Page last updated: 2024-08-07 12:31:32

hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (498)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
catecholHomo sapiens (human)Potency12.589320
chlordeconeHomo sapiens (human)Potency40.870810
4-aminophenolHomo sapiens (human)Potency50.118710
3,4-dihydroxyphenylacetic acidHomo sapiens (human)Potency15.848920
hydroquinoneHomo sapiens (human)Potency1.995320
1,10-phenanthrolineHomo sapiens (human)Potency10.752730
1,3-dipropyl-8-cyclopentylxanthineHomo sapiens (human)Potency10.000020
s,s'-1,4-phenylene-bis(1,2-ethanediyl)bis-isothioureaHomo sapiens (human)Potency25.118920
1h-(1,2,4)oxadiazolo(4,3-a)quinoxalin-1-oneHomo sapiens (human)Potency12.589320
3,4-dichloroisocoumarinHomo sapiens (human)Potency31.622820
3-nitropropionic acidHomo sapiens (human)Potency25.118920
p-chloromercuribenzoic acidHomo sapiens (human)Potency19.952620
4-hydroxybenzoic acid hydrazideHomo sapiens (human)Potency25.118920
4-nonylphenolHomo sapiens (human)Potency79.432810
6-chloromelatoninHomo sapiens (human)Potency12.589320
6-nitroso-1,2-benzopyroneHomo sapiens (human)Potency25.118920
aa 861Homo sapiens (human)Potency7.943320
acemetacinHomo sapiens (human)Potency5.050020
rtki cpdHomo sapiens (human)Potency15.848920
tyrphostin a23Homo sapiens (human)Potency10.000020
tyrphostin 25Homo sapiens (human)Potency10.000020
ambroxolHomo sapiens (human)Potency12.589320
amfonelic acidHomo sapiens (human)Potency25.118920
p-aminohippuric acidHomo sapiens (human)Potency5.011920
theophyllineHomo sapiens (human)Potency3.162320
amiodaroneHomo sapiens (human)Potency31.622820
amoxapineHomo sapiens (human)Potency7.943320
amsacrineHomo sapiens (human)Potency5.011920
aurintricarboxylic acidHomo sapiens (human)Potency12.589320
2,2-bis(4-glycidyloxyphenyl)propaneHomo sapiens (human)Potency79.432810
benzbromaroneHomo sapiens (human)Potency2.714520
benzethoniumHomo sapiens (human)Potency10.000020
berberineHomo sapiens (human)Potency2.511920
bay h 4502Homo sapiens (human)Potency1.258920
bisacodylHomo sapiens (human)Potency0.647720
bithionolHomo sapiens (human)Potency16.611530
bufexamacHomo sapiens (human)Potency10.266320
bumetanideHomo sapiens (human)Potency2.120120
buspironeHomo sapiens (human)Potency12.589320
cgs 15943Homo sapiens (human)Potency5.011920
chelerythrineHomo sapiens (human)Potency31.622820
chlorambucilHomo sapiens (human)Potency10.286920
clemizoleHomo sapiens (human)Potency11.896120
clioquinolHomo sapiens (human)Potency4.538530
clofazimineHomo sapiens (human)Potency5.227620
clonidineHomo sapiens (human)Potency12.589320
clotrimazoleHomo sapiens (human)Potency5.011920
dephostatinHomo sapiens (human)Potency10.000020
dequaliniumHomo sapiens (human)Potency5.997620
ddtHomo sapiens (human)Potency79.432810
dichlorophenHomo sapiens (human)Potency39.810710
diflunisalHomo sapiens (human)Potency5.011920
dilazepHomo sapiens (human)Potency3.981120
n,n-di-n-propyldopamineHomo sapiens (human)Potency12.589320
dipyridamoleHomo sapiens (human)Potency25.118920
2,3-dimethoxy-1,4-naphthoquinoneHomo sapiens (human)Potency7.943320
domperidoneHomo sapiens (human)Potency2.511920
droperidolHomo sapiens (human)Potency3.981120
ebselenHomo sapiens (human)Potency17.559420
ellipticineHomo sapiens (human)Potency16.408020
emodinHomo sapiens (human)Potency10.000020
ethacrynic acidHomo sapiens (human)Potency34.870530
ethoxyquinHomo sapiens (human)Potency1.258920
ethoxzolamideHomo sapiens (human)Potency0.010020
fenbufenHomo sapiens (human)Potency10.000020
fipexideHomo sapiens (human)Potency3.981120
