Page last updated: 2024-08-07 20:57:39

thioredoxin reductase

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (2740)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
dinitrochlorobenzeneRattus norvegicus (Norway rat)Potency2.818410
3-hydroxyanthranilic acidRattus norvegicus (Norway rat)Potency79.432810
gamma-aminobutyric acidRattus norvegicus (Norway rat)Potency19.952610
5-aminovaleric acidRattus norvegicus (Norway rat)Potency8.436820
agmatineRattus norvegicus (Norway rat)Potency0.562310
quinacrineRattus norvegicus (Norway rat)Potency6.610220
aminooxyacetic acidRattus norvegicus (Norway rat)Potency3.233620
catecholRattus norvegicus (Norway rat)Potency13.785630
chlordeconeRattus norvegicus (Norway rat)Potency100.000010
salicylic acidRattus norvegicus (Norway rat)Potency63.095710
4-methylumbelliferyl acetateRattus norvegicus (Norway rat)Potency25.118910
4-amino-1,2-oxazolidin-3-oneRattus norvegicus (Norway rat)Potency0.023810
4-aminophenolRattus norvegicus (Norway rat)Potency11.519020
bupropionRattus norvegicus (Norway rat)Potency3.162310
[3-carboxy-2-(1-oxohexadecoxy)propyl]-trimethylammoniumRattus norvegicus (Norway rat)Potency17.558220
taxifolinRattus norvegicus (Norway rat)Potency18.186520
3,4-dihydroxyphenylacetic acidRattus norvegicus (Norway rat)Potency18.944620
cysteineRattus norvegicus (Norway rat)Potency50.118710
histamineRattus norvegicus (Norway rat)Potency23.778110
hydroquinoneRattus norvegicus (Norway rat)Potency32.850210
hydroxylamineRattus norvegicus (Norway rat)Potency0.794310
indol-3-yl pyruvic acidRattus norvegicus (Norway rat)Potency50.118710
racepinephrineRattus norvegicus (Norway rat)Potency5.972820
melatoninRattus norvegicus (Norway rat)Potency13.766220
n-acetylserotoninRattus norvegicus (Norway rat)Potency21.192310
naphthaleneRattus norvegicus (Norway rat)Potency89.125110
norepinephrine, (+,-)-isomerRattus norvegicus (Norway rat)Potency12.657620
pyrazinamideRattus norvegicus (Norway rat)Potency0.004710
pyrazinoic acidRattus norvegicus (Norway rat)Potency89.125110
quinolinic acidRattus norvegicus (Norway rat)Potency0.381420
spermidineRattus norvegicus (Norway rat)Potency0.398110
spermineRattus norvegicus (Norway rat)Potency0.354810
2,3-dichloro-alpha-methylbenzylamineRattus norvegicus (Norway rat)Potency0.707910
sk&f 81297Rattus norvegicus (Norway rat)Potency23.778120
7-hydroxy-2-n,n-dipropylaminotetralinRattus norvegicus (Norway rat)Potency15.067730
sk&f 82958Rattus norvegicus (Norway rat)Potency23.299220
1-hydroxy-3-amino-2-pyrrolidoneRattus norvegicus (Norway rat)Potency37.685810
gallopamilRattus norvegicus (Norway rat)Potency1.000010
normetanephrineRattus norvegicus (Norway rat)Potency1.000010
sk&f 77434Rattus norvegicus (Norway rat)Potency15.848910
sk&f-38393Rattus norvegicus (Norway rat)Potency3.577130
perillic acidRattus norvegicus (Norway rat)Potency1.337110
mandelic acidRattus norvegicus (Norway rat)Potency79.432810
dimethylphenylpiperazinium iodideRattus norvegicus (Norway rat)Potency1.000010
1,10-diaminodecaneRattus norvegicus (Norway rat)Potency0.474410
1,3-diethyl-8-phenylxanthineRattus norvegicus (Norway rat)Potency37.685810
1,3-dipropyl-8-cyclopentylxanthineRattus norvegicus (Norway rat)Potency37.685810
1,3-dipropyl-8-(4-sulfophenyl)xanthineRattus norvegicus (Norway rat)Potency18.909740
1,5-dihydroxyisoquinolineRattus norvegicus (Norway rat)Potency31.622810
1-(1-naphthyl)piperazineRattus norvegicus (Norway rat)Potency25.118910
1-(2-methoxyphenyl)piperazineRattus norvegicus (Norway rat)Potency17.658820
1-(5-isoquinolinylsulfonyl)-3-methylpiperazineRattus norvegicus (Norway rat)Potency42.284120
1-anilino-8-naphthalenesulfonateRattus norvegicus (Norway rat)Potency70.794610
1h-(1,2,4)oxadiazolo(4,3-a)quinoxalin-1-oneRattus norvegicus (Norway rat)Potency26.407620
2,2'-dipyridylRattus norvegicus (Norway rat)Potency0.054410
2,4-dichlorophenoxyacetic acidRattus norvegicus (Norway rat)Potency1.122010
4-(2,4-dichlorophenoxy)butyric acidRattus norvegicus (Norway rat)Potency89.125110
2-amino-5,6-dihydro-6-methyl-4h-1,3-thiazineRattus norvegicus (Norway rat)Potency3.162310
pyrithioneRattus norvegicus (Norway rat)Potency11.220210
3,4-dichloroisocoumarinRattus norvegicus (Norway rat)Potency6.139920
phaclofenRattus norvegicus (Norway rat)Potency0.398110
3-bromo-7-nitroindazoleRattus norvegicus (Norway rat)Potency28.340410
enprofyllineRattus norvegicus (Norway rat)Potency3.768620
3-nitropropionic acidRattus norvegicus (Norway rat)Potency0.707910
mdl 72222Rattus norvegicus (Norway rat)Potency42.284120
4,5,6,7-tetrabromo-2-azabenzimidazoleRattus norvegicus (Norway rat)Potency26.679510
cgp 52411Rattus norvegicus (Norway rat)Potency37.685810
(4-amidinophenyl)methanesulfonyl fluorideRattus norvegicus (Norway rat)Potency0.316210
4-amino-1,8-naphthalimideRattus norvegicus (Norway rat)Potency35.636710
4-aminopyridineRattus norvegicus (Norway rat)Potency89.125120
p-chloromercuribenzoic acidRattus norvegicus (Norway rat)Potency0.676730
homovanillic acidRattus norvegicus (Norway rat)Potency42.284110
4-phenyl-3-furoxancarbonitrileRattus norvegicus (Norway rat)Potency9.466210
5,5-dimethyl-1-pyrroline-1-oxideRattus norvegicus (Norway rat)Potency29.934910
phenytoinRattus norvegicus (Norway rat)Potency1.000010
5,7-dichlorokynurenic acidRattus norvegicus (Norway rat)Potency8.436840
5-dimethylamilorideRattus norvegicus (Norway rat)Potency37.685810
5-(n,n-hexamethylene)amilorideRattus norvegicus (Norway rat)Potency59.727920
ethylisopropylamilorideRattus norvegicus (Norway rat)Potency26.679510
5-fluoroindole-2-carboxylic acidRattus norvegicus (Norway rat)Potency32.708120
hydroxyindoleacetic acidRattus norvegicus (Norway rat)Potency22.252930
6,7-dichloroquinoxaline-2,3-dioneRattus norvegicus (Norway rat)Potency40.918830
6-fluoronorepinephrineRattus norvegicus (Norway rat)Potency9.466220
6-hydroxymelatoninRattus norvegicus (Norway rat)Potency17.925620
6-methoxytryptolineRattus norvegicus (Norway rat)Potency26.237610
6-nitroso-1,2-benzopyroneRattus norvegicus (Norway rat)Potency27.483130
7-nitroindazoleRattus norvegicus (Norway rat)Potency0.316210
8-(4-sulfophenyl)theophyllineRattus norvegicus (Norway rat)Potency21.497840
8-phenyltheophyllineRattus norvegicus (Norway rat)Potency2.889220
tacrineRattus norvegicus (Norway rat)Potency7.519320
N-(2-aminoethyl)-5-chloro-1-naphthalenesulfonamideRattus norvegicus (Norway rat)Potency3.162310
aa 861Rattus norvegicus (Norway rat)Potency26.604220
abt 702Rattus norvegicus (Norway rat)Potency15.904930
acetazolamideRattus norvegicus (Norway rat)Potency0.927520
acetochlorRattus norvegicus (Norway rat)Potency31.622810
acetohexamideRattus norvegicus (Norway rat)Potency1.258910
acridoneRattus norvegicus (Norway rat)Potency56.607220
beta-aminoethyl isothioureaRattus norvegicus (Norway rat)Potency14.125410
ag 127Rattus norvegicus (Norway rat)Potency37.685810
rtki cpdRattus norvegicus (Norway rat)Potency0.316220
tyrphostin a23Rattus norvegicus (Norway rat)Potency31.591420
tyrphostin 25Rattus norvegicus (Norway rat)Potency50.118710
tyrphostin a1Rattus norvegicus (Norway rat)Potency28.243830
tyrphostin ag957Rattus norvegicus (Norway rat)Potency56.234110
1-aminoindan-1,5-dicarboxylic acidRattus norvegicus (Norway rat)Potency16.603030
alachlorRattus norvegicus (Norway rat)Potency89.125110
albuterolRattus norvegicus (Norway rat)Potency3.235720
alfuzosinRattus norvegicus (Norway rat)Potency18.647730
alpha-methyltyrosine methyl esterRattus norvegicus (Norway rat)Potency16.833610
altretamineRattus norvegicus (Norway rat)Potency8.912510
amantadineRattus norvegicus (Norway rat)Potency6.297320
aminoglutethimideRattus norvegicus (Norway rat)Potency21.236510
theophyllineRattus norvegicus (Norway rat)Potency14.125410
dan 2163Rattus norvegicus (Norway rat)Potency21.192310
amitriptylineRattus norvegicus (Norway rat)Potency28.183810
amoxapineRattus norvegicus (Norway rat)Potency79.432810
amsacrineRattus norvegicus (Norway rat)Potency23.487730
6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diolRattus norvegicus (Norway rat)Potency13.525930
aprindineRattus norvegicus (Norway rat)Potency16.833610
arecolineRattus norvegicus (Norway rat)Potency1.000010
aspirinRattus norvegicus (Norway rat)Potency16.599120
2-amino-3-(5-tert-butyl-3-oxo-4-isoxazolyl)propanoic acidRattus norvegicus (Norway rat)Potency0.029910
aurintricarboxylic acidRattus norvegicus (Norway rat)Potency34.269220
azathioprineRattus norvegicus (Norway rat)Potency14.659720
azinphosmethylRattus norvegicus (Norway rat)Potency28.183810
azepexoleRattus norvegicus (Norway rat)Potency20.814230
baclofenRattus norvegicus (Norway rat)Potency8.421610
benserazideRattus norvegicus (Norway rat)Potency3.665230
benzamideRattus norvegicus (Norway rat)Potency5.972810
bicalutamideRattus norvegicus (Norway rat)Potency0.398110
biperidenRattus norvegicus (Norway rat)Potency0.562310
brimonidineRattus norvegicus (Norway rat)Potency11.976040
b 169Rattus norvegicus (Norway rat)Potency33.587520
bumetanideRattus norvegicus (Norway rat)Potency46.402110
verapamilRattus norvegicus (Norway rat)Potency0.398110
calmidazoliumRattus norvegicus (Norway rat)Potency17.782810
carbazilquinoneRattus norvegicus (Norway rat)Potency50.118710
carisoprodolRattus norvegicus (Norway rat)Potency29.934910
3-[[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-8-oxo-7-[[1-oxo-2-(1-tetrazolyl)ethyl]amino]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidRattus norvegicus (Norway rat)Potency35.481310
cgs 15943Rattus norvegicus (Norway rat)Potency28.112820
chelerythrineRattus norvegicus (Norway rat)Potency39.810720
chlorambucilRattus norvegicus (Norway rat)Potency23.021720
chlormezanoneRattus norvegicus (Norway rat)Potency0.125910
chloroquineRattus norvegicus (Norway rat)Potency0.354810
chloroxineRattus norvegicus (Norway rat)Potency56.234110
chlorpromazineRattus norvegicus (Norway rat)Potency1.995310
chlorpropamideRattus norvegicus (Norway rat)Potency0.891310
cilostamideRattus norvegicus (Norway rat)Potency17.782810
cilostazolRattus norvegicus (Norway rat)Potency0.446710
cinoxacinRattus norvegicus (Norway rat)Potency28.982230
ciprofibrateRattus norvegicus (Norway rat)Potency13.371410
citalopramRattus norvegicus (Norway rat)Potency1.061020
5,7-dimethoxycoumarinRattus norvegicus (Norway rat)Potency22.983320
clemastineRattus norvegicus (Norway rat)Potency37.685810
clioquinolRattus norvegicus (Norway rat)Potency43.688010
clofibrateRattus norvegicus (Norway rat)Potency0.398110
clofoctolRattus norvegicus (Norway rat)Potency50.118710
clotrimazoleRattus norvegicus (Norway rat)Potency0.631010
cx546Rattus norvegicus (Norway rat)Potency2.687720
cystamineRattus norvegicus (Norway rat)Potency11.389440
decamethoniumRattus norvegicus (Norway rat)Potency3.548110
dephostatinRattus norvegicus (Norway rat)Potency1.555420
dequaliniumRattus norvegicus (Norway rat)Potency0.891320
desipramineRattus norvegicus (Norway rat)Potency8.436810
diphenyleneiodoniumRattus norvegicus (Norway rat)Potency17.499220
dipyridamoleRattus norvegicus (Norway rat)Potency36.953520
disulfiramRattus norvegicus (Norway rat)Potency18.892620
2-amino-7-phosphonoheptanoic acidRattus norvegicus (Norway rat)Potency1.778310
racemetirosineRattus norvegicus (Norway rat)Potency37.685820
2,3-dimethoxy-1,4-naphthoquinoneRattus norvegicus (Norway rat)Potency30.868920
domperidoneRattus norvegicus (Norway rat)Potency3.162310
adtnRattus norvegicus (Norway rat)Potency7.018220
doxazosinRattus norvegicus (Norway rat)Potency29.285730
dsp 4Rattus norvegicus (Norway rat)Potency4.807930
ebastineRattus norvegicus (Norway rat)Potency8.912510
ebselenRattus norvegicus (Norway rat)Potency14.771520
nsc-526417Rattus norvegicus (Norway rat)Potency89.125110
edrophoniumRattus norvegicus (Norway rat)Potency4.744420
ellipticineRattus norvegicus (Norway rat)Potency20.595030
emodinRattus norvegicus (Norway rat)Potency9.469820
epinastineRattus norvegicus (Norway rat)Potency31.622810
etazolateRattus norvegicus (Norway rat)Potency16.001420
ethacrynic acidRattus norvegicus (Norway rat)Potency29.881610
profenamineRattus norvegicus (Norway rat)Potency29.934920
ethosuximideRattus norvegicus (Norway rat)Potency29.934910
ethoxyquinRattus norvegicus (Norway rat)Potency89.125110
etodolacRattus norvegicus (Norway rat)Potency1.584910
fenoldopamRattus norvegicus (Norway rat)Potency11.297030
berotekRattus norvegicus (Norway rat)Potency37.685810
fipexideRattus norvegicus (Norway rat)Potency10.000010
flufenamic acidRattus norvegicus (Norway rat)Potency100.000010
flumazenilRattus norvegicus (Norway rat)Potency0.133720
fluorouracilRattus norvegicus (Norway rat)Potency0.446710
fluoxetineRattus norvegicus (Norway rat)Potency1.122010
fluspirileneRattus norvegicus (Norway rat)Potency6.684830
4-androsten-4-ol-3,17-dioneRattus norvegicus (Norway rat)Potency0.398110
fpl 64176Rattus norvegicus (Norway rat)Potency18.887610
furafyllineRattus norvegicus (Norway rat)Potency0.891310
gabaculineRattus norvegicus (Norway rat)Potency2.238710
gallamine triethiodideRattus norvegicus (Norway rat)Potency7.317830
4-amino-5-hexynoic acidRattus norvegicus (Norway rat)Potency1.683410
gbr 12935Rattus norvegicus (Norway rat)Potency0.891310
2,5-dihydroxybenzoic acidRattus norvegicus (Norway rat)Potency50.118710
glyburideRattus norvegicus (Norway rat)Potency2.993520
gossypolRattus norvegicus (Norway rat)Potency30.546140
gr 89696Rattus norvegicus (Norway rat)Potency39.810710
granisetronRattus norvegicus (Norway rat)Potency35.481310
guanfacineRattus norvegicus (Norway rat)Potency1.000010
gyki 52466Rattus norvegicus (Norway rat)Potency28.183810
1-(5-isoquinolinesulfonyl)-2-methylpiperazineRattus norvegicus (Norway rat)Potency50.118710
haloperidolRattus norvegicus (Norway rat)Potency2.667920
2,2',3,3',4,4'-hexahydroxy-1,1'-biphenyl-6,6'-dimethanol dimethyl etherRattus norvegicus (Norway rat)Potency14.125410
hemicholinium 3Rattus norvegicus (Norway rat)Potency6.102720
tele-methylhistamineRattus norvegicus (Norway rat)Potency0.446710
hydralazineRattus norvegicus (Norway rat)Potency18.887620
hydroxyureaRattus norvegicus (Norway rat)Potency16.352230
atropine sulfateRattus norvegicus (Norway rat)Potency1.995310
ibudilastRattus norvegicus (Norway rat)Potency19.635420
lidocaineRattus norvegicus (Norway rat)Potency0.538920
imetitRattus norvegicus (Norway rat)Potency2.818410
amrinoneRattus norvegicus (Norway rat)Potency64.775820
indole-3-carbinolRattus norvegicus (Norway rat)Potency50.118710
iodoacetamideRattus norvegicus (Norway rat)Potency22.982120
isoetharineRattus norvegicus (Norway rat)Potency35.636720
4-piperidinecarboxylic acidRattus norvegicus (Norway rat)Potency0.597310
isoproterenolRattus norvegicus (Norway rat)Potency11.795820
isradipineRattus norvegicus (Norway rat)Potency79.432810
1-(2-naphthalenyl)-3-[(phenylmethyl)-propan-2-ylamino]-1-propanoneRattus norvegicus (Norway rat)Potency12.510230
jl 18Rattus norvegicus (Norway rat)Potency30.741020
nsc 664704Rattus norvegicus (Norway rat)Potency28.054430
ketorolacRattus norvegicus (Norway rat)Potency26.679520
labetalolRattus norvegicus (Norway rat)Potency19.430530
lamotrigineRattus norvegicus (Norway rat)Potency28.425430
lansoprazoleRattus norvegicus (Norway rat)Potency1.258910
beta-lapachoneRattus norvegicus (Norway rat)Potency24.079340
lavendustin bRattus norvegicus (Norway rat)Potency39.810710
2-hydroxy-5-(2,5-dihydrobenzyl)aminobenzoic acidRattus norvegicus (Norway rat)Potency39.810710
leflunomideRattus norvegicus (Norway rat)Potency0.631010
tetramisoleRattus norvegicus (Norway rat)Potency0.251210
qx-314Rattus norvegicus (Norway rat)Potency0.631010
lomefloxacinRattus norvegicus (Norway rat)Potency25.067430
loratadineRattus norvegicus (Norway rat)Potency0.446710
loxoprofenRattus norvegicus (Norway rat)Potency3.006430
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-oneRattus norvegicus (Norway rat)Potency32.464820
maprotilineRattus norvegicus (Norway rat)Potency0.084420
edaravoneRattus norvegicus (Norway rat)Potency79.432810
1,5-(diethylamino)piperidineRattus norvegicus (Norway rat)Potency0.281810
meclofenamic acid(1-)Rattus norvegicus (Norway rat)Potency0.354810
sarkolysinRattus norvegicus (Norway rat)Potency20.622530
memantineRattus norvegicus (Norway rat)Potency0.794310
metaproterenolRattus norvegicus (Norway rat)Potency35.481310
methoctramineRattus norvegicus (Norway rat)Potency8.436810
doxorubicin hydrochlorideRattus norvegicus (Norway rat)Potency25.118910
methoxychlorRattus norvegicus (Norway rat)Potency89.125110
3-Hydroxy-alpha-methyl-DL-tyrosineRattus norvegicus (Norway rat)Potency8.291520
methergineRattus norvegicus (Norway rat)Potency84.279020
metolazoneRattus norvegicus (Norway rat)Potency39.482430
metyraponeRattus norvegicus (Norway rat)Potency31.622810
milrinoneRattus norvegicus (Norway rat)Potency0.546720
minoxidilRattus norvegicus (Norway rat)Potency0.597310
mitotaneRattus norvegicus (Norway rat)Potency21.076620
ml 7Rattus norvegicus (Norway rat)Potency37.685820
ml 9Rattus norvegicus (Norway rat)Potency5.972820
acecainideRattus norvegicus (Norway rat)Potency3.162310
ethylmaleimideRattus norvegicus (Norway rat)Potency10.621310
fg 7142Rattus norvegicus (Norway rat)Potency49.502130
n-methyldeoxynojirimycinRattus norvegicus (Norway rat)Potency0.891310
deoxyepinephrineRattus norvegicus (Norway rat)Potency9.347320
apneaRattus norvegicus (Norway rat)Potency3.882230
naftopidilRattus norvegicus (Norway rat)Potency29.934910
nan 190Rattus norvegicus (Norway rat)Potency15.144820
niclosamideRattus norvegicus (Norway rat)Potency0.005310
nifedipineRattus norvegicus (Norway rat)Potency32.518530
nilutamideRattus norvegicus (Norway rat)Potency21.587710
nimesulideRattus norvegicus (Norway rat)Potency37.685810
nimodipineRattus norvegicus (Norway rat)Potency17.053530
nitrendipineRattus norvegicus (Norway rat)Potency17.614320
no 711Rattus norvegicus (Norway rat)Potency10.000010
nomifensineRattus norvegicus (Norway rat)Potency0.562310
masoprocolRattus norvegicus (Norway rat)Potency19.952610
5-nitro-2-(3-phenylpropylamino)benzoic acidRattus norvegicus (Norway rat)Potency0.751910
ns 1619Rattus norvegicus (Norway rat)Potency38.603130
octopamineRattus norvegicus (Norway rat)Potency8.436810
ofloxacinRattus norvegicus (Norway rat)Potency29.750630
oxaprozinRattus norvegicus (Norway rat)Potency31.622810
oxiracetamRattus norvegicus (Norway rat)Potency37.685810
oxolinic acidRattus norvegicus (Norway rat)Potency14.222130
oxotremorine mRattus norvegicus (Norway rat)Potency0.354810
oxyphenbutazoneRattus norvegicus (Norway rat)Potency7.943310
quinoneRattus norvegicus (Norway rat)Potency30.302610
fenclonineRattus norvegicus (Norway rat)Potency39.810710
papaverineRattus norvegicus (Norway rat)Potency0.335920
1,7-dimethylxanthineRattus norvegicus (Norway rat)Potency1.258910
pd 169316Rattus norvegicus (Norway rat)Potency44.668410
pd 98059Rattus norvegicus (Norway rat)Potency0.562310
5-hydroxy-4-methoxy-5-(1-methylethenyl)-2-furanoneRattus norvegicus (Norway rat)Potency14.125410
pentoxifyllineRattus norvegicus (Norway rat)Potency5.168810
phenyl biguanideRattus norvegicus (Norway rat)Potency19.952610
phloretinRattus norvegicus (Norway rat)Potency19.455920
pinacidilRattus norvegicus (Norway rat)Potency1.375110
pindololRattus norvegicus (Norway rat)Potency2.463810
piracetamRattus norvegicus (Norway rat)Potency0.843710
pirenperoneRattus norvegicus (Norway rat)Potency39.810710
praziquantelRattus norvegicus (Norway rat)Potency2.387120
prazosinRattus norvegicus (Norway rat)Potency25.853330
procaineRattus norvegicus (Norway rat)Potency0.398110
promazineRattus norvegicus (Norway rat)Potency89.125110
promethazineRattus norvegicus (Norway rat)Potency10.920130
propachlorRattus norvegicus (Norway rat)Potency19.952610
propafenoneRattus norvegicus (Norway rat)Potency0.678320
propranololRattus norvegicus (Norway rat)Potency42.239520
protoporphyrin ixRattus norvegicus (Norway rat)Potency25.072220
protriptylineRattus norvegicus (Norway rat)Potency39.810710
pyrilamineRattus norvegicus (Norway rat)Potency0.596620
riluzoleRattus norvegicus (Norway rat)Potency16.833610
risperidoneRattus norvegicus (Norway rat)Potency15.003010
rolipramRattus norvegicus (Norway rat)Potency4.259720
sanguinarineRattus norvegicus (Norway rat)Potency31.622810
carbamylhydrazineRattus norvegicus (Norway rat)Potency0.446710
linsidomineRattus norvegicus (Norway rat)Potency42.284120
spiperoneRattus norvegicus (Norway rat)Potency1.584910
sq 22536Rattus norvegicus (Norway rat)Potency4.152720
ACar 18-0Rattus norvegicus (Norway rat)Potency0.398110
succinylcholineRattus norvegicus (Norway rat)Potency1.584910
sulfadimethoxineRattus norvegicus (Norway rat)Potency5.011910
sulfaphenazoleRattus norvegicus (Norway rat)Potency100.000010
sulmazoleRattus norvegicus (Norway rat)Potency79.432810
sulpirideRattus norvegicus (Norway rat)Potency0.562310
gatifloxacinRattus norvegicus (Norway rat)Potency56.234110
1,4-bis(2-(3,5-dichloropyridyloxy))benzeneRattus norvegicus (Norway rat)Potency18.122210
tegafurRattus norvegicus (Norway rat)Potency89.125110
telenzepineRattus norvegicus (Norway rat)Potency0.067020
terazosinRattus norvegicus (Norway rat)Potency40.868630
terbutalineRattus norvegicus (Norway rat)Potency0.223910
tetraethylammoniumRattus norvegicus (Norway rat)Potency37.685820
tetrahydrozolineRattus norvegicus (Norway rat)Potency14.125410
thiotepaRattus norvegicus (Norway rat)Potency89.125110
tolazamideRattus norvegicus (Norway rat)Potency47.775510
ici 136,753Rattus norvegicus (Norway rat)Potency22.807520
trazodoneRattus norvegicus (Norway rat)Potency24.702820
triamtereneRattus norvegicus (Norway rat)Potency30.405640
trimipramineRattus norvegicus (Norway rat)Potency0.398110
tropicamideRattus norvegicus (Norway rat)Potency0.112210
tulobuterolRattus norvegicus (Norway rat)Potency0.538920
tyrphostin a9Rattus norvegicus (Norway rat)Potency29.102140
u 101958Rattus norvegicus (Norway rat)Potency30.300120
u 99194Rattus norvegicus (Norway rat)Potency0.400820
urapidilRattus norvegicus (Norway rat)Potency19.093520
5-methylurapidilRattus norvegicus (Norway rat)Potency0.354810
venlafaxineRattus norvegicus (Norway rat)Potency1.778310
vesamicolRattus norvegicus (Norway rat)Potency3.048820
vigabatrinRattus norvegicus (Norway rat)Potency0.631010
n-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-n-(2-pyridinyl)cyclohexanecarboxamideRattus norvegicus (Norway rat)Potency4.533920
8-(4-((2-aminoethyl)aminocarbonylmethyloxy)phenyl)-1,3-dipropylxanthineRattus norvegicus (Norway rat)Potency20.268530
xylometazolineRattus norvegicus (Norway rat)Potency5.974330
3-(5'-hydroxymethyl-2'-furyl)-1-benzylindazoleRattus norvegicus (Norway rat)Potency27.141440
corticosteroneRattus norvegicus (Norway rat)Potency39.810710
reserpineRattus norvegicus (Norway rat)Potency32.310510
isoproterenol hydrochlorideRattus norvegicus (Norway rat)Potency45.599510
4-[(1S)-1-hydroxy-2-(propan-2-ylamino)ethyl]benzene-1,2-diolRattus norvegicus (Norway rat)Potency6.884320
thyroxineRattus norvegicus (Norway rat)Potency89.125110
pentolinium tartrateRattus norvegicus (Norway rat)Potency0.262020
promazine hydrochlorideRattus norvegicus (Norway rat)Potency42.284110
pilocarpineRattus norvegicus (Norway rat)Potency0.827220
pentylenetetrazoleRattus norvegicus (Norway rat)Potency14.125410
racepinephrine hydrochlorideRattus norvegicus (Norway rat)Potency17.852610
(4-(m-chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium chlorideRattus norvegicus (Norway rat)Potency13.893410
methyldimethylaminoazobenzeneRattus norvegicus (Norway rat)Potency89.125110
hexamethonium bromideRattus norvegicus (Norway rat)Potency0.047410
cystamine dihydrochlorideRattus norvegicus (Norway rat)Potency3.358710
tetraethylammonium chlorideRattus norvegicus (Norway rat)Potency37.685810
glutamineRattus norvegicus (Norway rat)Potency1.778310
vincristineRattus norvegicus (Norway rat)Potency79.432810
physostigmineRattus norvegicus (Norway rat)Potency29.934910
aminopyrineRattus norvegicus (Norway rat)Potency100.000010
methyltestosteroneRattus norvegicus (Norway rat)Potency70.794610
promethazine hydrochlorideRattus norvegicus (Norway rat)Potency11.917310
pyridoxine hydrochlorideRattus norvegicus (Norway rat)Potency50.118710
cephalothinRattus norvegicus (Norway rat)Potency44.668410
phenylephrineRattus norvegicus (Norway rat)Potency1.122010
levodopaRattus norvegicus (Norway rat)Potency29.934920
cysteamineRattus norvegicus (Norway rat)Potency12.534140
methoxamineRattus norvegicus (Norway rat)Potency4.572420
n-methyltryptamineRattus norvegicus (Norway rat)Potency56.234110
berlitionRattus norvegicus (Norway rat)Potency45.008210
ethyl methanesulfonateRattus norvegicus (Norway rat)Potency100.000010
dimethylnitrosamineRattus norvegicus (Norway rat)Potency100.000010
colchicineRattus norvegicus (Norway rat)Potency10.272130
quinacrine monohydrochlorideRattus norvegicus (Norway rat)Potency23.778110
chlorpromazine hydrochlorideRattus norvegicus (Norway rat)Potency26.679510
cytarabine hydrochlorideRattus norvegicus (Norway rat)Potency1.191710
cytarabineRattus norvegicus (Norway rat)Potency0.891310
trifluridineRattus norvegicus (Norway rat)Potency100.000010
perthaneRattus norvegicus (Norway rat)Potency89.125110
tryptophanRattus norvegicus (Norway rat)Potency30.710920
quinethazoneRattus norvegicus (Norway rat)Potency79.432810
arginineRattus norvegicus (Norway rat)Potency0.281810
dehydrocholic acidRattus norvegicus (Norway rat)Potency70.794610
rotenoneRattus norvegicus (Norway rat)Potency21.192310
skimmianineRattus norvegicus (Norway rat)Potency56.234110
9,10-phenanthrenequinoneRattus norvegicus (Norway rat)Potency6.581220
brompheniramineRattus norvegicus (Norway rat)Potency0.100010
7-amino-4-hydroxy-2-naphthalenesulfonic acidRattus norvegicus (Norway rat)Potency50.910020
Ethyl 2-aminobenzoateRattus norvegicus (Norway rat)Potency28.183810
anthranilamideRattus norvegicus (Norway rat)Potency79.432810
1-naphthylphenylamineRattus norvegicus (Norway rat)Potency25.118910
quinoxalinesRattus norvegicus (Norway rat)Potency3.162310
uvitex swnRattus norvegicus (Norway rat)Potency79.432810
2-naphthylamineRattus norvegicus (Norway rat)Potency56.234110
dehydrothio-4-toluidineRattus norvegicus (Norway rat)Potency29.903320
synephrineRattus norvegicus (Norway rat)Potency34.023920
3,4-xylidineRattus norvegicus (Norway rat)Potency100.000010
3,4-dichlorophenolRattus norvegicus (Norway rat)Potency89.125110
2-amino-4-methylphenolRattus norvegicus (Norway rat)Potency44.668410
p-tert-butyl catecholRattus norvegicus (Norway rat)Potency22.387210
alpha-methylstyrolRattus norvegicus (Norway rat)Potency89.125110
3-dimethylaminophenolRattus norvegicus (Norway rat)Potency100.000010
n-isopropyl-n-phenyl-4-phenylenediamineRattus norvegicus (Norway rat)Potency50.118710
n-oxydiethylene-2-benzothiazole sulfenamideRattus norvegicus (Norway rat)Potency12.589310
cyclohexanoneRattus norvegicus (Norway rat)Potency100.000010
methylergonovineRattus norvegicus (Norway rat)Potency14.412740
imipramine hydrochlorideRattus norvegicus (Norway rat)Potency26.679510
diphenylacetic acidRattus norvegicus (Norway rat)Potency89.125120
dithiodibenzoic acidRattus norvegicus (Norway rat)Potency3.548110
sulfan blueRattus norvegicus (Norway rat)Potency44.668410
suramin sodiumRattus norvegicus (Norway rat)Potency9.466210
pyrazolanthroneRattus norvegicus (Norway rat)Potency38.449420
diatrizoate meglumineRattus norvegicus (Norway rat)Potency56.234110
3-amino-9-ethylcarbazoleRattus norvegicus (Norway rat)Potency56.234110
2-Phenylethyl 2-aminobenzoateRattus norvegicus (Norway rat)Potency84.279020
amibenRattus norvegicus (Norway rat)Potency89.125110
neozoneRattus norvegicus (Norway rat)Potency28.187720
2-aminobenzothiazoleRattus norvegicus (Norway rat)Potency0.707910
chelidamic acidRattus norvegicus (Norway rat)Potency51.774010
4-nitrosodimethylanilineRattus norvegicus (Norway rat)Potency42.222420
4'-(chloroacetyl)acetanilideRattus norvegicus (Norway rat)Potency70.794610
diphenhydramine hydrochlorideRattus norvegicus (Norway rat)Potency89.125110
1,2-dihydro-2,2,4-trimethylquinolineRattus norvegicus (Norway rat)Potency79.432810
catechinRattus norvegicus (Norway rat)Potency40.070410
cysteamine hydrochlorideRattus norvegicus (Norway rat)Potency50.312610
benzo(e)pyreneRattus norvegicus (Norway rat)Potency21.679420
fluorantheneRattus norvegicus (Norway rat)Potency35.481310
benz(c)acridineRattus norvegicus (Norway rat)Potency22.387210
phenanthridineRattus norvegicus (Norway rat)Potency100.000010
acridinesRattus norvegicus (Norway rat)Potency79.432810
phenoxathiinRattus norvegicus (Norway rat)Potency89.125110
propantheline bromideRattus norvegicus (Norway rat)Potency0.794310
diiodotyrosineRattus norvegicus (Norway rat)Potency41.692010
muscarineRattus norvegicus (Norway rat)Potency23.778110
norchlorcyclizineRattus norvegicus (Norway rat)Potency15.848910
3-phenylsalicylic acidRattus norvegicus (Norway rat)Potency39.810710
2,3-dimercaptosuccinic acidRattus norvegicus (Norway rat)Potency28.183810
ethamivanRattus norvegicus (Norway rat)Potency0.766210
opipramolRattus norvegicus (Norway rat)Potency5.834930
aminophyllineRattus norvegicus (Norway rat)Potency1.683410
orphenadrine hydrochlorideRattus norvegicus (Norway rat)Potency1.337110
methysergideRattus norvegicus (Norway rat)Potency11.605320
cyproterone acetateRattus norvegicus (Norway rat)Potency57.902310
nandroloneRattus norvegicus (Norway rat)Potency89.125110
2-aminopurineRattus norvegicus (Norway rat)Potency15.848910
boldineRattus norvegicus (Norway rat)Potency17.782810
emetineRattus norvegicus (Norway rat)Potency3.548110
bicucullineRattus norvegicus (Norway rat)Potency70.794610
kainic acidRattus norvegicus (Norway rat)Potency0.354810
methyl redRattus norvegicus (Norway rat)Potency50.118710
3,4-toluenediamineRattus norvegicus (Norway rat)Potency100.000010
dihydroergotamineRattus norvegicus (Norway rat)Potency4.228420
hematoxylinRattus norvegicus (Norway rat)Potency10.750910
luminolRattus norvegicus (Norway rat)Potency44.668410
herniarinRattus norvegicus (Norway rat)Potency50.118710
methoxyhydroxyphenylglycolRattus norvegicus (Norway rat)Potency9.466220
nitrophenideRattus norvegicus (Norway rat)Potency39.810710
decamethonium dibromideRattus norvegicus (Norway rat)Potency22.387210
maleimideRattus norvegicus (Norway rat)Potency1.995310
aniline mustardRattus norvegicus (Norway rat)Potency44.668410
carbamylhydrazine monohydrochlorideRattus norvegicus (Norway rat)Potency10.621310
betaine hydrochlorideRattus norvegicus (Norway rat)Potency26.679510
3-aminophenolRattus norvegicus (Norway rat)Potency10.000010
pentabromophenolRattus norvegicus (Norway rat)Potency31.622810
apocodeineRattus norvegicus (Norway rat)Potency39.810710
2-phenylbenzimidazoleRattus norvegicus (Norway rat)Potency56.234110
phosmetRattus norvegicus (Norway rat)Potency35.481310
diphenyl disulfideRattus norvegicus (Norway rat)Potency50.118710
isopropylmethanesulfonateRattus norvegicus (Norway rat)Potency100.000010
5-aminobenzimidazoleRattus norvegicus (Norway rat)Potency2.818410
2-phenylindoleRattus norvegicus (Norway rat)Potency56.234110
estradiol valerateRattus norvegicus (Norway rat)Potency79.432810
c 137Rattus norvegicus (Norway rat)Potency89.125110
2,2'-diaminodiphenyldisulfideRattus norvegicus (Norway rat)Potency10.000010
n-acetylmelphalanRattus norvegicus (Norway rat)Potency31.622810
2-amino-4-phenylphenolRattus norvegicus (Norway rat)Potency79.432810
dehydroepiandrosterone acetateRattus norvegicus (Norway rat)Potency89.125110
carmineRattus norvegicus (Norway rat)Potency50.118710
lysergolRattus norvegicus (Norway rat)Potency18.738320
tetrachloroisophthalonitrileRattus norvegicus (Norway rat)Potency0.281810
amiloride hydrochloride, anhydrousRattus norvegicus (Norway rat)Potency79.432810
amilorideRattus norvegicus (Norway rat)Potency19.571020
2-methoxy-1,4-naphthoquinoneRattus norvegicus (Norway rat)Potency39.810710
1-methylpyreneRattus norvegicus (Norway rat)Potency79.432810
ethyl violetRattus norvegicus (Norway rat)Potency17.782810
dexbrompheniramineRattus norvegicus (Norway rat)Potency0.316210
