Page last updated: 2024-08-07 19:40:54

TPA: protein transporter TIM10

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (64)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
1,10-phenanthrolineSaccharomyces cerevisiae S288CIC5012.300010
3,4-dichloroisocoumarinSaccharomyces cerevisiae S288CIC5060.050020
ebselenSaccharomyces cerevisiae S288CIC505.290020
dehydrothio-4-toluidineSaccharomyces cerevisiae S288CIC5017.400010
pyrazolanthroneSaccharomyces cerevisiae S288CIC5073.400020
clomipramine hydrochlorideSaccharomyces cerevisiae S288CIC5037.800010
magnololSaccharomyces cerevisiae S288CIC5068.300010
honokiolSaccharomyces cerevisiae S288CIC5048.800010
prochlorperazine edisylate saltSaccharomyces cerevisiae S288CIC5029.100010
paxillineSaccharomyces cerevisiae S288CIC5033.550010
4-methoxy-1-vinylcarbolineSaccharomyces cerevisiae S288CIC5025.000010
tosylphenylalanyl chloromethyl ketoneSaccharomyces cerevisiae S288CIC500.640010
menadione sodium bisulfite, trihydrateSaccharomyces cerevisiae S288CIC507.140010
4-chloro-N-(4-chloro-2,5-dimethoxyphenyl)-5-dithiazolimineSaccharomyces cerevisiae S288CIC508.075020
3-(4-methoxyphenyl)-8-(6-methyl-2-phenyl-4-pyrimidinyl)-8-azabicyclo[3.2.1]octan-3-olSaccharomyces cerevisiae S288CIC5018.200010
r 59949Saccharomyces cerevisiae S288CIC5012.700010
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenolSaccharomyces cerevisiae S288CIC5061.100010
5,8-dichloro-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-oneSaccharomyces cerevisiae S288CIC5047.800010
dienestrolSaccharomyces cerevisiae S288CIC5025.600010
5-(4-cyclohexylphenyl)-1,2-dihydropyrazol-3-oneSaccharomyces cerevisiae S288CIC5029.500010
1-(4-methoxyphenyl)-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ureaSaccharomyces cerevisiae S288CIC5014.500010
4-(6-methyl-4-phenyl-2-quinazolinyl)-1-piperazinecarboxaldehydeSaccharomyces cerevisiae S288CIC509.880010
N-[4-(2-methyl-4-thiazolyl)phenyl]benzamideSaccharomyces cerevisiae S288CIC508.180010
1-[[(1-methyl-2-benzimidazolyl)amino]methyl]-2-naphthalenolSaccharomyces cerevisiae S288CIC50100.000010
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrileSaccharomyces cerevisiae S288CIC50100.000010
4-(3-methylphenyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneSaccharomyces cerevisiae S288CIC5037.500010
3-amino-6-cyclopropyl-4-(4-methoxyphenyl)-2-thieno[2,3-b]pyridinecarbonitrileSaccharomyces cerevisiae S288CIC508.580020
2-(2-methoxyphenyl)-1H-indoleSaccharomyces cerevisiae S288CIC5046.900010
3-[(2-chloro-6-fluorophenyl)methylthio]-4-ethyl-5-(2-furanyl)-1,2,4-triazoleSaccharomyces cerevisiae S288CIC5024.300010
curcuminSaccharomyces cerevisiae S288CIC5019.700010
2,2-dimethyl-N-[[2-(4-methyl-1-piperidinyl)anilino]-sulfanylidenemethyl]propanamideSaccharomyces cerevisiae S288CIC5075.800010
3-chloro-N-[3-nitro-5-(2-pyridinylthio)phenyl]benzamideSaccharomyces cerevisiae S288CIC5034.900010
3-[(1,3-benzothiazol-2-ylthio)methyl]-4-cyclohexyl-1H-1,2,4-triazole-5-thioneSaccharomyces cerevisiae S288CIC50100.000010
2-(2-bromophenyl)-5-[(2-chlorophenoxy)methyl]-1,3,4-oxadiazoleSaccharomyces cerevisiae S288CIC5022.250020
2-chloro-N-[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]acetamideSaccharomyces cerevisiae S288CIC5044.682540
