Page last updated: 2024-08-07 22:47:21

ClpP

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (1108)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
4-methylumbelliferyl acetateBacillus subtilisPotency25.118910
melatoninBacillus subtilisPotency28.183810
my 5445Bacillus subtilisPotency25.118910
2-aminofluoreneBacillus subtilisPotency11.220210
pyrithioneBacillus subtilisPotency3.981110
homovanillic acidBacillus subtilisPotency10.000010
6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diolBacillus subtilisPotency25.118910
aurintricarboxylic acidBacillus subtilisPotency21.671210
2,3-dimethoxy-1,4-naphthoquinoneBacillus subtilisPotency22.387210
ellipticineBacillus subtilisPotency17.782810
embelinBacillus subtilisPotency10.000010
nsc-39661Bacillus subtilisPotency35.481310
doxorubicin hydrochlorideBacillus subtilisPotency15.848910
methyclothiazideBacillus subtilisPotency14.125410
omeprazoleBacillus subtilisPotency22.387210
1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineBacillus subtilisPotency19.952610
tosufloxacinBacillus subtilisPotency8.912510
vincaBacillus subtilisPotency15.848910
phentolamineBacillus subtilisPotency22.387210
2-hydroxybenzylbenzimidazoleBacillus subtilisPotency15.848910
etiocholanoloneBacillus subtilisPotency31.622810
tetraethylammonium chlorideBacillus subtilisPotency0.707910
n,n'-diphenyl-4-phenylenediamineBacillus subtilisPotency12.589310
carbazoleBacillus subtilisPotency35.481310
salicylanilideBacillus subtilisPotency31.622810
2-naphthylamineBacillus subtilisPotency39.810710
4-biphenylamineBacillus subtilisPotency28.183810
efloxateBacillus subtilisPotency31.622810
dianisidineBacillus subtilisPotency3.548110
2-tolidineBacillus subtilisPotency5.011910
3-amino-9-ethylcarbazoleBacillus subtilisPotency39.810710
yohimbineBacillus subtilisPotency14.125410
benz(c)acridineBacillus subtilisPotency35.481310
triphenyltetrazolium chlorideBacillus subtilisPotency31.622810
flavanoneBacillus subtilisPotency15.848910
diphenylamineBacillus subtilisPotency31.622810
n-hydroxy-4-acetylaminostilbeneBacillus subtilisPotency31.622810
fenadiazoleBacillus subtilisPotency31.622810
2-amino-4-phenylphenolBacillus subtilisPotency31.622810
padimate-oBacillus subtilisPotency35.481310
k 308Bacillus subtilisPotency35.481310
pirfenidoneBacillus subtilisPotency31.622810
amlodipine besylateBacillus subtilisPotency11.220210
orbifloxacinBacillus subtilisPotency2.818410
5-AminoacenaphtheneBacillus subtilisPotency14.125410
benzoclidineBacillus subtilisPotency31.622810
aloxistatinBacillus subtilisPotency35.481310
pyrrolo(1,2-a)quinoxalineBacillus subtilisPotency2.511910
2-aminodiphenylamineBacillus subtilisPotency28.183810
2-(2'-pyridyl)benzimidazoleBacillus subtilisPotency28.183810
etidinBacillus subtilisPotency28.183810
masoprocolBacillus subtilisPotency0.631010
methyl 3-aminopyrazine-2-carboxylateBacillus subtilisPotency1.258910
methyl fluorone blackBacillus subtilisPotency25.118910
pr-d-92Bacillus subtilisPotency3.548110
EvoxineBacillus subtilisPotency7.079510
1-naphthoxyacetic acidBacillus subtilisPotency15.848910
8-methyl-4-oxo-3-pyrido[1,2-a]pyrimidinecarboxylic acid ethyl esterBacillus subtilisPotency2.511910
2-(1H-benzimidazol-2-yl)anilineBacillus subtilisPotency1.995310
1-(10h-phenothiazin-2-yl)ethanoneBacillus subtilisPotency31.622810
6-aminoindazoleBacillus subtilisPotency15.848910
witisolBacillus subtilisPotency14.125410
8-(4-tolylsulfonylamino)quinolineBacillus subtilisPotency28.183810
picloram-methylBacillus subtilisPotency31.622810
4-methylumbelliferyl butyrateBacillus subtilisPotency25.118910
8-(trifluoromethyl)-1H-quinolin-4-oneBacillus subtilisPotency28.183810
diflufenicanBacillus subtilisPotency35.481310
n-(2,6-difluorophenyl)-5-methyl(1,2,4)-triazol(1,5-a)pyrimidine-2-sulfonamideBacillus subtilisPotency31.622810
malic acid, (r)-isomerBacillus subtilisPotency3.981110
methylene bis(methylanthranilate)Bacillus subtilisPotency28.183810
ska-31Bacillus subtilisPotency3.548110
2-methyl-4-methoxymethyl-5-cyano-6-oxypyridineBacillus subtilisPotency2.818410
4,5-diphenyl-1,5-dihydroimidazol-2-oneBacillus subtilisPotency3.162310
8-cyclopropyltheophyllineBacillus subtilisPotency25.118910
wr 158122Bacillus subtilisPotency39.810710
diphyllinBacillus subtilisPotency21.154610
7-amino-4-trifluoromethylcoumarinBacillus subtilisPotency39.810710
7,9-dimethyl-9aH-quinolizine-1,2,3,4-tetracarboxylic acid tetramethyl esterBacillus subtilisPotency31.622810
gamma-fagarineBacillus subtilisPotency15.848910
quifenadine hydrochlorideBacillus subtilisPotency31.622810
methotrexateBacillus subtilisPotency23.735810
N-(1,3-dioxo-4-isoindolyl)acetamideBacillus subtilisPotency14.125410
teomorfolinBacillus subtilisPotency31.622810
2-phenylbenzotriazoleBacillus subtilisPotency25.118910
harmalanBacillus subtilisPotency15.848910
epiberberineBacillus subtilisPotency39.810710
metralindole monohydrochlorideBacillus subtilisPotency28.183810
rufloxacin hydrochlorideBacillus subtilisPotency28.183810
2-[(2-methoxy-2-oxoethyl)thio]benzoic acid methyl esterBacillus subtilisPotency25.118910
2-[2-[2-(2-aminophenoxy)ethoxy]ethoxy]anilineBacillus subtilisPotency22.387210
4,5-dimethoxy-2,3-dihydroinden-1-oneBacillus subtilisPotency28.183810
6-methyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileBacillus subtilisPotency1.000010
6-hydroxynicotineBacillus subtilisPotency31.622810
