Page last updated: 2024-08-07 22:52:36

NPC intracellular cholesterol transporter 1 precursor

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (1338)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
quinacrineHomo sapiens (human)Potency58.047910
catecholHomo sapiens (human)Potency115.821010
hydroquinoneHomo sapiens (human)Potency91.999710
octoclothepineHomo sapiens (human)Potency91.999710
s,s'-1,4-phenylene-bis(1,2-ethanediyl)bis-isothioureaHomo sapiens (human)Potency23.109310
2-aminofluoreneHomo sapiens (human)Potency3.981110
5-(n,n-hexamethylene)amilorideHomo sapiens (human)Potency2.818410
ag 1295Homo sapiens (human)Potency1.258910
amlexanoxHomo sapiens (human)Potency0.316210
anisindioneHomo sapiens (human)Potency5.623410
calmidazoliumHomo sapiens (human)Potency58.047910
cantharidinHomo sapiens (human)Potency36.625710
chelerythrineHomo sapiens (human)Potency58.047910
citalopramHomo sapiens (human)Potency20.596210
dequaliniumHomo sapiens (human)Potency183.564010
diphenyleneiodoniumHomo sapiens (human)Potency183.564010
ebastineHomo sapiens (human)Potency46.109110
ellipticineHomo sapiens (human)Potency30.605110
emodinHomo sapiens (human)Potency20.596210
fluoxetineHomo sapiens (human)Potency58.047910
fluspirileneHomo sapiens (human)Potency58.047910
vanoxerineHomo sapiens (human)Potency58.047910
gossypolHomo sapiens (human)Potency91.999710
hexachloropheneHomo sapiens (human)Potency3.162310
hydralazineHomo sapiens (human)Potency2.592910
phenelzineHomo sapiens (human)Potency10.322510
indirubin-3'-monoximeHomo sapiens (human)Potency4.610910
indoprofenHomo sapiens (human)Potency0.089110
ipriflavoneHomo sapiens (human)Potency0.647810
1-(2-naphthalenyl)-3-[(phenylmethyl)-propan-2-ylamino]-1-propanoneHomo sapiens (human)Potency58.047910
nsc 664704Homo sapiens (human)Potency0.517410
ketorolacHomo sapiens (human)Potency10.322510
lansoprazoleHomo sapiens (human)Potency3.036810
leflunomideHomo sapiens (human)Potency1.199010
loratadineHomo sapiens (human)Potency58.047910
maprotilineHomo sapiens (human)Potency58.047910
methiothepinHomo sapiens (human)Potency73.078010
nocodazoleHomo sapiens (human)Potency7.307810
mitoxantroneHomo sapiens (human)Potency115.821010
fg 7142Homo sapiens (human)Potency12.995310
clorgylineHomo sapiens (human)Potency16.360110
nabumetoneHomo sapiens (human)Potency2.818410
nicardipineHomo sapiens (human)Potency115.821010
niclosamideHomo sapiens (human)Potency0.052410
nortriptylineHomo sapiens (human)Potency58.047910
5-nitro-2-(3-phenylpropylamino)benzoic acidHomo sapiens (human)Potency20.596210
pd 98059Homo sapiens (human)Potency2.310910
perphenazineHomo sapiens (human)Potency58.047910
prazosinHomo sapiens (human)Potency58.047910
riluzoleHomo sapiens (human)Potency10.322510
ritanserinHomo sapiens (human)Potency58.047910
aurinHomo sapiens (human)Potency3.548110
sanguinarineHomo sapiens (human)Potency145.810010
sb 206553Homo sapiens (human)Potency3.662610
spiperoneHomo sapiens (human)Potency94.593710
streptonigrinHomo sapiens (human)Potency0.562310
terfenadineHomo sapiens (human)Potency91.999710
thiabendazoleHomo sapiens (human)Potency3.548110
thioridazineHomo sapiens (human)Potency58.047910
trifluoperazineHomo sapiens (human)Potency58.047910
triflupromazineHomo sapiens (human)Potency58.047910
tyrphostin a9Homo sapiens (human)Potency37.168410
3-(5'-hydroxymethyl-2'-furyl)-1-benzylindazoleHomo sapiens (human)Potency184.126210
methyldimethylaminoazobenzeneHomo sapiens (human)Potency0.631010
strophanthidinHomo sapiens (human)Potency1.778310
cycloheximideHomo sapiens (human)Potency0.446710
1-amino-2-methylanthraquinoneHomo sapiens (human)Potency3.162310
quinophthaloneHomo sapiens (human)Potency5.623410
rotenoneHomo sapiens (human)Potency290.929010
9,10-phenanthrenequinoneHomo sapiens (human)Potency3.548110
1-(2-pyridylazo)-2-naphtholHomo sapiens (human)Potency1.258910
dehydrothio-4-toluidineHomo sapiens (human)Potency0.316210
triclocarbanHomo sapiens (human)Potency5.623410
2-aminoanthraquinoneHomo sapiens (human)Potency3.548110
pyrazolanthroneHomo sapiens (human)Potency10.322510
naphthyl redHomo sapiens (human)Potency3.548110
2-Phenylethyl 2-aminobenzoateHomo sapiens (human)Potency1.122010
peucedaninHomo sapiens (human)Potency2.818410
cepharanthineHomo sapiens (human)Potency3.981110
emetineHomo sapiens (human)Potency58.047910
podophyllotoxinHomo sapiens (human)Potency0.501210
flavoneHomo sapiens (human)Potency5.623410
4,4'-diaminoazobenzeneHomo sapiens (human)Potency0.501210
aminacrineHomo sapiens (human)Potency2.818410
2-phenylbenzimidazoleHomo sapiens (human)Potency3.548110
2,5-diphenyloxazoleHomo sapiens (human)Potency1.584910
2-phenylindoleHomo sapiens (human)Potency3.548110
c 137Homo sapiens (human)Potency3.981110
bromindioneHomo sapiens (human)Potency3.548110
digoxigeninHomo sapiens (human)Potency3.981110
4-hydroxyazobenzeneHomo sapiens (human)Potency6.309610
drometrizoleHomo sapiens (human)Potency3.162310
nsc 3852Homo sapiens (human)Potency3.981110
2-(alpha-thenoylamino)-2-nitro-5-thiazoleHomo sapiens (human)Potency0.891310
nitroxolineHomo sapiens (human)Potency6.309610
4-(4-dimethylaminophenylazo)benzoic acidHomo sapiens (human)Potency0.012610
helenalinHomo sapiens (human)Potency0.794310
marmesin, (r)-isomerHomo sapiens (human)Potency2.511910
metergolineHomo sapiens (human)Potency58.047910
1-(4-carboxyethylphenyl)-3,3-dimethyltriazeneHomo sapiens (human)Potency5.623410
frentizoleHomo sapiens (human)Potency5.623410
N-fluorenylacetamideHomo sapiens (human)Potency3.548110
paclitaxelHomo sapiens (human)Potency3.548110
isovelleralHomo sapiens (human)Potency3.548110
nitazoxanideHomo sapiens (human)Potency0.501210
s-2678Homo sapiens (human)Potency6.309610
dinalineHomo sapiens (human)Potency12.006320
idarubicinHomo sapiens (human)Potency115.821010
paroxetineHomo sapiens (human)Potency58.047910
chaetochrominHomo sapiens (human)Potency1.412510
idazoxanHomo sapiens (human)Potency58.047910
mibefradilHomo sapiens (human)Potency58.047910
daunorubicin hydrochlorideHomo sapiens (human)Potency0.316210
3,4-dihydro-2(1h)-quinolinoneHomo sapiens (human)Potency1.000010
nile redHomo sapiens (human)Potency0.562310
xanthyletineHomo sapiens (human)Potency3.162310
rutecarpineHomo sapiens (human)Potency4.266410
pifexoleHomo sapiens (human)Potency3.399810
toxoflavinHomo sapiens (human)Potency1.412510
dimidium bromideHomo sapiens (human)Potency1.000010
sertralineHomo sapiens (human)Potency58.047910
2-(2'-pyridyl)benzimidazoleHomo sapiens (human)Potency3.981110
6-hydroxyflavoneHomo sapiens (human)Potency2.818410
hesperetinHomo sapiens (human)Potency5.623410
2-phenyl-4,5-dichloro-3-pyridazinoneHomo sapiens (human)Potency3.162310
tryptanthrineHomo sapiens (human)Potency2.818410
4'-methoxyflavoneHomo sapiens (human)Potency2.511910
2-(4-Morpholinyl)benzothiazoleHomo sapiens (human)Potency3.548110
N-(4-ethoxyphenyl)-3-hydroxy-2-naphthalenecarboxamideHomo sapiens (human)Potency1.258910
2-methyl-4-nitroquinoline 1-oxideHomo sapiens (human)Potency2.818410
2-(1H-benzimidazol-2-yl)anilineHomo sapiens (human)Potency3.981110
witisolHomo sapiens (human)Potency1.122010
5,7-dimethoxyflavoneHomo sapiens (human)Potency2.238710
pyridabenHomo sapiens (human)Potency0.089110
phenylisopropyladenosineHomo sapiens (human)Potency16.360110
coumarin 7Homo sapiens (human)Potency0.281810
efuamideHomo sapiens (human)Potency1.412510
2-(2'-hydroxy-3'-methoxyphenyl)benzothiazoleHomo sapiens (human)Potency5.623410
girinimbineHomo sapiens (human)Potency3.162310
zpckHomo sapiens (human)Potency91.999710
n(6)-phenyladenosineHomo sapiens (human)Potency9.064610
4'-methoxyflavanoneHomo sapiens (human)Potency5.623410
cp-55,940Homo sapiens (human)Potency58.047910
beta-carboline-3-carboxylic acid ethyl esterHomo sapiens (human)Potency3.162310
sudan yellow 3gHomo sapiens (human)Potency3.162310
triptolideHomo sapiens (human)Potency0.089110
benzamilHomo sapiens (human)Potency25.929010
pefloxacin mesylateHomo sapiens (human)Potency1.258910
tetradecanoylphorbol acetateHomo sapiens (human)Potency58.047910
nsc 607097Homo sapiens (human)Potency0.251210
indatralineHomo sapiens (human)Potency58.047910
sr 2640Homo sapiens (human)Potency23.109310
8-cyclopentyl-3-(3-((4-(fluorosulfonyl)benzoyl)oxy)propyl)-1-propylxanthineHomo sapiens (human)Potency91.999710
l 741626Homo sapiens (human)Potency58.047910
1,4-di(2'-thienyl)-1,4-butadioneHomo sapiens (human)Potency1.258910
sch 45752Homo sapiens (human)Potency1.584910
enniatin bHomo sapiens (human)Potency4.466810
4'-hydroxyflavanoneHomo sapiens (human)Potency5.623410
fiduxosinHomo sapiens (human)Potency58.047910
sch 58261Homo sapiens (human)Potency5.804810
4',6-dihydroxyflavoneHomo sapiens (human)Potency5.623410
N-(4-methoxyphenyl)carbamic acid propan-2-yl esterHomo sapiens (human)Potency1.995310
phenserineHomo sapiens (human)Potency9.200010
fonsecinHomo sapiens (human)Potency2.511910
N-(4-methoxyphenyl)-1,3-benzothiazol-2-amineHomo sapiens (human)Potency2.511910
N-tert-butyl-6-ethyl-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency3.981110
gossypol acetic acidHomo sapiens (human)Potency3.981110
4'-hydroxyflavoneHomo sapiens (human)Potency5.623410
N-(3-chlorophenyl)carbamic acid 2-pyridinylmethyl esterHomo sapiens (human)Potency4.466810
(R)-RoemerineHomo sapiens (human)Potency62.841710
2-pyridin-4-yl-1,3-benzothiazoleHomo sapiens (human)Potency3.162310
N-(3-fluorophenyl)benzamideHomo sapiens (human)Potency2.511910
1',2'-dihydrorotenoneHomo sapiens (human)Potency1.122010
1-(2,4-Dihydroxyphenyl)-2-(4-methoxyphenyl)ethanoneHomo sapiens (human)Potency3.548110
nsc 95397Homo sapiens (human)Potency59.491610
2-chloro-3-(4-methylanilino)naphthalene-1,4-dioneHomo sapiens (human)Potency6.309610
methylnaphthazarinHomo sapiens (human)Potency1.584910
aromaticinHomo sapiens (human)Potency3.548110
1-(4-chlorophenyl)-3-(2-ethoxyphenyl)ureaHomo sapiens (human)Potency0.631010
2-(4-aminophenyl)quinolineHomo sapiens (human)Potency1.458110
4-methoxyxanthoneHomo sapiens (human)Potency3.162310
2-[[[4-(methylthio)anilino]-oxomethyl]amino]benzamideHomo sapiens (human)Potency2.511910
nsc228155Homo sapiens (human)Potency3.981110
N-[2-(1-azepanyl)-1,3-benzothiazol-6-yl]carbamic acid ethyl esterHomo sapiens (human)Potency0.446710
4-amino-N-(4-methoxyphenyl)-2-(methylthio)-5-thiazolecarboxamideHomo sapiens (human)Potency3.162310
pifithrin muHomo sapiens (human)Potency73.078010
5-(1,3-benzodioxol-5-yl)-N-(2,4-dimethylphenyl)-1,3,4-oxadiazol-2-amineHomo sapiens (human)Potency3.548110
(5-amino-3-triazolo[1,5-a]quinazolinyl)-(4-morpholinyl)methanoneHomo sapiens (human)Potency3.162310
6-(4-chlorophenyl)-2,3-dihydroimidazo[2,1-b]thiazoleHomo sapiens (human)Potency1.778310
11,12-dihydro-4-methoxydibenz(b,f)(1,4)oxazepine-8-carboxylateHomo sapiens (human)Potency2.511910
N-phenylcarbamic acid 2-phenoxyethyl esterHomo sapiens (human)Potency3.981110
3-phenyl-1H-quinoxalin-2-oneHomo sapiens (human)Potency3.162310
DubamineHomo sapiens (human)Potency0.562310
7-(4-methoxyphenyl)-5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency3.981110
2,3-diaminophenazineHomo sapiens (human)Potency5.011910
ouabainHomo sapiens (human)Potency77.266810
digitoxinHomo sapiens (human)Potency0.251210
angustibalinHomo sapiens (human)Potency0.631010
doxorubicin hydrochlorideHomo sapiens (human)Potency0.251210
resveratrolHomo sapiens (human)Potency11.989910
thapsigarginHomo sapiens (human)Potency145.810010
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolHomo sapiens (human)Potency58.047910
6-bromoindirubin-3'-oximeHomo sapiens (human)Potency3.228710
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency1.584910
4-(2-oxazolo[4,5-b]pyridinyl)anilineHomo sapiens (human)Potency3.162310
2-[(4-nitrophenyl)methylthio]-1,3-benzoxazoleHomo sapiens (human)Potency0.631010
2-[(2-nitrophenyl)methylthio]-1,3-benzoxazoleHomo sapiens (human)Potency3.162310
2-(4-chlorophenyl)-1-phthalazinoneHomo sapiens (human)Potency1.412510
3-(4-chlorophenyl)-6-(1-pyrrolidinyl)-1,2,4,5-tetrazineHomo sapiens (human)Potency1.995310
2-(1H-benzimidazol-2-ylthio)-1-thiophen-2-ylethanoneHomo sapiens (human)Potency1.258910
2-(3-nitrophenyl)-5-phenyl-1,3,4-oxadiazoleHomo sapiens (human)Potency2.818410
5-(2-furanyl)-3-(3-pyridinyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency3.162310
3-(1-azepanylazo)benzoic acidHomo sapiens (human)Potency0.100010
4-[[7-bicyclo[4.1.0]heptanyl(oxo)methyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency2.238710
3-(4-fluoroanilino)-1-(3-nitrophenyl)-1-propanoneHomo sapiens (human)Potency5.623410
4-[2-(4-methoxycarbonylphenyl)iminohydrazinyl]benzoic acid methyl esterHomo sapiens (human)Potency0.199510
3-(4-bromophenyl)-1,2,3-benzotriazin-4-oneHomo sapiens (human)Potency3.162310
6-propan-2-yl-1,3-benzothiazol-2-amineHomo sapiens (human)Potency1.584910
5-methoxy-3-methyl-1H-indole-2-carboxylic acid ethyl esterHomo sapiens (human)Potency5.623410
4-(2-pyridinylthio)benzofuro[3,2-d]pyrimidineHomo sapiens (human)Potency3.548110
cabreuvinHomo sapiens (human)Potency2.818410
2,3-diphenyl-6-quinoxalinecarboxylic acidHomo sapiens (human)Potency3.162310
piplartineHomo sapiens (human)Potency6.309610
7-methoxyisoflavoneHomo sapiens (human)Potency0.707910
piperineHomo sapiens (human)Potency2.511910
ilepcimideHomo sapiens (human)Potency3.548110
cgp 60474Homo sapiens (human)Potency0.794310
3-(2-phenoxyethyl)-1,3-benzothiazol-2-oneHomo sapiens (human)Potency2.238710
N-[2-(1-cyclohexenyl)ethyl]-4-(4-morpholinylmethyl)benzamideHomo sapiens (human)Potency2.818410
1-[2,5-diethoxy-4-(1-tetrazolyl)phenyl]sulfonyl-4-(4-fluorophenyl)-3,6-dihydro-2H-pyridineHomo sapiens (human)Potency3.548110
2-oxo-N-(2-pyridinylmethyl)-1-benzopyran-3-carboxamideHomo sapiens (human)Potency3.162310
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency2.818410
4-[[2-(1-benzotriazolyl)-1-oxoethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency3.548110
4-chloro-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)benzamideHomo sapiens (human)Potency3.548110
3-methyl-4-(7-methyl-2-indolizinyl)-1,2,5-oxadiazoleHomo sapiens (human)Potency3.981110
N,N-dimethyl-6-phenyl-3-pyridazinamineHomo sapiens (human)Potency1.584910
2-(4-bromophenyl)-5-(2-methylphenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency1.995310
N-(1,3-benzothiazol-2-yl)-N-methylbenzamideHomo sapiens (human)Potency0.281810
4-[2-[1-(4-methoxyphenyl)sulfonyl-2-benzimidazolyl]ethyl]morpholineHomo sapiens (human)Potency1.258910
5-(2-furanyl)-3-[2-methoxy-6-(4-methylphenyl)-3-pyridinyl]-1,2,4-oxadiazoleHomo sapiens (human)Potency3.548110
N-cyclohexyl-N,4-dimethyl-5-thieno[3,2-b]pyrrolecarboxamideHomo sapiens (human)Potency3.981110
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-N-[2-(4-morpholinyl)phenyl]acetamideHomo sapiens (human)Potency1.584910
5-[3-(dimethylamino)phenyl]-N-methyl-1,3,4-thiadiazol-2-amineHomo sapiens (human)Potency6.309610
