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Adenosine receptor A2b
An adenosine receptor A2b that is encoded in the genome of mouse. [OMA:Q60614, PRO:DNx]
Synonyms
Research
Bioassay Publications (6)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 4 (66.67) | 29.6817 |
| 2010's | 2 (33.33) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (10)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| caffeine | Mus musculus (house mouse) | Ki | 23.0000 | 1 | 1 |
| psb 1115 | Mus musculus (house mouse) | Ki | 1.9400 | 1 | 1 |
| mrs 1754 | Mus musculus (house mouse) | Ki | 0.0033 | 2 | 2 |
Drugs with Activation Measurements
Drugs with Other Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| enprofylline | Mus musculus (house mouse) | Kb | 18.0000 | 1 | 1 |
| theophylline | Mus musculus (house mouse) | Kb | 16.0000 | 1 | 1 |
| caffeine | Mus musculus (house mouse) | Kb | 25.0000 | 1 | 1 |
| cvt-6883 | Mus musculus (house mouse) | Kb | 0.0020 | 1 | 1 |
| psb 11 | Mus musculus (house mouse) | Kb | 2.1000 | 1 | 1 |
Fluorescent-Labeled Selective Adenosine AJournal of medicinal chemistry, , 05-24, Volume: 61, Issue:10, 2018
Imidazo[2,1-i]purin-5-ones and related tricyclic water-soluble purine derivatives: potent A(2A)- and A(3)-adenosine receptor antagonists.Journal of medicinal chemistry, , Aug-01, Volume: 45, Issue:16, 2002
AJournal of medicinal chemistry, , 04-25, Volume: 62, Issue:8, 2019
AJournal of medicinal chemistry, , 04-25, Volume: 62, Issue:8, 2019
1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity.Journal of medicinal chemistry, , Jul-09, Volume: 52, Issue:13, 2009