Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
3-hydroxyanthranilic acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
amoxapine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
bay h 4502 | Homo sapiens (human) | Potency | 70.7946 | 1 | 0 |
clotrimazole | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
diazinon | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
dipyridamole | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
thiorphan | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ebselen | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ethacrynic acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
ethotoin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
isoconazole | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
loratadine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
pomiferin | Homo sapiens (human) | Potency | 48.3939 | 2 | 0 |
protoporphyrin ix | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
sulfinpyrazone | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
dimethylphenylpiperazinium iodide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
methylene blue | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
7-amino-4-hydroxy-2-naphthalenesulfonic acid | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
pyronine | Homo sapiens (human) | Potency | 18.4927 | 1 | 0 |
2-amino-5-nitrothiazole | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
sulfan blue | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
imperatorin | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
beclomethasone dipropionate | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
diacerein | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
thymolphthalein | Homo sapiens (human) | Potency | 16.1652 | 2 | 0 |
butoconazole nitrate | Homo sapiens (human) | Potency | 63.0957 | 1 | 0 |
lovastatin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
sulconazole, mononitrate, (+-)-isomer | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
Isobergapten | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2,3-trimethylene-4-quinazolone | Homo sapiens (human) | Potency | 43.6381 | 2 | 0 |
miconazole nitrate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
econazole nitrate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
cresolphthalein | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
5-aminovaleric acid hydrochloride | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
lobaric acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
stictic acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
9,10-phenanthrenequinone monoxime | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-(4-hydroxyphenyl)-5,6,7,8-tetrahydroxy-4H-1-benzopyran-4-one | Homo sapiens (human) | Potency | 70.7946 | 1 | 0 |
diphyllin | Homo sapiens (human) | Potency | 32.6049 | 3 | 0 |
purpactin a | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
cryptotanshinone | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
8-(4-benzenesulfonylamino)quinoline | Homo sapiens (human) | Potency | 41.3999 | 1 | 0 |
ajmalicine, hydrochloride(19alpha)-isomer | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
gant58 | Homo sapiens (human) | Potency | 39.7679 | 3 | 0 |
medrogestone | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
oxopurpureine | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
discretamine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
mometasone furoate | Homo sapiens (human) | Potency | 22.1969 | 2 | 0 |
amcinonide | Homo sapiens (human) | Potency | 10.6025 | 2 | 0 |
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
menadione sodium bisulfite, trihydrate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
4-chloro-N-(4-chloro-2,5-dimethoxyphenyl)-5-dithiazolimine | Homo sapiens (human) | Potency | 45.5600 | 1 | 0 |
averufin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
calmidazolium | Homo sapiens (human) | Potency | 23.4648 | 3 | 0 |
3-(benzenesulfonyl)-2-imino-1-(2-oxolanylmethyl)-5-dipyrido[1,2-d-3',4'-f]pyrimidinone | Homo sapiens (human) | Potency | 28.1152 | 2 | 0 |