[3-[3-(5-methyl-2-furanyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]-phenylmethanoneHomo sapiens (human)Potency3.162310
N-[4-[oxo-(2-pyridinylamino)methyl]phenyl]-2-furancarboxamideHomo sapiens (human)Potency2.238710
N-(3-fluoro-4-methylphenyl)-1-(2-pyrimidinyl)-3-piperidinecarboxamideHomo sapiens (human)Potency3.548110
N-[2-(4-methoxyphenyl)-6-methyl-5-benzotriazolyl]-3-pyridinecarboxamideHomo sapiens (human)Potency3.548110
5-(2-ethoxyphenyl)-3-(2-methoxy-6-methyl-3-pyridinyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency4.466810
N-(1,3-benzodioxol-5-yl)-3-[(2-methyl-1-oxopropyl)amino]benzamideHomo sapiens (human)Potency2.818410
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-1-(1-piperidinyl)ethanoneHomo sapiens (human)Potency0.562310
1-(4-methoxyphenyl)-2-(5-thiophen-2-yl-2-tetrazolyl)ethanoneHomo sapiens (human)Potency3.548110
N-(3-dibenzofuranyl)-4-morpholinecarboxamideHomo sapiens (human)Potency3.548110
1-(3-chlorophenyl)-3-[4-[4-morpholinyl(oxo)methyl]phenyl]ureaHomo sapiens (human)Potency3.548110
N-[2-methoxy-4-[(2-methyl-1-oxopropyl)amino]phenyl]-2-furancarboxamideHomo sapiens (human)Potency3.981110
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency3.162310
2-(ethylthio)-5-(4-methoxyphenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency2.818410
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-methoxyacetamideHomo sapiens (human)Potency1.995310
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2-pyrimidinyl)-3-piperidinecarboxamideHomo sapiens (human)Potency0.398110
1-cyclohexyl-5-(2-phenoxyethylthio)tetrazoleHomo sapiens (human)Potency0.562310
N-(5-methoxy-1,3-benzothiazol-2-yl)-3-methylbutanamideHomo sapiens (human)Potency4.466810
6-phenyl-4-(1-pyrrolyl)furo[2,3-d]pyrimidineHomo sapiens (human)Potency6.309610
N,N-diethyl-2-[(3-thiophen-2-yl-7-isothiazolo[4,5-d]pyrimidinyl)thio]acetamideHomo sapiens (human)Potency3.548110
5-amino-2-(4-methylphenyl)isoindole-1,3-dioneHomo sapiens (human)Potency3.548110
N-[3-chloro-4-(4-morpholinyl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency1.412510
5-[(2-fluoroanilino)methyl]-8-quinolinolHomo sapiens (human)Potency1.258910
2-(4,5-dihydrothiazol-2-ylthio)-N-(6-methoxy-1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)Potency3.981110
1-[5-(2-amino-5-methyl-4-thiazolyl)-2,3-dihydroindol-1-yl]-1-butanoneHomo sapiens (human)Potency5.623410
6,7-dimethoxy-2-(2-thiazolyl)-3H-isoindol-1-oneHomo sapiens (human)Potency2.511910
N-(3-methoxyphenyl)-2-(2-pyridinylthio)acetamideHomo sapiens (human)Potency5.623410
2-[[2-(3-methoxyphenoxy)-1-oxoethyl]amino]benzamideHomo sapiens (human)Potency3.548110
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)Potency3.981110
N-(1,3-benzodioxol-5-yl)-5-bromo-3-pyridinecarboxamideHomo sapiens (human)Potency2.511910
N-[2-(1-cyclohexenyl)ethyl]-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency1.778310
2-(4-chlorophenyl)-5-(methylamino)-4-oxazolecarbonitrileHomo sapiens (human)Potency2.511910
N-(2-oxolanylmethyl)-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency1.995310
1-phenyl-N-(3-propan-2-yloxypropyl)-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency1.412510
2-[2-[[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]amino]ethoxy]ethanolHomo sapiens (human)Potency1.122010
1-(4-chlorophenyl)-N-(1-methoxypropan-2-yl)-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency0.707910
1-[1-(4-methoxyphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-4-piperidinecarboxamideHomo sapiens (human)Potency3.548110
2-[2-[(1-phenyl-4-pyrazolo[3,4-d]pyrimidinyl)amino]ethoxy]ethanolHomo sapiens (human)Potency2.238710
1-methyl-2-[(phenylthio)methyl]-3-indolecarbonitrileHomo sapiens (human)Potency2.238710
1-[(4-methylphenyl)methyl]-4-[4-(4-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineHomo sapiens (human)Potency3.548110
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency3.981110
4-(2-furanyl)-3-methyl-5-(4-methylphenyl)-2,4-dihydropyrrolo[3,4-c]pyrazol-6-oneHomo sapiens (human)Potency3.981110
LSM-32400Homo sapiens (human)Potency0.794310
2-(4-benzofuro[3,2-d]pyrimidinylthio)-1-thiophen-2-ylethanoneHomo sapiens (human)Potency2.818410
2-methoxy-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-methoxyphenyl)acetamideHomo sapiens (human)Potency5.623410
3-phenyl-1H-cinnolin-4-oneHomo sapiens (human)Potency2.238710
3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpropanamideHomo sapiens (human)Potency2.818410
N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-furancarboxamideHomo sapiens (human)Potency3.981110
N-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency2.818410
2-[[3-[4-(dimethylamino)phenyl]-4,5-dihydroisoxazol-5-yl]methyl]-1,1-dioxo-1,2-benzothiazol-3-oneHomo sapiens (human)Potency3.162310
7-methyl-3-(3-methylbutylamino)-1-(1-pyrrolidinyl)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileHomo sapiens (human)Potency0.112210
N-(3,4-dihydro-1H-[1,4]thiazino[4,3-a]benzimidazol-8-yl)pentanamideHomo sapiens (human)Potency3.548110
4-[[1-oxo-2-(3-oxo-2-thiomorpholinyl)ethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency2.238710
N-(3,4-dihydro-1H-[1,4]thiazino[4,3-a]benzimidazol-8-yl)butanamideHomo sapiens (human)Potency3.548110
3,3',4,5'-tetrahydroxystilbeneHomo sapiens (human)Potency6.513110
N-(4-phenylmethoxyphenyl)methanesulfonamideHomo sapiens (human)Potency2.818410
N-(4-acetylphenyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency2.818410
4-methoxy-N-(5-methyl-3-isoxazolyl)benzamideHomo sapiens (human)Potency1.995310
2,4-difluoro-N-[[(5-methyl-1H-pyrazol-3-yl)amino]-oxomethyl]benzamideHomo sapiens (human)Potency0.501210
3,4-methylenedioxy-beta-nitrostyreneHomo sapiens (human)Potency58.047910
5-[(1,3-benzothiazol-2-ylthio)methyl]-2-furancarboxylic acid methyl esterHomo sapiens (human)Potency2.818410
N-(2-fluorophenyl)-4-phenylmethoxybenzamideHomo sapiens (human)Potency3.162310
N-[4-(diethylamino)phenyl]-2-furancarboxamideHomo sapiens (human)Potency1.584910
1-[1-(4-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-(4-methyl-1-piperidinyl)ethanoneHomo sapiens (human)Potency2.238710
te 5Homo sapiens (human)Potency2.238710
4-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamideHomo sapiens (human)Potency3.548110
5-hydroxy-2-methyl-3-benzo[g]benzofurancarboxylic acid ethyl esterHomo sapiens (human)Potency5.623410
2-(cyclohexylamino)-N-(4-ethylphenyl)-2-sulfanylideneacetamideHomo sapiens (human)Potency0.794310
4-methyl-N-[4-(4-morpholinyl)phenyl]benzamideHomo sapiens (human)Potency2.818410
2-[[anilino(oxo)methyl]amino]-4,5-dimethyl-3-thiophenecarboxamideHomo sapiens (human)Potency5.623410
3-[[2-benzofuranyl(oxo)methyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency1.000010
N-(4-fluorophenyl)-2,1,3-benzothiadiazole-5-carboxamideHomo sapiens (human)Potency3.548110
2-(4-bromophenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency3.548110
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-benzothiazol-2-amineHomo sapiens (human)Potency3.981110
5-(1,3-benzodioxol-5-yl)-2-[(2-chloro-6-fluorophenyl)methyl]tetrazoleHomo sapiens (human)Potency3.981110
6-methoxy-2-(4-methoxyphenyl)-1-benzopyran-4-oneHomo sapiens (human)Potency0.501210
2-methoxy-N-(2-pyridinyl)benzamideHomo sapiens (human)Potency2.511910
2-(2-furanyl)-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency1.995310
2-chloro-N-(2-phenylethyl)benzamideHomo sapiens (human)Potency0.354810
N-[2-(1-cyclohexenyl)ethyl]-4-fluorobenzamideHomo sapiens (human)Potency0.398110
4-phenyl-N-(3-pyridinyl)-2-thiazolamineHomo sapiens (human)Potency3.548110
4-thiomorpholinecarbodithioic acid [2-(4-chlorophenyl)-2-oxoethyl] esterHomo sapiens (human)Potency3.162310
2-(4-ethylphenoxy)-N-(1H-1,2,4-triazol-5-yl)acetamideHomo sapiens (human)Potency3.162310
2-[(4-chloro-2-methylphenoxy)methyl]imidazo[1,2-a]pyrimidineHomo sapiens (human)Potency3.548110
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethyl-3-furamideHomo sapiens (human)Potency5.623410
4-chloro-1-methyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency3.548110
1-[4-[(2-methyl-4-quinolinyl)amino]phenyl]ethanoneHomo sapiens (human)Potency3.162310
N1-(6-bromo-4-quinazolinyl)-N4,N4-dimethylbenzene-1,4-diamineHomo sapiens (human)Potency2.818410
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterHomo sapiens (human)Potency2.818410
1-(1,3-benzodioxol-5-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterHomo sapiens (human)Potency3.162310
5-[2-[(4-chlorophenyl)thio]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid methyl esterHomo sapiens (human)Potency3.981110
2-(3,4-dichlorophenyl)imidazo[1,2-a]pyrimidineHomo sapiens (human)Potency3.162310
N-cyclohexyl-2,3-dihydroindole-1-carboxamideHomo sapiens (human)Potency2.818410
N-(7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)benzamideHomo sapiens (human)Potency2.818410
N-[(3-nitroanilino)-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency2.511910
N-tert-butyl-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency0.354810
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(4-oxo-3-quinazolinyl)acetamideHomo sapiens (human)Potency2.238710
6-(chloromethyl)-N2-(2,5-dimethoxyphenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency3.981110
2-methoxy-6-[[(1-methyl-2-benzimidazolyl)amino]methyl]phenolHomo sapiens (human)Potency1.000010
4-fluorophenyl-L-alanineHomo sapiens (human)Potency16.360110
5-(2,3-dihydro-1H-inden-5-yloxymethyl)-2-furancarbohydrazideHomo sapiens (human)Potency1.000010
5-[(4-ethylphenoxy)methyl]-N-(2-pyridinylmethyl)-2-furancarboxamideHomo sapiens (human)Potency1.995310
N-(5-methyl-3-isoxazolyl)-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency2.511910
phenylthiazolylthioureaHomo sapiens (human)Potency2.285810
vu0038882Homo sapiens (human)Potency3.162310
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-methoxybenzamideHomo sapiens (human)Potency3.162310
2-[(3-methyl-2-thiophenyl)methylidene]indene-1,3-dioneHomo sapiens (human)Potency3.548110
4-(1H-benzimidazol-2-yl)quinolineHomo sapiens (human)Potency4.466810
2-anilino-N-(4-fluorophenyl)acetamideHomo sapiens (human)Potency3.981110
4-[[2-furanyl(oxo)methyl]amino]benzoic acid propan-2-yl esterHomo sapiens (human)Potency2.511910
N-(2,5-dimethylphenyl)-2-benzofurancarboxamideHomo sapiens (human)Potency3.162310
N-(4-methoxyphenyl)-2-benzofurancarboxamideHomo sapiens (human)Potency1.584910
1-(1,3-benzothiazol-2-yl)-3-phenylureaHomo sapiens (human)Potency2.818410
4-hydroxy-1-(4-methylphenyl)-3-pyrazolecarboxylic acid ethyl esterHomo sapiens (human)Potency4.466810
1-(4-fluorophenyl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterHomo sapiens (human)Potency5.623410
N-[4-(diethylamino)phenyl]-N'-phenylureaHomo sapiens (human)Potency0.891310
4-bromo-N-phenacylbenzamideHomo sapiens (human)Potency2.818410
4-bromo-2-phenyl-5-(1-piperidinyl)-3-pyridazinoneHomo sapiens (human)Potency3.548110
N-(5-acetyl-4-methyl-2-thiazolyl)-4-tert-butylbenzamideHomo sapiens (human)Potency1.584910
N-[4-(3,4-dimethylphenyl)-2-thiazolyl]-2-furancarboxamideHomo sapiens (human)Potency2.238710
1-[4-[(4,6-dimethyl-2-pyrimidinyl)amino]phenyl]ethanoneHomo sapiens (human)Potency3.162310
N-[4-(4-ethylphenyl)-2-thiazolyl]carbamic acid phenyl esterHomo sapiens (human)Potency2.818410
2-phenylmethoxy-1-naphthalenecarboxaldehydeHomo sapiens (human)Potency3.162310
1-benzoyl-4-phenyl-3-thiosemicarbazideHomo sapiens (human)Potency3.162310
1-(2,3-dihydroindol-1-yl)-2-(phenylthio)ethanoneHomo sapiens (human)Potency3.548110
5,7-dimethyl-2-phenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency3.981110
N-[6-methyl-2-(4-methylphenyl)-5-benzotriazolyl]-3-pyridinecarboxamideHomo sapiens (human)Potency3.548110
N-[[(5-chloro-2-pyridinyl)amino]-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency5.623410
N-[[(6-methyl-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency3.548110
N-(3,4,5,6-tetrahydro-2H-azepin-7-yl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amineHomo sapiens (human)Potency3.162310
2-(2-bromo-4-methylphenoxy)-N-(2-pyridinylmethyl)acetamideHomo sapiens (human)Potency4.466810
1-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-3-(4-chlorophenyl)ureaHomo sapiens (human)Potency2.511910
1-(4-methoxyphenyl)-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ureaHomo sapiens (human)Potency3.981110
5-amino-1-(2-pyridinyl)-4-pyrazolecarboxylic acid ethyl esterHomo sapiens (human)Potency3.981110
1-cyclohexyl-3-(2-phenylethyl)ureaHomo sapiens (human)Potency1.122010
3-(2,4-dioxo-6-methyl-5-pyrimidinyl)acrylic acidHomo sapiens (human)Potency1.258910
acetic acid [4-[oxo-(2-phenylethylamino)methyl]phenyl] esterHomo sapiens (human)Potency0.398110
N-phenethyl-2-furamideHomo sapiens (human)Potency3.162310
8-(1H-indol-3-ylmethylidene)-6,10-dioxaspiro[4.5]decane-7,9-dioneHomo sapiens (human)Potency1.122010
4-[2-(1-methyl-2-benzimidazolyl)ethyl]anilineHomo sapiens (human)Potency3.162310
acetic acid (4-oxo-3-phenyl-1-benzopyran-7-yl) esterHomo sapiens (human)Potency5.623410
4-amino-2-(phenacylthio)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency3.162310
2-[[(4-chlorophenyl)thio]methyl]imidazo[1,2-a]pyridineHomo sapiens (human)Potency3.548110
N-(4-methoxyphenyl)carbamic acid (9-fluorenylideneamino) esterHomo sapiens (human)Potency3.548110
N-cyclopentyl-2-benzo[e]benzofurancarboxamideHomo sapiens (human)Potency1.412510
nsc185058Homo sapiens (human)Potency2.201610
2-[(2-fluorophenyl)methylthio]-5-(4-methylphenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency0.794310
2-[(4-fluorophenyl)methylthio]-5-(2-methylphenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency2.818410
2-[(2-methoxyphenoxy)methyl]-1H-benzimidazoleHomo sapiens (human)Potency2.511910
2-(4-fluorophenyl)-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidineHomo sapiens (human)Potency3.981110
N-(3,4-dimethoxyphenyl)-4-methoxybenzamideHomo sapiens (human)Potency3.981110
2-fluoro-N-phenacylbenzamideHomo sapiens (human)Potency0.446710
N-(4-ethylphenyl)-4-oxo-3H-phthalazine-1-carboxamideHomo sapiens (human)Potency3.162310
2-(4-chlorophenyl)-5-(4-fluorophenyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency1.995310
5-nitro-2-phenyl-1,3-benzoxazoleHomo sapiens (human)Potency2.238710
N-[2-(4-methoxyphenyl)-5-benzotriazolyl]butanamideHomo sapiens (human)Potency0.562310
5,7-dimethyl-2-(4-methylphenyl)pyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency3.548110
N-[1-(4-methylphenyl)-5-benzimidazolyl]acetamideHomo sapiens (human)Potency1.122010
3-(4-methylphenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneHomo sapiens (human)Potency2.511910
2-(2-phenylethyl)-1,3-benzoxazol-5-amineHomo sapiens (human)Potency2.511910
3-(8-methyl-2-imidazo[1,2-a]pyridinyl)-1-benzopyran-2-oneHomo sapiens (human)Potency0.112210
4-[(1H-benzimidazol-2-ylthio)methyl]-2-thiazolamineHomo sapiens (human)Potency2.511910
