[no definition available]
EC 3.2.1.18;
Neuraminidase
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (25.00) | 29.6817 |
2010's | 6 (75.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
oseltamivir | Clostridium perfringens | IC50 | 61.1000 | 1 | 1 |
2-deoxy-2,3-dehydro-n-acetylneuraminic acid | Clostridium perfringens | IC50 | 20.0000 | 1 | 1 |
osajin | Clostridium perfringens | IC50 | 3.0600 | 1 | 1 |
osajin | Clostridium perfringens | Ki | 3.2100 | 1 | 1 |
cristacarpin | Clostridium perfringens | IC50 | 2.2800 | 1 | 1 |
cristacarpin | Clostridium perfringens | Ki | 0.3100 | 1 | 1 |
bcx 1812 | Clostridium perfringens | IC50 | 39.6000 | 1 | 1 |
8-deoxygartanin | Clostridium perfringens | IC50 | 29.2000 | 1 | 1 |
8-deoxygartanin | Clostridium perfringens | Ki | 15.5000 | 1 | 1 |
gs 4071 | Clostridium perfringens | IC50 | 0.0010 | 1 | 1 |
6,8-diprenylgenistein | Clostridium perfringens | IC50 | 4.0400 | 1 | 1 |
6,8-diprenylgenistein | Clostridium perfringens | Ki | 4.2900 | 1 | 1 |
quercetin | Clostridium perfringens | IC50 | 9.9200 | 5 | 5 |
apigenin | Clostridium perfringens | IC50 | 17.4000 | 2 | 2 |
luteolin | Clostridium perfringens | IC50 | 4.3000 | 1 | 1 |
herbacetin | Clostridium perfringens | IC50 | 1.4000 | 1 | 1 |
gossypetin | Clostridium perfringens | IC50 | 0.8000 | 1 | 1 |
apigetrin | Clostridium perfringens | IC50 | 39.3000 | 1 | 1 |
rutin | Clostridium perfringens | IC50 | 30.9000 | 1 | 1 |
kaempferol | Clostridium perfringens | IC50 | 8.0000 | 1 | 1 |
genistein | Clostridium perfringens | IC50 | 12.0500 | 1 | 1 |
gartanin | Clostridium perfringens | IC50 | 2.9000 | 1 | 1 |
gartanin | Clostridium perfringens | Ki | 2.0183 | 2 | 2 |
3-hydroxyblancoxanthone | Clostridium perfringens | IC50 | 0.1860 | 1 | 1 |
3-hydroxyblancoxanthone | Clostridium perfringens | Ki | 0.2901 | 2 | 2 |
mangiferin | Clostridium perfringens | IC50 | 16.2000 | 1 | 1 |
mangostin | Clostridium perfringens | IC50 | 12.2000 | 1 | 1 |
mangostin | Clostridium perfringens | Ki | 5.8000 | 1 | 1 |
astragalin | Clostridium perfringens | IC50 | 29.4000 | 1 | 1 |
kaempferol-3-o-rutinoside | Clostridium perfringens | IC50 | 55.5000 | 1 | 1 |
auriculasin | Clostridium perfringens | IC50 | 0.3000 | 1 | 1 |
auriculasin | Clostridium perfringens | Ki | 0.1300 | 1 | 1 |
gamma-mangostin | Clostridium perfringens | IC50 | 2.2000 | 1 | 1 |
gamma-mangostin | Clostridium perfringens | Ki | 4.1050 | 2 | 2 |
beta-Mangostin | Clostridium perfringens | IC50 | 60.7000 | 1 | 1 |
beta-Mangostin | Clostridium perfringens | Ki | 24.9000 | 1 | 1 |
9-Hydroxycalabaxanthone | Clostridium perfringens | IC50 | 20.1000 | 1 | 1 |
9-Hydroxycalabaxanthone | Clostridium perfringens | Ki | 5.9000 | 1 | 1 |
2,3,6,8-tetrahydroxy-1-(3-methylbut-2-enyl)-5-(2-methylbut-3-en-2-yl)-9h-xanthen-9-one | Clostridium perfringens | IC50 | 0.2450 | 1 | 1 |
2,3,6,8-tetrahydroxy-1-(3-methylbut-2-enyl)-5-(2-methylbut-3-en-2-yl)-9h-xanthen-9-one | Clostridium perfringens | Ki | 0.1748 | 2 | 2 |
cudraxanthone l | Clostridium perfringens | IC50 | 0.2280 | 1 | 1 |
cudraxanthone l | Clostridium perfringens | Ki | 0.3528 | 2 | 2 |
1-methoxyerythrabyssin ii | Clostridium perfringens | IC50 | 0.0900 | 1 | 1 |
1-methoxyerythrabyssin ii | Clostridium perfringens | Ki | 0.1100 | 1 | 1 |