flufenamic acidHomo sapiens (human)Potency7.506020
fluspirileneHomo sapiens (human)Potency25.118920
fpl 64176Homo sapiens (human)Potency2.511920
furafyllineHomo sapiens (human)Potency7.943320
fusaric acidHomo sapiens (human)Potency9.180420
gallamine triethiodideHomo sapiens (human)Potency12.589320
vanoxerineHomo sapiens (human)Potency18.966220
gbr 12935Homo sapiens (human)Potency25.118920
glimepirideHomo sapiens (human)Potency7.943320
glutaralHomo sapiens (human)Potency39.810710
glyburideHomo sapiens (human)Potency2.578820
gossypolHomo sapiens (human)Potency10.000020
fluorometholoneHomo sapiens (human)Potency3.981120
guanfacineHomo sapiens (human)Potency10.000020
bis(2-guanidinoethyl)disulfideHomo sapiens (human)Potency15.848920
gyki 52466Homo sapiens (human)Potency12.589320
n-(2-aminoethyl)-5-isoquinolinesulfonamideHomo sapiens (human)Potency25.118920
hexachloropheneHomo sapiens (human)Potency50.118710
hexamethylene bisacetamideHomo sapiens (human)Potency12.589320
hycanthoneHomo sapiens (human)Potency5.011920
amrinoneHomo sapiens (human)Potency3.981120
indirubin-3'-monoximeHomo sapiens (human)Potency25.118920
indomethacinHomo sapiens (human)Potency7.539720
iodoquinolHomo sapiens (human)Potency0.199520
ipriflavoneHomo sapiens (human)Potency6.309620
itraconazoleHomo sapiens (human)Potency2.511920
1-(2-naphthalenyl)-3-[(phenylmethyl)-propan-2-ylamino]-1-propanoneHomo sapiens (human)Potency31.622820
nsc 664704Homo sapiens (human)Potency3.162320
kinetinHomo sapiens (human)Potency12.589320
lansoprazoleHomo sapiens (human)Potency11.896120
beta-lapachoneHomo sapiens (human)Potency31.622820
loratadineHomo sapiens (human)Potency15.848920
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-oneHomo sapiens (human)Potency7.943320
mebendazoleHomo sapiens (human)Potency1.978320
meclofenamate sodium anhydrousHomo sapiens (human)Potency12.924420
mefenamic acidHomo sapiens (human)Potency10.000020
vitamin k 3Homo sapiens (human)Potency12.589320
mesalamineHomo sapiens (human)Potency10.000020
nocodazoleHomo sapiens (human)Potency1.097420
mitotaneHomo sapiens (human)Potency63.095710
mitoxantroneHomo sapiens (human)Potency10.266320
moxisylyteHomo sapiens (human)Potency25.118920
clorgylineHomo sapiens (human)Potency25.118920
deoxyepinephrineHomo sapiens (human)Potency6.309620
nan 190Homo sapiens (human)Potency15.848920
niclosamideHomo sapiens (human)Potency2.253620
nifedipineHomo sapiens (human)Potency0.667520
niflumic acidHomo sapiens (human)Potency11.079220
nimesulideHomo sapiens (human)Potency6.581220
nitrendipineHomo sapiens (human)Potency10.000020
masoprocolHomo sapiens (human)Potency5.011920
oxatomideHomo sapiens (human)Potency17.559420
oxethazaineHomo sapiens (human)Potency7.943320
oxibendazoleHomo sapiens (human)Potency2.511920
benoxinateHomo sapiens (human)Potency10.000020
4-(2'-methoxyphenyl)-1-(2'-(n-(2''-pyridinyl)-4-iodobenzamido)ethyl)piperazineHomo sapiens (human)Potency15.848920
papaverineHomo sapiens (human)Potency6.256020
phenazopyridineHomo sapiens (human)Potency0.631020
phenolsulfonphthaleinHomo sapiens (human)Potency0.199520
piretanideHomo sapiens (human)Potency1.000020
pomiferinHomo sapiens (human)Potency3.981120
prazosinHomo sapiens (human)Potency12.589320
prochlorperazineHomo sapiens (human)Potency25.118920
promazineHomo sapiens (human)Potency15.065420
propofolHomo sapiens (human)Potency25.118920
ritanserinHomo sapiens (human)Potency12.589320
sanguinarineHomo sapiens (human)Potency8.971620
sb 206553Homo sapiens (human)Potency12.589320