2-[[2-(1-benzotriazolyl)-1-oxoethyl]-(2-furanylmethyl)amino]-N-cyclohexyl-2-(2-fluorophenyl)acetamide | Homo sapiens (human) | Potency | 12.1560 | 2 | 0 |
N-(1,3-benzodioxol-5-yl)-N-[1-(4-chlorophenyl)-2-(cyclohexylamino)-2-oxoethyl]-2-pyrazinecarboxamide | Homo sapiens (human) | Potency | 35.3950 | 2 | 0 |
2-[[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]thio]-3-ethyl-4-quinazolinone | Homo sapiens (human) | Potency | 41.3999 | 1 | 0 |
LSM-26505 | Homo sapiens (human) | Potency | 23.2809 | 1 | 0 |
9,10-dimethoxy-2-(2-pyridinylmethylamino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-one | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrile | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
LSM-34582 | Homo sapiens (human) | Potency | 26.2574 | 3 | 0 |
1,4,8-trimethyl-12-quinolino[2,3-b]quinolinamine | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
2-[[2-[4-(4-chlorophenyl)-1-piperazinyl]-2-oxoethyl]thio]-3-ethyl-4-quinazolinone | Homo sapiens (human) | Potency | 11.6681 | 1 | 0 |
6-(4-benzoyl-1-piperazinyl)-3,3-dimethyl-8-propan-2-yl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrile | Homo sapiens (human) | Potency | 25.8480 | 2 | 0 |
4-chloro-N-[3-chloro-4-(4-morpholinyl)phenyl]benzamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
6-bromo-3-(4-morpholinyl)-4-phenyl-1H-quinolin-2-one | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acid | Homo sapiens (human) | Potency | 28.5992 | 4 | 0 |
2-[[(2,3-dimethoxyphenyl)-oxomethyl]amino]-5-propan-2-yl-3-thiophenecarboxamide | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
5-(2,3-dihydroindol-1-ylsulfonyl)-1,3-diethyl-2-benzimidazolone | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(3-pyridinyl)-4-quinolinecarboxamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
5-[(5-tert-butyl-2,3-dimethylphenyl)sulfonylamino]-2-hydroxybenzoic acid | Homo sapiens (human) | Potency | 37.3176 | 2 | 0 |
9-(3-bromo-4-hydroxyphenyl)-10-phenyl-3,4,5,6,7,9-hexahydro-2H-acridine-1,8-dione | Homo sapiens (human) | Potency | 27.2500 | 2 | 0 |
2-[2,5-dimethyl-3-[(2,4,6-trioxo-1,3-diazinan-5-ylidene)methyl]-1-pyrrolyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid ethyl ester | Homo sapiens (human) | Potency | 19.2989 | 3 | 0 |
[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-thiophen-2-ylmethanone | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
8,9-dimethyl-N-(3-methylphenyl)-3-[2-(4-morpholinyl)ethyl]-4H-[1,3]thiazino[6,5-b]quinolin-2-imine | Homo sapiens (human) | Potency | 12.9547 | 2 | 0 |
4,6-bis(1-imidazolyl)-N,N-diphenyl-1,3,5-triazin-2-amine | Homo sapiens (human) | Potency | 20.8002 | 2 | 0 |
3-(benzenesulfonyl)-2-imino-1-propyl-5-dipyrido[1,2-d-3',4'-f]pyrimidinone | Homo sapiens (human) | Potency | 29.8816 | 2 | 0 |
(2S)-3-(1H-indol-3-yl)-2-[[2-[(4-methyl-6-oxo-3-benzo[c][1]benzopyranyl)oxy]-1-oxoethyl]amino]propanoic acid | Homo sapiens (human) | Potency | 63.0957 | 1 | 0 |
N,N-dibutyl-2-(pyridin-4-yl)quinazolin-4-amine | Homo sapiens (human) | Potency | 32.8851 | 1 | 0 |
3-cyclohexyl-10-methyl-2-thiophen-2-ylpyrimido[4,5-b]quinoline-4,5-dione | Homo sapiens (human) | Potency | 26.3733 | 2 | 0 |
mcb-613 | Homo sapiens (human) | Potency | 41.8711 | 2 | 0 |
N-(4-ethoxyphenyl)-4-[[4-(methylthio)phenyl]sulfonylamino]benzenesulfonamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
reversan | Homo sapiens (human) | Potency | 32.8851 | 1 | 0 |
2-(2-chlorophenyl)-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-4-quinolinecarboxamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
2-pyridin-4-yl-N-[4-(2-thiazolylsulfamoyl)phenyl]-4-quinolinecarboxamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4,5-diphenyl-2-thiazolyl)acetamide | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanone | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamide | Homo sapiens (human) | Potency | 57.1210 | 3 | 0 |
5-(3,4-dimethoxyphenyl)-2-methyl-4-(4-methyl-1-piperidinyl)thieno[2,3-d]pyrimidine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]thio]-3-ethyl-5,6-dimethyl-4-thieno[2,3-d]pyrimidinone | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
