14.7500	4	10
Calcium/calmodulin-dependent protein kinase type 1	Homo sapiens (human)	Kd	4.0307	3	6
Calcium/calmodulin-dependent protein kinase type 1D	Homo sapiens (human)	Kd	3.5674	3	6
Calcium/calmodulin-dependent protein kinase type 1G	Homo sapiens (human)	Kd	7.7570	4	7
Calcium/calmodulin-dependent protein kinase type II subunit alpha	Homo sapiens (human)	Kd	4.0001	3	5
Calcium/calmodulin-dependent protein kinase type II subunit beta	Homo sapiens (human)	Kd	4.0011	3	5
Calcium/calmodulin-dependent protein kinase type II subunit delta	Homo sapiens (human)	Kd	17.0001	4	10
Calcium/calmodulin-dependent protein kinase type II subunit gamma	Homo sapiens (human)	Kd	15.5557	4	9
Calcium/calmodulin-dependent protein kinase type IV	Homo sapiens (human)	Kd	20.0082	3	10
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	Kd	18.8931	3	9
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	Kd	17.5072	3	8
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	Kd	30.0000	1	3
cAMP-dependent protein kinase catalytic subunit PRKX	Homo sapiens (human)	Kd	5.0065	2	4
cAMP-dependent protein kinase type II-alpha regulatory subunit	Homo sapiens (human)	Kd	30.0000	1	4
Cannabinoid receptor 1	Mus musculus (house mouse)	EC50	0.1850	1	1
Cannabinoid receptor 2	Mus musculus (house mouse)	EC50	0.1850	1	1
Carbonic anhydrase 2	Homo sapiens (human)	Kd	2,000.0000	1	1
Casein kinase I isoform alpha	Homo sapiens (human)	Kd	20.1742	2	6
Casein kinase I isoform alpha-like	Homo sapiens (human)	Kd	0.9750	2	4
Casein kinase I isoform delta	Homo sapiens (human)	Kd	15.6092	3	8
Casein kinase I isoform epsilon	Homo sapiens (human)	Kd	12.8630	4	12
Casein kinase I isoform gamma-1	Homo sapiens (human)	Kd	18.7200	4	10
Casein kinase I isoform gamma-2	Homo sapiens (human)	Kd	15.8844	4	9
Casein kinase I isoform gamma-3	Homo sapiens (human)	Kd	21.1111	3	9
Casein kinase II subunit alpha	Homo sapiens (human)	Kd	5.2440	2	4
Casein kinase II subunit alpha'	Homo sapiens (human)	Kd	17.5296	3	8
Cell division control protein 2 homolog	Plasmodium falciparum 3D7	Kd	5.4000	1	2
cell division cycle 42 (GTP binding protein, 25kDa), partial	Homo sapiens (human)	EC50	30.0000	4	4
Cell division cycle 7-related protein kinase	Homo sapiens (human)	Kd	30.0000	1	4
cGMP-dependent protein kinase 1	Homo sapiens (human)	Kd	17.5080	3	8
cGMP-dependent protein kinase 2	Homo sapiens (human)	Kd	5.0080	2	4
Chain A, BCL-2-RELATED PROTEIN A1	Homo sapiens (human)	EC50	350.0000	1	1
Chain A, CITRATE SYNTHASE	Sus scrofa (pig)	Kd	10.0000	1	1
Chain A, Glycogen phosphorylase, liver form	Homo sapiens (human)	Kd	100.0000	1	8
Chain A, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1	Homo sapiens (human)	Kd	21.6000	1	1
Chain A, Phospholipase A2 isoform 3	Naja sagittifera	Kd	6.4000	1	1
Chain A, probable fosfomycin resistance protein	Pseudomonas aeruginosa PAO1	Kd	0.2000	1	1
Chain A, Transthyretin	Homo sapiens (human)	Kd	2.1222	1	9
Chain A, Troponin C, slow skeletal and cardiac muscles	Homo sapiens (human)	Kd	1,100.0000	1	1
Chain B, CITRATE SYNTHASE	Sus scrofa (pig)	Kd	10.0000	1	1
Chain B, EUKARYOTIC TRANSLATION INITIATION FACTOR 4E	Homo sapiens (human)	Kd	110,000.0000	1	1
Chain B, probable fosfomycin resistance protein	Pseudomonas aeruginosa PAO1	Kd	0.2000	1	1
Chain B, Transthyretin	Homo sapiens (human)	Kd	2.1000	1	2
Choline-phosphate cytidylyltransferase A	Homo sapiens (human)	Kd	30.0000	1	4
Chromodomain-helicase-DNA-binding protein 4	Homo sapiens (human)	Kd	30.0000	1	4
Citron Rho-interacting kinase	Homo sapiens (human)	Kd	17.5495	3	8
Cyclin-dependent kinase 1	Homo sapiens (human)	Kd	30.0000	1	4
Cyclin-dependent kinase 10	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 11A	Homo sapiens (human)	Kd	10.0000	2	4
Cyclin-dependent kinase 11B	Homo sapiens (human)	Kd	10.0000	2	4
Cyclin-dependent kinase 12	Homo sapiens (human)	Kd	23.3700	1	4
Cyclin-dependent kinase 13	Homo sapiens (human)	Kd	17.4313	2	6
Cyclin-dependent kinase 14	Homo sapiens (human)	Kd	5.0800	2	4
Cyclin-dependent kinase 15	Homo sapiens (human)	Kd	5.1300	1	2
Cyclin-dependent kinase 16	Homo sapiens (human)	Kd	15.4775	4	11
Cyclin-dependent kinase 17	Homo sapiens (human)	Kd	17.5240	3	8
Cyclin-dependent kinase 18	Homo sapiens (human)	Kd	13.4233	3	6
Cyclin-dependent kinase 19	Homo sapiens (human)	Kd	5.0950	2	4
Cyclin-dependent kinase 2	Homo sapiens (human)	Kd	22.1111	5	11
Cyclin-dependent kinase 3	Homo sapiens (human)	Kd	15.7229	3	7
Cyclin-dependent kinase 4	Homo sapiens (human)	Kd	18.8967	3	9
Cyclin-dependent kinase 6	Homo sapiens (human)	Kd	30.0000	1	4
Cyclin-dependent kinase 7	Homo sapiens (human)	Kd	17.5112	3	8
Cyclin-dependent kinase 8	Homo sapiens (human)	Kd	5.2550	2	4
Cyclin-dependent kinase 9	Homo sapiens (human)	Kd	14.3064	3	8
Cyclin-dependent kinase-like 1	Homo sapiens (human)	Kd	5.1650	1	2
Cyclin-dependent kinase-like 2	Homo sapiens (human)	Kd	5.2550	1	2
Cyclin-dependent kinase-like 3	Homo sapiens (human)	Kd	7.5500	1	2
Cyclin-dependent kinase-like 5	Homo sapiens (human)	Kd	17.5850	2	4
Cyclin-dependent-like kinase 5	Homo sapiens (human)	Kd	15.5841	4	9
Cyclin-G-associated kinase	Homo sapiens (human)	Kd	12.5181	4	12
Cysteine--tRNA ligase, cytoplasmic	Homo sapiens (human)	Kd	30.0000	1	4
Cystic fibrosis transmembrane conductance regulator	Homo sapiens (human)	EC50	8.2900	5	5
Cystic fibrosis transmembrane conductance regulator	Homo sapiens (human)	Kd	25.6000	1	1
Cystic fibrosis transmembrane conductance regulator	Rattus norvegicus (Norway rat)	Kd	40.0000	1	1
Cytochrome c1, heme protein, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	4
Cytochrome P450 1A1	Homo sapiens (human)	EC50	8.8000	1	1
Cytochrome P450 1A1	Homo sapiens (human)	Kd	19.1000	1	1
Cytochrome P450 1B1	Homo sapiens (human)	EC50	1.1000	1	1
Cytochrome P450 2B6	Homo sapiens (human)	EC50	1.3000	1	1
Cytochrome P450 2C8	Homo sapiens (human)	EC50	0.1850	1	1
Cytochrome P450 3A4	Homo sapiens (human)	EC50	0.2820	2	2
Cytochrome P450 3A4	Homo sapiens (human)	Kd	0.0130	1	1
Cytoplasmic tyrosine-protein kinase BMX	Homo sapiens (human)	Kd	4.1500	3	5
dCTP pyrophosphatase 1	Homo sapiens (human)	Kd	30.0000	1	5
Death-associated protein kinase 1	Homo sapiens (human)	Kd	5.0007	2	4
Death-associated protein kinase 2	Homo sapiens (human)	Kd	3.4360	3	6
Death-associated protein kinase 3	Homo sapiens (human)	Kd	3.9891	4	8
Delta-type opioid receptor	Homo sapiens (human)	EC50	0.3714	7	7
Delta-type opioid receptor	Rattus norvegicus (Norway rat)	EC50	0.0030	1	1
Delta(24)-sterol reductase	Homo sapiens (human)	Kd	30.0000	1	5
Deoxycytidine kinase	Homo sapiens (human)	Kd	30.0000	1	4
Discoidin domain-containing receptor 2	Homo sapiens (human)	Kd	16.2605	3	8
DNA replication licensing factor MCM4	Homo sapiens (human)	Kd	30.0000	1	4
DNA topoisomerase 2-alpha	Homo sapiens (human)	Kd	30.0000	1	4
DNA topoisomerase 2-beta	Homo sapiens (human)	Kd	30.0000	1	4
DnaJ homolog subfamily A member 1	Homo sapiens (human)	Kd	30.0000	1	4
Dual serine/threonine and tyrosine protein kinase	Homo sapiens (human)	Kd	5.0055	1	2
Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	Kd	13.7630	3	8
Dual specificity mitogen-activated protein kinase kinase 2	Homo sapiens (human)	Kd	13.6581	3	8
Dual specificity mitogen-activated protein kinase kinase 3	Homo sapiens (human)	Kd	18.8900	3	9
Dual specificity mitogen-activated protein kinase kinase 4	Homo sapiens (human)	Kd	10.0280	3	5
Dual specificity mitogen-activated protein kinase kinase 5	Homo sapiens (human)	Kd	20.2338	2	6
Dual specificity mitogen-activated protein kinase kinase 6	Homo sapiens (human)	Kd	17.5008	3	8
Dual specificity mitogen-activated protein kinase kinase 7	Homo sapiens (human)	Kd	5.0150	1	2
Dual specificity protein kinase CLK1	Homo sapiens (human)	Kd	12.2492	4	9
Dual specificity protein kinase CLK2	Homo sapiens (human)	Kd	14.0328	4	10