5-bromo-N-(2,4-dichlorophenyl)-2-furancarboxamideHomo sapiens (human)Potency2.238710
N-[3-chloro-4-(1-pyrrolidinyl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency1.412510
1-(4,5-dihydrothiazol-2-yl)-3-phenylureaHomo sapiens (human)Potency1.412510
N-(4-methoxyphenyl)-3,4-dihydroquinolin-2-amineHomo sapiens (human)Potency2.818410
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazineHomo sapiens (human)Potency3.162310
4-chloro-N-(4-methyl-2-thiazolyl)-2-nitrobenzamideHomo sapiens (human)Potency2.511910
2-(phenylmethylthio)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoleHomo sapiens (human)Potency0.316210
5-methyl-N-(4,5,6-trimethyl-2-pyrimidinyl)-1,3-benzoxazol-2-amineHomo sapiens (human)Potency1.584910
4-acetamido-N-(2-phenylethyl)benzamideHomo sapiens (human)Potency3.548110
1-(4-methoxyphenyl)-3-(6-methyl-2-pyridinyl)ureaHomo sapiens (human)Potency3.548110
[5-(4-nitrophenyl)-2-furanyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency3.981110
3-ethoxy-N-(2-thiazolyl)benzamideHomo sapiens (human)Potency5.011910
2-bromo-N-(3-methoxyphenyl)benzamideHomo sapiens (human)Potency3.981110
2,4-dimethoxy-n-naphthalen-2-yl-benzamideHomo sapiens (human)Potency3.548110
N-[[(4,6-dimethyl-2-pyrimidinyl)amino]-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency3.162310
3-[[(2,5-dimethyl-3-furanyl)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency3.548110
N-(1,3-benzodioxol-5-ylmethyl)-1H-benzimidazol-2-amineHomo sapiens (human)Potency3.162310
1,3-bis(2-phenylethyl)thioureaHomo sapiens (human)Potency4.466810
5-ethyl-3-[[4-(2-methylpropoxy)phenyl]methylthio]-1H-1,2,4-triazoleHomo sapiens (human)Potency3.162310
4-chloro-1-ethyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency3.548110
[4-[(2-fluorophenyl)methoxy]phenyl]-(1-pyrrolidinyl)methanethioneHomo sapiens (human)Potency1.778310
1-ethyl-2-[(4-methylphenoxy)methyl]benzimidazoleHomo sapiens (human)Potency2.818410
4-methyl-N-(3-nitrophenyl)-5-phenyl-3-thiophenecarboxamideHomo sapiens (human)Potency0.707910
9-oxo-3-fluorenecarboxylic acid (phenylmethyl) esterHomo sapiens (human)Potency3.162310
5-bromo-N-(4-propan-2-ylphenyl)-2-furancarboxamideHomo sapiens (human)Potency0.891310
N-(2,4-difluorophenyl)-3-methoxybenzamideHomo sapiens (human)Potency3.548110
N-[2-(2-methylpropyl)-1,3-dioxo-5-isoindolyl]-2-furancarboxamideHomo sapiens (human)Potency3.981110
2-(2-furanyl)-6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-b][1,3]oxazin-4-oneHomo sapiens (human)Potency3.162310
N-(1,3-benzothiazol-2-yl)-2-cyclohexylacetamideHomo sapiens (human)Potency1.778310
5-bromo-N-[(2-pyridinylamino)-sulfanylidenemethyl]-3-pyridinecarboxamideHomo sapiens (human)Potency1.778310
5-(3-chloro-4-methylphenyl)-3-pyridin-4-yl-1,2,4-oxadiazoleHomo sapiens (human)Potency1.995310
5-(phenylmethyl)-3-(2-pyridinyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency2.238710
N-(4-fluorophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxamideHomo sapiens (human)Potency3.981110
N-(4-hydroxyphenyl)-3-methoxy-2-naphthalenecarboxamideHomo sapiens (human)Potency1.412510
6-(1,3-benzoxazol-2-yl)-1,3-benzothiazol-2-amineHomo sapiens (human)Potency1.122010
7,8-dimethoxy-5-methyl-3-phenylpyrazolo[3,4-c]isoquinolineHomo sapiens (human)Potency3.548110
N-(4-methylphenyl)carbamic acid (cyclopentylideneamino) esterHomo sapiens (human)Potency3.981110
N-(cyclopentylideneamino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamideHomo sapiens (human)Potency2.511910
6-(4-chlorophenyl)-2-methyl-3-pyridinecarboxylic acid methyl esterHomo sapiens (human)Potency1.584910
2-methyl-N-(2-naphthalenyl)-3-furancarboxamideHomo sapiens (human)Potency1.412510
N-[[(5-chloro-2-pyridinyl)amino]-sulfanylidenemethyl]-3-methylbutanamideHomo sapiens (human)Potency2.818410
N-[[(6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-4-phenylbenzamideHomo sapiens (human)Potency2.818410
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency0.631010
1-(2-naphthalenyl)hexane-1,4-dioneHomo sapiens (human)Potency3.548110
2-[[(3-methylphenyl)-oxomethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acidHomo sapiens (human)Potency2.511910
N-(2-furanylmethyl)-1-(4-methoxyphenyl)-5-benzimidazolamineHomo sapiens (human)Potency2.818410
N-(1-propyl-5-benzimidazolyl)-2-thiophenecarboxamideHomo sapiens (human)Potency3.548110
N-(1-tert-butyl-5-benzimidazolyl)-2-thiophenecarboxamideHomo sapiens (human)Potency2.511910
5-[anilino(oxo)methyl]-4-methyl-2-(1-oxopropylamino)-3-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency0.794310
4-methyl-N,5-diphenyl-3-thiophenecarboxamideHomo sapiens (human)Potency1.122010
N-(2-pyridinyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency3.162310
5-[(2-chlorophenoxy)methyl]-3-pyridin-4-yl-1,2,4-oxadiazoleHomo sapiens (human)Potency2.818410
2-(2,4-dichlorophenyl)-3,5-dihydro-1H-pyrazolo[3,4-d]triazol-6-amineHomo sapiens (human)Potency5.623410
2-methyl-3,7-diphenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency2.511910
N-(4-bromo-2-fluorophenyl)-2-methyl-3-furancarboxamideHomo sapiens (human)Potency4.466810
6-(1H-benzimidazol-2-yl)-2-methyl-1H-benzimidazoleHomo sapiens (human)Potency1.412510
2-chloro-4-methyl-N-[4-(4-methyl-1-piperazinyl)phenyl]benzamideHomo sapiens (human)Potency3.548110
2-[[(5-bromo-2-furanyl)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency3.548110
3-amino-5-phenyl-2-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency5.623410
N-(4-methoxyphenyl)-3-methyl-1,3-benzothiazol-2-imineHomo sapiens (human)Potency2.511910
N-[4-(4-chlorophenyl)-3,5-dimethyl-2-thiazolylidene]-2-furancarboxamideHomo sapiens (human)Potency2.511910
10,11-dihydroxy-n-allylnoraporphineHomo sapiens (human)Potency58.047910
2-(ethylthio)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency3.548110
3-[[(3-chloro-4-ethoxyphenyl)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency0.100010
N-[1-[(4-fluorophenyl)methyl]-3-pyrazolyl]-5-methyl-2-furancarboxamideHomo sapiens (human)Potency3.548110
N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-pyrazinecarboxamideHomo sapiens (human)Potency3.981110
N-(1,3-benzodioxol-5-yl)-5-methyl-2-furancarboxamideHomo sapiens (human)Potency2.818410
3-chloro-6-methyl-N-(3-pyridinyl)-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency2.818410
3,6-dichloro-N-(4-methyl-2-pyridinyl)-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency0.125910
2-methoxy-N-(4-methylphenyl)-4-(methylthio)benzamideHomo sapiens (human)Potency3.548110
1-(2-methylphenyl)-3-[[(5-methyl-3-thiophenyl)-oxomethyl]amino]thioureaHomo sapiens (human)Potency3.162310
1-(3-methylphenyl)-3-[[oxo-(5-propyl-3-thiophenyl)methyl]amino]thioureaHomo sapiens (human)Potency3.548110
1-cyclohexyl-3-(2,3-dihydro-1,4-benzodioxin-6-yl)ureaHomo sapiens (human)Potency0.631010
2-[(3-fluorophenyl)methylthio]pyrimidine-4,6-diamineHomo sapiens (human)Potency2.818410
4,5-dimethyl-2-[4-(3-nitrophenyl)-2-thiazolyl]-1H-pyrazol-3-oneHomo sapiens (human)Potency3.981110
2-(4-fluoro-N-methylsulfonylanilino)-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency3.162310
N-(1-acetyl-2,3-dihydroindol-5-yl)-4-methylbenzamideHomo sapiens (human)Potency0.794310
2-[(1-ethyl-2,5-dimethyl-3-pyrrolyl)methylidene]indene-1,3-dioneHomo sapiens (human)Potency3.548110
1-(4-methoxyphenyl)-3-[[oxo(thiophen-2-yl)methyl]amino]thioureaHomo sapiens (human)Potency49.916910
N-(6-ethoxy-1,3-benzothiazol-2-yl)butanamideHomo sapiens (human)Potency2.818410
4-(4-phenylmethoxyphenyl)thiadiazoleHomo sapiens (human)Potency1.778310
N2,N4-bis(4-methoxyphenyl)pyrimidine-2,4-diamineHomo sapiens (human)Potency1.995310
2-(3-methoxyphenyl)-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency4.466810
5-methyl-1-phenyl-4-pyrazolecarboxylic acid (4-methoxyphenyl) esterHomo sapiens (human)Potency3.162310
2-methoxy-3-methyl-N-[4-(4-morpholinylmethyl)phenyl]benzamideHomo sapiens (human)Potency3.162310
N-(2-phenyl-6-imidazo[1,2-a]pyridinyl)acetamideHomo sapiens (human)Potency1.000010
N,N-dimethylcarbamic acid [4-[6-(trifluoromethyl)-2-imidazo[1,2-a]pyridinyl]phenyl] esterHomo sapiens (human)Potency3.548110
N-(6-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-3-phenylpropanamideHomo sapiens (human)Potency3.548110
5-(4-methylphenyl)-2-phenyl-3-pyrazolamineHomo sapiens (human)Potency1.122010
2-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]thio]-1-(1-piperidinyl)ethanoneHomo sapiens (human)Potency3.981110
5-(4-fluorophenyl)-2-thiophen-2-yloxazoleHomo sapiens (human)Potency3.981110
N-(2-chlorophenyl)-2-[[cyclopropyl(oxo)methyl]amino]-4-methyl-5-thiazolecarboxamideHomo sapiens (human)Potency3.548110
5-(4-propan-2-ylphenyl)-2H-tetrazoleHomo sapiens (human)Potency6.309610
2-(4-methoxyphenyl)-5-(3-pyridinyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency3.981110
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-benzimidazolamineHomo sapiens (human)Potency2.818410
N-(4-fluorophenyl)-1-(3-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency3.162310
2-[[5-(4-ethoxyphenyl)-1,3,4-oxadiazol-2-yl]thio]-1-(4-morpholinyl)ethanoneHomo sapiens (human)Potency2.511910
1-(4-fluorophenyl)-2-(2-pyridinylthio)ethanoneHomo sapiens (human)Potency4.466810
5-(3,5-dimethoxyphenyl)-3-phenyl-1,2,4-oxadiazoleHomo sapiens (human)Potency5.623410
2-[(2-chlorophenyl)methylthio]-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoleHomo sapiens (human)Potency3.981110
N'-[(4-chlorophenyl)-oxomethyl]-2-hydroxy-3-methylbenzohydrazideHomo sapiens (human)Potency2.511910
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-4-methylbenzamideHomo sapiens (human)Potency1.122010
N-[2-(4-fluorophenyl)ethyl]-4-nitrobenzamideHomo sapiens (human)Potency2.511910
N-(2-fluorophenyl)-3-phenylpropanamideHomo sapiens (human)Potency3.548110
N-[[(6-methoxy-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency3.162310
1-(1-azepanyl)-2-(4-bromophenyl)ethanoneHomo sapiens (human)Potency3.981110
3-(4-methoxyphenyl)-5-(4-methylphenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency1.995310
4-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]benzoic acid ethyl esterHomo sapiens (human)Potency3.162310
2-chloro-4,5-difluoro-N-(5-methyl-2-pyridinyl)benzamideHomo sapiens (human)Potency1.778310
n-(2-methoxybenzyl)-2-(phenylthio)acetamideHomo sapiens (human)Potency2.511910
N-[(3-acetylanilino)-sulfanylidenemethyl]-3-chlorobenzamideHomo sapiens (human)Potency3.548110
N-(1,3-benzodioxol-5-yl)-4-(4-morpholinylmethyl)benzamideHomo sapiens (human)Potency3.981110
1-azepanyl-[4-[(phenylthio)methyl]phenyl]methanoneHomo sapiens (human)Potency3.162310
4-chloro-N-[4-(2-imidazo[1,2-a]pyridinyl)phenyl]benzamideHomo sapiens (human)Potency1.995310
4-propan-2-yl-N-(3-pyridinyl)benzamideHomo sapiens (human)Potency1.584910
3-(4-methoxyphenyl)-5-(2-phenylethyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency3.162310
2-(2-phenylethylthio)-3-pyridinecarboxylic acidHomo sapiens (human)Potency0.446710
3-[[[3-(4-methoxyphenyl)phenyl]-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency3.162310
5-(2-furanylmethylamino)-2-(4-methoxyphenyl)-4-oxazolecarbonitrileHomo sapiens (human)Potency3.162310
3-[(4-ethoxyphenoxy)methyl]-N,N-diethylbenzamideHomo sapiens (human)Potency0.251210
5-[(4-ethoxyphenoxy)methyl]-N-(3-pyridinyl)-2-furancarboxamideHomo sapiens (human)Potency0.562310
N-[4-[[acetamido(sulfanylidene)methyl]amino]phenyl]-2-thiophenecarboxamideHomo sapiens (human)Potency3.981110
N-[anilino(sulfanylidene)methyl]-5-bromo-2-furancarboxamideHomo sapiens (human)Potency3.548110
4-phenyl-N-(2-propyl-5-tetrazolyl)benzamideHomo sapiens (human)Potency2.511910
6-methoxy-4-methyl-2-[(2-methylphenyl)methylthio]quinazolineHomo sapiens (human)Potency6.309610
N-[3-[methyl(methylsulfonyl)amino]phenyl]-2-phenoxyacetamideHomo sapiens (human)Potency4.466810
4-[methyl(methylsulfonyl)amino]-N-(2-phenylethyl)benzamideHomo sapiens (human)Potency1.412510
N-(4-phenylmethoxyphenyl)carbamic acid methyl esterHomo sapiens (human)Potency3.162310
N-(5-acetyl-4-methyl-2-thiazolyl)-5-bromo-2-furancarboxamideHomo sapiens (human)Potency3.548110
4-[2-(3-methoxyphenyl)-2-oxoethoxy]benzoic acid methyl esterHomo sapiens (human)Potency1.995310
4-phenacyloxybenzoic acid methyl esterHomo sapiens (human)Potency3.162310
2-(3-acetamidophenoxy)-N-phenylacetamideHomo sapiens (human)Potency3.548110
4-[[(cyclohexylamino)-oxomethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency3.548110
4-tert-butyl-N-(4-methyl-3-nitrophenyl)benzamideHomo sapiens (human)Potency3.548110
2-(2-cyclohexylidenehydrazinyl)benzoic acidHomo sapiens (human)Potency3.981110
N2-(4-methylphenyl)-6-[(2-pyrimidinylthio)methyl]-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency2.238710
4-[[(2-methyl-1,3-benzothiazol-6-yl)-oxomethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency0.841020
N-(4-ethoxyphenyl)-1,2,5-thiadiazole-3-carboxamideHomo sapiens (human)Potency1.412510
N-(3,4-dimethyl-2-thiazolylidene)benzamideHomo sapiens (human)Potency3.162310
N-[5-(2-chlorophenyl)-1H-1,2,4-triazol-3-yl]-4,6-dimethyl-2-pyrimidinamineHomo sapiens (human)Potency4.466810
N-(3-methoxyphenyl)-4-[(2-methyl-1-oxopropyl)amino]benzamideHomo sapiens (human)Potency3.548110
3-acetamidobenzoic acid [2-(2-chlorophenyl)-2-oxoethyl] esterHomo sapiens (human)Potency3.548110
4-(1-oxopropylamino)benzoic acid (2-chlorophenyl)methyl esterHomo sapiens (human)Potency2.238710
N-(4,5-dimethyl-2-thiazolyl)cyclohexanecarboxamideHomo sapiens (human)Potency3.548110
N-(2,3-dihydro-1H-inden-5-yl)-2-methyl-3-nitrobenzamideHomo sapiens (human)Potency5.623410
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency2.511910
5-[(4-methylphenoxy)methyl]-3-phenyl-1,2,4-oxadiazoleHomo sapiens (human)Potency3.162310
3-(2-methoxy-6-methyl-3-pyridinyl)-5-(2-methoxyphenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency3.981110
7,8-dichloropyrido[1,2-a]benzimidazoleHomo sapiens (human)Potency6.309610
N'-(1,3-benzoxazol-2-yl)benzohydrazideHomo sapiens (human)Potency0.398110
1-(cycloheptylideneamino)-3-(4-fluorophenyl)thioureaHomo sapiens (human)Potency1.412510
4-methoxy-N-[[(phenylmethyl)amino]-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency5.623410
N-(4,5-dihydrothiazol-2-yl)-2-(2-methylphenoxy)acetamideHomo sapiens (human)Potency1.778310
3-amino-2-(4-methylphenyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency1.258910
3-(2-benzo[cd]indolylamino)benzoic acidHomo sapiens (human)Potency0.446710
N2-(4-fluorophenyl)-6-(3-methyl-2-benzofuranyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency2.238710
6-(chloromethyl)-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency3.162310
5-(2-furanylmethylamino)-2-(3-methylphenyl)-4-oxazolecarbonitrileHomo sapiens (human)Potency4.466810
N-cyclopropyl-3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency2.818410