2-(2-bromo-4-tert-butylphenoxy)-N-(2-furanylmethyl)acetamideSaccharomyces cerevisiae S288CIC5012.200010
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneSaccharomyces cerevisiae S288CIC5011.000010
N-(4-tert-butyl-2-thiazolyl)-5-methyl-2-thiophenecarboxamideSaccharomyces cerevisiae S288CIC5020.900010
(4-chlorophenyl)-[6,7-dichloro-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-3-benzofuranyl]methanoneSaccharomyces cerevisiae S288CIC5018.600010
2-(difluoromethyl)-4-benzo[h][1]benzopyranoneSaccharomyces cerevisiae S288CIC5081.260020
4-[3-[[(2,5-dichloroanilino)-methyliminomethyl]thio]-2,5-dioxo-1-pyrrolidinyl]benzoic acid methyl esterSaccharomyces cerevisiae S288CIC509.465020
4-[[2-(4-ethyl-3-oxo-2-morpholinyl)-1-oxoethyl]amino]benzoic acid ethyl esterSaccharomyces cerevisiae S288CIC505.590020
2-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methylthio]-3-pyridinecarboxylic acid propan-2-yl esterSaccharomyces cerevisiae S288CIC5071.200020
5-hydroxy-2-methyl-4-[1-piperidinyl(3-pyridinyl)methyl]-3-benzo[g]benzofurancarboxylic acid ethyl esterSaccharomyces cerevisiae S288CIC5036.100010
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinolSaccharomyces cerevisiae S288CIC5018.000010
2-[[2-(1-adamantyl)-2-oxoethyl]thio]-6-amino-4-(4-chlorophenyl)pyridine-3,5-dicarbonitrileSaccharomyces cerevisiae S288CIC5041.600010
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[4-(2-methoxyphenyl)-1-piperazinyl]acetamideSaccharomyces cerevisiae S288CIC5058.700010
N-(1-adamantyl)-6-(3,5-dimethyl-1-pyrazolyl)-1,2,4,5-tetrazin-3-amineSaccharomyces cerevisiae S288CIC5046.400010
4-chloro-N-(1,3,4-thiadiazol-2-yl)-5-dithiazolimineSaccharomyces cerevisiae S288CIC502.600010
1-(3,4-dichlorophenyl)-3-(1,3,5-trimethyl-4-pyrazolyl)ureaSaccharomyces cerevisiae S288CIC5022.400010
3-[(4-methyl-1-piperazinyl)sulfonyl]-N-(4-phenyl-2-thiazolyl)-N-prop-2-enylbenzamideSaccharomyces cerevisiae S288CIC5046.800010
2-[4-(4-chloro-2-nitrophenyl)-1-piperazinyl]phenolSaccharomyces cerevisiae S288CIC5032.300010
5-[(2,4-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]-4-pyrazolyl]-2-furancarboxamideSaccharomyces cerevisiae S288CIC5025.500010
galanginSaccharomyces cerevisiae S288CIC5067.750020
[2-(1-piperidinyl)-1,3-benzothiazol-6-yl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneSaccharomyces cerevisiae S288CIC5046.100010
3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5,7-dihydroxy-2-methyl-1-benzopyran-4-oneSaccharomyces cerevisiae S288CIC5010.700010
N-methyl-6-phenyl-3-(2-pyridinyl)-1,2,4-triazin-5-amineSaccharomyces cerevisiae S288CIC5029.800010
fluphenazineSaccharomyces cerevisiae S288CIC5031.300010
homochlorocyclizine monohydrochlorideSaccharomyces cerevisiae S288CIC5030.900010
2-[2-fluoro-5-(4-methyl-1-piperazinyl)-4-nitrophenyl]-3,4-dihydro-1H-isoquinolineSaccharomyces cerevisiae S288CIC5071.600010
chlorhexidine hydrochlorideSaccharomyces cerevisiae S288CIC5056.050020
(3R)-3-(2-fluoro-5-methylphenyl)-7-phenyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneSaccharomyces cerevisiae S288CIC5011.095020
6-chloro-N2-cyclopentyl-N4-(3,5-difluorophenyl)-1,3,5-triazine-2,4-diamineSaccharomyces cerevisiae S288CIC5037.700010
1-[amino-[(6-methoxy-4-methyl-2-quinazolinyl)amino]methylidene]-3-phenylureaSaccharomyces cerevisiae S288CIC5047.300010