Proteins > G-protein coupled receptor 55
Page last updated: 2024-08-07 15:19:04

G-protein coupled receptor 55

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (64)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
bisacodylHomo sapiens (human)IC500.908410
nitrendipineHomo sapiens (human)IC501.465210
phenolphthaleinHomo sapiens (human)IC506.667210
1,6-bismaleimidohexaneHomo sapiens (human)IC509.790710
helenalinHomo sapiens (human)IC502.642310
angustibalinHomo sapiens (human)IC504.494410
4-[1-(4-hydroxyphenyl)ethenyl]phenolHomo sapiens (human)IC501.753910
1-[(4-methylphenyl)methyl]-4-[4-(4-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineHomo sapiens (human)IC5032.000010
2-(4-methoxyphenyl)-5-(3-pyridinyl)-1,3,4-oxadiazoleHomo sapiens (human)IC5032.000010
3-phenyl-5-(2-phenylphenyl)-1,2,4-oxadiazoleHomo sapiens (human)IC506.085310
4-(4-anilinoanilino)-2-quinazolinecarboxylic acid ethyl esterHomo sapiens (human)IC502.481110
4-(3-bromophenyl)-2-(4-bromophenyl)-7-methylpyrazolo[3,4-d]pyridazineHomo sapiens (human)IC500.904020
4-(3-bromophenyl)-7-methyl-2-(4-methylphenyl)pyrazolo[3,4-d]pyridazineHomo sapiens (human)IC501.723220
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(3-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)IC501.002520
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(2-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)IC500.299730
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)IC501.265820
2-furanyl-[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]methanoneHomo sapiens (human)IC501.140420
[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-thiophen-2-ylmethanoneHomo sapiens (human)IC504.130010
1-[(4-methylphenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineHomo sapiens (human)IC5032.000010
1-[(4-chlorophenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineHomo sapiens (human)IC5032.000010
2-phenyl-N-[4-(2-thiazolylsulfamoyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)IC505.750010
3-chloro-N-[3-[[(3-chloro-4-nitrophenyl)-oxomethyl]amino]-2,2-dimethylpropyl]-4-nitrobenzamideHomo sapiens (human)IC503.112310
N-[4-[(4,6-dimethyl-2-pyrimidinyl)sulfamoyl]phenyl]-2-phenyl-4-quinolinecarboxamideHomo sapiens (human)IC5013.700010
2-(2-chlorophenyl)-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-4-quinolinecarboxamideHomo sapiens (human)IC504.630010
2-pyridin-4-yl-N-[4-(2-thiazolylsulfamoyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)IC5032.000010
5-cyano-6-phenoxy-2-phenyl-3-pyridinecarboxylic acid ethyl esterHomo sapiens (human)IC501.688610
N-[4-(butylsulfamoyl)phenyl]-2-phenyl-2-(phenylthio)acetamideHomo sapiens (human)IC501.124910
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamideHomo sapiens (human)IC506.557810
2-[[2,2,2-trichloro-1-[(2,2-dimethyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterHomo sapiens (human)IC502.006010
9-(1H-indol-3-yl)acridineHomo sapiens (human)IC504.831610
[4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)IC500.507530
N-ethyl-N-(2-ethylphenyl)-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideHomo sapiens (human)IC501.059610
3,3-bis(4-hydroxyphenyl)-7-methyl-1,3-dihydro-2h-indol-2-oneHomo sapiens (human)IC501.329720
4-chloro-5-(2,3-dihydro-1,4-benzodioxin-3-yl)thieno[2,3-d]pyrimidineHomo sapiens (human)IC503.379510
3,3-bis(4-hydroxy-2-methylphenyl)-1-isobenzofuranoneHomo sapiens (human)IC503.464810
perhexiline maleateHomo sapiens (human)IC503.188810
fendiline hydrochlorideHomo sapiens (human)IC503.103810
4-[3-[(3-chloro-4-fluoroanilino)-oxomethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid tert-butyl esterHomo sapiens (human)IC501.176820
2-[(1R,3S)-3-(7-bromo-2-methyl-1H-indol-3-yl)-2,2-dimethylcyclopropyl]acetonitrileHomo sapiens (human)IC501.490110
cid-2745687Homo sapiens (human)IC509.080010
cid16020046Homo sapiens (human)IC501.178410
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esterHomo sapiens (human)IC502.546310
3-[1-[[1-(4-methoxyphenyl)cyclopropyl]-oxomethyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneHomo sapiens (human)IC509.550010
3-[1-[[1-(4-methylphenyl)cyclopropyl]-oxomethyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneHomo sapiens (human)IC502.682220
3-[1-[oxo-(1-phenylcyclopropyl)methyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneHomo sapiens (human)IC5017.400010
3-[1-[[1-(4-chlorophenyl)cyclopropyl]-oxomethyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneHomo sapiens (human)IC500.719920

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
isovelleralHomo sapiens (human)EC500.500010
nile redHomo sapiens (human)EC500.500010
5-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)EC5032.000010
3-(4-methoxyphenyl)-8-(6-methyl-2-phenyl-4-pyrimidinyl)-8-azabicyclo[3.2.1]octan-3-olHomo sapiens (human)EC507.353610
1-[(1-cyclopentyl-5-tetrazolyl)-thiophen-2-ylmethyl]-4-(2-methoxyphenyl)piperazineHomo sapiens (human)EC506.330110
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamideHomo sapiens (human)EC5017.676610
N-(2-furanylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)EC5032.000010
2-[(7-methoxy-4-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)thio]-N-methyl-N-(4-phenyl-2-thiazolyl)acetamideHomo sapiens (human)EC5032.000010
5-bromo-N-(4-methoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)EC5032.000010
3-[[4-(2,3-dimethylphenyl)-1-piperazinyl]-oxomethyl]-N,N-dimethyl-4-(1-pyrrolidinyl)benzenesulfonamideHomo sapiens (human)EC500.385420
2-[(5-chloro-1,3-benzothiazol-2-yl)thio]-N-[3-(4-morpholinylsulfonyl)phenyl]propanamideHomo sapiens (human)EC500.860820
4-(3,5-dimethyl-1-pyrazolyl)-N-[2-methoxy-5-(4-morpholinylsulfonyl)phenyl]benzamideHomo sapiens (human)EC500.831010
2-(4-methoxyphenyl)-N-[2-(4-morpholinyl)-5-(4-morpholinylsulfonyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)EC501.684510
N-[3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxo-1-pyrrolidinyl)benzamideHomo sapiens (human)EC501.370010
N,N-dimethyl-3-[[4-(4-nitrophenyl)-1-piperazinyl]-oxomethyl]-4-(1-pyrrolidinyl)benzenesulfonamideHomo sapiens (human)EC500.674720
5233705 compoundHomo sapiens (human)EC5032.000010
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneHomo sapiens (human)EC5032.000010
N-[2-methoxy-5-(4-morpholinylsulfonyl)phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHomo sapiens (human)EC500.414420