silymarinHomo sapiens (human)Potency12.589320
spiperoneHomo sapiens (human)Potency12.691420
sulfasalazineHomo sapiens (human)Potency0.223910
tetraisopropylpyrophosphamideHomo sapiens (human)Potency3.162320
thiabendazoleHomo sapiens (human)Potency2.511920
todralazineHomo sapiens (human)Potency7.943320
trazodoneHomo sapiens (human)Potency12.589320
trequinsinHomo sapiens (human)Potency6.309620
triamtereneHomo sapiens (human)Potency33.144330
tyrphostin a9Homo sapiens (human)Potency0.125920
5-methylurapidilHomo sapiens (human)Potency15.848920
3-(5'-hydroxymethyl-2'-furyl)-1-benzylindazoleHomo sapiens (human)Potency12.589320
hydrocortisone acetateHomo sapiens (human)Potency0.125920
corticosteroneHomo sapiens (human)Potency0.063120
3,3',5-triiodothyroacetic acidHomo sapiens (human)Potency6.309620
3,3',5-triiodothyropropionic acidHomo sapiens (human)Potency12.589320
prednisolone acetateHomo sapiens (human)Potency0.025120
prednisoneHomo sapiens (human)Potency35.481310
1,2,5,6-dibenzanthraceneHomo sapiens (human)Potency44.668410
dimethylphenylpiperazinium iodideHomo sapiens (human)Potency12.589320
cantharidinHomo sapiens (human)Potency2.511920
chlordanHomo sapiens (human)Potency79.432810
9,10-dimethyl-1,2-benzanthraceneHomo sapiens (human)Potency44.668410
promethazine hydrochlorideHomo sapiens (human)Potency12.589320
phenylephrineHomo sapiens (human)Potency0.251220
levodopaHomo sapiens (human)Potency10.000020
papaverine hydrochlorideHomo sapiens (human)Potency6.309620
fluocinolone acetonideHomo sapiens (human)Potency0.001320
cycloserineHomo sapiens (human)Potency1.584920
dinitrofluorobenzeneHomo sapiens (human)Potency50.118710
dichlorodiphenyldichloroethaneHomo sapiens (human)Potency79.432810
tryptophanHomo sapiens (human)Potency12.589320
triamcinolone acetonideHomo sapiens (human)Potency0.010020
hexachlorocyclopentadieneHomo sapiens (human)Potency12.589310
tetrabromobisphenol aHomo sapiens (human)Potency44.964710
quinophthaloneHomo sapiens (human)Potency0.398120
methylprednisoloneHomo sapiens (human)Potency0.050120
uvitex swnHomo sapiens (human)Potency44.668410
4,4'-thiobis(6-tert-butyl-3-cresol)Homo sapiens (human)Potency25.118910
fentichlorHomo sapiens (human)Potency39.810710
diglycidyl resorcinol etherHomo sapiens (human)Potency50.118710
monobenzoneHomo sapiens (human)Potency10.000020
phenforminHomo sapiens (human)Potency6.309620
dicofolHomo sapiens (human)Potency31.622810
chloranilHomo sapiens (human)Potency39.810710
cloropheneHomo sapiens (human)Potency79.432810
benzethonium chlorideHomo sapiens (human)Potency79.432810
suramin sodiumHomo sapiens (human)Potency12.589320
pyrazolanthroneHomo sapiens (human)Potency15.848920
dioxybenzoneHomo sapiens (human)Potency5.011920
captanHomo sapiens (human)Potency35.716810
2-Phenylethyl 2-aminobenzoateHomo sapiens (human)Potency50.118710
ziramHomo sapiens (human)Potency12.589310
4-nitrosodimethylanilineHomo sapiens (human)Potency50.118710
4'-(chloroacetyl)acetanilideHomo sapiens (human)Potency25.118910
sterogenolHomo sapiens (human)Potency50.118710
2-chloroadenosineHomo sapiens (human)Potency6.309620
benzo(b)fluorantheneHomo sapiens (human)Potency44.668410
benzo(k)fluorantheneHomo sapiens (human)Potency31.622810
chlormadinone acetateHomo sapiens (human)Potency0.100020
fluocinonideHomo sapiens (human)Potency0.001020
3,5-dinitro-4-chloro-alpha,alpha,alpha-trifluorotolueneHomo sapiens (human)Potency79.432810
fluorometholoneHomo sapiens (human)Potency0.010020
lithocholic acidHomo sapiens (human)Potency50.118710
boldineHomo sapiens (human)Potency1.995320