4-chloro-N-(1,2-dimethyl-5-benzimidazolyl)benzamideHomo sapiens (human)Potency0.281810
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-3-methylbenzamideHomo sapiens (human)Potency0.501210
N-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency5.623410
N-(1,3-benzodioxol-5-yl)-4-(2-furanylmethyl)-1-piperazinecarbothioamideHomo sapiens (human)Potency3.162310
1-(2,4-dichlorophenyl)-3-(1-methyl-3-pyrazolyl)ureaHomo sapiens (human)Potency3.548110
4-[[1-azepanyl(oxo)methyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency1.122010
1-[[(2-methyl-3-furanyl)-oxomethyl]amino]-3-[2-(trifluoromethyl)phenyl]thioureaHomo sapiens (human)Potency2.818410
N-(1,3-benzothiazol-2-yl)-2-[(1-methyl-2-imidazolyl)thio]acetamideHomo sapiens (human)Potency2.818410
1-(3-acetylphenyl)-3-(2-pyridinylmethyl)ureaHomo sapiens (human)Potency3.548110
1-(4-acetylphenyl)-3-[2-(4-fluorophenyl)ethyl]thioureaHomo sapiens (human)Potency2.818410
N-[4-[2-[(4-methyl-2-pyridinyl)amino]-4-thiazolyl]phenyl]acetamideHomo sapiens (human)Potency1.412510
4-[2-(3-methoxyanilino)-4-thiazolyl]phenolHomo sapiens (human)Potency3.548110
4-(3,4-dimethoxyphenyl)-N-(3-methyl-2-pyridinyl)-2-thiazolamineHomo sapiens (human)Potency3.981110
3-[[(5-bromo-2-furanyl)-oxomethyl]amino]-2-methylbenzoic acidHomo sapiens (human)Potency3.981110
N-[3-[[(3,5-dimethoxyphenyl)-oxomethyl]amino]phenyl]carbamic acid ethyl esterHomo sapiens (human)Potency1.000010
(5-phenyl-3-isoxazolyl)-(1-pyrrolidinyl)methanoneHomo sapiens (human)Potency0.794310
2-(4-methylanilino)-4-pyrido[3,2-e][1,3]thiazinoneHomo sapiens (human)Potency3.162310
1-(1-naphthalenylmethoxy)benzotriazoleHomo sapiens (human)Potency3.548110
N-(2-pyridinyl)-2-[[5-(3-pyridinyl)-1,3,4-oxadiazol-2-yl]thio]acetamideHomo sapiens (human)Potency3.162310
N-(3-chloro-4-methylphenyl)-2-(2-formylphenoxy)acetamideHomo sapiens (human)Potency1.995310
N-(2-hydroxy-5-methylphenyl)-1,3-dioxo-2-propyl-5-isoindolecarboxamideHomo sapiens (human)Potency2.238710
1-phenyl-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneHomo sapiens (human)Potency3.548110
7-amino-2-(4-tert-butylphenyl)-6-pyrazolo[1,5-a]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency1.258910
N-(7-bromo-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-3-methoxybenzamideHomo sapiens (human)Potency2.818410
1-[4-(4-bromophenyl)-2-thiazolyl]-4-piperidinecarboxamideHomo sapiens (human)Potency2.958210
umi-77Homo sapiens (human)Potency6.309610
2-[[4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency0.891310
N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-(3-methyl-N-methylsulfonylanilino)acetamideHomo sapiens (human)Potency3.162310
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamideHomo sapiens (human)Potency3.548110
N-[[3-(hydroxymethyl)anilino]-sulfanylidenemethyl]-4-phenylbenzamideHomo sapiens (human)Potency1.000010
N-[(3-acetylanilino)-sulfanylidenemethyl]-5-bromo-3-pyridinecarboxamideHomo sapiens (human)Potency2.511910
5-bromo-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideHomo sapiens (human)Potency1.584910
3-[[(3,5-dichloro-4-ethoxyphenyl)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency0.562310
N-[[(5-methyl-1H-pyrazol-3-yl)amino]-oxomethyl]-3-(1,1,2,2-tetrafluoroethoxy)benzamideHomo sapiens (human)Potency2.511910
N-[[3-chloro-4-(4-morpholinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency3.162310
pyridine-2-carboxylic acid thiazol-2-ylamideHomo sapiens (human)Potency3.548110
3-[2-(4-aminoanilino)-4-thiazolyl]-1-benzopyran-2-oneHomo sapiens (human)Potency3.548110
8-[1-(3-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-1,4-dioxa-8-azaspiro[4.5]decaneHomo sapiens (human)Potency2.818410
2-[[cyclohexyl(oxo)methyl]amino]-1,3-benzothiazole-6-carboxylic acid methyl esterHomo sapiens (human)Potency0.891310
3-(4-chlorophenyl)-5-propyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneHomo sapiens (human)Potency6.309610
3-(4-methoxyphenyl)-6-phenyl-4-thieno[2,3-d]pyrimidinoneHomo sapiens (human)Potency0.562310
N-[2-(2-pyridinyl)-3H-benzimidazol-5-yl]cyclohexanecarboxamideHomo sapiens (human)Potency2.511910
N-(2-methyl-1,3-benzothiazol-6-yl)-2-furancarboxamideHomo sapiens (human)Potency3.162310
1-methyl-N-(2-naphthalenyl)-5-benzotriazolecarboxamideHomo sapiens (human)Potency0.891310
N-(1-naphthalenyl)-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineHomo sapiens (human)Potency3.162310
N-[4-[2-[(6-methyl-2-pyridinyl)amino]-4-thiazolyl]phenyl]acetamideHomo sapiens (human)Potency1.778310
N-[3-[2-[(4-methyl-2-pyridinyl)amino]-4-thiazolyl]phenyl]acetamideHomo sapiens (human)Potency2.511910
3-[2-(3-methylphenoxy)ethyl]-1,3-benzothiazol-2-oneHomo sapiens (human)Potency2.511910
3-[2-(4-methylphenoxy)ethyl]-1,3-benzothiazol-2-oneHomo sapiens (human)Potency3.548110
5-(4-methylphenyl)-N-(3-pyridinylmethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency5.623410
LSM-16285Homo sapiens (human)Potency6.309610
3-methoxy-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)benzamideHomo sapiens (human)Potency3.548110
N-[4-(1-pyrrolidinyl)phenyl]-2-naphthalenecarboxamideHomo sapiens (human)Potency1.258910
2-[(3-cyano-6-methoxy-2-quinolinyl)thio]-N-(2-methyl-1,3-benzothiazol-5-yl)acetamideHomo sapiens (human)Potency3.548110
N-[3-chloro-4-[[2-furanyl(oxo)methyl]amino]phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency3.548110
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acidHomo sapiens (human)Potency1.412510
5-[2-[(4-chlorophenyl)thio]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterHomo sapiens (human)Potency3.548110
1-[2,5-dimethyl-1-(4-methylphenyl)-3-pyrrolyl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneHomo sapiens (human)Potency0.891310
4-[[7-methoxy-4-oxo-2-(trifluoromethyl)-1-benzopyran-3-yl]oxy]benzoic acidHomo sapiens (human)Potency0.501210
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterHomo sapiens (human)Potency6.309610
2-(4-chloro-3-methylphenoxy)acetic acid [4-[(4-methylanilino)-oxomethyl]phenyl] esterHomo sapiens (human)Potency2.238710
2-(3-chlorophenoxy)acetic acid [4-[(4-methylanilino)-oxomethyl]phenyl] esterHomo sapiens (human)Potency2.818410
2-(4-chloro-2-methylphenoxy)acetic acid [4-[(4-methylanilino)-oxomethyl]phenyl] esterHomo sapiens (human)Potency3.981110
3-(1,3-dioxo-2-isoindolyl)propanoic acid [4-[(4-methylanilino)-oxomethyl]phenyl] esterHomo sapiens (human)Potency3.162310
n-(1,3-benzothiazol-2-yl)-n-(4,5-dihydro-1h-imidazol-2-yl)amineHomo sapiens (human)Potency3.981110
N-(4-chlorophenyl)carbamic acid 2-pyridinylmethyl esterHomo sapiens (human)Potency2.511910
N-(4-methylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency3.162310
3-(2-phenyl-5-tetrazolyl)pyridineHomo sapiens (human)Potency3.981110
4-chloro-1-methyl-N-[1-[(4-methylphenyl)methyl]-3-pyrazolyl]-3-pyrazolecarboxamideHomo sapiens (human)Potency3.981110
N-[(4-ethylanilino)-sulfanylidenemethyl]-3-methylbutanamideHomo sapiens (human)Potency3.548110
3-[(4-bromophenoxy)methyl]-N-(5-methyl-3-isoxazolyl)benzamideHomo sapiens (human)Potency0.354810
2-(2-bromo-4-chlorophenoxy)-N-cyclohexyl-N-methylacetamideHomo sapiens (human)Potency5.623410
3-[[(2-cyclohexyl-1,3-dioxo-5-isoindolyl)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency1.584910
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency0.955920
LSM-27108Homo sapiens (human)Potency3.162310
2-(1,2-benzoxazol-3-yl)-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency3.981110
N-[4-[(N-methylanilino)-oxomethyl]phenyl]-2-furancarboxamideHomo sapiens (human)Potency5.623410
N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency2.818410
N-(5-tert-butyl-3-isoxazolyl)-3-nitrobenzamideHomo sapiens (human)Potency2.238710
5-bromo-N-[2-(4-chlorophenyl)ethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency3.981110
3-chloro-4-fluoro-N-(3-pyridinyl)-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency3.981110
5-bromo-N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency0.501210
N-[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency3.548110
2-benzamido-4,5-dihydrobenzo[g][1]benzothiole-3-carboxamideHomo sapiens (human)Potency4.466810
N-[2-(4-fluorophenyl)ethyl]-5-methyl-2-thiophenecarboxamideHomo sapiens (human)Potency1.412510
3-[[oxo-[3-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl]methoxy]methyl]benzoic acid ethyl esterHomo sapiens (human)Potency1.995310
N-(3-hydroxyphenyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency5.011910
N-[(3-methoxyphenyl)methyl]-1-propyl-5-benzimidazolamineHomo sapiens (human)Potency3.162310
3-[[[3-(1-azepanylsulfonyl)-4-chlorophenyl]-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency0.316210
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamideHomo sapiens (human)Potency2.818410
N-[2-(5-bromo-3-pyridinyl)-1,3-benzoxazol-5-yl]butanamideHomo sapiens (human)Potency1.584910
2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(2-pyridinyl)acetamideHomo sapiens (human)Potency0.668220
[2-(4-propylphenyl)-4-quinolinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency0.354810
2-(4-propylphenyl)-N-[2-(4-sulfamoylphenyl)ethyl]-4-quinolinecarboxamideHomo sapiens (human)Potency2.511910
2-(3-bromophenyl)-6-methyl-N-(1,2,4-triazol-4-yl)-4-quinolinecarboxamideHomo sapiens (human)Potency5.623410
N-(4-methyl-2-thiazolyl)-2-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]acetamideHomo sapiens (human)Potency15.785110
7-(2-oxopropoxy)-3-phenyl-1-benzopyran-2-oneHomo sapiens (human)Potency1.122010
5-(4-ethylbenzylidene)-2-thioxothiazolidin-4-oneHomo sapiens (human)Potency10.322510
2-[[2-[(4-chlorophenyl)thio]-1-oxoethyl]amino]-N-(4-methoxyphenyl)benzamideHomo sapiens (human)Potency3.981110
4-methoxy-N-[2-[(4-nitrophenyl)methylthio]-4-oxo-3-quinazolinyl]benzamideHomo sapiens (human)Potency2.511910
4-morpholinecarbodithioic acid [4-amino-6-(4-methylanilino)-1,3,5-triazin-2-yl]methyl esterHomo sapiens (human)Potency2.818410
2-bromo-N-[4-(4-methyl-1-piperazinyl)phenyl]benzamideHomo sapiens (human)Potency3.162310
2-(4-bromophenoxy)-N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideHomo sapiens (human)Potency3.981110
vu0405601Homo sapiens (human)Potency5.623410
4-(5-amino-4-phenyl-1-pyrazolyl)benzoic acidHomo sapiens (human)Potency0.446710
5-bromo-N-[[(3-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideHomo sapiens (human)Potency3.981110
1-(1-azepanyl)-2-(2-bromo-4-propan-2-ylphenoxy)ethanoneHomo sapiens (human)Potency3.162310
4-[[diethylamino(oxo)methyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency3.162310
N-[3-(2-chlorophenyl)-4-oxo-2-thiazolidinylidene]benzamideHomo sapiens (human)Potency2.818410
3-methyl-1,5-dithiophen-2-ylpentane-1,5-dioneHomo sapiens (human)Potency2.818410
5-[(3-aminoanilino)-oxomethyl]-4-methyl-2-(1-oxobutylamino)-3-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency3.162310
2-bromo-N'-[(3-chlorophenyl)-oxomethyl]benzohydrazideHomo sapiens (human)Potency5.623410
3-(3,4-dimethoxyphenyl)-7-(2-oxopropoxy)-1-benzopyran-2-oneHomo sapiens (human)Potency3.981110
N-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]carbamic acid methyl esterHomo sapiens (human)Potency3.548110
1-(2-fluorophenyl)-3-[5-(2-fluorophenyl)-1,3,4-thiadiazol-2-yl]ureaHomo sapiens (human)Potency2.511910
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzothiazoleHomo sapiens (human)Potency3.162310
N-(4-methylphenyl)-4-benzofuro[3,2-d]pyrimidinamineHomo sapiens (human)Potency2.511910
N-(6-chloro-1,3-benzothiazol-2-yl)-2-diphenylphosphorylacetamideHomo sapiens (human)Potency1.258910
N-(1,3-benzodioxol-5-yl)-4-methyl-1-phthalazinamineHomo sapiens (human)Potency3.548110
2-[[5-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-ethyl-1,3,4-thiadiazol-2-yl)acetamideHomo sapiens (human)Potency2.818410
6-[[2-(4-morpholinyl)-2-oxoethyl]thio]-[1,3]dioxolo[4,5-g]quinoline-7-carbonitrileHomo sapiens (human)Potency1.258910
N-[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]-2-methoxyacetamideHomo sapiens (human)Potency1.122010
N-[6-[[cyclohexyl(oxo)methyl]amino]-3-pyridinyl]-2-pyridinecarboxamideHomo sapiens (human)Potency3.162310
N-[5-[(2,2-dimethyl-1-oxopropyl)amino]-2-pyridinyl]-2-furancarboxamideHomo sapiens (human)Potency1.778310
N-[4-(1-methylsulfonyl-2,3-dihydroindol-5-yl)-2-thiazolyl]acetamideHomo sapiens (human)Potency3.548110
N-(2,3-dihydro-1H-inden-5-yl)-5-methyl-2-pyrazinecarboxamideHomo sapiens (human)Potency1.000010
5-(6-chloro-3-pyridinyl)-3-(3-methoxyphenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency3.548110
2-[(4-fluorophenyl)sulfonyl-(2-pyridinyl)amino]-N-phenylacetamideHomo sapiens (human)Potency5.623410
5-[1-(benzenesulfonyl)-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency2.238710
5-[1-[(4-methylphenyl)methyl]-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency2.818410
5-[1-(4-fluorophenyl)sulfonyl-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency5.623410
5-[1-[(4-fluorophenyl)methyl]-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency3.981110
4-(4-chlorophenyl)-1-(6-fluoro-2-pyridinyl)-3-pyrazolamineHomo sapiens (human)Potency2.511910
3-phenyl-5-[(phenylthio)methyl]isoxazoleHomo sapiens (human)Potency3.548110
3-(4-chlorophenyl)-5-[(phenylthio)methyl]isoxazoleHomo sapiens (human)Potency4.466810
4-chloro-5-(dimethylamino)-2-(4-methylphenyl)-3-pyridazinoneHomo sapiens (human)Potency0.398110
3-phenyl-2H-1,4-benzoxazineHomo sapiens (human)Potency5.623410
2-(4-methylsulfonylphenyl)-6-imidazo[1,2-a]pyridinecarboxylic acid methyl esterHomo sapiens (human)Potency4.466810
4-(2-quinoxalinylamino)benzoic acid ethyl esterHomo sapiens (human)Potency2.238710
4-[4-(2,4-dichlorophenyl)-2-thiazolyl]benzoic acidHomo sapiens (human)Potency1.584910
N,N-dimethylcarbamothioic acid O-[4-[2-[(4-chlorophenyl)thio]-1-oxoethyl]-2,6-dimethylphenyl] esterHomo sapiens (human)Potency2.818410
2-(2,4-dichlorophenyl)-5-[2-(methylthio)phenyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency3.162310
r-7050Homo sapiens (human)Potency6.309610
N,N-dimethylcarbamic acid [4-[2-(benzenesulfonyl)-1-oxoethyl]-2,6-dimethylphenyl] esterHomo sapiens (human)Potency3.162310
3-chloro-N-(2-methyl-3-oxo-1,2,4-thiadiazol-5-yl)benzamideHomo sapiens (human)Potency3.548110
2-(6-chloro-3-pyridinyl)-1H-benzimidazoleHomo sapiens (human)Potency5.623410
N,N-dimethylcarbamic acid [4-[2-(4-fluorophenyl)sulfonyl-1-oxoethyl]-2,6-dimethylphenyl] esterHomo sapiens (human)Potency3.981110
1-(6-methyl-2-pyridinyl)-N-(3-pyridinyl)-4-imidazolecarboxamideHomo sapiens (human)Potency2.818410
6-methyl-5-[2-(2-methylphenoxy)ethyl]-2-sulfanylidene-1H-pyrimidin-4-oneHomo sapiens (human)Potency0.707910
3,4-dichloro-N-(2-thiophen-2-ylethyl)benzamideHomo sapiens (human)Potency3.162310
N2,N2-dimethyl-6-[[[1-(1-naphthalenyl)-5-tetrazolyl]thio]methyl]-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency3.981110
LSM-19448Homo sapiens (human)Potency3.162310