Dual specificity protein kinase CLK3	Homo sapiens (human)	Kd	16.1467	4	9
Dual specificity protein kinase CLK4	Homo sapiens (human)	Kd	14.0294	4	10
Dual specificity protein kinase TTK	Homo sapiens (human)	Kd	15.4433	4	12
Dual specificity testis-specific protein kinase 1	Homo sapiens (human)	Kd	18.9600	3	9
Dual specificity testis-specific protein kinase 2	Homo sapiens (human)	Kd	30.0000	1	4
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Homo sapiens (human)	Kd	21.6673	2	6
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Homo sapiens (human)	Kd	13.3427	3	6
Dual specificity tyrosine-phosphorylation-regulated kinase 2	Homo sapiens (human)	Kd	5.1250	1	2
Dynamin-like 120 kDa protein, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	4
Egl nine homolog 1	Homo sapiens (human)	EC50	50.0000	1	1
Egl nine homolog 1	Homo sapiens (human)	Kd	200.0000	1	1
eIF-2-alpha kinase GCN2	Homo sapiens (human)	Kd	5.0080	2	4
EKC/KEOPS complex subunit TP53RK	Homo sapiens (human)	Kd	30.0000	1	5
Electron transfer flavoprotein subunit beta	Homo sapiens (human)	Kd	30.0000	1	4
Elongation factor Tu, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	4
endoribonuclease toxin MazF	Escherichia coli str. K-12 substr. MG1655	EC50	99.0000	2	4
Env polyprotein	Human immunodeficiency virus 1	EC50	100.0000	1	1
Ephrin type-A receptor 1	Homo sapiens (human)	Kd	17.5750	3	8
Ephrin type-A receptor 2	Homo sapiens (human)	Kd	15.9189	4	9
Ephrin type-A receptor 3	Homo sapiens (human)	Kd	32.0156	4	7
Ephrin type-A receptor 4	Homo sapiens (human)	Kd	15.6989	4	9
Ephrin type-A receptor 5	Homo sapiens (human)	Kd	15.5933	4	9
Ephrin type-A receptor 6	Homo sapiens (human)	Kd	0.6440	3	5
Ephrin type-A receptor 7	Homo sapiens (human)	Kd	13.9938	4	8
Ephrin type-A receptor 8	Homo sapiens (human)	Kd	4.1360	3	5
Ephrin type-B receptor 1	Homo sapiens (human)	Kd	4.2140	3	5
Ephrin type-B receptor 2	Homo sapiens (human)	Kd	18.7500	4	10
Ephrin type-B receptor 3	Homo sapiens (human)	Kd	21.1111	3	9
Ephrin type-B receptor 4	Homo sapiens (human)	Kd	20.2444	3	9
Ephrin type-B receptor 6	Homo sapiens (human)	Kd	20.5517	2	6
Epidermal growth factor receptor	Homo sapiens (human)	Kd	3.3517	24	50
Epithelial discoidin domain-containing receptor 1	Homo sapiens (human)	Kd	16.8931	3	9
Estrogen receptor	Homo sapiens (human)	EC50	0.8199	6	8
Estrogen receptor beta	Homo sapiens (human)	EC50	0.2460	9	11
Eukaryotic peptide chain release factor GTP-binding subunit ERF3B	Homo sapiens (human)	Kd	30.0000	1	3
Eukaryotic translation initiation factor 2-alpha kinase 1	Homo sapiens (human)	Kd	23.3333	2	6
Eukaryotic translation initiation factor 4E	Homo sapiens (human)	Kd	0.0005	1	1
Eukaryotic translation initiation factor 5B	Homo sapiens (human)	Kd	30.0000	1	4
Exosome RNA helicase MTR4	Homo sapiens (human)	Kd	30.0000	1	4
Fatty acid-binding protein, intestinal	Homo sapiens (human)	Kd	4.4100	1	1
Fatty acid-binding protein, liver	Rattus norvegicus (Norway rat)	Kd	3.1029	16	23
Ferrochelatase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	4
Fibroblast growth factor receptor 1	Homo sapiens (human)	Kd	17.0240	4	10
Fibroblast growth factor receptor 2	Homo sapiens (human)	Kd	4.0720	3	5
Fibroblast growth factor receptor 3	Homo sapiens (human)	Kd	4.5451	5	9
Fibroblast growth factor receptor 4	Homo sapiens (human)	Kd	5.1250	2	4
Focal adhesion kinase 1	Homo sapiens (human)	Kd	15.5773	4	9
Free fatty acid receptor 1	Homo sapiens (human)	EC50	812.8310	1	1
Free fatty acid receptor 3	Homo sapiens (human)	EC50	10.1000	1	1
G protein-coupled receptor	Human betaherpesvirus 5	EC50	0.3306	1	2
G protein-coupled receptor kinase 4	Homo sapiens (human)	Kd	5.0185	1	2
G protein-coupled receptor kinase 6	Homo sapiens (human)	Kd	30.0000	1	4
G-protein coupled bile acid receptor 1	Homo sapiens (human)	EC50	2.3367	5	6
G-protein coupled receptor 35	Homo sapiens (human)	EC50	8.4675	2	8
G-protein coupled receptor homolog US28	Human herpesvirus 5 strain AD169	EC50	0.3524	1	2
GABA theta subunit	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
GABA theta subunit	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	EC50	50.0000	1	4
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	Kd	0.1622	1	1
General transcription and DNA repair factor IIH helicase subunit XPD	Homo sapiens (human)	Kd	30.0000	1	4
Glucose-dependent insulinotropic receptor	Homo sapiens (human)	EC50	2.3043	7	7
Glucose-dependent insulinotropic receptor	Mus musculus (house mouse)	EC50	2.9000	1	1
Glutamate receptor ionotropic, NMDA 1	Homo sapiens (human)	EC50	60.0000	1	1
Glutamate receptor ionotropic, NMDA 2A	Homo sapiens (human)	EC50	60.0000	1	1
Glutamate receptor ionotropic, NMDA 2B	Homo sapiens (human)	EC50	60.0000	1	1
Glutamate receptor ionotropic, NMDA 2C	Homo sapiens (human)	EC50	60.0000	1	1
Glutamate receptor ionotropic, NMDA 2D	Homo sapiens (human)	EC50	60.0000	1	1
Glutamate receptor ionotropic, NMDA 3A	Homo sapiens (human)	EC50	60.0000	1	1
Glutamate receptor ionotropic, NMDA 3B	Homo sapiens (human)	EC50	60.0000	1	1
Glycine receptor subunit alpha-1	Homo sapiens (human)	EC50	0.4000	1	1
Glycine--tRNA ligase	Homo sapiens (human)	Kd	30.0000	1	5
Glycogen phosphorylase, brain form	Homo sapiens (human)	Kd	30.0000	1	4
Glycogen phosphorylase, liver form	Homo sapiens (human)	Kd	30.0000	1	4
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	Kd	18.9200	3	9
Glycogen synthase kinase-3 beta	Homo sapiens (human)	EC50	3,000.0000	1	1
Glycogen synthase kinase-3 beta	Homo sapiens (human)	Kd	15.4422	3	8
glycogen synthase kinase-3 beta isoform 1	Homo sapiens (human)	EC50	109.1300	1	3
GTP-binding nuclear protein Ran	Homo sapiens (human)	Kd	30.0000	1	4
GTP-binding protein (rab7)	Canis lupus familiaris (dog)	EC50	30.0000	2	2
Guanine nucleotide-binding protein G(i) subunit alpha-2	Homo sapiens (human)	Kd	30.0000	1	3
Hemagglutinin	Influenza A virus (A/Puerto Rico/8/1934(H1N1))	Kd	46.5000	1	1
Heme oxygenase 2	Homo sapiens (human)	Kd	30.0000	1	4
Heparanase	Homo sapiens (human)	Kd	1,000.0000	1	1
Hepatocyte growth factor receptor	Homo sapiens (human)	Kd	14.5038	5	13
Heterogeneous nuclear ribonucleoprotein A1	Homo sapiens (human)	Kd	5.3000	1	2
High affinity nerve growth factor receptor	Homo sapiens (human)	Kd	15.5567	4	9
Histamine H1 receptor	Homo sapiens (human)	Kd	0.1900	1	1
Histidine decarboxylase	Rattus norvegicus (Norway rat)	EC50	0.0030	1	1
Histone deacetylase 1	Homo sapiens (human)	EC50	3.5000	2	2
Histone deacetylase 1	Homo sapiens (human)	Kd	0.0137	1	2
Histone deacetylase 2	Homo sapiens (human)	Kd	0.0137	1	2
Histone deacetylase 4	Homo sapiens (human)	EC50	2.5000	1	2
Histone deacetylase 6	Homo sapiens (human)	EC50	0.0052	1	1
HLA class I histocompatibility antigen, A alpha chain	Homo sapiens (human)	Kd	15.7000	1	1
Homeodomain-interacting protein kinase 1	Homo sapiens (human)	Kd	6.3500	1	2
Homeodomain-interacting protein kinase 2	Homo sapiens (human)	Kd	5.0950	1	2
Homeodomain-interacting protein kinase 3	Homo sapiens (human)	Kd	5.0375	1	2
Homeodomain-interacting protein kinase 4	Homo sapiens (human)	Kd	5.1950	1	2
Hormonally up-regulated neu tumor-associated kinase	Homo sapiens (human)	Kd	5.3100	1	2
Hsf1 protein	Mus musculus (house mouse)	EC50	98.6595	2	2
Inhibitor of nuclear factor kappa-B kinase subunit alpha	Homo sapiens (human)	Kd	5.0029	1	2
Inhibitor of nuclear factor kappa-B kinase subunit beta	Homo sapiens (human)	Kd	5.0155	1	2
Inhibitor of nuclear factor kappa-B kinase subunit epsilon	Homo sapiens (human)	Kd	17.5013	3	8
Inosine-5'-monophosphate dehydrogenase 2	Homo sapiens (human)	Kd	30.0000	1	4
Insulin receptor	Homo sapiens (human)	Kd	15.5881	4	9
Insulin receptor-related protein	Homo sapiens (human)	Kd	5.0405	2	4
Insulin-like growth factor 1 receptor	Homo sapiens (human)	Kd	18.9356	3	9
Insulin-like growth factor-binding protein 5	Homo sapiens (human)	Kd	696,000.0000	7	7