nsc 74859Bacillus subtilisPotency28.183810
3-([1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-a]pyridineBacillus subtilisPotency25.118910
n-acetyl-1-aminopyreneBacillus subtilisPotency14.125410
1,5-bis(2-methoxyphenyl)penta-1,4-dien-3-oneBacillus subtilisPotency28.183810
a-301Bacillus subtilisPotency28.183810
7-Acetoxy-2-methylisoflavoneBacillus subtilisPotency28.183810
u-29409Bacillus subtilisPotency25.118910
4-methoxyxanthoneBacillus subtilisPotency22.387210
6-methoxy-3-methyl-1,3-benzothiazol-2-imineBacillus subtilisPotency25.118910
5-(3,4,5-trimethoxyphenyl)-3H-1,3,4-oxadiazol-2-oneBacillus subtilisPotency15.848910
3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinecarboxylic acid ethyl esterBacillus subtilisPotency28.183810
medicarpinBacillus subtilisPotency0.707910
6-Methoxy-2-naphthoic acidBacillus subtilisPotency22.387210
3H-benzo[e]indole-2-carboxylic acidBacillus subtilisPotency22.387210
nsc 674495Bacillus subtilisPotency1.258910
3-imino-1,5,5-trimethyl-2-oxabicyclo[2.2.1]heptane-4,7,7-tricarbonitrileBacillus subtilisPotency31.622810
5f-203Bacillus subtilisPotency15.848910
7-(4-methoxyphenyl)-5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineBacillus subtilisPotency31.622810
resveratrolBacillus subtilisPotency25.118910
ferulic acidBacillus subtilisPotency19.952610
4-(2,3-Dihydroxy-3-methylbutoxy)furo(3,2-g)chromen-7-oneBacillus subtilisPotency28.183810
2-methyl-1H-pyrimido[1,2-a]benzimidazol-4-oneBacillus subtilisPotency14.125410
3-Furan-3-yl-3a,7-dimethyl-3a,4,5,6-tetrahydro-3H-isobenzofuran-1-oneBacillus subtilisPotency25.118910
3-methoxy-9H-carbazoleBacillus subtilisPotency35.481310
t-2 toxinBacillus subtilisPotency31.622810
N'-[(2-chlorophenyl)-oxomethyl]-5-(trifluoromethoxy)-1H-indole-2-carbohydrazideBacillus subtilisPotency15.848910
2-(3-oxo-4H-quinoxalin-2-yl)propanoic acid ethyl esterBacillus subtilisPotency28.183810
1-(2-pyridin-4-yl-1-oxa-3,4-diazaspiro[4.6]undec-2-en-4-yl)ethanoneBacillus subtilisPotency3.162310
5-methoxy-3-methyl-1H-indole-2-carboxylic acid ethyl esterBacillus subtilisPotency14.125410
TCMDC-138263Bacillus subtilisPotency31.622810
4,7-dimethoxy-2,3-dihydroinden-1-oneBacillus subtilisPotency31.622810
2-amino-3-cyano-5,6,7,8-tetrahydroquinoline-4-carboxylic acid methyl esterBacillus subtilisPotency28.183810
2,3-diphenyl-6-quinoxalinecarboxylic acidBacillus subtilisPotency22.387210
2-(4-hydroxy-3-methoxyphenyl)-3-(2-methoxyphenyl)-1,2-dihydroquinazolin-4-oneBacillus subtilisPotency31.622810
6-amino-2-methyl-8-phenyl-1,6,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrileBacillus subtilisPotency28.183810
2-[(6-chloro-2-oxo-4-propyl-1-benzopyran-7-yl)oxy]-N,N-dimethylacetamideBacillus subtilisPotency2.511910
3,6-dimethoxy-9H-carbazoleBacillus subtilisPotency39.810710
2-(2,5-dimethoxyphenyl)-5-(5-methyl-2-furanyl)-1,3,4-oxadiazoleBacillus subtilisPotency2.511910
2-[[5-[4-(1-piperidinylsulfonyl)phenyl]-1H-1,2,4-triazol-3-yl]thio]-N-(2-thiazolyl)acetamideBacillus subtilisPotency28.183810
N-[2-(cyclopentylamino)-1-(5-methyl-2-furanyl)-2-oxoethyl]-N-[(4-fluorophenyl)methyl]-4-thiadiazolecarboxamideBacillus subtilisPotency39.810710
1-[3-(dimethylamino)propyl]-3-(4-fluorophenyl)-1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]ureaBacillus subtilisPotency31.622810
1-[3-(dimethylamino)propyl]-1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-phenylureaBacillus subtilisPotency22.387210
1-[2,5-diethoxy-4-(1-tetrazolyl)phenyl]sulfonyl-4-(4-fluorophenyl)-3,6-dihydro-2H-pyridineBacillus subtilisPotency14.125410
2-oxo-N-(2-pyridinylmethyl)-1-benzopyran-3-carboxamideBacillus subtilisPotency31.622810
LSM-19079Bacillus subtilisPotency31.622810
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid ethyl esterBacillus subtilisPotency28.183810
2-[[3-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]acetic acid methyl esterBacillus subtilisPotency28.183810
N-methyl-N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)-3-oxolanecarboxamideBacillus subtilisPotency19.952610
2-(6-cyano-1-indolyl)-N-cyclohexylacetamideBacillus subtilisPotency14.125410
9-methyl-6H-benzo[c][1,2]benzothiazine 5,5-dioxideBacillus subtilisPotency28.183810
5-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideBacillus subtilisPotency35.481310
N-[1-[(4-methylphenyl)methyl]-2-benzimidazolyl]-2-furancarboxamideBacillus subtilisPotency25.118910
3-amino-5-methoxy-2-benzofurancarboxylic acid methyl esterBacillus subtilisPotency15.848910
2-[(3,4-dimethoxyphenyl)methyl]-5-[4-(4-methoxyphenyl)phenyl]-1,3,4-oxadiazoleBacillus subtilisPotency4.051620
3-[(1-tert-butyl-5-tetrazolyl)-[2-furanylmethyl(2-oxolanylmethyl)amino]methyl]-6-methoxy-1H-quinolin-2-oneBacillus subtilisPotency19.952610
5-(4-fluorophenyl)-N-[2-(1-piperidinyl)phenyl]-4-oxazolecarboxamideBacillus subtilisPotency28.183810
1-(1,3-benzodioxol-5-ylmethyl)-3-hydroxy-3-[2-(4-methylphenyl)-2-oxoethyl]-2-indoloneBacillus subtilisPotency15.848910
5-hydroxy-N,N-dimethyl-2-phenyl-3-benzofurancarboxamideBacillus subtilisPotency19.952610
11-[2-(4-morpholinyl)ethylamino]-7,8,9,10-tetrahydrobenzimidazolo[1,2-b]isoquinoline-6-carbonitrileBacillus subtilisPotency17.782810
2-(4-bromophenyl)-5-(2-methylphenyl)-1,3,4-oxadiazoleBacillus subtilisPotency25.118910
3-(benzenesulfonyl)-2-imino-1-(2-oxolanylmethyl)-5-dipyrido[1,2-d-3',4'-f]pyrimidinoneBacillus subtilisPotency1.995310