thiourea | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
5-(4-Chloro-benzenesulfonyl)-pyrimidine-2,4-diamine | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
2-[4-[[4-[bis(2-hydroxyethyl)amino]-2-chlorophenyl]-(2-chlorophenyl)methyl]-3-chloro-N-(2-hydroxyethyl)anilino]ethanol | Homo sapiens (human) | Potency | 23.6309 | 3 | 0 |
1-[8-chloro-4-(1-naphthalenyl)-3,3a,4,9b-tetrahydrocyclopenta[c]quinolin-5-yl]ethanone | Homo sapiens (human) | Potency | 20.2698 | 3 | 0 |
4-(3-methoxyphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazoline-2-thione | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dione | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
1-(2,4-dimethoxyphenyl)-3-[4-(4-morpholinyl)anilino]pyrrolidine-2,5-dione | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
N-[3-chloro-4-(4-morpholinyl)phenyl]-1,1-dioxo-1,2-benzothiazol-3-amine | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[[4-methyl-5-(2-methyl-3-furanyl)-1,2,4-triazol-3-yl]thio]ethanone | Homo sapiens (human) | Potency | 13.0918 | 1 | 0 |
2-[(4-chlorophenyl)-[2-[5-(4-chlorophenyl)-2-thiazolyl]-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]propanedinitrile | Homo sapiens (human) | Potency | 70.7946 | 1 | 0 |
2-[(3-cyano-4,6-diphenyl-2-pyridinyl)thio]-3-methylbutanoic acid | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
3-[[5,6-bis(4-methoxyphenyl)-4-furo[2,3-d]pyrimidinyl]amino]-1-propanol | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
6-amino-5,7,7-tricyano-8-pyridin-4-yl-1,3,8,8a-tetrahydroisoquinoline-2-carboxylic acid (phenylmethyl) ester | Homo sapiens (human) | Potency | 47.0795 | 3 | 0 |
N-cyclohexyl-2-[3-methoxy-N-(1-oxo-2-thiophen-2-ylethyl)-4-(1-tetrazolyl)anilino]-2-(4-methylphenyl)acetamide | Homo sapiens (human) | Potency | 15.1802 | 2 | 0 |
CID 3192987 | Homo sapiens (human) | Potency | 21.9889 | 3 | 0 |
N-[2-(cyclohexylamino)-2-oxo-1-thiophen-2-ylethyl]-2,2,2-trifluoro-N-(4-methylphenyl)acetamide | Homo sapiens (human) | Potency | 12.9547 | 2 | 0 |
2-(4-ethoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acid | Homo sapiens (human) | Potency | 36.6799 | 3 | 0 |
N,N-diethyl-4-[[5-oxo-6-(phenylmethyl)-7H-pyrrolo[3,4-b]pyridin-7-yl]amino]benzenesulfonamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
1-methyl-N-(2-methylcyclohexyl)-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamide | Homo sapiens (human) | Potency | 17.7395 | 2 | 0 |
benzoic acid [4-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)-2-methoxyphenyl] ester | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
4-[[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholine | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
3-(3-bromoanilino)-2-oxo-1H-indole-3-carbonitrile | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
2-chloro-N-(2-methyl-6-oxo-5H-benzo[b][1,4]benzoxazepin-8-yl)acetamide | Homo sapiens (human) | Potency | 30.0653 | 3 | 0 |
N-(2,2,4-trimethyl-3H-benzofuran-7-yl)benzenesulfonamide | Homo sapiens (human) | Potency | 9.2683 | 1 | 0 |
1-bromo-3-(5,5-dimethyl-3-phenyl-4H-pyrazolo[4,3-a]carbazol-10-yl)-2-propanol | Homo sapiens (human) | Potency | 29.3089 | 1 | 0 |
2-[(2,6-dichlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinone | Homo sapiens (human) | Potency | 17.4372 | 2 | 0 |
2-[(4-hydroxy-3-nitrophenyl)sulfonylamino]benzoic acid [2-(4-methoxyphenyl)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 52.1194 | 1 | 0 |
3,3-bis(4-hydroxy-2-methylphenyl)-1-isobenzofuranone | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
2-[[6-amino-2-(4-methoxyanilino)-5-nitro-4-pyrimidinyl]amino]ethanol | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
LSM-16826 | Homo sapiens (human) | Potency | 34.5598 | 2 | 0 |
2-(3-oxo-2,4-dihydroquinoxalin-1-yl)-2-phenyl-N-(4-propan-2-ylphenyl)acetamide | Homo sapiens (human) | Potency | 32.4648 | 2 | 0 |
LSM-28572 | Homo sapiens (human) | Potency | 46.4515 | 1 | 0 |
[5-(4-fluorophenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[2-(3-pyridinyl)-1-piperidinyl]methanone | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazole | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