3-(4-phenylphenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepineHomo sapiens (human)Potency3.981110
fluoxetineHomo sapiens (human)Potency58.047910
epalrestatHomo sapiens (human)Potency3.548110
N-[4-(4-morpholinyl)phenyl]carbamic acid butyl esterHomo sapiens (human)Potency2.818410
4-(4-chlorophenoxy)-1-(1-piperidinyl)-1-butanoneHomo sapiens (human)Potency25.017710
N-[(phenacylamino)-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency4.466810
2-chloro-N-heptyl-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency6.309610
4-(5-formyl-2-furanyl)benzoic acid propyl esterHomo sapiens (human)Potency0.316210
fm19g11Homo sapiens (human)Potency0.398110
N-cyano-N'-(2-fluorophenyl)carbamimidothioic acid [2-(tert-butylamino)-2-oxoethyl] esterHomo sapiens (human)Potency3.981110
3-(1H-benzimidazol-2-yl)-N-(3-pyridinylmethyl)anilineHomo sapiens (human)Potency2.818410
3-amino-N-(2-fluorophenyl)-6-(2-furanyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency2.511910
cuspin-1Homo sapiens (human)Potency39.650410
2-(4-bromophenyl)-1-(2,4-dihydroxyphenyl)ethanoneHomo sapiens (human)Potency3.162310
N-[(2-methoxyanilino)-oxomethyl]benzamideHomo sapiens (human)Potency2.511910
N-[4-[[2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]thio]phenyl]acetamideHomo sapiens (human)Potency1.584910
1-(2,4-dimethylphenyl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneHomo sapiens (human)Potency1.995310
4-methoxy-N-(3-methyl-2-thiazolylidene)benzamideHomo sapiens (human)Potency3.981110
3-[(2-chloro-4-fluorophenoxy)methyl]-1,2,3-benzotriazin-4-oneHomo sapiens (human)Potency3.162310
N-(3-cyano-2-thiophenyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]acetamideHomo sapiens (human)Potency2.818410
2-(2-bromophenyl)-5-[(2-chlorophenoxy)methyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency3.548110
4-[4-(phenylmethyl)-1-piperidinyl]thieno[2,3-d]pyrimidineHomo sapiens (human)Potency2.818410
3-(4-methoxyphenyl)-1-phenyl-4-pyrazolamineHomo sapiens (human)Potency3.548110
3-methoxy-N-(2,3,4-trifluorophenyl)benzamideHomo sapiens (human)Potency3.981110
2-ethoxy-3-pyridinecarboxylic acid [2-[1-(2-furanylmethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)Potency0.354810
N-phenyl-5-(propan-2-ylthio)-1,3,4-thiadiazol-2-amineHomo sapiens (human)Potency3.981110
2-(1H-benzimidazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneHomo sapiens (human)Potency0.125910
[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-(2-ethoxy-3-pyridinyl)methanoneHomo sapiens (human)Potency0.501210
2-phenylacetic acid [2-[4-[(4-ethoxyanilino)-oxomethyl]anilino]-2-oxoethyl] esterHomo sapiens (human)Potency2.511910
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-quinolinecarboxamideHomo sapiens (human)Potency2.511910
N-(3,4-dihydro-2H-pyrrol-5-yl)-5-phenyl-1,3,4-oxadiazol-2-amineHomo sapiens (human)Potency0.501210
N-(3,4-dihydro-2H-pyrrol-5-yl)-5-(2-furanyl)-1,3,4-oxadiazol-2-amineHomo sapiens (human)Potency3.548110
5-(4-ethoxyphenyl)-N-(3,4,5,6-tetrahydro-2H-azepin-7-yl)-1,3,4-oxadiazol-2-amineHomo sapiens (human)Potency0.501210
2-(4-formylphenoxy)acetic acid [2-(4-methylanilino)-4-thiazolyl]methyl esterHomo sapiens (human)Potency2.511910
1-(1,3-benzothiazol-2-yl)-3-propylureaHomo sapiens (human)Potency2.238710
5-bromo-N-(6-sulfamoyl-1,3-benzothiazol-2-yl)-2-furancarboxamideHomo sapiens (human)Potency3.548110
3-cyclohexyl-N-(1,3-dimethyl-2,6-dioxo-4-pyrimidinyl)propanamideHomo sapiens (human)Potency3.981110
N-(4-fluoro-3-methyl-1,3-benzothiazol-2-ylidene)-2-nitrobenzamideHomo sapiens (human)Potency0.562310
N-[2-(methylthio)-1,3-benzothiazol-6-yl]-2-furancarboxamideHomo sapiens (human)Potency2.818410
2-(1H-indol-3-yl)-2-oxo-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency3.548110
2-[2-(1-naphthalenyloxy)ethylthio]pyrimidineHomo sapiens (human)Potency2.511910
2-[2-(4-chlorophenoxy)ethylthio]pyrimidineHomo sapiens (human)Potency2.511910
1-cyclohexyl-3-(6-ethoxy-1,3-benzothiazol-2-yl)ureaHomo sapiens (human)Potency1.778310
5-bromo-N-[[(4-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideHomo sapiens (human)Potency6.309610
N-[5-(3-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamideHomo sapiens (human)Potency3.548110
N-[2-(1-naphthalenyl)-1,3-benzoxazol-5-yl]-1H-1,2,4-triazole-5-carboxamideHomo sapiens (human)Potency2.818410
1-(4-bromo-2-chlorophenyl)-3-(3-methyl-2-pyridinyl)thioureaHomo sapiens (human)Potency3.162310
N-[5-(2-methoxyethylthio)-1,3,4-thiadiazol-2-yl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency5.623410
2-butoxy-7-hydroxy-9-fluorenoneHomo sapiens (human)Potency3.548110
N-(4-chlorophenyl)-4-methyl-2-thiazolamineHomo sapiens (human)Potency3.981110
2,3-dimethyl-6-quinoxalinecarboxylic acid (2-bromophenyl)methyl esterHomo sapiens (human)Potency3.162310
1-[oxo-(2-oxo-1-benzopyran-3-yl)methyl]-4-piperidinecarboxylic acid methyl esterHomo sapiens (human)Potency3.981110
N-(3-acetylphenyl)-5,7-dimethyl-2-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency1.584910
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneHomo sapiens (human)Potency1.122010
4-chloro-N-[(2-methylpropylamino)-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency5.623410
2-[[[5-(3-chlorophenyl)-2-furanyl]-oxomethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency5.623410
N-(3-acetylphenyl)-2-naphthalenecarboxamideHomo sapiens (human)Potency3.162310
4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-[4-(1-piperidinylsulfonyl)phenyl]benzamideHomo sapiens (human)Potency0.562310
1-[2-(2-chlorophenoxy)ethoxy]-2-methoxy-4-methylbenzeneHomo sapiens (human)Potency5.623410
5-bromo-N-(4-methoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency3.162310
N-(1H-benzimidazol-2-yl)-4-(dimethylsulfamoyl)benzamideHomo sapiens (human)Potency4.466810
2-bromo-N-(4-ethylphenyl)benzamideHomo sapiens (human)Potency1.412510
2-(1,3-benzothiazol-2-yl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamineHomo sapiens (human)Potency3.162310
2-(4,6-dimethyl-2-pyrimidinyl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamineHomo sapiens (human)Potency2.511910
7-methyl-3-(phenylhydrazo)-1,5-benzodiazepin-2-oneHomo sapiens (human)Potency3.981110
3-methyl-N,1-diphenyl-4-pyrazolecarbothioamideHomo sapiens (human)Potency5.623410
1-(2-chlorophenyl)-3-[[(1-ethyl-2-methyl-5-benzimidazolyl)-oxomethyl]amino]thioureaHomo sapiens (human)Potency3.162310
6-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]-2-[3-(trifluoromethyl)phenyl]benzo[de]isoquinoline-1,3-dioneHomo sapiens (human)Potency3.548110
5,6,7,8-tetrafluoro-2-(2,3,4,5,6-pentafluorophenyl)-4h-1-benzopyran-4-oneHomo sapiens (human)Potency3.548110
1-(2-chlorophenyl)-2-(3,5-dimethyl-4-nitro-1-pyrazolyl)ethanoneHomo sapiens (human)Potency3.548110
1-(5-isoquinolinyl)-3-(2-phenylethyl)thioureaHomo sapiens (human)Potency2.818410
N-(3,5-dichloro-2-pyridinyl)-2-methoxy-4-(methylthio)benzamideHomo sapiens (human)Potency3.981110
4-(diethylsulfamoyl)benzoic acid [2-[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]-2-oxoethyl] esterHomo sapiens (human)Potency0.398110
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(3,5-dimethyl-1-pyrazolyl)benzamideHomo sapiens (human)Potency3.548110
4-(dimethylamino)benzoic acid [2-(2-methoxyphenyl)-2-oxoethyl] esterHomo sapiens (human)Potency3.162310
4-methylbenzoic acid [2-(1H-indol-3-yl)-2-oxoethyl] esterHomo sapiens (human)Potency2.511910
3-oxo-2,4-dihydroquinoxaline-1-carboxylic acid (phenylmethyl) esterHomo sapiens (human)Potency5.623410
2,5-dimethyl-3-furancarboxylic acid [2-(2,3-dihydroindol-1-yl)-2-oxoethyl] esterHomo sapiens (human)Potency3.981110
2-[(1-oxido-2-pyridin-1-iumyl)thio]-1-(4-phenylphenyl)ethanoneHomo sapiens (human)Potency3.548110
n-benzyl-n,1-dimethyl-2-propynylamineHomo sapiens (human)Potency3.981110
5-methyl-N-(4-propan-2-ylphenyl)-2-pyrazinecarboxamideHomo sapiens (human)Potency3.548110
5-(4-propylphenyl)-1H-pyrazol-3-amineHomo sapiens (human)Potency4.466810
2-(1H-benzimidazol-2-yl)-1-(3-nitrophenyl)ethanoneHomo sapiens (human)Potency3.162310
4-methoxy-N-[1-methyl-2-oxo-6-(trifluoromethyl)-3-pyridinyl]benzamideHomo sapiens (human)Potency2.818410
2-(4-methoxyphenyl)-5-(2-methylpropylthio)-1,3,4-oxadiazoleHomo sapiens (human)Potency1.000010
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideHomo sapiens (human)Potency6.309610
N-(2-phenylethyl)-1,3-benzothiazol-2-amineHomo sapiens (human)Potency3.981110
thiocyanic acid [4-[(2-chloro-1-oxoethyl)amino]-3,5-dimethylphenyl] esterHomo sapiens (human)Potency5.623410
2-(phenylmethyl)benzoic acid [2-[4-(difluoromethylthio)anilino]-2-oxoethyl] esterHomo sapiens (human)Potency5.623410
N-[4-(1-piperidinyl)phenyl]-2-quinolinecarboxamideHomo sapiens (human)Potency5.623410
2-chloro-N-[3-[(2-chlorophenyl)methyl]-2-thiazolylidene]acetamideHomo sapiens (human)Potency1.258910
3-[(4-chlorophenyl)thio]-1-[4-(4-hydroxyphenyl)-1-piperazinyl]-1-propanoneHomo sapiens (human)Potency3.548110
5-bromo-2-furancarboxylic acid [2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)Potency3.162310
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-quinolinecarboxamideHomo sapiens (human)Potency5.623410
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)Potency3.548110
N-(4,5,6-trifluoro-1,3-benzothiazol-2-yl)-2-furancarboxamideHomo sapiens (human)Potency2.238710
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideHomo sapiens (human)Potency5.623410
N-(4-tert-butyl-2-thiazolyl)-5-methyl-2-thiophenecarboxamideHomo sapiens (human)Potency2.511910
N-(1H-indazol-6-yl)-2,4-dimethoxybenzamideHomo sapiens (human)Potency5.011910
2-[2-(difluoromethoxy)anilino]-1-(2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency3.162310
2-[[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]thio]-1-(1H-pyrrol-2-yl)ethanoneHomo sapiens (human)Potency3.162310
2-hydroxy-4-methoxybenzoic acid (2-methyl-4-thiazolyl)methyl esterHomo sapiens (human)Potency3.548110
4-[[5-(1,3-benzothiazol-2-yl)-2-thiophenyl]-oxomethyl]-1-piperazinecarboxaldehydeHomo sapiens (human)Potency1.778310
5-bromo-N-(4-methyl-2-thiazolyl)-3-pyridinecarboxamideHomo sapiens (human)Potency2.818410
N-(4-tert-butyl-2-thiazolyl)-6-quinoxalinecarboxamideHomo sapiens (human)Potency2.511910
3,5-dimethyl-1H-pyrrole-2,4-dicarboxylic acid O4-ethyl ester O2-[(2-fluorophenyl)methyl] esterHomo sapiens (human)Potency1.584910
4-methyl-N-[4-(2-methyl-4-thiazolyl)phenyl]benzamideHomo sapiens (human)Potency2.238710
N-tert-butyl-2-[[4-(4-fluorophenyl)-2-thiazolyl]thio]acetamideHomo sapiens (human)Potency3.548110
2-(4-chlorophenyl)-5-[[(4-methyl-2-thiazolyl)thio]methyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency2.818410
4-(3,4-dimethoxyphenyl)-2-thiophen-2-ylthiazoleHomo sapiens (human)Potency2.818410
2-oxo-1H-pyridine-3-carboxylic acid [2-(2,5-dimethyl-1-propyl-3-pyrrolyl)-2-oxoethyl] esterHomo sapiens (human)Potency1.258910
N-(4-chloro-2-fluorophenyl)-3-(methoxymethyl)-2-benzofurancarboxamideHomo sapiens (human)Potency6.309610
4-hydroxybenzoic acid [2-[1-(2-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)Potency5.011910
4-methyl-N'-(4-quinazolinyl)benzohydrazideHomo sapiens (human)Potency3.162310
5-methoxy-3-methyl-N-(3-methylbutyl)-2-benzofurancarboxamideHomo sapiens (human)Potency3.162310
4-[[6-[(2-methyl-5-thieno[2,3-e][1,3]benzothiazolyl)oxy]-3-pyridinyl]sulfonyl]morpholineHomo sapiens (human)Potency3.548110
2-[[[1-(2-methoxy-5-methylphenyl)-5-tetrazolyl]thio]methyl]-1,3-benzothiazoleHomo sapiens (human)Potency5.623410
2-(2,3-dihydro-1H-inden-5-yloxy)-1-(2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency2.818410
2-(1,3-benzoxazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneHomo sapiens (human)Potency0.631010
7-[(4-acetylphenoxy)methyl]-5-thiazolo[3,2-a]pyrimidinoneHomo sapiens (human)Potency3.981110
4-[(2,4-dioxo-1,3-diazaspiro[4.5]decan-3-yl)methyl]benzoic acid methyl esterHomo sapiens (human)Potency5.623410
1-[1-(3-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(1-methyl-5-tetrazolyl)thio]ethanoneHomo sapiens (human)Potency3.981110
2-(2,4-dibromophenoxy)-N-[oxo-(propan-2-ylamino)methyl]acetamideHomo sapiens (human)Potency1.000010
3-bromo-N-(4-methyl-2-oxo-1-benzopyran-7-yl)benzamideHomo sapiens (human)Potency0.501210
3-(difluoromethoxy)-N-(4,5-dihydrothiazol-2-yl)benzamideHomo sapiens (human)Potency2.238710
N-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-fluorobenzamideHomo sapiens (human)Potency3.548110
3-methoxy-N-(4-methyl-2-thiazolyl)benzamideHomo sapiens (human)Potency3.162310
digoxinHomo sapiens (human)Potency0.223910
4-phenoxyphenyl 4-hydroxypiperidine-1-carboxylateHomo sapiens (human)Potency3.162310
N-(2-methyl-1,3-benzothiazol-6-yl)benzamideHomo sapiens (human)Potency2.818410
N-(2-chlorophenyl)-4-(1-pyrrolyl)-1,3,5-triazin-2-amineHomo sapiens (human)Potency2.818410
2-(4-methylphenyl)-1,9b-dihydropyrazolo[1,5-b]isoindol-5-oneHomo sapiens (human)Potency2.818410
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency6.309610
tamoxifenHomo sapiens (human)Potency58.047910
3-(4-chlorophenyl)-2-methyl-3,3a,4,5-tetrahydrobenzo[g]indazoleHomo sapiens (human)Potency1.778310
N-[4-(5-oxazolyl)phenyl]benzamideHomo sapiens (human)Potency3.162310
N,N-diethyl-5-thiophen-2-yl-2-thiophenecarboxamideHomo sapiens (human)Potency2.511910
4-(2-fluorophenyl)-N-(2-methylbut-3-yn-2-yl)benzamideHomo sapiens (human)Potency3.162310
N-(4-chlorophenyl)-2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolecarboxamideHomo sapiens (human)Potency0.707910
N-(3,5-dimethylphenyl)-2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolecarboxamideHomo sapiens (human)Potency1.122010
4-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-2-methylthiazoleHomo sapiens (human)Potency1.778310
3-(methylthio)-5-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazoleHomo sapiens (human)Potency3.162310
1-[2-[(4-chlorophenoxy)methyl]-4-thiazolyl]ethanoneHomo sapiens (human)Potency0.891310
1-piperidinyl-(5-thiophen-2-yl-3-isoxazolyl)methanoneHomo sapiens (human)Potency1.000010
4-[3-(2,4-dichlorophenyl)-5-isoxazolyl]-2-pyrimidinamineHomo sapiens (human)Potency0.354810
N-(2-chlorophenyl)-2-[[5-[5-(trifluoromethyl)-2-pyridinyl]-1,3,4-oxadiazol-2-yl]thio]acetamideHomo sapiens (human)Potency2.238710
3-(4-methylphenyl)-2,1-benzoxazole-5-carboxaldehydeHomo sapiens (human)Potency2.238710
3-[5-[anilino(oxo)methyl]-2-furanyl]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency3.548110
4-(4-methylphenyl)-2-(3-nitrophenyl)-3-pyrazolamineHomo sapiens (human)Potency2.238710
3-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency2.238710
statticHomo sapiens (human)Potency91.999710
cgp 74514aHomo sapiens (human)Potency58.047910
N-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-2-furancarboxamideHomo sapiens (human)Potency3.981110
N'-(4-tert-butyl-2-thiazolyl)-4-chlorobenzohydrazideHomo sapiens (human)Potency5.623410