1,2-benzisothiazoline-3-oneRattus norvegicus (Norway rat)Potency28.183810
6-chrysenamineRattus norvegicus (Norway rat)Potency19.952610
1,2-diphenyl-3,5-pyrazolidinedioneRattus norvegicus (Norway rat)Potency25.118910
2-amino-3-chloro-1,4-naphthoquinoneRattus norvegicus (Norway rat)Potency12.589310
4-amino-2-hydroxytolueneRattus norvegicus (Norway rat)Potency19.952610
dibromoacetonitrileRattus norvegicus (Norway rat)Potency79.432810
n-(4-dimethylamino-3,5-dinitrophenyl)maleimideRattus norvegicus (Norway rat)Potency2.818410
phenoxyacetic acidRattus norvegicus (Norway rat)Potency100.000010
nitroxolineRattus norvegicus (Norway rat)Potency75.113720
Bis(2-furanylmethyl) disulfideRattus norvegicus (Norway rat)Potency39.810710
acetylthiocholineRattus norvegicus (Norway rat)Potency12.589310
methylglutaronitrileRattus norvegicus (Norway rat)Potency100.000010
1,6-bismaleimidohexaneRattus norvegicus (Norway rat)Potency0.707910
1-methyl-5-chloro-4-nitroimidazoleRattus norvegicus (Norway rat)Potency28.183810
trimetazidineRattus norvegicus (Norway rat)Potency44.668410
mexiletine hydrochlorideRattus norvegicus (Norway rat)Potency89.125110
beclomethasone dipropionateRattus norvegicus (Norway rat)Potency79.432810
vidarabineRattus norvegicus (Norway rat)Potency89.125110
octocryleneRattus norvegicus (Norway rat)Potency56.234110
6,7-Dimethoxy-1-methyl-3,4-dihydroisoquinolineRattus norvegicus (Norway rat)Potency26.651420
helenalinRattus norvegicus (Norway rat)Potency56.234110
ormetoprimRattus norvegicus (Norway rat)Potency79.432810
levodopa methyl esterRattus norvegicus (Norway rat)Potency21.252540
isoetharine mesylateRattus norvegicus (Norway rat)Potency54.683810
molindoneRattus norvegicus (Norway rat)Potency20.577620
zalcitabineRattus norvegicus (Norway rat)Potency10.455830
2-Propenyl 2-aminobenzoateRattus norvegicus (Norway rat)Potency22.387210
propionylpromazine hydrochlorideRattus norvegicus (Norway rat)Potency1.000010
propionylpromazineRattus norvegicus (Norway rat)Potency7.519310
camptothecinRattus norvegicus (Norway rat)Potency10.432540
hydroxyzine pamoateRattus norvegicus (Norway rat)Potency79.432810
n-methylisatoic anhydrideRattus norvegicus (Norway rat)Potency40.676520
pyrazophosRattus norvegicus (Norway rat)Potency0.100010
apazoneRattus norvegicus (Norway rat)Potency70.794610
marmesin, (r)-isomerRattus norvegicus (Norway rat)Potency79.432810
salenRattus norvegicus (Norway rat)Potency0.100010
levamisoleRattus norvegicus (Norway rat)Potency0.631010
benserazide hydrochlorideRattus norvegicus (Norway rat)Potency12.980410
tetridaminRattus norvegicus (Norway rat)Potency89.125110
metizolineRattus norvegicus (Norway rat)Potency28.425830
metergolineRattus norvegicus (Norway rat)Potency33.245120
1-(trimethylsilyl)-1h-imidazoleRattus norvegicus (Norway rat)Potency100.000010
bromocriptineRattus norvegicus (Norway rat)Potency19.952610
triamcinoloneRattus norvegicus (Norway rat)Potency29.760720
butylated hydroxytolueneRattus norvegicus (Norway rat)Potency35.481310
benzonidazoleRattus norvegicus (Norway rat)Potency79.432810
dihydro-beta-erythroidineRattus norvegicus (Norway rat)Potency15.467420
glutamic acidRattus norvegicus (Norway rat)Potency7.079510
cefazolinRattus norvegicus (Norway rat)Potency50.118710
2-n-octyl-4-isothiazolin-3-oneRattus norvegicus (Norway rat)Potency31.622810
timololRattus norvegicus (Norway rat)Potency1.412510
carbidopaRattus norvegicus (Norway rat)Potency19.813510
proroxan hydrochlorideRattus norvegicus (Norway rat)Potency0.281810
propafenone hydrochlorideRattus norvegicus (Norway rat)Potency8.436810
dobutamineRattus norvegicus (Norway rat)Potency14.125410
butaclamolRattus norvegicus (Norway rat)Potency7.519310
10-carboxymethyl-9-acridanoneRattus norvegicus (Norway rat)Potency67.833420
methyldopaRattus norvegicus (Norway rat)Potency10.438420
bezafibrateRattus norvegicus (Norway rat)Potency28.990020
diltiazemRattus norvegicus (Norway rat)Potency4.744420
nimustineRattus norvegicus (Norway rat)Potency14.445820
lonidamineRattus norvegicus (Norway rat)Potency0.446710
ng-nitroarginine methyl esterRattus norvegicus (Norway rat)Potency0.501210
albuterol sulfateRattus norvegicus (Norway rat)Potency0.532310
quisqualic acidRattus norvegicus (Norway rat)Potency2.150830
pirfenidoneRattus norvegicus (Norway rat)Potency7.629330
idarubicinRattus norvegicus (Norway rat)Potency26.679520
terazosin hydrochloride anhydrousRattus norvegicus (Norway rat)Potency66.225420
chlorsulfuronRattus norvegicus (Norway rat)Potency89.125110
cefaclor anhydrousRattus norvegicus (Norway rat)Potency50.118710
alo 2145Rattus norvegicus (Norway rat)Potency33.587510
flupirtineRattus norvegicus (Norway rat)Potency31.448630
idazoxanRattus norvegicus (Norway rat)Potency7.519320
quinpiroleRattus norvegicus (Norway rat)Potency2.484010
raloxifene hydrochlorideRattus norvegicus (Norway rat)Potency55.158710
mifepristoneRattus norvegicus (Norway rat)Potency12.380720
imazodanRattus norvegicus (Norway rat)Potency13.693710
salmeterol xinafoateRattus norvegicus (Norway rat)Potency17.220620
ranolazineRattus norvegicus (Norway rat)Potency0.946620
quineloraneRattus norvegicus (Norway rat)Potency13.005120
orbifloxacinRattus norvegicus (Norway rat)Potency44.668410
mibefradilRattus norvegicus (Norway rat)Potency0.428020
eliprodilRattus norvegicus (Norway rat)Potency0.751910
duloxetineRattus norvegicus (Norway rat)Potency50.118710
irinotecanRattus norvegicus (Norway rat)Potency35.490620
aptiganel hydrochlorideRattus norvegicus (Norway rat)Potency0.053210
3-iodobenzylguanidineRattus norvegicus (Norway rat)Potency8.912510
2-Amino-5-(5-nitro-2-furyl)-1,3,4-thiadiazoleRattus norvegicus (Norway rat)Potency1.122010
5-AminoacenaphtheneRattus norvegicus (Norway rat)Potency19.952610
ici 63197Rattus norvegicus (Norway rat)Potency26.059840
paroxetine hydrochlorideRattus norvegicus (Norway rat)Potency89.125110
trazodone hydrochlorideRattus norvegicus (Norway rat)Potency70.012820
verapamil hydrochlorideRattus norvegicus (Norway rat)Potency17.782810
doxazosin mesylateRattus norvegicus (Norway rat)Potency56.451620
terfenadineRattus norvegicus (Norway rat)Potency89.125110
src-820 rRattus norvegicus (Norway rat)Potency0.089110
nelfinavir mesylateRattus norvegicus (Norway rat)Potency63.095710
n(4)-acetylsulfadiazineRattus norvegicus (Norway rat)Potency0.398110
norharmanRattus norvegicus (Norway rat)Potency79.432810
desipramine hydrochlorideRattus norvegicus (Norway rat)Potency3.358710
dopamine hydrochlorideRattus norvegicus (Norway rat)Potency16.833610
4-nitrobenzylthioinosineRattus norvegicus (Norway rat)Potency33.587510
rutecarpineRattus norvegicus (Norway rat)Potency32.643120
telmisartanRattus norvegicus (Norway rat)Potency79.432810
thioridazine hydrochlorideRattus norvegicus (Norway rat)Potency22.387210
trifluoperazine hydrochlorideRattus norvegicus (Norway rat)Potency15.848910
siquilRattus norvegicus (Norway rat)Potency37.685810
alprenolol hydrochlorideRattus norvegicus (Norway rat)Potency0.056210
2-methoxyestradiolRattus norvegicus (Norway rat)Potency22.779820
toxoflavinRattus norvegicus (Norway rat)Potency48.022420
pyrrolo(1,2-a)quinoxalineRattus norvegicus (Norway rat)Potency33.552020
7-(trifluoromethyl)-1H-quinolin-4-oneRattus norvegicus (Norway rat)Potency44.668410
harmolRattus norvegicus (Norway rat)Potency32.464820
dimidium bromideRattus norvegicus (Norway rat)Potency89.125110
2,6-dimethoxy-1,4-benzoquinoneRattus norvegicus (Norway rat)Potency31.622810
dyclonine hydrochlorideRattus norvegicus (Norway rat)Potency3.162310
11h-pyrido(2,1-b)quinazolin-11-oneRattus norvegicus (Norway rat)Potency31.622810
clomipramine hydrochlorideRattus norvegicus (Norway rat)Potency89.125110
prazosin hydrochlorideRattus norvegicus (Norway rat)Potency67.833420
mianserin hydrochlorideRattus norvegicus (Norway rat)Potency37.685810
econazole nitrateRattus norvegicus (Norway rat)Potency25.118910
lomefloxacin hydrochlorideRattus norvegicus (Norway rat)Potency44.668410
sanguinarine chlorideRattus norvegicus (Norway rat)Potency79.432810
plasmenylserineRattus norvegicus (Norway rat)Potency0.398110
cefaloramRattus norvegicus (Norway rat)Potency12.589310
n-(2-carboxyphenyl)glycineRattus norvegicus (Norway rat)Potency79.432810
5,6-benzocoumarin-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency46.682720
n-acetyltryptamineRattus norvegicus (Norway rat)Potency0.188910
spirodecanoneRattus norvegicus (Norway rat)Potency63.095710
propipocaine monohydrochlorideRattus norvegicus (Norway rat)Potency50.118710
2-MethoxyxanthoneRattus norvegicus (Norway rat)Potency56.234110
D-serineRattus norvegicus (Norway rat)Potency0.354820
masoprocolRattus norvegicus (Norway rat)Potency17.780620
pirenzepine dihydrochlorideRattus norvegicus (Norway rat)Potency1.122010
labetalol hydrochlorideRattus norvegicus (Norway rat)Potency67.833420
loperamide hydrochlorideRattus norvegicus (Norway rat)Potency0.751910
opipramol hydrochlorideRattus norvegicus (Norway rat)Potency0.422810
thioxoloneRattus norvegicus (Norway rat)Potency100.000010
3-octadecanamido-2-ethoxypropylphosphocholineRattus norvegicus (Norway rat)Potency13.223010
sesaminRattus norvegicus (Norway rat)Potency89.125110
chelerythrine chlorideRattus norvegicus (Norway rat)Potency18.887610
carbobenzoxyvalylphenylalanine aldehydeRattus norvegicus (Norway rat)Potency0.501210
methyl 3-aminopyrazine-2-carboxylateRattus norvegicus (Norway rat)Potency0.756320
9-hydroxyphenylfluoronRattus norvegicus (Norway rat)Potency10.000010
3-aminophenoxazoneRattus norvegicus (Norway rat)Potency56.234110
2-phenyl-4,5-dichloro-3-pyridazinoneRattus norvegicus (Norway rat)Potency14.125410
3-methylbenzotriazin-4-oneRattus norvegicus (Norway rat)Potency89.125110
tetrandrineRattus norvegicus (Norway rat)Potency35.481310
tosyllysine chloromethyl ketoneRattus norvegicus (Norway rat)Potency43.084510
tosyllysine chloromethyl ketoneRattus norvegicus (Norway rat)Potency25.955330
nodakeninRattus norvegicus (Norway rat)Potency79.432810
amperozideRattus norvegicus (Norway rat)Potency37.685820
EvoxineRattus norvegicus (Norway rat)Potency60.456620
ergocornineRattus norvegicus (Norway rat)Potency52.487020
agroclavineRattus norvegicus (Norway rat)Potency3.628220
n-benzylmaleimideRattus norvegicus (Norway rat)Potency0.398110
habaRattus norvegicus (Norway rat)Potency89.125110
6-hydroxy-2-phenylpyridazin-3-oneRattus norvegicus (Norway rat)Potency39.810710
1-benzyl-1h-indazol-3-olRattus norvegicus (Norway rat)Potency56.234110
1-hydroxybenzotriazoleRattus norvegicus (Norway rat)Potency89.125110
bis(phenylsulfonyl)methaneRattus norvegicus (Norway rat)Potency11.220210
4'-methoxyflavoneRattus norvegicus (Norway rat)Potency20.386620
2-aminopyrazineRattus norvegicus (Norway rat)Potency63.095710
5-amino-1-phenyl-1H-pyrazole-4-carbonitrileRattus norvegicus (Norway rat)Potency39.810710
n-benzyl-4-toluidineRattus norvegicus (Norway rat)Potency5.011910
8-methyl-4-oxo-3-pyrido[1,2-a]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency75.113720
2-(1H-benzimidazol-2-yl)anilineRattus norvegicus (Norway rat)Potency31.225620
1-(2-phenanthrenyl)ethanoneRattus norvegicus (Norway rat)Potency25.118910
5-phenoxysulfonyl-1-methyl-4-nitroimidazoleRattus norvegicus (Norway rat)Potency0.316210
n,n'-2-phenylenedimaleimideRattus norvegicus (Norway rat)Potency0.316210
4-methylumbelliferyl butyrateRattus norvegicus (Norway rat)Potency37.618820
6-methoxy-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-oneRattus norvegicus (Norway rat)Potency29.903320
5-aminoindazoleRattus norvegicus (Norway rat)Potency79.432810
7-(diethylamino)-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency28.183810
methionine sulfoximineRattus norvegicus (Norway rat)Potency0.562310
nicotineRattus norvegicus (Norway rat)Potency44.668410
sennoside BRattus norvegicus (Norway rat)Potency11.220210
mephentermineRattus norvegicus (Norway rat)Potency100.000010
gliquidoneRattus norvegicus (Norway rat)Potency79.432810
fluazinamRattus norvegicus (Norway rat)Potency25.118910
L-2-aminoadipic acidRattus norvegicus (Norway rat)Potency0.100010
columbianetin, (s)-isomerRattus norvegicus (Norway rat)Potency25.285520
D-dopaRattus norvegicus (Norway rat)Potency26.679510
7-amino-4-methylcoumarinRattus norvegicus (Norway rat)Potency51.453220
n-(4,4-diphenyl-3-butenyl)nipecotic acidRattus norvegicus (Norway rat)Potency39.810710
1-(4'-nitrophenyl)-2-aminopropane-1,3-diolRattus norvegicus (Norway rat)Potency89.125120
methylene bis(methylanthranilate)Rattus norvegicus (Norway rat)Potency22.387210
1-piperonylpiperazineRattus norvegicus (Norway rat)Potency79.432810
3-(n-salicyloyl)amino-1,2,4-triazoleRattus norvegicus (Norway rat)Potency56.234110
ska-31Rattus norvegicus (Norway rat)Potency89.125110
2-methyl-4-methoxymethyl-5-cyano-6-oxypyridineRattus norvegicus (Norway rat)Potency22.387210
4,5-diphenyl-1,5-dihydroimidazol-2-oneRattus norvegicus (Norway rat)Potency45.857720
6-(4-nitrobenzylthio)guanosineRattus norvegicus (Norway rat)Potency42.284120
2-(4-hydroxyphenyl)-5,6,7,8-tetrahydroxy-4H-1-benzopyran-4-oneRattus norvegicus (Norway rat)Potency15.848910
3,5,7,3',4'-pentamethoxyflavoneRattus norvegicus (Norway rat)Potency56.234110
3-aminopropylphosphonic acidRattus norvegicus (Norway rat)Potency5.323310
1-(1,2-dihydroacenaphthylen-5-yl)ethanoneRattus norvegicus (Norway rat)Potency56.234110
3,3'-DihydroxyhexestrolRattus norvegicus (Norway rat)Potency7.943310
5-benzyloxytryptophanRattus norvegicus (Norway rat)Potency79.432810
4-hydroxyantipyrineRattus norvegicus (Norway rat)Potency70.794610
6,6'-methylene bis(2,2,4-trimethyl-1,2-dihydroquinoline)Rattus norvegicus (Norway rat)Potency17.782810
9-methoxyacridineRattus norvegicus (Norway rat)Potency84.279020
3,7-dimethyl-1-propargylxanthineRattus norvegicus (Norway rat)Potency0.597310
zpckRattus norvegicus (Norway rat)Potency26.751420
2-(4-pyridyl)thiazolidine-4-carboxylic acidRattus norvegicus (Norway rat)Potency50.118710
diphyllinRattus norvegicus (Norway rat)Potency12.589310
jjc 323Rattus norvegicus (Norway rat)Potency8.912510
n-acetyldopamineRattus norvegicus (Norway rat)Potency26.679510
7-amino-4-trifluoromethylcoumarinRattus norvegicus (Norway rat)Potency56.234110
7,9-dimethyl-9aH-quinolizine-1,2,3,4-tetracarboxylic acid tetramethyl esterRattus norvegicus (Norway rat)Potency62.050620
n(6)-phenyladenosineRattus norvegicus (Norway rat)Potency0.501210
moxifloxacin hydrochlorideRattus norvegicus (Norway rat)Potency50.118710
lobelineRattus norvegicus (Norway rat)Potency0.631010
n-methyladenosineRattus norvegicus (Norway rat)Potency0.571220
fulvestrantRattus norvegicus (Norway rat)Potency13.371420
alphaxaloneRattus norvegicus (Norway rat)Potency0.631010
bicuculline methochlorideRattus norvegicus (Norway rat)Potency8.436820
cp-55,940Rattus norvegicus (Norway rat)Potency36.013130
chlorethylclonidineRattus norvegicus (Norway rat)Potency25.255220
methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylateRattus norvegicus (Norway rat)Potency44.668410
cv 3988Rattus norvegicus (Norway rat)Potency9.290930
beta-carboline-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency50.118710
dihydroergocristineRattus norvegicus (Norway rat)Potency0.026720
6-hydroxydopaRattus norvegicus (Norway rat)Potency27.644820
gamma-fagarineRattus norvegicus (Norway rat)Potency22.387210
cl 218872Rattus norvegicus (Norway rat)Potency89.125110
betaxolol hydrochlorideRattus norvegicus (Norway rat)Potency0.125910
1-(2-methoxyphenyl)-4-(4-(2-phthalimido)butyl)piperazineRattus norvegicus (Norway rat)Potency29.934910
s-methylthiocitrullineRattus norvegicus (Norway rat)Potency2.238710
dihydrocapsaicinRattus norvegicus (Norway rat)Potency41.352920
ml 9Rattus norvegicus (Norway rat)Potency2.377810
sphondinRattus norvegicus (Norway rat)Potency56.234110
benzamilRattus norvegicus (Norway rat)Potency22.387210
sch 28080Rattus norvegicus (Norway rat)Potency37.685810
tanshinoneRattus norvegicus (Norway rat)Potency39.810710
1-(carboxymethylthio)tetradecaneRattus norvegicus (Norway rat)Potency23.778120
olprinoneRattus norvegicus (Norway rat)Potency13.371410
3-(1-piperidinyl)-1-(4-propan-2-yloxyphenyl)-1-propanoneRattus norvegicus (Norway rat)Potency0.707910
2-methyl-4-isothiazolin-3-one hydrochlorideRattus norvegicus (Norway rat)Potency56.234110
n-(phenylthio)-epsilon-caprolactamRattus norvegicus (Norway rat)Potency0.281810
pefloxacin mesylateRattus norvegicus (Norway rat)Potency89.125110
buthionine sulfoximineRattus norvegicus (Norway rat)Potency33.587510
sm 1213Rattus norvegicus (Norway rat)Potency1.778310
uh 301Rattus norvegicus (Norway rat)Potency0.354810
san 58035Rattus norvegicus (Norway rat)Potency0.316210
a 68930Rattus norvegicus (Norway rat)Potency11.220210
pd 128042Rattus norvegicus (Norway rat)Potency26.770020
tetradecanoylphorbol acetateRattus norvegicus (Norway rat)Potency17.453530
imatinib mesylateRattus norvegicus (Norway rat)Potency0.281810
mk 912Rattus norvegicus (Norway rat)Potency0.842820
1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidineRattus norvegicus (Norway rat)Potency0.562310
nnc 711Rattus norvegicus (Norway rat)Potency0.891310
n,n-dimethylarginineRattus norvegicus (Norway rat)Potency1.122010
sk&f 86466Rattus norvegicus (Norway rat)Potency0.446710
l 687384Rattus norvegicus (Norway rat)Potency0.005320
furamidineRattus norvegicus (Norway rat)Potency57.457020
2-phenyl-3-(n,n-dimethylaminopropyl)-1,3-thiazolidin-4-oneRattus norvegicus (Norway rat)Potency2.818410
methotrexateRattus norvegicus (Norway rat)Potency34.851530
sr 2640Rattus norvegicus (Norway rat)Potency0.067010
rufinamideRattus norvegicus (Norway rat)Potency0.867520
ici 204448Rattus norvegicus (Norway rat)Potency0.946610
sr 57227aRattus norvegicus (Norway rat)Potency0.446710
n,n-di-n-hexyl-2-(4-fluorophenyl)indole-3-acetamideRattus norvegicus (Norway rat)Potency36.576440
4-(benzodioxan-5-yl)-1-(indan-2-yl)piperazineRattus norvegicus (Norway rat)Potency0.251210
3,5-bis(trifluoromethyl)benzyl n-acetyltryptophanRattus norvegicus (Norway rat)Potency39.810710
omega-n-methylarginineRattus norvegicus (Norway rat)Potency1.412510
sk&f 83959Rattus norvegicus (Norway rat)Potency0.354810
alpha-ergocryptineRattus norvegicus (Norway rat)Potency30.258620
n-(3,5-dimethyl-4-isoxazolylmethyl)phthalimideRattus norvegicus (Norway rat)Potency15.848910
tilarginine acetateRattus norvegicus (Norway rat)Potency79.432810
alpha-guanidinoglutaric acidRattus norvegicus (Norway rat)Potency0.631010
N-(1,3-dioxo-4-isoindolyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
imidazole-4-acetic acid hydrochlorideRattus norvegicus (Norway rat)Potency0.532310
isodibutRattus norvegicus (Norway rat)Potency25.118910
1-(1,3-benzodioxol-5-yl)-3-(1-piperidinyl)-1-propanoneRattus norvegicus (Norway rat)Potency0.316210
sk&f-38393Rattus norvegicus (Norway rat)Potency15.003010
nsc-141549Rattus norvegicus (Norway rat)Potency62.050620
levofloxacinRattus norvegicus (Norway rat)Potency56.234110
dichloro-1,2-diaminocyclohexane platinum complexRattus norvegicus (Norway rat)Potency0.316210
sandoz-21-009Rattus norvegicus (Norway rat)Potency31.622810
2-phenylbenzotriazoleRattus norvegicus (Norway rat)Potency19.952610
idazoxan hydrochlorideRattus norvegicus (Norway rat)Potency53.176410
n,n-dipropylcarboxamidotryptamineRattus norvegicus (Norway rat)Potency7.079510
alpha-methylhistamineRattus norvegicus (Norway rat)Potency8.539820
tetrahydroharmineRattus norvegicus (Norway rat)Potency53.882020
oxidopamine hydrochlorideRattus norvegicus (Norway rat)Potency56.234110
cryptotanshinoneRattus norvegicus (Norway rat)Potency28.183810
cyc 202Rattus norvegicus (Norway rat)Potency0.037710
2-methyl-4-(phenylimino)naphth(2,3-d)oxazol-9-oneRattus norvegicus (Norway rat)Potency17.782810
Serotonin hydrochlorideRattus norvegicus (Norway rat)Potency0.150010
n-phthaloylglutamic acidRattus norvegicus (Norway rat)Potency28.642020
ag 3-5Rattus norvegicus (Norway rat)Potency16.833610
2,4-dinitropyrimidinyl-2-thiophenolRattus norvegicus (Norway rat)Potency31.622810
tanshinone ii aRattus norvegicus (Norway rat)Potency17.782810
enniatin bRattus norvegicus (Norway rat)Potency89.125120
2-phenyl-1,2-benzisothiazol-3-(2h)-oneRattus norvegicus (Norway rat)Potency14.125410
cystamine hydrochlorideRattus norvegicus (Norway rat)Potency79.432810
n-n-propylnorapomorphineRattus norvegicus (Norway rat)Potency19.824530
azepexole, dihydrochlorideRattus norvegicus (Norway rat)Potency9.466210
abt 980Rattus norvegicus (Norway rat)Potency63.095710
carboline-3-carboxylic acidRattus norvegicus (Norway rat)Potency63.120820
2,10,11-trihydroxy-n-n-propylnoraporphineRattus norvegicus (Norway rat)Potency13.371410
sk&f 75670Rattus norvegicus (Norway rat)Potency8.594220
esatenololRattus norvegicus (Norway rat)Potency0.398110
rufloxacin hydrochlorideRattus norvegicus (Norway rat)Potency19.952610
sb 216763Rattus norvegicus (Norway rat)Potency0.299310
sch 58261Rattus norvegicus (Norway rat)Potency5.715220
4-methoxy-1-vinylcarbolineRattus norvegicus (Norway rat)Potency39.810710
3-chloro-7-methoxy-4-methyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency36.253020
dizocilpineRattus norvegicus (Norway rat)Potency5.972820
memantine hydrochlorideRattus norvegicus (Norway rat)Potency15.832610
moracin mRattus norvegicus (Norway rat)Potency56.234110
pongidaeRattus norvegicus (Norway rat)Potency0.047410
phenserineRattus norvegicus (Norway rat)Potency1.258910
sb 205384Rattus norvegicus (Norway rat)Potency4.744410
4-(2-methyl-5-phenyl-1-pyrrolyl)benzoic acidRattus norvegicus (Norway rat)Potency70.794610
fonsecinRattus norvegicus (Norway rat)Potency89.125110
brazilinRattus norvegicus (Norway rat)Potency4.466810
cortisoneRattus norvegicus (Norway rat)Potency32.817720
equilinRattus norvegicus (Norway rat)Potency28.183810
nsc13345Rattus norvegicus (Norway rat)Potency11.220210
carbamothioic acid S-[2-(2-methoxyanilino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency12.589310
4,5-dimethoxy-2,3-dihydroinden-1-oneRattus norvegicus (Norway rat)Potency85.894320
vincaleukoblastineRattus norvegicus (Norway rat)Potency11.220210
PorfiromycineRattus norvegicus (Norway rat)Potency56.234110
2-hydroxyestradiolRattus norvegicus (Norway rat)Potency35.481310
6-methyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency21.712320
1,10-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,9-diolRattus norvegicus (Norway rat)Potency28.183810
anisomycinRattus norvegicus (Norway rat)Potency39.810710
n-methylserotonin oxalate saltRattus norvegicus (Norway rat)Potency0.335910
showdomycinRattus norvegicus (Norway rat)Potency7.079510
nsc 95397Rattus norvegicus (Norway rat)Potency24.539240
5-(2-naphthalenylmethylidene)-1,3-diazinane-2,4,6-trioneRattus norvegicus (Norway rat)Potency14.125410
2-chloro-3-(4-methylanilino)naphthalene-1,4-dioneRattus norvegicus (Norway rat)Potency3.548110
noscapineRattus norvegicus (Norway rat)Potency0.398110
dimethyl 2-(2-nitrobenzylidene)malonateRattus norvegicus (Norway rat)Potency56.234110
N-butyl-1H-benzimidazol-2-amineRattus norvegicus (Norway rat)Potency5.011910
2-(3-nitrophenyl)-3,1-benzoxazin-4-oneRattus norvegicus (Norway rat)Potency0.446710
2-(4-aminophenyl)quinolineRattus norvegicus (Norway rat)Potency35.481310
2-(2-oxolanylmethyl)benzo[de]isoquinoline-1,3-dioneRattus norvegicus (Norway rat)Potency25.118910
4-[(1-naphthalenylamino)-oxomethyl]benzene-1,3-dicarboxylic acidRattus norvegicus (Norway rat)Potency79.432820
nsc228155Rattus norvegicus (Norway rat)Potency1.584910
a-130aRattus norvegicus (Norway rat)Potency63.095710
hematoxylinRattus norvegicus (Norway rat)Potency10.000010
pifithrin muRattus norvegicus (Norway rat)Potency7.871430
(5-amino-3-triazolo[1,5-a]quinazolinyl)-(4-morpholinyl)methanoneRattus norvegicus (Norway rat)Potency6.309610
3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
7-methoxycoumarin-4-acetic acidRattus norvegicus (Norway rat)Potency70.794610
N-phenylcarbamic acid 2-phenoxyethyl esterRattus norvegicus (Norway rat)Potency100.000010
3-phenyl-1H-quinoxalin-2-oneRattus norvegicus (Norway rat)Potency39.810710
5-[(4-chlorophenyl)methylthio]-1,3,4-thiadiazol-2-amineRattus norvegicus (Norway rat)Potency10.000010
nsc606985Rattus norvegicus (Norway rat)Potency31.832620
DubamineRattus norvegicus (Norway rat)Potency31.622810
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneRattus norvegicus (Norway rat)Potency0.158510
1-methyl-3-phenylpyrazino[1,2-a]benzimidazoleRattus norvegicus (Norway rat)Potency56.234110
nsc 674495Rattus norvegicus (Norway rat)Potency3.162310
nsc681152Rattus norvegicus (Norway rat)Potency56.234110
5,7-dimethoxy-4-methyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency25.118910
7-methoxy-4-methyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency70.794610
nsc697923Rattus norvegicus (Norway rat)Potency0.354810
5f-203Rattus norvegicus (Norway rat)Potency3.162310
7-(4-methoxyphenyl)-5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency63.095710
1-methoxy-10H-acridin-9-oneRattus norvegicus (Norway rat)Potency84.279020
dichloro-1,2-diaminocyclohexane platinum complexRattus norvegicus (Norway rat)Potency0.251210
macbecin iiRattus norvegicus (Norway rat)Potency3.162310
canavanineRattus norvegicus (Norway rat)Potency1.584910
5-hydroxytryptophanRattus norvegicus (Norway rat)Potency27.691420
ouabainRattus norvegicus (Norway rat)Potency37.685810
tosylphenylalanyl chloromethyl ketoneRattus norvegicus (Norway rat)Potency42.984020
monoiodotyrosineRattus norvegicus (Norway rat)Potency9.560010
nitroarginineRattus norvegicus (Norway rat)Potency0.672410
mimosineRattus norvegicus (Norway rat)Potency0.357120
cortodoxoneRattus norvegicus (Norway rat)Potency42.284110
pancuroniumRattus norvegicus (Norway rat)Potency0.005310
decursinolRattus norvegicus (Norway rat)Potency56.234110
angustibalinRattus norvegicus (Norway rat)Potency56.234110
genipinRattus norvegicus (Norway rat)Potency29.934920
naringinRattus norvegicus (Norway rat)Potency79.432810
s-(4-azidophenacyl)glutathioneRattus norvegicus (Norway rat)Potency26.679510
n-formylmethionine leucyl-phenylalanineRattus norvegicus (Norway rat)Potency89.125110
hydroxylamine hydrochlorideRattus norvegicus (Norway rat)Potency0.597310
L-isoprenalineRattus norvegicus (Norway rat)Potency4.336120
3,5-dihydroxyphenylglycineRattus norvegicus (Norway rat)Potency1.258910
actinoninRattus norvegicus (Norway rat)Potency1.268510
vinpocetineRattus norvegicus (Norway rat)Potency6.309610
flumethasone pivalateRattus norvegicus (Norway rat)Potency100.000010
tretinoinRattus norvegicus (Norway rat)Potency23.962520
resveratrolRattus norvegicus (Norway rat)Potency20.517820
retinolRattus norvegicus (Norway rat)Potency50.118710
oleic acidRattus norvegicus (Norway rat)Potency89.125110
thapsigarginRattus norvegicus (Norway rat)Potency24.146640
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolRattus norvegicus (Norway rat)Potency39.467140
adenosine-5'-(n-ethylcarboxamide)Rattus norvegicus (Norway rat)Potency2.107620
L-cycloserineRattus norvegicus (Norway rat)Potency0.891310
visnadinRattus norvegicus (Norway rat)Potency28.183810
ketoconazoleRattus norvegicus (Norway rat)Potency23.778110
melphalanRattus norvegicus (Norway rat)Potency79.432810
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneRattus norvegicus (Norway rat)Potency42.800020
cefmetazole(1-)Rattus norvegicus (Norway rat)Potency23.935920
4-(2-oxazolo[4,5-b]pyridinyl)anilineRattus norvegicus (Norway rat)Potency56.234110
2-methyl-1H-pyrimido[1,2-a]benzimidazol-4-oneRattus norvegicus (Norway rat)Potency31.622810
9,14-Dimethyl-5-methylidene-3,13-dioxatetracyclo[8.4.0.02,6.012,14]tetradec-9-ene-4,11-dioneRattus norvegicus (Norway rat)Potency8.912510
IPA-3Rattus norvegicus (Norway rat)Potency1.888810
2-chloro-N-(5-methyl-3-isoxazolyl)acetamideRattus norvegicus (Norway rat)Potency70.794610
5-(2-methylthioethyl)hydantoinRattus norvegicus (Norway rat)Potency8.912510
2-(2-phenoxyethylsulfonyl)-1H-benzimidazoleRattus norvegicus (Norway rat)Potency44.668410
3-(4-fluoroanilino)-1-(3-nitrophenyl)-1-propanoneRattus norvegicus (Norway rat)Potency3.548110
5-[[[(5-tert-butyl-2-methyl-3-furanyl)-oxomethyl]amino]methyl]-2-furancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency25.118910
2-(3-oxo-4H-quinoxalin-2-yl)propanoic acid ethyl esterRattus norvegicus (Norway rat)Potency44.668410
1-(2-pyridin-4-yl-1-oxa-3,4-diazaspiro[4.6]undec-2-en-4-yl)ethanoneRattus norvegicus (Norway rat)Potency27.005020
lomatinRattus norvegicus (Norway rat)Potency56.234110
4-chloro-N-(4-chloro-2,5-dimethoxyphenyl)-5-dithiazolimineRattus norvegicus (Norway rat)Potency22.387210
4,7-dimethoxy-2,3-dihydroinden-1-oneRattus norvegicus (Norway rat)Potency56.234110
4-oxo-10H-pyrimido[1,2-a]benzimidazole-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency30.258620
2-amino-3-cyano-5,6,7,8-tetrahydroquinoline-4-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency31.622810
4-[[bis(2-hydroxyethyl)amino]methyl]-2,6-ditert-butylphenolRattus norvegicus (Norway rat)Potency3.548110
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineRattus norvegicus (Norway rat)Potency67.833420
1,3-dichloro-7-methyl-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileRattus norvegicus (Norway rat)Potency30.669420
LSM-31955Rattus norvegicus (Norway rat)Potency17.782810
2,3-diphenyl-6-quinoxalinecarboxylic acidRattus norvegicus (Norway rat)Potency79.432810
2-[(4,4-dimethyl-2,6-dioxocyclohexyl)-(3-pyridinyl)methyl]-5,5-dimethylcyclohexane-1,3-dioneRattus norvegicus (Norway rat)Potency35.481310
pirarubicin hydrochlorideRattus norvegicus (Norway rat)Potency56.234110
niflumic acidRattus norvegicus (Norway rat)Potency89.125110
chalconeRattus norvegicus (Norway rat)Potency100.000010
isoliquiritigeninRattus norvegicus (Norway rat)Potency34.872820
3-Hydroxy-1-(4-hydroxyphenyl)-1-propanoneRattus norvegicus (Norway rat)Potency79.432810
dibenzylidene acetoneRattus norvegicus (Norway rat)Potency56.234110
cefazolin(1-)Rattus norvegicus (Norway rat)Potency11.917320
gw9662Rattus norvegicus (Norway rat)Potency1.584910
calmidazoliumRattus norvegicus (Norway rat)Potency32.464810
2-(4-hydroxy-3-methoxyphenyl)-3-(2-methoxyphenyl)-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency25.118910
6-amino-2-methyl-8-phenyl-1,6,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrileRattus norvegicus (Norway rat)Potency50.118710
N-[(8-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-oxolanylmethyl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency15.848910
2-imino-N,8-dimethyl-5-oxo-1-propan-2-yl-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency45.639820
2-(2,5-dimethoxyphenyl)-5-(5-methyl-2-furanyl)-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency61.087620
1-[4-[4-[(4-methylphenyl)methylamino]phenyl]-1-piperazinyl]ethanoneRattus norvegicus (Norway rat)Potency79.432810
N-(cyclohexylmethyl)-5,6,7,8-tetrahydrotetrazolo[5,1-b]quinazolin-9-amineRattus norvegicus (Norway rat)Potency4.466810
1-(2,3-dihydroindol-1-yl)-2-[(5,5-dimethyl-6H-[1,2,4]triazolo[3,4-a]isoquinolin-3-yl)thio]ethanoneRattus norvegicus (Norway rat)Potency1.258910
2-[5-(4-butoxyphenyl)-2-tetrazolyl]-N-(2-furanylmethyl)acetamideRattus norvegicus (Norway rat)Potency100.000010
LSM-19079Rattus norvegicus (Norway rat)Potency56.234110
2-(4-chlorophenoxy)-N-(2-pyridin-4-yl-1,3-benzoxazol-5-yl)acetamideRattus norvegicus (Norway rat)Potency63.095710
1-(2,5-dimethoxyphenyl)-2-[[5-(2-furanyl)-4-propyl-1,2,4-triazol-3-yl]thio]ethanoneRattus norvegicus (Norway rat)Potency39.810710
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
2-[[2-[[4-(2-furanylmethyl)-5-(phenylmethyl)-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideRattus norvegicus (Norway rat)Potency10.000010
9-methyl-6H-benzo[c][1,2]benzothiazine 5,5-dioxideRattus norvegicus (Norway rat)Potency56.234110
2-[2,2-dimethyl-6-[4-morpholinyl(oxo)methyl]-3-oxo-1,4-benzoxazin-4-yl]-N-phenylacetamideRattus norvegicus (Norway rat)Potency79.432810
3-amino-5-methoxy-2-benzofurancarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency31.622810