rheinHomo sapiens (human)Potency12.589320
podophyllotoxinHomo sapiens (human)Potency0.015820
medroxyprogesteroneHomo sapiens (human)Potency0.079420
domiphen bromideHomo sapiens (human)Potency31.622810
dicyclohexylcarbodiimideHomo sapiens (human)Potency79.432810
gentian violetHomo sapiens (human)Potency15.848910
chlorotrianiseneHomo sapiens (human)Potency10.000020
isoxsuprine hydrochlorideHomo sapiens (human)Potency0.125920
megestrol acetateHomo sapiens (human)Potency7.943320
pentabromophenolHomo sapiens (human)Potency39.810710
2-anthramineHomo sapiens (human)Potency50.118710
n-(1,3-dimethylbutyl)-n'-phenyl-1,4-phenylenediamineHomo sapiens (human)Potency50.118710
ethidium bromideHomo sapiens (human)Potency39.810710
flurandrenoloneHomo sapiens (human)Potency0.006320
pimozideHomo sapiens (human)Potency2.927620
benperidolHomo sapiens (human)Potency0.794320
flumethasoneHomo sapiens (human)Potency0.005020
azaribineHomo sapiens (human)Potency2.511920
hydrocortisone hemisuccinateHomo sapiens (human)Potency0.794320
antazoline hydrochlorideHomo sapiens (human)Potency12.589320
pontamine sky blueHomo sapiens (human)Potency6.309620
ethamsylateHomo sapiens (human)Potency0.398120
dichloroacetonitrileHomo sapiens (human)Potency31.622810
palmatineHomo sapiens (human)Potency12.589320
pentaerythrityl triacrylateHomo sapiens (human)Potency31.622810
diloxanide furoateHomo sapiens (human)Potency2.511920
2,2',4'-trichloroacetophenoneHomo sapiens (human)Potency25.118910
beclomethasoneHomo sapiens (human)Potency1.000020
2,2'-dihydroxy-6,6'-dinaphthyldisulfideHomo sapiens (human)Potency39.810710
methylene bis(thiocyanate)Homo sapiens (human)Potency19.952610
c.i. acid red 114, disodium saltHomo sapiens (human)Potency39.810710
levodopa methyl esterHomo sapiens (human)Potency15.848920
isoetharine mesylateHomo sapiens (human)Potency1.995320
camptothecinHomo sapiens (human)Potency0.102720
potassium dichromateHomo sapiens (human)Potency15.848910
hydroxyzine pamoateHomo sapiens (human)Potency7.943320
pyrithione zincHomo sapiens (human)Potency3.162310
parbendazoleHomo sapiens (human)Potency0.316220
tetraethylene glycol diacrylateHomo sapiens (human)Potency50.118710
ergocristineHomo sapiens (human)Potency10.000020
thiodiacetic acidHomo sapiens (human)Potency0.031620
triamcinoloneHomo sapiens (human)Potency0.031620
thymolphthaleinHomo sapiens (human)Potency3.162320
2-n-octyl-4-isothiazolin-3-oneHomo sapiens (human)Potency79.432810
moricizineHomo sapiens (human)Potency1.584920
ciclopirox olamineHomo sapiens (human)Potency0.316220
lonidamineHomo sapiens (human)Potency15.848920
torsemideHomo sapiens (human)Potency3.981120
lovastatinHomo sapiens (human)Potency33.144330
flupirtineHomo sapiens (human)Potency3.981120
3-chloro-4-(dichloromethyl)-5-hydroxy-2(5h)-furanoneHomo sapiens (human)Potency50.118710
remoxiprideHomo sapiens (human)Potency1.995320
eticloprideHomo sapiens (human)Potency10.000020
mibefradilHomo sapiens (human)Potency25.118920
topotecan hydrochlorideHomo sapiens (human)Potency0.251220
3-iodobenzylguanidineHomo sapiens (human)Potency12.589320
saquinavir monomethanesulfonateHomo sapiens (human)Potency79.432810
trichloropheneHomo sapiens (human)Potency3.162320
daunorubicin hydrochlorideHomo sapiens (human)Potency5.871030
nelfinavir mesylateHomo sapiens (human)Potency39.810710
amodiaquine hydrochlorideHomo sapiens (human)Potency5.011920
cyclenHomo sapiens (human)Potency12.589320
sulconazole, mononitrate, (+-)-isomerHomo sapiens (human)Potency10.000020