5-(2,3-dihydrobenzofuran-5-yl)-3-(4-fluorophenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency0.562310
2-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrimidineHomo sapiens (human)Potency1.778310
N-[4-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]phenyl]-3,4-dimethylbenzamideHomo sapiens (human)Potency3.162310
N-(2-quinolinyl)cyclohexanecarboxamideHomo sapiens (human)Potency1.122010
2-[(7-chloro-4-quinazolinyl)oxy]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethanoneHomo sapiens (human)Potency3.162310
N-(1H-indol-5-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency1.584910
N-[(2-hydroxyphenyl)-oxomethyl]-2,3-dihydrobenzofuran-5-carboxamideHomo sapiens (human)Potency1.412510
5-[[(4-methoxyanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid ethyl esterHomo sapiens (human)Potency0.281810
1,4-bis[2-(4-hydroxyphenyl)ethylamino]anthracene-9,10-dioneHomo sapiens (human)Potency58.047910
2-(3,4-dimethoxyphenyl)quinolineHomo sapiens (human)Potency2.238710
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)Potency3.162310
N-(2-chlorophenyl)-5-(2-pyridinyl)-2-thiophenecarboxamideHomo sapiens (human)Potency1.995310
2-[(4-chlorophenyl)methoxy]-6-methoxybenzonitrileHomo sapiens (human)Potency0.707910
N-phenyl-2-benzo[g][1]benzothiolecarboxamideHomo sapiens (human)Potency4.466810
N-[(2-chloroanilino)-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency3.162310
N'-[3-bicyclo[2.2.1]heptanyl(oxo)methyl]-3-chloro-1-benzothiophene-2-carbohydrazideHomo sapiens (human)Potency5.623410
N-(4-methyl-2-nitrophenyl)-2-furancarboxamideHomo sapiens (human)Potency2.818410
1-(4-tert-butylphenoxy)-3-(1H-1,2,4-triazol-5-ylthio)-2-propanolHomo sapiens (human)Potency0.446710
1-hexadecyl-3-methylimidazolium bromideHomo sapiens (human)Potency2.818410
N-(4-propan-2-ylphenyl)-3-bicyclo[2.2.1]heptanecarboxamideHomo sapiens (human)Potency3.548110
2-[[oxo(thiophen-2-yl)methyl]amino]-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency3.548110
N'-[(4-methoxyphenyl)methyl]-N-phenylcarbamimidothioic acid (2,5-dioxo-3-pyrrolidinyl) esterHomo sapiens (human)Potency5.623410
1-ethoxy-3-(2-methoxy-4-prop-2-enylphenoxy)-2-propanolHomo sapiens (human)Potency2.511910
N-[2-furanyl-(8-hydroxy-7-quinolinyl)methyl]-2-methylpropanamideHomo sapiens (human)Potency6.309610
N-(2-hydroxy-5-methylphenyl)-2-furancarboxamideHomo sapiens (human)Potency3.981110
3-(4-methoxyphenyl)-3-(4-methylphenyl)sulfonyl-1-phenyl-1-propanoneHomo sapiens (human)Potency2.238710
N-[5-[(4-methylphenyl)methyl]-2-thiazolyl]-2-oxolanecarboxamideHomo sapiens (human)Potency1.122010
2-chlorobenzoic acid [2-(4-methoxyphenyl)-2-oxo-1-phenylethyl] esterHomo sapiens (human)Potency3.981110
N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-5-ethyl-2-furancarboxamideHomo sapiens (human)Potency3.981110
4-chloro-3-(diethylsulfamoyl)-N-(2-nitrophenyl)benzamideHomo sapiens (human)Potency3.162310
(3-amino-5-nitro-2-benzofuranyl)-phenylmethanoneHomo sapiens (human)Potency3.548110
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(4-methoxyphenyl)methyl]acetamideHomo sapiens (human)Potency5.623410
2-nitrobenzoic acid [1-(4-methylphenyl)-1-oxopropan-2-yl] esterHomo sapiens (human)Potency0.891310
N-(4-carbamoylphenyl)-2-(4-methoxyphenyl)-4-quinolinecarboxamideHomo sapiens (human)Potency3.162310
2,4-dimethoxy-N-(5-nitro-2-pyridinyl)benzamideHomo sapiens (human)Potency1.122010
4-[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-2,6-dimethylmorpholineHomo sapiens (human)Potency1.122010
1-(4-methoxyphenyl)-N,N-dipropyl-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency0.707910
[3-[(2-chlorophenoxy)methyl]phenyl]-(2,6-dimethyl-4-morpholinyl)methanoneHomo sapiens (human)Potency3.548110
4-phenoxy-1-[4-(2-pyridinyl)-1-piperazinyl]-1-butanoneHomo sapiens (human)Potency1.258910
N-(4-anilinophenyl)-3-(hydroxymethyl)-1-piperidinecarbothioamideHomo sapiens (human)Potency2.511910
5-(4-methoxyanilino)-2-[(3-methylphenoxy)methyl]-4-oxazolecarbonitrileHomo sapiens (human)Potency3.981110
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-phenoxybutanamideHomo sapiens (human)Potency3.548110
N-[6-(dimethylsulfamoyl)-1,3-benzothiazol-2-yl]-2-thiophenecarboxamideHomo sapiens (human)Potency1.412510
2-[[(4-chlorophenyl)thio]methyl]-5-methylimidazo[1,2-a]pyridineHomo sapiens (human)Potency3.162310
N-(2-methoxy-3-dibenzofuranyl)-2-oxolanecarboxamideHomo sapiens (human)Potency3.981110
N-(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-3-isoxazolecarboxamideHomo sapiens (human)Potency1.778310
1-[(4-tert-butylphenyl)methyl]-4-(4-nitrophenyl)imidazoleHomo sapiens (human)Potency3.548110
N-[3-chloro-4-(4-morpholinyl)phenyl]-1,1-dioxo-1,2-benzothiazol-3-amineHomo sapiens (human)Potency2.238710
N-cycloheptyl-2-(cyclohexylamino)-2-sulfanylideneacetamideHomo sapiens (human)Potency2.511910
N-[(2-chlorophenyl)methyl]-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-hydroxy-5-nitro-4-triazolimineHomo sapiens (human)Potency5.011910
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methoxy-4-propan-2-yloxybenzamideHomo sapiens (human)Potency3.162310
N-[4-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-oxolanecarboxamideHomo sapiens (human)Potency0.794310
5-(2-nitrophenyl)-N-(2-thiazolyl)-2-furancarboxamideHomo sapiens (human)Potency2.818410
3-methyl-4-oxo-1,5,6,7-tetrahydroindole-2-carboxylic acid (4-methylcyclohexyl) esterHomo sapiens (human)Potency0.501210
2-[(2-furanylmethylthio)methyl]-5-methylimidazo[1,2-a]pyridineHomo sapiens (human)Potency1.122010
6-[(phenylmethylthio)methyl]imidazo[2,1-b]thiazoleHomo sapiens (human)Potency2.818410
2-methyl-1-cyclopropanecarboxylic acid (7-bromo-4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl esterHomo sapiens (human)Potency2.511910
1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)-2-(1-phthalazinyloxy)ethanoneHomo sapiens (human)Potency1.412510
N-(3-methyl-1,3-benzothiazol-2-ylidene)-2-pyrazinecarboxamideHomo sapiens (human)Potency1.995310
3-hydroxy-1-adamantanecarboxylic acid [2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)Potency0.354810
N-(1,3-benzothiazol-2-yl)-2-oxolanecarboxamideHomo sapiens (human)Potency1.122010
2-[2-[2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolyl]-2-oxoethyl]isoindole-1,3-dioneHomo sapiens (human)Potency0.501210
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-4-thiophen-2-ylbutanamideHomo sapiens (human)Potency2.818410
2-(2-amino-4H-[1,3,5]triazino[2,1-b][1,3]benzoxazol-4-yl)propanedioic acid diethyl esterHomo sapiens (human)Potency2.818410
2-[2-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-2-oxoethyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dioneHomo sapiens (human)Potency0.562310
6-methyl-2-(phenylethynyl)pyridineHomo sapiens (human)Potency5.804810
asterric acidHomo sapiens (human)Potency0.281810
N-(2-hydroxy-5-nitrophenyl)-3-nitrobenzamideHomo sapiens (human)Potency5.623410
N'-[4-(dimethylamino)phenyl]-N-propyloxamideHomo sapiens (human)Potency5.623410
5-methyl-N-(3-methylphenyl)-4-nitro-1H-pyrazol-3-amineHomo sapiens (human)Potency2.511910
1-(1-benzotriazolyl)-3-(2-methylphenoxy)-2-propanolHomo sapiens (human)Potency2.511910
3-(benzenesulfonyl)-3-(4-methoxyphenyl)-1-phenyl-1-propanoneHomo sapiens (human)Potency3.548110
1-[4-(6-bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]ethanoneHomo sapiens (human)Potency3.162310
4-amino-2-(butylthio)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency5.623410
N-[4-(1H-benzimidazol-2-yl)phenyl]-2-methyl-4-nitro-3-pyrazolecarboxamideHomo sapiens (human)Potency4.466810
2-(4-chlorophenoxy)-N-(5-nitro-2-thiazolyl)acetamideHomo sapiens (human)Potency0.562310
2-furanyl-[3-hydroxy-3-(trifluoromethyl)-3a,4,5,6,7,8-hexahydrocyclohepta[c]pyrazol-2-yl]methanoneHomo sapiens (human)Potency1.412510
1-(3-hydroxy-2,4,4-trimethyl-1-oxido-5-thiophen-2-yl-2-imidazol-1-iumyl)ethanoneHomo sapiens (human)Potency0.100010
5-hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazole-1-carboxylic acid ethyl esterHomo sapiens (human)Potency0.891310
5-(3,4-dimethoxyphenyl)-2-methylsulfonyl-3-thiophen-2-yl-3,4-dihydropyrazoleHomo sapiens (human)Potency2.511910
N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency5.623410
N-[2-[1-methyl-5-[[(4-methylphenyl)-oxomethyl]amino]-2-benzimidazolyl]ethyl]-2-furancarboxamideHomo sapiens (human)Potency3.548110
N-[3-chloro-4-(4-methyl-1-piperazinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency3.548110
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency3.162310
2-(2-furanyl)-2-[(4-methoxyphenyl)methyl-[2-[5-(5-methyl-2-furanyl)-2-tetrazolyl]-1-oxoethyl]amino]-N-(2-oxolanylmethyl)acetamideHomo sapiens (human)Potency0.100010
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-1-(2-methyl-2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency3.548110
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[(1-propan-2-yl-5-tetrazolyl)thio]ethanoneHomo sapiens (human)Potency3.548110
3,4-dihydro-2H-quinolin-1-yl-[4-(phenylmethyl)-5-thieno[3,2-b]pyrrolyl]methanoneHomo sapiens (human)Potency3.162310
1-[3-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]-1-butanoneHomo sapiens (human)Potency3.548110
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(4-methyl-2-thiazolyl)acetamideHomo sapiens (human)Potency3.548110
N-[2-(1-cyclohexenyl)ethyl]-3-(1,3-dioxo-2-isoindolyl)propanamideHomo sapiens (human)Potency3.981110
2-[(3-fluorophenyl)methylthio]-1-(4-phenyl-1-piperazinyl)ethanoneHomo sapiens (human)Potency3.162310
5-(2-furanyl)-N-(3-pyridinylmethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency3.548110
2-[(3-methoxyphenyl)-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency3.548110
(7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl)-(4-morpholinyl)methanoneHomo sapiens (human)Potency3.981110
N-[1-[(4-chlorophenyl)methyl]-5-methyl-3-pyrazolyl]-5-(3,4-dimethoxyphenyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency3.981110
3-chloro-N-(5-chloro-2-pyridinyl)-4-ethoxybenzamideHomo sapiens (human)Potency2.511910
4-[(1-methyl-2-oxo-4-quinolinyl)oxy]-N-(4-methyl-2-pyridinyl)butanamideHomo sapiens (human)Potency5.623410
5-(4-bromophenyl)-N,N-diethyl-3-isoxazolecarboxamideHomo sapiens (human)Potency1.995310
N-[4-[5-[(2-methylphenoxy)methyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideHomo sapiens (human)Potency3.981110
1-(2-methoxyethyl)-2-[(4-methylphenoxy)methyl]benzimidazoleHomo sapiens (human)Potency3.162310
1,7,7-trimethyl-9-oxo-N-(2-oxolanylmethyl)-8H-furo[3,2-f][1]benzopyran-2-carboxamideHomo sapiens (human)Potency5.623410
2-(3-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency3.981110
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency3.548110
3-[[oxo(2-quinoxalinyl)methyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency0.501210
4-[2-[[2-[[4-(1,3-benzodioxol-5-yl)-2-thiazolyl]amino]-2-oxoethyl]thio]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency2.818410
N-(2-methoxyethyl)-5-(3-methoxyphenyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency3.548110
1-[4-[(4-ethyl-1-piperazinyl)methyl]phenyl]-3-thiophen-2-ylureaHomo sapiens (human)Potency1.000010
3-methyl-N,6-diphenyl-2-imidazo[2,1-b]thiazolecarboxamideHomo sapiens (human)Potency3.981110
3-[5-amino-3-(4-chlorophenyl)-1-pyrazolyl]propanoic acid ethyl esterHomo sapiens (human)Potency2.511910
N-(2-methoxyethyl)-4-[4-(2-methoxyethylsulfamoyl)phenyl]benzenesulfonamideHomo sapiens (human)Potency0.891310
N-(1,3-benzodioxol-5-yl)-5-oxo-2,3-dihydrothiazolo[3,2-a]pyrimidine-6-carboxamideHomo sapiens (human)Potency3.548110
2-[(3-bromo-5,7-dimethyl-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzoxazoleHomo sapiens (human)Potency5.623410
N-[2-(2-methyl-1-indolyl)ethyl]benzamideHomo sapiens (human)Potency1.995310
2-[(5-anilino-1,3,4-thiadiazol-2-yl)thio]ethanolHomo sapiens (human)Potency5.623410
3-[[oxo-[3-(1-piperidinylsulfonyl)phenyl]methyl]amino]benzoic acidHomo sapiens (human)Potency1.995310
3,4-dihydro-2H-quinolin-1-yl-[5-(4-methoxyphenyl)-3-isoxazolyl]methanoneHomo sapiens (human)Potency3.162310
3-(4-methoxyphenyl)-3-(1-pyrrolyl)-N-(2-thiazolyl)propanamideHomo sapiens (human)Potency2.818410
N-(4-ethoxyphenyl)-2-(hydroxymethyl)benzamideHomo sapiens (human)Potency3.981110
5-(4-methoxyphenyl)-N-propan-2-yl-3-isoxazolecarboxamideHomo sapiens (human)Potency2.511910
[1-(3-methylphenyl)-5-benzimidazolyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency5.623410
N-(1,3-benzodioxol-5-yl)-2-[[6-methyl-4-oxo-3-(phenylmethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideHomo sapiens (human)Potency3.981110
N-(4-acetylphenyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideHomo sapiens (human)Potency1.122010
N-(2-furanylmethyl)-5-(3-methoxyphenyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency3.162310
2-(7-methyl-4-oxo-3-furo[3,4]pyrrolo[3,5-c][1,2,4]triazinyl)acetic acid methyl esterHomo sapiens (human)Potency3.162310
5-(4-chlorophenyl)-N-(2-furanylmethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency3.162310
5-(4-bromophenyl)-N-propan-2-yl-3-isoxazolecarboxamideHomo sapiens (human)Potency1.412510
N,3-diphenyl-1-pyrrolidinecarboxamideHomo sapiens (human)Potency1.584910
N-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideHomo sapiens (human)Potency2.511910
3-(4-methylphenyl)-N-phenyl-1-pyrrolidinecarboxamideHomo sapiens (human)Potency4.466810
N-(1,3-benzodioxol-5-yl)-3-ethyl-5-methyl-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideHomo sapiens (human)Potency3.162310
1-[(6-methoxy-2-furo[2,3-b]quinolinyl)-oxomethyl]-4-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency3.548110
2-(2-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency2.511910
N-cyclohexyl-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideHomo sapiens (human)Potency2.238710
n-(1-methyl-5-indolyl)-n'-(3-methyl-5-isothiazolyl)ureaHomo sapiens (human)Potency7.307810
3-(phenylthio)-1-(1-pyrrolidinyl)-1-propanoneHomo sapiens (human)Potency2.511910
2-[(1-oxo-3-phenylpropyl)amino]-3-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency5.623410
2-phenoxy-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamideHomo sapiens (human)Potency3.548110
5-methyl-2-(2-phenoxyethyl)-4-phenyl-1,2,4-triazol-3-oneHomo sapiens (human)Potency3.162310
2-(dichloromethyl)-4-(4-methylphenyl)-6-(methylthio)-1,3,5-triazineHomo sapiens (human)Potency3.548110
N-(2-chloro-3-pyridinyl)-3-oxo-3-phenylpropanamideHomo sapiens (human)Potency5.011910
N-[2-(4-morpholinyl)ethyl]-2-(4-propan-2-yloxyphenyl)-4-quinolinecarboxamideHomo sapiens (human)Potency3.548110
5-[[(3,4-dichloroanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterHomo sapiens (human)Potency0.631010
2-[(5-chloro-2-thiophenyl)-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency2.818410
2-[[2-(4-methoxyphenyl)-6-methyl-1-benzopyran-4-ylidene]amino]-4-methylpentanoic acidHomo sapiens (human)Potency2.818410
