Proteins > ubiquitin carboxyl-terminal hydrolase 2 isoform a
Page last updated: 2024-08-07 19:23:47

ubiquitin carboxyl-terminal hydrolase 2 isoform a

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (623)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
quinacrineHomo sapiens (human)Potency14.689210
thyroxineHomo sapiens (human)Potency25.118910
5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)-3,4-dihydro-2H-chromen-3-yl 3,4,5-trihydroxybenzoateHomo sapiens (human)Potency25.118910
4-amino-1,8-naphthalimideHomo sapiens (human)Potency14.689210
5,8,11,14-eicosatetraynoic acidHomo sapiens (human)Potency28.183810
tyrphostin 25Homo sapiens (human)Potency25.118910
amoxapineHomo sapiens (human)Potency19.952610
anthralinHomo sapiens (human)Potency25.118910
astemizoleHomo sapiens (human)Potency8.800610
aurintricarboxylic acidHomo sapiens (human)Potency7.371530
benzbromaroneHomo sapiens (human)Potency0.631010
bay h 4502Homo sapiens (human)Potency25.118910
broxyquinolineHomo sapiens (human)Potency3.981110
bumetanideHomo sapiens (human)Potency6.309610
busulfanHomo sapiens (human)Potency15.848910
calmidazoliumHomo sapiens (human)Potency13.091810
candesartan cilexetilHomo sapiens (human)Potency0.794310
chelerythrineHomo sapiens (human)Potency25.118910
chromone-2-carboxylic acidHomo sapiens (human)Potency31.622810
clioquinolHomo sapiens (human)Potency1.790110
clofoctolHomo sapiens (human)Potency10.000010
clotrimazoleHomo sapiens (human)Potency18.933810
dephostatinHomo sapiens (human)Potency15.848910
dichlorophenHomo sapiens (human)Potency25.118910
diflunisalHomo sapiens (human)Potency6.309610
dipyridamoleHomo sapiens (human)Potency10.449030
domperidoneHomo sapiens (human)Potency10.000010
adtnHomo sapiens (human)Potency1.166810
embelinHomo sapiens (human)Potency3.162310
erythrosineHomo sapiens (human)Potency11.220210
fenofibrateHomo sapiens (human)Potency6.309610
fluphenazineHomo sapiens (human)Potency18.854110
fluspirileneHomo sapiens (human)Potency7.943310
fosfosalHomo sapiens (human)Potency3.981110
gabapentinHomo sapiens (human)Potency14.689210
gossypolHomo sapiens (human)Potency13.069730
hexachloropheneHomo sapiens (human)Potency10.253830
batyl alcoholHomo sapiens (human)Potency25.118910
indirubin-3'-monoximeHomo sapiens (human)Potency25.118910
iodoacetamideHomo sapiens (human)Potency25.118910
iodoquinolHomo sapiens (human)Potency0.316210
jugloneHomo sapiens (human)Potency12.589310
lidoflazineHomo sapiens (human)Potency10.000010
loperamideHomo sapiens (human)Potency5.011910
loratadineHomo sapiens (human)Potency12.589310
mebendazoleHomo sapiens (human)Potency15.848910
meclofenamate sodium anhydrousHomo sapiens (human)Potency10.000010
vitamin k 3Homo sapiens (human)Potency6.309610
methyl methanesulfonateHomo sapiens (human)Potency15.848910
mitoxantroneHomo sapiens (human)Potency14.689210
etoposide phosphateHomo sapiens (human)Potency10.000010
papaverineHomo sapiens (human)Potency12.589310
pargylineHomo sapiens (human)Potency5.011910
pentoxifyllineHomo sapiens (human)Potency25.118910
perphenazineHomo sapiens (human)Potency12.589310
phenazopyridineHomo sapiens (human)Potency3.981110
pipobromanHomo sapiens (human)Potency10.000010
pirenzepineHomo sapiens (human)Potency12.589310
piretanideHomo sapiens (human)Potency7.943310
piribedilHomo sapiens (human)Potency3.981110
pomiferinHomo sapiens (human)Potency10.000010
protoporphyrin ixHomo sapiens (human)Potency14.689210
1,2,5,8-tetrahydroxy anthraquinoneHomo sapiens (human)Potency3.981110
quipazineHomo sapiens (human)Potency5.011910
raloxifeneHomo sapiens (human)Potency5.011910
riluzoleHomo sapiens (human)Potency5.011910
roxarsoneHomo sapiens (human)Potency1.258910
saccharinHomo sapiens (human)Potency19.952610
sanguinarineHomo sapiens (human)Potency25.118910
spiperoneHomo sapiens (human)Potency15.848910
sulfamethoxazoleHomo sapiens (human)Potency43.239710
sulfanilamideHomo sapiens (human)Potency10.000010
sulfasalazineHomo sapiens (human)Potency6.309610
ticlopidineHomo sapiens (human)Potency10.000010
ici 136,753Homo sapiens (human)Potency7.943310
trigonellineHomo sapiens (human)Potency12.589310
6,18,30-trimethyl-3,9,12,15,21,24,27,33,36-nona(propan-2-yl)-1,7,13,19,25,31-hexaoxa-4,10,16,22,28,34-hexazacyclohexatriacontane-2,5,8,11,14,17,20,23,26,29,32,35-dodeconeHomo sapiens (human)Potency12.589310
alloxanHomo sapiens (human)Potency10.000010
levodopaHomo sapiens (human)Potency20.749110
papaverine hydrochlorideHomo sapiens (human)Potency12.589310
quinacrine monohydrochlorideHomo sapiens (human)Potency0.631010
7,8-dimethyl-10-[(2R,3R,4S)-2,3,4,5-tetrahydroxypentyl]benzo[g]pteridine-2,4-dioneHomo sapiens (human)Potency10.000010
acriflavine chlorideHomo sapiens (human)Potency0.631010
pyronineHomo sapiens (human)Potency11.220210
betazoleHomo sapiens (human)Potency5.011910
methylergonovineHomo sapiens (human)Potency14.689210
benzethonium chlorideHomo sapiens (human)Potency25.732420
2,4-dihydroxybenzophenoneHomo sapiens (human)Potency11.220210
amprolium hydrochlorideHomo sapiens (human)Potency2.511910
triflusalHomo sapiens (human)Potency5.011910
chrysophanic acidHomo sapiens (human)Potency25.118910
gentian violetHomo sapiens (human)Potency10.000010
2-amino-4-phenylphenolHomo sapiens (human)Potency3.162310
lysergolHomo sapiens (human)Potency3.981110
5-hydroxyindoleHomo sapiens (human)Potency7.943310
pimozideHomo sapiens (human)Potency2.511910
pontamine sky blueHomo sapiens (human)Potency10.000010
piperacetazineHomo sapiens (human)Potency5.011910
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazineHomo sapiens (human)Potency2.238710
hydroxyzine pamoateHomo sapiens (human)Potency5.011910
diacereinHomo sapiens (human)Potency25.118910
metergolineHomo sapiens (human)Potency10.000010
methyldopaHomo sapiens (human)Potency22.387210
s-2678Homo sapiens (human)Potency14.125410
idarubicinHomo sapiens (human)Potency16.481610
mitoxantrone hydrochlorideHomo sapiens (human)Potency25.118910
chaetochrominHomo sapiens (human)Potency11.679930
topotecan hydrochlorideHomo sapiens (human)Potency10.000010
daunorubicin hydrochlorideHomo sapiens (human)Potency10.000010
verapamil hydrochlorideHomo sapiens (human)Potency10.000010
diacetylfluoresceinHomo sapiens (human)Potency7.079510
sulconazole, mononitrate, (+-)-isomerHomo sapiens (human)Potency25.118910
telmisartanHomo sapiens (human)Potency10.000010
trifluoperazine hydrochlorideHomo sapiens (human)Potency15.848910
xanthoxylineHomo sapiens (human)Potency15.848910
fluphenazine hydrochlorideHomo sapiens (human)Potency10.000010
2,3-trimethylene-4-quinazoloneHomo sapiens (human)Potency3.981110
2,6-dimethoxy-1,4-benzoquinoneHomo sapiens (human)Potency7.943310
miconazole nitrateHomo sapiens (human)Potency25.118910
econazole nitrateHomo sapiens (human)Potency19.952610
masoprocolHomo sapiens (human)Potency31.622810
aceclofenacHomo sapiens (human)Potency3.162310
fluphenacurHomo sapiens (human)Potency12.589310
nonoxynol-9Homo sapiens (human)Potency2.511910
coumarin 153Homo sapiens (human)Potency3.981110
methyl fluorone blackHomo sapiens (human)Potency28.183810
9-hydroxyphenylfluoronHomo sapiens (human)Potency28.183810
ergocornineHomo sapiens (human)Potency11.220210
pramoxine hydrochlorideHomo sapiens (human)Potency12.589310
atovaquoneHomo sapiens (human)Potency10.000010