Integrase	Human immunodeficiency virus 1	Kd	3.0000	1	1
Integrin-linked protein kinase	Homo sapiens (human)	Kd	30.0000	1	4
Interferon-induced, double-stranded RNA-activated protein kinase	Homo sapiens (human)	Kd	5.1800	2	4
Interleukin-1 receptor-associated kinase 1	Homo sapiens (human)	Kd	21.6733	2	6
Interleukin-1 receptor-associated kinase 3	Homo sapiens (human)	Kd	17.5032	3	8
Interleukin-1 receptor-associated kinase 4	Homo sapiens (human)	Kd	21.6670	2	6
Interstitial collagenase	Homo sapiens (human)	Kd	51.8000	1	1
Isoleucine--tRNA ligase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	2
Kappa-type opioid receptor	Homo sapiens (human)	EC50	0.4443	6	6
Kappa-type opioid receptor	Mus musculus (house mouse)	EC50	0.4000	1	1
Kappa-type opioid receptor	Rattus norvegicus (Norway rat)	EC50	0.0030	1	1
LAP4	Saccharomyces cerevisiae (brewer's yeast)	EC50	4.8230	1	1
Leucine-rich repeat serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	5.0009	2	4
Leukocyte tyrosine kinase receptor	Homo sapiens (human)	Kd	5.0185	2	4
Leukotriene C4 synthase	Cavia porcellus (domestic guinea pig)	Kd	6.7500	1	2
LIM domain kinase 1	Homo sapiens (human)	Kd	15.7389	4	9
LIM domain kinase 2	Homo sapiens (human)	Kd	20.9333	3	9
Long-chain-fatty-acid--CoA ligase 5	Homo sapiens (human)	Kd	30.0000	1	2
Lymphocyte antigen 96	Homo sapiens (human)	Kd	379.0000	1	1
Macrophage colony-stimulating factor 1 receptor	Homo sapiens (human)	Kd	5.0060	2	4
Macrophage-stimulating protein receptor	Homo sapiens (human)	Kd	22.9143	2	7
MAP kinase-activated protein kinase 2	Homo sapiens (human)	Kd	17.7200	3	8
MAP kinase-activated protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
MAP kinase-activated protein kinase 5	Homo sapiens (human)	Kd	17.1814	3	7
MAP kinase-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	5.0850	2	4
MAP kinase-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	3.5093	3	6
MAP/microtubule affinity-regulating kinase 3	Homo sapiens (human)	Kd	17.5007	3	8
MAP/microtubule affinity-regulating kinase 4	Homo sapiens (human)	Kd	17.5014	3	8
Mas-related G-protein coupled receptor member X2	Homo sapiens (human)	EC50	6.4000	2	2
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	Kd	4.8486	16	31
Maternal embryonic leucine zipper kinase	Homo sapiens (human)	Kd	13.9985	3	8
Megakaryocyte-associated tyrosine-protein kinase	Homo sapiens (human)	Kd	5.1300	1	2
Melatonin receptor type 1A	Gallus gallus (chicken)	EC50	0.0226	1	1
Melatonin receptor type 1A	Homo sapiens (human)	EC50	0.0008	11	11
Melatonin receptor type 1B	Gallus gallus (chicken)	EC50	0.0226	1	1
Melatonin receptor type 1B	Homo sapiens (human)	EC50	0.0025	12	12
Melatonin receptor type 1C	Gallus gallus (chicken)	EC50	0.0226	1	1
Melatonin receptor type 1C	Xenopus laevis (African clawed frog)	EC50	0.0001	3	3
Membrane-associated progesterone receptor component 1	Homo sapiens (human)	Kd	30.0000	1	1
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	Homo sapiens (human)	Kd	20.0000	3	8
Methionine--tRNA ligase, mitochondrial	Homo sapiens (human)	EC50	7.9000	1	1
Methyl-accepting chemotaxis protein NahY	Pseudomonas putida	Kd	20.4500	1	2
Microtubule-associated serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	5.0750	1	2
Midasin	Homo sapiens (human)	Kd	30.0000	1	5
Misshapen-like kinase 1	Homo sapiens (human)	Kd	17.5002	2	4
Mitogen-activated protein kinase 1	Homo sapiens (human)	Kd	20.5111	3	9
Mitogen-activated protein kinase 10	Homo sapiens (human)	Kd	11.5938	5	13
Mitogen-activated protein kinase 11	Homo sapiens (human)	EC50	0.0600	1	1
Mitogen-activated protein kinase 11	Homo sapiens (human)	Kd	15.4909	5	11
Mitogen-activated protein kinase 12	Homo sapiens (human)	EC50	0.0600	1	1
Mitogen-activated protein kinase 12	Homo sapiens (human)	Kd	0.9108	4	8
Mitogen-activated protein kinase 13	Homo sapiens (human)	EC50	0.0600	1	1
Mitogen-activated protein kinase 13	Homo sapiens (human)	Kd	3.4167	2	3
Mitogen-activated protein kinase 14	Homo sapiens (human)	EC50	0.0600	2	2
Mitogen-activated protein kinase 14	Homo sapiens (human)	Kd	11.6731	7	12
Mitogen-activated protein kinase 14	Mus musculus (house mouse)	Kd	0.0200	2	2
Mitogen-activated protein kinase 15	Homo sapiens (human)	Kd	17.5088	3	8
Mitogen-activated protein kinase 3	Homo sapiens (human)	Kd	19.6000	3	8
Mitogen-activated protein kinase 4	Homo sapiens (human)	Kd	10.0000	2	4
Mitogen-activated protein kinase 6	Homo sapiens (human)	Kd	8.2750	2	4
Mitogen-activated protein kinase 7	Homo sapiens (human)	Kd	17.9000	3	8
Mitogen-activated protein kinase 8	Homo sapiens (human)	Kd	10.3800	5	12
Mitogen-activated protein kinase 9	Homo sapiens (human)	Kd	12.5025	5	13
Mitogen-activated protein kinase kinase kinase 1	Homo sapiens (human)	Kd	21.7250	2	6
Mitogen-activated protein kinase kinase kinase 10	Homo sapiens (human)	Kd	5.0260	2	4
Mitogen-activated protein kinase kinase kinase 11	Homo sapiens (human)	Kd	15.5622	4	9
Mitogen-activated protein kinase kinase kinase 12	Homo sapiens (human)	Kd	5.7500	1	2
Mitogen-activated protein kinase kinase kinase 13	Homo sapiens (human)	Kd	5.1050	1	2
Mitogen-activated protein kinase kinase kinase 15	Homo sapiens (human)	Kd	5.0012	1	2
Mitogen-activated protein kinase kinase kinase 19	Homo sapiens (human)	Kd	5.0004	1	2
Mitogen-activated protein kinase kinase kinase 2	Homo sapiens (human)	Kd	22.8575	2	7
Mitogen-activated protein kinase kinase kinase 20	Homo sapiens (human)	Kd	19.8667	3	9
Mitogen-activated protein kinase kinase kinase 3	Homo sapiens (human)	Kd	23.2571	2	7
Mitogen-activated protein kinase kinase kinase 4	Homo sapiens (human)	Kd	16.0667	4	9
Mitogen-activated protein kinase kinase kinase 5	Homo sapiens (human)	Kd	15.4955	5	11
Mitogen-activated protein kinase kinase kinase 6	Homo sapiens (human)	Kd	21.7100	2	6
Mitogen-activated protein kinase kinase kinase 7	Homo sapiens (human)	Kd	5.0335	1	2
Mitogen-activated protein kinase kinase kinase 9	Homo sapiens (human)	Kd	5.0050	2	4
Mitogen-activated protein kinase kinase kinase kinase 1	Homo sapiens (human)	Kd	17.5011	3	8
Mitogen-activated protein kinase kinase kinase kinase 2	Homo sapiens (human)	Kd	21.6681	2	6
Mitogen-activated protein kinase kinase kinase kinase 3	Homo sapiens (human)	Kd	17.5020	3	8
Mitogen-activated protein kinase kinase kinase kinase 4	Homo sapiens (human)	Kd	15.9310	3	8
Mitogen-activated protein kinase kinase kinase kinase 5	Homo sapiens (human)	Kd	18.1875	4	11
Mitotic checkpoint serine/threonine-protein kinase BUB1	Homo sapiens (human)	Kd	30.0000	1	4
Mu-type opioid receptor	Homo sapiens (human)	EC50	0.1302	26	27
Mu-type opioid receptor	Mus musculus (house mouse)	EC50	0.0750	2	2
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	EC50	0.1118	7	7
mu-type opioid receptor isoform MOR-1	Homo sapiens (human)	EC50	92.4750	1	2
Multidrug resistance protein MdtK	Escherichia coli K-12	Kd	9.8000	1	1
Multidrug resistance-associated protein 1	Homo sapiens (human)	EC50	21.8500	2	2
Multifunctional protein ADE2	Homo sapiens (human)	Kd	30.0000	1	5
Muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	EC50	191.2333	2	9
Muscarinic acetylcholine receptor M2	Rattus norvegicus (Norway rat)	EC50	191.2333	2	9
Muscarinic acetylcholine receptor M3	Rattus norvegicus (Norway rat)	EC50	191.2333	2	9
Muscarinic acetylcholine receptor M4	Rattus norvegicus (Norway rat)	EC50	191.2333	2	9
Muscarinic acetylcholine receptor M5	Rattus norvegicus (Norway rat)	EC50	191.2333	2	9
Muscle, skeletal receptor tyrosine-protein kinase	Homo sapiens (human)	Kd	5.0430	2	4
Myosin light chain kinase 2, skeletal/cardiac muscle	Homo sapiens (human)	Kd	4.0464	3	5
Myosin light chain kinase 3	Homo sapiens (human)	Kd	21.6900	2	6
Myosin light chain kinase family member 4	Homo sapiens (human)	Kd	5.2350	2	4
Myosin light chain kinase, smooth muscle	Gallus gallus (chicken)	Kd	5.0700	1	2