rutecarpineHomo sapiens (human)Potency15.848920
17 beta-estradiol hemisuccinateHomo sapiens (human)Potency5.011920
salicylhydroxamic acidHomo sapiens (human)Potency3.981120
miconazole nitrateHomo sapiens (human)Potency5.011920
econazole nitrateHomo sapiens (human)Potency17.207630
rilmenidineHomo sapiens (human)Potency25.118920
4-aminobenzo-2,1,3-thiadiazoleHomo sapiens (human)Potency3.162320
clobetasone butyrateHomo sapiens (human)Potency0.000820
masoprocolHomo sapiens (human)Potency7.943320
diflorasone diacetateHomo sapiens (human)Potency0.010020
hesperetinHomo sapiens (human)Potency5.011920
paceinHomo sapiens (human)Potency1.995320
tosyllysine chloromethyl ketoneHomo sapiens (human)Potency15.848920
ergocornineHomo sapiens (human)Potency0.398120
crystal violet lactoneHomo sapiens (human)Potency19.952610
atovaquoneHomo sapiens (human)Potency6.309620
5-aminoindazoleHomo sapiens (human)Potency10.000020
carbetapentane citrateHomo sapiens (human)Potency12.589320
salsolinolHomo sapiens (human)Potency1.995320
gliquidoneHomo sapiens (human)Potency2.511920
sk&f 95282Homo sapiens (human)Potency10.000020
meclizine hydrochlorideHomo sapiens (human)Potency12.589320
tarenflurbilHomo sapiens (human)Potency1.995320
corynanthineHomo sapiens (human)Potency15.848920
21-deoxycortisolHomo sapiens (human)Potency0.199520
cortisol octanoateHomo sapiens (human)Potency0.794320
azomethine hHomo sapiens (human)Potency1.258920
zpckHomo sapiens (human)Potency25.118920
n-acetyldopamineHomo sapiens (human)Potency12.589320
cp-55,940Homo sapiens (human)Potency31.622820
chlorethylclonidineHomo sapiens (human)Potency15.848920
methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylateHomo sapiens (human)Potency10.000020
vinpocetineHomo sapiens (human)Potency3.981120
benzamilHomo sapiens (human)Potency8.800620
carboxyamido-triazoleHomo sapiens (human)Potency3.162320
ponceau mxHomo sapiens (human)Potency0.079420
l 655240Homo sapiens (human)Potency12.589320
levalbuterolHomo sapiens (human)Potency0.337020
sr 2640Homo sapiens (human)Potency31.622820
n-(2-chloroethyl)-4-piperidinyl diphenylacetateHomo sapiens (human)Potency15.848920
n,n-di-n-hexyl-2-(4-fluorophenyl)indole-3-acetamideHomo sapiens (human)Potency25.118920
8-cyclopentyl-3-(3-((4-(fluorosulfonyl)benzoyl)oxy)propyl)-1-propylxanthineHomo sapiens (human)Potency31.622820
d-glutamineHomo sapiens (human)Potency10.000020
corbadrineHomo sapiens (human)Potency1.831820
17 alpha-hydroxyprogesterone caproateHomo sapiens (human)Potency3.981120
2-[carboxymethyl-[2-(2,6-diethylanilino)-2-oxoethyl]amino]acetic acidHomo sapiens (human)Potency0.501220
sb 216763Homo sapiens (human)Potency3.981120
ketoprofenHomo sapiens (human)Potency15.848920
chrysene-1,4-dioneHomo sapiens (human)Potency7.943320
n-(4-isothiocyanatophenethyl)spiperoneHomo sapiens (human)Potency15.848920
epinastineHomo sapiens (human)Potency0.007920
nsc 95397Homo sapiens (human)Potency6.309620
oxolamine citrateHomo sapiens (human)Potency12.589320
1-amino-9,10-dioxo-4-(3-sulfamoylanilino)anthracene-2-sulfonic acidHomo sapiens (human)Potency0.631020
6,11-dioxo-12-naphtho[2,3-b]indolizinecarboxylic acid ethyl esterHomo sapiens (human)Potency1.584920
graveolineHomo sapiens (human)Potency7.943320
nsc668394Homo sapiens (human)Potency0.158520
nsc681152Homo sapiens (human)Potency6.309620
methylmercuric chlorideHomo sapiens (human)Potency39.810710
nsc 146109Homo sapiens (human)Potency0.251220
nsc354961Homo sapiens (human)Potency5.011920
tosylphenylalanyl chloromethyl ketoneHomo sapiens (human)Potency25.118920