1,8-diazabicyclo(5.4.0)undec-7-eneHomo sapiens (human)Potency15.848910
2-butyl-6-(butylamino)-1h-benzo(de)isoquinoline-1,3(2h)-dioneHomo sapiens (human)Potency6.309610
sennoside BHomo sapiens (human)Potency1.995310
prochlorperazine edisylate saltHomo sapiens (human)Potency12.589310
coumarin 7Homo sapiens (human)Potency0.430120
osajinHomo sapiens (human)Potency15.848910
4-methoxydalbergioneHomo sapiens (human)Potency12.589310
alexidine dihydrchlorideHomo sapiens (human)Potency31.622810
cv 3988Homo sapiens (human)Potency14.689210
6-hydroxydopaHomo sapiens (human)Potency14.420020
alpha-ergocryptineHomo sapiens (human)Potency11.220210
harmalol hydrochlorideHomo sapiens (human)Potency1.584910
sb 216763Homo sapiens (human)Potency16.481610
chrysene-1,4-dioneHomo sapiens (human)Potency3.162310
benfluorex hydrochlorideHomo sapiens (human)Potency25.118910
gossypol acetic acidHomo sapiens (human)Potency5.623410
methylnaphthazarinHomo sapiens (human)Potency22.387210
nsc-260594Homo sapiens (human)Potency17.437220
4-amino-N-(4-methoxyphenyl)-2-(methylthio)-5-thiazolecarboxamideHomo sapiens (human)Potency25.118910
5-demethylnobiletinHomo sapiens (human)Potency10.000010
2,3-diaminophenazineHomo sapiens (human)Potency15.848910
s-(4-azidophenacyl)glutathioneHomo sapiens (human)Potency14.689210
doxorubicin hydrochlorideHomo sapiens (human)Potency10.000010
arachidonic acidHomo sapiens (human)Potency3.162310
retinolHomo sapiens (human)Potency10.000010
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolHomo sapiens (human)Potency25.118910
diethylstilbestrolHomo sapiens (human)Potency25.118910
6-bromoindirubin-3'-oximeHomo sapiens (human)Potency12.589310
isotetrandrineHomo sapiens (human)Potency10.000010
IPA-3Homo sapiens (human)Potency14.689210
2-furancarboxylic acid [4-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterHomo sapiens (human)Potency3.162310
2-[[(6-bromo-1H-benzimidazol-2-yl)thio]methyl]-1-methylbenzimidazoleHomo sapiens (human)Potency6.309610
tolfenamic acidHomo sapiens (human)Potency10.000010
4-(2-pyridinylthio)benzofuro[3,2-d]pyrimidineHomo sapiens (human)Potency3.981110
calmidazoliumHomo sapiens (human)Potency14.880630
N-(2-fluorophenyl)-2-(3-methoxyphenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamideHomo sapiens (human)Potency15.848910
3-[[2-[[4-ethyl-5-[(4-methylanilino)methyl]-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency10.000010
3-[(1-cyclopentyl-5-tetrazolyl)-(3,4-dihydro-1H-isoquinolin-2-yl)methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency5.011910
3-[[1,3-benzodioxol-5-ylmethyl-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency6.309610
1-(2-furanyl)-N-[[1-[(4-methylphenyl)sulfonylmethyl]-5-tetrazolyl]methyl]-N-(thiophen-2-ylmethyl)methanamineHomo sapiens (human)Potency12.589310
N-[2-(cyclohexylamino)-1-(2-furanyl)-2-oxoethyl]-N-(2-furanylmethyl)-2-furancarboxamideHomo sapiens (human)Potency5.011910
LSM-19079Homo sapiens (human)Potency10.000010
3-amino-N-cyclopentyl-6-thiophen-2-yl-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency5.011910
2-[[4-(3-methoxyphenyl)-5-[(4-methylphenoxy)methyl]-1,2,4-triazol-3-yl]thio]acetic acidHomo sapiens (human)Potency12.589310
2-[(5,5-dimethyl-6H-[1,2,4]triazolo[3,4-a]isoquinolin-3-yl)thio]-1-[4-(2-methoxyphenyl)-1-piperazinyl]ethanoneHomo sapiens (human)Potency12.589310
2-[[3-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]acetic acid methyl esterHomo sapiens (human)Potency12.589310
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[[1-(3,4-dimethoxyphenyl)-5-tetrazolyl]thio]acetamideHomo sapiens (human)Potency7.943310
2-[[2-[[4-(2-furanylmethyl)-5-(phenylmethyl)-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideHomo sapiens (human)Potency10.000010
2-(6-cyano-1-indolyl)-N-cyclohexylacetamideHomo sapiens (human)Potency25.118910
6-[[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]quinolineHomo sapiens (human)Potency5.011910
6-amino-4-(2-methoxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileHomo sapiens (human)Potency12.589310
7,8-dimethyl-1-[2-oxo-2-(1-pyrrolidinyl)ethyl]-4-phenyl-3H-1,5-benzodiazepin-2-oneHomo sapiens (human)Potency10.000010
4-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-2-methyl-5-thieno[3,2-b]pyrrolecarboxylic acid ethyl esterHomo sapiens (human)Potency5.011910
N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-cyclohexyl-2-furancarboxamideHomo sapiens (human)Potency10.000010
5-(diethylsulfamoyl)-3-hydroxy-2-naphthalenecarboxylic acidHomo sapiens (human)Potency6.309610
N-[4-[3-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-2-hydroxypropoxy]phenyl]acetamideHomo sapiens (human)Potency10.000010
N,N-dimethyl-6-phenyl-3-pyridazinamineHomo sapiens (human)Potency3.162310
3-[[1,3-benzodioxol-5-ylmethyl-[(1-cyclopentyl-5-tetrazolyl)methyl]amino]methyl]-6-ethyl-1H-quinolin-2-oneHomo sapiens (human)Potency5.011910
1-(1-adamantyl)-3-[8-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]ureaHomo sapiens (human)Potency12.589310
2-[cyclohexyl-(2,4,6-trimethylphenyl)sulfonylamino]-N-(3-pyridinylmethyl)acetamideHomo sapiens (human)Potency12.589310
1-(4-chlorophenyl)sulfonyl-N-[3-methoxy-4-(1-tetrazolyl)phenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency12.589310
2-[(5-amino-1-phenacyl-1,2,4-triazol-3-yl)thio]-N-(3-cyano-4,5-dimethyl-2-thiophenyl)acetamideHomo sapiens (human)Potency15.848910
3-[[[1-[1-(2-furanylmethyl)-5-tetrazolyl]-2-methylpropyl]-(2-oxolanylmethyl)amino]methyl]-8-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency25.118910
N-[4-[[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]sulfonyl]phenyl]acetamideHomo sapiens (human)Potency12.589310
4-[4-[[1-[(4-methoxyphenyl)methyl]-5-tetrazolyl]-(3-pyridinyl)methyl]-1-piperazinyl]phenolHomo sapiens (human)Potency19.952610
8-[(1-cyclohexyl-5-tetrazolyl)methyl]-3-(4-fluorophenyl)-8-azabicyclo[3.2.1]octan-3-olHomo sapiens (human)Potency12.589310
4-methoxy-1,3-dimethyl-6-thiophen-2-yl-8-cyclohepta[c]furanoneHomo sapiens (human)Potency7.943310
6-methyl-3-[[[1-(phenylmethyl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency12.589310
4-[2-[1-(4-methoxyphenyl)sulfonyl-2-benzimidazolyl]ethyl]morpholineHomo sapiens (human)Potency25.118910
5-(2-furanyl)-3-[2-methoxy-6-(4-methylphenyl)-3-pyridinyl]-1,2,4-oxadiazoleHomo sapiens (human)Potency7.943310
6-ethoxy-3-[[2-oxolanylmethyl-[[1-(2-phenylethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
3-[1-azepanyl-[1-(phenylmethyl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency12.589310
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-[[3-(2-furanylmethyl)-4-oxo-2-quinazolinyl]thio]acetamideHomo sapiens (human)Potency5.011910
5-(1,3-benzodioxol-5-yl)-1-methyl-2-imidazolamineHomo sapiens (human)Potency15.848910
4,5-dichloro-3-isothiazolecarboxylic acid [1-(2-furanylmethylamino)-1-oxopropan-2-yl] esterHomo sapiens (human)Potency12.589310
3-[[[1-(2-furanylmethyl)-5-tetrazolyl]methyl-[(2-methoxyphenyl)methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency2.511910
2-[4-(4-fluorophenyl)sulfonyl-1-piperazinyl]-4-(3-methoxyphenyl)thiazoleHomo sapiens (human)Potency7.943310
N-[4-[oxo-(2-pyridinylamino)methyl]phenyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
1-(1,3-benzodioxol-5-ylmethyl)-3-(4-methylphenyl)-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]ureaHomo sapiens (human)Potency3.981110
