An acyl-CoA desaturase 1 that is encoded in the genome of rat. [OMA:P07308, PRO:DNx]
EC 1.14.19.1;
Delta(9)-desaturase 1;
Delta-9 desaturase 1;
Fatty acid desaturase 1;
Stearoyl-CoA desaturase 1
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 7 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
tacrine | Rattus norvegicus (Norway rat) | IC50 | 0.0470 | 1 | 1 |
rivastigmine | Rattus norvegicus (Norway rat) | IC50 | 1.7100 | 1 | 1 |
u 69593 | Rattus norvegicus (Norway rat) | Ki | 0.0035 | 1 | 1 |
morphine | Rattus norvegicus (Norway rat) | Ki | 0.2990 | 1 | 1 |
mf 438 | Rattus norvegicus (Norway rat) | IC50 | 0.0537 | 3 | 3 |
mk 8245 | Rattus norvegicus (Norway rat) | IC50 | 0.0355 | 4 | 4 |
cabozantinib | Rattus norvegicus (Norway rat) | IC50 | 0.0013 | 1 | 1 |
pf 8380 | Rattus norvegicus (Norway rat) | IC50 | 0.0084 | 1 | 1 |
gsk 1363089 | Rattus norvegicus (Norway rat) | IC50 | 0.0004 | 1 | 1 |
dcc-2701 | Rattus norvegicus (Norway rat) | IC50 | 0.0027 | 1 | 1 |