n-acetyl-d-tryptophanHomo sapiens (human)Potency1.000020
norpseudoephedrineHomo sapiens (human)Potency6.309620
raubasineHomo sapiens (human)Potency5.011920
L-isoprenalineHomo sapiens (human)Potency0.276720
sb 228357Homo sapiens (human)Potency3.981120
difluprednateHomo sapiens (human)Potency0.004020
doxorubicin hydrochlorideHomo sapiens (human)Potency6.674630
vinpocetineHomo sapiens (human)Potency6.309620
amcinonideHomo sapiens (human)Potency0.001320
flumethasone pivalateHomo sapiens (human)Potency0.000820
tretinoinHomo sapiens (human)Potency0.251220
resveratrolHomo sapiens (human)Potency10.000020
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolHomo sapiens (human)Potency25.118920
diethylstilbestrolHomo sapiens (human)Potency63.095710
purvalanol aHomo sapiens (human)Potency10.000020
dactinomycinHomo sapiens (human)Potency0.251210
aphidicolinHomo sapiens (human)Potency1.995320
melphalanHomo sapiens (human)Potency50.118710
nsc 45641Homo sapiens (human)Potency0.015820
tolfenamic acidHomo sapiens (human)Potency10.000020
opc-2009Homo sapiens (human)Potency2.511920
diethylstilbestrol dipropionateHomo sapiens (human)Potency1.995320
fludarabineHomo sapiens (human)Potency6.309620
dithizoneHomo sapiens (human)Potency10.000020
physostigmine salicylateHomo sapiens (human)Potency2.511920
r 59949Homo sapiens (human)Potency5.011920
1H-indazole-3-carboxylic acid methyl esterHomo sapiens (human)Potency10.000020
3,7-dimethyl-1-(phenylmethyl)-8-[(phenylmethyl)amino]purine-2,6-dioneHomo sapiens (human)Potency10.000020
6-ethyl-6-methyl-5,8-dihydro-1H-thiopyrano[2,3]thieno[2,4-b]pyrimidine-2,4-dioneHomo sapiens (human)Potency10.000020
2'-amino-5',6'-dimethoxy-1'-spiro[cyclopentane-1,3'-indene]carbonitrileHomo sapiens (human)Potency6.309620
6,6,7-trimethyl-1-(4-morpholinyl)-3-(phenylmethylthio)-5,8-dihydro-2,7-naphthyridine-4-carbonitrileHomo sapiens (human)Potency0.199520
2-[(3-oxo-5-phenyl-1,2-dihydropyrazol-4-yl)-(3-thiophenyl)methyl]propanedinitrileHomo sapiens (human)Potency10.000020
3-(4-butyl-3,5-dimethyl-1-pyrazolyl)-5-methyl-[1,2,4]triazino[5,6-b]indoleHomo sapiens (human)Potency0.398120
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3,3,3-trifluoro-2-methyl-2-(trifluoromethyl)propanamideHomo sapiens (human)Potency3.981120
2-amino-4-(2-chlorophenyl)-6-(ethylthio)pyridine-3,5-dicarbonitrileHomo sapiens (human)Potency3.981120
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2,2-bis(trifluoromethyl)butanamideHomo sapiens (human)Potency2.511920
1-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)Potency12.589320
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)Potency0.631020
4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl esterHomo sapiens (human)Potency12.589320
2-[[(4-chloro-1-methyl-3-pyrazolyl)-oxomethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterHomo sapiens (human)Potency10.000020
4-amino-5,8-dimethoxy-2-(1,1,2,2,2-pentafluoroethyl)-3-quinolinecarbonitrileHomo sapiens (human)Potency10.000020
5-[(3-ethoxycarbonyl-4-thiophen-2-yl-2-thiophenyl)amino]-5-oxopentanoic acidHomo sapiens (human)Potency1.584920
5-bromo-3-ethyl-1H-indole-2-carboxylic acidHomo sapiens (human)Potency10.000020
2-(4-methoxyphenyl)-1-(2-methylprop-2-enyl)benzimidazoleHomo sapiens (human)Potency12.589320
7-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxoethyl]amino]-5H-[1,3]dioxolo[4,5-f]indole-6-carboxylic acid ethyl esterHomo sapiens (human)Potency1.995320
arachinHomo sapiens (human)Potency5.011920
N-(3-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideHomo sapiens (human)Potency7.943320