N'-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]-N'-(3-fluorophenyl)-N-(3-pyridinyl)butanediamideHomo sapiens (human)Potency15.848910
1-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-3,4-dihydro-2H-quinolineHomo sapiens (human)Potency10.000010
N-(1,3-benzodioxol-5-yl)-1-[(4-fluorophenyl)methyl]-4-triazolecarboxamideHomo sapiens (human)Potency7.943310
N-tert-butyl-2-(2-furanyl)-2-[[2-[5-(5-methyl-2-furanyl)-2-tetrazolyl]-1-oxoethyl]-(thiophen-2-ylmethyl)amino]acetamideHomo sapiens (human)Potency12.589310
2-[(1-cyclohexyl-5-tetrazolyl)thio]-N-(6-ethoxy-1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)Potency12.589310
[5-(2-furanyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency15.848910
2-[4-[(1-cyclopentyl-5-tetrazolyl)-(6-quinolinyl)methyl]-1-piperazinyl]-1,3-benzothiazoleHomo sapiens (human)Potency3.981110
1-(3,5-dimethyl-1-pyrazolyl)-3-[2-(4-methoxyphenyl)-1-indolyl]-2-propanolHomo sapiens (human)Potency12.589310
1-(4-fluorophenyl)-4-[[1-(2-phenylethyl)-5-tetrazolyl]-thiophen-2-ylmethyl]piperazineHomo sapiens (human)Potency12.589310
6,7-dimethoxy-2-[[2-[4-(4-methoxyphenyl)-1-piperazinyl]-2-oxoethyl]thio]-3-quinolinecarbonitrileHomo sapiens (human)Potency5.011910
N-[4-[(tert-butylamino)-oxomethyl]phenyl]-2,3-dihydro-1,4-benzodioxin-3-carboxamideHomo sapiens (human)Potency12.589310
N-(2,5-diethoxyphenyl)-2-[(3-methyl-2-imidazo[4,5-b]pyridinyl)thio]acetamideHomo sapiens (human)Potency0.251210
2,5-diethoxy-N-[2-(2-methylphenyl)ethyl]-4-(1-tetrazolyl)benzenesulfonamideHomo sapiens (human)Potency3.162310
6-chloro-2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-piperidinyl]-1H-benzimidazoleHomo sapiens (human)Potency12.589310
4-[[4-ethyl-5-[(2-methylphenoxy)methyl]-1,2,4-triazol-3-yl]thio]-N-(2-methoxyphenyl)-3-oxobutanamideHomo sapiens (human)Potency10.000010
3-(3-chlorophenyl)-1-(3-hydroxypropyl)-1-[(8-methyl-2-oxo-1H-quinolin-3-yl)methyl]ureaHomo sapiens (human)Potency12.589310
4-bromo-N-[(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-hydroxyethyl)benzamideHomo sapiens (human)Potency19.952610
6-ethoxy-3-[[[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency19.952610
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency5.011910
2-[[5-(phenoxymethyl)-4-(2-phenylethyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency12.589310
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency10.000010
N'-[2-(cyclopentylamino)-2-oxoethyl]-N'-(3,4-dimethylphenyl)-N-(2-pyridinyl)pentanediamideHomo sapiens (human)Potency5.011910
N-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-[[4-propyl-5-(2-pyridinyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency10.000010
3-(2-chlorophenyl)-1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-[2-(1-pyrrolidinyl)ethyl]ureaHomo sapiens (human)Potency12.589310
2-[4-(benzenesulfonyl)phenyl]-5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency7.943310
4-(1-methylsulfonyl-2,3-dihydroindol-5-yl)-N-(2-oxolanylmethyl)-2-thiazolamineHomo sapiens (human)Potency25.118910
1-[4-(2-methoxyphenyl)-1-piperazinyl]-2-[[5-(2-methyl-3-furanyl)-1,3,4-oxadiazol-2-yl]thio]ethanoneHomo sapiens (human)Potency12.589310
8-[(1-tert-butyl-5-tetrazolyl)-thiomorpholin-4-ylmethyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneHomo sapiens (human)Potency10.000010
1-[1-[1-(1,3-benzodioxol-5-ylmethyl)-5-tetrazolyl]-2-methylpropyl]-4-phenylpiperazineHomo sapiens (human)Potency19.952610
1-cyclopentyl-1-[(7-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-(2-methoxyphenyl)ureaHomo sapiens (human)Potency10.000010
3-[2-(3-phenoxypropyl)-5-tetrazolyl]pyridineHomo sapiens (human)Potency12.589310
2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)thio]-N-(4-phenyl-2-thiazolyl)acetamideHomo sapiens (human)Potency6.309610
2-[(5,5-dimethyl-6H-[1,2,4]triazolo[3,4-a]isoquinolin-3-yl)thio]-1-(4-phenyl-1-piperazinyl)ethanoneHomo sapiens (human)Potency10.000010
2-[2-[[2-[[1-(4-methoxyphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esterHomo sapiens (human)Potency10.000010
1-[1-[[1-[(4-methylphenyl)methyl]-5-tetrazolyl]methyl]-4-piperidinyl]-5-(trifluoromethyl)benzotriazoleHomo sapiens (human)Potency3.981110
N-(1,3-benzodioxol-5-yl)-N-[1-(4-chlorophenyl)-2-(cyclohexylamino)-2-oxoethyl]-2-pyrazinecarboxamideHomo sapiens (human)Potency5.011910
LSM-34623Homo sapiens (human)Potency10.000010
LSM-34679Homo sapiens (human)Potency12.589310
2-[(3-cyano-5,7-dimethyl-2-quinolinyl)thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency3.981110
3-[[cyclopentyl-[[1-[(4-methoxyphenyl)methyl]-5-tetrazolyl]methyl]amino]methyl]-7-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
1-(2-methoxyphenyl)-4-[(4-methylphenyl)-(1-propan-2-yl-5-tetrazolyl)methyl]piperazineHomo sapiens (human)Potency10.000010
N,N-diethyl-2-[(3-thiophen-2-yl-7-isothiazolo[4,5-d]pyrimidinyl)thio]acetamideHomo sapiens (human)Potency3.162310
3-[[1-(1,3-benzodioxol-5-ylmethyl)-5-tetrazolyl]-(1-pyrrolidinyl)methyl]-8-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency12.589310
N-(2-ethoxyphenyl)-1-[4-(1-pyrrolidinylsulfonyl)phenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency12.589310
2-(2-cyanophenoxy)-N-[2-[cyclopropyl(oxo)methyl]-3-benzofuranyl]acetamideHomo sapiens (human)Potency6.309610
3-[[1-[1-(2-furanylmethyl)-5-tetrazolyl]propyl-(2-phenylethyl)amino]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency5.011910
1-[(5,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-furanylmethyl)-3-phenylureaHomo sapiens (human)Potency25.118910
N-[2-[1,3-benzodioxol-5-yl-[2-(tert-butylamino)-2-oxo-1-pyridin-4-ylethyl]amino]-2-oxoethyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
N-(2-furanylmethyl)-N-[(7-methyl-4-tetrazolo[1,5-a]quinolinyl)methyl]-2-phenoxyacetamideHomo sapiens (human)Potency19.952610
2-[5-(3,4-diethoxyphenyl)-2-tetrazolyl]-N-(3-methoxyphenyl)acetamideHomo sapiens (human)Potency10.000010
6-amino-4-[3-ethoxy-4-[2-(4-morpholinyl)ethoxy]phenyl]-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileHomo sapiens (human)Potency10.000010
5-[(2-fluoroanilino)methyl]-8-quinolinolHomo sapiens (human)Potency5.011910
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(thiophen-2-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamideHomo sapiens (human)Potency10.000010
benzoic acid [5-amino-1-(4-methoxyphenyl)sulfonyl-3-pyrazolyl] esterHomo sapiens (human)Potency1.258910
2-[[5-(4-methylphenyl)-3-thiazolo[2,3-c][1,2,4]triazolyl]thio]-N-(6-methyl-2-pyridinyl)acetamideHomo sapiens (human)Potency7.943310
N-[2-(4-chloro-N-[2-(cyclohexylamino)-2-oxoethyl]anilino)-2-oxoethyl]-2-furancarboxamideHomo sapiens (human)Potency6.309610
N'-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]-N-(5-methyl-3-isoxazolyl)-N'-phenylbutanediamideHomo sapiens (human)Potency12.589310
N-[4-(diethylsulfamoyl)phenyl]-2-(2-oxo-1,3-benzothiazol-3-yl)acetamideHomo sapiens (human)Potency7.943310
2-[[5-[(2,3-dimethylphenoxy)methyl]-4-methyl-1,2,4-triazol-3-yl]thio]-1-thiophen-2-ylethanoneHomo sapiens (human)Potency15.848910
1-(4,6-dimethyl-2-pyrimidinyl)-4-piperidinecarboxylic acidHomo sapiens (human)Potency7.943310
N-(3,4-dimethylphenyl)-2-[[5-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency12.589310
3-[[4-(1-benzotriazolyl)-1-piperidinyl]sulfonyl]-N-cyclopentylbenzenesulfonamideHomo sapiens (human)Potency6.309610
