Page last updated: 2024-08-07 23:10:03
Pancreatic triacylglycerol lipase
[no definition available]
Synonyms
PL;
PTL;
Pancreatic lipase;
EC 3.1.1.3
Research
Bioassay Publications (19)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 17 (89.47) | 24.3611 |
2020's | 2 (10.53) | 2.80 |
Compounds (42)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
gallic acid | Sus scrofa (pig) | IC50 | 1,000.0000 | 1 | 1 |
vanillin | Sus scrofa (pig) | IC50 | 74.4000 | 1 | 1 |
phloretin | Sus scrofa (pig) | IC50 | 50.4000 | 1 | 1 |
phlorhizin | Sus scrofa (pig) | IC50 | 300.0000 | 1 | 1 |
rotenone | Sus scrofa (pig) | IC50 | 500.0000 | 1 | 1 |
vanillic acid | Sus scrofa (pig) | IC50 | 250.0000 | 1 | 1 |
catechin | Sus scrofa (pig) | IC50 | 500.0000 | 1 | 1 |
aromadedrin | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
moracin c | Sus scrofa (pig) | IC50 | 32.0000 | 1 | 1 |
moracin m | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
naringenin | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
lusianthridin | Sus scrofa (pig) | Ki | 4.9600 | 1 | 1 |
Hircinol | Sus scrofa (pig) | Ki | 8.5700 | 1 | 1 |
6,8-diprenylgenistein | Sus scrofa (pig) | IC50 | 65.0000 | 1 | 1 |
8-isopentenylnaringenin | Sus scrofa (pig) | IC50 | 76.9000 | 1 | 1 |
hydroxyphenethylferulate | Sus scrofa (pig) | IC50 | 50.0000 | 1 | 1 |
chalcone | Sus scrofa (pig) | IC50 | 84.4100 | 1 | 1 |
caffeic acid | Sus scrofa (pig) | IC50 | 1,000.0000 | 1 | 1 |
orlistat | Sus scrofa (pig) | IC50 | 0.4214 | 14 | 14 |
orlistat | Sus scrofa (pig) | Ki | 5.0300 | 2 | 2 |
quercetin | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
biochanin a | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
quercetin 3-o-glucopyranoside | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
kaempferol | Sus scrofa (pig) | IC50 | 85.0000 | 2 | 2 |
genistein | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
5,7-dihydroxychromone | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
3-methylquercetin | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
morin | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
trans-2,3',4,5'-tetrahydroxystilbene | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
wighteone | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
astragalin | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
broussonin a | Sus scrofa (pig) | IC50 | 98.7000 | 1 | 1 |
broussonin b | Sus scrofa (pig) | IC50 | 75.4000 | 1 | 1 |
3'-o-methylorobol | Sus scrofa (pig) | IC50 | 100.0000 | 1 | 1 |
Norartocarpetin | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
lipstatin | Sus scrofa (pig) | IC50 | 0.1400 | 1 | 1 |
morachalcone a | Sus scrofa (pig) | IC50 | 6.2000 | 1 | 1 |
1,7-bis(4-hydroxyphenyl)-1,4,6-heptatrien-3-one | Sus scrofa (pig) | Ki | 3.3400 | 1 | 1 |
batatasin-iii | Sus scrofa (pig) | Ki | 6.7900 | 1 | 1 |
1,7-bis(4-hydroxyphenyl)hepta-4E-6E-dien-3-one | Sus scrofa (pig) | Ki | 1.9200 | 1 | 1 |
Norartocarpanone | Sus scrofa (pig) | IC50 | 70.0000 | 1 | 1 |
cudraflavanone a | Sus scrofa (pig) | IC50 | 6.5000 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
orlistat | Sus scrofa (pig) | Km | 225.8400 | 3 | 3 |
caffeic acid phenethyl ester | Sus scrofa (pig) | ED50 | 10.0000 | 1 | 1 |