luteolin-7-glucoside | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
gamma-linolenic acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
indocyanine green | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
prostaglandin f2 methyl ester | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
neoglycyrol | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
4-amino-6,7-diphenyl-3H-pteridine-2-thione | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
morusinol | Homo sapiens (human) | Potency | 70.7946 | 1 | 0 |
3,3'-diethylthiacarbocyanine iodide | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
2-[[6-[(5-chloro-2,4-dimethoxyanilino)-oxomethyl]-1,2,3,4-tetrahydroacridin-9-yl]thio]acetic acid | Homo sapiens (human) | Potency | 40.1516 | 2 | 0 |
4-[3-[(3-chloro-4-fluoroanilino)-oxomethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid tert-butyl ester | Homo sapiens (human) | Potency | 16.9600 | 3 | 0 |
1-[2-(2,5-dimethylphenoxy)ethyl]-3-indolecarboxylic acid | Homo sapiens (human) | Potency | 32.8851 | 1 | 0 |
u 74389g | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
lissamine rhodamine b | Homo sapiens (human) | Potency | 2.2387 | 1 | 0 |
cnidicin | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
pimaric acid | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
5-methoxy-8,8-dimethyl-2-phenyl-4H,8H-pyrano[2,3-h]chromen-4-one | Homo sapiens (human) | Potency | 30.1272 | 3 | 0 |
glabrol | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
Dihydro-beta-erythroidine hydrobromide | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
efaroxan hydrochloride | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
microcolin a | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
5-[[3-bromo-4-[(2-fluorophenyl)methoxy]-5-methoxyphenyl]methylamino]-1,3-dihydrobenzimidazol-2-one | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
3-bromo-N-[5-(4-morpholinylsulfonyl)-1,3,4-thiadiazol-2-yl]benzamide | Homo sapiens (human) | Potency | 43.0341 | 1 | 0 |
3-[3-(4-fluorophenyl)-2,5,7-trimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-(2-methoxyphenyl)propanamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
[5-(4-bromophenyl)-3-(2-hydroxyphenyl)-3,4-dihydropyrazol-2-yl]-pyridin-4-ylmethanone | Homo sapiens (human) | Potency | 25.6651 | 2 | 0 |
N-[1,4-dimethyl-2,3-dioxo-7-(1-piperidinyl)-6-quinoxalinyl]-4-ethylbenzenesulfonamide | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
acid blue 129 | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
N-[5-Ethyl-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chloride | Homo sapiens (human) | Potency | 38.7463 | 3 | 0 |
N-[5-Bromo-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chloride | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
N-[5-Fluoro-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chloride | Homo sapiens (human) | Potency | 58.4789 | 1 | 0 |
6-(3-cyclopentyloxy-4-methoxyphenyl)-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
6-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-3-(2-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
N-(2-aminophenyl)-4-[[[(2S,3S)-10-[[cyclohexyl(oxo)methyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl-methylamino]methyl]benzamide | Homo sapiens (human) | Potency | 37.5543 | 3 | 0 |
1-[[(2S,3S)-10-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]urea | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
1-[[(2S,3S)-10-(dimethylamino)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]urea | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
N-[4-[2-[3-(dimethylsulfamoyl)anilino]-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamide | Homo sapiens (human) | Potency | 41.3999 | 1 | 0 |
N-[4-[2-(2-methoxyethylamino)-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamide | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
LSM-20825 | Homo sapiens (human) | Potency | 13.9143 | 2 | 0 |
N-[4-[2-(2-oxolanylmethylamino)-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamide | Homo sapiens (human) | Potency | 37.5392 | 3 | 0 |