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	Kd	18.8922	3	9
Myosin-10	Homo sapiens (human)	Kd	30.0000	1	5
Myosin-14	Homo sapiens (human)	Kd	30.0000	1	4
Myosin-IIIa	Homo sapiens (human)	Kd	5.2500	2	4
Myosin-IIIb	Homo sapiens (human)	Kd	5.1500	2	4
Myotonin-protein kinase	Homo sapiens (human)	Kd	5.0018	2	4
NAD kinase	Homo sapiens (human)	Kd	1.7800	1	1
NAD-dependent protein deacetylase sirtuin-6	Homo sapiens (human)	Kd	183.5000	4	4
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13	Homo sapiens (human)	Kd	30.0000	1	4
Neuronal acetylcholine receptor subunit alpha-7	Homo sapiens (human)	EC50	11.6000	1	1
Non-receptor tyrosine-protein kinase TNK1	Homo sapiens (human)	Kd	17.5006	3	8
Non-receptor tyrosine-protein kinase TYK2	Homo sapiens (human)	Kd	14.5212	4	10
NPYLR7B	Aedes aegypti (yellow fever mosquito)	EC50	20.0000	1	2
NT-3 growth factor receptor	Homo sapiens (human)	Kd	5.0085	2	4
NUAK family SNF1-like kinase 1	Homo sapiens (human)	Kd	5.0022	2	4
NUAK family SNF1-like kinase 2	Homo sapiens (human)	Kd	15.7143	3	7
Nuclear factor erythroid 2-related factor 2	Homo sapiens (human)	EC50	21.0000	1	1
Nuclear hormone receptor family member daf-12	Caenorhabditis elegans	EC50	67.4900	1	1
Nuclear receptor subfamily 1 group I member 2	Homo sapiens (human)	EC50	4.6740	11	20
Nuclear receptor subfamily 1 group I member 2	Rattus norvegicus (Norway rat)	EC50	25.1000	1	1
Nuclear receptor subfamily 4 group A member 2	Homo sapiens (human)	EC50	5.1000	1	1
Nucleolar GTP-binding protein 1	Homo sapiens (human)	Kd	30.0000	1	5
Obg-like ATPase 1	Homo sapiens (human)	Kd	30.0000	1	4
ORF73	Human gammaherpesvirus 8	EC50	75.0000	1	2
oxysterols receptor LXR-beta isoform 1	Homo sapiens (human)	EC50	67.4900	1	1
Palmitoleoyl-protein carboxylesterase NOTUM	Homo sapiens (human)	EC50	45.8000	1	1
Palmitoleoyl-protein carboxylesterase NOTUM	Homo sapiens (human)	Kd	85.0000	1	1
PAS domain-containing serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	4
Peptidyl-prolyl cis-trans isomerase A	Homo sapiens (human)	Kd	0.6225	11	11
Peptidyl-prolyl cis-trans isomerase B	Homo sapiens (human)	Kd	0.0098	1	1
Peptidyl-prolyl cis-trans isomerase D	Homo sapiens (human)	Kd	0.0215	2	2
Peptidyl-prolyl cis-trans isomerase FKBP1A	Homo sapiens (human)	EC50	0.0364	1	1
Peptidyl-prolyl cis-trans isomerase FKBP1B	Homo sapiens (human)	Kd	0.0002	1	1
Peripheral plasma membrane protein CASK	Homo sapiens (human)	Kd	5.0095	1	2
Peroxisomal acyl-coenzyme A oxidase 1	Homo sapiens (human)	Kd	30.0000	1	4
Peroxisomal acyl-coenzyme A oxidase 3	Homo sapiens (human)	Kd	30.0000	1	4
Peroxisome proliferator-activated receptor alpha	Homo sapiens (human)	EC50	31.6797	30	38
Peroxisome proliferator-activated receptor alpha	Mus musculus (house mouse)	EC50	62.0000	2	4
Peroxisome proliferator-activated receptor alpha	Rattus norvegicus (Norway rat)	EC50	29.5000	2	2
Peroxisome proliferator-activated receptor delta	Homo sapiens (human)	EC50	41.0709	11	11
Peroxisome proliferator-activated receptor delta	Mus musculus (house mouse)	EC50	110.0000	2	2
Peroxisome proliferator-activated receptor gamma	Homo sapiens (human)	EC50	49.7244	50	56
Peroxisome proliferator-activated receptor gamma	Mus musculus (house mouse)	EC50	143.5400	3	6
Peroxisome proliferator-activated receptor gamma	Homo sapiens (human)	Kd	0.8710	1	1
Phenylalanine--tRNA ligase beta subunit	Homo sapiens (human)	Kd	30.0000	1	4
Phosphatidylethanolamine-binding protein 1	Homo sapiens (human)	Kd	30.0000	1	4
Phosphatidylinositol 4-kinase beta	Homo sapiens (human)	Kd	5.2300	1	2
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta	Homo sapiens (human)	Kd	10.0000	1	2
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma	Homo sapiens (human)	Kd	5.2150	1	2
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha	Homo sapiens (human)	Kd	5.0215	2	4
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma	Homo sapiens (human)	Kd	2.6500	1	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	Kd	9.2162	13	25
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	Kd	6.6692	2	3
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	Homo sapiens (human)	Kd	6.6685	2	3
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Homo sapiens (human)	Kd	3.9383	2	3
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha	Homo sapiens (human)	Kd	30.0000	1	4
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta	Homo sapiens (human)	Kd	5.0385	2	4
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma	Homo sapiens (human)	Kd	23.3333	2	6
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform	Homo sapiens (human)	Kd	14.0481	4	10
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform	Homo sapiens (human)	Kd	4.0004	3	5
Platelet-derived growth factor receptor alpha	Homo sapiens (human)	Kd	5.0050	2	4
Platelet-derived growth factor receptor beta	Homo sapiens (human)	Kd	15.5563	4	9
Polycomb protein EED	Homo sapiens (human)	Kd	15.1000	1	1
Polypeptide N-acetylgalactosaminyltransferase 2	Homo sapiens (human)	Kd	0.6475	1	2
POsterior Segregation	Caenorhabditis elegans	EC50	16.2407	1	3
Potassium channel subfamily K member 2	Homo sapiens (human)	EC50	377.0000	1	1
Probable ATP-dependent RNA helicase DDX6	Homo sapiens (human)	Kd	30.0000	1	4
Procathepsin L	Homo sapiens (human)	EC50	83.4000	1	1
Programmed cell death protein 4	Homo sapiens (human)	EC50	0.0500	1	1
Prolyl hydroxylase EGLN2	Homo sapiens (human)	EC50	50.0000	1	1
Prolyl hydroxylase EGLN3	Homo sapiens (human)	EC50	50.0000	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	Kd	3.6397	2	3
Protein kinase C alpha type	Homo sapiens (human)	Kd	24.0100	2	5
Protein kinase C beta type	Homo sapiens (human)	Kd	30.0000	1	4
Protein kinase C delta type	Homo sapiens (human)	Kd	14.3490	3	8
Protein kinase C epsilon type	Homo sapiens (human)	Kd	5.0001	2	4
Protein kinase C eta type	Homo sapiens (human)	Kd	5.0024	2	4
Protein kinase C iota type	Homo sapiens (human)	Kd	21.6710	2	6
Protein kinase C theta type	Homo sapiens (human)	Kd	17.5021	3	8
Protein kinase C zeta type	Homo sapiens (human)	Kd	30.0000	1	3
Protein-tyrosine kinase 2-beta	Homo sapiens (human)	Kd	17.5009	3	8
Protein-tyrosine kinase 6	Homo sapiens (human)	Kd	15.7111	4	9
Proteinase-activated receptor 1	Homo sapiens (human)	EC50	0.0037	1	2
Prothrombin	Homo sapiens (human)	Kd	0.0387	1	1
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	Kd	11.2571	7	16
Proto-oncogene tyrosine-protein kinase ROS	Homo sapiens (human)	Kd	5.0150	2	4
Proto-oncogene tyrosine-protein kinase Src	Gallus gallus (chicken)	Kd	0.2960	1	1
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	Kd	14.6255	5	11
Putative heat shock protein HSP 90-beta 2	Homo sapiens (human)	Kd	30.0000	1	4
Pyridoxal kinase	Homo sapiens (human)	Kd	30.0000	1	5
Pyruvate kinase PKM	Homo sapiens (human)	EC50	0.0009	2	2
Rab-like protein 3	Homo sapiens (human)	Kd	30.0000	1	1
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	EC50	0.4600	2	2
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	Kd	17.5050	3	8
RAC-beta serine/threonine-protein kinase	Homo sapiens (human)	Kd	17.5110	3	8
RAC-gamma serine/threonine-protein kinase	Homo sapiens (human)	Kd	17.5425	3	8
Rac1 protein	Homo sapiens (human)	EC50	33.2632	4	4
RAF proto-oncogene serine/threonine-protein kinase	Homo sapiens (human)	Kd	5.4900	2	4
ras protein, partial	Homo sapiens (human)	EC50	30.0000	4	4
Ras-related C3 botulinum toxin substrate 1	Homo sapiens (human)	Kd	30.0000	1	1
Ras-related protein Rab-10	Homo sapiens (human)	Kd	30.0000	1	5
Ras-related protein Rab-27A	Homo sapiens (human)	Kd	30.0000	1	4
Ras-related protein Rab-2A	Canis lupus familiaris (dog)	EC50	30.0000	2	2
Ras-related protein Rab-6A	Homo sapiens (human)	Kd	30.0000	1	4
Receptor tyrosine-protein kinase erbB-2	Homo sapiens (human)	Kd	7.5475	2	4
