An alpha-2A adrenergic receptor that is encoded in the genome of cow. [OMA:Q28838, PRO:DNx]
Alpha-2A adrenoreceptor;
Alpha-2A adrenoceptor;
Alpha-2AAR;
Alpha-2D adrenergic receptor
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 3 (42.86) | 18.7374 |
1990's | 2 (28.57) | 18.2507 |
2000's | 2 (28.57) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
alpha-methylserotonin | Bos taurus (cattle) | IC50 | 0.0196 | 1 | 1 |
buspirone | Bos taurus (cattle) | IC50 | 0.0250 | 1 | 1 |
clonidine | Bos taurus (cattle) | IC50 | 0.0020 | 1 | 1 |
oxymetazoline | Bos taurus (cattle) | Ki | 0.0015 | 1 | 1 |
prazosin | Bos taurus (cattle) | Ki | 0.1060 | 1 | 1 |
5-methoxy-alpha-methyltryptamine | Bos taurus (cattle) | IC50 | 0.0864 | 1 | 1 |
gepirone | Bos taurus (cattle) | IC50 | 0.1140 | 1 | 1 |
ipsapirone | Bos taurus (cattle) | Ki | 0.2200 | 1 | 2 |
mianserin hydrochloride | Bos taurus (cattle) | IC50 | 0.1087 | 3 | 3 |
1,2,3,4,6,7,12,12b-octahydroindolo(2,3-a)quinolizine | Bos taurus (cattle) | Ki | 0.0603 | 1 | 1 |
rauwolscine | Bos taurus (cattle) | Ki | 0.0034 | 1 | 1 |
4-iodo-2,5-dimethoxyphenylisopropylamine, (r)-isomer | Bos taurus (cattle) | IC50 | 3.8430 | 1 | 1 |