N,N-dimethyl-4-[[4-(5-methyl-1-benzotriazolyl)-1-piperidinyl]sulfonyl]benzamideHomo sapiens (human)Potency12.589310
2-[4-[1-[1-[(4-methylphenyl)sulfonylmethyl]-5-tetrazolyl]propyl]-1-piperazinyl]-1,3-benzothiazoleHomo sapiens (human)Potency10.000010
2-[[5-[[2-(3-chloroanilino)-4-thiazolyl]methyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]thio]acetic acid methyl esterHomo sapiens (human)Potency12.589310
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideHomo sapiens (human)Potency10.996330
8-(2-furanyl)-6-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3,3-dimethyl-1,4-dihydrothiopyrano[3,4-c]pyridine-5-carbonitrileHomo sapiens (human)Potency17.261830
5-bromo-3-[[2-(4-cyclohexyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency10.000010
2-amino-1-(1,3-benzodioxol-5-yl)-N-[2-(4-morpholinyl)ethyl]-3-pyrrolo[3,2-b]quinoxalinecarboxamideHomo sapiens (human)Potency7.943310
5-chloro-3-[[2-(4-ethoxycarbonyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency10.000010
2-(pyridin-4-yl)-4-(pyrrolidin-1-yl)quinazolineHomo sapiens (human)Potency12.589310
3,4,5-trimethoxy-N-[2-(4-sulfamoylphenyl)ethyl]benzamideHomo sapiens (human)Potency12.589310
2-cyano-N-(2-furanylmethyl)-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetamideHomo sapiens (human)Potency12.589310
LSM-27020Homo sapiens (human)Potency10.000010
2-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-1-(8-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)ethanoneHomo sapiens (human)Potency7.943310
2-(2-oxo-3H-1,4-benzoxazin-4-yl)acetic acid [2-(3-bromo-4-methoxyphenyl)-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
5,6-dimethoxy-3-[[(3-methoxyphenyl)-oxomethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency10.000010
2-(butan-2-ylamino)-N-[4-[5-[[2-(butan-2-ylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideHomo sapiens (human)Potency10.000010
2-(butylamino)-N-[4-[5-[[2-(butylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideHomo sapiens (human)Potency10.000010
5-(2,4-dimethoxyphenyl)-7-(3,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency12.589310
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid cyclohexyl esterHomo sapiens (human)Potency10.000010
2-[5-[(2-chlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)Potency15.848910
6-(4-methoxyphenyl)-3-phenyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency15.848910
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid hexyl esterHomo sapiens (human)Potency3.162310
4-[4-(1H-benzimidazol-2-ylmethyl)-1-piperazinyl]benzofuro[3,2-d]pyrimidineHomo sapiens (human)Potency12.589310
8-(1,3-benzothiazol-2-ylthio)-3-methyl-7-pentylpurine-2,6-dioneHomo sapiens (human)Potency12.589310
2-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-3a,4,7,7a-tetrahydroisoindole-1,3-dioneHomo sapiens (human)Potency25.118910
4-(1H-benzimidazol-2-ylmethylthio)-2-methylbenzofuro[3,2-d]pyrimidineHomo sapiens (human)Potency12.589310
(2S)-4-methyl-2-[[oxo-(1,2,3,4-tetrahydronaphthalen-1-ylamino)methyl]amino]pentanoic acid methyl esterHomo sapiens (human)Potency15.848910
3-methoxy-2-(3-pyridinylmethylthio)-4-quinazolinoneHomo sapiens (human)Potency3.162310
N-[7-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideHomo sapiens (human)Potency12.589310
1-(thiophen-2-ylmethyl)-3-thiophen-2-ylsulfonyl-2-pyrrolo[3,2-b]quinoxalinamineHomo sapiens (human)Potency12.589310
3-[[2-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency12.589310
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dioneHomo sapiens (human)Potency6.309610
3-[[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-1-oxoethyl]amino]-5-ethoxy-1H-indole-2-carboxylic acid ethyl esterHomo sapiens (human)Potency25.118910
9,10-dimethoxy-2-(2-pyridinylmethylamino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-oneHomo sapiens (human)Potency1.258910
(3aR,6aS)-3-(2-chlorophenyl)-5-(2,5-dimethoxyphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dioneHomo sapiens (human)Potency25.118910
N-(4-chlorophenyl)-2-[3-(2-furanylmethyl)-4-imino-6,6-dimethyl-2-oxo-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-1-yl]acetamideHomo sapiens (human)Potency10.000010
Glyceryl lactopalmitateHomo sapiens (human)Potency13.650530
N-[5-(4-chlorophenyl)-7-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-furancarboxamideHomo sapiens (human)Potency5.011910
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanolHomo sapiens (human)Potency10.000010
LSM-32568Homo sapiens (human)Potency12.589310
2-[3-(2-furanylmethyl)-4-imino-6,6-dimethyl-2-oxo-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-1-yl]-N-phenylacetamideHomo sapiens (human)Potency25.118910
3-[(3aR,6aS)-6'-chloro-5-(4-chlorophenyl)-7'-methyl-2',4,6-trioxo-1-spiro[1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3,3'-1H-indole]yl]propanamideHomo sapiens (human)Potency12.589310
7-(3,4-dimethoxyphenyl)-4-methyl-2-[4-(phenylmethyl)-1-piperazinyl]-7,8-dihydro-6H-quinazolin-5-oneHomo sapiens (human)Potency12.589310
7-butyl-8-[[4-(3-chlorophenyl)-1-piperazinyl]methyl]-1,3-dimethylpurine-2,6-dioneHomo sapiens (human)Potency10.000010
3-(1-benzotriazolylmethyl)-6-(2-phenylethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency10.000010
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency0.794310
3-(4-fluorophenyl)-6-(4-methoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency5.011910
2-amino-4-(3-chlorophenyl)-6-(2-furanylmethyl)-7-methyl-5-oxo-4H-pyrano[3,2-c]pyridine-3-carboxylic acid methyl esterHomo sapiens (human)Potency15.848910
6-amino-1-(4-fluorophenyl)-3-methyl-4-thiophen-2-yl-5-pyrazolo[3,4-b]pyridinecarbonitrileHomo sapiens (human)Potency12.589310
6-[[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]methyl]-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency10.000010
4-(3,4-dihydro-2H-quinolin-1-yl)-6-[(4-phenyl-1-piperazinyl)methyl]-1,3,5-triazin-2-amineHomo sapiens (human)Potency10.000010
3-(1-benzimidazolylmethyl)-6-[(4-methoxyphenoxy)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency10.000010
2-[[[5-(3-chlorophenyl)-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-1H-benzimidazoleHomo sapiens (human)Potency10.000010
3-(2,3-dihydro-1,4-benzodioxin-3-yl)-6-(4-fluorophenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency12.589310
2-[[2-furanyl(oxo)methyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid ethyl esterHomo sapiens (human)Potency25.118910
N-(2-furanylmethyl)-2-benzofurancarboxamideHomo sapiens (human)Potency12.589310
3,4'-dihydroxyflavoneHomo sapiens (human)Potency12.589310
5-(5-chloro-2-methoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneHomo sapiens (human)Potency10.000010
spiro[1,3-dihydroperimidine-2,1'-cycloheptane]Homo sapiens (human)Potency3.162310
N-(4-methyl-2-thiazolyl)-3-(2-oxo-1,3-benzothiazol-3-yl)propanamideHomo sapiens (human)Potency22.387210
4-[(4-phenyl-2-thiazolyl)amino]benzenesulfonamideHomo sapiens (human)Potency21.671210
2-[[2-(5,6-dimethyl-1-benzimidazolyl)-1-oxoethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency3.162310
4-methyl-N-[1-[2-(1-pyrrolidinyl)ethyl]-2-benzimidazolyl]benzamideHomo sapiens (human)Potency12.589310
N-(1-naphthalenyl)-4-(phenylmethyl)-1-piperazinecarboxamideHomo sapiens (human)Potency10.000010
3,5-dimethyl-1-[(7-methyl-2-naphthalenyl)sulfonyl]pyrazoleHomo sapiens (human)Potency3.162310
