Page last updated: 2024-08-07 13:34:43

Alpha-2A adrenergic receptor

An alpha-2A adrenergic receptor that is encoded in the genome of cow. [OMA:Q28838, PRO:DNx]

Synonyms

Alpha-2A adrenoreceptor;
Alpha-2A adrenoceptor;
Alpha-2AAR;
Alpha-2D adrenergic receptor

Research

Bioassay Publications (7)

TimeframeStudies on this Protein(%)All Drugs %
pre-19903 (42.86)18.7374
1990's2 (28.57)18.2507
2000's2 (28.57)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (12)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
alpha-methylserotoninBos taurus (cattle)IC500.019611
buspironeBos taurus (cattle)IC500.025011
clonidineBos taurus (cattle)IC500.002011
oxymetazolineBos taurus (cattle)Ki0.001511
prazosinBos taurus (cattle)Ki0.106011
5-methoxy-alpha-methyltryptamineBos taurus (cattle)IC500.086411
gepironeBos taurus (cattle)IC500.114011
ipsapironeBos taurus (cattle)Ki0.220012
mianserin hydrochlorideBos taurus (cattle)IC500.108733
1,2,3,4,6,7,12,12b-octahydroindolo(2,3-a)quinolizineBos taurus (cattle)Ki0.060311
rauwolscineBos taurus (cattle)Ki0.003411
4-iodo-2,5-dimethoxyphenylisopropylamine, (r)-isomerBos taurus (cattle)IC503.843011