Receptor tyrosine-protein kinase erbB-3	Homo sapiens (human)	Kd	10.0000	1	2
Receptor tyrosine-protein kinase erbB-4	Homo sapiens (human)	Kd	2.7850	1	2
Receptor-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	4
Receptor-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	16.4707	4	12
Receptor-interacting serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	4
Receptor-interacting serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	5.0550	1	2
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	Kd	8.0011	15	30
recombinase A	Mycobacterium tuberculosis H37Rv	EC50	124.0550	2	2
Renin	Homo sapiens (human)	EC50	0.1850	1	1
Replicase polyprotein 1a	Severe acute respiratory syndrome-related coronavirus	EC50	83.4000	2	2
Replicase polyprotein 1ab	Betacoronavirus England 1	EC50	83.4000	1	1
Replicase polyprotein 1ab	Human coronavirus 229E	EC50	83.4000	2	2
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	EC50	24.5075	3	4
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	EC50	44.9350	3	4
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	Kd	18.4000	3	3
Reverse transcriptase/RNaseH	Human immunodeficiency virus 1	Kd	7.1500	2	2
Rho-associated protein kinase 1	Homo sapiens (human)	Kd	16.8177	2	6
Rho-associated protein kinase 2	Homo sapiens (human)	Kd	16.3777	3	8
Rhodopsin kinase GRK1	Homo sapiens (human)	Kd	5.0005	1	2
Rhodopsin kinase GRK7	Homo sapiens (human)	Kd	5.0004	1	2
Ribosomal protein S6 kinase alpha-1	Homo sapiens (human)	Kd	11.9272	5	12
Ribosomal protein S6 kinase alpha-2	Homo sapiens (human)	Kd	4.2608	5	10
Ribosomal protein S6 kinase alpha-3	Homo sapiens (human)	Kd	15.5776	4	9
Ribosomal protein S6 kinase alpha-4	Homo sapiens (human)	Kd	13.7200	5	12
Ribosomal protein S6 kinase alpha-5	Homo sapiens (human)	Kd	11.6846	6	14
Ribosomal protein S6 kinase alpha-6	Homo sapiens (human)	Kd	12.2613	5	12
Ribosomal protein S6 kinase beta-1	Homo sapiens (human)	Kd	21.6669	2	6
Ribosyldihydronicotinamide dehydrogenase [quinone]	Homo sapiens (human)	Kd	23.1127	1	4
RNA cytidine acetyltransferase	Homo sapiens (human)	Kd	30.0000	1	5
RPL19A	Saccharomyces cerevisiae (brewer's yeast)	EC50	0.8525	2	2
S-adenosylmethionine synthase isoform type-2	Homo sapiens (human)	Kd	30.0000	1	4
Septin-9	Homo sapiens (human)	Kd	30.0000	1	5
Serine/threonine-protein kinase 10	Homo sapiens (human)	Kd	15.5556	4	9
Serine/threonine-protein kinase 16	Homo sapiens (human)	Kd	14.1250	4	10
Serine/threonine-protein kinase 17A	Homo sapiens (human)	Kd	3.6918	3	6
Serine/threonine-protein kinase 17B	Homo sapiens (human)	Kd	4.0136	3	5
Serine/threonine-protein kinase 24	Homo sapiens (human)	Kd	13.3733	3	6
Serine/threonine-protein kinase 25	Homo sapiens (human)	Kd	5.0550	2	4
Serine/threonine-protein kinase 26	Homo sapiens (human)	Kd	17.5350	3	8
Serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	17.5000	3	8
Serine/threonine-protein kinase 3	Mus musculus (house mouse)	Kd	0.1101	1	2
Serine/threonine-protein kinase 32A	Homo sapiens (human)	Kd	0.6565	1	2
Serine/threonine-protein kinase 32B	Homo sapiens (human)	Kd	1.0990	2	4
Serine/threonine-protein kinase 32C	Homo sapiens (human)	Kd	5.1550	2	4
Serine/threonine-protein kinase 33	Homo sapiens (human)	Kd	5.0009	2	4
serine/threonine-protein kinase 33 isoform a	Homo sapiens (human)	EC50	15.3800	1	2
Serine/threonine-protein kinase 35	Homo sapiens (human)	Kd	5.0700	1	2
Serine/threonine-protein kinase 36	Homo sapiens (human)	Kd	3.2933	3	6
Serine/threonine-protein kinase 38	Homo sapiens (human)	Kd	5.0280	1	2
Serine/threonine-protein kinase 38-like	Homo sapiens (human)	Kd	3.7388	3	6
Serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	15.6546	4	11
Serine/threonine-protein kinase A-Raf	Homo sapiens (human)	Kd	30.0000	1	4
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	Kd	13.5400	5	12
Serine/threonine-protein kinase BRSK1	Homo sapiens (human)	Kd	5.0130	2	4
Serine/threonine-protein kinase BRSK2	Homo sapiens (human)	Kd	5.0018	2	4
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	Kd	17.5008	3	8
Serine/threonine-protein kinase Chk2	Homo sapiens (human)	Kd	5.0370	1	2
Serine/threonine-protein kinase D1	Homo sapiens (human)	Kd	5.0135	2	4
Serine/threonine-protein kinase D2	Homo sapiens (human)	Kd	14.5700	3	8
Serine/threonine-protein kinase D3	Homo sapiens (human)	Kd	16.6721	3	8
Serine/threonine-protein kinase DCLK1	Homo sapiens (human)	Kd	5.0550	2	4
Serine/threonine-protein kinase DCLK2	Homo sapiens (human)	Kd	5.0365	2	4
Serine/threonine-protein kinase DCLK3	Homo sapiens (human)	Kd	5.0085	2	4
Serine/threonine-protein kinase ICK	Homo sapiens (human)	Kd	17.5040	2	4
Serine/threonine-protein kinase LATS1	Homo sapiens (human)	Kd	14.2818	3	8
Serine/threonine-protein kinase LATS2	Homo sapiens (human)	Kd	5.0085	2	4
Serine/threonine-protein kinase MAK	Homo sapiens (human)	Kd	6.3000	1	2
Serine/threonine-protein kinase MARK1	Homo sapiens (human)	Kd	5.0020	2	4
Serine/threonine-protein kinase MARK2	Homo sapiens (human)	Kd	14.1801	4	10
Serine/threonine-protein kinase MRCK alpha	Homo sapiens (human)	Kd	16.5642	3	8
Serine/threonine-protein kinase MRCK beta	Homo sapiens (human)	Kd	17.2760	3	9
Serine/threonine-protein kinase MRCK gamma	Homo sapiens (human)	Kd	15.1092	3	8
Serine/threonine-protein kinase mTOR	Homo sapiens (human)	Kd	5.8405	3	5
Serine/threonine-protein kinase N1	Homo sapiens (human)	Kd	13.8554	3	8
Serine/threonine-protein kinase N2	Homo sapiens (human)	Kd	14.0755	3	8
Serine/threonine-protein kinase N3	Homo sapiens (human)	Kd	22.5248	1	4
Serine/threonine-protein kinase Nek1	Homo sapiens (human)	Kd	17.7150	3	8
Serine/threonine-protein kinase Nek11	Homo sapiens (human)	Kd	6.5500	1	2
Serine/threonine-protein kinase Nek2	Homo sapiens (human)	Kd	15.8044	4	9
Serine/threonine-protein kinase Nek3	Homo sapiens (human)	Kd	23.3333	2	6
Serine/threonine-protein kinase Nek4	Homo sapiens (human)	Kd	10.0000	1	2
Serine/threonine-protein kinase Nek5	Homo sapiens (human)	Kd	5.4050	2	4
Serine/threonine-protein kinase Nek6	Homo sapiens (human)	Kd	10.0000	2	4
Serine/threonine-protein kinase Nek7	Homo sapiens (human)	Kd	14.8333	3	6
Serine/threonine-protein kinase Nek9	Homo sapiens (human)	Kd	16.9889	4	9
Serine/threonine-protein kinase NIM1	Homo sapiens (human)	Kd	5.0700	1	2
Serine/threonine-protein kinase NLK	Homo sapiens (human)	Kd	15.0612	3	8
Serine/threonine-protein kinase OSR1	Homo sapiens (human)	Kd	5.2200	1	2
Serine/threonine-protein kinase PAK 1	Homo sapiens (human)	Kd	4.0006	3	5
Serine/threonine-protein kinase PAK 2	Homo sapiens (human)	Kd	17.5008	3	8
Serine/threonine-protein kinase PAK 3	Homo sapiens (human)	Kd	4.0029	3	5
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	Kd	17.0021	4	10
Serine/threonine-protein kinase PAK 5	Homo sapiens (human)	Kd	4.0011	3	5
Serine/threonine-protein kinase PAK 6	Homo sapiens (human)	Kd	8.3336	4	6
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	Kd	12.7316	5	11
Serine/threonine-protein kinase pim-2	Homo sapiens (human)	Kd	7.2097	4	7
Serine/threonine-protein kinase pim-3	Homo sapiens (human)	Kd	5.0003	2	4
Serine/threonine-protein kinase PknB	Mycobacterium tuberculosis H37Rv	Kd	5.0440	1	2
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	Kd	20.0380	3	10
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	Kd	5.1000	1	2
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	Kd	5.4550	2	4
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	Kd	14.0772	4	10
Serine/threonine-protein kinase PRP4 homolog	Homo sapiens (human)	Kd	5.1100	1	2
Serine/threonine-protein kinase receptor R3	Homo sapiens (human)	Kd	16.6667	3	6
Serine/threonine-protein kinase RIO1	Homo sapiens (human)	Kd	5.0650	2	4
Serine/threonine-protein kinase RIO2	Homo sapiens (human)	Kd	5.1950	1	2
Serine/threonine-protein kinase RIO3	Homo sapiens (human)	Kd	3.3846	3	6
Serine/threonine-protein kinase SBK1	Homo sapiens (human)	Kd	5.0016	1	2