2-methyl-N-(2-naphthalenyl)-3-furancarboxamideHomo sapiens (human)Potency12.589310
(2'-(4-aminophenyl)-(2,5'-bi-1h-benzimidazol)-5-amine)Homo sapiens (human)Potency19.904020
4,5-dimethylcyclopenta[c]quinolizine-1,2-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency14.125410
2-(4-methoxyphenoxy)-N-(2-methoxyphenyl)acetamideHomo sapiens (human)Potency3.162310
4-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]benzoic acid ethyl esterHomo sapiens (human)Potency10.000010
N-(1,3-benzodioxol-5-yl)-4-(4-morpholinylmethyl)benzamideHomo sapiens (human)Potency7.943310
lupitidineHomo sapiens (human)Potency12.589310
N-[3-[(1,3-dioxo-5-isoindolyl)oxy]phenyl]-2-furancarboxamideHomo sapiens (human)Potency25.118910
N2-(4-fluorophenyl)-6-(3-methyl-2-benzofuranyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency6.309610
thiothixeneHomo sapiens (human)Potency10.000010
N-(2-hydroxy-5-methoxy-1H-indol-3-yl)acetamideHomo sapiens (human)Potency12.589310
N-(3-chlorophenyl)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-4-methylbenzenesulfonamideHomo sapiens (human)Potency17.782810
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency28.183810
2-(3-pyridinyl)-4-[4-(1-pyrrolidinylsulfonyl)phenyl]thiazoleHomo sapiens (human)Potency12.589310
4-[[[2,3-bis(2-pyridinyl)-6-quinoxalinyl]amino]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
2-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]thio]-N-(4-methyl-2-thiazolyl)acetamideHomo sapiens (human)Potency12.589310
4-[[[3-(4-morpholinylsulfonyl)phenyl]-oxomethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency15.848910
N-[4-[4-[(2-methylphenyl)-oxomethyl]-1-piperazinyl]phenyl]propanamideHomo sapiens (human)Potency12.589310
N-(2-furanylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency3.981110
4-[4-(benzenesulfonyl)-1-piperazinyl]-2-methylquinolineHomo sapiens (human)Potency3.981110
N-(2-furanylmethyl)-2-(4-oxo-6-phenyl-3-thieno[2,3-d]pyrimidinyl)acetamideHomo sapiens (human)Potency18.835940
1-(3,4-dimethoxyphenyl)sulfonyl-4-(2-methoxyphenyl)piperazineHomo sapiens (human)Potency10.000010
N-(3-carbamoyl-5-propyl-2-thiophenyl)-2-methyl-3-furancarboxamideHomo sapiens (human)Potency5.011910
[4-(2-methylphenyl)-1-piperazinyl]-(5-propyl-3-thiophenyl)methanoneHomo sapiens (human)Potency10.000010
1,4-dioxa-8-azaspiro[4.5]decan-8-yl(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)methanoneHomo sapiens (human)Potency19.952610
N-[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency10.000010
2-[(4-chlorophenyl)thio]-N-(5-oxo-1-phenyl-4H-pyrazol-3-yl)acetamideHomo sapiens (human)Potency12.589310
2-[[2-(3,4-dimethylanilino)-2-oxoethyl]thio]acetamideHomo sapiens (human)Potency10.000010
1-methylsulfonyl-N-(6,7,8,9-tetrahydrodibenzofuran-2-yl)-2,3-dihydroindole-5-sulfonamideHomo sapiens (human)Potency10.000010
2-[2-chloro-4-(2,3-dihydroindol-1-ylsulfonyl)phenoxy]-N-(2-pyridinylmethyl)acetamideHomo sapiens (human)Potency12.589310
N-[2-(4-acetyl-1-piperazinyl)phenyl]-2-(5-methyl-2-propan-2-ylphenoxy)acetamideHomo sapiens (human)Potency12.589310
N-(2-furanylmethyl)-2-imino-5-oxo-1-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideHomo sapiens (human)Potency10.000010
N-[3-[2-(1-azepanyl)-4,5-dicyanophenoxy]phenyl]acetamideHomo sapiens (human)Potency15.848910
3-phenyl-5-[[[4-phenyl-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-1,2,4-oxadiazoleHomo sapiens (human)Potency3.162310
2-[[2-[[1-(2,4-dimethylphenyl)-5-tetrazolyl]thio]-1-oxoethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency10.000010
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency3.981110
N-[6-(diethylsulfamoyl)-1,3-benzothiazol-2-yl]-2-thiophenecarboxamideHomo sapiens (human)Potency19.952610
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-5-methyl-3-phenyl-4-isoxazolecarboxamideHomo sapiens (human)Potency15.848910
2-[[4-(1,3-dioxo-2-isoindolyl)-1-oxobutyl]amino]-N-(2-furanylmethyl)-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideHomo sapiens (human)Potency12.589310
[4-[(2,4-dichlorophenoxy)methyl]phenyl]-(4-methyl-1-piperazinyl)methanoneHomo sapiens (human)Potency12.589310
N-[4-[4-(4-hydroxyphenyl)-1-piperazinyl]phenyl]carbamic acid phenyl esterHomo sapiens (human)Potency3.162310
darunavir ethanolateHomo sapiens (human)Potency15.848910
1-[2,3-bis(2-furanyl)-6-quinoxalinyl]-3-[4-(4-morpholinyl)phenyl]thioureaHomo sapiens (human)Potency11.220210
N-[3-[[2-(2-bromo-4,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamideHomo sapiens (human)Potency3.162310
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-(2-methoxyphenyl)acetamideHomo sapiens (human)Potency10.000010
4-(dimethylsulfamoyl)-N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamideHomo sapiens (human)Potency3.981110
N-(3,4-dimethoxyphenyl)-4-[(4-phenyl-1-piperazinyl)methyl]benzamideHomo sapiens (human)Potency6.309610
1-(3-chlorophenyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazineHomo sapiens (human)Potency12.589310
cis-resveratrolHomo sapiens (human)Potency10.000010
4-(4-chlorophenoxy)-1-(4-morpholinyl)-1-butanoneHomo sapiens (human)Potency5.011910
2-phenyl-N-[4-(2-thiazolylsulfamoyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)Potency1.544420
N-(9-ethyl-3-carbazolyl)-2-[[4-ethyl-5-(2-furanyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency1.584910
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[methyl-(phenylmethyl)sulfamoyl]benzamideHomo sapiens (human)Potency10.000010
N-(9-ethyl-3-carbazolyl)-2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]acetamideHomo sapiens (human)Potency1.258910
7-[[[5-(2,4-dimethylanilino)-1,3,4-thiadiazol-2-yl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneHomo sapiens (human)Potency10.000010
3-methyl-2-benzofurancarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] esterHomo sapiens (human)Potency10.000010
N-(3-cyano-2-thiophenyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]acetamideHomo sapiens (human)Potency12.589310
4-(1,3-benzothiazol-2-ylthio)butanoic acid [2-[(3-cyano-2-thiophenyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
N-(1,3-benzodioxol-5-ylmethyl)-2-[(3-methyl-4-oxo-5-thiophen-2-yl-2-thieno[2,3-d]pyrimidinyl)thio]acetamideHomo sapiens (human)Potency10.000010
1-[4-(benzenesulfonyl)-1-piperazinyl]-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]ethanoneHomo sapiens (human)Potency15.848910
1-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]-2-(2-methyl-4-thiazolyl)ethanoneHomo sapiens (human)Potency10.000010
2-[[2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]-1-oxoethyl]amino]-5-phenyl-3-thiophenecarboxamideHomo sapiens (human)Potency3.162310
6-[1-oxo-2-[[4-(phenylmethyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]thio]ethyl]-4H-1,4-benzoxazin-3-oneHomo sapiens (human)Potency10.000010
4-(2-oxo-1-pyrrolidinyl)benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
4-[bis(2-methylpropyl)sulfamoyl]-N-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideHomo sapiens (human)Potency3.162310
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterHomo sapiens (human)Potency12.589310
N-(3-dibenzofuranyl)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)thio]acetamideHomo sapiens (human)Potency5.011910
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-2-benzofurancarboxamideHomo sapiens (human)Potency3.981110