3-[(1-tert-butyl-5-tetrazolyl)-[2-furanylmethyl(2-oxolanylmethyl)amino]methyl]-6-methoxy-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency22.387210
2-(2-ethyl-6-methyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(5-methyl-2-furanyl)methyl]-N-(3-pyridinylmethyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
3-(benzenesulfonyl)-2-imino-1-(2-oxolanylmethyl)-5-dipyrido[1,2-d-3',4'-f]pyrimidinoneRattus norvegicus (Norway rat)Potency31.622810
N-[2-(2-furanylmethylthio)ethyl]-4-methoxybenzenesulfonamideRattus norvegicus (Norway rat)Potency89.125110
6,8-dimethyl-3-[(3-methyl-1-piperidinyl)-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency56.234110
2-[5-[4-(dimethylamino)phenyl]-2-tetrazolyl]-N-[2-(4-morpholinyl)phenyl]acetamideRattus norvegicus (Norway rat)Potency100.000010
6-amino-4-[4-(2-amino-2-oxoethoxy)-2-chloro-5-methoxyphenyl]-5-cyano-2-methyl-4H-pyran-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency44.668410
3-[(2-chlorophenyl)methyl]-N-phenyl-7-triazolo[4,5-d]pyrimidinamineRattus norvegicus (Norway rat)Potency17.782810
2-[benzenesulfonyl(2-pyridinyl)amino]acetic acid methyl esterRattus norvegicus (Norway rat)Potency31.622810
5-(2-furanyl)-3-[2-methoxy-6-(4-methylphenyl)-3-pyridinyl]-1,2,4-oxadiazoleRattus norvegicus (Norway rat)Potency20.483920
6-ethoxy-3-[[2-oxolanylmethyl-[[1-(2-phenylethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency0.891310
N-[2-[1,3-benzodioxol-5-yl-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]amino]-2-oxoethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency28.183810
3-[1-azepanyl-[1-(phenylmethyl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency50.118710
N-[2-(3-acetamidophenyl)-3H-benzimidazol-5-yl]acetamideRattus norvegicus (Norway rat)Potency89.716420
[3-[3-(5-methyl-2-furanyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]-phenylmethanoneRattus norvegicus (Norway rat)Potency56.234110
4,5-dichloro-3-isothiazolecarboxylic acid [1-(2-furanylmethylamino)-1-oxopropan-2-yl] esterRattus norvegicus (Norway rat)Potency50.118710
3-[(1-cyclopentyl-5-tetrazolyl)-[4-(2-methoxyphenyl)-1-piperazinyl]methyl]-7-methyl-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency15.848910
7-[[1-(2-oxolanylmethyl)-5-tetrazolyl]-(1-pyrrolidinyl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-oneRattus norvegicus (Norway rat)Potency36.041520
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]propanoic acid ethyl esterRattus norvegicus (Norway rat)Potency5.530320
2-(3,4-diethoxyphenyl)-5-(2-furanyl)-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency28.183810
5,6,7-trimethoxy-1-methyl-2-indolecarboxylic acidRattus norvegicus (Norway rat)Potency56.234110
9,10-dimethoxy-2,4,6,7-tetrahydro-[1,3]oxazino[4,3-a]isoquinoline-1-carbonitrileRattus norvegicus (Norway rat)Potency12.589310
2-[[5-(2,4-dichlorophenyl)-1,3,4-oxadiazol-2-yl]thio]acetic acid butyl esterRattus norvegicus (Norway rat)Potency3.162310
2-[[1-(2-methoxyethyl)-5-tetrazolyl]thio]-1-phenylethanoneRattus norvegicus (Norway rat)Potency0.891310
1-(ethylamino)-3-[3-(ethylamino)-2-hydroxypropoxy]-2-propanolRattus norvegicus (Norway rat)Potency22.387210
[5-(2-furanyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneRattus norvegicus (Norway rat)Potency39.810710
5,7-dimethyl-2-(1-pyrrolidinyl)-3-quinolinecarbonitrileRattus norvegicus (Norway rat)Potency39.810710
3-cyclohexyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-1-[2-(1-pyrrolidinyl)ethyl]ureaRattus norvegicus (Norway rat)Potency63.095710
N-[2-(2-ethyl-5-tetrazolyl)phenyl]-3-(1-tetrazolyl)benzamideRattus norvegicus (Norway rat)Potency42.741420
1-[4-[4-[(phenylmethyl)amino]phenyl]-1-piperazinyl]ethanoneRattus norvegicus (Norway rat)Potency44.668410
4-[2-(3-fluorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]morpholineRattus norvegicus (Norway rat)Potency56.234110
6,7-dimethoxy-2-[[2-[4-(4-methoxyphenyl)-1-piperazinyl]-2-oxoethyl]thio]-3-quinolinecarbonitrileRattus norvegicus (Norway rat)Potency50.118710
5-cyano-6-[[2-(2,3-dimethylanilino)-2-oxoethyl]thio]-4-(2-furanyl)-2-methyl-N-phenyl-1,4-dihydropyridine-3-carboxamideRattus norvegicus (Norway rat)Potency19.622220
N-methyl-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineRattus norvegicus (Norway rat)Potency37.618820
N-[2-[(3-cyano-6-ethoxy-2-quinolinyl)amino]ethyl]propanamideRattus norvegicus (Norway rat)Potency50.118710
1-(4-chlorophenyl)-1-cyclohexyl-3-(4-morpholinyl)-1-propanolRattus norvegicus (Norway rat)Potency31.622810
N-[1-[4-(4-methylphenyl)-2-thiazolyl]-4-piperidinyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideRattus norvegicus (Norway rat)Potency0.891310
2,5-diethoxy-N-[2-(2-methylphenyl)ethyl]-4-(1-tetrazolyl)benzenesulfonamideRattus norvegicus (Norway rat)Potency31.622810
8-[2-(4-methoxyphenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-1,4-dioxa-8-azaspiro[4.5]decaneRattus norvegicus (Norway rat)Potency26.651420
5-[(4-chloro-1-pyrazolyl)methyl]-N-(6-methyl-1,3-benzothiazol-2-yl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency70.794610
N-butyl-N-[5-(3,4,5-trimethoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency56.234110
2-acetyl-6-amino-8-(2-phenylethyl)-1,3,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrileRattus norvegicus (Norway rat)Potency25.118910
4-[2-(3-fluorophenyl)-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-9-yl]morpholineRattus norvegicus (Norway rat)Potency42.800020
N-(4-methylphenyl)-2-(3-oxo-5,6-dihydroimidazo[2,1-b]thiazol-2-yl)acetamideRattus norvegicus (Norway rat)Potency44.668410
1-(3-cyano-7-methoxy-2-quinolinyl)-4-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency89.125110
6-ethoxy-3-[[[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency56.234110
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency56.234110
2-[4-(benzenesulfonyl)phenyl]-5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency59.621820
N-[2,5-diethoxy-4-[[oxo-(3,4,5-trimethoxyphenyl)methyl]amino]phenyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency50.118710
4-[3-(1,3-dioxo-2-isoindolyl)propylamino]-2-methylisoindole-1,3-dioneRattus norvegicus (Norway rat)Potency70.794610
8-[(1-tert-butyl-5-tetrazolyl)-thiomorpholin-4-ylmethyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneRattus norvegicus (Norway rat)Potency50.118710
2-(2,5-dimethoxyphenyl)-5-[4-(4-methoxyphenyl)phenyl]-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency45.857720
2-methoxy-N-methyl-N-[5-(5-methyl-2-pyrazinyl)-1,3,4-thiadiazol-2-yl]acetamideRattus norvegicus (Norway rat)Potency31.622810
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-6-methyl-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency25.118910
2-fluoro-N-[2-(4-fluorophenyl)-1,3-benzoxazol-5-yl]benzamideRattus norvegicus (Norway rat)Potency50.118710
7-(2-methyl-2,3-dihydroindol-1-yl)-3-(phenylmethyl)triazolo[4,5-d]pyrimidineRattus norvegicus (Norway rat)Potency50.118710
1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-[5-[4-(dimethylamino)phenyl]-2-tetrazolyl]ethanoneRattus norvegicus (Norway rat)Potency56.607220
7-(methoxymethyl)-3-(2-methoxyphenyl)-1H-[1,2,4]triazolo[4,3-a]pyrimidin-5-oneRattus norvegicus (Norway rat)Potency35.481310
6-ethoxy-3-[[2-furanylmethyl-[[1-(phenylmethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency32.122020
3-[1-azepanyl-[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl]-6,7-dimethoxy-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency0.891310
2-(3-methylphenoxy)-N-[4-(4-methylsulfonyl-1-piperazinyl)phenyl]acetamideRattus norvegicus (Norway rat)Potency2.818410
9-[3-(4-acetyl-3,5-dimethyl-1-pyrazolyl)-2-hydroxypropyl]-6-methyl-3,4-dihydro-2H-carbazol-1-oneRattus norvegicus (Norway rat)Potency50.118710
N-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(3-hydroxypropyl)benzenesulfonamideRattus norvegicus (Norway rat)Potency39.810710
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneRattus norvegicus (Norway rat)Potency30.300120
6-methoxy-3-[[2-oxolanylmethyl-[[1-(phenylmethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency70.794610
1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-(phenylmethyl)-1-(3-pyridinylmethyl)ureaRattus norvegicus (Norway rat)Potency79.432810
6-phenyl-4-(1-pyrrolyl)furo[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency56.234110
4-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5-furo[3,2-b]pyrrolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency50.118710
LSM-34623Rattus norvegicus (Norway rat)Potency44.668410
2-[(3-chlorophenyl)-(3-oxo-5-propyl-1,2-dihydropyrazol-4-yl)methyl]propanedinitrileRattus norvegicus (Norway rat)Potency1.778310
4-methyl-6-(methylthio)-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency26.968020
2-[[4-(3,4-dimethoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
2-[(3-cyano-5,7-dimethyl-2-quinolinyl)thio]-N-(2-furanylmethyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
6-amino-4-(2,4-dimethoxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileRattus norvegicus (Norway rat)Potency31.622810
2-[[5-(2-furanyl)-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]-1-(4-morpholinyl)ethanoneRattus norvegicus (Norway rat)Potency15.848910
N-(2,1,3-benzothiadiazol-4-yl)-3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency39.810710
4-[2-(4-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]morpholineRattus norvegicus (Norway rat)Potency7.996020
3-[2-methoxy-6-(4-methylphenyl)-3-pyridinyl]-5-(3-pyridinyl)-1,2,4-oxadiazoleRattus norvegicus (Norway rat)Potency37.646020
N-methyl-N-[5-(5-methyl-2-pyrazinyl)-1,3,4-thiadiazol-2-yl]-2-oxolanecarboxamideRattus norvegicus (Norway rat)Potency36.041520
4-amino-N5-[1-(2-furanyl)-2-(3-methylbutylamino)-2-oxoethyl]-N5-(2-methoxyphenyl)isothiazole-3,5-dicarboxamideRattus norvegicus (Norway rat)Potency35.716820
6-amino-4-[3-ethoxy-4-[2-(4-morpholinyl)ethoxy]phenyl]-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileRattus norvegicus (Norway rat)Potency89.125110
6-methoxy-3-[[[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl-(2-phenylethyl)amino]methyl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency89.125110
N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]butanamideRattus norvegicus (Norway rat)Potency48.022420
5-[(2-fluoroanilino)methyl]-8-quinolinolRattus norvegicus (Norway rat)Potency0.707910
4-[[4-(1,3-benzothiazol-2-yl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-2-methoxyphenolRattus norvegicus (Norway rat)Potency2.238710
1-piperidinecarboxylic acid (5-chloro-8-quinolinyl) esterRattus norvegicus (Norway rat)Potency31.622810
2-[[2-[3-cyano-4-(methoxymethyl)-6-methyl-2-oxo-1-pyridinyl]-1-oxoethyl]amino]benzoic acid methyl esterRattus norvegicus (Norway rat)Potency50.118710
3-[3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-5,7-dimethyl-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency35.481310
3-[1-(2-furanylmethyl)-5-phenyl-2-pyrrolyl]propanoic acidRattus norvegicus (Norway rat)Potency12.589310
2-[(5-methyl-1H-1,2,4-triazol-3-yl)thio]-1-phenylethanoneRattus norvegicus (Norway rat)Potency79.432810
1-(4-chlorophenyl)-2-[[4-ethyl-5-(2-methyl-3-furanyl)-1,2,4-triazol-3-yl]thio]ethanoneRattus norvegicus (Norway rat)Potency12.589310
cefsulodin sodiumRattus norvegicus (Norway rat)Potency30.258610
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideRattus norvegicus (Norway rat)Potency39.810710
5-(2-furanyl)-N-(4-methylphenyl)-3-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency17.782810
diethylstilbestrol dipropionateRattus norvegicus (Norway rat)Potency100.000010
methamilane methiodideRattus norvegicus (Norway rat)Potency100.000010
physostigmine salicylateRattus norvegicus (Norway rat)Potency44.668410
n(6)-cyclopentyladenosineRattus norvegicus (Norway rat)Potency0.631010
1-cyclohexyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-amineRattus norvegicus (Norway rat)Potency15.848910
6-ethyl-6-methyl-5,8-dihydro-1H-thiopyrano[2,3]thieno[2,4-b]pyrimidine-2,4-dioneRattus norvegicus (Norway rat)Potency22.535820
2-[[3-cyano-4-(5-methyl-2-furanyl)-5,6,7,8-tetrahydroquinolin-2-yl]thio]acetic acid methyl esterRattus norvegicus (Norway rat)Potency70.794610
2-[(3-oxo-5-phenyl-1,2-dihydropyrazol-4-yl)-(3-thiophenyl)methyl]propanedinitrileRattus norvegicus (Norway rat)Potency39.810710
1-amino-5-(4-morpholinyl)-6,7,8,9-tetrahydrothieno[2,3-c]isoquinoline-2-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency22.535820
2-[(7-methyl-4-oxo-3-phenyl-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-2-yl)thio]acetic acid methyl esterRattus norvegicus (Norway rat)Potency79.432810
6-amino-4-(5-bromo-2-thiophenyl)-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileRattus norvegicus (Norway rat)Potency28.183810
2-[2-hydroxy-6,7-dimethoxy-4-(4-morpholinyl)-1-naphthalenyl]-N-phenylacetamideRattus norvegicus (Norway rat)Potency12.589310
8-(2-furanyl)-6-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3,3-dimethyl-1,4-dihydrothiopyrano[3,4-c]pyridine-5-carbonitrileRattus norvegicus (Norway rat)Potency13.516020
3-amino-5-methyl-4-[[3-(4-morpholinyl)propylamino]-oxomethyl]-2-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency89.125110
LSM-19776Rattus norvegicus (Norway rat)Potency56.234110
5-chloro-3-[[2-(4-ethoxycarbonyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency89.125110
7-diethylaminocoumarin-3-carboxylic acidRattus norvegicus (Norway rat)Potency44.668410
6-[2-(dimethylamino)ethylamino]-8-(2-furanyl)-3,3-dimethyl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrileRattus norvegicus (Norway rat)Potency79.432820
N-(2,1,3-benzothiadiazol-5-yl)-2,4-dimethyl-6-oxo-3-pyrancarboxamideRattus norvegicus (Norway rat)Potency89.125110
4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl esterRattus norvegicus (Norway rat)Potency9.180420
2-cyano-N-(2-furanylmethyl)-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetamideRattus norvegicus (Norway rat)Potency19.952610
LSM-27020Rattus norvegicus (Norway rat)Potency28.183810
2-(6-bromo-2-methyl-4-oxo-1-quinolinyl)-N-(2-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency15.848910
2-[[(4-chloro-1-methyl-3-pyrazolyl)-oxomethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency31.622810
2-[[5-cyano-2-(3,4-dimethoxyphenyl)-4-oxo-2,3-dihydro-1,3-thiazin-6-yl]thio]acetic acid ethyl esterRattus norvegicus (Norway rat)Potency31.622810
3-(6-methyl-4-oxo-2-sulfanylidene-1H-pyrimidin-5-yl)propanoic acid methyl esterRattus norvegicus (Norway rat)Potency5.623410
N-ethyl-2-imino-10-methyl-1-[(4-methylphenyl)methyl]-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency13.534620
2-(4-chlorophenyl)-5-(methylamino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency39.810720
2-(butan-2-ylamino)-N-[4-[5-[[2-(butan-2-ylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideRattus norvegicus (Norway rat)Potency31.622810
2-(4-chlorophenyl)-5-(1-piperidinyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency43.321820
2-[(2-fluorophenoxy)methyl]-5-[3-(1-imidazolyl)propylamino]-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency56.234110
2-(butylamino)-N-[4-[5-[[2-(butylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideRattus norvegicus (Norway rat)Potency22.387210
3-benzamido-5-bromo-2-benzofurancarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency50.118710
5-(4-methoxyphenyl)-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency11.220210
7-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxoethyl]amino]-5H-[1,3]dioxolo[4,5-f]indole-6-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.810710
LSM-23818Rattus norvegicus (Norway rat)Potency39.810710
2-amino-4-(2-ethoxyphenyl)-7-methyl-5-oxo-6-(2-pyridinylmethyl)-4H-pyrano[3,2-c]pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency14.125410
N-(3-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideRattus norvegicus (Norway rat)Potency4.466810
2-(4-chlorophenyl)-3-(2-furanylmethyl)imidazo[4,5-b]quinoxalineRattus norvegicus (Norway rat)Potency44.668410
5-(2,4-dimethoxyphenyl)-7-(3,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency12.589310
2-[(6-chloro-4-ethyl-2-oxo-1-benzopyran-7-yl)oxy]propanoic acidRattus norvegicus (Norway rat)Potency50.118710
1-(3,5-dichlorophenyl)-3-(N-hydroxyanilino)pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency19.952610
5-(4-methoxyphenyl)-7-(4-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency35.481310
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-phenyl-2-furancarboxamideRattus norvegicus (Norway rat)Potency56.234110
1-(3,4-dichlorophenyl)-2-[[4-(2-furanylmethyl)-5-(3-pyridinyl)-1,2,4-triazol-3-yl]thio]ethanoneRattus norvegicus (Norway rat)Potency44.668410
2-[5-[(2-chlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineRattus norvegicus (Norway rat)Potency89.125110
3-methyl-N-(1-propyl-3-pyrazolo[3,4-b]quinolinyl)butanamideRattus norvegicus (Norway rat)Potency70.794610
2-[5-[(2,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineRattus norvegicus (Norway rat)Potency44.668410
LSM-32147Rattus norvegicus (Norway rat)Potency79.432810
2-amino-4-pyridin-4-yl-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency56.234110
5-(4-bromophenyl)-4-(4-hydroxy-3-methoxyphenyl)-3-methyl-2,4-dihydropyrrolo[3,4-c]pyrazol-6-oneRattus norvegicus (Norway rat)Potency7.943310
2-[4-[(4-chlorophenyl)methoxy]phenyl]-5-(dimethylamino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency7.811720
N-[7-(2-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideRattus norvegicus (Norway rat)Potency40.676520
5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-(2-furanyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency19.952610
2-(4-methoxyphenyl)-3-propylimidazo[4,5-b]quinoxalineRattus norvegicus (Norway rat)Potency40.870820
N-[3-(2-furanylmethylamino)-2-quinoxalinyl]-3-methylbenzenesulfonamideRattus norvegicus (Norway rat)Potency44.668410
3-[[2-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-1-oxoethyl]amino]-6-methyl-1H-indole-2-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency14.125410
2-(2-furanyl)-5-(2-furanylmethylamino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency39.810710
5-[(2-chlorophenyl)methylamino]-2-(3,4-dimethoxyphenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency26.651420
5-(1-azepanyl)-2-(3,4-dimethoxyphenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency55.302620
1-[4-cyano-2-(2-furanyl)-5-oxazolyl]-4-piperidinecarboxamideRattus norvegicus (Norway rat)Potency89.716420
1-[3-[(8-methyl-5H-pyrimido[5,4-b]indol-4-yl)amino]propyl]-2-pyrrolidinoneRattus norvegicus (Norway rat)Potency15.848910
5-[4-(diphenylmethyl)-1-piperazinyl]-2-(2-methoxyphenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency2.238710
2-(2-methoxyphenyl)-5-[2-(4-methoxyphenyl)ethylamino]-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency19.952610
5-[(4-fluorophenyl)methylamino]-2-(2-methoxyphenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency56.234110
LSM-28231Rattus norvegicus (Norway rat)Potency6.309610
2-(3-methylphenyl)sulfonyl-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetonitrileRattus norvegicus (Norway rat)Potency79.432810
2-[[6,6-dimethyl-2-(propan-2-ylthio)-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-4-yl]thio]-N-(2-furanylmethyl)acetamideRattus norvegicus (Norway rat)Potency31.622810
2-methoxy-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
N-[7-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideRattus norvegicus (Norway rat)Potency17.782810
N-(1-ethyl-7-methyl-3-pyrazolo[3,4-b]quinolinyl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency70.794610
1-(thiophen-2-ylmethyl)-3-thiophen-2-ylsulfonyl-2-pyrrolo[3,2-b]quinoxalinamineRattus norvegicus (Norway rat)Potency56.234110
5-[2-(3,4-dimethoxyphenyl)ethylamino]-2-(1-naphthalenylmethyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency2.511910
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dioneRattus norvegicus (Norway rat)Potency8.912510
2,6-dimethyl-4-(1-phenyl-4-pyrazolyl)furo[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency10.610120
N-[5-(3,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-yl]carbamic acid ethyl esterRattus norvegicus (Norway rat)Potency7.079510
3-[[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-1-oxoethyl]amino]-5-ethoxy-1H-indole-2-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency28.183810
LSM-28489Rattus norvegicus (Norway rat)Potency12.589310
4,8-dimethyl-3-(phenylmethyl)-7-(2H-tetrazol-5-ylmethoxy)-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency28.183810
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterRattus norvegicus (Norway rat)Potency0.398110
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanolRattus norvegicus (Norway rat)Potency28.183810
2-amino-4-(2-furanyl)-6-(2-pyridinyl)-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency31.622820
1-[1-oxo-2-[(4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl)oxy]ethyl]-4-piperidinecarboxylic acidRattus norvegicus (Norway rat)Potency7.943310
LSM-32980Rattus norvegicus (Norway rat)Potency79.432810
7-(2-methoxyethyl)-3-methyl-8-(phenylthio)purine-2,6-dioneRattus norvegicus (Norway rat)Potency50.118710
3-[4,8-dimethyl-2-oxo-7-(2H-tetrazol-5-ylmethoxy)-1-benzopyran-3-yl]propanoic acid ethyl esterRattus norvegicus (Norway rat)Potency30.669420
2-methyl-3-phenyl-5-propyl-7-[4-(2-pyridinyl)-1-piperazinyl]pyrazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency29.903320
5-(3-methoxyphenyl)-N-(2-oxolanylmethyl)-7-(trifluoromethyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency89.125110
LSM-20899Rattus norvegicus (Norway rat)Potency56.234110
3,4,7-trimethyl-5-(3-oxobutan-2-yloxy)-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency56.234110
2-amino-6-[3-(1-imidazolyl)propyl]-4-(2-methoxyphenyl)-7-methyl-5-oxo-4H-pyrano[3,2-c]pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency89.125110
4-(1-benzotriazolyl)-5-(2-methoxyphenoxy)benzene-1,2-dicarbonitrileRattus norvegicus (Norway rat)Potency0.251210
6-amino-4-(4-fluorophenyl)-3-methyl-1-phenyl-5-pyrazolo[3,4-b]pyridinecarbonitrileRattus norvegicus (Norway rat)Potency49.692720
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency24.803310
(3aR,6aS)-3-(3,4-dimethoxyphenyl)-5-(2,4-dimethylphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dioneRattus norvegicus (Norway rat)Potency22.387210
3-methyl-6-(1-naphthalenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleRattus norvegicus (Norway rat)Potency44.668410
3-(2-furanylmethyl)-8-(4-methoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrileRattus norvegicus (Norway rat)Potency50.118710
N2-(4-fluorophenyl)-6-[[4-(2-pyridinyl)-1-piperazinyl]methyl]-1,3,5-triazine-2,4-diamineRattus norvegicus (Norway rat)Potency50.118710
4,9-dimethyl-3-(2H-tetrazol-5-ylmethoxy)-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-6-oneRattus norvegicus (Norway rat)Potency55.302620
8-methoxy-5-methyl-3-[2-(1-pyrrolidinyl)ethyl]-4-pyrimido[5,4-b]indoloneRattus norvegicus (Norway rat)Potency17.782810
2-amino-6-(2-furanylmethyl)-7-methyl-5-oxo-4-(3-pyridinyl)-4H-pyrano[3,2-c]pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency44.668410
LSM-33283Rattus norvegicus (Norway rat)Potency19.952610
1-(4-fluorophenyl)-2-[[4-(2-furanylmethyl)-5-(phenoxymethyl)-1,2,4-triazol-3-yl]thio]ethanoneRattus norvegicus (Norway rat)Potency50.118710
3,3',4,5'-tetrahydroxystilbeneRattus norvegicus (Norway rat)Potency11.663730
5-(1-imidazolylsulfonyl)-8-methoxyquinolineRattus norvegicus (Norway rat)Potency35.481310
3,4-methylenedioxy-beta-nitrostyreneRattus norvegicus (Norway rat)Potency5.742940
5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency31.622810
(2R)-1-[(4,8-dimethoxy-7-furo[2,3-b]quinolinyl)oxy]-3-methylbutane-2,3-diolRattus norvegicus (Norway rat)Potency79.432810
2-[[2-furanyl(oxo)methyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency66.945220
carbidopa, (r)-isomerRattus norvegicus (Norway rat)Potency5.407320
2-amino-4-(5-methyl-2-furanyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrileRattus norvegicus (Norway rat)Potency31.622810
1-(diethylamino)-3-methyl-4-pyrido[1,2-a]benzimidazolecarbonitrileRattus norvegicus (Norway rat)Potency19.952610
sch-202676Rattus norvegicus (Norway rat)Potency21.135020
2-amino-4-phenyl-6-(1-pyrrolidinyl)pyridine-3,5-dicarbonitrileRattus norvegicus (Norway rat)Potency79.432810
levosulpirideRattus norvegicus (Norway rat)Potency0.492920
caffeic acidRattus norvegicus (Norway rat)Potency1.062110
3-(4-methylbenzoyl)acrylic acidRattus norvegicus (Norway rat)Potency2.818410
2-oxo-N-(3-pyridinylmethyl)-1-benzopyran-3-carboxamideRattus norvegicus (Norway rat)Potency31.622810
N-[(2-phenylethylamino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency22.387210
2-(8-quinolinylthio)acetic acidRattus norvegicus (Norway rat)Potency56.234110
4-phenyl-N-(3-pyridinyl)-2-thiazolamineRattus norvegicus (Norway rat)Potency0.251210
1-(3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinyl)ethanoneRattus norvegicus (Norway rat)Potency15.848910
2-(4-ethylphenoxy)-N-(1H-1,2,4-triazol-5-yl)acetamideRattus norvegicus (Norway rat)Potency56.234110
N-[(4-pyrimidinylthio)methyl]benzamideRattus norvegicus (Norway rat)Potency12.589310
4-chloro-1-methyl-3-nitro-2-quinolinoneRattus norvegicus (Norway rat)Potency2.238710
2-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxy]acetic acid propan-2-yl esterRattus norvegicus (Norway rat)Potency56.234110
nitrofurylacrylic acidRattus norvegicus (Norway rat)Potency10.000010
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency25.118910
1-(1,3-benzodioxol-5-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
2-(4-chloro-3-methylphenoxy)-N-(1H-1,2,4-triazol-5-yl)acetamideRattus norvegicus (Norway rat)Potency39.810710
3-methyl-N-[4-(4-oxo-3,1-benzoxazin-2-yl)phenyl]butanamideRattus norvegicus (Norway rat)Potency42.871220
5-methyl-4-[(2-oxo-1-benzopyran-7-yl)oxymethyl]-2-furancarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency19.952610
N-(4-hydroxy-2-methyl-5-propan-2-ylphenyl)-4-methoxybenzenesulfonamideRattus norvegicus (Norway rat)Potency31.622810
2-(3,4-dichlorophenyl)imidazo[1,2-a]pyrimidineRattus norvegicus (Norway rat)Potency39.810710
5-(2-phenyl-4-triazolyl)-2H-tetrazoleRattus norvegicus (Norway rat)Potency44.668410
1-(2-methoxyphenyl)-3-(2-pyridinyl)thioureaRattus norvegicus (Norway rat)Potency28.183810
N-cyclohexyl-2,3-dihydroindole-1-carboxamideRattus norvegicus (Norway rat)Potency8.912510
3-[1-(carboxymethyl)-5-phenyl-2-pyrrolyl]propanoic acidRattus norvegicus (Norway rat)Potency21.450920
N-[(3-nitroanilino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency31.622810
2-methyl-5-(5-methyl-2-furanyl)-3-(1-pyrrolyl)-4-thieno[2,3-d]pyrimidinoneRattus norvegicus (Norway rat)Potency56.234110
1-[2-(dimethylamino)ethyl]-5-methoxy-N-methyl-2-indolecarboxamideRattus norvegicus (Norway rat)Potency79.432810
2-mercaptobenzoxazoleRattus norvegicus (Norway rat)Potency79.432810
6-methoxy-2-oxo-N-(3-pyridinylmethyl)-1-benzopyran-3-carboxamideRattus norvegicus (Norway rat)Potency79.432810
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileRattus norvegicus (Norway rat)Potency15.848910
2-[[2-furanyl(oxo)methyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency56.234110
phenylthiazolylthioureaRattus norvegicus (Norway rat)Potency4.863230
vu0038882Rattus norvegicus (Norway rat)Potency10.000010
5-cyano-2-methyl-6-sulfanylidene-1H-pyridine-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency7.943310
4-Acetyl-3-methyl-5-(methylthio)thiophene-2-carboxylic acidRattus norvegicus (Norway rat)Potency0.089110
7,9-dibromo-3,4-dihydropyrido[2,1-c][1,2,4]thiadiazine 2,2-dioxideRattus norvegicus (Norway rat)Potency31.622810
4-(1H-benzimidazol-2-yl)quinolineRattus norvegicus (Norway rat)Potency28.183810
2-(Phenylthio)nicotinic acidRattus norvegicus (Norway rat)Potency1.258910
2-(3-nitrophenyl)-2,3-dihydro-1H-perimidineRattus norvegicus (Norway rat)Potency50.118710
5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency64.775820
1-hydroxy-2-phenyl-1,5,6,7-tetrahydro-4H-benzimidazol-4-oneRattus norvegicus (Norway rat)Potency28.183810
4,5-dimethylaminobenzylidene-2-thiobarbituric acidRattus norvegicus (Norway rat)Potency6.990610
2-[[oxo(phenoxy)methyl]amino]benzene-1,4-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency79.432810
(4-Methyl-2-oxochromen-7-yl) furan-2-carboxylateRattus norvegicus (Norway rat)Potency75.113720
1-(2-furanyl)-2-([1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-ylthio)ethanoneRattus norvegicus (Norway rat)Potency12.589310
1-(2,5-dimethoxyphenyl)-3-phenylthioureaRattus norvegicus (Norway rat)Potency0.316210
N-[4-(3,4-dimethylphenyl)-2-thiazolyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency89.125110
5-(methoxymethyl)-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneRattus norvegicus (Norway rat)Potency28.183810
3-[(6-methyl-4-phenyl-2-quinazolinyl)amino]propanoic acidRattus norvegicus (Norway rat)Potency79.432810
N-(2-phenyl-3-imidazo[1,2-a]pyridinyl)carbamic acid methyl esterRattus norvegicus (Norway rat)Potency3.981110
2-[[(4-phenyl-1,2,4-triazol-3-yl)thio]methyl]imidazo[1,2-a]pyrimidineRattus norvegicus (Norway rat)Potency36.253020
2-amino-4-(4-chlorophenyl)-6-methyl-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency31.622810
4-[2-(1-methyl-2-benzimidazolyl)ethyl]anilineRattus norvegicus (Norway rat)Potency0.100010
4-pyridin-4-yl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrileRattus norvegicus (Norway rat)Potency14.125410
N-(3-chloro-4-hydroxy-2,5-dimethylphenyl)benzenesulfonamideRattus norvegicus (Norway rat)Potency44.668410
4-(2,5-dimethylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency2.511910
2-amino-5-ethyl-4-(2-furanyl)-6-propyl-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency15.848910
N-cyclopentyl-2-benzo[e]benzofurancarboxamideRattus norvegicus (Norway rat)Potency56.234110
7,7-dimethyl-2-(1-pyrrolidinyl)-5,8-dihydropyrano[4,3-b]pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency31.622820
3-(4-chlorophenyl)-2,5-dimethyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneRattus norvegicus (Norway rat)Potency56.234110
3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinecarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency56.234110
6-methoxy-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazineRattus norvegicus (Norway rat)Potency17.782810
2-methyl-N-(1-methyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-yl)propanamideRattus norvegicus (Norway rat)Potency44.668410
N-(3,4-dimethoxyphenyl)-4-methoxybenzamideRattus norvegicus (Norway rat)Potency0.891310
2-[(1-acetyl-3-indolyl)amino]benzoic acidRattus norvegicus (Norway rat)Potency39.810710
4-(1-ethyl-2-benzimidazolyl)anilineRattus norvegicus (Norway rat)Potency35.481310
N-(4-ethylphenyl)-4-oxo-3H-phthalazine-1-carboxamideRattus norvegicus (Norway rat)Potency15.848910
2-(4-chlorophenyl)-5-(4-fluorophenyl)-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency25.118910
4-(2-furanylmethyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency56.234110
N-[2-(4-methoxyphenyl)-5-benzotriazolyl]butanamideRattus norvegicus (Norway rat)Potency25.118910
(3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolyl)-(3-methyl-1-pyrazolyl)methanoneRattus norvegicus (Norway rat)Potency31.622810
1-[(4-phenyl-1-piperazinyl)methyl]-2-naphthalenolRattus norvegicus (Norway rat)Potency79.432810
3-(8-methyl-2-imidazo[1,2-a]pyridinyl)-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency14.125410
N-(1-methyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-yl)-2-(1-pyrrolidinyl)acetamideRattus norvegicus (Norway rat)Potency79.432810
1-methyl-4-[(4-methylphenyl)thio]-3-nitro-2-quinolinoneRattus norvegicus (Norway rat)Potency1.995310
4-(6-methyl-4-phenyl-2-quinazolinyl)-1-piperazinecarboxaldehydeRattus norvegicus (Norway rat)Potency15.848910
6-chloro-N4-cyclohexyl-N2-propan-2-yl-1,3,5-triazine-2,4-diamineRattus norvegicus (Norway rat)Potency31.622810