Serine/threonine-protein kinase Sgk3	Homo sapiens (human)	Kd	5.0017	1	2
Serine/threonine-protein kinase SIK1	Homo sapiens (human)	Kd	5.0011	2	4
Serine/threonine-protein kinase SIK2	Homo sapiens (human)	Kd	17.5003	3	8
Serine/threonine-protein kinase SIK3	Homo sapiens (human)	Kd	20.6501	2	6
Serine/threonine-protein kinase STK11	Homo sapiens (human)	Kd	17.5153	3	8
Serine/threonine-protein kinase TAO1	Homo sapiens (human)	Kd	21.6667	2	6
Serine/threonine-protein kinase TAO2	Homo sapiens (human)	Kd	21.6687	2	6
Serine/threonine-protein kinase TAO3	Homo sapiens (human)	Kd	22.8572	2	7
Serine/threonine-protein kinase TBK1	Homo sapiens (human)	Kd	21.6668	2	6
Serine/threonine-protein kinase TNNI3K	Homo sapiens (human)	Kd	2.2500	2	4
Serine/threonine-protein kinase tousled-like 1	Homo sapiens (human)	Kd	5.0135	2	4
Serine/threonine-protein kinase tousled-like 2	Homo sapiens (human)	Kd	5.0080	2	4
Serine/threonine-protein kinase ULK1	Homo sapiens (human)	Kd	21.6683	2	6
Serine/threonine-protein kinase ULK2	Homo sapiens (human)	Kd	5.0004	1	2
Serine/threonine-protein kinase ULK3	Homo sapiens (human)	Kd	22.8573	2	7
Serine/threonine-protein kinase ULK3	Mus musculus (house mouse)	Kd	0.3415	1	2
Serine/threonine-protein kinase VRK2	Homo sapiens (human)	Kd	10.0000	1	2
Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens (human)	Kd	21.6702	2	6
Serine/threonine-protein kinase/endoribonuclease IRE2	Homo sapiens (human)	Kd	30.0000	1	4
Sex hormone-binding globulin	Homo sapiens (human)	Kd	19.9085	1	2
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	EC50	30.0000	1	2
Sigma non-opioid intracellular receptor 1	Rattus norvegicus (Norway rat)	EC50	30.0000	2	2
Sigma non-opioid intracellular receptor 1	Rattus norvegicus (Norway rat)	Kd	0.1600	1	1
Signal recognition particle receptor subunit alpha	Homo sapiens (human)	Kd	30.0000	1	4
Signal transducer and activator of transcription 1-alpha/beta	Homo sapiens (human)	Kd	0.7000	1	1
SNF-related serine/threonine-protein kinase	Homo sapiens (human)	Kd	5.0450	1	2
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	EC50	7.2513	1	3
Sodium-dependent serotonin transporter	Rattus norvegicus (Norway rat)	EC50	30.0000	1	1
Sodium/bile acid cotransporter	Homo sapiens (human)	Kd	64.3000	1	1
Spike glycoprotein	Betacoronavirus England 1	EC50	83.4000	1	1
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	EC50	83.4000	1	1
SRSF protein kinase 1	Homo sapiens (human)	Kd	5.0028	2	4
SRSF protein kinase 2	Homo sapiens (human)	Kd	5.0335	2	4
SRSF protein kinase 3	Homo sapiens (human)	Kd	5.0365	1	2
STE20-like serine/threonine-protein kinase	Homo sapiens (human)	Kd	12.2091	4	11
STE20-related kinase adapter protein alpha	Homo sapiens (human)	Kd	30.0000	1	4
STE20/SPS1-related proline-alanine-rich protein kinase	Homo sapiens (human)	Kd	5.0650	1	2
streptokinase A precursor	Streptococcus pyogenes M1 GAS	EC50	1.3815	1	2
Structural maintenance of chromosomes protein 1A	Homo sapiens (human)	Kd	30.0000	1	4
Structural maintenance of chromosomes protein 2	Homo sapiens (human)	Kd	30.0000	1	4
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	6
SWI/SNF related, matrix associated, actin dependent regulator of chromatin, subfamily a, member 2, isoform CRA_a	Homo sapiens (human)	EC50	91.1400	1	1
Testis-specific serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	5.0120	2	4
TGF-beta receptor type-1	Homo sapiens (human)	Kd	17.2750	3	8
TGF-beta receptor type-2	Homo sapiens (human)	Kd	17.9500	3	8
Thyroid hormone receptor-associated protein 3	Homo sapiens (human)	Kd	30.0000	1	4
TRAF2 and NCK-interacting protein kinase	Homo sapiens (human)	Kd	11.2396	4	11
Transcription factor AP-1	Homo sapiens (human)	EC50	0.8100	2	2
Transient receptor potential cation channel subfamily A member 1	Homo sapiens (human)	EC50	19.2703	3	4
Transient receptor potential cation channel subfamily A member 1	Mus musculus (house mouse)	EC50	3.8000	1	1
Transient receptor potential cation channel subfamily M member 6	Homo sapiens (human)	Kd	10.0000	1	2
Transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	EC50	2.0575	4	4
Translocator protein	Rattus norvegicus (Norway rat)	EC50	0.0156	1	1
Transmembrane prolyl 4-hydroxylase	Homo sapiens (human)	EC50	50.0000	1	1
Transmembrane protease serine 2	Homo sapiens (human)	EC50	83.4000	1	1
Transthyretin	Homo sapiens (human)	EC50	26.8000	3	5
Transthyretin	Homo sapiens (human)	Kd	0.4000	2	2
Tubulin alpha-1A chain	Rattus norvegicus (Norway rat)	Kd	5.3850	1	2
Tyrosine--tRNA ligase, cytoplasmic	Homo sapiens (human)	Kd	30.0000	1	4
Tyrosine-protein kinase ABL1	Homo sapiens (human)	Kd	6.0803	30	55
Tyrosine-protein kinase ABL2	Homo sapiens (human)	Kd	17.0380	4	10
Tyrosine-protein kinase Blk	Homo sapiens (human)	Kd	5.0075	2	4
Tyrosine-protein kinase BTK	Homo sapiens (human)	Kd	15.6811	4	9
Tyrosine-protein kinase CSK	Homo sapiens (human)	Kd	15.6778	4	9
Tyrosine-protein kinase Fer	Homo sapiens (human)	Kd	15.5642	4	9
Tyrosine-protein kinase Fes/Fps	Homo sapiens (human)	Kd	17.5058	3	8
Tyrosine-protein kinase Fgr	Homo sapiens (human)	Kd	15.5627	4	9
Tyrosine-protein kinase FRK	Homo sapiens (human)	Kd	12.8350	4	10
Tyrosine-protein kinase Fyn	Homo sapiens (human)	Kd	18.1925	4	11
Tyrosine-protein kinase HCK	Homo sapiens (human)	Kd	15.5613	4	9
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	Kd	5.0095	2	4
Tyrosine-protein kinase JAK1	Homo sapiens (human)	Kd	17.0006	4	10
Tyrosine-protein kinase JAK2	Homo sapiens (human)	Kd	11.4331	4	7
Tyrosine-protein kinase JAK3	Homo sapiens (human)	Kd	5.0055	2	4
Tyrosine-protein kinase Lck	Homo sapiens (human)	Kd	13.9644	4	9
Tyrosine-protein kinase Lyn	Homo sapiens (human)	Kd	18.2082	4	11
Tyrosine-protein kinase Mer	Homo sapiens (human)	Kd	10.0026	3	5
Tyrosine-protein kinase receptor Tie-1	Homo sapiens (human)	Kd	5.0325	2	4
Tyrosine-protein kinase receptor TYRO3	Homo sapiens (human)	Kd	5.1400	2	4
Tyrosine-protein kinase receptor UFO	Homo sapiens (human)	Kd	5.0034	2	4
Tyrosine-protein kinase Srms	Homo sapiens (human)	Kd	5.3700	2	4
Tyrosine-protein kinase SYK	Homo sapiens (human)	EC50	27.6000	3	5
Tyrosine-protein kinase SYK	Homo sapiens (human)	Kd	15.5594	4	9
Tyrosine-protein kinase Tec	Homo sapiens (human)	Kd	17.8250	3	8
Tyrosine-protein kinase TXK	Homo sapiens (human)	Kd	2.3650	2	4
Tyrosine-protein kinase Yes	Homo sapiens (human)	Kd	15.5726	4	9
Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	Kd	5.0220	2	4
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	Kd	1,600.0000	1	1
U5 small nuclear ribonucleoprotein 200 kDa helicase	Homo sapiens (human)	Kd	30.0000	1	4
UDP-galactopyranose mutase	Klebsiella pneumoniae	Kd	69.0000	1	1
UDP-galactopyranose mutase	Mycobacterium tuberculosis H37Rv	Kd	653.0000	1	1
UMP-CMP kinase	Homo sapiens (human)	Kd	30.0000	1	5
Uncharacterized aarF domain-containing protein kinase 5	Homo sapiens (human)	Kd	30.0000	1	3
Uncharacterized protein FLJ45252	Homo sapiens (human)	Kd	30.0000	1	5
Uncharacterized serine/threonine-protein kinase SBK3	Homo sapiens (human)	Kd	5.0125	1	2
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	Kd	5.0750	2	4
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	Kd	4.1420	3	5
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	Kd	4.0174	3	5
Very long-chain specific acyl-CoA dehydrogenase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	5
Vitamin D3 receptor	Homo sapiens (human)	EC50	17.3801	3	3
Vitamin D3 receptor	Mus musculus (house mouse)	EC50	0.9000	1	1
Vitamin D3 receptor	Homo sapiens (human)	Kd	9.5733	3	3
voltage-dependent T-type calcium channel subunit alpha-1H isoform a	Homo sapiens (human)	EC50	5.1500	1	1
Wee1-like protein kinase	Homo sapiens (human)	Kd	17.9000	3	8
Wee1-like protein kinase 2	Homo sapiens (human)	Kd	10.0000	1	2
Zinc finger protein mex-5	Caenorhabditis elegans	EC50	7.2513	1	3