4-methyl-N-[2-(phenylmethyl)-3,4-dihydro-1H-pyrazino[1,2-a]benzimidazol-8-yl]benzenesulfonamideHomo sapiens (human)Potency7.943310
2-[[1-oxo-2-(1H-1,2,4-triazol-5-ylthio)ethyl]amino]-4-thiophen-2-yl-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
N-(2-furanylmethyl)-2-[3-(1-oxo-2-phenoxyethyl)-1-indolyl]acetamideHomo sapiens (human)Potency12.589310
N-[3-[[2-(2,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamideHomo sapiens (human)Potency10.000010
1-(3-chlorophenyl)-3-[3-[methyl(methylsulfonyl)amino]phenyl]ureaHomo sapiens (human)Potency28.183810
2-(3,5-dimethylphenoxy)-N-[3-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideHomo sapiens (human)Potency3.981110
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-dibenzofuransulfonamideHomo sapiens (human)Potency25.118910
1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(5,7-diphenyl-2-pyrazolo[1,5-a]pyrimidinyl)methanoneHomo sapiens (human)Potency12.589310
2-(2,4-dichloro-6-methylphenoxy)-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency3.162310
1-chloro-2-[2-(2-methoxy-4-methylphenoxy)ethoxy]-4-methylbenzeneHomo sapiens (human)Potency11.220210
4-[3-(2,5-dimethyl-1-pyrrolyl)-4-(1-pyrrolidinyl)phenyl]sulfonylmorpholineHomo sapiens (human)Potency2.818410
LSM-19724Homo sapiens (human)Potency12.589310
2-(1H-benzimidazol-2-ylthio)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamideHomo sapiens (human)Potency5.011910
4-amino-2-[[4-(1-azepanylsulfonyl)phenyl]-oxomethyl]isoindole-1,3-dioneHomo sapiens (human)Potency12.589310
N-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-2-[(6-methyl-1H-benzimidazol-2-yl)thio]acetamideHomo sapiens (human)Potency5.011910
3-[5-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-1,3,4-oxadiazol-2-yl]-1-benzopyran-2-oneHomo sapiens (human)Potency3.162310
[1-(4-fluorophenyl)sulfonyl-4-piperidinyl]-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methanoneHomo sapiens (human)Potency19.952610
N-(2,4-dichlorophenyl)-2-[[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]thio]acetamideHomo sapiens (human)Potency10.000010
2-[[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)thio]methyl]-1,3-benzothiazoleHomo sapiens (human)Potency12.589310
5-[2-[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
2-(1,3-benzodioxol-5-yl)-5-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methylthio]-1,3,4-oxadiazoleHomo sapiens (human)Potency12.589310
2-[[[2-[(5-methoxycarbonyl-2-furanyl)methoxy]-2-oxoethyl]thio]methyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
4-cyclopropyl-2-[[2-[(3,5-dimethyl-4-isoxazolyl)methylthio]-1-oxoethyl]amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency19.952610
N-[5-chloro-2-(4-methyl-1-piperazinyl)phenyl]-3-(dimethylsulfamoyl)benzamideHomo sapiens (human)Potency15.848910
5-(4-chloroanilino)-3-oxo-4-isothiazolecarbonitrileHomo sapiens (human)Potency13.699620
2-amino-7-methyl-5-oxo-4-(2,3,4-trimethoxyphenyl)-4,6,7,8-tetrahydro-1-benzopyran-3-carbonitrileHomo sapiens (human)Potency25.118910
1-hexadecyl-3-methylimidazolium bromideHomo sapiens (human)Potency22.834020
4-[[3-methoxy-4-[(4-nitrophenyl)methoxy]phenyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneHomo sapiens (human)Potency11.904820
3,4,5-trimethoxy-N-[4-[(2-methyl-1-piperidinyl)sulfonyl]phenyl]benzamideHomo sapiens (human)Potency10.000010
1-(2-furanylmethyl)-3-[(4-methylphenyl)methyl]pyrrolidine-2,5-dioneHomo sapiens (human)Potency10.000010
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dioneHomo sapiens (human)Potency10.000010
2-[(9-tert-butyl-1,5-dicyano-2-oxo-3-azaspiro[5.5]undec-4-en-4-yl)thio]-N-cyclohexylacetamideHomo sapiens (human)Potency12.589310
2-methyl-3-[(2-methyl-1H-indol-3-yl)-(2-pyridinyl)methyl]-1H-indoleHomo sapiens (human)Potency28.183810
N-[4-[4-(1-pyrrolidinylsulfonyl)phenyl]-2-thiazolyl]-2,3-dihydro-1,4-benzodioxin-3-carboxamideHomo sapiens (human)Potency12.589310
3-hydroxy-3-[2-oxo-2-[4-(1-pyrrolyl)phenyl]ethyl]-1H-indol-2-oneHomo sapiens (human)Potency10.000010
N-(5-chloro-2-hydroxyphenyl)-2-ethoxybenzamideHomo sapiens (human)Potency12.589310
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-phenoxybutanamideHomo sapiens (human)Potency12.589310
N-[2-[(2-furanylmethylamino)-oxomethyl]phenyl]-4-methyl-3-(1-piperidinylsulfonyl)benzamideHomo sapiens (human)Potency12.589310
3-[2-(2,4-dimethyl-3-furanyl)-2-oxoethyl]-3-hydroxy-1-(2-phenylethyl)-2-indoloneHomo sapiens (human)Potency12.589310
N-[3-chloro-4-[4-[oxo-(4-propoxyphenyl)methyl]-1-piperazinyl]phenyl]propanamideHomo sapiens (human)Potency6.309610
3-fluoro-N-[4-[[4-(4-methoxyphenyl)-1-piperazinyl]-oxomethyl]phenyl]benzenesulfonamideHomo sapiens (human)Potency19.952610
1-[2-(hydroxymethyl)-1-benzimidazolyl]-3-(1-indolyl)-2-propanolHomo sapiens (human)Potency25.118910
1-[3-[4-(2-chloro-5-methoxyphenyl)-1-piperazinyl]propyl]-3-(4-methylphenyl)ureaHomo sapiens (human)Potency7.943310
9-oxo-N-(1-phenylethyl)-3-bicyclo[3.3.1]nonanecarboxamideHomo sapiens (human)Potency5.011910
N-(3-carbamoyl-5-propyl-2-thiophenyl)-2-oxolanecarboxamideHomo sapiens (human)Potency10.000010
6-(2-chlorophenyl)-3-methyl-2-[4-morpholinyl(oxo)methyl]-1,5,6,7-tetrahydroindol-4-oneHomo sapiens (human)Potency12.589310
N-[3-chloro-4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]phenyl]-2-(4-chlorophenyl)acetamideHomo sapiens (human)Potency5.011910
4-(1,3-benzodioxol-5-yl)-6-[[2-(4-chlorophenyl)ethylamino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
1-[2-furanyl(oxo)methyl]-6-(1-pyrrolidinylsulfonyl)-2-benzo[cd]indoloneHomo sapiens (human)Potency12.589310
2-[[[4-(4-methoxyphenyl)-5-phenyl-1,2,4-triazol-3-yl]thio]methyl]-5-phenyl-1,3,4-oxadiazoleHomo sapiens (human)Potency12.589310
3-[5-(dimethylsulfamoyl)-1-ethyl-2-benzimidazolyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)propanamideHomo sapiens (human)Potency5.011910
7-[[[1-(3-methylphenyl)-2-benzimidazolyl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneHomo sapiens (human)Potency10.000010
2-(4-cyanophenoxy)-N-(2-methyl-1-phenyl-5-benzimidazolyl)acetamideHomo sapiens (human)Potency5.011910
1-[4-(benzenesulfonyl)-1-piperazinyl]-2-[[1-(2-methylpropyl)-2-benzimidazolyl]thio]ethanoneHomo sapiens (human)Potency12.589310
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamideHomo sapiens (human)Potency12.589310
1-butyl-2-[(1,3-dioxo-2-isoindolyl)methylthio]-5-benzimidazolesulfonamideHomo sapiens (human)Potency10.000010
3-(2,5-dimethyl-3-furanyl)-5,6-diphenyl-1,2,4-triazineHomo sapiens (human)Potency10.000010
1-(4-fluorophenyl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxylic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)Potency10.000010
7-[3-[4-(2-ethoxyphenyl)-1-piperazinyl]-2-hydroxypropoxy]-4-methyl-1-benzopyran-2-oneHomo sapiens (human)Potency6.309610
3-[(4-phenyl-1-piperazinyl)sulfonyl]benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterHomo sapiens (human)Potency1.995310
1-butyl-2-[(5-phenyl-2-oxazolyl)methylthio]-5-benzimidazolesulfonamideHomo sapiens (human)Potency12.589310
2-[(5,6-dithiophen-2-yl-1,2,4-triazin-3-yl)oxy]-N-methyl-N-phenylacetamideHomo sapiens (human)Potency15.848910
3-ethyl-4-oxo-1-phthalazinecarboxylic acid [2-(1H-indol-3-yl)-2-oxoethyl] esterHomo sapiens (human)Potency25.118910