2-(8-quinolinylthio)acetic acid phenacyl esterRattus norvegicus (Norway rat)Potency89.125110
1-(3-nitrophenyl)-3-phenyl-2-propyn-1-oneRattus norvegicus (Norway rat)Potency0.100010
2-methoxy-4-[[2-(methylthio)anilino]methyl]phenolRattus norvegicus (Norway rat)Potency5.011910
2-(1-methyl-2-phenyl-3-indolyl)ethanolRattus norvegicus (Norway rat)Potency67.833420
6-ethyl-5-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-oneRattus norvegicus (Norway rat)Potency56.234110
N-(1-acetyl-2-chloro-3-indolyl)-2-chloroacetamideRattus norvegicus (Norway rat)Potency12.589310
2-(3-cyano-4,5,6-trimethyl-1H-pyridin-2-ylidene)propanedinitrileRattus norvegicus (Norway rat)Potency35.481310
N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-5-nitro-2-furancarboxamideRattus norvegicus (Norway rat)Potency79.432810
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrileRattus norvegicus (Norway rat)Potency43.928420
[5-(4-nitrophenyl)-2-furanyl]-(1-piperidinyl)methanoneRattus norvegicus (Norway rat)Potency22.387210
3-chloro-6-phenyl-[1,2,4]triazolo[4,3-b]pyridazineRattus norvegicus (Norway rat)Potency15.848910
N4,N4-dimethyl-N1-(4-nitro-1,1-dioxo-2,5-dihydrothiophen-3-yl)benzene-1,4-diamineRattus norvegicus (Norway rat)Potency0.251210
N-[4-(1-azepanyl)phenyl]-2-chloroacetamideRattus norvegicus (Norway rat)Potency56.234110
3-chloro-1-(2-chlorophenyl)-4-(4-morpholinyl)pyrrole-2,5-dioneRattus norvegicus (Norway rat)Potency0.281810
4-chloro-1-ethyl-3-nitro-2-quinolinoneRattus norvegicus (Norway rat)Potency2.511910
3-(3-nitrophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency56.234110
2-(2,4-dimethylphenyl)-5-benzotriazolamineRattus norvegicus (Norway rat)Potency79.432810
LSM-20909Rattus norvegicus (Norway rat)Potency31.622810
2-[[4-amino-2-(ethylamino)-5-thiazolyl]-phenylmethylidene]propanedinitrileRattus norvegicus (Norway rat)Potency43.928420
2-(3,4-dimethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)ethanoneRattus norvegicus (Norway rat)Potency1.258910
2-oxo-3-benzo[h][1]benzopyrancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.310620
2-furancarboxylic acid (2-acetyl-1-benzothiophen-3-yl) esterRattus norvegicus (Norway rat)Potency89.125110
5-(4-chlorophenyl)-2-furanpropionic acidRattus norvegicus (Norway rat)Potency17.782810
6-(1,3-benzoxazol-2-yl)-1,3-benzothiazol-2-amineRattus norvegicus (Norway rat)Potency31.622810
3-prop-2-enyl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-[1]benzothiolo[2,3-d]pyrimidin-4-oneRattus norvegicus (Norway rat)Potency3.981110
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneRattus norvegicus (Norway rat)Potency39.810710
2-(2,5-dimethylphenyl)-3H-benzimidazol-5-amineRattus norvegicus (Norway rat)Potency39.810720
4-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency1.995310
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideRattus norvegicus (Norway rat)Potency3.981110
(2'-(4-aminophenyl)-(2,5'-bi-1h-benzimidazol)-5-amine)Rattus norvegicus (Norway rat)Potency15.789630
3-propyl-1-(2-pyridinylmethylamino)-4-pyrido[1,2-a]benzimidazolecarbonitrileRattus norvegicus (Norway rat)Potency15.848910
N-(3-phenyl-1,3-benzothiazol-2-ylidene)-2-propenamideRattus norvegicus (Norway rat)Potency22.387210
6-(1H-benzimidazol-2-yl)-2-methyl-1H-benzimidazoleRattus norvegicus (Norway rat)Potency70.794610
2-[[4-(1-pyrrolidinylsulfonyl)phenyl]hydrazinylidene]propanedinitrileRattus norvegicus (Norway rat)Potency22.387210
10,11-dihydroxy-n-allylnoraporphineRattus norvegicus (Norway rat)Potency4.274330
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]acetamideRattus norvegicus (Norway rat)Potency28.183810
3-(1,3-dimethyl-4-pyrazolyl)-4-(2-methoxyphenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency3.162310
3-(1,3-benzodioxol-5-yl)-4-(2,5-dimethylphenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency0.562310
3-(1-benzothiophen-3-yl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency39.810710
3-(4,5-dimethyl-3-thiophenyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency8.912510
4,5-dimethyl-2-[4-(3-nitrophenyl)-2-thiazolyl]-1H-pyrazol-3-oneRattus norvegicus (Norway rat)Potency89.125110
LSM-31933Rattus norvegicus (Norway rat)Potency31.622810
6-(2-phenylethyl)-3-(phenylmethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleRattus norvegicus (Norway rat)Potency35.481310
N-(2-phenyl-6-imidazo[1,2-a]pyridinyl)acetamideRattus norvegicus (Norway rat)Potency22.387210
N-[[6-cyano-5-(ethylamino)-3-methyl-2-pyrazinyl]methyl]-N-phenylacetamideRattus norvegicus (Norway rat)Potency19.952610
isoeugenolRattus norvegicus (Norway rat)Potency5.011910
5-[2-(6-hydroxy-3-methyl-2-benzofuranyl)-2-oxoethyl]-2-furancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency31.354020
5-(3,3-dimethyl-2-oxobutoxy)-4-ethyl-7-methyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency79.432810
3-(3,4-dimethylanilino)-1-thiophen-2-yl-1-propanoneRattus norvegicus (Norway rat)Potency4.466810
5-(4-fluorophenyl)-2-thiophen-2-yloxazoleRattus norvegicus (Norway rat)Potency16.372420
2-chloro-N-[5-ethyl-3-[(4-methylphenyl)-oxomethyl]-2-thiophenyl]acetamideRattus norvegicus (Norway rat)Potency31.622810
2-(4-methoxyphenyl)-5-(3-pyridinyl)-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency29.396920
3-amino-6-cyclopropyl-4-(4-methoxyphenyl)-2-thieno[2,3-b]pyridinecarbonitrileRattus norvegicus (Norway rat)Potency19.952610
2-[[oxo(thiophen-2-yl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid propan-2-yl esterRattus norvegicus (Norway rat)Potency50.118710
(4-(3-chlorophenyl)piperazin-1-yl)(2-ethoxyphenyl)methanoneRattus norvegicus (Norway rat)Potency0.112210
N-[[(6-methyl-4-pyrimidinyl)thio]methyl]benzamideRattus norvegicus (Norway rat)Potency11.220210
2-[[anilino(oxo)methyl]amino]-4,5-dimethoxybenzoic acidRattus norvegicus (Norway rat)Potency56.234110
5-(1-methyl-2-benzimidazolyl)-2-thiophenecarboxaldehydeRattus norvegicus (Norway rat)Potency53.882020
6,7-dimethoxy-3-phenyl-1H-quinazoline-2,4-dioneRattus norvegicus (Norway rat)Potency17.782810
N-(2-methyl-1,3-dioxo-5-isoindolyl)-1-naphthalenecarboxamideRattus norvegicus (Norway rat)Potency56.234110
3-(4-bromoanilino)-1-(3-nitrophenyl)-1-propanoneRattus norvegicus (Norway rat)Potency15.848910
3-anilino-1-(3-nitrophenyl)-1-propanoneRattus norvegicus (Norway rat)Potency1.584910
4-(4-morpholinylmethyl)-3-quinolinolRattus norvegicus (Norway rat)Potency31.622810
4-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]benzoic acid ethyl esterRattus norvegicus (Norway rat)Potency31.622810
2-amino-9-ethyl-3-pyrido[2,3-b]indolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency63.095710
4-sulfanylidene-1,6,7,8,9,10-hexahydropyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrileRattus norvegicus (Norway rat)Potency10.000010
7-methoxy-4,8-dimethyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency31.622810
3-bromo-N-[(tert-butylamino)-sulfanylidenemethyl]-4-methoxybenzamideRattus norvegicus (Norway rat)Potency28.183810
N-[(3-acetylanilino)-sulfanylidenemethyl]-3-chlorobenzamideRattus norvegicus (Norway rat)Potency14.125410
4-(3-pyridinyloxy)benzene-1,2-dicarbonitrileRattus norvegicus (Norway rat)Potency1.122010
5-acetyloxy-2-[[cyclohexyl(oxo)methyl]amino]benzoic acidRattus norvegicus (Norway rat)Potency56.234110
1-(2-methylpropyl)-2-thiophen-2-ylbenzimidazoleRattus norvegicus (Norway rat)Potency56.234110
2-(3,4-dimethylphenoxy)ethanethioic acid S-(4-methylphenyl) esterRattus norvegicus (Norway rat)Potency8.912510
2-[(3-ethyl-4-methyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid methyl esterRattus norvegicus (Norway rat)Potency35.481310
N-(2-furanylmethyl)-1,3-dioxo-2-propyl-5-isoindolecarboxamideRattus norvegicus (Norway rat)Potency70.794610
5-(2-furanylmethylamino)-2-(4-methoxyphenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency72.679620
N-(2-cyano-1-cyclopentenyl)-1-ethyl-3-pyrazolecarboxamideRattus norvegicus (Norway rat)Potency25.118910
N-[(2-methoxyphenyl)methyl]-4-(1-piperidinyl)anilineRattus norvegicus (Norway rat)Potency15.848910
2-(4-methoxyphenyl)-5-(2-phenylethylamino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency49.489220
5-(4-morpholinyl)-2-thiophen-2-yl-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency41.524220
N-(2,4-dimethylphenyl)-4-(phenylmethyl)-1-piperazinecarbothioamideRattus norvegicus (Norway rat)Potency56.234110
N-[4-[[acetamido(sulfanylidene)methyl]amino]phenyl]-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency50.118710
5-amino-3-(2-methylphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.810710
6-methoxy-4-methyl-2-[(2-methylphenyl)methylthio]quinazolineRattus norvegicus (Norway rat)Potency100.000010
3-[1-(4-acetylphenyl)-5-thiophen-2-yl-2-pyrrolyl]propanoic acidRattus norvegicus (Norway rat)Potency25.787710
[2-(5-methyl-2-thiophenyl)-4-quinolinyl]-(1-pyrrolidinyl)methanoneRattus norvegicus (Norway rat)Potency79.432810
N-(3-methyl-4-oxo-1-benzopyran-2-yl)carbamic acid ethyl esterRattus norvegicus (Norway rat)Potency89.125110
2-(2-methoxyphenyl)-1H-indoleRattus norvegicus (Norway rat)Potency84.279020
1-(6,8-dimethyl-2,3-dihydropyrrolo[2,3-g]quinolin-1-yl)ethanoneRattus norvegicus (Norway rat)Potency56.234110
3-(3,5-dimethyl-7-oxo-6-furo[3,2-g][1]benzopyranyl)propanoic acidRattus norvegicus (Norway rat)Potency79.432810
deltoinRattus norvegicus (Norway rat)Potency31.622810
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneRattus norvegicus (Norway rat)Potency57.457020
5-hydroxy-2-[[(4-methylphenyl)thio]methyl]-3-benzofurancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency3.548110
3-[2-methoxy-6-(4-methoxyphenyl)-3-pyridinyl]-5-(methoxymethyl)-1,2,4-oxadiazoleRattus norvegicus (Norway rat)Potency39.310620
4-chloro-N-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]benzamideRattus norvegicus (Norway rat)Potency1.995310
1-ethyl-3-(4-methylphenyl)sulfonylthioureaRattus norvegicus (Norway rat)Potency15.848910
7-methoxy-2-oxo-1-benzopyran-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency57.731520
2-(4-chlorophenyl)-4-propan-2-yloxyquinazolineRattus norvegicus (Norway rat)Potency89.125110
7,8-dichloropyrido[1,2-a]benzimidazoleRattus norvegicus (Norway rat)Potency15.848910
2-(2-furanyl)-3-(4-methylphenyl)imidazo[4,5-b]quinoxalineRattus norvegicus (Norway rat)Potency39.810710
1-(cycloheptylideneamino)-3-(4-fluorophenyl)thioureaRattus norvegicus (Norway rat)Potency1.122010
4-methoxy-N-[[(phenylmethyl)amino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency22.387210
7-acetoxycoumarinRattus norvegicus (Norway rat)Potency76.110420
2-(2-cyclohexylidenehydrazinyl)-1-cyclohepta-2,4,6-trienoneRattus norvegicus (Norway rat)Potency70.794610
2-(2-fluorophenyl)-5-(4-methyl-1-piperidinyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency84.279020
5-(2-furanylmethylamino)-2-(3-methylphenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency22.387210
8-(9-methyl-5H-pyrimido[5,4-b]indol-4-yl)-1,4-dioxa-8-azaspiro[4.5]decaneRattus norvegicus (Norway rat)Potency79.432810
1-methyl-5-(1-naphthalenyloxy)-4-nitroimidazoleRattus norvegicus (Norway rat)Potency8.912510
3-(isopropylideneamino)-2,2-dimethyl-2,3-dihydroquinazolin-4(1h)-oneRattus norvegicus (Norway rat)Potency17.782810
3-amino-4-thiophen-2-yl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency44.668410
2-(2-fluorophenyl)-5-(4-methoxyanilino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency31.622810
3-[5-(2-furanyl)-1H-pyrazol-3-yl]-4-(2-methoxyphenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency44.668410
N-[[(phenylmethyl)amino]-sulfanylidenemethyl]-1,3-benzodioxole-5-carboxamideRattus norvegicus (Norway rat)Potency17.782810
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-3-methylbenzamideRattus norvegicus (Norway rat)Potency28.183810
terazosinRattus norvegicus (Norway rat)Potency76.110420
curcuminRattus norvegicus (Norway rat)Potency50.118710
2-[[(4-methyl-1-pyrazolyl)-oxomethyl]amino]benzoic acid methyl esterRattus norvegicus (Norway rat)Potency63.095710
1-(4-methoxyphenyl)-3-(6-quinoxalinyl)thioureaRattus norvegicus (Norway rat)Potency15.848910
3-[(2-ethyl-1-oxobutyl)amino]-N-(2-furanylmethyl)benzamideRattus norvegicus (Norway rat)Potency19.952610
1-(1-pyrrolidinyl)-2-(8-quinolinylthio)ethanoneRattus norvegicus (Norway rat)Potency16.082520
2-(methanesulfonamido)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency70.794610
1-(4-bromophenyl)-3-(2-fluorophenyl)thioureaRattus norvegicus (Norway rat)Potency14.125410
7-amino-2-(4-tert-butylphenyl)-6-pyrazolo[1,5-a]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency0.141310
3-tert-butyl-7-[[2-(4-methylphenyl)-2-oxoethyl]thio]-[1,3,4]thiadiazolo[2,3-c][1,2,4]triazin-4-oneRattus norvegicus (Norway rat)Potency1.995310
N-[(3-bromo-4-ethoxy-5-methoxyphenyl)methyl]-2,3-dihydro-1,4-benzodioxin-6-amineRattus norvegicus (Norway rat)Potency3.981110
N-[(1-ethyl-2-oxo-6-benzo[cd]indolyl)sulfonyl]-N-(4-methoxyphenyl)-3-pyridinecarboxamideRattus norvegicus (Norway rat)Potency89.125120
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideRattus norvegicus (Norway rat)Potency56.234110
3-[(4-benzoyl-1-piperazinyl)-oxomethyl]-8-methoxy-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency6.309610
umi-77Rattus norvegicus (Norway rat)Potency22.387210
4-[(2-bromophenoxy)methyl]-N-[4-[(3,5-dimethyl-1-pyrazolyl)methyl]phenyl]benzamideRattus norvegicus (Norway rat)Potency56.234110
1-[[[2-(difluoromethoxy)phenyl]-oxomethyl]amino]-3-(4-fluorophenyl)thioureaRattus norvegicus (Norway rat)Potency63.095710
N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-(3-methyl-N-methylsulfonylanilino)acetamideRattus norvegicus (Norway rat)Potency50.118710
2-[(3-cyano-4-phenyl-6-thiophen-2-yl-2-pyridinyl)thio]-N-propan-2-ylacetamideRattus norvegicus (Norway rat)Potency84.279020
2-[9-(4-methoxyphenyl)-1,8-dioxo-3,4,5,6,7,9-hexahydro-2H-acridin-10-yl]acetic acidRattus norvegicus (Norway rat)Potency56.234110
2-[(5-bromo-2-thiophenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideRattus norvegicus (Norway rat)Potency39.810710
N-[[3-(hydroxymethyl)anilino]-sulfanylidenemethyl]-4-phenylbenzamideRattus norvegicus (Norway rat)Potency17.782810
N-[(3-acetylanilino)-sulfanylidenemethyl]-5-bromo-3-pyridinecarboxamideRattus norvegicus (Norway rat)Potency22.387210
4-[[[[oxo-(4-phenylphenyl)methyl]amino]-sulfanylidenemethyl]amino]benzoic acidRattus norvegicus (Norway rat)Potency15.848910
2-(1,3-dimethyl-2,6-dioxo-9-purinyl)-N-[2-(4-morpholinyl)-5-(trifluoromethyl)phenyl]acetamideRattus norvegicus (Norway rat)Potency0.141310
3,4-dimethoxy-N-[[4-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency3.981110
4-[[4-bromo-5-(4-morpholinyl)-2-furanyl]methylideneamino]phenolRattus norvegicus (Norway rat)Potency31.622810
N-[3-[oxo-(3-pyridinylmethylamino)methyl]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency22.387210
5-ethyl-2-[[oxo-(3,4,5-trimethoxyphenyl)methyl]amino]-3-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency34.411720
N-[[3-chloro-4-(4-morpholinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency44.668410
2-[3-(4-methoxyphenyl)-1-benzo[f]quinolinyl]acetic acid ethyl esterRattus norvegicus (Norway rat)Potency25.118910
rhi002Rattus norvegicus (Norway rat)Potency44.668410
4-[[[2,3-bis(2-pyridinyl)-6-quinoxalinyl]amino]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency56.234110
1-[(4-fluorophenyl)methyl]-4-(3,4,5-trimethoxyphenyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency63.095710
1-[(4-methylphenyl)methyl]-4-(3,4,5-trimethoxyphenyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency44.668410
1-cyclopropyl-4-[4-(trifluoromethyl)phenyl]-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency19.952610
N-cyclopentyl-2-imino-1-[3-(4-morpholinyl)propyl]-5-oxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency22.387210
N-[(2-chlorophenyl)methyl]-1-(4-methylphenyl)sulfonyl-4-piperidinecarboxamideRattus norvegicus (Norway rat)Potency0.354810
N-[2-[2-[2-(4-ethoxyanilino)-2-oxoethyl]-5-tetrazolyl]phenyl]-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency50.118710
N-[2-(2-pyridinyl)-3H-benzimidazol-5-yl]cyclohexanecarboxamideRattus norvegicus (Norway rat)Potency15.848910
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N,N-diethylacetamideRattus norvegicus (Norway rat)Potency11.220210
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency70.794610
2-(2,4,5-trimethoxyphenyl)-1,3-benzothiazoleRattus norvegicus (Norway rat)Potency50.118710
5-(4-bromophenyl)-2-phenyl-7-pyrazolo[1,5-a]pyrimidinamineRattus norvegicus (Norway rat)Potency0.631010
N-(3-methylphenyl)-4-tetrazolo[1,5-a]quinoxalinamineRattus norvegicus (Norway rat)Potency79.432810
[7-(difluoromethyl)-5-(4-methoxyphenyl)-3-pyrazolo[1,5-a]pyrimidinyl]-(1-piperidinyl)methanoneRattus norvegicus (Norway rat)Potency15.848910
2-(4-methylphenoxy)-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]acetamideRattus norvegicus (Norway rat)Potency12.589310
1-[(3,4-dimethoxyphenyl)methyl]-4-(4-hydroxyphenyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency59.621820
N-[2,2-dichloro-1-(4-chlorophenyl)sulfonylethenyl]benzamideRattus norvegicus (Norway rat)Potency44.668410
N-(2-furanylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency42.800020
N-(2-furanylmethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency44.668410
2-[[[3-[2-(4-methylphenyl)sulfonylethylthio]phenyl]-oxomethyl]amino]benzoic acidRattus norvegicus (Norway rat)Potency28.183810
2-[N-(benzenesulfonyl)-4-ethoxyanilino]-N-(2-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency100.000010
2-(2-methylphenoxy)-N-[2-(4-methylphenyl)-5-benzotriazolyl]acetamideRattus norvegicus (Norway rat)Potency79.432810
5-(3,4-dimethoxyphenyl)-N-(2-furanylmethyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency70.794610
6-(4,5-dihydrothiazol-2-ylthio)-N2,N4-bis(2-methylphenyl)-1,3,5-triazine-2,4-diamineRattus norvegicus (Norway rat)Potency1.000010
2-[[3-cyano-6-(4-methoxyphenyl)-4-phenyl-2-pyridinyl]thio]-N-(5-methyl-2-thiazolyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
[2-methoxy-4-(methylthio)phenyl]-[4-(phenylmethyl)-1-piperidinyl]methanoneRattus norvegicus (Norway rat)Potency0.188920
5-bromo-N-[3-(2-oxo-1-benzopyran-3-yl)phenyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency35.481310
2-[9-(3-chloro-4-methoxyphenyl)-1,8-dioxo-3,4,5,6,7,9-hexahydro-2H-acridin-10-yl]acetic acidRattus norvegicus (Norway rat)Potency72.679620
2-(4-methoxyphenyl)-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]acetamideRattus norvegicus (Norway rat)Potency8.912510
LSM-16774Rattus norvegicus (Norway rat)Potency56.234110
2-[[5-(1-benzotriazolylmethyl)-4-methyl-1,2,4-triazol-3-yl]thio]-1-(2-fluorophenyl)ethanoneRattus norvegicus (Norway rat)Potency44.668410
3-[[4-(1,3-benzodioxol-5-yl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(2-furanylmethyl)propanamideRattus norvegicus (Norway rat)Potency63.095710
2-(6-amino-2-methyl-4-oxo-3-quinazolinyl)-N-(2-methylphenyl)acetamideRattus norvegicus (Norway rat)Potency25.118910
6-amino-3-[(2-chlorophenyl)methyl]-2-propyl-4-quinazolinoneRattus norvegicus (Norway rat)Potency35.481310
N-(2-furanylmethyl)-2-(4-oxo-6-phenyl-3-thieno[2,3-d]pyrimidinyl)acetamideRattus norvegicus (Norway rat)Potency31.622810
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterRattus norvegicus (Norway rat)Potency2.818410
3-chloro-4-[2-(3,4-dimethoxyphenyl)ethylamino]-1-(2-phenylethyl)pyrrole-2,5-dioneRattus norvegicus (Norway rat)Potency25.118910
N-(2-ethylphenyl)-2-[[2-(4-methoxyphenyl)-4-oxo-1-benzopyran-6-yl]oxy]acetamideRattus norvegicus (Norway rat)Potency15.848910
2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)acetamideRattus norvegicus (Norway rat)Potency19.952610
10-(4-methoxyphenyl)-3,4,5,6,7,9-hexahydro-2H-acridine-1,8-dioneRattus norvegicus (Norway rat)Potency35.481310
3-methoxy-4-(2-methoxy-3-methoxycarbonyl-1-naphthalenyl)-2-naphthalenecarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency31.622820
N-(2-phenylethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideRattus norvegicus (Norway rat)Potency28.934220
3-imino-2-benzo[f][1]benzopyrancarbothioamideRattus norvegicus (Norway rat)Potency78.117120
5-(2,4-dichlorophenyl)-N-(4-methyl-2-thiazolyl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency89.125110
5-(4-fluorophenyl)sulfonyl-1-(2-methylpropyl)-4-nitro-2-propan-2-ylimidazoleRattus norvegicus (Norway rat)Potency0.891310
1-benzimidazolyl-[2-(4-methoxyphenyl)-4-quinolinyl]methanoneRattus norvegicus (Norway rat)Potency28.183810
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[5-[(4-chlorophenoxy)methyl]-2-furanyl]methanoneRattus norvegicus (Norway rat)Potency31.622810
2',4',6'-TrihydroxydihydrochalconeRattus norvegicus (Norway rat)Potency19.952610
7-anilino-1-(4-methylphenyl)-5-oxo-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency10.000010
LSM-16526Rattus norvegicus (Norway rat)Potency12.380720
3,5-dimethoxy-N-[(2-phenylethylamino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency39.810710
2-[[(5-ethyl-2-thiophenyl)-oxomethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency19.952610
2-(2-fluorophenyl)-4-(4-fluorophenyl)sulfonyl-5-(1-piperidinyl)oxazoleRattus norvegicus (Norway rat)Potency50.118710
N-(2-carbamoylphenyl)-4-ethyl-5-methyl-3-thiophenecarboxamideRattus norvegicus (Norway rat)Potency25.118910
N-(2-furanylmethyl)-5-methyl-4-phenyl-3-thiophenecarboxamideRattus norvegicus (Norway rat)Potency14.125410
2-benzamido-4,5-dihydrobenzo[g][1]benzothiole-3-carboxamideRattus norvegicus (Norway rat)Potency79.432810
LSM-33266Rattus norvegicus (Norway rat)Potency39.810710
3-[[[4-(4-methoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]methyl]benzoic acidRattus norvegicus (Norway rat)Potency89.125110
LSM-28559Rattus norvegicus (Norway rat)Potency50.118710
N-(3,5-dichlorophenyl)-2-(methanesulfonamido)benzamideRattus norvegicus (Norway rat)Potency9.698520
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamideRattus norvegicus (Norway rat)Potency79.432810
7-(2-oxopropoxy)-3-phenyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency35.481310
2-thioxantheneRattus norvegicus (Norway rat)Potency1.778310
2,6-dithiopurineRattus norvegicus (Norway rat)Potency5.011910
5-(4-ethylbenzylidene)-2-thioxothiazolidin-4-oneRattus norvegicus (Norway rat)Potency39.985040
4-(5-methyl-2-furanyl)-2-[[2-(4-morpholinyl)-1-oxoethyl]amino]-3-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.810710
N-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamideRattus norvegicus (Norway rat)Potency11.220210
N-[[2-methyl-5-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency70.794610
2-[[(3,4-dimethoxyphenyl)-oxomethyl]amino]-N-(2-furanylmethyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideRattus norvegicus (Norway rat)Potency39.810710
N-(2-furanylmethyl)-2-imino-5-oxo-1-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency79.432810
2,4-dimethyl-N-[[4-(4-morpholinyl)anilino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency39.810710
2-(1,3-benzodioxol-5-ylmethylthio)-5-(2-furanyl)-3-prop-2-enyl-4-thieno[2,3-d]pyrimidinoneRattus norvegicus (Norway rat)Potency50.118710
2-(4-chlorophenyl)-N-[[2-(4-morpholinyl)anilino]-sulfanylidenemethyl]acetamideRattus norvegicus (Norway rat)Potency12.589310
2-[[5-[(2-methyl-8-quinolinyl)oxymethyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]acetamideRattus norvegicus (Norway rat)Potency79.432810
N-[4-[4-(ethylsulfonylamino)-3-methoxyphenyl]-2-methoxyphenyl]ethanesulfonamideRattus norvegicus (Norway rat)Potency56.234110
2-(4-methoxyphenyl)-N-[4-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideRattus norvegicus (Norway rat)Potency17.782810
3-(2,3-dimethyl-1H-indol-5-yl)-4-(3-methoxyphenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency14.125410
1-[2-(difluoromethoxy)-4-methylphenyl]-3-(2,4-difluorophenyl)ureaRattus norvegicus (Norway rat)Potency7.079510
4-[[2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterRattus norvegicus (Norway rat)Potency89.125110
N-[(3,5-dimethoxyanilino)-sulfanylidenemethyl]-3-phenylpropanamideRattus norvegicus (Norway rat)Potency35.481310
4-(5-amino-4-phenyl-1-pyrazolyl)benzoic acidRattus norvegicus (Norway rat)Potency100.000010
5-bromo-N-[[(3-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideRattus norvegicus (Norway rat)Potency31.622810
2-(1-naphthalenyl)-N-(2-phenyl-1,3-benzoxazol-5-yl)acetamideRattus norvegicus (Norway rat)Potency63.095720
N-cyclohexyl-2-[(8-methoxy-6-oxo-3-benzo[c][1]benzopyranyl)oxy]acetamideRattus norvegicus (Norway rat)Potency17.782810
2-imino-10-methyl-N-[2-(4-morpholinyl)ethyl]-5-oxo-1-(3-pyridinylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency61.193620
5-methyl-4-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxymethyl]-2-furancarboxylic acidRattus norvegicus (Norway rat)Potency44.668410
2-[[(4-bromo-1-ethyl-3-pyrazolyl)-oxomethyl]amino]-4-phenyl-3-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency35.481310
darunavir ethanolateRattus norvegicus (Norway rat)Potency19.952610
5-bromo-N-[(2-carbamoylanilino)-sulfanylidenemethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency25.118910
5-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxymethyl]-2-furancarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency17.559420
4-methyl-3-(phenylmethyl)-7-[(3,4,5-trimethoxyphenyl)methoxy]-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency47.393620
2-chloro-5-[[[[(3,5-dimethoxyphenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]benzoic acidRattus norvegicus (Norway rat)Potency7.943310
N-(2-furanylmethyl)-2-[[oxo-(3,4,5-trimethoxyphenyl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideRattus norvegicus (Norway rat)Potency44.668410
[2-(4-methoxyphenyl)-6-methyl-4-quinolinyl]-(4-morpholinyl)methanoneRattus norvegicus (Norway rat)Potency28.183810
1-[2,3-bis(2-furanyl)-6-quinoxalinyl]-3-[4-(4-morpholinyl)phenyl]thioureaRattus norvegicus (Norway rat)Potency2.511910
5-(3,3-dimethyl-2-oxobutoxy)-3,4,7-trimethyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency79.432810
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-(2-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency25.118910
3-(3-oxo-2-benzo[f][1]benzopyranyl)-1-phenyl-4-pyrazolecarboxaldehydeRattus norvegicus (Norway rat)Potency3.981110
7-[4-(4-acetamidophenyl)sulfonyl-1-piperazinyl]-1-ethyl-6-fluoro-4-oxo-3-quinolinecarboxylic acidRattus norvegicus (Norway rat)Potency79.432810
5-bromo-N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency44.668410
N-(2-phenyl-5-benzotriazolyl)-2,3-dihydro-1,4-benzodioxin-6-carboxamideRattus norvegicus (Norway rat)Potency35.481310
2-benzo[b][1]benzoxepinamineRattus norvegicus (Norway rat)Potency39.810710
3-(3,4-dimethoxyphenyl)-7-(2-oxopropoxy)-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency100.000010
Methyl 7-methoxycoumarin-4-acetateRattus norvegicus (Norway rat)Potency44.668410
3-[[3-(4-morpholinyl)-1,4-dioxo-2-naphthalenyl]amino]benzoic acidRattus norvegicus (Norway rat)Potency79.432810
3-(4-methoxyphenyl)-2,4-dihydrothiazolo[3,2-a][1,3,5]triazin-6-oneRattus norvegicus (Norway rat)Potency35.481310
1-(2-fluorophenyl)-3-[5-(2-fluorophenyl)-1,3,4-thiadiazol-2-yl]ureaRattus norvegicus (Norway rat)Potency89.125110
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzothiazoleRattus norvegicus (Norway rat)Potency56.234110
1-(3,4-dihydroxyphenyl)-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneRattus norvegicus (Norway rat)Potency79.432810
2-(4-fluorophenoxy)-N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)acetamideRattus norvegicus (Norway rat)Potency39.810710
N-(1,3-benzodioxol-5-yl)-4-methyl-1-phthalazinamineRattus norvegicus (Norway rat)Potency3.548110
3-bromo-5-[[4-[hydroxy(diphenyl)methyl]-1-piperidinyl]-oxomethyl]-2-pyranoneRattus norvegicus (Norway rat)Potency25.118910
N-(4-methoxyphenyl)-2-(3-nitrophenyl)-4-quinazolinamineRattus norvegicus (Norway rat)Potency2.511910
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-propan-2-yl-2-furancarboxamideRattus norvegicus (Norway rat)Potency56.234110
2-[[5-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-ethyl-1,3,4-thiadiazol-2-yl)acetamideRattus norvegicus (Norway rat)Potency15.848910
2-[[5-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-[4-(1-pyrrolidinylsulfonyl)phenyl]acetamideRattus norvegicus (Norway rat)Potency79.432810
4-[[3-[(2-chlorophenyl)methyl]-5-cyclopropyl-7-triazolo[4,5-d]pyrimidinyl]amino]-N,N-dimethylbenzenesulfonamideRattus norvegicus (Norway rat)Potency34.487420
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency19.952610
7-methyl-2-[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]-3-quinolinecarbonitrileRattus norvegicus (Norway rat)Potency63.514420
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-phenylethyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
N',2-dimethyl-N'-[3-(trifluoromethyl)-2-quinoxalinyl]benzohydrazideRattus norvegicus (Norway rat)Potency0.177810
2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]-7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency50.118720
2-[benzenesulfonyl(2-pyridinyl)amino]acetic acidRattus norvegicus (Norway rat)Potency56.234110
2-[(4-chlorophenyl)sulfonyl-(2-pyridinyl)amino]acetic acidRattus norvegicus (Norway rat)Potency70.794610
6-(4-fluorophenyl)-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency22.387210
4-[5-(carboxymethyl)-4-phenyl-2-thiazolyl]benzoic acidRattus norvegicus (Norway rat)Potency25.118910
3-[5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazol-2-yl]-1-(phenylmethyl)-2-pyridinoneRattus norvegicus (Norway rat)Potency30.300120
5-(6-chloro-3-pyridinyl)-3-(3-methoxyphenyl)-1,2,4-oxadiazoleRattus norvegicus (Norway rat)Potency10.000010
4-(2,6-dimethylphenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidineRattus norvegicus (Norway rat)Potency89.125110
N-[2,5-dioxo-6-(4-phenoxyphenyl)-3-pyrano[3,2-c]pyridinyl]benzamideRattus norvegicus (Norway rat)Potency35.481310
5-[1-[(4-methylphenyl)methyl]-3-pyrazolyl]-2-phenylthiazoleRattus norvegicus (Norway rat)Potency27.005020
5-[1-[(4-fluorophenyl)methyl]-3-pyrazolyl]-2-phenylthiazoleRattus norvegicus (Norway rat)Potency33.552020
4-(4-chlorophenyl)sulfinyl-6-(methoxymethyl)-2-methylpyrimidineRattus norvegicus (Norway rat)Potency14.125410
6-(4-methyl-1-piperazinyl)-2-(3,4,5-trimethoxyphenyl)-1H-benzimidazoleRattus norvegicus (Norway rat)Potency26.651420
4-(4-chlorophenyl)-1-(6-fluoro-2-pyridinyl)-3-pyrazolamineRattus norvegicus (Norway rat)Potency15.848910
6-tert-butyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency39.810710
7-(4-chlorophenyl)-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]-[1,2,4]triazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency39.810710
4-chloro-6-(4-methoxyphenyl)-2-phenyl-5-pyrimidinecarbonitrileRattus norvegicus (Norway rat)Potency70.794610
2-(4-methylsulfonylphenyl)-6-imidazo[1,2-a]pyridinecarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency19.952610
2-(methylthio)-7-(4-phenylphenyl)-[1,2,4]triazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency21.712320
5-[3-[(2,4-dichlorophenyl)methoxy]-2-thiophenyl]-1,2-dihydro-1,2,4-triazole-3-thioneRattus norvegicus (Norway rat)Potency19.952610
2-(benzenesulfonylmethyl)-5-(4-chlorophenyl)cyclohexane-1,3-dioneRattus norvegicus (Norway rat)Potency25.118910
N,N-dimethylcarbamic acid [4-[2-(benzenesulfonyl)-1-oxoethyl]-2,6-dimethylphenyl] esterRattus norvegicus (Norway rat)Potency56.234110
3-(5-chloro-1,3-benzoxazol-2-yl)-N-(phenylmethyl)-2-pyridinamineRattus norvegicus (Norway rat)Potency30.300120
2-(6-chloro-3-pyridinyl)-1H-benzimidazoleRattus norvegicus (Norway rat)Potency22.387210
2-[(2,4-dichlorophenyl)methylthio]-6,7-dimethoxy-3-(thiophen-2-ylmethyl)-4-quinazolinimineRattus norvegicus (Norway rat)Potency0.281810
5-cyano-2-phenyl-6-[4-(2-pyridinyl)-1-piperazinyl]-3-pyridinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency31.622810