5-[[1-oxo-3-(3-oxo-4H-quinoxalin-2-yl)propoxy]methyl]-2-furancarboxylic acid ethyl esterBacillus subtilisPotency31.622810
1-[3-(4-morpholinyl)propyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-3-phenylureaBacillus subtilisPotency31.622810
N-[(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl]-4-fluoro-N-(2-hydroxyethyl)benzamideBacillus subtilisPotency22.387210
N-methyl-N-[5-(2-pyridinyl)-1,3,4-thiadiazol-2-yl]-3-oxolanecarboxamideBacillus subtilisPotency28.183810
3-acetamido-5-chloro-2-benzofurancarboxylic acidBacillus subtilisPotency17.782810
2-[benzenesulfonyl(2-pyridinyl)amino]acetic acid methyl esterBacillus subtilisPotency11.220210
5-(2-furanyl)-3-[2-methoxy-6-(4-methylphenyl)-3-pyridinyl]-1,2,4-oxadiazoleBacillus subtilisPotency28.183810
6-ethoxy-3-[[2-oxolanylmethyl-[[1-(2-phenylethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneBacillus subtilisPotency17.782810
2-methoxy-N-methyl-N-[5-(2-pyridinyl)-1,3,4-thiadiazol-2-yl]acetamideBacillus subtilisPotency25.118910
N,N-bis(but-2-ynyl)-3-methoxy-4-(1-tetrazolyl)benzenesulfonamideBacillus subtilisPotency28.183810
5-[3-(dimethylamino)phenyl]-N-methyl-1,3,4-thiadiazol-2-amineBacillus subtilisPotency7.943310
3-[[[1-(2-furanylmethyl)-5-tetrazolyl]methyl-[(2-methoxyphenyl)methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneBacillus subtilisPotency35.481310
7-[[1-(2-oxolanylmethyl)-5-tetrazolyl]-(1-pyrrolidinyl)methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-oneBacillus subtilisPotency31.622810
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]propanoic acid ethyl esterBacillus subtilisPotency35.481310
1-(1,3-benzodioxol-5-ylmethyl)-3-(4-methylphenyl)-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]ureaBacillus subtilisPotency31.622810
N-[(7-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(3-pyridinylmethyl)benzenesulfonamideBacillus subtilisPotency25.118910
2-(3,4-diethoxyphenyl)-5-(2-furanyl)-1,3,4-oxadiazoleBacillus subtilisPotency22.387210
N-[2-(4-methoxyphenyl)-6-methyl-5-benzotriazolyl]-3-pyridinecarboxamideBacillus subtilisPotency25.118910
5,6,7-trimethoxy-1-methyl-2-indolecarboxylic acidBacillus subtilisPotency12.589310
5-(2-ethoxyphenyl)-3-(2-methoxy-6-methyl-3-pyridinyl)-1,2,4-oxadiazoleBacillus subtilisPotency28.183810
5,7-dimethyl-2-(1-pyrrolidinyl)-3-quinolinecarbonitrileBacillus subtilisPotency25.118910
2-acetamido-N-[1-(3-cyano-4,6-dimethyl-2-pyridinyl)-4-piperidinyl]-3-(3-methoxyphenyl)propanamideBacillus subtilisPotency39.810710
3-cyclohexyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-1-[2-(1-pyrrolidinyl)ethyl]ureaBacillus subtilisPotency35.481310
1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-(4-methoxyphenyl)-1-(2-oxolanylmethyl)ureaBacillus subtilisPotency31.622810
3-[3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-6-ethyl-1H-quinolin-2-oneBacillus subtilisPotency39.810710
2-methoxy-N-(5-thiophen-2-yl-1,3,4-thiadiazol-2-yl)acetamideBacillus subtilisPotency39.810710
1-(3,5-dimethyl-1-pyrazolyl)-3-[2-(4-methoxyphenyl)-1-indolyl]-2-propanolBacillus subtilisPotency22.387210
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-methylphenyl)propanamideBacillus subtilisPotency28.183810
N-[2-(2-ethyl-5-tetrazolyl)phenyl]-3-(1-tetrazolyl)benzamideBacillus subtilisPotency25.118910
N-[3-(4-morpholinyl)propyl]-2-oxo-1-benzopyran-3-carboxamideBacillus subtilisPotency28.183810
4-[2-(3-fluorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]morpholineBacillus subtilisPotency35.481310
N-[1-[2-(2-chlorophenoxy)ethyl]-2-benzimidazolyl]acetamideBacillus subtilisPotency35.481310
1-[2-(dimethylamino)ethyl]-1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-(phenylmethyl)ureaBacillus subtilisPotency25.118910
5-cyano-6-[[2-(2,3-dimethylanilino)-2-oxoethyl]thio]-4-(2-furanyl)-2-methyl-N-phenyl-1,4-dihydropyridine-3-carboxamideBacillus subtilisPotency35.481310
2-pyridin-4-yl-2,3-dihydro-1H-quinazolin-4-oneBacillus subtilisPotency28.183810
2-[[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]amino]benzoic acid methyl esterBacillus subtilisPotency31.622810
N-methyl-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineBacillus subtilisPotency2.511910
N-[2-[(3-cyano-6-ethoxy-2-quinolinyl)amino]ethyl]propanamideBacillus subtilisPotency28.183810
2,5-diethoxy-N-[2-(2-methylphenyl)ethyl]-4-(1-tetrazolyl)benzenesulfonamideBacillus subtilisPotency31.622810
8-[2-(4-methoxyphenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-1,4-dioxa-8-azaspiro[4.5]decaneBacillus subtilisPotency5.965620
3-[2-hydroxyethyl-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]sulfamoyl]benzoic acid ethyl esterBacillus subtilisPotency35.481310
5-[(4-chloro-1-pyrazolyl)methyl]-N-(6-methyl-1,3-benzothiazol-2-yl)-2-furancarboxamideBacillus subtilisPotency39.810710
N-butyl-N-[5-(3,4,5-trimethoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-furancarboxamideBacillus subtilisPotency11.220210
6-methoxy-3-[[[1-(2-methoxyethyl)-5-tetrazolyl]methyl-(3-pyridinylmethyl)amino]methyl]-1H-quinolin-2-oneBacillus subtilisPotency19.952610
4-[2-(3-fluorophenyl)-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolin-9-yl]morpholineBacillus subtilisPotency31.622810
4-bromo-N-[(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-hydroxyethyl)benzamideBacillus subtilisPotency31.622810
1-(3-cyano-7-methoxy-2-quinolinyl)-4-piperidinecarboxylic acid ethyl esterBacillus subtilisPotency25.118910