Other Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
2-5A-dependent ribonuclease	Homo sapiens (human)	Activity	30.0000	1	1
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	Activity	0.0100	1	1
5-hydroxytryptamine receptor 1B	Homo sapiens (human)	Activity	0.0280	1	1
5-hydroxytryptamine receptor 1D	Homo sapiens (human)	Activity	0.0009	1	1
5-hydroxytryptamine receptor 1D	Homo sapiens (human)	KA	35.0000	1	1
5-hydroxytryptamine receptor 1D	Rattus norvegicus (Norway rat)	Kb	0.0140	1	1
5-hydroxytryptamine receptor 1E	Homo sapiens (human)	Activity	1.6590	1	1
5-hydroxytryptamine receptor 2A	Homo sapiens (human)	Activity	0.0071	1	1
5-hydroxytryptamine receptor 2B	Homo sapiens (human)	Activity	0.0026	1	1
5-hydroxytryptamine receptor 2C	Rattus norvegicus (Norway rat)	Activity	0.0095	1	1
5-hydroxytryptamine receptor 3A	Homo sapiens (human)	Activity	10.0000	1	1
5-hydroxytryptamine receptor 4	Homo sapiens (human)	Activity	1.2740	1	1
5-hydroxytryptamine receptor 5A	Homo sapiens (human)	Activity	0.5620	1	1
5-hydroxytryptamine receptor 6	Homo sapiens (human)	Activity	0.0910	1	1
5-hydroxytryptamine receptor 6	Homo sapiens (human)	Kb	0.0168	2	2
5-hydroxytryptamine receptor 7	Homo sapiens (human)	Activity	0.0180	1	1
5-hydroxytryptamine receptor 7	Homo sapiens (human)	Kb	0.0001	2	2
Acetylcholinesterase	Electrophorus electricus (electric eel)	EC24	250.0000	1	1
Adenosine receptor A1	Homo sapiens (human)	Affinity constant	30.0000	1	1
Adenosine receptor A1	Rattus norvegicus (Norway rat)	Kb	60.0000	1	4
Adenosine receptor A1	Homo sapiens (human)	KD hydro	150,000.0000	1	1
Adenosine receptor A2a	Homo sapiens (human)	Affinity constant	30.0000	1	1
Adenosine receptor A2a	Rattus norvegicus (Norway rat)	Kb	36.0000	1	1
Adenosine receptor A2a	Rattus norvegicus (Norway rat)	Ratio	48.0000	1	2
Adenosine receptor A2b	Homo sapiens (human)	Affinity constant	30.0000	1	1
Adenosine receptor A2b	Mus musculus (house mouse)	Kb	25.0000	1	1
Adenosine receptor A2b	Rattus norvegicus (Norway rat)	Ratio	48.0000	1	2
Adenylate cyclase type 1	Homo sapiens (human)	Kb	30.0000	1	1
Alcohol dehydrogenase E chain	Equus caballus (horse)	Km	22.3000	1	1
Alcohol dehydrogenase S chain	Equus caballus (horse)	Km	22.3000	1	1
Alpha-1A adrenergic receptor	Homo sapiens (human)	Activity	0.0300	1	1
Alpha-1B adrenergic receptor	Homo sapiens (human)	Activity	0.1230	1	1
Alpha-1D adrenergic receptor	Homo sapiens (human)	Activity	0.0910	1	1
Alpha-2A adrenergic receptor	Homo sapiens (human)	Activity	0.0310	1	1
Alpha-2B adrenergic receptor	Homo sapiens (human)	Activity	0.0410	1	1
Alpha-2C adrenergic receptor	Homo sapiens (human)	Activity	0.0300	1	1
Amine oxidase [flavin-containing] A	Mus musculus (house mouse)	Activity	0.0010	2	6
Amine oxidase [flavin-containing] A	Rattus norvegicus (Norway rat)	Activity	0.0011	1	2
Amine oxidase [flavin-containing] B	Mus musculus (house mouse)	Activity	0.0009	2	6
Amine oxidase [flavin-containing] B	Rattus norvegicus (Norway rat)	Activity	0.0011	1	2
Amyloid-beta precursor protein	Homo sapiens (human)	DC50	0.7550	2	2
Androgen receptor	Homo sapiens (human)	EC150	26.3333	1	3
Arginase	Leishmania amazonensis	Kis	6.9000	1	1
Arylacetamide deacetylase	Homo sapiens (human)	Km	200.0000	1	2
ATP-dependent translocase ABCB1	Homo sapiens (human)	Activity	9.0333	3	3
ATP-dependent translocase ABCB1	Homo sapiens (human)	Ki1	200.0000	1	1
ATP-dependent translocase ABCB1	Homo sapiens (human)	Ki2	1,750.0000	1	1
ATP-dependent translocase ABCB1	Homo sapiens (human)	Km	4.1233	3	3
cAMP-dependent protein kinase catalytic subunit alpha isoform Calpha1	Homo sapiens (human)	AC50	0.8403	2	3
Carbonic anhydrase	Brucella suis 1330	Kinact	0.0180	1	1
Carbonic anhydrase 1	Homo sapiens (human)	KA	4.8667	3	3
Carbonic anhydrase 1	Homo sapiens (human)	Kinact	412.5000	1	2
Carbonic anhydrase 2	Homo sapiens (human)	KA	35.0000	2	2
Carbonic anhydrase 2	Homo sapiens (human)	Kinact	9.6000	1	2
Carbonic anhydrase 4	Bos taurus (cattle)	KA	18.0000	2	2
Carbonic anhydrase 4	Homo sapiens (human)	KA	15.0000	1	1
Carbonic anhydrase 5A, mitochondrial	Homo sapiens (human)	Kinact	0.0990	1	2
Carbonic anhydrase 5B, mitochondrial	Homo sapiens (human)	Kinact	0.0975	1	2
Caspase 6, apoptosis-related cysteine peptidase	Homo sapiens (human)	AC50	0.4610	1	1
Caspase-7	Homo sapiens (human)	AC50	5.4000	1	1
Chain A, BCL-2-RELATED PROTEIN A1	Homo sapiens (human)	AC50	697.4500	2	2
Cholinesterase	Equus caballus (horse)	EC16	250.0000	1	1
Cyclic AMP-responsive element-binding protein 1	Homo sapiens (human)	AC50	13.5000	1	1
Cyclin-dependent kinase 1	Homo sapiens (human)	ID50	0.2175	2	2
cystic fibrosis transmembrane conductance regulator ATP-binding cassette sub-family C member 7	Homo sapiens (human)	AC50	7.7400	1	1
Cytochrome P450 1A1	Homo sapiens (human)	Km	803.0000	1	1
Cytochrome P450 1A1	Rattus norvegicus (Norway rat)	Ks	870.0000	1	1
Cytochrome P450 1A2	Homo sapiens (human)	INH	10.0000	1	1
Cytochrome P450 1A2	Homo sapiens (human)	Km	120.0000	1	1
Cytochrome P450 2B1	Rattus norvegicus (Norway rat)	Ks	800.0000	1	1
Cytochrome P450 2D6	Homo sapiens (human)	INH	3.6000	1	1
Cytochrome P450 3A4	Homo sapiens (human)	INH	10.0000	1	1
D(1A) dopamine receptor	Homo sapiens (human)	Activity	0.0090	1	1
D(2) dopamine receptor	Homo sapiens (human)	Activity	0.0740	1	1
D(3) dopamine receptor	Rattus norvegicus (Norway rat)	Activity	0.0140	1	1
D(4) dopamine receptor	Homo sapiens (human)	Activity	0.0049	1	1
Delta-type opioid receptor	Homo sapiens (human)	Activity	0.0189	1	1
Delta-type opioid receptor	Rattus norvegicus (Norway rat)	Activity	0.6115	2	2
Delta-type opioid receptor	Homo sapiens (human)	ED50	0.3160	1	1
Delta-type opioid receptor	Mus musculus (house mouse)	Ke	0.0074	1	1
Dihydrofolate reductase	Homo sapiens (human)	Activity	0.9200	1	1
Dihydroxyacetone phosphate acyltransferase	Homo sapiens (human)	Radius of inhibition zone	9,214.2857	7	7
DNA repair protein RAD52 homolog isoform a	Homo sapiens (human)	AC50	13.6600	1	1
DNA topoisomerase 1	Homo sapiens (human)	MIC	27.5000	1	2
dual specificity tyrosine-phosphorylation-regulated kinase 1A	Rattus norvegicus (Norway rat)	AC50	7.7737	1	3
Egl nine homolog 1	Homo sapiens (human)	Km	180.0000	1	1
EWS/FLI fusion protein	Homo sapiens (human)	AbsAC35_uM	40.2500	1	1
FAD-linked sulfhydryl oxidase ALR	Homo sapiens (human)	AC50	0.5280	1	2
FATTY-ACID-CoA LIGASE FADD28 (FATTY-ACID-CoA SYNTHETASE) (FATTY-ACID-CoA SYNTHASE)	Mycobacterium tuberculosis H37Rv	AC50	63.7200	1	2
fibroblast growth factor 22 isoform 1 precursor	Homo sapiens (human)	AbsAC1_uM	4.3700	1	1
fMet-Leu-Phe receptor	Homo sapiens (human)	IC20	3.6000	1	1
G2/mitotic-specific cyclin-B1	Homo sapiens (human)	ID50	0.2175	2	2
G2/mitotic-specific cyclin-B2	Homo sapiens (human)	ID50	0.2175	2	2
G2/mitotic-specific cyclin-B3	Homo sapiens (human)	ID50	0.2175	2	2
Glucocorticoid receptor	Homo sapiens (human)	EC150	26.3333	1	3
Glutamate dehydrogenase 1, mitochondrial	Bos taurus (cattle)	Km	20.0000	1	1
glycogen synthase kinase-3 alpha	Homo sapiens (human)	AC50	114.3043	1	3
heat shock protein 90, putative	Plasmodium falciparum 3D7	AC50	5.7407	1	3
heat shock protein HSP 90-alpha isoform 2	Homo sapiens (human)	AC50	4.7830	1	3
Histamine H1 receptor	Homo sapiens (human)	Activity	0.0982	1	1
Histamine H2 receptor	Homo sapiens (human)	Activity	0.1040	1	1
Histamine H2 receptor	Cavia porcellus (domestic guinea pig)	K0.5	0.0003	1	2
Histamine H4 receptor	Homo sapiens (human)	Activity	0.0127	1	1
Histone deacetylase 1	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 1	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 11	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 11	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 2	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 2	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 3	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 3	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 4	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 4	Homo sapiens (human)	EC1000	0.0200	1	1