6-methyl-5-[2-(2-methylphenoxy)ethyl]-2-sulfanylidene-1H-pyrimidin-4-oneRattus norvegicus (Norway rat)Potency15.848910
4-[1-[(3-methoxyphenyl)methyl]-2-benzimidazolyl]-1,2,5-oxadiazol-3-amineRattus norvegicus (Norway rat)Potency12.589310
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-oneRattus norvegicus (Norway rat)Potency25.118910
4-methoxy-N-(8-methyl-[1,3]dioxolo[4,5-g]quinazolin-6-yl)benzamideRattus norvegicus (Norway rat)Potency89.125120
3-(benzenesulfonyl)-2-imino-1-propyl-5-dipyrido[1,2-d-3',4'-f]pyrimidinoneRattus norvegicus (Norway rat)Potency22.387210
N-[2-[(phenylmethyl)amino]-1,3-benzodioxol-2-yl]carbamic acid ethyl esterRattus norvegicus (Norway rat)Potency31.622810
1-[[2-[[4-(4-chlorophenyl)-5-phenyl-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-3-phenylthioureaRattus norvegicus (Norway rat)Potency8.912510
cinnarizineRattus norvegicus (Norway rat)Potency0.354810
2-[[[4-(diethylsulfamoyl)phenyl]-oxomethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency50.118710
sulindacRattus norvegicus (Norway rat)Potency35.481310
sulindacRattus norvegicus (Norway rat)Potency26.679520
fluoxetineRattus norvegicus (Norway rat)Potency0.446710
cysteine sulfinic acidRattus norvegicus (Norway rat)Potency18.887610
1,4-benzoquinone guanylhydrazone thiosemicarbazoneRattus norvegicus (Norway rat)Potency19.952610
cyqualonRattus norvegicus (Norway rat)Potency35.035610
1-[[2-(1,3-benzothiazol-2-ylthio)-1-oxoethyl]amino]-3-phenylthioureaRattus norvegicus (Norway rat)Potency11.220210
6-(1,3-dioxo-2-isoindolyl)hexanoic acid (4-methyl-2-oxo-1-benzopyran-7-yl) esterRattus norvegicus (Norway rat)Potency28.183810
3-chloro-1-(2,4-dimethylphenyl)-4-(2-hydroxyethylamino)pyrrole-2,5-dioneRattus norvegicus (Norway rat)Potency70.794610
2-(4-chlorophenyl)-5-(prop-2-enylamino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency56.234110
N-[[4-[(5-ethyl-1,3,4-thiadiazol-2-yl)sulfamoyl]anilino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency28.183810
1-(4-fluorophenyl)-7-(4-methylphenyl)-5,5-bis(trifluoromethyl)-8H-pyrimido[4,5-d]pyrimidine-2,4-dioneRattus norvegicus (Norway rat)Potency94.562620
2-chloro-N-heptyl-N-(3-methylphenyl)acetamideRattus norvegicus (Norway rat)Potency39.810710
2-chloro-4,6-diphenyl-5-pyrimidinamineRattus norvegicus (Norway rat)Potency25.118910
4-(5-formyl-2-furanyl)benzoic acid propyl esterRattus norvegicus (Norway rat)Potency38.145620
ac 55649Rattus norvegicus (Norway rat)Potency31.622820
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneRattus norvegicus (Norway rat)Potency17.782810
N-[4-[[(1-oxohexylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency11.220210
3-(5,8-dinitro-1,3-dioxo-2-benzo[de]isoquinolinyl)benzoic acidRattus norvegicus (Norway rat)Potency11.220210
fm19g11Rattus norvegicus (Norway rat)Potency14.125410
N-[3-(dimethylamino)propyl]-9H-carbazole-3-carboxamideRattus norvegicus (Norway rat)Potency44.668410
N-(3-phenylpropyl)methanesulfonamideRattus norvegicus (Norway rat)Potency3.548110
1-[2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]-1-oxoethyl]-4-phenyl-4-piperidinecarboxylic acidRattus norvegicus (Norway rat)Potency56.234110
5-[(4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl)oxymethyl]-2-furancarboxylic acidRattus norvegicus (Norway rat)Potency15.848910
1-ethyl-3-[[[2-(2-methylpropyl)-4-quinolinyl]-oxomethyl]amino]thioureaRattus norvegicus (Norway rat)Potency19.952610
umbellipreninRattus norvegicus (Norway rat)Potency63.095710
4-[[[1-oxo-2-[(2-oxo-3-phenyl-1-benzopyran-7-yl)oxy]ethyl]amino]methyl]-1-cyclohexanecarboxylic acidRattus norvegicus (Norway rat)Potency24.702820
3-bromo-4-methoxy-N-[(propan-2-ylamino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency10.000010
4-(1-benzotriazolyl)-3,5-dinitrobenzonitrileRattus norvegicus (Norway rat)Potency15.848910
5-bromo-N-(2-fluorophenyl)-6-oxo-3-pyrancarboxamideRattus norvegicus (Norway rat)Potency28.183810
4-(2,5-dimethoxyphenyl)-3-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency44.668410
5-tert-butyl-3-(4-chlorophenyl)-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineRattus norvegicus (Norway rat)Potency85.894320
N-[[(5-chloro-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency10.000010
9-methoxy-6-[(4-methoxyphenyl)methyl]indolo[3,2-b]quinoxalineRattus norvegicus (Norway rat)Potency10.000010
6-chloro-5,7-dimethyl-N-(thiophen-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineRattus norvegicus (Norway rat)Potency19.952610
N-[[(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-5-methyl-3-phenyl-4-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency4.466810
2-[3-(2-furanylmethyl)-2,4-dioxo-6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-b]pyrimidin-1-yl]acetamideRattus norvegicus (Norway rat)Potency28.183810
4,5-dichloro-2-methyl-1-(2-phenoxyethyl)imidazoleRattus norvegicus (Norway rat)Potency5.623410
N-(9-ethyl-3-carbazolyl)-2-[[4-ethyl-5-(2-furanyl)-1,2,4-triazol-3-yl]thio]acetamideRattus norvegicus (Norway rat)Potency2.818410
tg 003Rattus norvegicus (Norway rat)Potency18.887620
amn082Rattus norvegicus (Norway rat)Potency1.000010
2-amino-4-[[2-(4-bromophenyl)-2-oxoethyl]thio]-3-azaspiro[5.5]undeca-1,4-diene-1,5-dicarbonitrileRattus norvegicus (Norway rat)Potency89.125110
2-amino-1-[2-(4-morpholinyl)ethyl]-3-pyrrolo[3,2-b]quinoxalinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency25.118910
2-amino-1-[2-(4-morpholinyl)ethyl]-N-prop-2-enyl-3-pyrrolo[3,2-b]quinoxalinecarboxamideRattus norvegicus (Norway rat)Potency22.387210
4-[[3-[(2-methoxyanilino)-oxomethyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidRattus norvegicus (Norway rat)Potency39.810710
2-(2-furanyl)-3,5-dimethyl-4-oxido-6-phenylpyrazin-1-ium 1-oxideRattus norvegicus (Norway rat)Potency28.183810
6-chloro-4-phenyl-2-(prop-2-enylthio)quinazolineRattus norvegicus (Norway rat)Potency28.183810
1-[2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl]-3-phenylureaRattus norvegicus (Norway rat)Potency79.432810
1-[[(4-ethoxyanilino)-sulfanylidenemethyl]amino]-3-[3-(trifluoromethyl)phenyl]thioureaRattus norvegicus (Norway rat)Potency31.622810
N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamideRattus norvegicus (Norway rat)Potency53.176420
3-[(6-methyl-4-phenyl-2-quinazolinyl)amino]-1-propanolRattus norvegicus (Norway rat)Potency89.125110
5-[(6-hydroxy-4-oxo-1-benzopyran-3-yl)methylidene]-1,3-diazinane-2,4,6-trioneRattus norvegicus (Norway rat)Potency17.782810
3-amino-N-(2-fluorophenyl)-6-(2-furanyl)-2-thieno[2,3-b]pyridinecarboxamideRattus norvegicus (Norway rat)Potency4.466810
2-[5-(4-chlorophenyl)-1,3,5-dithiazinan-2-ylidene]-2-diethoxyphosphorylacetonitrileRattus norvegicus (Norway rat)Potency12.589310
2-(4-fluorophenyl)-3-(2-furanylmethyl)-10-methylpyrimido[4,5-b]quinoline-4,5-dioneRattus norvegicus (Norway rat)Potency15.848910
4-(2,5-dimethoxyphenyl)-3-(3-phenyl-1H-pyrazol-5-yl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)Potency50.118710
5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidineRattus norvegicus (Norway rat)Potency56.234110
LSM-20401Rattus norvegicus (Norway rat)Potency17.782810
2-amino-N-(3-ethoxypropyl)-1-(4-sulfamoylphenyl)-3-pyrrolo[3,2-b]quinoxalinecarboxamideRattus norvegicus (Norway rat)Potency2.818410
N-[5-methyl-2-(4-methylphenyl)-3-pyrazolyl]-2-[(7-methyl-4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-9-yl)oxy]acetamideRattus norvegicus (Norway rat)Potency50.118710
5-tert-butyl-2-methyl-3-phenyl-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineRattus norvegicus (Norway rat)Potency89.125110
3,4-dimethoxy-N-[[[oxo(2-pyrazinyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency56.234110
4-methoxybenzoic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency94.562620
3-methoxy-N-[[(2-oxo-1-benzopyran-6-yl)amino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency10.000010
4,6-dimethyl-2-[3-(4-morpholinyl)propylamino]-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency50.118710
4-bromobenzoic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency15.848910
N-[2-(3,4-dimethoxyphenyl)ethyl]-8-ethoxy-5H-pyrimido[5,4-b]indol-4-amineRattus norvegicus (Norway rat)Potency35.481310
2-benzofurancarboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency37.646020
2-tert-butyl-4-[(4-chlorophenyl)thio]-5-methyl-1H-pyrazol-3-oneRattus norvegicus (Norway rat)Potency50.118710
(4,7-dichloro-1,3-benzothiazol-2-yl)hydrazineRattus norvegicus (Norway rat)Potency70.794610
4-(4-chlorophenyl)-1-(2-methoxyethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency28.183810
4-(3,4-dimethoxyphenyl)-1-(2-methoxyethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency44.668410
2-[[(4-bromo-1-ethyl-3-pyrazolyl)-oxomethyl]amino]-4,5-dimethyl-3-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency32.983820
1-(3-chlorophenyl)-3-(thiophen-2-ylmethyl)thioureaRattus norvegicus (Norway rat)Potency1.412510
3-(4-methylphenyl)sulfonylpropanoic acid [2-[(3,5-dichloro-2-pyridinyl)amino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency79.432810
3-[3-[[2-oxo-2-(1,2,5-trimethyl-3-pyrrolyl)ethyl]thio]propyl]-1H-benzimidazol-2-oneRattus norvegicus (Norway rat)Potency17.782810
N-(4,5-dihydrothiazol-2-yl)-2-thiophen-2-yl-4-quinolinecarboxamideRattus norvegicus (Norway rat)Potency56.234110
2-(4-methoxyphenyl)-4-quinolinecarboxylic acid [2-oxo-2-(propan-2-ylamino)ethyl] esterRattus norvegicus (Norway rat)Potency62.050620
2-(2-furanyl)-4-quinolinecarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency10.300620
3-methyl-2-benzo[g]benzofurancarboxylic acid [2-[N-(2-cyanoethyl)anilino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency70.794610
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideRattus norvegicus (Norway rat)Potency44.668410
1-[4-(benzenesulfonyl)-1-piperazinyl]-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]ethanoneRattus norvegicus (Norway rat)Potency0.281810
2-chloro-1-[2,5-dimethyl-1-(5-methyl-3-isoxazolyl)-3-pyrrolyl]ethanoneRattus norvegicus (Norway rat)Potency70.794610
2-chloro-N-[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]acetamideRattus norvegicus (Norway rat)Potency44.668410
1-cyclopropyl-7-[4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-1-piperazinyl]-6-fluoro-4-oxo-3-quinolinecarboxylic acidRattus norvegicus (Norway rat)Potency39.810710
2-[7-chloro-2,3-dioxo-4-(phenylmethyl)-1-quinoxalinyl]-N-(3-fluorophenyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
3-(4-methoxyphenyl)-1-phenyl-4-pyrazolamineRattus norvegicus (Norway rat)Potency22.387210
3-methoxy-N-(2,3,4-trifluorophenyl)benzamideRattus norvegicus (Norway rat)Potency39.810710
3-methyl-1-[2-(2H-tetrazol-5-yl)ethyl]-4,6-bis(trifluoromethyl)pyrazolo[3,4-b]pyridineRattus norvegicus (Norway rat)Potency56.234110
[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-(2-ethoxy-3-pyridinyl)methanoneRattus norvegicus (Norway rat)Potency31.622810
2-chloro-N-(2-phenyl-5-propyl-3-pyrazolyl)acetamideRattus norvegicus (Norway rat)Potency50.118710
2-[[2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]-1-oxoethyl]amino]-5-phenyl-3-thiophenecarboxamideRattus norvegicus (Norway rat)Potency50.118710
3-methyl-6-thiophen-2-yl-4-isoxazolo[5,4-b]pyridinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency10.000010
2,6-dichloro-N-[2-(methylthio)-1,3-benzothiazol-6-yl]benzenesulfonamideRattus norvegicus (Norway rat)Potency89.125110
2-(4-formylphenoxy)acetic acid [2-(4-methylanilino)-4-thiazolyl]methyl esterRattus norvegicus (Norway rat)Potency0.141310
5-(3,4-dimethoxyphenyl)-3-(4-methoxyphenyl)-1H-imidazole-2-thioneRattus norvegicus (Norway rat)Potency56.234110
5-(3,4-dimethoxyphenyl)-3-(4-ethoxyphenyl)-1H-imidazole-2-thioneRattus norvegicus (Norway rat)Potency39.810710
N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency31.622810
N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamideRattus norvegicus (Norway rat)Potency3.162310
2-(2,4-dioxo-1H-pyrimidin-6-yl)-N-[2-(4-morpholinyl)ethyl]acetamideRattus norvegicus (Norway rat)Potency22.387210
3-phenyl-2-sulfanylidene-1H-benzofuro[3,2-d]pyrimidin-4-oneRattus norvegicus (Norway rat)Potency22.387210
(4-tert-butylphenyl)-[2-(4-fluorophenyl)-8-methyl-3-sulfanylidene-1,4,8-triazaspiro[4.5]dec-1-en-4-yl]methanoneRattus norvegicus (Norway rat)Potency31.622810
2-[[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-oxomethyl]imino-1-(2-methylpropyl)-5-oxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency56.234110
6-propyladenineRattus norvegicus (Norway rat)Potency0.398110
2-(4-benzofuro[3,2-d]pyrimidinylthio)-N-(2-ethoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency100.000010
LSM-26967Rattus norvegicus (Norway rat)Potency89.716420
4-[ethyl-(phenylmethyl)sulfamoyl]-N-[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideRattus norvegicus (Norway rat)Potency8.912510
2-[2-furanyl(oxo)methyl]imino-5-oxo-1-propan-2-yl-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency28.183810
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterRattus norvegicus (Norway rat)Potency10.000010
1-[2,3-bis(2-pyridinyl)-6-quinoxalinyl]-3-propylthioureaRattus norvegicus (Norway rat)Potency28.183810
thiocyanic acid [2-(1-naphthalenyl)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency56.234110
mcb-613Rattus norvegicus (Norway rat)Potency56.234110
3-[4-[(4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-ylidene)methyl]-3-(2-oxo-1-benzopyran-3-yl)-1-pyrazolyl]propanoic acidRattus norvegicus (Norway rat)Potency7.079510
1-cyclohexyl-3-(6-ethoxy-1,3-benzothiazol-2-yl)ureaRattus norvegicus (Norway rat)Potency12.589310
N-(2-methoxyphenyl)-5-methyl-3-(1-naphthalenylmethyl)-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency89.125110
2,3-dichloro-4-methoxy-N-(3-methoxypropyl)benzenesulfonamideRattus norvegicus (Norway rat)Potency10.000010
3-methoxy-N-[2-(3-methoxyphenoxy)ethyl]benzamideRattus norvegicus (Norway rat)Potency28.183810
N-(2-furanylmethyl)-2-(6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-d]pyrimidin-4-ylthio)acetamideRattus norvegicus (Norway rat)Potency28.183810
N-[5-(3-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency89.125110
2,5-dimethoxybenzenesulfonic acid (1,3-dioxo-2-isoindolyl) esterRattus norvegicus (Norway rat)Potency1.778310
2-(2-bromo-4-tert-butylphenoxy)-N-(2-furanylmethyl)acetamideRattus norvegicus (Norway rat)Potency11.220210
2-[2-nitro-4-(trifluoromethyl)phenyl]sulfinylacetic acid (4-chlorophenyl) esterRattus norvegicus (Norway rat)Potency50.118710
1-[[(4-ethyl-5-methyl-3-thiophenyl)-oxomethyl]amino]-3-(2-phenylethyl)thioureaRattus norvegicus (Norway rat)Potency0.089110
N-(2-furanylmethyl)-2-[4-(propylsulfamoyl)phenoxy]acetamideRattus norvegicus (Norway rat)Potency31.622810
1-[[(4-bromo-2-methyl-3-pyrazolyl)-oxomethyl]amino]-3-(2-methoxy-5-methylphenyl)thioureaRattus norvegicus (Norway rat)Potency70.794610
1-(4-bromo-2-chlorophenyl)-3-(3-methyl-2-pyridinyl)thioureaRattus norvegicus (Norway rat)Potency89.125110
4-(5-methyl-2-furanyl)-2-[[1-oxo-2-(1H-1,2,4-triazol-5-ylthio)ethyl]amino]-3-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.810710
3-(3-bromoanilino)-1-(5-methyl-2-furanyl)-1-propanoneRattus norvegicus (Norway rat)Potency19.952610
3-[1-(3-methoxypropyl)-5-thiophen-2-yl-2-pyrrolyl]propanoic acidRattus norvegicus (Norway rat)Potency25.515420
N-[4-(cyanomethyl)phenyl]-4-cyclohexylbenzenesulfonamideRattus norvegicus (Norway rat)Potency0.251210
2-(5-bromo-2-furanyl)-6-methyl-3,1-benzoxazin-4-oneRattus norvegicus (Norway rat)Potency79.432810
4-(3-hydroxyphenyl)-1-(thiophen-2-ylmethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency35.481310
N-(2-fluorophenyl)-4-methoxy-2,5-dimethylbenzenesulfonamideRattus norvegicus (Norway rat)Potency0.398110
4-methyl-6-(2,2,3,3,4,4,5,5-octafluoropentoxy)-2-pyrimidinamineRattus norvegicus (Norway rat)Potency0.562310
2-[(3,4-dimethyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid prop-2-enyl esterRattus norvegicus (Norway rat)Potency50.118710
2-[(3,4,8-trimethyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid prop-2-enyl esterRattus norvegicus (Norway rat)Potency39.810710
4-chloro-N-[(2-methylpropylamino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency14.125410
4-[benzenesulfonyl(methyl)amino]-N-[2-[(4-chlorophenyl)methylthio]ethyl]benzamideRattus norvegicus (Norway rat)Potency10.000010
2-[2-[[3-(1,3-benzoxazol-2-yl)anilino]-oxomethyl]phenyl]benzoic acidRattus norvegicus (Norway rat)Potency39.810710
1,3-dimethyl-5-[[5-(phenylthio)-2-furanyl]methylidene]-1,3-diazinane-2,4,6-trioneRattus norvegicus (Norway rat)Potency10.000010
N-(2,1,3-benzothiadiazol-4-yl)-5-(3-chlorophenyl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency35.481310
2-(2,4-dichloro-6-methylphenoxy)-N-(2-furanylmethyl)acetamideRattus norvegicus (Norway rat)Potency39.810710
N-[3-[[diethylamino(sulfanylidene)methyl]thio]-1-oxopropyl]carbamic acid (4-propan-2-ylphenyl) esterRattus norvegicus (Norway rat)Potency79.432810
1,3-dimethyl-5-[[2-[2-(4-nitrophenoxy)ethoxy]phenyl]methylidene]-1,3-diazinane-2,4,6-trioneRattus norvegicus (Norway rat)Potency11.220210
N-(3-dibenzofuranyl)-2-[2-oxo-2-(2,4,6-trimethylanilino)ethoxy]benzamideRattus norvegicus (Norway rat)Potency56.234110
reversanRattus norvegicus (Norway rat)Potency28.183810
2-(4-methoxyphenyl)-N-[2-(4-morpholinyl)ethyl]-4-quinolinecarboxamideRattus norvegicus (Norway rat)Potency79.432810
N'-(3,4-dihydro-2H-pyrrol-5-yl)-2-(2-naphthalenylamino)acetohydrazideRattus norvegicus (Norway rat)Potency89.125110
N-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethenyl]-4-morpholinecarboxamideRattus norvegicus (Norway rat)Potency89.125110
4-[3-(2,5-dimethyl-1-pyrrolyl)-4-(1-pyrrolidinyl)phenyl]sulfonylmorpholineRattus norvegicus (Norway rat)Potency1.584910
2-[(4-ethoxyphenyl)sulfonylamino]-N-[2-(4-morpholinyl)phenyl]benzamideRattus norvegicus (Norway rat)Potency89.716420
2-[(2,5-dimethylphenyl)sulfonylamino]-N-[4-(2-pyrimidinylsulfamoyl)phenyl]benzamideRattus norvegicus (Norway rat)Potency63.095710
4-(4-chlorophenyl)-4-oxobutanoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency44.668410
3-methoxy-2-naphthalenecarboxylic acid [2-(4-morpholinyl)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency89.125110
4-(diethylsulfamoyl)benzoic acid [2-[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency79.432810
2,3-dihydro-1,4-dioxin-5-carboxylic acid [2-[4-[4-(2-methylbutan-2-yl)phenoxy]anilino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency25.118910
3-(1-azepanylsulfonyl)-4-chloro-N-(1H-1,2,4-triazol-5-yl)benzamideRattus norvegicus (Norway rat)Potency14.125410
N,N-diethyl-2-[(4-fluorophenyl)methylthio]-1,3-benzoxazole-5-sulfonamideRattus norvegicus (Norway rat)Potency12.589310
N-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency79.432810
1-(4-ethoxyphenyl)-3-(5-isoquinolinyl)thioureaRattus norvegicus (Norway rat)Potency79.432810
3-[3-oxo-4-(2-phenylethyl)-2-quinoxalinyl]propanoic acidRattus norvegicus (Norway rat)Potency56.234110
N-[(1-adamantylamino)-oxomethyl]-2-chloroacetamideRattus norvegicus (Norway rat)Potency14.125410
1-(2-methoxyethyl)-7-thiophen-2-yl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dioneRattus norvegicus (Norway rat)Potency15.848910
1-butyl-2,4-dioxo-7-thiophen-2-yl-5-pyrido[2,3-d]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency3.162310
3-[2-(cyclohexylamino)-4-(4-methoxyphenyl)-5-thiazolyl]propanoic acid methyl esterRattus norvegicus (Norway rat)Potency89.125110
N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)-4-oxo-4-thiophen-2-ylbutanamideRattus norvegicus (Norway rat)Potency39.810710
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideRattus norvegicus (Norway rat)Potency31.622810
thiocyanic acid [4-[(2-chloro-1-oxoethyl)amino]-3,5-dimethylphenyl] esterRattus norvegicus (Norway rat)Potency50.118710
2-phenoxybenzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency31.622810
2-(2-furanylmethylamino)benzoic acid [2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl] esterRattus norvegicus (Norway rat)Potency26.651420
2-hydroxy-4-methylbenzoic acid [2-(2-chloroanilino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency22.387210
2-[[[[(4-fluorophenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-4-(5-methyl-2-furanyl)-3-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency15.848910
2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]-N-(2-pyridinylmethyl)acetamideRattus norvegicus (Norway rat)Potency44.668410
2-chloro-N-[3-[(2-chlorophenyl)methyl]-2-thiazolylidene]acetamideRattus norvegicus (Norway rat)Potency25.118910
1-(2-furanyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneRattus norvegicus (Norway rat)Potency44.668410
1-(2-cyanoethyl)-6-(2-fluoro-4-methoxyphenyl)-3-methyl-4-pyrazolo[3,4-b]pyridinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency25.285520
[4-(2-ethoxyphenyl)-1-piperazinyl]-(1-oxido-4-pyridin-1-iumyl)methanoneRattus norvegicus (Norway rat)Potency56.234110
2-[(2-hydroxy-1-naphthalenyl)methyl-methylamino]-N-[4-(4-morpholinyl)phenyl]acetamideRattus norvegicus (Norway rat)Potency3.981110
N-(6-methoxy-1,3-benzothiazol-2-yl)-3-(4-morpholinylsulfonyl)benzamideRattus norvegicus (Norway rat)Potency70.794610
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4-methyl-5-phenyl-2-thiazolyl)-N-prop-2-enylacetamideRattus norvegicus (Norway rat)Potency6.309610
1-(2,6-diethylphenyl)-3-[2-(3,4-dihydroxyphenyl)ethyl]thioureaRattus norvegicus (Norway rat)Potency6.309610
1-[4-(4-hydroxyphenyl)-1-piperazinyl]-3-(1H-indol-3-yl)-1-propanoneRattus norvegicus (Norway rat)Potency0.100010
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneRattus norvegicus (Norway rat)Potency7.943310
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideRattus norvegicus (Norway rat)Potency56.234110
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideRattus norvegicus (Norway rat)Potency19.952610
2-chloro-1-[4-[(3-methylphenyl)methyl]-1-piperazinyl]ethanoneRattus norvegicus (Norway rat)Potency11.220210
2-anilinobenzoic acid [2-(4-acetylanilino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency89.125110
2-chloro-N-[(5-chloro-2-thiophenyl)methyl]-N-methylacetamideRattus norvegicus (Norway rat)Potency8.912510
4-[2-(4-fluoroanilino)-2-oxoethoxy]-3-methoxy-N-[4-(4-methoxyphenyl)-5-methyl-2-thiazolyl]benzamideRattus norvegicus (Norway rat)Potency44.668410
2-(butylamino)benzoic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterRattus norvegicus (Norway rat)Potency79.432810
2-[[4-(4-fluorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]thio]-N-[(2-furanylmethylamino)-oxomethyl]acetamideRattus norvegicus (Norway rat)Potency39.810710
2-[[5-(5-bromo-2-furanyl)-4-(phenylmethyl)-1,2,4-triazol-3-yl]thio]-1-(2-fluorophenyl)ethanoneRattus norvegicus (Norway rat)Potency44.668410
2-[2-(2,3-dimethoxyphenyl)-4-thiazolyl]acetic acidRattus norvegicus (Norway rat)Potency28.183810
1-[2,5-dimethyl-1-(phenylmethyl)-3-pyrrolyl]-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]ethanoneRattus norvegicus (Norway rat)Potency70.794610
4-[[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-oxomethyl]-2-ethyl-1-phthalazinoneRattus norvegicus (Norway rat)Potency12.589310
5-[2-[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
N-[3-[4-[(2-methoxyphenyl)sulfamoyl]anilino]-3-oxopropyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency39.810710
5-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acidRattus norvegicus (Norway rat)Potency50.118710
2-(1,3-benzodioxol-5-yl)-5-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methylthio]-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency15.848910
2-chloro-N-(2-chloro-5-methylsulfonylphenyl)acetamideRattus norvegicus (Norway rat)Potency12.589310
5-chloro-1-[(2-chlorophenyl)methyl]-3-methyl-4-pyrazolecarboxylic acid [2-[(5-methyl-3-isoxazolyl)amino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency44.668410
4,5-dichloro-2-[2-[2,5-dimethyl-1-(2,2,2-trifluoroethyl)-3-pyrrolyl]-2-oxoethyl]-3-pyridazinoneRattus norvegicus (Norway rat)Potency28.183810
N-[3-(4-morpholinyl)propyl]-3-(3-pyridinyl)-7,8-dihydro-6H-cyclopenta[4,5]thieno[1,2-c]pyrimidin-1-amineRattus norvegicus (Norway rat)Potency22.387210
[4-(3-chlorophenyl)-1-piperazinyl]-(2,5-dimethyl-3-furanyl)methanoneRattus norvegicus (Norway rat)Potency31.622810
3-[ethyl(phenyl)sulfamoyl]-4-methylbenzoic acid (4-methyl-2-oxo-1-benzopyran-7-yl) esterRattus norvegicus (Norway rat)Potency79.432810
2-[(2,4-dimethoxyphenyl)methyl-methylamino]-N-(2-methoxy-3-dibenzofuranyl)acetamideRattus norvegicus (Norway rat)Potency39.810710
4-bromotetramisole, oxalate (1:1), salt(s)-isomerRattus norvegicus (Norway rat)Potency100.000010
mercaptopurineRattus norvegicus (Norway rat)Potency79.432810
2-oxo-6-phenyl-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency30.258620
2-(methylamino)-6-thiophen-2-yl-4-(trifluoromethyl)-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency14.219120
4-phenoxyphenyl 4-hydroxypiperidine-1-carboxylateRattus norvegicus (Norway rat)Potency1.258910
1-(3-methylphenyl)-3-(2-pyridinyl)thioureaRattus norvegicus (Norway rat)Potency39.810710
mecysteine hydrochlorideRattus norvegicus (Norway rat)Potency79.432810
capsazepineRattus norvegicus (Norway rat)Potency51.051420
diphenyleneiodium chlorideRattus norvegicus (Norway rat)Potency22.983310
azetidine-2,4-dicarboxylic acid, (cis)-isomerRattus norvegicus (Norway rat)Potency26.393020
tamoxifen citrateRattus norvegicus (Norway rat)Potency42.284110
8-fluoro-4H-thieno[3,2-c][1]benzopyran-2-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency11.519020
4-(2-fluorophenyl)-N-(2-methylbut-3-yn-2-yl)benzamideRattus norvegicus (Norway rat)Potency3.548110
5-methoxy-N-(1-methoxypropan-2-yl)-1H-indole-2-carboxamideRattus norvegicus (Norway rat)Potency17.782810
N-butyl-5-methoxy-1H-indole-2-carboxamideRattus norvegicus (Norway rat)Potency39.810710
5-cyano-2-(methoxymethyl)-6-sulfanylidene-1H-pyridine-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency14.125410
1-piperidinyl-(5-thiophen-2-yl-3-isoxazolyl)methanoneRattus norvegicus (Norway rat)Potency31.622810
N-(3,5-dichlorophenyl)-2-[[4-methyl-5-[4-methyl-2-(5-methyl-3-isoxazolyl)-5-thiazolyl]-1,2,4-triazol-3-yl]thio]acetamideRattus norvegicus (Norway rat)Potency84.279020
N-(4-chlorophenyl)-2-[[4-methyl-5-[4-methyl-2-(5-methyl-3-isoxazolyl)-5-thiazolyl]-1,2,4-triazol-3-yl]thio]acetamideRattus norvegicus (Norway rat)Potency89.125110
4-(2-furanyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency50.118710
5-oxo-3-(4-phenylphenyl)-2H-furan-4-carbonitrileRattus norvegicus (Norway rat)Potency39.810710
[5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-yl]hydrazineRattus norvegicus (Norway rat)Potency56.234110
LSM-20838Rattus norvegicus (Norway rat)Potency33.527820
1-[(3-chlorophenyl)methyl]-3-[5-(methylthio)-1,3,4-oxadiazol-2-yl]-2-pyridinoneRattus norvegicus (Norway rat)Potency31.622810
2,6-dichlorobenzoic acid [3-cyano-6-(3-methoxyphenyl)-2-pyridinyl] esterRattus norvegicus (Norway rat)Potency84.279020
4-chlorobenzoic acid [3-cyano-6-(3-methoxyphenyl)-2-pyridinyl] esterRattus norvegicus (Norway rat)Potency79.432810
2-(4-methylphenyl)thiazolidineRattus norvegicus (Norway rat)Potency50.118710
monoacetylphloroglucinolRattus norvegicus (Norway rat)Potency3.548110
4-oxo-2-(trifluoromethyl)-1H-thieno[3,4-b]pyridine-7-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency70.794610
statticRattus norvegicus (Norway rat)Potency1.579930
5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-amineRattus norvegicus (Norway rat)Potency25.118910
2-{4-[(2-aminophenyl)thio]-3-nitrobenzoyl}benzoic acidRattus norvegicus (Norway rat)Potency0.100010
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineRattus norvegicus (Norway rat)Potency0.316210
8-methoxy-4-oxo-1H-quinoline-2-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency50.118710
2-(4-chlorophenyl)-6-(methylthio)-4-oxo-2,3-dihydro-1,3-thiazine-5-carbonitrileRattus norvegicus (Norway rat)Potency28.183810
2-(4-morpholinyl)-5-[[oxo-[2-(trifluoromethyl)-5-[4-(trifluoromethyl)phenyl]-3-furanyl]methyl]amino]benzoic acid methyl esterRattus norvegicus (Norway rat)Potency0.631010
1H-indol-3-yl(pyridin-2-yl)methanolRattus norvegicus (Norway rat)Potency89.125110
1-(4-fluorophenyl)-3-[2-methyl-5-(1-piperidinylsulfonyl)-3-furanyl]ureaRattus norvegicus (Norway rat)Potency15.848910
5-(tert-butyl)-2-methyl-N-(5-methyl-3-isoxazolyl)-3-furamideRattus norvegicus (Norway rat)Potency44.668410
2-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrimidineRattus norvegicus (Norway rat)Potency54.195620
5-[4-(2-furylcarbonyl)piperazino]-5-oxo-3-phenylpentanoic acidRattus norvegicus (Norway rat)Potency14.125410
5-(4-morpholinoanilino)-5-oxo-3-phenylpentanoic acidRattus norvegicus (Norway rat)Potency10.000010
LSM-28486Rattus norvegicus (Norway rat)Potency31.225620
3-oxo-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)thio]butanoic acid ethyl esterRattus norvegicus (Norway rat)Potency28.183810
2-oxo-4,6-dithiophen-2-yl-1H-pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency14.125410
5-[[(4-methoxyanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency56.234110
3-(2,4-dimethoxyphenyl)-6-phenyl-2-sulfanylidene-1H-thieno[2,3-d]pyrimidin-4-oneRattus norvegicus (Norway rat)Potency15.848910
5-(methoxymethyl)-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-oneRattus norvegicus (Norway rat)Potency11.464220
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileRattus norvegicus (Norway rat)Potency19.952610
3,3-dimethyl-1-[[9-(methylthio)-5,6-dihydrothieno[3,4-h]quinazolin-2-yl]thio]-2-butanoneRattus norvegicus (Norway rat)Potency50.118710
8-methylsulfinyl-4,5-dihydrothieno[3,4-g][2,1]benzoxazole-6-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency31.622810
1-(3,5-dichlorophenyl)-3-[2-(2-furanylmethylthio)ethyl]ureaRattus norvegicus (Norway rat)Potency79.432810
2-(2-pyrenyl)acetonitrileRattus norvegicus (Norway rat)Potency63.514420
2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-phenylacetamideRattus norvegicus (Norway rat)Potency70.794610
3-(4-ethyl-1-piperazinyl)-5-methylpyridazino[3,4-b][1,4]benzoxazineRattus norvegicus (Norway rat)Potency31.622810
N-[[1,3-dioxo-2-(phenylmethyl)-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]-4-methoxybenzamideRattus norvegicus (Norway rat)Potency25.118910
N-[(2-chloroanilino)-sulfanylidenemethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency22.387210
dihydrosamidineRattus norvegicus (Norway rat)Potency89.125110
oreoseloneRattus norvegicus (Norway rat)Potency56.234110
3-benzylbenzothiazoliumRattus norvegicus (Norway rat)Potency79.432810
5-cyclopentylidene-2-sulfanylidene-4-thiazolidinoneRattus norvegicus (Norway rat)Potency70.794610
1-(9-anthracenylmethyl)-3-piperidinolRattus norvegicus (Norway rat)Potency47.359320
2-(difluoromethyl)-4-benzo[h][1]benzopyranoneRattus norvegicus (Norway rat)Potency44.668410
3,7-dimethyl-2-[4-(2-pyridinyl)-1-piperazinyl]quinolineRattus norvegicus (Norway rat)Potency89.125110
2-(4,6,7-Trimethyl-2-quinazolinyl)guanidineRattus norvegicus (Norway rat)Potency79.432810
4-ethyl-2-methoxy-3-phenyl-3,3a,9,9a-tetrahydropyrrolo[2,3-b]quinoxalineRattus norvegicus (Norway rat)Potency19.952610
nemadipine-aRattus norvegicus (Norway rat)Potency28.796820
4-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) esterRattus norvegicus (Norway rat)Potency89.125110
2-[[oxo(thiophen-2-yl)methyl]amino]-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideRattus norvegicus (Norway rat)Potency25.118910
2-[[1-(4-ethoxyphenyl)-2,5-dioxo-3-pyrrolidinyl]amino]acetonitrileRattus norvegicus (Norway rat)Potency22.387210
N-(3-acetyl-2-methyl-5-benzofuranyl)-N-(4-chloro-3-nitrophenyl)sulfonylacetamideRattus norvegicus (Norway rat)Potency7.943310
N'-[4-(1-adamantyl)-2-thiazolyl]-N-[(4-fluorophenyl)methyl]oxamideRattus norvegicus (Norway rat)Potency5.623410
6-amino-4-(3-chlorophenyl)-3-methyl-1-(phenylmethyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrileRattus norvegicus (Norway rat)Potency44.668410