6-ethyl-2,5-dimethyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrileBacillus subtilisPotency19.952610
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideBacillus subtilisPotency31.622810
1-[3-(dimethylamino)propyl]-1-[(5,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-3-(phenylmethyl)ureaBacillus subtilisPotency13.931820
N-[2-(2-ethyl-5-tetrazolyl)phenyl]-4-(1-tetrazolyl)benzamideBacillus subtilisPotency31.622810
3-(2-chlorophenyl)-1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-[2-(1-pyrrolidinyl)ethyl]ureaBacillus subtilisPotency31.622810
2-[4-(benzenesulfonyl)phenyl]-5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazoleBacillus subtilisPotency39.810710
8-[(1-tert-butyl-5-tetrazolyl)-thiomorpholin-4-ylmethyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneBacillus subtilisPotency25.118910
2-(2,5-dimethoxyphenyl)-5-[4-(4-methoxyphenyl)phenyl]-1,3,4-oxadiazoleBacillus subtilisPotency15.848910
2-fluoro-N-[2-(4-fluorophenyl)-1,3-benzoxazol-5-yl]benzamideBacillus subtilisPotency7.079510
2-[[2-(4-methoxyphenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]amino]ethanolBacillus subtilisPotency10.000010
5-(3,4-dimethoxyphenyl)-1H-1,2,4-triazol-3-amineBacillus subtilisPotency14.125410
N-[2-methoxy-4-[[2-[(3-methyl-4-oxo-2-quinazolinyl)thio]-1-oxoethyl]amino]phenyl]-2-furancarboxamideBacillus subtilisPotency22.387210
N-(2-pyridin-4-yl-1,3-benzoxazol-5-yl)butanamideBacillus subtilisPotency28.183810
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-methoxyacetamideBacillus subtilisPotency3.162310
2-fluoro-N-(2-hydroxyethyl)-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]benzamideBacillus subtilisPotency19.952610
1-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-[5-[4-(dimethylamino)phenyl]-2-tetrazolyl]ethanoneBacillus subtilisPotency28.183810
2-[2-[[2-[[1-(4-methoxyphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esterBacillus subtilisPotency39.810710
7-(methoxymethyl)-3-(2-methoxyphenyl)-1H-[1,2,4]triazolo[4,3-a]pyrimidin-5-oneBacillus subtilisPotency31.622810
6-ethoxy-3-[[2-furanylmethyl-[[1-(phenylmethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneBacillus subtilisPotency15.848910
N-(2-furanylmethyl)-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]benzamideBacillus subtilisPotency25.118910
9-[3-(4-acetyl-3,5-dimethyl-1-pyrazolyl)-2-hydroxypropyl]-6-methyl-3,4-dihydro-2H-carbazol-1-oneBacillus subtilisPotency7.943310
N-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(3-hydroxypropyl)benzenesulfonamideBacillus subtilisPotency12.589310
2-[[4-(4-methoxyphenyl)-2-pyrimidinyl]thio]-1-(4-morpholinyl)ethanoneBacillus subtilisPotency15.848910
N-propyl-N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamideBacillus subtilisPotency15.848910
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneBacillus subtilisPotency35.481310
6-methoxy-3-[[2-oxolanylmethyl-[[1-(phenylmethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneBacillus subtilisPotency28.183810
1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-(phenylmethyl)-1-(3-pyridinylmethyl)ureaBacillus subtilisPotency25.118910
1-(4-cyanophenyl)-3-[1-[(4-methoxyphenyl)methyl]-2-oxo-3-pyridinyl]ureaBacillus subtilisPotency12.589310
6-phenyl-4-(1-pyrrolyl)furo[2,3-d]pyrimidineBacillus subtilisPotency28.183810
4-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5-furo[3,2-b]pyrrolecarboxylic acid ethyl esterBacillus subtilisPotency15.848910
2-[(3-methyl-2,4-dioxo-5-thiazolidinyl)amino]benzoic acidBacillus subtilisPotency28.183810
4-methyl-6-(methylthio)-1H-quinolin-2-oneBacillus subtilisPotency35.481310
2-[[4-(3,4-dimethoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideBacillus subtilisPotency12.589310
3-cyclohexyl-1-[(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-[3-(4-morpholinyl)propyl]ureaBacillus subtilisPotency25.118910
N-(2-ethoxyphenyl)-1-[4-(1-pyrrolidinylsulfonyl)phenyl]-4-piperidinecarboxamideBacillus subtilisPotency35.481310
4-[2-(4-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]morpholineBacillus subtilisPotency18.947420
3-[2-methoxy-6-(4-methylphenyl)-3-pyridinyl]-5-(3-pyridinyl)-1,2,4-oxadiazoleBacillus subtilisPotency11.238420
6-[(2-fluorophenyl)methyl]-2,4-dimethyl-5-thieno[3,4]pyrrolo[1,3-d]pyridazinoneBacillus subtilisPotency39.810710
N-(2-furanylmethyl)-2-[(4-methoxyphenyl)sulfonylamino]benzamideBacillus subtilisPotency10.000010
N-methyl-N-[5-(5-methyl-2-pyrazinyl)-1,3,4-thiadiazol-2-yl]-2-oxolanecarboxamideBacillus subtilisPotency28.183810
4-amino-N5-[1-(2-furanyl)-2-(3-methylbutylamino)-2-oxoethyl]-N5-(2-methoxyphenyl)isothiazole-3,5-dicarboxamideBacillus subtilisPotency39.810710
6-methoxy-3-[[[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl-(2-phenylethyl)amino]methyl]-1H-quinolin-2-oneBacillus subtilisPotency25.118910
N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]butanamideBacillus subtilisPotency15.848910
1-piperidinecarboxylic acid (5-chloro-8-quinolinyl) esterBacillus subtilisPotency22.387210
2-[[2-[3-cyano-4-(methoxymethyl)-6-methyl-2-oxo-1-pyridinyl]-1-oxoethyl]amino]benzoic acid methyl esterBacillus subtilisPotency17.782810
1-(4,6-dimethyl-2-pyrimidinyl)-4-piperidinecarboxylic acidBacillus subtilisPotency19.952610
4-chloro-N-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-N-(2-oxolanylmethyl)benzenesulfonamideBacillus subtilisPotency11.220210