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenolHomo sapiens (human)Potency10.000020
5-(4-methoxyphenyl)-7-(4-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency10.000020
3-[(4-methoxyanilino)methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency10.000020
3-(4-chlorophenyl)-6-(thiophen-2-ylmethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency2.511920
dienestrolHomo sapiens (human)Potency10.000020
ag-213Homo sapiens (human)Potency10.000020
carbidopa, (r)-isomerHomo sapiens (human)Potency7.943320
curcuminHomo sapiens (human)Potency6.309620
cinnarizineHomo sapiens (human)Potency12.589320
cis-resveratrolHomo sapiens (human)Potency7.875820
malachite greenHomo sapiens (human)Potency12.589310
capsazepineHomo sapiens (human)Potency5.011920
tamoxifen citrateHomo sapiens (human)Potency31.622830
tetraoctylammonium bromideHomo sapiens (human)Potency15.848910
ranitidineHomo sapiens (human)Potency3.981120
bp 897Homo sapiens (human)Potency6.924120
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency5.011920
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency5.011920
6-(3-furanyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency1.584920
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency1.995320
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.398120
6-(3-methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency1.995320
6-(3-furanyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency1.000020
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency0.631020
mannonateHomo sapiens (human)Potency0.199520
cambinolHomo sapiens (human)Potency3.162320
nsc-134754Homo sapiens (human)Potency3.162320
n-(1-methyl-5-indolyl)-n'-(3-methyl-5-isothiazolyl)ureaHomo sapiens (human)Potency12.589320
sb-224289Homo sapiens (human)Potency31.622820
1,8-dinitro-4,5-dihydroxyanthraquinoneHomo sapiens (human)Potency19.952610
gw 7647Homo sapiens (human)Potency5.011920
ro 41-0960Homo sapiens (human)Potency5.011920
cgp 13501Homo sapiens (human)Potency6.309620
pd 168,077Homo sapiens (human)Potency5.011920
or486Homo sapiens (human)Potency15.848920
iik7Homo sapiens (human)Potency10.000020
sb 415286Homo sapiens (human)Potency12.589320
LY-310762Homo sapiens (human)Potency15.848920
sc 560Homo sapiens (human)Potency5.011920
ly 367265Homo sapiens (human)Potency25.118920
diclofenac sodiumHomo sapiens (human)Potency15.714220
cgp 7930Homo sapiens (human)Potency12.589320
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazoleHomo sapiens (human)Potency3.162320
sib 1757Homo sapiens (human)Potency12.589320
quercetinHomo sapiens (human)Potency10.000020
biochanin aHomo sapiens (human)Potency10.000020
prostaglandin b1Homo sapiens (human)Potency0.100020
acacetinHomo sapiens (human)Potency0.794320
apigeninHomo sapiens (human)Potency7.292320
luteolinHomo sapiens (human)Potency0.398120
scopoletinHomo sapiens (human)Potency12.589320
kaempferolHomo sapiens (human)Potency1.584920
prostaglandin a2Homo sapiens (human)Potency2.511920
harmineHomo sapiens (human)Potency6.309620
genisteinHomo sapiens (human)Potency5.011920
pulmicortHomo sapiens (human)Potency0.000820
methysergide maleateHomo sapiens (human)Potency1.000020
esculetinHomo sapiens (human)Potency10.000020
chrysinHomo sapiens (human)Potency6.309620
myricetinHomo sapiens (human)Potency1.995320
coumestrolHomo sapiens (human)Potency10.000020
n-oleoyldopamineHomo sapiens (human)Potency31.622820
tranilastHomo sapiens (human)Potency7.943320
hydrocortisone valerateHomo sapiens (human)Potency0.005020