N-(3-chloro-4-methylphenyl)-2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)acetamideRattus norvegicus (Norway rat)Potency89.125110
2-[4-(2,2-dimethyl-4-oxo-1,3,5,6-tetrahydrobenzo[a]phenanthridin-5-yl)-2-methoxyphenoxy]acetic acidRattus norvegicus (Norway rat)Potency71.264220
2-[[2-methyl-5-nitro-3-(phenylmethyl)-4-imidazolyl]thio]-6-nitro-1H-benzimidazoleRattus norvegicus (Norway rat)Potency2.511910
2-methoxy-N-(2-pyridinylmethyl)-3-dibenzofuranamineRattus norvegicus (Norway rat)Potency28.183810
[(2S)-1,3-dimethyl-3'-nitro-1'-spiro[cyclohepta[d]imidazol-3-ium-2,4'-cyclohexa-2,5-diene]ylidene]-dioxidoammoniumRattus norvegicus (Norway rat)Potency22.387210
1-(4-methylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency5.011910
1-(3,5-dimethylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency12.589310
kl001Rattus norvegicus (Norway rat)Potency19.952610
2-(2,4-dichlorophenyl)-3-(phenylmethyl)-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency28.183810
4-[5-(3-chloro-2-methylphenyl)-2-furanyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency22.387210
5-methyl-2-phenyl-5-(2-phenylethyl)-1,2,4-triazolidine-3-thioneRattus norvegicus (Norway rat)Potency50.118710
4-chloro-3-(diethylsulfamoyl)-N-(2-nitrophenyl)benzamideRattus norvegicus (Norway rat)Potency1.258910
4-bromobenzenesulfonic acid (1,3-dioxo-2-benzo[de]isoquinolinyl) esterRattus norvegicus (Norway rat)Potency39.810710
N-(4-chloro-3-nitrophenyl)-3-phenylbutanamideRattus norvegicus (Norway rat)Potency3.162310
4-(3-hydroxyphenyl)-1-(2-oxolanylmethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency14.333520
2-[[5-[(1,3-benzothiazol-2-ylthio)methyl]-4-methyl-1,2,4-triazol-3-yl]thio]-N-[2-(4-morpholinyl)ethyl]acetamideRattus norvegicus (Norway rat)Potency12.589310
2-(4-chlorophenyl)-5-(2-oxolanylmethylamino)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency56.234110
2-(4-fluorophenyl)-4-(4-methoxyanilino)-1-(4-methoxyphenyl)-2H-pyrrol-5-oneRattus norvegicus (Norway rat)Potency53.176420
3-(n,n-dimethylsulfonamido)-4-methyl-nitrobenzeneRattus norvegicus (Norway rat)Potency0.316210
5-[[(1-cyclohexyl-5-tetrazolyl)thio]methyl]-3-phenyl-1,2,4-oxadiazoleRattus norvegicus (Norway rat)Potency17.782810
1-cyclopentyl-2-imino-10-methyl-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency53.176420
3-(2-furanylmethyl)-2-phenyl-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency72.679620
1-(2-furanylmethyl)-3-[(4-methylphenyl)methyl]pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency50.118710
6-hydroxy-5-[(6-hydroxy-1-methyl-4-oxo-2-sulfanylidene-5-pyrimidinyl)-(2-pyridinyl)methyl]-1-methyl-2-sulfanylidene-4-pyrimidinoneRattus norvegicus (Norway rat)Potency35.481310
3-(2,5-dioxo-1-pyrrolidinyl)-N-(2-methyl-1,3-dioxo-5-isoindolyl)benzamideRattus norvegicus (Norway rat)Potency79.432810
4-[[1-[(3,4-dichlorophenyl)methyl]-3-indolyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneRattus norvegicus (Norway rat)Potency48.022420
N-(4-carbamoylphenyl)-2-(4-methoxyphenyl)-4-quinolinecarboxamideRattus norvegicus (Norway rat)Potency31.622810
2-[[1-(4-chlorophenyl)-2,5-dioxo-3-pyrrolidinyl]-methylamino]acetic acid methyl esterRattus norvegicus (Norway rat)Potency35.481310
4-(5-methyl-3-oxo-1H-pyrazol-2-yl)benzoic acidRattus norvegicus (Norway rat)Potency56.234110
5-(2-oxolanylmethylamino)-2-thiophen-2-yl-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency50.138720
2-[[1-(4-methoxy-2-nitrophenyl)-2,5-dioxo-3-pyrrolidinyl]thio]benzoic acidRattus norvegicus (Norway rat)Potency70.794610
2-methyl-3-[(2-methyl-1H-indol-3-yl)-(2-pyridinyl)methyl]-1H-indoleRattus norvegicus (Norway rat)Potency39.810710
N-[4-[4-(1-pyrrolidinylsulfonyl)phenyl]-2-thiazolyl]-2,3-dihydro-1,4-benzodioxin-3-carboxamideRattus norvegicus (Norway rat)Potency39.810710
1-(2,4-dimethoxyphenyl)-3-[4-(4-morpholinyl)anilino]pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency63.095710
3-nitro-N-[[4-[4-(1-oxopropyl)-1-piperazinyl]anilino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency17.782810
4-(5-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1h-pyrazol-1-yl)benzenesulfonamideRattus norvegicus (Norway rat)Potency16.597820
3-(2-pyrimidinylthio)-1-[2-(trifluoromethyl)phenyl]pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency70.794610
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-phenoxybutanamideRattus norvegicus (Norway rat)Potency31.622810
3-(2-furanyl)-3-(4-methylphenyl)-1-(4-morpholinyl)-1-propanoneRattus norvegicus (Norway rat)Potency44.668410
4-[[2-(4-ethyl-3-oxo-2-morpholinyl)-1-oxoethyl]amino]benzoic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
3-[2-(2,4-dimethyl-3-furanyl)-2-oxoethyl]-3-hydroxy-1-(2-phenylethyl)-2-indoloneRattus norvegicus (Norway rat)Potency15.848910
4-(4-nitrophenyl)-N-prop-2-enyl-1-piperazinecarbothioamideRattus norvegicus (Norway rat)Potency79.432810
2-[[(2-methoxy-4-nitroanilino)-sulfanylidenemethyl]amino]benzene-1,4-dicarboxylic acid diethyl esterRattus norvegicus (Norway rat)Potency62.050620
2-(1,3-benzothiazol-2-ylamino)-5-spiro[1,6,7,8-tetrahydroquinazoline-4,1'-cyclopentane]oneRattus norvegicus (Norway rat)Potency21.679420
5-(3,5-dimethyl-1-piperidinyl)-2-(2-furanyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency50.118710
4-[[[4-(2-furanylmethyl)-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]thio]methyl]benzonitrileRattus norvegicus (Norway rat)Potency39.810710
1-[4-[4-[[6-bromo-2-(3-pyridinyl)-4-quinolinyl]-oxomethyl]-1-piperazinyl]phenyl]ethanoneRattus norvegicus (Norway rat)Potency39.810710
5-chloro-7-[3-pyridinyl-(2-pyridinylamino)methyl]-8-quinolinolRattus norvegicus (Norway rat)Potency12.589310
3-[(1-methyl-5-tetrazolyl)thio]-1-phenylpyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency17.782810
2,4-dichloro-N-[2,4,6-trioxo-1-(phenylmethyl)-5-(trifluoromethyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzamideRattus norvegicus (Norway rat)Potency8.912510
cb 7969312Rattus norvegicus (Norway rat)Potency2.990410
3-[5-(4-methylphenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acidRattus norvegicus (Norway rat)Potency50.118710
2-[1-[[[(3-chloro-1-benzothiophen-2-yl)-oxomethyl]amino]-sulfanylidenemethyl]-3-oxo-2-piperazinyl]acetic acid methyl esterRattus norvegicus (Norway rat)Potency79.432810
2-[[4-(4-fluorophenyl)-6-(trifluoromethyl)-2-pyrimidinyl]sulfonyl]acetic acid ethyl esterRattus norvegicus (Norway rat)Potency3.981110
3-[5-(4-fluorophenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acidRattus norvegicus (Norway rat)Potency89.125110
4-(4-bromophenyl)-2-(3,5-dimethyl-1-pyrazolyl)-4-oxobutanoic acid methyl esterRattus norvegicus (Norway rat)Potency8.912510
2-[3-oxo-1-[[[oxo(thiophen-2-yl)methyl]amino]-sulfanylidenemethyl]-2-piperazinyl]acetic acid propan-2-yl esterRattus norvegicus (Norway rat)Potency79.432810
2-[1-[[[(4-methoxyphenyl)-oxomethyl]amino]-sulfanylidenemethyl]-3-oxo-2-piperazinyl]acetic acid propan-2-yl esterRattus norvegicus (Norway rat)Potency70.794610
4-(2-oxo-1-benzopyran-3-yl)-N-(3-pyridinylmethyl)benzamideRattus norvegicus (Norway rat)Potency44.668410
2,2-dimethyl-N-[[4-(pyridin-4-ylmethyl)anilino]-sulfanylidenemethyl]propanamideRattus norvegicus (Norway rat)Potency22.387210
3-methyl-N-[[(2-methyl-5-quinolinyl)amino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency12.589310
2-[[2-(4-ethyl-4-methyl-2,5-dioxo-1-imidazolidinyl)-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideRattus norvegicus (Norway rat)Potency25.118910
2-[(4-methylphenyl)sulfonylamino]acetic acid (2-oxo-3-oxolanyl) esterRattus norvegicus (Norway rat)Potency39.810710
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamideRattus norvegicus (Norway rat)Potency8.912510
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideRattus norvegicus (Norway rat)Potency39.810710
2-(1,3-diphenyl-4-pyrazolyl)-3-(2-furanylmethyl)-4-thiazolidinoneRattus norvegicus (Norway rat)Potency79.432810
3-(2,5-dimethyl-3-furanyl)-5,6-diphenyl-1,2,4-triazineRattus norvegicus (Norway rat)Potency31.622810
bis(1-ethenyl-2-imidazolyl)-(9-ethyl-3-carbazolyl)-sulfanylidenephosphoraneRattus norvegicus (Norway rat)Potency19.952610
1-(4-fluorophenyl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxylic acid (2-oxo-3-oxolanyl) esterRattus norvegicus (Norway rat)Potency63.095710
5-amino-3-[[[1-(2-furanylmethyl)-5-oxo-3-pyrrolidinyl]-oxomethoxy]methyl]thiophene-2,4-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency17.782810
3-[[5,5-dimethyl-3-(4-morpholinyl)-1-cyclohex-2-enylidene]amino]-N,N-dimethylanilineRattus norvegicus (Norway rat)Potency12.589310
zeranolRattus norvegicus (Norway rat)Potency0.100010
2-amino-4-chlorobenzoic acid [2-oxo-2-(3,3,5-trimethyl-7-azabicyclo[3.2.1]octan-7-yl)ethyl] esterRattus norvegicus (Norway rat)Potency39.810710
3-fluoro-6a,7,8,9,10,11-hexahydro-6H-azepino[2,1-c][1,2,4]benzothiadiazine 5,5-dioxideRattus norvegicus (Norway rat)Potency89.125110
1-butyl-2-[(5-phenyl-2-oxazolyl)methylthio]-5-benzimidazolesulfonamideRattus norvegicus (Norway rat)Potency79.432810
2-(2-amino-4H-[1,3,5]triazino[2,1-b][1,3]benzoxazol-4-yl)propanedioic acid diethyl esterRattus norvegicus (Norway rat)Potency42.239520
2-(2-furanyl)-N-(2-oxolanylmethyl)-4-quinolinecarboxamideRattus norvegicus (Norway rat)Potency53.138020
3-(4-methylphenyl)sulfonyl-1-(3-oxolanylmethyl)-2-pyrrolo[3,2-b]quinoxalinamineRattus norvegicus (Norway rat)Potency28.183810
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideRattus norvegicus (Norway rat)Potency89.125110
ly 73497Rattus norvegicus (Norway rat)Potency19.952610
LSM-1318Rattus norvegicus (Norway rat)Potency15.575030
6-methyl-2-(phenylethynyl)pyridineRattus norvegicus (Norway rat)Potency39.810710
thiophanateRattus norvegicus (Norway rat)Potency50.118710
ranitidine hydrochlorideRattus norvegicus (Norway rat)Potency47.286410
7-deacetylgeduninRattus norvegicus (Norway rat)Potency39.810710
emetine dihydrochlorideRattus norvegicus (Norway rat)Potency1.191710
2,2-dimethyl-N-[2,2,2-trichloro-1-(2-pyrimidinylthio)ethyl]propanamideRattus norvegicus (Norway rat)Potency7.079510
3-O-AcetylepisamarcandinRattus norvegicus (Norway rat)Potency42.800020
N-methyl-5-nitro-N-(phenylmethyl)-2-furancarboxamideRattus norvegicus (Norway rat)Potency14.125410
N-[[2-(4-chlorophenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]benzenesulfonamideRattus norvegicus (Norway rat)Potency10.000010
2-[[2,2,2-trichloro-1-[(2,2-dimethyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency6.309610
2-(2,3,3-trichloro-1-nitroprop-2-enylidene)-1,3-dihydrobenzimidazoleRattus norvegicus (Norway rat)Potency11.220210
2-[(4-chlorophenyl)-[2-[5-(4-chlorophenyl)-2-thiazolyl]-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]propanedinitrileRattus norvegicus (Norway rat)Potency11.220210
3-(4-fluorophenyl)-5-(2-furanyl)-2-phenyl-3,4-dihydropyrazoleRattus norvegicus (Norway rat)Potency17.138220
2-[[3-methyl-5-oxo-1-(phenylmethyl)-4H-pyrazol-4-yl]-phenylmethyl]propanedinitrileRattus norvegicus (Norway rat)Potency44.668410
4-[4-[2-hydroxy-3-(4-morpholinyl)propoxy]phenyl]benzonitrileRattus norvegicus (Norway rat)Potency22.387210
N-[2-[5-[(4-tert-butylphenyl)methylthio]-1,3,4-oxadiazol-2-yl]phenyl]benzamideRattus norvegicus (Norway rat)Potency11.220210
3-nitro-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency56.234110
3,4-dimethoxy-N-[(2-methyl-4-nitroanilino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency2.238710
3-[[5,6-bis(4-methoxyphenyl)-4-furo[2,3-d]pyrimidinyl]amino]-1-propanolRattus norvegicus (Norway rat)Potency22.387210
2-[(2-ethyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-3-yl)oxy]acetic acid methyl esterRattus norvegicus (Norway rat)Potency56.234110
1-[3-(benzenesulfonyl)-2-(1-piperidinyl)propyl]piperidineRattus norvegicus (Norway rat)Potency44.668410
1-(3-hydroxy-2,4,4-trimethyl-1-oxido-5-thiophen-2-yl-2-imidazol-1-iumyl)ethanoneRattus norvegicus (Norway rat)Potency15.848910
2-imino-1-[(4-methylphenyl)methyl]-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency31.622810
yl-109Rattus norvegicus (Norway rat)Potency44.668410
3-methyl-1-(3-propan-2-yloxypropylamino)-4-pyrido[1,2-a]benzimidazolecarbonitrileRattus norvegicus (Norway rat)Potency22.387210
N-(2-methoxyethyl)-1-methyl-2-oxo-6-benzo[cd]indolesulfonamideRattus norvegicus (Norway rat)Potency31.622810
2-(3-ethoxypropylamino)-8-methyl-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[1,2-pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency27.829820
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneRattus norvegicus (Norway rat)Potency25.118910
2-(1,5-dimethyl-4-pyrazolyl)-4-quinolinecarboxylic acidRattus norvegicus (Norway rat)Potency28.183810
3-ethyl-1-(2-furanylmethyl)-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]thioureaRattus norvegicus (Norway rat)Potency44.668410
N-[2-(tert-butylamino)-2-oxo-1-pyridin-4-ylethyl]-N-(2-furanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideRattus norvegicus (Norway rat)Potency31.622810
2-methoxy-4-[5-methyl-3-(2-oxolanylmethylamino)-2-imidazo[1,2-a]pyridinyl]phenolRattus norvegicus (Norway rat)Potency31.622810
CID 3192987Rattus norvegicus (Norway rat)Potency22.387210
4-[[4-(1,3-benzothiazol-2-yl)-1-piperazinyl]-[1-(2-phenylethyl)-5-tetrazolyl]methyl]phenolRattus norvegicus (Norway rat)Potency35.481310
4-[3-(1,3-benzodioxol-5-ylmethylamino)-7-methyl-2-imidazo[1,2-a]pyridinyl]phenolRattus norvegicus (Norway rat)Potency89.125110
2-butyl-3-[(3-chlorophenyl)methyl]-5-methyl-6-imidazo[4,5-b]pyridinamineRattus norvegicus (Norway rat)Potency56.234110
N-tert-butyl-2-[(2-chloro-1-oxoethyl)-(2-furanylmethyl)amino]-2-(4-chlorophenyl)acetamideRattus norvegicus (Norway rat)Potency12.589310
N-(1,3-benzodioxol-5-ylmethyl)-N-[2-(cyclohexylamino)-2-oxo-1-pyridin-4-ylethyl]-2,2,2-trifluoroacetamideRattus norvegicus (Norway rat)Potency39.810710
2-chloro-N-[1-[oxo(10-phenothiazinyl)methyl]-4-piperidinyl]benzamideRattus norvegicus (Norway rat)Potency1.412510
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid [1-(cyclohexylamino)-1-oxopropan-2-yl] esterRattus norvegicus (Norway rat)Potency50.118710
1-[3-[(7-cyano-[1,3]dioxolo[4,5-g]quinolin-6-yl)amino]propyl]-3-(3-methoxypropyl)thioureaRattus norvegicus (Norway rat)Potency39.810720
1-[3-[(7-cyano-[1,3]dioxolo[4,5-g]quinolin-6-yl)amino]propyl]-3-(3-ethoxypropyl)thioureaRattus norvegicus (Norway rat)Potency56.234110
N-[2-(cyclopentylamino)-2-oxoethyl]-4,7-dimethyl-N-(2-methylphenyl)-2-oxo-3H-pyrido[1,2-a]pyrimidine-4-carboxamideRattus norvegicus (Norway rat)Potency34.411720
3-[(2-chlorophenyl)methyl]-7-[4-[4-(trifluoromethyl)phenyl]-1-piperazinyl]triazolo[4,5-d]pyrimidineRattus norvegicus (Norway rat)Potency2.818410
1-(1-tert-butyl-5-tetrazolyl)-N-[(4-fluorophenyl)methyl]-N-(2-furanylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamineRattus norvegicus (Norway rat)Potency39.810710
N-[2-(3-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-N',N'-dimethylpropane-1,3-diamineRattus norvegicus (Norway rat)Potency22.387210
1-(3-methylphenyl)-3-[[1-[4-(4-morpholinylsulfonyl)phenyl]-4-piperidinyl]methyl]ureaRattus norvegicus (Norway rat)Potency79.432810
ml106Rattus norvegicus (Norway rat)Potency19.952610
2-[5-[[2-(3-methoxypropylamino)-2-oxoethyl]thio]-3-oxo-2H-imidazo[1,2-c]quinazolin-2-yl]-N-(phenylmethyl)acetamideRattus norvegicus (Norway rat)Potency14.125410
5-(2-furanyl)-N-(3-pyridinylmethyl)-3-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency50.118710
4-[butan-2-yl-[(3,4-dichloroanilino)-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency100.000010
5-bromo-N-[6-[[(5-bromo-2-furanyl)-oxomethyl]amino]-2-pyridinyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency31.622810
N-(2,4-dimethoxyphenyl)-3-[[2-(2-methoxyphenoxy)-1-oxoethyl]amino]-2-benzofurancarboxamideRattus norvegicus (Norway rat)Potency21.450920
3-(1,3-benzodioxol-5-ylmethyl)-7-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-2-sulfanylidene-1H-quinazolin-4-oneRattus norvegicus (Norway rat)Potency0.316210
(7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl)-(4-morpholinyl)methanoneRattus norvegicus (Norway rat)Potency19.952610
1-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methylsulfinyl]ethanoneRattus norvegicus (Norway rat)Potency12.589310
3-[[2-(4-fluorophenoxy)-1-oxoethyl]amino]-2-benzofurancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency89.716420
N-(2,4-dimethoxyphenyl)-3-[[2-furanyl(oxo)methyl]amino]-2-benzofurancarboxamideRattus norvegicus (Norway rat)Potency40.676520
5-[2-furanyl(4-morpholinyl)methyl]-2-methyl-6-thiazolo[3,2-b][1,2,4]triazololRattus norvegicus (Norway rat)Potency3.162310
7-(4-methoxyphenyl)-5-methyl-2-(methylthio)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidineRattus norvegicus (Norway rat)Potency79.432810
3-[2,4-dioxo-1-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl]-3-quinazolinyl]-N-(2-furanylmethyl)propanamideRattus norvegicus (Norway rat)Potency79.432810
2-phenyl-5-(1-piperidinyl)-4-triazolecarbonitrileRattus norvegicus (Norway rat)Potency26.651420
2-(2-methoxyethyl)-9-methyl-N-[3-(4-methyl-1-piperidinyl)propyl]-1-oxo-4-pyrido[3,4-b]indolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
1-(4-bromophenyl)sulfonyl-4-[(3-methoxyphenyl)methyl]-1,4-diazepaneRattus norvegicus (Norway rat)Potency22.387210
1-(1-naphthalenyl)-3-[3-(1-pyrrolidinyl)propyl]ureaRattus norvegicus (Norway rat)Potency70.794610
2-[[4-[(2,6-dimethyl-4-morpholinyl)sulfonyl]phenyl]-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency25.118910
4-[2-[(1'-acetyl-4-oxo-6-spiro[3,4-dihydro-2H-1-benzopyran-2,4'-piperidine]yl)oxy]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency24.702820
1-(4-chlorophenyl)sulfonyl-N-(2-thiazolyl)-1-cyclopropanecarboxamideRattus norvegicus (Norway rat)Potency0.112210
2-[(3-oxo-2-propan-2-yl-2H-imidazo[1,2-c]quinazolin-5-yl)thio]-N-[2-(4-sulfamoylphenyl)ethyl]acetamideRattus norvegicus (Norway rat)Potency63.095710
4-[(4-cyclohexyl-1-piperazinyl)-oxomethyl]-2-ethyl-6,7-dimethoxy-1-isoquinolinoneRattus norvegicus (Norway rat)Potency63.095710
1,7,7-trimethyl-9-oxo-N-(2-oxolanylmethyl)-8H-furo[3,2-f][1]benzopyran-2-carboxamideRattus norvegicus (Norway rat)Potency63.095710
N-[3-(1-imidazolyl)propyl]-7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamideRattus norvegicus (Norway rat)Potency15.848910
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideRattus norvegicus (Norway rat)Potency28.370820
2-(pyridin-4-ylmethylamino)benzoic acidRattus norvegicus (Norway rat)Potency22.387210
9-(4-methoxyphenyl)-3,3,6,6-tetramethyl-10-[2-(4-morpholinyl)ethyl]-4,5,7,9-tetrahydro-2H-acridine-1,8-dioneRattus norvegicus (Norway rat)Potency56.234110
N-[2-(2,3-dimethylphenyl)-5,5-dioxo-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-2-methoxybenzamideRattus norvegicus (Norway rat)Potency72.679620
5-(3,4-dimethoxyphenyl)-N-[1-[(2-methylphenyl)methyl]-4-pyrazolyl]-3-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency50.118710
N-(2-furanylmethyl)-2-[(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)thio]acetamideRattus norvegicus (Norway rat)Potency50.118710
4-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-6-(trifluoromethyl)pyrimidineRattus norvegicus (Norway rat)Potency44.964720
5a,6,7,8,9,10-hexahydro-5H-azepino[2,1-b]quinazolin-12-oneRattus norvegicus (Norway rat)Potency35.481310
2-cyclopentyl-4-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-9-methyl-1-pyrido[3,4-b]indoloneRattus norvegicus (Norway rat)Potency28.183810
4-[[[(1-ethyl-2-oxo-6-benzo[cd]indolyl)amino]-oxomethyl]amino]benzoic acid ethyl esterRattus norvegicus (Norway rat)Potency10.000010
LSM-18934Rattus norvegicus (Norway rat)Potency44.668410
5-(dimethylamino)-2-phenyl-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency26.632020
4-(2-furanyl)-N-(3-pyridinylmethyl)-6-(trifluoromethyl)-2-pyrimidinamineRattus norvegicus (Norway rat)Potency39.810710
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-methyl-4-oxo-1-phthalazinyl)acetamideRattus norvegicus (Norway rat)Potency35.481310
4-[[2-(3-ethylanilino)-3,4-dioxo-1-cyclobutenyl]amino]-1-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
3-[[(3-methoxyphenyl)-oxomethyl]amino]-2-benzofurancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency89.125120
2-[(3-bromo-5,7-dimethyl-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzoxazoleRattus norvegicus (Norway rat)Potency56.234110
4-[[2-[4-(4-chlorophenyl)-1-piperazinyl]-1-oxoethyl]amino]benzoic acid methyl esterRattus norvegicus (Norway rat)Potency10.000010
2-(2-methoxyethyl)-9-methyl-4-[(4-methyl-1-piperidinyl)-oxomethyl]-1-pyrido[3,4-b]indoloneRattus norvegicus (Norway rat)Potency39.810710
N-[3-(1-azepanyl)propyl]-2-(4-morpholinyl)-3-oxo-4H-1,4-benzothiazine-6-carboxamideRattus norvegicus (Norway rat)Potency22.387210
2-amino-4-[5-methyl-2-(methylthio)-3-thiophenyl]-5-oxo-1-(3-pyridinyl)-4,6,7,8-tetrahydroquinoline-3-carbonitrileRattus norvegicus (Norway rat)Potency8.912510
2-(1-ethoxycarbonyl-4-piperidinyl)-1,3-dioxo-5-isoindolecarboxylic acidRattus norvegicus (Norway rat)Potency0.100010
3-(2-furanylmethyl)-5-(2-methoxyethyl)-1,3,5-thiadiazinane-2-thioneRattus norvegicus (Norway rat)Potency17.782810
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-(7-methoxy-2-furo[2,3-b]quinolinyl)methanoneRattus norvegicus (Norway rat)Potency56.234110
7-[(4-methyl-1-piperazinyl)methyl]-5-(phenylmethoxymethyl)-8-quinolinolRattus norvegicus (Norway rat)Potency79.432810
3-methyl-N-[2-(4-morpholinyl)ethyl]-1-phenyl-5-thieno[2,3-c]pyrazolecarboxamideRattus norvegicus (Norway rat)Potency19.952610
3-(2-chlorophenyl)-5-methyl-N-[3-(3-methyl-2-imidazo[1,2-a]pyrimidinyl)phenyl]-4-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency26.468520
savirinRattus norvegicus (Norway rat)Potency15.649820
6,7-dimethoxy-4-(2-oxolanylmethylamino)-1H-quinazoline-2-thioneRattus norvegicus (Norway rat)Potency70.794610
2-(2-methoxyethyl)-9-methyl-1-oxo-N-(thiophen-2-ylmethyl)-4-pyrido[3,4-b]indolecarboxamideRattus norvegicus (Norway rat)Potency22.387210
2-chloro-6-[4-morpholinyl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneRattus norvegicus (Norway rat)Potency50.118710
4-[[9-methyl-2-(2-methylpropyl)-1-oxo-4-pyrido[3,4-b]indolyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency56.234110
N-(4-fluorophenyl)-6-methyl-1-propyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carboxamideRattus norvegicus (Norway rat)Potency1.000010
N-(2-chlorophenyl)-5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-methyl-2-benzofurancarboxamideRattus norvegicus (Norway rat)Potency5.011910
2-[3-[3-(2-furanylmethylamino)-3-oxopropyl]-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]acetic acid (phenylmethyl) esterRattus norvegicus (Norway rat)Potency35.481310
acetic acid [2-(1-acetyl-6-indolyl)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency44.668410
1-[(5,7-dimethyl-3-pyrazolo[1,5-a]pyrimidinyl)-oxomethyl]-4-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency31.622810
6,7-dimethoxy-N-[(5-methyl-2-furanyl)methyl]-2-(2-methylpropyl)-1-oxo-4-isoquinolinecarboxamideRattus norvegicus (Norway rat)Potency19.952610
N-(2-furanylmethyl)-N'-[4-methyl-2-(4-methyl-1-piperazinyl)-6-quinolinyl]butanediamideRattus norvegicus (Norway rat)Potency50.118710
3-[5-(4-fluorophenyl)-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-1-propanolRattus norvegicus (Norway rat)Potency39.310620
N-(3,4-dimethylphenyl)-5-(2-furanyl)-3-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
5-(1,3-benzodioxol-5-yl)-3-[3-(methylthio)phenyl]-1H-imidazol-2-oneRattus norvegicus (Norway rat)Potency15.848910
N-(2-furanylmethyl)-3-[3-[(4-methoxyphenyl)methyl]-2-imidazo[4,5-b]pyridinyl]propanamideRattus norvegicus (Norway rat)Potency56.234110
1-[(6-methoxy-2-furo[2,3-b]quinolinyl)-oxomethyl]-4-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency44.668410
N-(3,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideRattus norvegicus (Norway rat)Potency50.118710
N-[2-(dipropylamino)ethyl]-4-methyl-2-furo[3,2-c]quinolinecarboxamideRattus norvegicus (Norway rat)Potency89.125110
4-[[3-[(2-furanylmethylamino)-oxomethyl]-7-methoxy-1-benzopyran-2-ylidene]amino]benzoic acidRattus norvegicus (Norway rat)Potency89.125110
N-(2-furanylmethyl)-1-[2-(2-hydroxyethoxy)ethyl]-2-imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency22.387210
N-(3-methoxyphenyl)-2-(1-methyl-3-indolyl)acetamideRattus norvegicus (Norway rat)Potency28.183810
2-[[3-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]-N-(2-oxolanylmethyl)acetamideRattus norvegicus (Norway rat)Potency19.952610
6-methoxy-N-(thiophen-2-ylmethyl)-2-furo[2,3-b]quinolinecarboxamideRattus norvegicus (Norway rat)Potency14.125410
4-oxo-4-[5-(1,2,3,4-tetrahydronaphthalen-1-ylsulfamoyl)-2,3-dihydroindol-1-yl]butanoic acidRattus norvegicus (Norway rat)Potency0.794310
2-cyclohexyl-9-methyl-1-oxo-N-[3-(2-oxo-1-pyrrolidinyl)propyl]-4-pyrido[3,4-b]indolecarboxamideRattus norvegicus (Norway rat)Potency89.125110
N-[2-(3,4-diethoxyphenyl)ethyl]-1-[6-(4-morpholinyl)-3-pyridazinyl]-4-piperidinecarboxamideRattus norvegicus (Norway rat)Potency56.234110
cambinolRattus norvegicus (Norway rat)Potency29.934910
N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-[(5-methyl-2-furanyl)methylamino]-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]carbamic acid (phenylmethyl) esterRattus norvegicus (Norway rat)Potency56.234110
N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamineRattus norvegicus (Norway rat)Potency25.118910
5-amino-2-(3-nitrophenyl)-1-phenyl-2H-pyrrole-3,3,4-tricarbonitrileRattus norvegicus (Norway rat)Potency12.589310
LSM-28187Rattus norvegicus (Norway rat)Potency39.592620
2,6-dimethyl-4-(4-phenyl-2-quinolinyl)morpholineRattus norvegicus (Norway rat)Potency70.794610
N-[[4-(dimethylamino)phenyl]methyl]-1-ethyl-5-benzimidazolamineRattus norvegicus (Norway rat)Potency10.266310
2-(3-thiophenyl)acetic acid [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] esterRattus norvegicus (Norway rat)Potency35.481310
2-[(5-amino-1H-1,2,4-triazol-3-yl)thio]-N-(2-bromo-4-nitrophenyl)acetamideRattus norvegicus (Norway rat)Potency2.511910
5-hydroxy-2-methyl-4-[1-piperidinyl(3-pyridinyl)methyl]-3-benzo[g]benzofurancarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency7.079510
N-(5-acetyl-2-phenyl-4-sulfanylidene-1H-pyrimidin-6-yl)benzamideRattus norvegicus (Norway rat)Potency1.122010
1-(6-methyl-2-pyridinyl)-3-[3-(trifluoromethyl)phenyl]thioureaRattus norvegicus (Norway rat)Potency3.548110
1-(3-ethoxypropyl)-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency56.234110
2-(trifluoromethyl)-3-imidazo[1,2-a]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.810710
6-amino-5-cyano-2-(4-methoxyphenyl)-4-(3-pyridinyl)-4H-pyran-3-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
4-[[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholineRattus norvegicus (Norway rat)Potency50.118710
gw 7647Rattus norvegicus (Norway rat)Potency56.234110
N-(6-ethoxy-1,3-benzothiazol-2-yl)-4-methoxy-3-(4-morpholinylsulfonyl)benzamideRattus norvegicus (Norway rat)Potency89.125110
N-[4-[2-(2-ethyl-1-oxobutyl)-3-phenyl-3,4-dihydropyrazol-5-yl]phenyl]methanesulfonamideRattus norvegicus (Norway rat)Potency44.964720
2-(2-methoxyphenyl)-1-methyl-3,5-dinitro-2H-pyridineRattus norvegicus (Norway rat)Potency50.118710
5-[[(3,4-dichloroanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency1.258910
2-methyl-N'-[2-[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]benzohydrazideRattus norvegicus (Norway rat)Potency0.100010
2-fluoro-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)benzamideRattus norvegicus (Norway rat)Potency0.100010
2-[[2-(4-methoxyphenyl)-6-methyl-1-benzopyran-4-ylidene]amino]-4-methylpentanoic acidRattus norvegicus (Norway rat)Potency69.621920
1-butyl-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency44.668410
7-methoxy-2-(3-methoxyanilino)-3-quinolinecarbonitrileRattus norvegicus (Norway rat)Potency94.562620
N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-[4-methyl-4-(4-methylphenyl)-2,5-dioxo-1-imidazolidinyl]acetamideRattus norvegicus (Norway rat)Potency1.122010
N,N-dimethylcarbamodithioic acid (1-acetamido-2,2,2-trichloroethyl) esterRattus norvegicus (Norway rat)Potency19.952610
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinolRattus norvegicus (Norway rat)Potency89.125110
ro 41-0960Rattus norvegicus (Norway rat)Potency63.873920
7-[[2-(4-chloro-3-methyl-1-pyrazolyl)-1-oxopropyl]amino]-3-[[(1-methyl-5-tetrazolyl)thio]methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidRattus norvegicus (Norway rat)Potency28.183810
LSM-16990Rattus norvegicus (Norway rat)Potency25.118910
5-bromo-N-[3-[methyl(phenyl)sulfamoyl]phenyl]-3-pyridinecarboxamideRattus norvegicus (Norway rat)Potency39.810710
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinolRattus norvegicus (Norway rat)Potency4.466810
6-amino-5-cyano-4-(2-fluorophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyridine-3-carboxamideRattus norvegicus (Norway rat)Potency50.118710
1-(1,3-benzoxazol-2-yl)-N-[(4-ethylphenyl)methyl]-3-piperidinecarboxamideRattus norvegicus (Norway rat)Potency56.234110
N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-methyl-3-pyrazolecarboxamideRattus norvegicus (Norway rat)Potency31.622810
2-benzoylimino-1-(2-furanylmethyl)-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency45.857720
2-amino-4-(2-ethoxyphenyl)-6,7-dimethyl-5-oxo-4H-pyrano[3,2-c]pyridine-3-carbonitrileRattus norvegicus (Norway rat)Potency12.589310
N-[5-ethyl-3-[(4-fluorophenyl)-(4-morpholinyl)methyl]-2-thiophenyl]benzamideRattus norvegicus (Norway rat)Potency19.952610
valproateRattus norvegicus (Norway rat)Potency0.371620
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olRattus norvegicus (Norway rat)Potency12.589310
1-(4-methoxyphenyl)-3-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)pyrrolidine-2,5-dioneRattus norvegicus (Norway rat)Potency25.118910
N-(6-acetamido-3-prop-2-enyl-1,3-benzothiazol-2-ylidene)cyclohexanecarboxamideRattus norvegicus (Norway rat)Potency17.782810
4-[1-(4-bromophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneRattus norvegicus (Norway rat)Potency10.000010
2-chloro-8-[4-morpholinyl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneRattus norvegicus (Norway rat)Potency25.118910
N-(6-acetamido-3-prop-2-enyl-1,3-benzothiazol-2-ylidene)-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency44.668410
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-dimethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolamineRattus norvegicus (Norway rat)Potency64.775820
2-[2-[(5-chloro-2-thiophenyl)-oxomethyl]imino-6-fluoro-1,3-benzothiazol-3-yl]acetic acid methyl esterRattus norvegicus (Norway rat)Potency25.118910
4-[4-dimethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolyl]morpholineRattus norvegicus (Norway rat)Potency33.997220
obtusininRattus norvegicus (Norway rat)Potency32.464820
2-[4-methoxy-3-(4-morpholinylmethyl)phenyl]-3-(phenylmethyl)-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency84.279020
N-(4-fluorophenyl)-2-(3-methyl-5-oxo-1-phenyl-4H-pyrazol-4-yl)-2-oxoacetamideRattus norvegicus (Norway rat)Potency63.095710
N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]-5-nitro-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency56.234110
6-[2-(1-azepanyl)-2-oxoethoxy]-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-oneRattus norvegicus (Norway rat)Potency56.234110
1-[(2,6-dichlorophenyl)methyl]-5-(4-methylphenyl)-2-oxo-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency26.651420
2-thiophen-2-yl-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterRattus norvegicus (Norway rat)Potency28.183810
sb 242084Rattus norvegicus (Norway rat)Potency39.810710
pd 168,077Rattus norvegicus (Norway rat)Potency36.951030
acetic acid 2-(7-oxo-2,3-dihydrofuro[3,2-g][1]benzopyran-2-yl)propan-2-yl esterRattus norvegicus (Norway rat)Potency56.234110
brl 15572Rattus norvegicus (Norway rat)Potency21.192320