3-[3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-5,7-dimethyl-1H-quinolin-2-oneBacillus subtilisPotency31.622810
3-[1-(2-furanylmethyl)-5-phenyl-2-pyrrolyl]propanoic acidBacillus subtilisPotency28.183810
4-[(3-cyano-4,6-dimethyl-2-pyridinyl)thio]-3-oxobutanoic acid propan-2-yl esterBacillus subtilisPotency28.183810
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideBacillus subtilisPotency15.848910
5-(2-furanyl)-N-(4-methylphenyl)-3-isoxazolecarboxamideBacillus subtilisPotency35.481310
1-cyclohexyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-amineBacillus subtilisPotency14.125410
6-ethyl-6-methyl-5,8-dihydro-1H-thiopyrano[2,3]thieno[2,4-b]pyrimidine-2,4-dioneBacillus subtilisPotency35.481310
2-[[3-cyano-4-(5-methyl-2-furanyl)-5,6,7,8-tetrahydroquinolin-2-yl]thio]acetic acid methyl esterBacillus subtilisPotency31.622810
2-thiophen-2-yl-2,3-dihydro-1H-quinazolin-4-oneBacillus subtilisPotency31.622810
1-amino-5-(4-morpholinyl)-6,7,8,9-tetrahydrothieno[2,3-c]isoquinoline-2-carboxylic acid ethyl esterBacillus subtilisPotency31.622810
2-[(7-methyl-4-oxo-3-phenyl-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-2-yl)thio]acetic acid methyl esterBacillus subtilisPotency17.782810
6,7-dimethoxy-2-(2-thiazolyl)-3H-isoindol-1-oneBacillus subtilisPotency31.622810
2-[2-hydroxy-6,7-dimethoxy-4-(4-morpholinyl)-1-naphthalenyl]-N-phenylacetamideBacillus subtilisPotency28.183810
8-(2-furanyl)-6-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3,3-dimethyl-1,4-dihydrothiopyrano[3,4-c]pyridine-5-carbonitrileBacillus subtilisPotency39.810710
7-methyl-3-(4-morpholinyl)-1-(prop-2-enylamino)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileBacillus subtilisPotency15.848910
3-amino-5-methyl-4-[[3-(4-morpholinyl)propylamino]-oxomethyl]-2-thiophenecarboxylic acid ethyl esterBacillus subtilisPotency31.622810
LSM-19776Bacillus subtilisPotency25.118910
1-ethyl-6-methoxy-4-oxo-3-quinolinecarboxylic acidBacillus subtilisPotency31.622810
5-chloro-3-[[2-(4-ethoxycarbonyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterBacillus subtilisPotency25.118910
2-amino-4-(2-chlorophenyl)-6-(ethylthio)pyridine-3,5-dicarbonitrileBacillus subtilisPotency28.183810
6-[2-(dimethylamino)ethylamino]-8-(2-furanyl)-3,3-dimethyl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrileBacillus subtilisPotency39.810710
5-[4-morpholinyl(oxo)methyl]-2-pyranoneBacillus subtilisPotency31.622810
N-(2,1,3-benzothiadiazol-5-yl)-2,4-dimethyl-6-oxo-3-pyrancarboxamideBacillus subtilisPotency28.183810
3-(phenylmethyl)-1H-quinoxalin-2-oneBacillus subtilisPotency35.481310
4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl esterBacillus subtilisPotency28.183810
LSM-27020Bacillus subtilisPotency25.118910
4-(3-amino-5-bromo-2-benzofuranyl)-4-oxobutanoic acid methyl esterBacillus subtilisPotency15.848910
4-amino-5,8-dimethoxy-2-(1,1,2,2,2-pentafluoroethyl)-3-quinolinecarbonitrileBacillus subtilisPotency39.810710
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]-N-(2-phenylethyl)acetamideBacillus subtilisPotency39.810710
N-[2-(1-cyclohexenyl)ethyl]-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineBacillus subtilisPotency35.481310
N-ethyl-2-imino-10-methyl-1-[(4-methylphenyl)methyl]-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideBacillus subtilisPotency4.466810
N-(2-oxolanylmethyl)-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineBacillus subtilisPotency25.118910
2-(2-chlorophenyl)-5-(methylamino)-4-oxazolecarbonitrileBacillus subtilisPotency15.848910
2-[2-[[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]amino]ethoxy]ethanolBacillus subtilisPotency31.622810
2-(butan-2-ylamino)-N-[4-[5-[[2-(butan-2-ylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideBacillus subtilisPotency12.589310
1-(4-chlorophenyl)-N-(1-methoxypropan-2-yl)-4-pyrazolo[3,4-d]pyrimidinamineBacillus subtilisPotency28.183810
2-(4-methoxyphenyl)-1-(2-methylprop-2-enyl)benzimidazoleBacillus subtilisPotency15.848910
2-(butylamino)-N-[4-[5-[[2-(butylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideBacillus subtilisPotency3.981110
3-benzamido-5-bromo-2-benzofurancarboxylic acid methyl esterBacillus subtilisPotency28.183810
2-[2-[(1-phenyl-4-pyrazolo[3,4-d]pyrimidinyl)amino]ethoxy]ethanolBacillus subtilisPotency31.622810
5-(4-methoxyphenyl)-7-phenyl-[1,2,4]triazolo[1,5-a]pyrimidineBacillus subtilisPotency31.622810
7-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxoethyl]amino]-5H-[1,3]dioxolo[4,5-f]indole-6-carboxylic acid ethyl esterBacillus subtilisPotency3.162310
LSM-23818Bacillus subtilisPotency12.589310
5-methyl-6-pyridin-4-yl-6H-benzimidazolo[1,2-c]quinazolineBacillus subtilisPotency19.952610
1-[(4-methylphenyl)methyl]-4-[4-(4-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineBacillus subtilisPotency39.810710
2-[(6-chloro-4-ethyl-2-oxo-1-benzopyran-7-yl)oxy]propanoic acidBacillus subtilisPotency39.810710
5-(4-methoxyphenyl)-7-(4-methylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineBacillus subtilisPotency25.118910
cardionogen-2Bacillus subtilisPotency22.387210
LSM-32147Bacillus subtilisPotency12.589310
6-(4-methoxyphenyl)-3-phenyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleBacillus subtilisPotency35.481310
2-amino-4-pyridin-4-yl-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine-3-carbonitrileBacillus subtilisPotency22.387210