2-bromoergocryptine mesylateHomo sapiens (human)Potency3.162320
phenoxybenzamine hydrochlorideHomo sapiens (human)Potency18.814430
phenylephrine hydrochlorideHomo sapiens (human)Potency0.100020
quercetinHomo sapiens (human)Potency1.995320
tetrachlorvinphosHomo sapiens (human)Potency50.118710
toxapheneHomo sapiens (human)Potency79.432810
afimoxifeneHomo sapiens (human)Potency79.432810
fenretinideHomo sapiens (human)Potency39.810710
ic 261Homo sapiens (human)Potency0.050120
denopamineHomo sapiens (human)Potency2.511920
desoximetasoneHomo sapiens (human)Potency0.005020
l 745870Homo sapiens (human)Potency12.589320
su 6656Homo sapiens (human)Potency19.952620
ag 538Homo sapiens (human)Potency7.943320
tyrphostin ag 555Homo sapiens (human)Potency10.266320
tyrphostin ag-494Homo sapiens (human)Potency10.000020
ag-490Homo sapiens (human)Potency10.000020
ag 112Homo sapiens (human)Potency15.848920
molsidomineHomo sapiens (human)Potency0.316220
rg 13022Homo sapiens (human)Potency0.501220
fluvoxamineHomo sapiens (human)Potency11.896120
dichlorisone acetateHomo sapiens (human)Potency0.005020
trimebutine maleate saltHomo sapiens (human)Potency1.258920
vinblastine sulfateHomo sapiens (human)Potency0.031620
vincristine sulfateHomo sapiens (human)Potency0.063120
zimeldineHomo sapiens (human)Potency1.258920
s-trans,trans-farnesylthiosalicylic acidHomo sapiens (human)Potency25.118920
sulindac sulfoneHomo sapiens (human)Potency15.848920
ici 118551Homo sapiens (human)Potency12.589320
gw-5074Homo sapiens (human)Potency25.118920
7-chloro-4-hydroxy-2-phenyl-1,8-naphthyridineHomo sapiens (human)Potency3.981120
pregna-4,17-diene-3,16-dione, (17z)-isomerHomo sapiens (human)Potency79.432810
gw 1929Homo sapiens (human)Potency1.995320
a 77636Homo sapiens (human)Potency3.981120
b 43Homo sapiens (human)Potency31.622820
(8R)-7-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triolHomo sapiens (human)Potency2.511920
(8R)-7-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triolHomo sapiens (human)Potency2.511920
dihydrexidineHomo sapiens (human)Potency5.011920
4-(2-(phenylsulfonylamino)ethylthio)-2,6-difluorophenoxyacetamideHomo sapiens (human)Potency25.118920
gw2974Homo sapiens (human)Potency0.794320
l 750667Homo sapiens (human)Potency3.162320
l 162313Homo sapiens (human)Potency31.622820
5-(4-phenylbutoxy)psoralenHomo sapiens (human)Potency25.118920
sb 222200Homo sapiens (human)Potency19.952620
cycloheximideHomo sapiens (human)Potency0.063120
suloctidilHomo sapiens (human)Potency5.011920
methiazoleHomo sapiens (human)Potency3.162320
dibenzheptropine citrateHomo sapiens (human)Potency3.981120
chlorhexidineHomo sapiens (human)Potency31.622810
phenylmercuric acetateHomo sapiens (human)Potency2.511910
meclofenamate sodium anhydrousHomo sapiens (human)Potency6.309620
cytomelHomo sapiens (human)Potency10.000020
prednisolone sodium succinateHomo sapiens (human)Potency0.631020
cortisol succinate, sodium saltHomo sapiens (human)Potency0.631020
nafcillin sodiumHomo sapiens (human)Potency12.589320
oxytetracycline, anhydrousHomo sapiens (human)Potency7.943320
sepiapterinHomo sapiens (human)Potency10.000020
ganciclovirHomo sapiens (human)Potency3.981120
zaprinastHomo sapiens (human)Potency7.506020
hli 373Homo sapiens (human)Potency2.511920
azaguanineHomo sapiens (human)Potency7.943320
ag-879Homo sapiens (human)Potency0.631020
N-tert-butyl-3-(3-tert-butyl-1-methyl-7-oxo-4H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxybenzenesulfonamideHomo sapiens (human)Potency10.000020