N-[2-[(3-nitrophenyl)methylthio]-4-oxo-3-quinazolinyl]benzamideRattus norvegicus (Norway rat)Potency15.848910
5-[2-[3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]-2-(phenylmethyl)-3,4-dihydroisoquinolin-1-oneRattus norvegicus (Norway rat)Potency9.520920
5-(4-ethoxyphenyl)-1,3-diphenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-4,6-dioneRattus norvegicus (Norway rat)Potency79.432820
mrs 1523Rattus norvegicus (Norway rat)Potency59.530010
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideRattus norvegicus (Norway rat)Potency35.481310
ML162Rattus norvegicus (Norway rat)Potency14.125410
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideRattus norvegicus (Norway rat)Potency14.125410
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideRattus norvegicus (Norway rat)Potency11.220210
2-[(2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)oxy]-N-heptylacetamideRattus norvegicus (Norway rat)Potency15.848910
3-ethyl-2-sulfanylidene-5-thiophen-2-yl-1H-thieno[2,3-d]pyrimidin-4-oneRattus norvegicus (Norway rat)Potency1.122010
6-[(4-bromophenyl)-(1-pyrrolidinyl)methyl]-1,3-benzodioxol-5-olRattus norvegicus (Norway rat)Potency2.511910
2-[1-(2-methylphenyl)-3-oxo-3-thiophen-2-ylpropyl]propanedinitrileRattus norvegicus (Norway rat)Potency10.000010
10-[3-(dibutylamino)-2-hydroxypropyl]-9-acridinoneRattus norvegicus (Norway rat)Potency75.113720
5-[(4-chlorophenyl)-oxomethyl]-4-hydroxy-6-[5-(2-nitrophenyl)-2-furanyl]-4-(trifluoromethyl)-1,3-diazinan-2-oneRattus norvegicus (Norway rat)Potency50.118710
2-(4-ethoxyphenyl)-N-[3-(1-imidazolyl)propyl]-4-quinolinecarboxamideRattus norvegicus (Norway rat)Potency67.833420
7-ethoxy-3-[5-(2-furanyl)-2-methylsulfonyl-3,4-dihydropyrazol-3-yl]-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency19.952610
2-chloro-N-(2-methyl-6-oxo-5H-benzo[b][1,4]benzoxazepin-8-yl)acetamideRattus norvegicus (Norway rat)Potency56.234110
LSM-24581Rattus norvegicus (Norway rat)Potency79.432810
N-(4-bromophenyl)-5-methyl-4-nitro-1H-pyrazol-3-amineRattus norvegicus (Norway rat)Potency70.794610
l 152804Rattus norvegicus (Norway rat)Potency56.234110
2-methyl-3-nitro-N-[4-[[(1-oxopropylamino)-sulfanylidenemethyl]amino]phenyl]benzamideRattus norvegicus (Norway rat)Potency8.912510
2-amino-5-(1-benzotriazolyl)-6-methyl-4-phenyl-4H-pyran-3-carbonitrileRattus norvegicus (Norway rat)Potency50.118710
1-bromo-3-(5,5-dimethyl-3-phenyl-4H-pyrazolo[4,3-a]carbazol-10-yl)-2-propanolRattus norvegicus (Norway rat)Potency22.387210
LSM-17147Rattus norvegicus (Norway rat)Potency35.481310
3-methyl-N-[[[(4-nitrophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]butanamideRattus norvegicus (Norway rat)Potency19.974020
1-amino-N-methyl-5-(4-morpholinyl)-N-phenyl-6,7,8,9-tetrahydrothieno[2,3-c]isoquinoline-2-carboxamideRattus norvegicus (Norway rat)Potency28.183810
N-methyl-5-phenyl-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency31.622810
6-amino-4-(1-cyclohex-2-enyl)-3-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileRattus norvegicus (Norway rat)Potency70.794610
AnthraniloyllycoctonineRattus norvegicus (Norway rat)Potency35.481310
3,5-diethyl-2-(3-hydroxypropylamino)-5-methyl-6H-benzo[h]quinazolin-4-oneRattus norvegicus (Norway rat)Potency8.643820
N-[(5-quinolinylamino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency50.118710
2-Chloro-1-[5-(3,4-dimethoxyphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneRattus norvegicus (Norway rat)Potency7.943310
LSM-31277Rattus norvegicus (Norway rat)Potency56.234120
2-amino-4-(2-fluorophenyl)-6-(3-pyridinyl)-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency28.183810
N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideRattus norvegicus (Norway rat)Potency0.891310
3-(2,4-dichloro-5-methoxyphenyl)-2-sulfanyl-4(3h)-quinazolinoneRattus norvegicus (Norway rat)Potency0.141310
4-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-3-oxobutanoic acid ethyl esterRattus norvegicus (Norway rat)Potency3.162310
4-[[(2-methyl-5-nitro-1H-imidazol-4-yl)thio]methyl]-2-nitrophenolRattus norvegicus (Norway rat)Potency25.118910
3-(3,4-dimethylphenyl)sulfonyl-2-imino-1-prop-2-enyl-5-dipyrido[1,2-e-4',3'-f]pyrimidinoneRattus norvegicus (Norway rat)Potency69.621920
5-amino-2-(diethylamino)-N-(2-methoxyphenyl)benzenesulfonamideRattus norvegicus (Norway rat)Potency6.309610
N-(2-chlorophenyl)-4-[[(2-methoxy-4-nitroanilino)-sulfanylidenemethyl]hydrazo]-4-oxobutanamideRattus norvegicus (Norway rat)Potency8.912510
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleRattus norvegicus (Norway rat)Potency7.943310
or486Rattus norvegicus (Norway rat)Potency45.373610
3-(2-methoxyphenyl)-2-methyl-4-oxo-1H-quinazoline-2-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency28.183810
fg 9041Rattus norvegicus (Norway rat)Potency4.242120
4-chloro-5-(2,3-dihydro-1,4-benzodioxin-3-yl)thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency44.668410
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-methyl-2,5-dioxo-4-(2-phenylethyl)-1-imidazolidinyl]acetamideRattus norvegicus (Norway rat)Potency79.432810
suramin sodiumRattus norvegicus (Norway rat)Potency14.125410
(4-chlorophenyl)-[4-(8-nitro-5-quinolinyl)-1-piperazinyl]methanoneRattus norvegicus (Norway rat)Potency4.744410
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(2-methoxy-4-methylphenyl)-2-thiophenecarboxamideRattus norvegicus (Norway rat)Potency46.779120
N-[4-[[(4-tert-butylphenyl)-oxomethyl]amino]phenyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency33.117020
N-[4-[cyano-[3-(3-hydroxypropylamino)-2-quinoxalinyl]methyl]sulfonylphenyl]acetamideRattus norvegicus (Norway rat)Potency78.161420
2-amino-1-(dimethylamino)-4-(1-naphthalenyl)-5-oxo-7-phenyl-4,6,7,8-tetrahydroquinoline-3-carbonitrileRattus norvegicus (Norway rat)Potency0.141310
2-(1H-indol-3-yl)-8-methylimidazo[1,2-a]pyridineRattus norvegicus (Norway rat)Potency28.796820
4-(1H-benzimidazol-2-ylthio)-1-[4-(4-nitrophenyl)-1-piperazinyl]-1-butanoneRattus norvegicus (Norway rat)Potency3.162310
2-hydroxybenzoic acid [2-(2-ethoxyanilino)-2-oxo-1-phenylethyl] esterRattus norvegicus (Norway rat)Potency89.125110
N-(2,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideRattus norvegicus (Norway rat)Potency59.621820
[4-[(2-chlorophenyl)methylsulfonyl]-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneRattus norvegicus (Norway rat)Potency17.782810
2-amino-4-(3,4-dimethoxyphenyl)-7,7-dimethyl-5-oxo-1-(3-pyridinyl)-6,8-dihydro-4H-quinoline-3-carbonitrileRattus norvegicus (Norway rat)Potency17.782810
5-bromo-N-[(1,2-dimethyl-5-indolyl)methyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency8.912510
3-(2-chlorophenyl)-N-[5-(2,4-dichlorophenyl)-1,3,4-thiadiazol-2-yl]-5-methyl-4-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency31.622810
2-[[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]-1-oxo-5-isoquinolinyl]oxy]propanoic acid ethyl esterRattus norvegicus (Norway rat)Potency0.298820
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidRattus norvegicus (Norway rat)Potency79.432810
4-[4-diethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolyl]morpholineRattus norvegicus (Norway rat)Potency33.997220
3-hydroxy-6-(hydroxymethyl)-2-[(3-methoxyphenyl)-(2-pyridinylamino)methyl]-4-pyranoneRattus norvegicus (Norway rat)Potency70.794610
N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)-2,3-dihydro-1,4-benzodioxin-6-carboxamideRattus norvegicus (Norway rat)Potency44.668410
3-nitro-N-[(3-sulfamoylanilino)-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency12.589310
1-[[2-(2,4-dichlorophenoxy)-1-oxoethyl]amino]-3-(4-methoxyphenyl)thioureaRattus norvegicus (Norway rat)Potency15.848910
[4-(butan-2-ylamino)-6-chloro-1,3,5-triazin-2-yl]-[(1,1,3-trioxo-1,2-benzothiazol-2-yl)methyl]cyanamideRattus norvegicus (Norway rat)Potency79.432810
2-(4-tert-butylphenyl)sulfinyl-4,6-dimethyl-3-thieno[2,3-b]pyridinamineRattus norvegicus (Norway rat)Potency31.622810
N-[3-(1-azepanylsulfonyl)-4-methylphenyl]-2-(4-quinazolinylthio)acetamideRattus norvegicus (Norway rat)Potency25.118910
iik7Rattus norvegicus (Norway rat)Potency5.972810
2-[(3-fluorophenyl)-(2-pyridinylamino)methyl]-3-hydroxy-6-(hydroxymethyl)-4-pyranoneRattus norvegicus (Norway rat)Potency19.952610
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneRattus norvegicus (Norway rat)Potency28.183810
7-methoxy-N-(3-pyridinylmethyl)-2-furo[2,3-b]quinolinecarboxamideRattus norvegicus (Norway rat)Potency28.183810
2-(4-methoxyphenyl)sulfonylquinoxalineRattus norvegicus (Norway rat)Potency79.432810
sb 415286Rattus norvegicus (Norway rat)Potency9.704620
5-methyl-4-[(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-(3-nitrophenyl)methyl]-2-phenyl-1H-pyrazol-3-oneRattus norvegicus (Norway rat)Potency7.943310
2,6-dichloro-1,7-dimethylpyrazolo[1,2-a]pyrazole-3,5-dioneRattus norvegicus (Norway rat)Potency72.679620
3-(acetyloxymethyl)-7-[[3-(4-chloro-3,5-dimethyl-1-pyrazolyl)-2-methyl-1-oxopropyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acidRattus norvegicus (Norway rat)Potency89.716420
2-(2-bromophenyl)-3-[3-(4-morpholinyl)propyl]-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency56.234110
6-amino-5-cyano-2-[[(3-cyano-6-methyl-7,8-dihydro-5H-1,6-naphthyridin-2-yl)thio]methyl]-4-(4-fluorophenyl)-4H-pyran-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency14.125410
2-(2-furanylmethylamino)benzoic acid [2-[(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency10.000010
5-[[(2-methylanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency0.794310
N-[3-(N-(2-chloro-1-oxoethyl)-4-nitroanilino)propyl]-2,2,2-trifluoroacetamideRattus norvegicus (Norway rat)Potency39.810710
N-[[(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-5-methyl-3-phenyl-4-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency6.309610
3,5-diethyl-2-(2-hydroxyethylamino)-5-methyl-6H-benzo[h]quinazolin-4-oneRattus norvegicus (Norway rat)Potency19.952610
2-[4-(3-fluorophenyl)-3-methyl-5-oxo-1,2,4-triazol-1-yl]acetonitrileRattus norvegicus (Norway rat)Potency22.387210
4-(3-chlorophenyl)sulfonyl-N-cyclohexyl-N-methyl-3-nitrobenzamideRattus norvegicus (Norway rat)Potency50.118710
2-[[2-(3,4-dimethoxyanilino)-2-oxoethyl]thio]-3-pyridinecarboxylic acid propan-2-yl esterRattus norvegicus (Norway rat)Potency0.125910
sc 560Rattus norvegicus (Norway rat)Potency37.685810
5-bromo-N-[2-(2-methyl-1-indolyl)ethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency10.000010
1-(5-nitro-2-thiophenyl)piperidineRattus norvegicus (Norway rat)Potency56.234110
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]-4-methylbenzamideRattus norvegicus (Norway rat)Potency44.668410
sc-19220Rattus norvegicus (Norway rat)Potency89.125110
le 300Rattus norvegicus (Norway rat)Potency18.852230
5-[3-(2-chloro-6-methoxy-3-quinolinyl)-5-(2-furanyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acidRattus norvegicus (Norway rat)Potency39.810710
digitoxigeninRattus norvegicus (Norway rat)Potency89.125110
2-(N-(2-chloro-1-oxoethyl)-4-fluoroanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideRattus norvegicus (Norway rat)Potency14.125410
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideRattus norvegicus (Norway rat)Potency15.848910
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideRattus norvegicus (Norway rat)Potency6.309610
1-[3-(dimethylsulfamoyl)phenyl]-3-(2-furanylmethyl)thioureaRattus norvegicus (Norway rat)Potency79.432810
2-furanyl-[4-[(6-hydroxy-2-methyl-5-thiazolo[3,2-b][1,2,4]triazolyl)-thiophen-2-ylmethyl]-1-piperazinyl]methanoneRattus norvegicus (Norway rat)Potency31.622810
LSM-27960Rattus norvegicus (Norway rat)Potency22.387210
2-[4-(2,5-diphenyl-3,4-dihydropyrazol-3-yl)-2-methoxyphenoxy]acetic acidRattus norvegicus (Norway rat)Potency56.234110
4-[1-(4-fluorophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneRattus norvegicus (Norway rat)Potency70.794610
N-(1,3-dioxo-4-isoindolyl)-2-(2,5-dioxo-1-pyrrolidinyl)acetamideRattus norvegicus (Norway rat)Potency17.488220
1-(2-methoxy-3-dibenzofuranyl)-3-(3-methylphenyl)thioureaRattus norvegicus (Norway rat)Potency56.234110
2-Chloro-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneRattus norvegicus (Norway rat)Potency12.589310
N-[5-(phenylmethyl)-2-thiazolyl]-4,5-dihydro-1H-imidazole-2-carboxamideRattus norvegicus (Norway rat)Potency10.000010
4-(1,3-dioxo-2-benzo[de]isoquinolinyl)butanoic acid [2-(2-acetylanilino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency50.118710
LSM-16446Rattus norvegicus (Norway rat)Potency31.622810
1-(3-chloro-4-methoxyphenyl)-3-(2-fluorophenyl)ureaRattus norvegicus (Norway rat)Potency89.125110
3-chloro-N-[3-(2-methoxyethyl)-6-sulfamoyl-1,3-benzothiazol-2-ylidene]-1-benzothiophene-2-carboxamideRattus norvegicus (Norway rat)Potency43.928420
1-cyclohexyl-3-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)thioureaRattus norvegicus (Norway rat)Potency89.125110
N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]-4-[(2-methyl-1-piperidinyl)sulfonyl]benzamideRattus norvegicus (Norway rat)Potency89.125110
4-[7-(2-methoxyethyl)-2,6-dioxo-3-(phenylmethyl)-8-purinyl]benzonitrileRattus norvegicus (Norway rat)Potency79.432820
3-amino-4-[(4-chlorophenyl)thio]benzoic acid methyl esterRattus norvegicus (Norway rat)Potency31.622810
5-oxo-2-pyrrolidinecarboxylic acid [2-[3-(4-methoxyphenyl)-5-(2-naphthalenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency25.118910
4-(1-imidazolyl)-3,5-dinitrobenzoic acid methyl esterRattus norvegicus (Norway rat)Potency56.234110
4-(4-propan-2-ylphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazolin-2-oneRattus norvegicus (Norway rat)Potency79.432810
LSM-31434Rattus norvegicus (Norway rat)Potency100.000010
ly 367265Rattus norvegicus (Norway rat)Potency7.638010
3-(benzenesulfonyl)-1-cyclopropyl-2-pyrrolo[3,2-b]quinoxalinamineRattus norvegicus (Norway rat)Potency31.832620
2-bromo-6-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneRattus norvegicus (Norway rat)Potency44.668410
LSM-16483Rattus norvegicus (Norway rat)Potency56.234110
3-(4-chlorophenyl)-6-(4-methyl-1-piperazinyl)-1H-pyrimidine-2,4-dioneRattus norvegicus (Norway rat)Potency79.432810
2-(3-methoxyphenyl)-3,5,6,7,8,9-hexahydrocyclohepta[2,3]thieno[2,4-b]pyrimidin-4-oneRattus norvegicus (Norway rat)Potency27.292820
[4-(4-chlorophenyl)-4,5-dihydro-1H-pyrazol-3-yl]-(2-oxiranyl)methanoneRattus norvegicus (Norway rat)Potency50.118710
5-[[2-(diethylamino)-9-methyl-4-oxo-3-pyrido[1,2-a]pyrimidinyl]methylidene]-1,3-diazinane-2,4,6-trioneRattus norvegicus (Norway rat)Potency89.125110
2-(2-furanyl)-4-mercapto-3-(4-methylphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileRattus norvegicus (Norway rat)Potency3.981110
4-dimethoxyphosphoryl-2-(1-naphthalenyl)-N-(phenylmethyl)-5-oxazolamineRattus norvegicus (Norway rat)Potency50.118710
clodronic acidRattus norvegicus (Norway rat)Potency0.631010
4-chlorobenzoic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency15.848910
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency100.000010
1-(4-methoxyphenyl)-3-[3-(1-piperidinylsulfonyl)phenyl]thioureaRattus norvegicus (Norway rat)Potency7.079510
N-[4-(4-fluorophenyl)-2-thiazolyl]-3-methoxy-4-[2-(4-morpholinyl)-2-oxoethoxy]benzamideRattus norvegicus (Norway rat)Potency14.125410
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[[oxo-[(phenylmethyl)amino]methyl]amino]ethyl] esterRattus norvegicus (Norway rat)Potency17.782810
3-[4-(4-butan-2-ylphenyl)sulfonyl-1-piperazinyl]butanoic acidRattus norvegicus (Norway rat)Potency39.810710
4-[[[1-oxo-2-[(2-oxo-3-phenyl-1-benzopyran-7-yl)oxy]propyl]amino]methyl]-1-cyclohexanecarboxylic acidRattus norvegicus (Norway rat)Potency14.976320
acetic acid [1-[(4,8-dimethoxy-7-furo[2,3-b]quinolinyl)oxy]-3-hydroxy-3-methylbutan-2-yl] esterRattus norvegicus (Norway rat)Potency28.183810
2-[(4-acetamidophenyl)sulfonylamino]acetic acid [7-(ethoxycarbonylamino)-2-oxo-1-benzopyran-4-yl]methyl esterRattus norvegicus (Norway rat)Potency31.673420
LSM-24516Rattus norvegicus (Norway rat)Potency25.118910
LSM-28572Rattus norvegicus (Norway rat)Potency28.183810
2-(Chloroacetyl)-N,2-diphenylhydrazinecarboxamideRattus norvegicus (Norway rat)Potency7.943310
2-chloro-1-[1-(3-isoxazolyl)-2,5-dimethyl-3-pyrrolyl]ethanoneRattus norvegicus (Norway rat)Potency79.432810
N-[[[2-(2-naphthalenyloxy)-1-oxopropyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency22.387210
LSM-28172Rattus norvegicus (Norway rat)Potency36.041520
2-Chloro-1-[5-(furan-2-yl)-3-(5-methylfuran-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneRattus norvegicus (Norway rat)Potency22.387210
2-(2-chloro-1-oxoethyl)-3,4-dihydro-1H-isoquinoline-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency14.125410
5-(4-methylphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acidRattus norvegicus (Norway rat)Potency48.022420
N-[2-(4-methoxyphenyl)-4-oxo-1,2-dihydroquinazolin-3-yl]carbamic acid ethyl esterRattus norvegicus (Norway rat)Potency56.234110
cgp 7930Rattus norvegicus (Norway rat)Potency34.466520
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acidRattus norvegicus (Norway rat)Potency0.631010
[3-(2-hydroxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-thiophen-2-ylmethanoneRattus norvegicus (Norway rat)Potency79.432810
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazoleRattus norvegicus (Norway rat)Potency37.685810
N,N-dimethyl-3-(3-oxo-1,2-benzothiazol-2-yl)benzenesulfonamideRattus norvegicus (Norway rat)Potency14.125410
N-(3-oxo-2-benzo[f][1]benzopyranyl)acetamideRattus norvegicus (Norway rat)Potency21.314520
N-[4-methyl-2-(4-morpholinyl)-6-quinolinyl]cyclohexanecarboxamideRattus norvegicus (Norway rat)Potency79.432810
2-(4-fluoro-3-nitrophenyl)-4,4-dimethyl-5H-oxazoleRattus norvegicus (Norway rat)Potency17.782810
Meranzin hydrateRattus norvegicus (Norway rat)Potency28.183810
N-[1-[(4-fluorophenyl)methyl]-4-pyrazolyl]-5-(2-furanyl)-3-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency89.125110
5-(2,4-dichlorophenyl)-4,6-dioxo-3a,6a-dihydro-2H-pyrrolo[3,4-d]isoxazole-3,3-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency44.668410
2-[3-(2-furanylmethyl)-2-(4-methoxyphenyl)imino-4-oxo-5-thiazolidinyl]-N-(2-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency79.432810
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideRattus norvegicus (Norway rat)Potency0.707910
3,7-dibutyl-3,7-dimethyl-2,6-dihydro-[1,2,4]triazolo[1,2-a][1,2,4]triazole-1,5-dithioneRattus norvegicus (Norway rat)Potency25.118910
2-(4-acetyl-1-piperazinyl)-6-amino-4-(cyanomethyl)pyridine-3,5-dicarbonitrileRattus norvegicus (Norway rat)Potency7.943310
3-(5,7-diphenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-1-propanolRattus norvegicus (Norway rat)Potency79.432820
5-[(2,4-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]-4-pyrazolyl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency35.481310
4,5,6,7-tetrabromobenzimidazoleRattus norvegicus (Norway rat)Potency5.011910
4-[3-(2-chloro-1-oxoethyl)-2,5-dimethyl-1-pyrrolyl]-1,5-dimethyl-2-phenyl-3-pyrazoloneRattus norvegicus (Norway rat)Potency8.912510
2-[[3-butyl-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideRattus norvegicus (Norway rat)Potency39.810710
N-[[(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-2-methylbenzamideRattus norvegicus (Norway rat)Potency2.238710
ncgc00099374Rattus norvegicus (Norway rat)Potency7.951820
sib 1757Rattus norvegicus (Norway rat)Potency19.744920
5-(3,4-dimethoxyphenyl)-3-(2-furanylmethyl)-4-imino-5H-[1]benzopyrano[2,3-d]pyrimidin-8-olRattus norvegicus (Norway rat)Potency50.118710
2-[3-(1-benzotriazolylmethyl)-4-methoxyphenyl]-3-(4-methoxyphenyl)-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency79.432810
fraxinRattus norvegicus (Norway rat)Potency79.432810
fraxetinRattus norvegicus (Norway rat)Potency89.125110
quercetinRattus norvegicus (Norway rat)Potency23.778110
scopoletinRattus norvegicus (Norway rat)Potency28.183810
vitamin k semiquinone radicalRattus norvegicus (Norway rat)Potency35.481310
hymecromoneRattus norvegicus (Norway rat)Potency54.195620
daphnetinRattus norvegicus (Norway rat)Potency37.685810
quercetin 3-o-methyl etherRattus norvegicus (Norway rat)Potency44.668410
cyclosporineRattus norvegicus (Norway rat)Potency11.953840
senecionineRattus norvegicus (Norway rat)Potency25.118910
gamma-linolenic acidRattus norvegicus (Norway rat)Potency70.794610
alpha-linolenic acidRattus norvegicus (Norway rat)Potency79.432810
harmineRattus norvegicus (Norway rat)Potency56.234110
genisteinRattus norvegicus (Norway rat)Potency1.122010
prochlorperazine maleateRattus norvegicus (Norway rat)Potency18.887610
methysergide maleateRattus norvegicus (Norway rat)Potency89.716420
fucoxanthinRattus norvegicus (Norway rat)Potency35.481310
harmanRattus norvegicus (Norway rat)Potency46.769030
esculetinRattus norvegicus (Norway rat)Potency67.833420
pteryxinRattus norvegicus (Norway rat)Potency56.234110
7-hydroxycoumarinRattus norvegicus (Norway rat)Potency67.833420
morinRattus norvegicus (Norway rat)Potency38.815710
myricetinRattus norvegicus (Norway rat)Potency23.119730
7-hydroxy-6,4'-dimethoxyisoflavoneRattus norvegicus (Norway rat)Potency89.125110
coumestrolRattus norvegicus (Norway rat)Potency36.426110
daidzeinRattus norvegicus (Norway rat)Potency11.920430
caffeic acid phenethyl esterRattus norvegicus (Norway rat)Potency0.223910
acteosideRattus norvegicus (Norway rat)Potency44.668410
puerarinRattus norvegicus (Norway rat)Potency31.622810
rottlerinRattus norvegicus (Norway rat)Potency15.102720
n-oleoyldopamineRattus norvegicus (Norway rat)Potency49.427740
cilnidipineRattus norvegicus (Norway rat)Potency25.118910
domoic acidRattus norvegicus (Norway rat)Potency14.125410
trimipramine maleateRattus norvegicus (Norway rat)Potency0.211910
4-hydroxyestradiolRattus norvegicus (Norway rat)Potency19.952610
menatetrenoneRattus norvegicus (Norway rat)Potency17.782810
isotretinoinRattus norvegicus (Norway rat)Potency31.941820
xylometazoline hydrochlorideRattus norvegicus (Norway rat)Potency79.432810
ketotifen fumarateRattus norvegicus (Norway rat)Potency37.685810
indocyanine greenRattus norvegicus (Norway rat)Potency3.548110
triprolidineRattus norvegicus (Norway rat)Potency0.707920
10-octadecenoic acid, (z)-isomerRattus norvegicus (Norway rat)Potency25.553620
n-arachidonylglycineRattus norvegicus (Norway rat)Potency24.968420
n-oleoylethanolamineRattus norvegicus (Norway rat)Potency29.417030
phenoxybenzamine hydrochlorideRattus norvegicus (Norway rat)Potency44.668410
phenylephrine hydrochlorideRattus norvegicus (Norway rat)Potency1.337110
brefeldin aRattus norvegicus (Norway rat)Potency56.234110
fenretinideRattus norvegicus (Norway rat)Potency31.286740
ic 261Rattus norvegicus (Norway rat)Potency79.432810
as 605240Rattus norvegicus (Norway rat)Potency1.412510
su 9516Rattus norvegicus (Norway rat)Potency6.691810
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acidRattus norvegicus (Norway rat)Potency29.261740
7-hydroxy-8-[[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-4-methyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency33.997220
2-[3-(diethylamino)propylamino]-4-(methoxymethyl)-6-methyl-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency25.118910
8-(1-piperidinylsulfonyl)-6-pyrido[1,2-a]quinazolinoneRattus norvegicus (Norway rat)Potency89.716420
1-[(2-oxo-3,4-dihydro-1H-quinolin-6-yl)sulfonyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-piperidinecarboxamideRattus norvegicus (Norway rat)Potency7.079510
[4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-[1,2,4]triazolo[4,3-a]quinoxalin-8-yl]-phenylmethanoneRattus norvegicus (Norway rat)Potency79.432810
3-(4-chlorophenyl)-1-methyl-N-[(5-methyl-2-furanyl)methyl]-5-thieno[2,3-c]pyrazolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
2-[[5-methyl-2-(3-methylphenyl)-4-oxazolyl]methylsulfinyl]-N-(2-oxolanylmethyl)acetamideRattus norvegicus (Norway rat)Potency17.782810
3-(4-chlorophenyl)-1-methyl-N-[3-(1-pyrrolidinyl)propyl]-5-thieno[2,3-c]pyrazolecarboxamideRattus norvegicus (Norway rat)Potency89.125110
N-(4-ethylphenyl)-2-(2-furanylmethyl)-1,3-dioxo-5-isoindolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
N-(2-furanylmethyl)-3-(2,4,8,10-tetramethyl-3-pyrido[2,3]pyrazolo[2,4-a]pyrimidinyl)propanamideRattus norvegicus (Norway rat)Potency79.432810
4-[1-[(4-methyl-2-oxo-1-benzopyran-7-yl)amino]-3-oxo-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency11.392620
N-(6-acetyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenyl-3-pyrazolecarboxamideRattus norvegicus (Norway rat)Potency19.952610
N-[(2-methoxyphenyl)methyl]-1-(8-quinolinylsulfonyl)-4-piperidinecarboxamideRattus norvegicus (Norway rat)Potency0.022410
2-[[2-(3,4-dimethoxyphenyl)-5-methyl-4-oxazolyl]methylsulfinyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideRattus norvegicus (Norway rat)Potency28.183810
2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]-N-(2-oxolanylmethyl)acetamideRattus norvegicus (Norway rat)Potency89.125110
N-[2-(4-morpholinyl)ethyl]-4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazine-6-carboxamideRattus norvegicus (Norway rat)Potency28.183810
3-(4-chlorophenyl)-N-[2-(diethylamino)ethyl]-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
8-(2-chlorophenyl)-3-(4-ethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrileRattus norvegicus (Norway rat)Potency17.782810
N-(2-ethoxyphenyl)-[1,2,4]triazolo[4,3-a]quinoxalin-4-amineRattus norvegicus (Norway rat)Potency28.183810
N-[3-(4-methyl-1-piperazinyl)propyl]-4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazine-6-carboxamideRattus norvegicus (Norway rat)Potency84.279020
N-(4-methyl-1,3-benzothiazol-2-yl)-2-(1-pyrrolyl)acetamideRattus norvegicus (Norway rat)Potency28.183810
N-(5-methyl-3-isoxazolyl)-2-[[3-(3-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]acetamideRattus norvegicus (Norway rat)Potency89.125110
6-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-3-ethyl-1H-pyrimidine-2,4-dioneRattus norvegicus (Norway rat)Potency7.943310
1-(4-morpholinyl)-2-[[3-(2-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]ethanoneRattus norvegicus (Norway rat)Potency79.432810
2-(2-chlorophenyl)-9-(3-methylphenyl)-8-oxo-7H-purine-6-carboxamideRattus norvegicus (Norway rat)Potency5.011910
7-hydroxy-8-(4-morpholinylmethyl)-3-phenyl-1-benzopyran-4-oneRattus norvegicus (Norway rat)Potency79.432820
4-aminocrotonic acidRattus norvegicus (Norway rat)Potency42.284120
olvanilRattus norvegicus (Norway rat)Potency17.681230
preclamolRattus norvegicus (Norway rat)Potency10.189430
k 185Rattus norvegicus (Norway rat)Potency30.990530
l 655,708Rattus norvegicus (Norway rat)Potency4.228410
al 8810Rattus norvegicus (Norway rat)Potency0.631010
cytochalasin bRattus norvegicus (Norway rat)Potency60.456610
ml 10302Rattus norvegicus (Norway rat)Potency0.199510
pd 128907Rattus norvegicus (Norway rat)Potency0.455730
exp 655Rattus norvegicus (Norway rat)Potency0.707910
vinorelbineRattus norvegicus (Norway rat)Potency28.183810
(3r)-((2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl))methanoneRattus norvegicus (Norway rat)Potency15.003010
su 6656Rattus norvegicus (Norway rat)Potency24.891520
ro 4-6790Rattus norvegicus (Norway rat)Potency17.782810
7,7-dimethyl-5,8-eicosadienoic acidRattus norvegicus (Norway rat)Potency19.902510
3,5-dimethoxy-trans-stilbeneRattus norvegicus (Norway rat)Potency71.772220
neoglycyrolRattus norvegicus (Norway rat)Potency14.125410
salazinic acidRattus norvegicus (Norway rat)Potency50.118710
4-[(3aR,4S,9bS)-8-[(4-methoxyphenyl)sulfamoyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-4-yl]benzoic acidRattus norvegicus (Norway rat)Potency56.234110
furazolidoneRattus norvegicus (Norway rat)Potency11.220210
1-Ethyl-9H-pyrido[3,4-b]indoleRattus norvegicus (Norway rat)Potency56.234110
casein kinase iiRattus norvegicus (Norway rat)Potency8.436840
erbstatinRattus norvegicus (Norway rat)Potency70.794610
ag 538Rattus norvegicus (Norway rat)Potency19.163830
tyrphostin ag 555Rattus norvegicus (Norway rat)Potency28.294410
tyrphostin ag-494Rattus norvegicus (Norway rat)Potency25.125630
tyrphostin b44Rattus norvegicus (Norway rat)Potency54.350630
ag-490Rattus norvegicus (Norway rat)Potency23.899020
ag 112Rattus norvegicus (Norway rat)Potency25.725020
ag 183Rattus norvegicus (Norway rat)Potency79.432810
semaxinibRattus norvegicus (Norway rat)Potency14.673710
nifuroxazideRattus norvegicus (Norway rat)Potency19.952610
8-(3-chlorostyryl)caffeineRattus norvegicus (Norway rat)Potency14.220440
bay 11-7082Rattus norvegicus (Norway rat)Potency0.543730
bay 11-7085Rattus norvegicus (Norway rat)Potency1.393220
molsidomineRattus norvegicus (Norway rat)Potency26.679510
diamideRattus norvegicus (Norway rat)Potency50.118710
5,7-dihydroxy-4-methylcoumarinRattus norvegicus (Norway rat)Potency86.288520
1-(4-methylpiperazin-1-yl)-3-(5-nitrofuran-2-yl)prop-2-en-1-oneRattus norvegicus (Norway rat)Potency10.000010
styrylquinolineRattus norvegicus (Norway rat)Potency79.432820
7-hydroxy-3-(4-methoxyphenyl)-4-methylcoumarinRattus norvegicus (Norway rat)Potency53.138020
zimeldineRattus norvegicus (Norway rat)Potency1.778310
isoalloxazineRattus norvegicus (Norway rat)Potency13.540430
7-hydroxy-4-methyl-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency15.848910
5-deazaflavinRattus norvegicus (Norway rat)Potency79.432810
7-Hydroxy-2-methylisoflavoneRattus norvegicus (Norway rat)Potency79.432810
2-(5,7-dihydroxy-4-methyl-2-oxo-1-benzopyran-3-yl)acetic acid ethyl esterRattus norvegicus (Norway rat)Potency22.404820
vinblastine sulfateRattus norvegicus (Norway rat)Potency50.118710
(5R)-3'-phenyl-1-(phenylmethyl)spiro[1,3-diazinane-5,5'-2,4,4a,6-tetrahydro-1H-pyrazino[1,2-a]quinoline]-2,4,6-trioneRattus norvegicus (Norway rat)Potency70.794610
6-ethyl-7-hydroxy-4-[[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency79.432810
7-hydroxy-6-(4-morpholinylmethyl)-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-4-oneRattus norvegicus (Norway rat)Potency51.453220
N-(2,3-dimethylphenyl)-1-methyl-9H-pyrido[3,4-b]indole-3-carboxamideRattus norvegicus (Norway rat)Potency4.466810
1-methyl-beta-carboline-3-carboxylic acidRattus norvegicus (Norway rat)Potency67.833420
3-bromo-7-hydroxy-4,8-dimethyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency89.125110
5,7-dihydroxy-4-methyl-3-(phenylmethyl)-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency46.779120
nitrofurazoneRattus norvegicus (Norway rat)Potency7.079510
cisplatinRattus norvegicus (Norway rat)Potency0.503430
naloxone hydrochlorideRattus norvegicus (Norway rat)Potency70.794610
sulindac sulfoneRattus norvegicus (Norway rat)Potency9.068810
thunberginol bRattus norvegicus (Norway rat)Potency19.952610
norbinaltorphimineRattus norvegicus (Norway rat)Potency0.303020
8-(diethylaminomethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-7-hydroxy-1-benzopyran-4-oneRattus norvegicus (Norway rat)Potency56.234110
7-hydroxy-8-methyl-4-[[methyl-(phenylmethyl)amino]methyl]-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency89.125110
nylidrin hydrochlorideRattus norvegicus (Norway rat)Potency25.118910
triprolidine hydrochloride anhydrousRattus norvegicus (Norway rat)Potency2.818410
fenoterolRattus norvegicus (Norway rat)Potency23.778110
n-(2-aminoethyl)-4-chlorobenzamide hydrochlorideRattus norvegicus (Norway rat)Potency15.003010
2',3,4-trihydroxychalconeRattus norvegicus (Norway rat)Potency19.952610
CrotaoprostrinRattus norvegicus (Norway rat)Potency50.118710
2-(dimethylaminostyryl)-1-ethylpyridiniumRattus norvegicus (Norway rat)Potency50.118710
chloride of pseudoisocyanineRattus norvegicus (Norway rat)Potency56.234110
3,8-dibromo-7-hydroxy-4-methylchromen-2-oneRattus norvegicus (Norway rat)Potency25.118910
n,n,n-trimethyl-1-(4-stilbenoxy)-2-propylammonium iodideRattus norvegicus (Norway rat)Potency0.446710
nifuratroneRattus norvegicus (Norway rat)Potency14.125410
gw-5074Rattus norvegicus (Norway rat)Potency33.525420
6-(bromomethylene)tetrahydro-3-(1-naphthaleneyl)-2h-pyran-2-oneRattus norvegicus (Norway rat)Potency2.331620