N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-[4-methyl-4-(4-methylphenyl)-2,5-dioxo-1-imidazolidinyl]acetamideHomo sapiens (human)Potency1.778310
2-(2,4-dibromophenoxy)-N-[[3-(hydroxymethyl)anilino]-sulfanylidenemethyl]acetamideHomo sapiens (human)Potency0.354810
N-[2-(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)ethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency2.818410
2-[[1-(phenylmethyl)-3-indolyl]thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency3.162310
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olHomo sapiens (human)Potency6.309610
nsc 105827Homo sapiens (human)Potency0.316210
N-cycloheptyl-4-(2-oxolanylmethoxy)benzamideHomo sapiens (human)Potency3.548110
N-(6-acetamido-3-prop-2-enyl-1,3-benzothiazol-2-ylidene)-2-thiophenecarboxamideHomo sapiens (human)Potency1.995310
5-(3,4-dimethoxyphenyl)-N-(3-pyridinyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency2.238710
2-[(4-methylphenoxy)methyl]imidazo[1,2-a]pyrimidineHomo sapiens (human)Potency3.548110
N-(4-fluorophenyl)-2-(3-methyl-5-oxo-1-phenyl-4H-pyrazol-4-yl)-2-oxoacetamideHomo sapiens (human)Potency2.818410
6-[2-(1-azepanyl)-2-oxoethoxy]-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-oneHomo sapiens (human)Potency4.466810
sb 242084Homo sapiens (human)Potency58.047910
2-(4-methoxyphenyl)acetic acid [2-[4-[(4-ethoxyanilino)-oxomethyl]anilino]-2-oxoethyl] esterHomo sapiens (human)Potency3.548110
2-[(1-methyl-3-indolyl)thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency3.981110
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideHomo sapiens (human)Potency0.794310
ML162Homo sapiens (human)Potency0.891310
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency1.122010
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency3.548110
N-[2-[[2-(4-chlorophenyl)-2-oxoethyl]thio]-4-oxo-3-quinazolinyl]benzamideHomo sapiens (human)Potency3.162310
3-nitro-N-(2-phenylethyl)-2-pyridinamineHomo sapiens (human)Potency2.818410
N-(4-bromophenyl)-5-methyl-4-nitro-1H-pyrazol-3-amineHomo sapiens (human)Potency2.818410
(4-chlorophenyl)-(7-methyl-3-imidazo[1,2-a]pyridinyl)methanoneHomo sapiens (human)Potency3.548110
2-[4-(4-methoxyphenyl)-2-thiazolyl]guanidineHomo sapiens (human)Potency3.548110
N-methyl-5-phenyl-2-thiophenecarboxamideHomo sapiens (human)Potency3.162310
2-[4-[[(3-chlorophenyl)-oxomethyl]amino]phenyl]propanedioic acid dimethyl esterHomo sapiens (human)Potency2.511910
2-Chloro-1-[5-(3,4-dimethoxyphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneHomo sapiens (human)Potency6.309610
2-(4-phenyl-1-piperazinyl)quinoxalineHomo sapiens (human)Potency1.584910
5-methyl-2-[[(4-nitrophenyl)-oxomethyl]hydrazo]-4-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency5.623410
4-methyl-2-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentanoic acid [3-(4-nitrophenyl)-4-oxo-1-benzopyran-7-yl] esterHomo sapiens (human)Potency3.548110
2-[[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]amino]-1-butanolHomo sapiens (human)Potency0.446710
4-(2-fluorophenyl)-5-methyl-2-(2-phenoxyethyl)-1,2,4-triazol-3-oneHomo sapiens (human)Potency2.818410
N-(2-chlorophenyl)-4-[[(2-methoxy-4-nitroanilino)-sulfanylidenemethyl]hydrazo]-4-oxobutanamideHomo sapiens (human)Potency3.548110
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleHomo sapiens (human)Potency3.162310
N-cyclohexyl-1-(4-fluorophenyl)-2,5-dimethyl-3-pyrrolecarboxamideHomo sapiens (human)Potency2.818410
N-(4-fluorophenyl)-5-methyl-1H-indole-2-carboxamideHomo sapiens (human)Potency2.511910
2-(1H-benzimidazol-2-ylthio)-1-[2,5-dimethyl-1-(2-oxolanylmethyl)-3-pyrrolyl]ethanoneHomo sapiens (human)Potency0.100010
7-methoxy-2-phenylimino-1-benzopyran-3-carboxamideHomo sapiens (human)Potency3.548110
N-[3-(dimethylsulfamoyl)-4-methylphenyl]-2-quinolinecarboxamideHomo sapiens (human)Potency5.623410
3-(5-bromo-2-furanyl)-5-(4-methoxyphenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency0.631010
N-[(3-hydroxyanilino)-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency3.981110
butanoic acid [2-oxo-2-(4-phenyldiazenylanilino)ethyl] esterHomo sapiens (human)Potency2.238710
2-(1H-indol-3-yl)-8-methylimidazo[1,2-a]pyridineHomo sapiens (human)Potency3.162310
3,4-dimethoxy-N-(3-methyl-1,3-benzothiazol-2-ylidene)benzamideHomo sapiens (human)Potency2.511910
N-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]acetamideHomo sapiens (human)Potency4.466810
4-(4-ethoxyphenyl)-1-(4-methoxyphenyl)-2-(methylthio)imidazoleHomo sapiens (human)Potency3.548110
N-(2-oxo-1-benzopyran-3-yl)cyclohexanecarboxamideHomo sapiens (human)Potency0.446710
3-methoxy-N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)benzamideHomo sapiens (human)Potency2.818410
2-[(1-methyl-2-imidazolyl)thio]-1-(2-naphthalenyl)ethanoneHomo sapiens (human)Potency2.238710
1-(3-methyl-1-piperidinyl)-2-(2-quinoxalinylthio)ethanoneHomo sapiens (human)Potency5.623410
1-(1H-benzimidazol-2-yl)-3-cyclohexylureaHomo sapiens (human)Potency0.446710
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneHomo sapiens (human)Potency2.511910
2-methoxy-N-(5-phenyl-1,2,4-thiadiazol-3-yl)benzamideHomo sapiens (human)Potency1.412510
2-cyclopentylacetic acid [2-[(3-chloro-9,10-dioxo-2-anthracenyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency3.548110
5-[[(2-methylanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterHomo sapiens (human)Potency3.548110
N-[3-(N-(2-chloro-1-oxoethyl)-4-nitroanilino)propyl]-2,2,2-trifluoroacetamideHomo sapiens (human)Potency6.309610
N,N-dimethylsulfamic acid [3-[(4-methoxyanilino)-oxomethyl]phenyl] esterHomo sapiens (human)Potency1.584910
5-(4-methylphenyl)-2-methylsulfonyl-3-thiophen-2-yl-3,4-dihydropyrazoleHomo sapiens (human)Potency1.778310
4-(4-morpholinyl)-3-nitro-N-(2-thiazolyl)benzamideHomo sapiens (human)Potency1.778310
5-bromo-N-[2-(2-methyl-1-indolyl)ethyl]-2-furancarboxamideHomo sapiens (human)Potency2.818410
6-(2-methyl-1-piperidinyl)-5-nitro-4-pyrimidinamineHomo sapiens (human)Potency1.122010
3-[(4-bromophenoxy)methyl]benzohydrazideHomo sapiens (human)Potency0.316210
2-[[5-(cyclohexylamino)-1,3,4-thiadiazol-2-yl]thio]-N-(9,10-dioxo-2-anthracenyl)acetamideHomo sapiens (human)Potency3.548110
1-(4-methoxyphenyl)-N-(2-oxolanylmethyl)-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency0.562310
digitoxigeninHomo sapiens (human)Potency1.258910
2-(N-(2-chloro-1-oxoethyl)-4-fluoroanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideHomo sapiens (human)Potency1.122010
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideHomo sapiens (human)Potency2.238710
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideHomo sapiens (human)Potency3.162310
(4-methyl-1-piperazinyl)-(2-thieno[3,2-b][1]benzothiolyl)methanoneHomo sapiens (human)Potency0.631010
N-(1-adamantyl)-6-(3,5-dimethyl-1-pyrazolyl)-1,2,4,5-tetrazin-3-amineHomo sapiens (human)Potency1.995310
N2,N6-bis[4-(dimethylamino)phenyl]pyridine-2,6-dicarboxamideHomo sapiens (human)Potency2.818410
2-Chloro-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneHomo sapiens (human)Potency6.309610
2-(4-morpholinyl)-10-pyridazino[6,1-b]quinazolinoneHomo sapiens (human)Potency2.511910
2,6-diphenyl-7-pyrazolo[1,5-a]pyrimidinamineHomo sapiens (human)Potency1.412510
1-(3-chloro-4-methoxyphenyl)-3-(2-fluorophenyl)ureaHomo sapiens (human)Potency1.778310
N-(3-isoxazolyl)-3-nitro-4-(1-piperidinyl)benzamideHomo sapiens (human)Potency2.818410
5-(2-chlorophenyl)-N-(4-methoxyphenyl)-2-furancarboxamideHomo sapiens (human)Potency3.162310
N-(1H-benzimidazol-2-yl)-3-phenylbutanamideHomo sapiens (human)Potency4.466810
N-(7-methyl-2-thiazolo[4,5-g][1,3]benzothiazolyl)propanamideHomo sapiens (human)Potency3.548110
6-chloro-2-[(phenylmethylthio)methyl]imidazo[1,2-a]pyridineHomo sapiens (human)Potency1.584910
5-oxo-2-pyrrolidinecarboxylic acid [2-[3-(4-methoxyphenyl)-5-(2-naphthalenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] esterHomo sapiens (human)Potency1.584910
N-(1,3-dioxo-5-isoindolyl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency3.981110
3-amino-N2-(2,3-dichlorophenyl)-5-(2-methoxyphenyl)imino-2H-thiophene-2,4-dicarboxamideHomo sapiens (human)Potency3.548110
3,5-dimethyl-4-oxo-6-thieno[2,3-d]pyrimidinecarboxylic acid (4-methylphenyl) esterHomo sapiens (human)Potency2.818410
[5-(2-furanyl)-3-isoxazolyl]-(4-methyl-1-piperidinyl)methanoneHomo sapiens (human)Potency1.778310
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-2-oxolanecarboxamideHomo sapiens (human)Potency3.548110
LSM-16483Homo sapiens (human)Potency3.548110
2-(3-methoxyphenyl)-3,5,6,7,8,9-hexahydrocyclohepta[2,3]thieno[2,4-b]pyrimidin-4-oneHomo sapiens (human)Potency1.258910
5-acetyloxy-6-bromo-2-[[(6-but-3-enyl-3-cyano-2-pyridinyl)thio]methyl]-1-methyl-3-indolecarboxylic acid ethyl esterHomo sapiens (human)Potency3.162310
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-2-(2-fluorophenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxamideHomo sapiens (human)Potency5.623410
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterHomo sapiens (human)Potency3.981110
5-(4-nitrophenyl)-3-phenyl-1H-imidazole-2-thioneHomo sapiens (human)Potency1.778310
3-[2-(2,4-dichlorophenoxy)ethoxy]-6-methyl-2-nitropyridineHomo sapiens (human)Potency6.309610
N-(4-fluorophenyl)-2-[(6-methyl-2-nitro-3-pyridinyl)oxy]acetamideHomo sapiens (human)Potency6.309610
N-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxolanylmethoxy)benzamideHomo sapiens (human)Potency2.818410
2-[4-(4-methoxyphenyl)-4-methyl-2,5-dioxo-1-imidazolidinyl]-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]acetamideHomo sapiens (human)Potency3.981110
N-(1H-benzimidazol-2-yl)-2-nitrobenzamideHomo sapiens (human)Potency3.981110
N-(6-methoxy-3-pyridinyl)-7-methyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideHomo sapiens (human)Potency2.818410
N-(2-methoxy-3-dibenzofuranyl)-3-pyridinecarboxamideHomo sapiens (human)Potency3.548110
2-[[4-(3,4-dimethylphenyl)-1-phenyl-2-imidazolyl]thio]-N-(1,1-dioxo-3-thiolanyl)acetamideHomo sapiens (human)Potency3.162310
4-[(2-cyano-1-oxoethyl)amino]benzoic acid [2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl] esterHomo sapiens (human)Potency3.162310
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[[2-(2-pyridinyl)-1-benzimidazolyl]methyl]-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency3.981110
N-[2-[oxo-(2-phenoxyethylamino)methyl]phenyl]-2-oxolanecarboxamideHomo sapiens (human)Potency3.981110
[5-(4-fluorophenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[2-(3-pyridinyl)-1-piperidinyl]methanoneHomo sapiens (human)Potency3.981110
5-nitro-N-[(4-propan-2-ylphenyl)methyl]-2-pyridinamineHomo sapiens (human)Potency2.511910
2-Chloro-1-[5-(furan-2-yl)-3-(5-methylfuran-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneHomo sapiens (human)Potency6.309610
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideHomo sapiens (human)Potency3.548110
N-[[(6-methyl-2-pyridinyl)amino]-oxomethyl]benzamideHomo sapiens (human)Potency3.981110
6-(4-bromo-3,5-dimethyl-1-pyrazolyl)-N-cyclohexyl-1,2,4,5-tetrazin-3-amineHomo sapiens (human)Potency2.238710
3-(4-methyl-1,3-dioxan-2-yl)-1-benzopyran-4-oneHomo sapiens (human)Potency3.162310
N-(1,1-dioxo-3-thiolanyl)-N-[(4-ethoxyphenyl)methyl]-2-oxo-1-benzopyran-3-carboxamideHomo sapiens (human)Potency3.162310
6-(4-methoxyphenyl)-N,3-dimethyl-2-imidazo[2,1-b]thiazolecarboxamideHomo sapiens (human)Potency1.584910
N-(6-fluoro-1,3-benzothiazol-2-yl)-2-oxolanecarboxamideHomo sapiens (human)Potency1.122010
sib 1757Homo sapiens (human)Potency18.356410
N-(5-acetyl-4-methyl-2-thiazolyl)-2-(2,4-dichlorophenoxy)acetamideHomo sapiens (human)Potency3.548110
2-[3-(1-benzotriazolylmethyl)-4-methoxyphenyl]-3-(4-methoxyphenyl)-1,2-dihydroquinazolin-4-oneHomo sapiens (human)Potency5.011910
brl 52537Homo sapiens (human)Potency4,610.910010
biochanin aHomo sapiens (human)Potency2.238710
acacetinHomo sapiens (human)Potency5.623410
apigeninHomo sapiens (human)Potency5.804810
7,3'-dihydroxy-4'-methoxyisoflavoneHomo sapiens (human)Potency5.623410
genisteinHomo sapiens (human)Potency5.135810
sulfuretinHomo sapiens (human)Potency5.623410
hispidulinHomo sapiens (human)Potency4.466810
daidzeinHomo sapiens (human)Potency9.200010
pterostilbeneHomo sapiens (human)Potency2.511910
flupenthixolHomo sapiens (human)Potency58.047910
tectochrysinHomo sapiens (human)Potency5.623410
n-oleoyldopamineHomo sapiens (human)Potency91.999710
tranilastHomo sapiens (human)Potency0.534910
cyclosporineHomo sapiens (human)Potency4.466810
genistinHomo sapiens (human)Potency5.623410
brefeldin aHomo sapiens (human)Potency0.092710
as 604850Homo sapiens (human)Potency8.199510
as 605240Homo sapiens (human)Potency10.322510
su 9516Homo sapiens (human)Potency29.653410
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acidHomo sapiens (human)Potency8.199510
N-(3-chlorophenyl)-1H-imidazole-5-carboxamideHomo sapiens (human)Potency3.981110
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,5-dimethyl-4-pyrazolecarboxamideHomo sapiens (human)Potency1.584910
N-cycloheptyl-1-hydroxy-3-oxo-2-propyl-1H-isoindole-5-carboxamideHomo sapiens (human)Potency1.995310
N-cyclohexyl-5-propyl-3-isoxazolecarboxamideHomo sapiens (human)Potency3.981110
[4-(3-methoxyphenyl)-1-piperazinyl]-[2-(1-piperidinyl)-1,3-benzothiazol-6-yl]methanoneHomo sapiens (human)Potency1.778310
N-(2-oxolanylmethyl)-2-(1-piperidinyl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency1.995310
[5-(2-methoxyphenyl)-3-isoxazolyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency3.548110
N-(3-acetylphenyl)-5-propan-2-yl-3-isoxazolecarboxamideHomo sapiens (human)Potency0.631010
N-[(3-methyl-6-imidazo[2,1-b]thiazolyl)methyl]-1-propanesulfonamideHomo sapiens (human)Potency3.981110
6-methyl-3-(prop-2-enylthio)-5H-[1,2,4]triazino[5,6-b]indoleHomo sapiens (human)Potency3.548110
3-(3,5-dimethyl-1-pyrazolyl)-5-phenyl-1,2,4-triazineHomo sapiens (human)Potency3.162310
cytochalasin bHomo sapiens (human)Potency1.122010
sib 1893Homo sapiens (human)Potency12.995310
(3r)-((2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl))methanoneHomo sapiens (human)Potency58.047910
su 6656Homo sapiens (human)Potency3.020410
5,7-dihydroxy-4',6-dimethoxyflavoneHomo sapiens (human)Potency3.162310
casein kinase iiHomo sapiens (human)Potency58.047910
semaxinibHomo sapiens (human)Potency16.360110
2-pyridylcarboxaldehyde benzoylhydrazoneHomo sapiens (human)Potency2.818410
(2e)-3-phenyl-1-(2,3,4,5-tetrahydro-1,6-benzodioxocin-8-yl)prop-2-en-1-oneHomo sapiens (human)Potency1.000010
bay 11-7082Homo sapiens (human)Potency115.821010
bay 11-7085Homo sapiens (human)Potency73.078010
styrylquinolineHomo sapiens (human)Potency2.818410
7-hydroxy-3-(4-methoxyphenyl)-4-methylcoumarinHomo sapiens (human)Potency5.623410
1,2-bis(2-pyridyl)ethyleneHomo sapiens (human)Potency2.818410