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-methyl-4-pyridinecarboxamideBacillus subtilisPotency28.183810
LSM-17424Bacillus subtilisPotency17.782810
2-[4-[(4-chlorophenyl)methoxy]phenyl]-5-(dimethylamino)-4-oxazolecarbonitrileBacillus subtilisPotency15.848910
N-[7-(2-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideBacillus subtilisPotency31.622810
5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-(2-furanyl)-4-oxazolecarbonitrileBacillus subtilisPotency14.125410
2-(4-methoxyphenyl)-3-propylimidazo[4,5-b]quinoxalineBacillus subtilisPotency28.183810
3-(ethylaminomethyl)-6-methyl-1H-quinolin-2-oneBacillus subtilisPotency28.183810
2-[4-[(4-chlorophenyl)methoxy]phenyl]-5-(4-morpholinyl)-4-oxazolecarbonitrileBacillus subtilisPotency1.995310
2-(2-furanyl)-5-(2-furanylmethylamino)-4-oxazolecarbonitrileBacillus subtilisPotency3.162310
5-[(2-chlorophenyl)methylamino]-2-(3,4-dimethoxyphenyl)-4-oxazolecarbonitrileBacillus subtilisPotency3.162310
5-(1-azepanyl)-2-(3,4-dimethoxyphenyl)-4-oxazolecarbonitrileBacillus subtilisPotency39.810710
1-[3-[(8-methyl-5H-pyrimido[5,4-b]indol-4-yl)amino]propyl]-2-pyrrolidinoneBacillus subtilisPotency11.220210
5-[4-(diphenylmethyl)-1-piperazinyl]-2-(2-methoxyphenyl)-4-oxazolecarbonitrileBacillus subtilisPotency3.981110
LSM-19719Bacillus subtilisPotency28.183810
2-(2-furanyl)-5-[4-(phenylmethyl)-1-piperazinyl]-4-oxazolecarbonitrileBacillus subtilisPotency28.183810
2-[4-[(4-chlorophenyl)methoxy]phenyl]-5-[3-(1-imidazolyl)propylamino]-4-oxazolecarbonitrileBacillus subtilisPotency25.118910
2-(3-methylphenyl)sulfonyl-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetonitrileBacillus subtilisPotency28.183810
2-methoxy-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-methoxyphenyl)acetamideBacillus subtilisPotency28.183810
N-[7-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideBacillus subtilisPotency28.183810
1-(thiophen-2-ylmethyl)-3-thiophen-2-ylsulfonyl-2-pyrrolo[3,2-b]quinoxalinamineBacillus subtilisPotency31.622810
5-[2-(3,4-dimethoxyphenyl)ethylamino]-2-(1-naphthalenylmethyl)-4-oxazolecarbonitrileBacillus subtilisPotency12.589310
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(4-methylphenyl)-2-oxolanecarboxamideBacillus subtilisPotency28.183810
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-propan-2-yl-4-pyridinecarboxamideBacillus subtilisPotency15.848910
3-[[2-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterBacillus subtilisPotency17.782810
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-propyl-2-pyridinecarboxamideBacillus subtilisPotency31.622810
N-butyl-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-2-pyridinecarboxamideBacillus subtilisPotency19.952610
3-[[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-1-oxoethyl]amino]-5-ethoxy-1H-indole-2-carboxylic acid ethyl esterBacillus subtilisPotency25.118910
9,10-dimethoxy-2-(2-pyridinylmethylamino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-oneBacillus subtilisPotency28.183810
LSM-28489Bacillus subtilisPotency3.548110
9-chloro-3-[(1-ethyl-2-pyrrolidinyl)methyl]-5H-pyrimido[5,4-b]indol-4-oneBacillus subtilisPotency31.622810
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanolBacillus subtilisPotency17.782810
3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpropanamideBacillus subtilisPotency39.810710
LSM-32980Bacillus subtilisPotency35.481310
7-(3-chlorophenyl)-2-(4-phenyl-1-piperazinyl)-7,8-dihydro-6H-quinazolin-5-oneBacillus subtilisPotency35.481310
7-methyl-3-(3-methylbutylamino)-1-(1-pyrrolidinyl)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileBacillus subtilisPotency22.387210
2-methyl-3-phenyl-5-propyl-7-[4-(2-pyridinyl)-1-piperazinyl]pyrazolo[1,5-a]pyrimidineBacillus subtilisPotency28.183810
LSM-20899Bacillus subtilisPotency28.183810
3,4,7-trimethyl-5-(3-oxobutan-2-yloxy)-1-benzopyran-2-oneBacillus subtilisPotency3.162310
6-amino-4-(4-fluorophenyl)-3-methyl-1-phenyl-5-pyrazolo[3,4-b]pyridinecarbonitrileBacillus subtilisPotency17.782810
N-[4-(4-oxo-2,3-dihydro-1,3-benzoxazin-2-yl)phenyl]acetamideBacillus subtilisPotency28.183810
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamideBacillus subtilisPotency39.810710
3-methyl-6-(1-naphthalenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleBacillus subtilisPotency22.387210
2-methoxy-6-[[(1-propyl-5-benzimidazolyl)amino]methyl]phenolBacillus subtilisPotency12.589310
8-methoxy-5-methyl-3-[2-(1-pyrrolidinyl)ethyl]-4-pyrimido[5,4-b]indoloneBacillus subtilisPotency31.622810
LSM-33283Bacillus subtilisPotency2.818410
2-(2,3,4-trimethoxyphenyl)-2,3-dihydro-1,3-benzoxazin-4-oneBacillus subtilisPotency28.183810
5-(1-imidazolylsulfonyl)-8-methoxyquinolineBacillus subtilisPotency12.589310
2-[(2-ethoxy-2-oxoethyl)thio]-1-benzimidazolecarboxylic acid ethyl esterBacillus subtilisPotency15.848910
2-[[2-furanyl(oxo)methyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid ethyl esterBacillus subtilisPotency35.481310
dichloramine-tBacillus subtilisPotency25.118910
4-[4-(2-quinoxalinyl)phenoxy]benzene-1,2-dicarbonitrileBacillus subtilisPotency19.952610
6-methyl-2-(trifluoromethyl)-3,5-dihydroimidazo[4,5-f]benzimidazoleBacillus subtilisPotency31.622810
4-(1-benzotriazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidineBacillus subtilisPotency31.622810
2-amino-4-phenyl-6-(1-pyrrolidinyl)pyridine-3,5-dicarbonitrileBacillus subtilisPotency39.810710