Histone deacetylase 4	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 5	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 5	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 6	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 6	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 7	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 7	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 8	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 8	Homo sapiens (human)	Inhibition	0.0035	1	1
Histone deacetylase 9	Homo sapiens (human)	AC50	0.4000	1	1
Histone deacetylase 9	Homo sapiens (human)	Inhibition	0.0035	1	1
histone-lysine N-methyltransferase NSD2 isoform 1	Homo sapiens (human)	AC50	0.2930	1	1
HSP40, subfamily A [Plasmodium falciparum 3D7]	Plasmodium falciparum 3D7	AbsAC1000_uM	1.5580	1	1
Hypoxia-inducible factor 1-alpha inhibitor	Homo sapiens (human)	Km	260.0000	1	1
Inosine-5'-monophosphate dehydrogenase 1	Homo sapiens (human)	Km	100.0000	1	1
Inosine-5'-monophosphate dehydrogenase 2	Homo sapiens (human)	Km	100.0000	1	1
interferon gamma precursor	Homo sapiens (human)	AC50	18.5200	2	3
Kappa-type opioid receptor	Rattus norvegicus (Norway rat)	Activity	0.0331	2	2
Kappa-type opioid receptor	Homo sapiens (human)	ED50	1.1400	1	1
Kappa-type opioid receptor	Mus musculus (house mouse)	Ke	0.0288	2	2
L-lactate dehydrogenase B chain	Sus scrofa (pig)	Km	84.4000	1	1
Lactoperoxidase	Bos taurus (cattle)	Km	59.1333	1	3
Malate dehydrogenase, cytoplasmic	Sus scrofa (pig)	Km	33.9000	1	1
Microphthalmia-associated transcription factor	Homo sapiens (human)	AC50	9.1160	5	5
Microtubule-associated protein tau	Homo sapiens (human)	DC50	200.0000	1	1
Mitogen-activated protein kinase 3	Homo sapiens (human)	Activity	10.0000	1	1
Mu-type opioid receptor	Mus musculus (house mouse)	Activity	0.0010	1	1
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	Activity	0.0030	1	1
Mu-type opioid receptor	Homo sapiens (human)	ED50	0.0370	2	2
Mu-type opioid receptor	Mus musculus (house mouse)	Ke	0.0033	1	1
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	KiH	0.0025	1	1
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	KiL	0.1130	1	1
Muscarinic acetylcholine receptor	Cavia porcellus (domestic guinea pig)	Kb	25.0000	1	1
Muscarinic acetylcholine receptor M1	Homo sapiens (human)	Activity	0.0012	1	1
Muscarinic acetylcholine receptor M2	Homo sapiens (human)	Activity	0.0177	1	1
Muscarinic acetylcholine receptor M3	Homo sapiens (human)	Activity	0.0038	1	1
Muscarinic acetylcholine receptor M4	Homo sapiens (human)	Activity	0.0369	1	1
NAD-dependent protein deacetylase sirtuin-1	Homo sapiens (human)	Km	80.0000	1	1
NADP-dependent malic enzyme, mitochondrial	Homo sapiens (human)	Activity	960.0000	1	1
Non-lysosomal glucosylceramidase	Mus musculus (house mouse)	Activity	11.0000	1	1
Nuclear factor erythroid 2-related factor 2	Homo sapiens (human)	Activity	1.5080	5	5
Nuclear factor erythroid 2-related factor 2	Homo sapiens (human)	CD	60.0000	1	1
Pancreatic alpha-amylase	Sus scrofa (pig)	Kii	5.8700	1	1
Pancreatic alpha-amylase	Sus scrofa (pig)	Kis	31.6000	1	1
Peroxisome proliferator-activated receptor gamma	Homo sapiens (human)	Activity	3.1400	2	2
Phosphatidylinositol 3-kinase regulatory subunit alpha	Homo sapiens (human)	INH	0.0160	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	INH	0.0089	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	Imax	25.0000	2	2
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	INH	0.0170	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	Homo sapiens (human)	INH	0.0160	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Homo sapiens (human)	INH	0.0530	1	1
Photosystem I iron-sulfur center	Panicum virgatum (switchgrass)	Activity	110.0000	1	1
Polyamine deacetylase HDAC10	Homo sapiens (human)	AC50	0.4000	1	1
Polyamine deacetylase HDAC10	Homo sapiens (human)	Inhibition	0.0035	1	1
Polyphenol oxidase 2	Agaricus bisporus	ID50	70.0000	1	1
Polyunsaturated fatty acid 5-lipoxygenase	Rattus norvegicus (Norway rat)	Change	50.0000	2	2
Prenyltransferase homolog	Streptomyces coelicolor A3(2)	Km	330.0000	1	1
Prolyl 4-hydroxylase subunit alpha-1	Homo sapiens (human)	Km	300.0000	1	1
Prolyl hydroxylase EGLN2	Homo sapiens (human)	Km	170.0000	1	1
Prolyl hydroxylase EGLN3	Homo sapiens (human)	Km	140.0000	1	1
prostaglandin E2 receptor EP2 subtype	Homo sapiens (human)	Active Concentration	20.0000	1	1
Prostaglandin E2 receptor EP3 subtype	Homo sapiens (human)	Activity	0.0217	1	1
Prostaglandin E2 receptor EP4 subtype	Homo sapiens (human)	Activity	0.0152	1	1
Prostaglandin G/H synthase 1	Homo sapiens (human)	Inhibition	15.0000	1	1
Prostaglandin G/H synthase 1	Rattus norvegicus (Norway rat)	Change	0.6000	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	INH	26.0000	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	Inhibition	0.0280	1	1
Prostaglandin G/H synthase 2	Rattus norvegicus (Norway rat)	Change	0.6000	1	1
protein AF-9 isoform a	Homo sapiens (human)	AC50	6.3100	1	1
Proteinase-activated receptor 1	Homo sapiens (human)	Imax	25.0000	2	2
Quinone oxidoreductase	Mus musculus (house mouse)	Activity	4.6433	3	3
Quinone oxidoreductase	Mus musculus (house mouse)	CD	10.4000	3	4
replicative DNA helicase	Mycobacterium tuberculosis H37Rv	AC50	260.7200	2	3
scavenger receptor class B member 1 isoform 1	Mus musculus (house mouse)	AbsAC40_uM	35.0000	1	1
scavenger receptor class B member 1 isoform 1	Mus musculus (house mouse)	AC50	87.8300	1	1
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	Km	114.8000	2	2
Seed linoleate 13S-lipoxygenase-1	Glycine max (soybean)	Vmax	0.0070	2	2
serine/threonine-protein kinase 33 isoform a	Homo sapiens (human)	AC50	9.3400	2	3
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	-Log IC50	0.0900	1	2
Skn7p	Saccharomyces cerevisiae (brewer's yeast)	AbsAC40_uM	12.6100	1	1
Sodium channel protein type 4 subunit alpha	Homo sapiens (human)	Kr	1,440.0000	1	1
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	Activity	1.1320	1	1
Sodium-dependent serotonin transporter	Homo sapiens (human)	Activity	0.0897	1	1
Solute carrier family 22 member 1	Rattus norvegicus (Norway rat)	Km	147.1333	1	3
Solute carrier organic anion transporter family member 1A1	Rattus norvegicus (Norway rat)	Km	252.0000	1	1
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	Km	7.2500	2	2
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	Km	2.3000	1	1
Substance-P receptor	Cavia porcellus (domestic guinea pig)	CD	11.0000	1	1
Sulfate anion transporter 1	Mus musculus (house mouse)	Km	151.0000	1	1
Sulfotransferase 1A1	Rattus norvegicus (Norway rat)	Km	92.0000	1	1
toxin B	Clostridioides difficile 630	AC50	20.8700	1	1
Type II pantothenate kinase	Staphylococcus aureus subsp. aureus MSSA476	Km	19.0000	1	1
Type III pantothenate kinase	Pseudomonas aeruginosa PAO1	Km	20.0000	1	1
UDP-glucuronosyltransferase 1-6	Homo sapiens (human)	Km	2,200.0000	1	1
UDP-glucuronosyltransferase 1A1	Homo sapiens (human)	Km	9,400.0000	1	1
UDP-glucuronosyltransferase 1A3	Homo sapiens (human)	Km	1,755.0000	1	2
UDP-glucuronosyltransferase 1A9	Homo sapiens (human)	Km	20,900.0000	1	1
UDP-glucuronosyltransferase 2B7	Homo sapiens (human)	Km	128.5000	1	2
unnamed protein product	Saccharomyces cerevisiae (brewer's yeast)	AC50	0.0008	1	1
Vasopressin V2 receptor	Sus scrofa (pig)	Kb	30.0000	1	1
Vitamin D3 receptor	Homo sapiens (human)	Activity	2,159.0000	4	4
Vitamin D3 receptor	Homo sapiens (human)	K	100.0000	1	1
Xanthine dehydrogenase/oxidase	Bos taurus (cattle)	Km	65.3000	4	4

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