6-methyl-2-[[2-(4-morpholinyl)-1-oxoethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterHomo sapiens (human)Potency12.589310
2-(3,4-dimethoxyphenyl)-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)Potency10.000010
3-[(4-methylphenyl)sulfamoyl]benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterHomo sapiens (human)Potency10.286930
N-[1-(1H-benzimidazol-2-yl)-2-phenylethyl]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxo-3-pyrrolidinecarboxamideHomo sapiens (human)Potency19.952610
AvocadyneHomo sapiens (human)Potency12.589310
3-deoxyvasicine, hydrochlorideHomo sapiens (human)Potency12.589310
N-(2-furanylmethyl)-6-(3-methoxyphenyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency25.118910
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency12.589310
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency12.589310
6-(3-furanyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency7.943310
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency12.589310
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency10.000010
6-(2-chlorophenyl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency15.848910
nih-12848Homo sapiens (human)Potency5.011910
6-(3-furanyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency25.118910
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency15.848910
4-[butan-2-yl-[(3,4-dichloroanilino)-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
4-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-2-methyl-5-furo[3,2-b]pyrrolecarboxylic acid methyl esterHomo sapiens (human)Potency15.848910
2-[[3-(4-chlorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency19.952610
3-(1,3-benzodioxol-5-ylmethyl)-7-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency7.943310
N-[3-[4-(2,3-dimethylphenyl)-1-piperazinyl]-3-oxopropyl]-2-(1-oxo-2-isoquinolinyl)acetamideHomo sapiens (human)Potency10.000010
6-bromo-3-[4-oxo-4-[4-(2-pyridinyl)-1-piperazinyl]butyl]-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency12.589310
2-(2-methoxyphenyl)-N-[4-[5-(3-methoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]acetamideHomo sapiens (human)Potency12.589310
2-[8-[[bis(phenylmethyl)amino]methyl]-3-methyl-2,6-dioxo-7-purinyl]acetic acid ethyl esterHomo sapiens (human)Potency15.848910
N-(3-chlorophenyl)-2-[6,7-dimethoxy-2,4-dioxo-3-(2-oxolanylmethyl)-1-quinazolinyl]acetamideHomo sapiens (human)Potency12.589310
1-[2-[3-(N-ethylanilino)propylamino]-3,4-dioxo-1-cyclobutenyl]-4-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency19.952610
4-morpholinecarboxylic acid [4-[6-amino-5-cyano-3-(4-methylphenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]phenyl] esterHomo sapiens (human)Potency12.589310
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideHomo sapiens (human)Potency10.000010
N-(2,3-dihydro-1H-inden-5-yl)-2-[(4-hydroxy-6-oxo-1H-pyrimidin-2-yl)thio]acetamideHomo sapiens (human)Potency10.000010
3,4-dihydro-2H-quinolin-1-yl-(7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl)methanoneHomo sapiens (human)Potency25.118910
N-(5-chloro-2-methoxyphenyl)-2,4-dimethyl-5-oxazolecarboxamideHomo sapiens (human)Potency15.848910
1-(4-chlorophenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-4-pyrazolecarboxylic acidHomo sapiens (human)Potency12.589310
N-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-2-[[1-oxo-2-(1-oxo-2-isoquinolinyl)ethyl]amino]acetamideHomo sapiens (human)Potency10.000010
4-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-6-(trifluoromethyl)pyrimidineHomo sapiens (human)Potency10.000010
N-(3-chlorophenyl)-5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-methyl-2-benzofurancarboxamideHomo sapiens (human)Potency12.589310
4-[2-[[2-[[4-(1,3-benzodioxol-5-yl)-2-thiazolyl]amino]-2-oxoethyl]thio]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
1-[4-[2-(2,5-dimethyl-1-pyrrolyl)ethyl]-1-piperazinyl]-2-[[3-(4-morpholinyl)-2-quinoxalinyl]thio]ethanoneHomo sapiens (human)Potency19.952610
2-[(5-bromo-2-thiophenyl)sulfonyl-methylamino]-N-(6-methyl-1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)Potency10.000010
[1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-3-piperidinyl]-(2-methyl-2,3-dihydroindol-1-yl)methanoneHomo sapiens (human)Potency12.589310
2-(4-ethoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acidHomo sapiens (human)Potency12.589310
3-methyl-N,6-diphenyl-2-imidazo[2,1-b]thiazolecarboxamideHomo sapiens (human)Potency10.000010
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-piperidinecarboxamideHomo sapiens (human)Potency12.589310
1-[[4-[(4-fluorophenyl)methyl]-5-thieno[3,2-b]pyrrolyl]-oxomethyl]-N-(2-furanylmethyl)-4-piperidinecarboxamideHomo sapiens (human)Potency7.943310
4-[[2-(3-ethylanilino)-3,4-dioxo-1-cyclobutenyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
5-bromo-N-[2-(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)ethyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
N-[2-(dimethylamino)ethyl]-2-[3-(4-methylphenyl)-6-oxo-1-pyridazinyl]acetamideHomo sapiens (human)Potency25.118910
6-[(2-ethylphenyl)sulfamoyl]-N-(2-furanylmethyl)-4-oxo-1H-quinoline-3-carboxamideHomo sapiens (human)Potency12.589310
2-[[3-oxo-2-[3-oxo-3-(4-phenyl-1-piperazinyl)propyl]-2H-imidazo[1,2-c]quinazolin-5-yl]thio]acetonitrileHomo sapiens (human)Potency10.000010
2-amino-4-[5-methyl-2-(methylthio)-3-thiophenyl]-5-oxo-1-(3-pyridinyl)-4,6,7,8-tetrahydroquinoline-3-carbonitrileHomo sapiens (human)Potency19.952610
6-[(2-ethylphenyl)sulfamoyl]-4-oxo-N-(2-oxolanylmethyl)-1H-quinoline-3-carboxamideHomo sapiens (human)Potency12.589310
N-butyl-2-[[6-(4-morpholinyl)-4-oxo-3-(2-phenylethyl)-2-quinazolinyl]thio]acetamideHomo sapiens (human)Potency12.589310
4-(4-methyl-1-oxido-2-triazol-1-iumyl)benzoic acidHomo sapiens (human)Potency10.000010
N-(1,3-benzodioxol-5-yl)-2-[(1-ethyl-2-oxo-4-quinolinyl)thio]acetamideHomo sapiens (human)Potency15.848910
6-(1-azepanylsulfonyl)-1-ethyl-N-(2-furanylmethyl)-4-oxo-3-quinolinecarboxamideHomo sapiens (human)Potency12.589310
3-(2-chlorophenyl)-5-methyl-N-[3-(3-methyl-2-imidazo[1,2-a]pyrimidinyl)phenyl]-4-isoxazolecarboxamideHomo sapiens (human)Potency7.943310
N-(1,3-benzodioxol-5-yl)-5-bromo-1-[cyclopropyl(oxo)methyl]-N-ethyl-2,3-dihydroindole-7-sulfonamideHomo sapiens (human)Potency5.011910
N-[2-[4-(3-chlorophenyl)-1-piperazinyl]ethyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-amineHomo sapiens (human)Potency5.011910
2-furanyl-[4-(4-tetrazolo[1,5-a]quinoxalinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency7.943310
1-acetyl-5-bromo-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-2-methyl-2,3-dihydroindole-7-sulfonamideHomo sapiens (human)Potency25.118910
6-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-5-thieno[2,3-b]pyrrolecarboxylic acid methyl esterHomo sapiens (human)Potency12.589310
N-(3,4-dimethylphenyl)-2-[N-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-methoxyanilino]acetamideHomo sapiens (human)Potency12.589310
N-(1,3-benzodioxol-5-yl)-2-[[6-methyl-4-oxo-3-(phenylmethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideHomo sapiens (human)Potency12.589310
N-(2-chlorophenyl)-5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-methyl-2-benzofurancarboxamideHomo sapiens (human)Potency10.000010
2-amino-4-[4-(methylthio)phenyl]-5-oxo-1-phenyl-4,6,7,8-tetrahydroquinoline-3-carbonitrileHomo sapiens (human)Potency19.952610