4-(3-amino-2-imidazo[1,2-a]pyridinyl)-2-methoxyphenolBacillus subtilisPotency17.782810
2-oxo-N-(3-pyridinylmethyl)-1-benzopyran-3-carboxamideBacillus subtilisPotency17.782810
2-[(3-cyano-6-cyclopropyl-4-thiophen-2-yl-2-pyridinyl)thio]acetamideBacillus subtilisPotency15.848910
6-(2-methyl-3-benzofuranyl)-2,3-dihydroimidazo[2,1-b]thiazoleBacillus subtilisPotency19.952610
N4-(3-chlorophenyl)-6-methyl-N2-(phenylmethyl)pyrimidine-2,4-diamineBacillus subtilisPotency22.387210
1-(3-methylphenyl)-N-(2-pyridinylmethyl)-4-pyrazolo[3,4-d]pyrimidinamineBacillus subtilisPotency19.952610
1-(3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinyl)ethanoneBacillus subtilisPotency19.952610
benzylidenephthalideBacillus subtilisPotency25.118910
5-(5-chloro-2-methoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneBacillus subtilisPotency28.183810
2-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxy]acetic acid propan-2-yl esterBacillus subtilisPotency35.481310
1-(1,3-benzodioxol-5-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterBacillus subtilisPotency31.622810
3-methyl-N-[4-(4-oxo-3,1-benzoxazin-2-yl)phenyl]butanamideBacillus subtilisPotency11.220210
5-methyl-4-[(2-oxo-1-benzopyran-7-yl)oxymethyl]-2-furancarboxylic acid methyl esterBacillus subtilisPotency14.125410
2-(3,4-dichlorophenyl)imidazo[1,2-a]pyrimidineBacillus subtilisPotency11.220210
5-(2-phenyl-4-triazolyl)-2H-tetrazoleBacillus subtilisPotency35.481310
3-[1-(carboxymethyl)-5-phenyl-2-pyrrolyl]propanoic acidBacillus subtilisPotency31.622810
1-[2-(dimethylamino)ethyl]-5-methoxy-N-methyl-2-indolecarboxamideBacillus subtilisPotency28.183810
6-methoxy-2-oxo-N-(3-pyridinylmethyl)-1-benzopyran-3-carboxamideBacillus subtilisPotency28.183810
2-[(dimethylamino)methyl]-4-methyl-6-(1-methylcyclohexyl)phenolBacillus subtilisPotency22.387210
2-[[2-furanyl(oxo)methyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterBacillus subtilisPotency39.810710
N-(1,2-dihydroacenaphthylen-5-yl)methanesulfonamideBacillus subtilisPotency15.848910
4-Acetyl-3-methyl-5-(methylthio)thiophene-2-carboxylic acidBacillus subtilisPotency35.481310
7,9-dibromo-3,4-dihydropyrido[2,1-c][1,2,4]thiadiazine 2,2-dioxideBacillus subtilisPotency25.118910
4-(1H-benzimidazol-2-yl)quinolineBacillus subtilisPotency15.848910
5-(2,4-dichlorophenyl)-N-(2-methylphenyl)-2-furancarboxamideBacillus subtilisPotency39.810710
5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineBacillus subtilisPotency31.622810
2-[[oxo(phenoxy)methyl]amino]benzene-1,4-dicarboxylic acid dimethyl esterBacillus subtilisPotency2.818410
5-(methoxymethyl)-2-phenyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneBacillus subtilisPotency25.118910
3-(4-methoxyphenyl)imidazo[1,5-a]pyridineBacillus subtilisPotency39.810710
N-(2-phenyl-3-imidazo[1,2-a]pyridinyl)carbamic acid methyl esterBacillus subtilisPotency17.612820
2-[[(4-phenyl-1,2,4-triazol-3-yl)thio]methyl]imidazo[1,2-a]pyrimidineBacillus subtilisPotency3.162310
LSM-21110Bacillus subtilisPotency15.848910
2-amino-5-ethyl-4-(2-furanyl)-6-propyl-3-pyridinecarbonitrileBacillus subtilisPotency31.622810
3-(4-chlorophenyl)-2,5-dimethyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneBacillus subtilisPotency19.952610
2-(4-fluorophenyl)-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidineBacillus subtilisPotency28.183810
6-methoxy-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazineBacillus subtilisPotency28.183810
2-methyl-N-(1-methyl-2,3-dihydropyrrolo[2,3-b]quinolin-4-yl)propanamideBacillus subtilisPotency39.810710
2-[(1-acetyl-3-indolyl)amino]benzoic acidBacillus subtilisPotency39.810710
4-[bis(phenylmethyl)amino]-2-(dimethylamino)-3-pyridinecarbonitrileBacillus subtilisPotency35.481310
4-phenyl-N-(3-pyridinylmethyl)-6-(trifluoromethyl)-2-pyrimidinamineBacillus subtilisPotency39.810710
3-hydroxypyridine, sodium saltBacillus subtilisPotency31.622810
(3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolyl)-(3-methyl-1-pyrazolyl)methanoneBacillus subtilisPotency3.548110
1-[(4-phenyl-1-piperazinyl)methyl]-2-naphthalenolBacillus subtilisPotency31.622810
4-[(6-methoxy-2-naphthalenyl)sulfonyl]morpholineBacillus subtilisPotency31.622810
2-(8-quinolinylthio)acetic acid phenacyl esterBacillus subtilisPotency25.118910
n-benzamidothioureaBacillus subtilisPotency31.622810
2-methoxy-4-[[2-(methylthio)anilino]methyl]phenolBacillus subtilisPotency28.183810
2-(1-methyl-2-phenyl-3-indolyl)ethanolBacillus subtilisPotency28.183810
6-ethyl-5-methyl-2-thiophen-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-oneBacillus subtilisPotency22.387210
1-[[(1-methyl-2-benzimidazolyl)amino]methyl]-2-naphthalenolBacillus subtilisPotency22.387210
4-amino-N-(4-ethoxyphenyl)benzenesulfonamideBacillus subtilisPotency44.668410
4-(4-morpholinyl)-N-(pyridin-4-ylmethyl)anilineBacillus subtilisPotency31.622810
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrileBacillus subtilisPotency25.118910
3-chloro-6-phenyl-[1,2,4]triazolo[4,3-b]pyridazineBacillus subtilisPotency25.118910
N-(1-naphthalenyl)-4-(phenylmethyl)-1-piperazinecarboxamideBacillus subtilisPotency17.782810
3-[2-(4-fluorophenyl)-5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]propanoic acid ethyl esterBacillus subtilisPotency25.118910
[4-(2-methylphenyl)-1-piperazinyl]-(4-nitrophenyl)methanethioneBacillus subtilisPotency25.118910
