Page last updated: 2024-08-07 16:45:13
Melatonin receptor type 1C
[no definition available]
Synonyms
Mel-1C-R;
Mel1c (alpha) receptor;
Mel1c receptor
Research
Bioassay Publications (3)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (66.67) | 29.6817 |
| 2010's | 1 (33.33) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| luzindole | Xenopus laevis (African clawed frog) | IC50 | 2.4547 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| melatonin | Xenopus laevis (African clawed frog) | EC50 | 0.0001 | 3 | 3 |
Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists.MedChemComm, , Mar-01, Volume: 10, Issue:3, 2019
7-Substituted-melatonin and 7-substituted-1-methylmelatonin analogues: effect of substituents on potency and binding affinity.Bioorganic & medicinal chemistry, , Jul-01, Volume: 15, Issue:13, 2007
Design, synthesis and melatoninergic activity of new unsubstituted and beta,beta'-difunctionalised 2,3-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-6-alkanamides.European journal of medicinal chemistry, , Volume: 42, Issue:7, 2007