7-hydroxyisoflavoneHomo sapiens (human)Potency3.162310
7,4'-dimethoxy-5-hydroxyisoflavoneHomo sapiens (human)Potency0.631010
vinblastine sulfateHomo sapiens (human)Potency1.000010
vincristine sulfateHomo sapiens (human)Potency0.891310
3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5,7-dihydroxy-2-methyl-1-benzopyran-4-oneHomo sapiens (human)Potency3.548110
2-pyridylcarboxaldehyde isonicotinoylhydrazoneHomo sapiens (human)Potency2.511910
3-(dimethylamino)benzoic acid (7-hydroxy-2-oxo-1-benzopyran-4-yl)methyl esterHomo sapiens (human)Potency3.162310
dithiazanine iodideHomo sapiens (human)Potency0.281810
3,3'-diethylthiatricarbocyanine iodide, 3h-labeledHomo sapiens (human)Potency2.511910
3,3'-diethylthiacarbocyanine iodideHomo sapiens (human)Potency3.981110
2-(dimethylaminostyryl)-1-ethylpyridiniumHomo sapiens (human)Potency0.794310
5233705 compoundHomo sapiens (human)Potency6.309610
cladrinHomo sapiens (human)Potency3.162310
n,n,n-trimethyl-1-(4-stilbenoxy)-2-propylammonium iodideHomo sapiens (human)Potency25.929010
6-(bromomethylene)tetrahydro-3-(1-naphthaleneyl)-2h-pyran-2-oneHomo sapiens (human)Potency73.078010
alpha-(p-Methoxyphenyl)-2-pyridineacrylonitrileHomo sapiens (human)Potency1.995310
5-methoxy-3,6-diphenyl-1,2,4-triazineHomo sapiens (human)Potency5.623410
ciproxifanHomo sapiens (human)Potency2.310910
su 4312Homo sapiens (human)Potency1.458110
3-[[(3-methoxyanilino)-oxomethyl]amino]benzoic acidHomo sapiens (human)Potency0.316210
1-(1,3-benzodioxol-5-yl)-3-(6-methyl-2-pyridinyl)ureaHomo sapiens (human)Potency1.778310
1-(1,3-benzodioxol-5-yl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)ureaHomo sapiens (human)Potency0.398110
N-(1,3-benzodioxol-5-yl)-2-methyl-3-pyrazolecarboxamideHomo sapiens (human)Potency2.818410
(3S)-2-(2-chloro-1-oxoethyl)-1,1-dimethyl-4,9-dihydro-3H-pyrido[3,4-b]indole-3-carboxylic acid methyl esterHomo sapiens (human)Potency6.309610
emetine hydrochlorideHomo sapiens (human)Potency0.125910
a 77636Homo sapiens (human)Potency58.047910
b 43Homo sapiens (human)Potency115.821010
cycloheximideHomo sapiens (human)Potency0.316210
dinitrofluorobenzeneHomo sapiens (human)Potency16.360110
2-(1,3-benzothiazol-2-yl)-4-chloro-5-(3-chloroanilino)-3-pyridazinoneHomo sapiens (human)Potency3.981110
6-bromo-2-(1-pyrrolidinyl)-1,3-benzothiazoleHomo sapiens (human)Potency1.995310
dihydroouabainHomo sapiens (human)Potency2.818410
xct790Homo sapiens (human)Potency58.047910
2-[4-(2-pyrimidinyl)-1-piperazinyl]quinolineHomo sapiens (human)Potency1.412510
6-fluoro-N-phenyl-1,3-benzothiazol-2-amineHomo sapiens (human)Potency2.818410
4-fluoro-N-(4-fluoro-1,3-benzothiazol-2-yl)-1,3-benzothiazol-2-amineHomo sapiens (human)Potency6.309610
N-(6-fluoro-1,3-benzothiazol-2-yl)-6,7-dihydro-[1,4]dioxino[2,3-f][1,3]benzothiazol-2-amineHomo sapiens (human)Potency2.818410
3-(2-pyridinyl)-6-(2-pyridinylmethylthio)pyridazineHomo sapiens (human)Potency2.818410
N-(1,3-benzodioxol-5-yl)-3-[(2-methoxy-1-oxoethyl)amino]-2-benzofurancarboxamideHomo sapiens (human)Potency3.548110
N-cyclohexyl-2-[[6-(4-ethoxyphenyl)-3-pyridazinyl]thio]acetamideHomo sapiens (human)Potency1.995310
3-[(3-fluorophenyl)methylthio]-6-(2-furanyl)pyridazineHomo sapiens (human)Potency6.309610
3-[(4-chlorophenyl)methylthio]-6-(2-furanyl)pyridazineHomo sapiens (human)Potency3.548110
N-[3-(dimethylamino)propyl]-N-(6-methyl-1,3-benzothiazol-2-yl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency3.162310
1-[2-(4-methoxyphenyl)ethyl]-3,5-dimethyl-4-nitropyrazoleHomo sapiens (human)Potency3.162310
N-(4-methoxyphenyl)-2-[[1-(phenylmethyl)-2-imidazolyl]thio]acetamideHomo sapiens (human)Potency5.623410
N-[2-(2-methoxyphenoxy)ethyl]-2,3-dihydro-1H-indene-5-carboxamideHomo sapiens (human)Potency5.623410
1-ethyl-N-[[1-(phenylmethyl)-2-benzimidazolyl]methyl]-5-benzimidazolamineHomo sapiens (human)Potency3.548110
5-chloro-N-[4-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2-thiophenesulfonamideHomo sapiens (human)Potency2.818410
4-chloro-N-(4-ethylphenyl)-3-methyl-5-isoxazolecarboxamideHomo sapiens (human)Potency2.511910
hydralazine 4-anisaldehyde hydrazoneHomo sapiens (human)Potency0.281810
lassbio 294Homo sapiens (human)Potency2.511910
2-methyl-6-(phenylethynyl)pyridine hydrochlorideHomo sapiens (human)Potency3.162310
17-cyclopropylmethyl-6,7-didehydro-4,5-epoxy-5'-guanidinyl-3,14-dihydroxyindolo(2',3'-6,7)morphinanHomo sapiens (human)Potency58.047910
N(2)-([biphenyl]-4-ylsulfonyl)-N-hydroxy-N(2)-isopropoxy-D-valinamideHomo sapiens (human)Potency7,307.800010
protoapigenoneHomo sapiens (human)Potency3.981110
2-(4-butan-2-ylanilino)-3-pyridinecarbonitrileHomo sapiens (human)Potency3.162310
b 015Homo sapiens (human)Potency58.047910
calcimycinHomo sapiens (human)Potency146.025510
dihydroouabainHomo sapiens (human)Potency3.981110
2-ethyl-3-methoxy-N-(2-thiophen-2-ylethyl)-6-indazolecarboxamideHomo sapiens (human)Potency2.511910
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency1.122010
2-(4-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency1.000010
3-(benzenesulfonyl)-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]propanamideHomo sapiens (human)Potency0.562310
3-[(3-methylphenyl)methylthio]-6-thiophen-2-ylpyridazineHomo sapiens (human)Potency3.981110
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneHomo sapiens (human)Potency3.548110
dehydrocurvularinHomo sapiens (human)Potency3.162310
4-methoxybenzoic acid 2-(4-hydroxyphenyl)ethyl esterHomo sapiens (human)Potency3.981110
rabeprazole sodiumHomo sapiens (human)Potency3.162310
N-Cyclohexyl-5-(2-thienyl)-1,2-oxazole-3-carboxamideHomo sapiens (human)Potency3.162310
3-nitro-4-(2-oxolanylmethylamino)-N-(2-phenylethyl)benzamideHomo sapiens (human)Potency3.162310
N-(4-ethyl-1,2,5-oxadiazol-3-yl)-3,5,6-trimethyl-2-benzofurancarboxamideHomo sapiens (human)Potency1.778310
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)Potency3.162310
5-chloro-2-[(3-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)Potency3.162310
3-[3,5-dimethyl-1-[6-(1-piperidinyl)-3-pyridazinyl]-4-pyrazolyl]-N-(3-fluorophenyl)propanamideHomo sapiens (human)Potency2.818410
3-[3,5-dimethyl-1-[6-(1-piperidinyl)-3-pyridazinyl]-4-pyrazolyl]-N-(3-fluoro-4-methylphenyl)propanamideHomo sapiens (human)Potency1.995310
[4-(2,3-dimethylphenyl)-1-piperazinyl]-[5-[(4-methylphenyl)sulfonylmethyl]-2-furanyl]methanoneHomo sapiens (human)Potency1.000010
3-[2-(4-fluorophenyl)-5-tetrazolyl]-2-methoxypyridineHomo sapiens (human)Potency2.818410
2-chloro-3-[2-(4-methylphenyl)-5-tetrazolyl]pyridineHomo sapiens (human)Potency0.794310
3-[2-(4-methylphenyl)-5-tetrazolyl]quinolineHomo sapiens (human)Potency0.891310
2-chloro-3-[2-(3,4-dichlorophenyl)-5-tetrazolyl]pyridineHomo sapiens (human)Potency1.000010
N-(4-acetylphenyl)-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamideHomo sapiens (human)Potency0.794310
1-(1,4-dioxan-2-yl)-N-[[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-N-methylmethanamineHomo sapiens (human)Potency3.548110
dafadine CHomo sapiens (human)Potency2.238710
N,8-dimethyl-N-(3-methylphenyl)-4-oxo-5H-thieno[3,2-c]quinoline-2-carboxamideHomo sapiens (human)Potency2.511910
N-(4-methylphenyl)-4-tetrazolo[1,5-a]quinoxalinamineHomo sapiens (human)Potency2.818410
3-(3-pyridinylmethylthio)-6-thiophen-2-ylpyridazineHomo sapiens (human)Potency3.548110
N-(5-chloro-2-pyridinyl)-4H-thieno[3,2-c][1]benzopyran-2-carboxamideHomo sapiens (human)Potency3.548110
N-[5-[[2-(2-furanylmethylamino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency1.122010
2-[[6-(4-ethylphenyl)-3-pyridazinyl]thio]-N-(2-oxolanylmethyl)acetamideHomo sapiens (human)Potency5.623410
(2R,4S)-4-cyclohexyl-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamideHomo sapiens (human)Potency2.511910
2-[(5,6-dimethyl-4-thieno[2,3-d]pyrimidinyl)amino]-1-(4-nitrophenyl)ethanolHomo sapiens (human)Potency2.818410
3-methoxy-N-(5-methyl-2-pyridinyl)-2-naphthalenecarboxamideHomo sapiens (human)Potency5.623410
prunetin 4'-O-glucosideHomo sapiens (human)Potency1.584910
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideHomo sapiens (human)Potency3.162310
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideHomo sapiens (human)Potency6.309610
3-chloro-N-propan-2-yl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)Potency1.258910
N-(2-oxolanylmethyl)-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)Potency1.000010
N-[(2S)-1-hydroxypropan-2-yl]-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)Potency1.584910
N-(2-methoxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)Potency0.707910
N-(2-hydroxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)Potency1.122010
3-hex-1-ynyl-5H-indazolo[2,3-a][3,1]benzoxazineHomo sapiens (human)Potency0.354810
(3R,3aS,7R,7aS)-3-[5-(1-benzothiophen-2-yl)-2-methoxyphenyl]-7-methyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency3.162310
1-(2,3-dihydro-1H-inden-5-yl)-3-(2-ethoxyphenyl)ureaHomo sapiens (human)Potency0.562310
2-(2,5-dichlorophenoxy)-1-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-1-butanoneHomo sapiens (human)Potency0.891310
N-(3-nitrophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxamideHomo sapiens (human)Potency2.511910
1-(3-chlorophenyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)thioureaHomo sapiens (human)Potency3.162310
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-2-(1-piperidinyl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency0.446710
N-[3-[6-(1-azepanyl)-3-pyridazinyl]phenyl]-4-methylbenzenesulfonamideHomo sapiens (human)Potency5.623410
puromycin dihydrochlorideHomo sapiens (human)Potency2.238710
11,15>]Heptadec-14-yl]-5-hydrofuran-2-one, hydrateHomo sapiens (human)Potency0.089110
1-azepanyl-[5-[(4-chloro-3,5-dimethylphenoxy)methyl]-3-isoxazolyl]methanoneHomo sapiens (human)Potency2.818410
10-deacetyltaxolHomo sapiens (human)Potency0.251210
[5-[(3,4-difluorophenoxy)methyl]-3-isoxazolyl]-(3-propoxy-1-piperidinyl)methanoneHomo sapiens (human)Potency2.818410
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideHomo sapiens (human)Potency0.100010
[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-[5-[(4-chloro-2-methoxyphenoxy)methyl]-3-isoxazolyl]methanoneHomo sapiens (human)Potency3.162310
N,3-dimethyl-5-propyl-N-(2-thiazolylmethyl)-2-benzofurancarboxamideHomo sapiens (human)Potency2.511910
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-methyl-5-thiadiazolecarboxamideHomo sapiens (human)Potency1.412510
N-methyl-N-(3-pyridinylmethyl)-5-(5,6,7,8-tetrahydronaphthalen-2-yloxymethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency1.258910
5-[(3,4-dimethylphenoxy)methyl]-N-methyl-N-(4-oxanylmethyl)-3-isoxazolecarboxamideHomo sapiens (human)Potency2.818410
4-[oxo-[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]methyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency1.584910
[5-[(4-methoxy-1-naphthalenyl)oxymethyl]-3-isoxazolyl]-(4-methoxy-1-piperidinyl)methanoneHomo sapiens (human)Potency2.818410
N-[4-(1H-benzimidazol-2-yl)phenyl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-piperidinecarboxamideHomo sapiens (human)Potency2.818410
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideHomo sapiens (human)Potency0.112210
2-[3-(4-morpholinyl)propylamino]-9-xanthenoneHomo sapiens (human)Potency2.818410
3-[[1-(dimethylsulfamoyl)-4-piperidinyl]oxy]-N-[(3-methyl-5-isoxazolyl)methyl]benzamideHomo sapiens (human)Potency3.548110
[5-[(2-methoxyphenoxy)methyl]-3-isoxazolyl]-(4-methyl-3-phenyl-1-piperazinyl)methanoneHomo sapiens (human)Potency3.981110
5-[(2-chloro-4-methoxyphenoxy)methyl]-N-[(6-methyl-2-pyridinyl)methyl]-3-isoxazolecarboxamideHomo sapiens (human)Potency6.309610
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-(3,5-dimethyl-1-pyrazolyl)acetamideHomo sapiens (human)Potency3.162310
N-[5-[[2-(4-acetamidoanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-3-methoxybenzamideHomo sapiens (human)Potency2.818410
4-tert-butyl-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideHomo sapiens (human)Potency0.501210
4-ethoxy-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideHomo sapiens (human)Potency0.100010
bix 01294Homo sapiens (human)Potency58.047910
N-(2-furanylmethyl)-N-methyl-6-(1-methyl-5-indolyl)-4-quinazolinamineHomo sapiens (human)Potency3.548110
2-[5-(2-fluorophenyl)-2-furanyl]-3-hydroxy-1,2-dihydroquinazolin-4-oneHomo sapiens (human)Potency5.623410
6-(3-chloroanilino)-9-cyclopentyl-2-purinecarbonitrileHomo sapiens (human)Potency3.548110
2,3-dimethoxy-N-[4-(1-piperidinyl)phenyl]anilineHomo sapiens (human)Potency3.548110
N-[(5-chloro-8-hydroxy-7-quinolinyl)-cyclopropylmethyl]acetamideHomo sapiens (human)Potency6.309610
N-[(5-fluoro-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamideHomo sapiens (human)Potency4.802210
6-(3,5-difluoroanilino)-9-(2,2-difluoroethyl)-2-purinecarbonitrileHomo sapiens (human)Potency2.818410
6-(3-chloroanilino)-9-ethyl-2-purinecarbonitrileHomo sapiens (human)Potency3.548110
N-[(5-bromo-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamideHomo sapiens (human)Potency6.309610
(E,E)-1-bromo-2,5-bis-(4-hydroxystyryl)benzeneHomo sapiens (human)Potency3.662610
N-(2-chlorophenyl)-4-hydroxy-2-oxo-1-pentyl-3-quinolinecarboxamideHomo sapiens (human)Potency3.548110
kf38789Homo sapiens (human)Potency5.623410
salinazidHomo sapiens (human)Potency4.466810
phenylamilHomo sapiens (human)Potency2.059610
5-amino-2-phenyl-3H-triazolo[4,5-d]pyrimidin-7-oneHomo sapiens (human)Potency1.995310
N-(2,3-dimethylphenyl)-5-(2-fluorophenyl)-6H-1,3,4-thiadiazin-2-amineHomo sapiens (human)Potency3.162310
2-[(2-pyridinylthio)methyl]-1H-benzofuro[3,2-d]pyrimidin-4-oneHomo sapiens (human)Potency3.548110
N-[4-(6-chloro-5-nitro-1H-benzimidazol-2-yl)phenyl]acetamideHomo sapiens (human)Potency0.446710
2-(4-methoxyphenyl)-1H-quinazolin-4-oneHomo sapiens (human)Potency1.412510
N-[(3-methoxyphenyl)methyl]-4H-3,1-benzothiazin-2-amineHomo sapiens (human)Potency2.818410
N-butyl-5-(3,4-dimethylphenyl)-6H-1,3,4-thiadiazin-2-amineHomo sapiens (human)Potency2.818410
5-[1-[(2-chlorophenyl)methyl]-2,5-dimethyl-3-pyrrolyl]-N-(1-methoxypropan-2-yl)-6H-1,3,4-thiadiazin-2-amineHomo sapiens (human)Potency1.412510
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-oneHomo sapiens (human)Potency0.707910
N-(4-acetylphenyl)-2-[(4-oxo-1H-quinazolin-2-yl)thio]butanamideHomo sapiens (human)Potency6.309610
2-[(2-pyridinylthio)methyl]-1H-quinazolin-4-oneHomo sapiens (human)Potency2.511910
N'-(1h-indol-3-ylmethylene)benzohydrazideHomo sapiens (human)Potency5.623410
5-(4-chlorophenyl)-3-(4-nitrophenyl)-1H-pyrazoleHomo sapiens (human)Potency3.548110
5-(2,5-difluorophenyl)-N-(2-oxolanylmethyl)-6H-1,3,4-thiadiazin-2-amineHomo sapiens (human)Potency3.162310
5-[1-(4-chlorophenyl)-2,5-dimethyl-3-pyrrolyl]-N-methyl-6H-1,3,4-thiadiazin-2-amineHomo sapiens (human)Potency3.981110
fenobamHomo sapiens (human)Potency18.356410