Proteins > oxysterols receptor LXR-beta isoform 1
Page last updated: 2024-08-07 21:02:13
oxysterols receptor LXR-beta isoform 1
[no definition available]
Synonyms
Research
Bioassay Publications (0)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0) | 18.7374 |
1990's | 0 (0) | 18.2507 |
2000's | 0 (0) | 29.6817 |
2010's | 0 (0) | 24.3611 |
2020's | 0 (0) | 2.80 |
Compounds (34)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
quinophthalone | Homo sapiens (human) | IC50 | 67.5470 | 1 | 0 |
rutecarpine | Homo sapiens (human) | IC50 | 67.5740 | 1 | 0 |
4-methoxybenzophenone | Homo sapiens (human) | IC50 | 67.5610 | 1 | 0 |
2-(2'-hydroxy-3'-methoxyphenyl)benzothiazole | Homo sapiens (human) | IC50 | 67.5610 | 1 | 0 |
pinafide | Homo sapiens (human) | IC50 | 67.4750 | 1 | 0 |
nsc 674495 | Homo sapiens (human) | IC50 | 67.6490 | 1 | 0 |
5f-203 | Homo sapiens (human) | IC50 | 67.6220 | 1 | 0 |
5,7-dimethyl-2-phenylpyrazolo[1,5-a]pyrimidine | Homo sapiens (human) | IC50 | 67.4790 | 1 | 0 |
5,7-dimethyl-2-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine | Homo sapiens (human) | IC50 | 67.5470 | 1 | 0 |
2,4-dimethoxy-n-naphthalen-2-yl-benzamide | Homo sapiens (human) | IC50 | 67.5240 | 1 | 0 |
2-[(1-ethyl-2,5-dimethyl-3-pyrrolyl)methylidene]indene-1,3-dione | Homo sapiens (human) | IC50 | 67.5220 | 1 | 0 |
1-(1,3-benzodioxol-5-yl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)urea | Homo sapiens (human) | IC50 | 67.5740 | 1 | 0 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
ag 1295 | Homo sapiens (human) | EC50 | 67.4900 | 1 | 0 |
nsc-39661 | Homo sapiens (human) | EC50 | 67.5810 | 1 | 0 |
bromodeoxyuridine | Homo sapiens (human) | EC50 | 67.5260 | 1 | 0 |
quinophthalone | Homo sapiens (human) | EC50 | 67.5470 | 1 | 0 |
dinaline | Homo sapiens (human) | EC50 | 67.5610 | 1 | 0 |
l 10503 | Homo sapiens (human) | EC50 | 67.5340 | 1 | 0 |
nsc 674495 | Homo sapiens (human) | EC50 | 67.6490 | 1 | 0 |
2-(4-chlorophenyl)-1-phthalazinone | Homo sapiens (human) | EC50 | 67.5060 | 1 | 0 |
5-hydroxy-2-methyl-3-benzo[g]benzofurancarboxylic acid ethyl ester | Homo sapiens (human) | EC50 | 67.5350 | 1 | 0 |
5,7-dimethyl-2-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine | Homo sapiens (human) | EC50 | 67.5470 | 1 | 0 |
4-methyl-N,5-diphenyl-3-thiophenecarboxamide | Homo sapiens (human) | EC50 | 67.5160 | 1 | 0 |
N-(2-pyridinyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide | Homo sapiens (human) | EC50 | 67.5390 | 1 | 0 |
4-(4-chlorophenyl)-1-(6-fluoro-2-pyridinyl)-3-pyrazolamine | Homo sapiens (human) | EC50 | 67.5950 | 1 | 0 |
n-(fluorenyl-9-methoxycarbonyl)leucine | Homo sapiens (human) | EC50 | 67.5410 | 1 | 0 |
3-cyclohexyl-N-(1,3-dimethyl-2,6-dioxo-4-pyrimidinyl)propanamide | Homo sapiens (human) | EC50 | 67.5350 | 1 | 0 |
2-(4,6-dimethyl-2-pyrimidinyl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamine | Homo sapiens (human) | EC50 | 67.5200 | 1 | 0 |
4-(diethylsulfamoyl)benzoic acid [2-[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]-2-oxoethyl] ester | Homo sapiens (human) | EC50 | 67.5270 | 1 | 0 |
sr 3335 | Homo sapiens (human) | EC50 | 10.0000 | 1 | 0 |
3-methyl-4-oxo-1,5,6,7-tetrahydroindole-2-carboxylic acid (4-methylcyclohexyl) ester | Homo sapiens (human) | EC50 | 67.5330 | 1 | 0 |
5-methyl-N-(3-methylphenyl)-4-nitro-1H-pyrazol-3-amine | Homo sapiens (human) | EC50 | 67.5470 | 1 | 0 |
2-[(5-chloro-2-thiophenyl)-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl ester | Homo sapiens (human) | EC50 | 67.4870 | 1 | 0 |
N-cyclohexyl-1-(4-fluorophenyl)-2,5-dimethyl-3-pyrrolecarboxamide | Homo sapiens (human) | EC50 | 67.5470 | 1 | 0 |
6-(4-bromo-3,5-dimethyl-1-pyrazolyl)-N-cyclohexyl-1,2,4,5-tetrazin-3-amine | Homo sapiens (human) | EC50 | 67.5540 | 1 | 0 |
N-[(3-methyl-6-imidazo[2,1-b]thiazolyl)methyl]-1-propanesulfonamide | Homo sapiens (human) | EC50 | 67.5470 | 1 | 0 |
3-(2-pyridinyl)-6-(2-pyridinylmethylthio)pyridazine | Homo sapiens (human) | EC50 | 67.4750 | 1 | 0 |