2,5-dimethyl-4-(4-methyl-1-piperidinyl)-6-thieno[2,3-d]pyrimidinecarboxylic acidHomo sapiens (human)Potency10.000010
N-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-2-[(1-ethyl-2-oxo-4-quinolinyl)oxy]acetamideHomo sapiens (human)Potency12.589310
2-[[2-(3-methyl-1-oxo-2-isoquinolinyl)-1-oxoethyl]amino]acetic acid ethyl esterHomo sapiens (human)Potency25.118910
N-(2,3-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideHomo sapiens (human)Potency12.589310
7-(2,4-dichlorophenyl)-5-oxo-2,3-dihydrothiazolo[3,2-a]pyrimidine-6-carbonitrileHomo sapiens (human)Potency12.589310
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamideHomo sapiens (human)Potency3.981110
5-(1,3-benzodioxol-5-yl)-3-[3-(methylthio)phenyl]-1H-imidazol-2-oneHomo sapiens (human)Potency10.000010
N-butan-2-yl-6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-1H-quinoline-3-carboxamideHomo sapiens (human)Potency12.589310
7-[4-[4-(2-fluorophenyl)-1-piperazinyl]-4-oxobutyl]-6-sulfanylidene-5H-[1,3]dioxolo[4,5-g]quinazolin-8-oneHomo sapiens (human)Potency31.622810
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency25.118910
1-[2-(4-bromophenyl)-2-oxoethyl]-3-(2-furanylmethyl)-6,7-dimethoxyquinazoline-2,4-dioneHomo sapiens (human)Potency10.000010
8-[[4-(5-chloro-2-methylphenyl)-1-piperazinyl]methyl]-3-methyl-7-(2-phenylethyl)purine-2,6-dioneHomo sapiens (human)Potency12.589310
1-methyl-N-(2-methylcyclohexyl)-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamideHomo sapiens (human)Potency12.589310
2-(2-ethoxyphenyl)-8-oxo-9-phenyl-7H-purine-6-carboxamideHomo sapiens (human)Potency12.589310
cyclopentanecarboxylic acid [4-(benzenesulfonyl)-2-tert-butyl-5-methyl-3-pyrazolyl] esterHomo sapiens (human)Potency12.589310
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-3-piperidinecarboxamideHomo sapiens (human)Potency10.000010
1-[(2-ethoxyphenyl)methyl]-3-thiophen-2-ylureaHomo sapiens (human)Potency25.118910
gw 7647Homo sapiens (human)Potency23.280910
cgp 13501Homo sapiens (human)Potency12.589310
2,4-dihydroxyheptadec-16-enyl acetateHomo sapiens (human)Potency15.848910
suramin sodiumHomo sapiens (human)Potency3.288510
2,4-dihydroxyheptadec-16-ynyl acetateHomo sapiens (human)Potency15.848910
2-[[2-(3,4-dimethoxyanilino)-2-oxoethyl]thio]-3-pyridinecarboxylic acid propan-2-yl esterHomo sapiens (human)Potency25.118910
[2-(3,4-dimethylphenyl)-4-quinolinyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency24.315510
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazoleHomo sapiens (human)Potency28.872220
2-nitro-4-[(6-nitro-4-quinolinyl)amino]-N-[4-(pyridin-4-ylamino)phenyl]benzamideHomo sapiens (human)Potency8.154820
quercetinHomo sapiens (human)Potency25.057820
acacetinHomo sapiens (human)Potency12.589310
apigeninHomo sapiens (human)Potency10.000010
cyclosporineHomo sapiens (human)Potency10.000010
baicaleinHomo sapiens (human)Potency0.631010
mangostinHomo sapiens (human)Potency10.000010
morinHomo sapiens (human)Potency18.492710
myricetinHomo sapiens (human)Potency3.235420
Pinosylvin methyl etherHomo sapiens (human)Potency25.118910
rosmarinic acidHomo sapiens (human)Potency25.118910
ellagic acidHomo sapiens (human)Potency1.122010
n-oleoyldopamineHomo sapiens (human)Potency13.131120
10-octadecenoic acid, (z)-isomerHomo sapiens (human)Potency12.589310
n-arachidonylglycineHomo sapiens (human)Potency16.481610
quercetinHomo sapiens (human)Potency2.511910
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acidHomo sapiens (human)Potency18.492710
N-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-1-(1H-imidazol-5-ylsulfonyl)-3-piperidinecarboxamideHomo sapiens (human)Potency15.848910
2-[6-[(5-chloro-2-methoxyphenyl)sulfamoyl]-2-oxo-1,3-benzoxazol-3-yl]acetic acid ethyl esterHomo sapiens (human)Potency14.125410
4-amino-5-chloro-N-[(3R,4S)-1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamideHomo sapiens (human)Potency3.981110
7,7-dimethyl-5,8-eicosadienoic acidHomo sapiens (human)Potency23.280910
fumarprotocetraric acidHomo sapiens (human)Potency25.118910
salazinic acidHomo sapiens (human)Potency25.118910
ag 538Homo sapiens (human)Potency1.166810
semaxinibHomo sapiens (human)Potency16.481610
(5R)-3'-phenyl-1-(phenylmethyl)spiro[1,3-diazinane-5,5'-2,4,4a,6-tetrahydro-1H-pyrazino[1,2-a]quinoline]-2,4,6-trioneHomo sapiens (human)Potency12.677240
(3S,3'aR,8'aS,8'bS)-5-ethyl-2'-(phenylmethyl)spiro[1H-indole-3,4'-3a,6,7,8,8a,8b-hexahydropyrrolo[3,4-a]pyrrolizine]-1',2,3'-trioneHomo sapiens (human)Potency12.589310
3-(1-benzimidazolyl)-6-ethyl-7-hydroxy-1-benzopyran-4-oneHomo sapiens (human)Potency3.981110
aztreonamHomo sapiens (human)Potency12.589310
methylbenzethonium chlorideHomo sapiens (human)Potency19.084930
dithiazanine iodideHomo sapiens (human)Potency22.387210
5233705 compoundHomo sapiens (human)Potency20.637820
gw-5074Homo sapiens (human)Potency16.481610
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-1-(4-methoxyphenyl)ethanoneHomo sapiens (human)Potency20.895030
N3,N6-bis(2,5-dimethoxyphenyl)pyridazine-3,6-diamineHomo sapiens (human)Potency14.125410
l 162313Homo sapiens (human)Potency3.162310
LSM-6455Homo sapiens (human)Potency12.589310
Garcinolic acidHomo sapiens (human)Potency10.000010
xct790Homo sapiens (human)Potency16.481610
3-(1H-benzimidazol-2-yl)-1-[4-(2,4-dimethylphenyl)-1-piperazinyl]-1-propanoneHomo sapiens (human)Potency5.011910
sgd 301-76Homo sapiens (human)Potency25.118910
lissamine rhodamine bHomo sapiens (human)Potency11.220210
chlorhexidine hydrochlorideHomo sapiens (human)Potency28.183810
tanninsHomo sapiens (human)Potency5.011910
(1R,5S)-6-[[5-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl]-6-azabicyclo[3.2.1]octaneHomo sapiens (human)Potency14.125410
meclofenamate sodium anhydrousHomo sapiens (human)Potency7.943310
cytomelHomo sapiens (human)Potency22.387210
fractalsHomo sapiens (human)Potency28.183810
5-(1,3-benzodioxol-5-yl)-4-(1-methyltetrazol-5-yl)sulfanylthieno[2,3-d]pyrimidineHomo sapiens (human)Potency12.589310
oxytetracycline, anhydrousHomo sapiens (human)Potency28.183810
piroxicamHomo sapiens (human)Potency18.854110
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamideHomo sapiens (human)Potency7.943310
4-hydroxy-2-oxo-1-propyl-N-(pyridin-4-ylmethyl)-3-quinolinecarboxamideHomo sapiens (human)Potency25.118910
robustic acidHomo sapiens (human)Potency10.000010
mobiflexHomo sapiens (human)Potency5.011910
isoxicamHomo sapiens (human)Potency10.430410
acyclovirHomo sapiens (human)Potency12.589310
olanzapineHomo sapiens (human)Potency19.952610
zaprinastHomo sapiens (human)Potency7.195010
kf38789Homo sapiens (human)Potency3.162310
hemateinHomo sapiens (human)Potency10.000010
4-[[2-[(6-methyl-4-oxo-1H-pyrimidin-2-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency25.118910
tegaserod maleateHomo sapiens (human)Potency10.000010
N-(1,3-benzodioxol-5-ylmethyl)-3-methoxy-N-[(4-oxo-1H-quinazolin-2-yl)methyl]benzamideHomo sapiens (human)Potency12.589310
1-cyclopentyl-1-[(4-oxo-1H-quinazolin-2-yl)methyl]-3-(phenylmethyl)ureaHomo sapiens (human)Potency15.848910
N-[(4-oxo-1H-quinazolin-2-yl)methyl]-N-(2-phenylethyl)butanamideHomo sapiens (human)Potency10.000010
2-[(dimethylamino)methyl]-4-spiro[1,6-dihydrobenzo[h]quinazoline-5,1'-cyclohexane]oneHomo sapiens (human)Potency7.943310