[4-(3-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneRattus norvegicus (Norway rat)Potency15.848910
7-chloro-4-hydroxy-2-phenyl-1,8-naphthyridineRattus norvegicus (Norway rat)Potency22.139720
gr 46611Rattus norvegicus (Norway rat)Potency9.916020
6-chloro-4-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-hydroxy-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency79.432810
7-(hydroxyimino)cyclopropan(b)chromen-1a-carbxoylic acid ethyl esterRattus norvegicus (Norway rat)Potency42.284110
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-1-(4-methoxyphenyl)ethanoneRattus norvegicus (Norway rat)Potency8.912510
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-N-(3-methylphenyl)acetamideRattus norvegicus (Norway rat)Potency8.912510
diacetylmonoximeRattus norvegicus (Norway rat)Potency2.238710
sinequanRattus norvegicus (Norway rat)Potency31.622810
flupirtineRattus norvegicus (Norway rat)Potency37.301610
zimelidine hydrochlorideRattus norvegicus (Norway rat)Potency16.833610
sclerotiorinRattus norvegicus (Norway rat)Potency50.118710
columbianadinRattus norvegicus (Norway rat)Potency79.432810
oxotremorine sesquifumarateRattus norvegicus (Norway rat)Potency37.685810
ly 53857Rattus norvegicus (Norway rat)Potency0.125910
chaetoglobosin ARattus norvegicus (Norway rat)Potency50.118710
marminRattus norvegicus (Norway rat)Potency31.622810
su 4312Rattus norvegicus (Norway rat)Potency29.342140
3-[[(3-methoxyanilino)-oxomethyl]amino]benzoic acidRattus norvegicus (Norway rat)Potency15.848910
N-(1,3-benzodioxol-5-yl)-2-methyl-3-pyrazolecarboxamideRattus norvegicus (Norway rat)Potency89.125110
2-(1-ethyl-4-pyrazolyl)-4-quinolinecarboxylic acidRattus norvegicus (Norway rat)Potency50.118710
N-butan-2-yl-1-[2-(4-fluorophenyl)ethyl]-5-oxo-3-pyrrolidinecarboxamideRattus norvegicus (Norway rat)Potency3.162310
(3S)-2-(2-chloro-1-oxoethyl)-1,1-dimethyl-4,9-dihydro-3H-pyrido[3,4-b]indole-3-carboxylic acid methyl esterRattus norvegicus (Norway rat)Potency50.118710
a 77636Rattus norvegicus (Norway rat)Potency17.782810
n-(3-(cyclohexylidene-(1h-imidazol-4-ylmethyl))phenyl)ethanesulfonamideRattus norvegicus (Norway rat)Potency1.195810
b 43Rattus norvegicus (Norway rat)Potency12.589310
(8R)-7-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triolRattus norvegicus (Norway rat)Potency6.007630
(8R)-7-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triolRattus norvegicus (Norway rat)Potency14.662930
dilazep(2+)Rattus norvegicus (Norway rat)Potency0.891310
erythro-dihydrosphingosineRattus norvegicus (Norway rat)Potency16.833610
2-(3,3-diphenylpropylamino)acetamideRattus norvegicus (Norway rat)Potency2.511910
4-(2-(phenylsulfonylamino)ethylthio)-2,6-difluorophenoxyacetamideRattus norvegicus (Norway rat)Potency10.621310
8-hydroxy-2-(di-n-propylamino)tetralin, (r)-isomerRattus norvegicus (Norway rat)Potency1.000010
l 162313Rattus norvegicus (Norway rat)Potency26.862530
mrs 1754Rattus norvegicus (Norway rat)Potency31.622810
pd 404182Rattus norvegicus (Norway rat)Potency39.810710
sb 215505Rattus norvegicus (Norway rat)Potency21.192310
[4-(4-amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methanoneRattus norvegicus (Norway rat)Potency89.125110
nitrofurantoinRattus norvegicus (Norway rat)Potency35.481310
3,4-dichloro-n-methyl-n-(2-(1-pyrrolidinyl)cyclohexyl)-benzeneacetamide, (trans)-(-)-isomerRattus norvegicus (Norway rat)Potency0.223910
azetidine-2,4-dicarboxylic acidRattus norvegicus (Norway rat)Potency0.106210
sb 218795Rattus norvegicus (Norway rat)Potency39.591230
sb 269970Rattus norvegicus (Norway rat)Potency0.480220
ym 976Rattus norvegicus (Norway rat)Potency7.943310
2-(1,3-benzothiazol-2-yl)-4-chloro-5-(3-chloroanilino)-3-pyridazinoneRattus norvegicus (Norway rat)Potency70.794610
1-(3-amino-7-methoxy-1-pyrazolo[3,4-b]quinolinyl)-2-(4-chlorophenyl)ethanoneRattus norvegicus (Norway rat)Potency0.100010
2-(2-furanyl)-N-phenyl-3-imidazo[1,2-a]pyridinamineRattus norvegicus (Norway rat)Potency44.668410
1-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-N-(phenylmethyl)-3-piperidinecarboxamideRattus norvegicus (Norway rat)Potency89.125110
5-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-3-methyl-2-thiophenecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency39.810710
N-(4-ethoxyphenyl)-1,5-dimethyl-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamideRattus norvegicus (Norway rat)Potency79.432810
2-(4-methoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency28.370820
LSM-32377Rattus norvegicus (Norway rat)Potency8.539820
atomoxetineRattus norvegicus (Norway rat)Potency37.685820
epinephrine bitartrateRattus norvegicus (Norway rat)Potency10.407410
LSM-6455Rattus norvegicus (Norway rat)Potency50.118710
sk&f 89976-aRattus norvegicus (Norway rat)Potency41.177110
cv 1808Rattus norvegicus (Norway rat)Potency8.912510
edelfosineRattus norvegicus (Norway rat)Potency37.685820
ganaxoloneRattus norvegicus (Norway rat)Potency6.309610
altenusinRattus norvegicus (Norway rat)Potency0.794310
xct790Rattus norvegicus (Norway rat)Potency12.651120
cefalotin(1-)Rattus norvegicus (Norway rat)Potency16.833620
3-(3-methylphenyl)-2-sulfanylidene-1H-benzofuro[3,2-d]pyrimidin-4-oneRattus norvegicus (Norway rat)Potency15.848910
N-(1,3-dioxo-5-isoindolyl)butanamideRattus norvegicus (Norway rat)Potency56.234110
3-(ethylthio)-6-(2-furanyl)pyridazineRattus norvegicus (Norway rat)Potency25.118910
3-[(3-fluorophenyl)methylthio]-6-(2-furanyl)pyridazineRattus norvegicus (Norway rat)Potency50.118710
2-[[6-(2-furanyl)-3-pyridazinyl]thio]-N-(3-methylphenyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
5-Chloro-3-pyridinyl 2-furoateRattus norvegicus (Norway rat)Potency56.234110
parthenolideRattus norvegicus (Norway rat)Potency56.234110
5-(1-phenyl-5-tetrazolyl)-2-pyridin-4-yl-4-thiophen-2-ylpyrimidineRattus norvegicus (Norway rat)Potency17.782810
3-butyl-10-phenylpyrimido[4,5-b]quinoline-2,4-dioneRattus norvegicus (Norway rat)Potency22.387220
1-(3-ethylphenyl)-3-(1-naphthalenyl)thioureaRattus norvegicus (Norway rat)Potency70.794610
2-(3,5-dimethyl-1H-pyrrol-2-yl)-1,3-benzothiazoleRattus norvegicus (Norway rat)Potency28.183810
2-amino-3-methyl-7-(2-phenylethyl)-5H-pteridine-4,6-dioneRattus norvegicus (Norway rat)Potency56.234110
alpha-solanineRattus norvegicus (Norway rat)Potency70.794610
4-[[[4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazin-6-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency16.271020
5-chloro-N-[4-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2-thiophenesulfonamideRattus norvegicus (Norway rat)Potency28.183810
1-(3,4-dimethylphenyl)-2,5-dioxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarbonitrileRattus norvegicus (Norway rat)Potency14.129120
4-[[oxo-[4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazin-6-yl]methyl]amino]-1-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency53.176420
1'-acetyl-6-[2-(4-ethyl-1-piperazinyl)-2-oxoethoxy]-4-spiro[3,4-dihydro-2H-1-benzopyran-2,4'-piperidine]oneRattus norvegicus (Norway rat)Potency19.952610
4-methyl-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideRattus norvegicus (Norway rat)Potency56.234110
N-(phenylmethyl)-3-[3,4,6-trimethyl-1-(4-methylphenyl)-5-pyrazolo[3,4-b]pyridinyl]propanamideRattus norvegicus (Norway rat)Potency50.118710
2-[(1-amino-1-oxopropan-2-yl)thio]-3-butyl-4-oxo-7-quinazolinecarboxylic acid methyl esterRattus norvegicus (Norway rat)Potency22.387210
naloxone benzoylhydrazoneRattus norvegicus (Norway rat)Potency27.734310
cefotaxime sodiumRattus norvegicus (Norway rat)Potency15.430540
pnu-282987Rattus norvegicus (Norway rat)Potency1.000010
(R)-fluoxetine hydrochlorideRattus norvegicus (Norway rat)Potency0.211910
beta-aminoethylisothiuronium dihydrobromideRattus norvegicus (Norway rat)Potency79.432810
norfenfluramineRattus norvegicus (Norway rat)Potency1.584910
17-cyclopropylmethyl-6,7-didehydro-4,5-epoxy-5'-guanidinyl-3,14-dihydroxyindolo(2',3'-6,7)morphinanRattus norvegicus (Norway rat)Potency25.248730
n(6)-cyclohexyladenosineRattus norvegicus (Norway rat)Potency2.993520
fursultiamin monohydrochlorideRattus norvegicus (Norway rat)Potency17.782810
molindone hydrochlorideRattus norvegicus (Norway rat)Potency66.896810
qx-314 bromideRattus norvegicus (Norway rat)Potency0.059710
(S)-fluoxetine hydrochlorideRattus norvegicus (Norway rat)Potency42.284110
a 134974Rattus norvegicus (Norway rat)Potency0.398110
u 74389gRattus norvegicus (Norway rat)Potency79.432810
y 27632, dihydrochloride, (4(r)-trans)-isomerRattus norvegicus (Norway rat)Potency0.597310
1-(2,3-dichlorobenzoyl)-5-methoxy-2-methyl-(2-(mopholin-4-yl)ethyl)-1h-indoleRattus norvegicus (Norway rat)Potency0.501210
a 77636Rattus norvegicus (Norway rat)Potency23.858810
2-methyl-N-(5-methyl-2-thiazolyl)-1,1,4-trioxo-3H-1$l^{6},2-benzothiazine-3-carboxamideRattus norvegicus (Norway rat)Potency56.234110
((2-n-butyl-6,7-dichloro-2-cyclopentyl-2,3-dihydro-1-oxo-1h-inden-5-yl)oxy)acetic acid, (+)-isomerRattus norvegicus (Norway rat)Potency27.227130
(5R)-9-bromo-5-phenyl-3-prop-2-enyl-1,2,4,5-tetrahydro-3-benzazepine-7,8-diolRattus norvegicus (Norway rat)Potency10.000010
cefotaxime sodiumRattus norvegicus (Norway rat)Potency54.240210
Pseudopterosin G-J aglyconeRattus norvegicus (Norway rat)Potency89.125110
mrs 1845Rattus norvegicus (Norway rat)Potency37.082630
3-hydroxybenzylhydrazine hydrochlorideRattus norvegicus (Norway rat)Potency44.668410
(r)-n-(benzimidazol-2-yl)-1,2,3,4-tetrahydro-1-naphthylamineRattus norvegicus (Norway rat)Potency15.003010
as 252424Rattus norvegicus (Norway rat)Potency21.192320
cgp 57380Rattus norvegicus (Norway rat)Potency0.398110
protoapigenoneRattus norvegicus (Norway rat)Potency70.794610
2-(4-butan-2-ylanilino)-3-pyridinecarbonitrileRattus norvegicus (Norway rat)Potency25.118910
N-[(1,3-dioxo-2-phenyl-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl)methyl]-4-methylbenzenesulfonamideRattus norvegicus (Norway rat)Potency2.818410
N-(2-methoxyethyl)-2-[[3-[(4-methoxyphenyl)methyl]-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideRattus norvegicus (Norway rat)Potency31.622820
1-aminocyclopropane-1-carboxylic acid hydrochlorideRattus norvegicus (Norway rat)Potency42.284110
6-fluoronorepinephrine monohydrochloride, (+-)-isomerRattus norvegicus (Norway rat)Potency54.218410
dsp 4 hydrochlorideRattus norvegicus (Norway rat)Potency23.316010
calcimycinRattus norvegicus (Norway rat)Potency21.476840
(2-(2',6'-dimethoxy)phenoxyethylamino)methylbenzodioxan hydrochlorideRattus norvegicus (Norway rat)Potency0.150010
adtnRattus norvegicus (Norway rat)Potency29.934910
2-hydroxyapomorphine, (r)-isomerRattus norvegicus (Norway rat)Potency31.622810
fenoldopam hydrobromideRattus norvegicus (Norway rat)Potency36.533820
dextrothyroxineRattus norvegicus (Norway rat)Potency28.183810
metoprololRattus norvegicus (Norway rat)Potency0.398110
tele-methylhistamineRattus norvegicus (Norway rat)Potency23.778110
alpha-methyltyrosine methyl ester, monohydrochlorideRattus norvegicus (Norway rat)Potency1.258910
2-(n-phenethyl-n-propyl)amino-5-hydroxytetralin hydrochlorideRattus norvegicus (Norway rat)Potency37.685810
du 24565Rattus norvegicus (Norway rat)Potency54.683810
ro 25-6981Rattus norvegicus (Norway rat)Potency4.268410
sk&f 77434Rattus norvegicus (Norway rat)Potency21.192310
3-[(6aR,9R,10aR)-7-methyl-6,6a,8,9,10,10a-hexahydro-4H-indolo[4,3-fg]quinoline-9-yl]-1,1-diethylureaRattus norvegicus (Norway rat)Potency14.125410
2-ethyl-3-methoxy-N-(2-thiophen-2-ylethyl)-6-indazolecarboxamideRattus norvegicus (Norway rat)Potency28.183810
N-(1-adamantylmethyl)-2-ethyl-3-methoxy-6-indazolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
3-ethoxy-N-[(4-methoxyphenyl)methyl]-2-propyl-6-indazolecarboxamideRattus norvegicus (Norway rat)Potency56.234110
1-(4-bromophenyl)-3-[[[4-(4-morpholinyl)-3-nitrophenyl]-oxomethyl]amino]thioureaRattus norvegicus (Norway rat)Potency12.589310
N-(3-fluorophenyl)-2-(9-oxo-10-acridinyl)acetamideRattus norvegicus (Norway rat)Potency2.511910
4-[(2-methyl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)hydrazo]-4-oxo-N-propan-2-ylbutanamideRattus norvegicus (Norway rat)Potency0.079410
[4-(2-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(phenylmethyl)-1-piperazinyl]methanoneRattus norvegicus (Norway rat)Potency10.000010
4-chloro-N-(3,4-dimethoxyphenyl)-2-thieno[3,2-c]quinolinecarboxamideRattus norvegicus (Norway rat)Potency89.125110
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency12.589310
2-(4-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideRattus norvegicus (Norway rat)Potency10.000010
2-[(2-chloro-1-oxoethyl)-(2,2-dimethoxyethyl)amino]-2-(4-chlorophenyl)-N-cyclohexylacetamideRattus norvegicus (Norway rat)Potency35.481310
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamideRattus norvegicus (Norway rat)Potency70.794610
1-(4-fluorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaRattus norvegicus (Norway rat)Potency15.848910
1-(4-methylphenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaRattus norvegicus (Norway rat)Potency10.000010
1-(3-chlorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaRattus norvegicus (Norway rat)Potency7.943310
4-[3-(3-fluorophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamideRattus norvegicus (Norway rat)Potency27.565320
3-(benzenesulfonyl)-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]propanamideRattus norvegicus (Norway rat)Potency56.234110
[9-(benzenesulfonyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinolin-8-yl]-(4-methylphenyl)methanoneRattus norvegicus (Norway rat)Potency12.589310
N-[2-methyl-5-(2-thiazolo[5,4-b]pyridinyl)phenyl]-5,6,7,8-tetrahydronaphthalene-2-sulfonamideRattus norvegicus (Norway rat)Potency0.501210
(2S)-2-[[(3,5-dimethoxyphenyl)-oxomethyl]amino]-3-methylbutanoic acid [2-oxo-2-(4-propan-2-ylanilino)ethyl] esterRattus norvegicus (Norway rat)Potency10.000010
2-(4-fluorophenyl)-6-methoxy-1,3-benzothiazoleRattus norvegicus (Norway rat)Potency19.952610
(1S)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-6-methoxy-2-methyl-2-oxido-3,4-dihydro-1H-isoquinolin-2-ium-7-olRattus norvegicus (Norway rat)Potency28.183810
prim-o-glucosylcimifuginRattus norvegicus (Norway rat)Potency44.668410
2',3'-dihydroxy-4',6'-dimethoxychalconeRattus norvegicus (Norway rat)Potency89.125110
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneRattus norvegicus (Norway rat)Potency15.848910
dehydrocurvularinRattus norvegicus (Norway rat)Potency11.220210
Moracin PRattus norvegicus (Norway rat)Potency79.432810
4'-o-beta-d-glucosyl-5-o-methylvisamminolRattus norvegicus (Norway rat)Potency31.622810
3-[2-(4-chlorophenyl)-5,7-dimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]propanamideRattus norvegicus (Norway rat)Potency89.125120
N'-butan-2-yl-N-[2-(3,5-dimethyl-1-piperidinyl)-4-methyl-6-quinolinyl]butanediamideRattus norvegicus (Norway rat)Potency19.952610
3-[2-(3,5-dimethoxyphenyl)-5,7-dimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-(phenylmethyl)propanamideRattus norvegicus (Norway rat)Potency89.125120
2-(8-methoxy-4-methyl-1-oxo-[1,2,4]triazino[4,5-a]indol-2-yl)-N-(3-propan-2-yloxypropyl)acetamideRattus norvegicus (Norway rat)Potency56.234110
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency21.421510
5-chloro-2-[(3-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency16.099210
N-[5-[ethyl(phenyl)sulfamoyl]-1,3,4-thiadiazol-2-yl]-2-furancarboxamideRattus norvegicus (Norway rat)Potency70.794610
2-(5,8-dimethyl-2,4-dioxo-3-phenyl-1-pyrimido[5,4-b]indolyl)-N-(2-oxolanylmethyl)acetamideRattus norvegicus (Norway rat)Potency42.800010
3-[[(3R,4S)-2-(4-bromophenyl)-5-(3-chlorophenyl)-4-(2-methoxyphenyl)-3,4-dihydropyrazol-3-yl]-oxomethyl]-2-oxazolidinoneRattus norvegicus (Norway rat)Potency84.279020
tanninsRattus norvegicus (Norway rat)Potency70.794610
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]methanoneRattus norvegicus (Norway rat)Potency56.234110
[4-(3-chlorophenyl)-1-piperazinyl]-[1-[4-(2-pyridinyl)-1-piperazinyl]-4-isoquinolinyl]methanoneRattus norvegicus (Norway rat)Potency17.039020
8-methyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-5H-thieno[3,2-c]quinoline-2-carboxamideRattus norvegicus (Norway rat)Potency17.782810
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-4-nitro-3-isoxazolecarboxamideRattus norvegicus (Norway rat)Potency15.848910
N-(4-acetylphenyl)-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamideRattus norvegicus (Norway rat)Potency50.118710
N,8-dimethyl-N-(3-methylphenyl)-4-oxo-5H-thieno[3,2-c]quinoline-2-carboxamideRattus norvegicus (Norway rat)Potency3.162310
N-[2-(3,4-dimethoxyphenyl)ethyl]-N'-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)oxamideRattus norvegicus (Norway rat)Potency14.125410
1,2-dihydroacenaphthylen-5-yl-[1-(2-pyridinylmethyl)-3-piperidinyl]methanoneRattus norvegicus (Norway rat)Potency79.432810
1-[3-[(6-methoxy-2-naphthalenyl)-oxomethyl]-1-piperidinyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)thio]ethanoneRattus norvegicus (Norway rat)Potency79.432810
2-(2,4-dimethoxyphenyl)-5-methyl-4-[[4-(4-quinazolinyl)-1-piperazinyl]methyl]oxazoleRattus norvegicus (Norway rat)Potency39.810710
(3aS,5S,9aS)-2-[(2-methylphenyl)methyl]-5-(1-methyl-3-phenyl-4-pyrazolyl)-3a,4,5,7,8,9-hexahydro-3H-pyrrolo[3,4-h]pyrrolizin-1-oneRattus norvegicus (Norway rat)Potency44.668410
1-[[3-(2-fluorophenyl)-1-methyl-4-pyrazolyl]methyl]-3-propoxypiperidineRattus norvegicus (Norway rat)Potency79.432810
N-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]-4-phenyl-1-piperazinecarbothioamideRattus norvegicus (Norway rat)Potency19.952610
N-(5-chloro-2-pyridinyl)-4H-thieno[3,2-c][1]benzopyran-2-carboxamideRattus norvegicus (Norway rat)Potency33.117020
violaceol IIRattus norvegicus (Norway rat)Potency50.118710
LSM-24185Rattus norvegicus (Norway rat)Potency63.095710
LSM-16753Rattus norvegicus (Norway rat)Potency19.622220
6-chloro-3-[2-[4-[2,3-dihydro-1,4-benzodioxin-3-yl(oxo)methyl]-1-piperazinyl]-2-oxoethyl]-7-hydroxy-4-methyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency22.874120
2-imino-8-methyl-5-oxo-1-(2-oxolanylmethyl)-N-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency67.833420
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency44.668410
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideRattus norvegicus (Norway rat)Potency25.118910
N-[(2S)-1-hydroxypropan-2-yl]-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideRattus norvegicus (Norway rat)Potency56.234110
N-(2-methoxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideRattus norvegicus (Norway rat)Potency79.432810
N-(2-hydroxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideRattus norvegicus (Norway rat)Potency44.668410
thimerosalRattus norvegicus (Norway rat)Potency0.562310
6-[(3E,5E,7S)-5,7-dimethyl-2-oxonona-3,5-dienyl]-2,4-dihydroxy-3-methylbenzaldehydeRattus norvegicus (Norway rat)Potency70.794610
3-(4-methylphenyl)-5-oxo-N-propyl-8-thiazolo[2,3-b]quinazolinecarboxamideRattus norvegicus (Norway rat)Potency14.125410
8-[3-(diethylamino)-1-(4-methoxyphenyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency22.387210
(3R,3aS,7R,7aS)-3-[4-[4-(dimethylamino)phenyl]-2-fluorophenyl]-7-methyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneRattus norvegicus (Norway rat)Potency28.183810
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esterRattus norvegicus (Norway rat)Potency79.432810
valproate sodiumRattus norvegicus (Norway rat)Potency42.284110
gdc 0941Rattus norvegicus (Norway rat)Potency141.254010
cloprostenol sodiumRattus norvegicus (Norway rat)Potency89.125110
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methoxyphenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)Potency12.589310
6-(3,5-dimethyl-4-isoxazolyl)-N-[(2-ethoxyphenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)Potency89.125110
6-(3,5-dimethyl-4-isoxazolyl)-N-[1-(2-furanyl)ethyl]-4-quinazolinamineRattus norvegicus (Norway rat)Potency56.234110
sl 80.0750Rattus norvegicus (Norway rat)Potency79.432810
N-[[3-(4-nitrophenyl)sulfonyl-2-oxazolidinyl]methyl]-N'-(2-pyridinylmethyl)oxamideRattus norvegicus (Norway rat)Potency89.125110
cefotiam hydrochlorideRattus norvegicus (Norway rat)Potency79.432810
N-[2-(2,5-dimethoxyphenyl)ethyl]-4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazine-6-carboxamideRattus norvegicus (Norway rat)Potency67.833420
N-[(5-bromo-2-methoxyphenyl)methyl]-4-methyl-2,3-dihydro-1,4-benzothiazine-6-carboxamideRattus norvegicus (Norway rat)Potency31.099020
5-fluoro-2-phenyl-1,2-benzothiazol-3-oneRattus norvegicus (Norway rat)Potency50.118710
2-(4-fluorophenyl)-1,2-benzothiazol-3-oneRattus norvegicus (Norway rat)Potency50.118710
4-[4-(4-fluorophenyl)-1-piperazinyl]-N-[4-methyl-2-(4-morpholinyl)-6-quinolinyl]-4-oxobutanamideRattus norvegicus (Norway rat)Potency22.387210
3-[1-[oxo-(1-phenylcyclopropyl)methyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneRattus norvegicus (Norway rat)Potency100.000010
4'-epichaetoviridin ARattus norvegicus (Norway rat)Potency25.118910
2-[[4-(5-chloro-2-propan-2-yloxyanilino)-6-(1-pyrrolidinyl)-1,3,5-triazin-2-yl]amino]ethanolRattus norvegicus (Norway rat)Potency56.234110
cilastatin sodiumRattus norvegicus (Norway rat)Potency70.794610
montelukast sodiumRattus norvegicus (Norway rat)Potency63.095710
cefmetazole sodiumRattus norvegicus (Norway rat)Potency15.003010
cefoxitin sodiumRattus norvegicus (Norway rat)Potency79.432810
deoxycholic acid, monosodium saltRattus norvegicus (Norway rat)Potency89.125110
zinacefRattus norvegicus (Norway rat)Potency63.095710
cephapirin sodiumRattus norvegicus (Norway rat)Potency33.587510
sodium cephalothinRattus norvegicus (Norway rat)Potency18.887610
cefazolin sodiumRattus norvegicus (Norway rat)Potency18.887610
naproxen sodiumRattus norvegicus (Norway rat)Potency33.587510
sodium 2,6-dichloroindophenolRattus norvegicus (Norway rat)Potency1.584910
leu-ser-glu-ala-leuRattus norvegicus (Norway rat)Potency39.810710
3-[(2-chlorophenyl)methyl]-N-(2-fluorophenyl)-5-methyl-7-triazolo[4,5-d]pyrimidinamineRattus norvegicus (Norway rat)Potency89.125110
cefsulodinRattus norvegicus (Norway rat)Potency5.329020
3-[[1-[1-(methylthio)propan-2-yl]-4-piperidinyl]oxy]-N-(2-pyridinylmethyl)benzamideRattus norvegicus (Norway rat)Potency8.912510
pci 32765Rattus norvegicus (Norway rat)Potency79.432810
norepinephrine bitartrateRattus norvegicus (Norway rat)Potency79.432810
(3S)-3-(2-methylpropyl)-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency1.995310
(3S)-3-(4-methoxyphenyl)-4-oxo-3-propan-2-yldiazetidine-1,2-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency28.183810
(3S)-4-oxo-3-phenyl-3-propan-2-yldiazetidine-1,2-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency17.782810
4-(4-acetyloxyphenyl)benzoic acid [2-[[2-(2-chloroanilino)-2-oxoethyl]-methylamino]-2-oxoethyl] esterRattus norvegicus (Norway rat)Potency89.125110
(3S)-3-cyclopentyl-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterRattus norvegicus (Norway rat)Potency8.912510
(3R)-3-(4-chlorophenyl)-4-oxo-3-propan-2-yldiazetidine-1,2-dicarboxylic acid diethyl esterRattus norvegicus (Norway rat)Potency44.668410
zonisamide monosodiumRattus norvegicus (Norway rat)Potency31.622810
mk 2206Rattus norvegicus (Norway rat)Potency56.234110
bix 01294Rattus norvegicus (Norway rat)Potency30.461230
4-(2,6-difluorophenyl)sulfonyl-1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)piperidineRattus norvegicus (Norway rat)Potency112.202010
N-[2-[(2,6-difluorophenyl)sulfonylamino]ethyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideRattus norvegicus (Norway rat)Potency0.707910
3-[(2-fluorophenyl)methyl]-5-methyl-4-thieno[3,4]pyrrolo[1,3-d]pyrimidinoneRattus norvegicus (Norway rat)Potency56.234110
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)Potency15.848910
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)Potency19.952610
6-(1,3-benzodioxol-5-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)Potency25.118910
5-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]methyl]-8-quinolinolRattus norvegicus (Norway rat)Potency28.183810
N-[4-cyano-2-(1-naphthalenyl)-5-oxazolyl]acetamideRattus norvegicus (Norway rat)Potency28.183810
2-[(4-methylphenyl)methylthio]-5-(1-naphthalenyl)-1,3,4-oxadiazoleRattus norvegicus (Norway rat)Potency21.450920
5-amino-2-(1-naphthalenyl)-4-oxazolecarbonitrileRattus norvegicus (Norway rat)Potency26.651420
4-[5-(3-hydroxy-4-oxo-1,2-dihydroquinazolin-2-yl)-2-furanyl]benzonitrileRattus norvegicus (Norway rat)Potency7.079510
2-[5-(2-fluorophenyl)-2-furanyl]-3-hydroxy-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency79.432810
3-hydroxy-2-(5-thiophen-2-yl-2-furanyl)-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency44.964720
3-hydroxy-2-[5-[4-(trifluoromethyl)phenyl]-2-furanyl]-1,2-dihydroquinazolin-4-oneRattus norvegicus (Norway rat)Potency56.234110
2-methoxybenzoic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency44.668410
2-naphthalenecarboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency14.721420
1H-indole-4-carboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterRattus norvegicus (Norway rat)Potency19.952610
3-(2-chlorophenyl)-6-(3-cyclopentyloxy-4-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineRattus norvegicus (Norway rat)Potency7.079510
6-(3-chloroanilino)-9-cyclopentyl-2-purinecarbonitrileRattus norvegicus (Norway rat)Potency89.125120
4-[(1-methyl-5-tetrazolyl)thio]-5-[2-(trifluoromethyl)phenyl]thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency25.118910
4-[4-[(1-methyl-5-tetrazolyl)thio]-5-thieno[2,3-d]pyrimidinyl]benzonitrileRattus norvegicus (Norway rat)Potency89.125110
4-[(1-methyl-5-tetrazolyl)thio]-5-(4-nitrophenyl)thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency79.432810
5-(2-benzofuranyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency12.589310
4-[(1-methyl-5-tetrazolyl)thio]-5-(1H-pyrrol-2-yl)thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency50.118710
5-(3-methylsulfonylphenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency89.125110
5-bromo-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineRattus norvegicus (Norway rat)Potency5.623410
6-(3-chloroanilino)-9-ethyl-2-purinecarbonitrileRattus norvegicus (Norway rat)Potency35.481310
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimineRattus norvegicus (Norway rat)Potency12.589310
4-[3-(3-bromophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamideRattus norvegicus (Norway rat)Potency31.622810
N-[[(2R,3S)-10-(dimethylamino)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-N-methylmethanesulfonamideRattus norvegicus (Norway rat)Potency39.810710
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-2-[[[(4-methoxyanilino)-oxomethyl]-methylamino]methyl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]cyclohexanecarboxamideRattus norvegicus (Norway rat)Potency89.125110
3-cyclohexyl-1-[[(2S,3R)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-10-[[oxo-(propan-2-ylamino)methyl]amino]-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methylureaRattus norvegicus (Norway rat)Potency22.387210
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-(methylaminomethyl)-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]cyclopropanecarboxamideRattus norvegicus (Norway rat)Potency70.794610
(2S,3S)-10-(dimethylamino)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl(pyridin-4-ylmethyl)amino]methyl]-3,4-dihydro-2H-1,5-benzoxazocin-6-oneRattus norvegicus (Norway rat)Potency79.432810
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[oxo-[4-(trifluoromethyl)anilino]methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-4-pyridinecarboxamideRattus norvegicus (Norway rat)Potency17.782810
1-[(2R,3R)-2-[[benzenesulfonyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-[4-(trifluoromethyl)phenyl]ureaRattus norvegicus (Norway rat)Potency70.794610
(E,E)-1-bromo-2,5-bis-(4-hydroxystyryl)benzeneRattus norvegicus (Norway rat)Potency19.711940
unc 0321Rattus norvegicus (Norway rat)Potency36.253020
oxytetracycline, anhydrousRattus norvegicus (Norway rat)Potency35.481310
piroxicamRattus norvegicus (Norway rat)Potency2.667910
LSM-16789Rattus norvegicus (Norway rat)Potency79.432810
lfm a13Rattus norvegicus (Norway rat)Potency0.504520
LSM-17430Rattus norvegicus (Norway rat)Potency10.000010
4-hydroxy-2-oxo-N-[3-(trifluoromethyl)phenyl]-1H-quinoline-3-carboxamideRattus norvegicus (Norway rat)Potency89.125110
4,7-Dihydroxy-2H-1-benzopyran-2-oneRattus norvegicus (Norway rat)Potency39.810710
demeclocyclineRattus norvegicus (Norway rat)Potency23.479420
6-chloro-4-hydroxy-3-(phenylmethyl)-1H-quinolin-2-oneRattus norvegicus (Norway rat)Potency35.481310
1-ethyl-N-(2-fluorophenyl)-4-hydroxy-2-oxo-3-quinolinecarboxamideRattus norvegicus (Norway rat)Potency35.481310
hispidinRattus norvegicus (Norway rat)Potency9.876720
N3-phenyl-4-hydroxy-1,5,6-trimethyl-2,2-dioxo-1,2-dihydro-26-thieno[2,3-c][1,2]thiazine-3-carboxamideRattus norvegicus (Norway rat)Potency10.000010
N-(4-hydroxy-2-oxo-1H-quinolin-3-yl)pentanamideRattus norvegicus (Norway rat)Potency25.118910
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-[4-oxo-2-(phenylmethyl)-3-quinazolinyl]-5,6,7,8-tetrahydroquinoline-3-carboxamideRattus norvegicus (Norway rat)Potency35.481310
acyclovirRattus norvegicus (Norway rat)Potency2.993510
sepiapterinRattus norvegicus (Norway rat)Potency44.340530
isoxanthopterinRattus norvegicus (Norway rat)Potency9.892540
clozapineRattus norvegicus (Norway rat)Potency22.984430
ganciclovirRattus norvegicus (Norway rat)Potency7.079510
oxypurinolRattus norvegicus (Norway rat)Potency0.100010
zaprinastRattus norvegicus (Norway rat)Potency0.501210
suptopin 2Rattus norvegicus (Norway rat)Potency28.183810
syringaldazineRattus norvegicus (Norway rat)Potency26.632020
4-oxo-2-(trifluoromethyl)-1H-quinazoline-6-carboxylic acid ethyl esterRattus norvegicus (Norway rat)Potency22.387210
6-[5-[[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]methyl]-2-oxo-1,3-dihydroimidazol-4-yl]-6-oxohexanoic acid ethyl esterRattus norvegicus (Norway rat)Potency22.387210
phenylamilRattus norvegicus (Norway rat)Potency17.895630
hemateinRattus norvegicus (Norway rat)Potency15.848910
thiolactomycinRattus norvegicus (Norway rat)Potency37.685810
2,4-diaminohypoxanthineRattus norvegicus (Norway rat)Potency38.705620
5-amino-2-phenyl-3H-triazolo[4,5-d]pyrimidin-7-oneRattus norvegicus (Norway rat)Potency17.900820
trichloroethyleneRattus norvegicus (Norway rat)Potency26.840740
norclozapineRattus norvegicus (Norway rat)Potency31.118420
2-[[3-[(2-ethoxy-2-oxoethyl)thio]-5-oxo-2H-1,2,4-triazin-6-yl]amino]acetic acid butyl esterRattus norvegicus (Norway rat)Potency11.220210
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-6-methyl-1H-pyrimidin-4-oneRattus norvegicus (Norway rat)Potency56.234110
1-cyclopentyl-1-[(4-oxo-1H-quinazolin-2-yl)methyl]-3-(phenylmethyl)ureaRattus norvegicus (Norway rat)Potency25.118910
quazinoneRattus norvegicus (Norway rat)Potency0.566120
2-amino-4-hydroxy-6-trifluoromethylpyrimidineRattus norvegicus (Norway rat)Potency70.794610
ag-879Rattus norvegicus (Norway rat)Potency30.458630
lomofunginRattus norvegicus (Norway rat)Potency56.234110
6-methyl-3-sulfanylidene-1,2-dihydro-[1,2,4]triazolo[4,3-b][1,2,4]triazin-7-oneRattus norvegicus (Norway rat)Potency19.952610
N-[4-[2-(2-methoxyethylamino)-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamideRattus norvegicus (Norway rat)Potency0.446710
pyridoxal 4-methoxybenzoyl hydrazoneRattus norvegicus (Norway rat)Potency79.432810
2-[5-(3-chlorophenyl)-2-furanyl]-1H-quinazolin-4-oneRattus norvegicus (Norway rat)Potency50.118710
5,5-diethyl-2-(2-hydroxyethylamino)-1,6-dihydrobenzo[h]quinazolin-4-oneRattus norvegicus (Norway rat)Potency28.183810
3-ethyl-2-[(4-oxo-1H-quinazolin-2-yl)methylthio]-4-quinazolinoneRattus norvegicus (Norway rat)Potency14.125410
5,5-diethyl-2-hydrazinyl-1,6-dihydrobenzo[h]quinazolin-4-oneRattus norvegicus (Norway rat)Potency56.234110