3-(2,3-dimethyl-1H-indol-5-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency25.118910
1-ethyl-2-[(4-methylphenoxy)methyl]benzimidazoleBacillus subtilisPotency35.481310
LSM-20909Bacillus subtilisPotency35.481310
3-phenyl-5,6,7,8-tetrahydro-1H-pyrazolo[5,1-b]quinazolin-9-oneBacillus subtilisPotency28.183810
5-(4-chlorophenyl)-2-furanpropionic acidBacillus subtilisPotency31.622810
3-amino-5H-pyrimido[5,4-b]indol-4-oneBacillus subtilisPotency19.952610
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneBacillus subtilisPotency25.118910
2-(2,5-dimethylphenyl)-3H-benzimidazol-5-amineBacillus subtilisPotency39.810710
N,4-dimethyl-5-phenyl-2-thiophenecarboxamideBacillus subtilisPotency31.622810
2-chloro-5-methyl-1-oxo-3-phenyl-4-pyrido[1,2-a]benzimidazolecarbonitrileBacillus subtilisPotency28.183810
1-(2-naphthalenyl)hexane-1,4-dioneBacillus subtilisPotency19.952610
1-(3-chlorophenyl)-3-(phenylmethyl)thioureaBacillus subtilisPotency28.183810
LSM-20487Bacillus subtilisPotency22.387210
3-amino-5-phenyl-2-thiophenecarboxylic acid ethyl esterBacillus subtilisPotency28.183810
3-(2-furanyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency10.000010
3-(4-ethyl-5-methyl-3-thiophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency28.183810
3-(1,3-benzodioxol-5-yl)-4-(2,5-dimethylphenyl)-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency28.183810
LSM-31933Bacillus subtilisPotency15.848910
2-(4-methyl-1-piperazinyl)-N-(5-thiophen-2-yl-1,3,4-thiadiazol-2-yl)acetamideBacillus subtilisPotency22.387210
N-(2-phenyl-6-imidazo[1,2-a]pyridinyl)acetamideBacillus subtilisPotency12.609620
N,N-dimethylcarbamic acid [4-[6-(trifluoromethyl)-2-imidazo[1,2-a]pyridinyl]phenyl] esterBacillus subtilisPotency10.000010
1-cyclohexyl-3-(2-ethylphenyl)ureaBacillus subtilisPotency3.162310
5-[2-(6-hydroxy-3-methyl-2-benzofuranyl)-2-oxoethyl]-2-furancarboxylic acid ethyl esterBacillus subtilisPotency31.622810
3-methyl-5-propyl-7-furo[3,2-g][1]benzopyranoneBacillus subtilisPotency14.125410
5-(4-fluorophenyl)-2-thiophen-2-yloxazoleBacillus subtilisPotency5.876620
2-(4-methoxyphenyl)-5-(3-pyridinyl)-1,3,4-oxadiazoleBacillus subtilisPotency5.011910
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-benzimidazolamineBacillus subtilisPotency15.848910
3-amino-6-cyclopropyl-4-(4-methoxyphenyl)-2-thieno[2,3-b]pyridinecarbonitrileBacillus subtilisPotency25.118910
2-[[oxo(thiophen-2-yl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid propan-2-yl esterBacillus subtilisPotency31.622810
2-[6-(carboxymethyl)-9-ethyl-3-carbazolyl]acetic acidBacillus subtilisPotency15.848910
2-[[anilino(oxo)methyl]amino]-4,5-dimethoxybenzoic acidBacillus subtilisPotency31.622810
5-(1-methyl-2-benzimidazolyl)-2-thiophenecarboxaldehydeBacillus subtilisPotency25.118910
6,7-dimethoxy-3-phenyl-1H-quinazoline-2,4-dioneBacillus subtilisPotency25.118910
4-(4-morpholinylmethyl)-3-quinolinolBacillus subtilisPotency19.952610
4-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]benzoic acid ethyl esterBacillus subtilisPotency31.622810
2-amino-9-ethyl-3-pyrido[2,3-b]indolecarboxylic acid ethyl esterBacillus subtilisPotency15.848910
7-methoxy-4,8-dimethyl-1-benzopyran-2-oneBacillus subtilisPotency3.548110
5-(4-chlorophenyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-furancarboxamideBacillus subtilisPotency14.125410
4-chloro-N-[4-(2-imidazo[1,2-a]pyridinyl)phenyl]benzamideBacillus subtilisPotency11.220210
8-chloro-7-propan-2-yloxy-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-4-oneBacillus subtilisPotency7.943310
5-acetyloxy-2-[[cyclohexyl(oxo)methyl]amino]benzoic acidBacillus subtilisPotency28.183810
1-propylsulfonyl-4-(2-pyridinyl)piperazineBacillus subtilisPotency15.848910
N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-thiophen-2-ylacetamideBacillus subtilisPotency10.000010
2-[(3-ethyl-4-methyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid methyl esterBacillus subtilisPotency14.125410
2-(4-methoxyphenyl)-5-(2-phenylethylamino)-4-oxazolecarbonitrileBacillus subtilisPotency31.622810
3-[5-(4-fluorophenyl)-1-(2-furanylmethyl)-2-pyrrolyl]propanoic acidBacillus subtilisPotency25.118910
6-methoxy-4-methyl-2-[(2-methylphenyl)methylthio]quinazolineBacillus subtilisPotency7.079510
3-[5-(4-methoxyphenyl)-1-prop-2-enyl-2-pyrrolyl]propanoic acidBacillus subtilisPotency25.118910
N-(3-methyl-4-oxo-1-benzopyran-2-yl)carbamic acid ethyl esterBacillus subtilisPotency5.011910
2-(2-methoxyphenyl)-1H-indoleBacillus subtilisPotency39.810710
1-(6,8-dimethyl-2,3-dihydropyrrolo[2,3-g]quinolin-1-yl)ethanoneBacillus subtilisPotency25.118910
2-(2,6-dichloroanilino)-3-pyridinesulfonamideBacillus subtilisPotency28.183810
3-(2-methoxy-6-methyl-3-pyridinyl)-5-(2-methoxyphenyl)-1,2,4-oxadiazoleBacillus subtilisPotency14.125410
7,8-dichloropyrido[1,2-a]benzimidazoleBacillus subtilisPotency14.113520
N-(2-methyl-5-tetrazolyl)-2-naphthalenecarboxamideBacillus subtilisPotency22.387210
2-[2-(2-furanyl)-5-methyl-7-oxo-1H-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]acetic acid methyl esterBacillus subtilisPotency28.183810
2-[(2,5-dimethoxyphenyl)sulfonyl-methylamino]acetic acidBacillus subtilisPotency39.810710
8-methoxy-1-(4-methoxyphenyl)-3-methyl-2-oxidobenzofuro[3,2-c]pyridin-2-iumBacillus subtilisPotency31.622810
8-(9-methyl-5H-pyrimido[5,4-b]indol-4-yl)-1,4-dioxa-8-azaspiro[4.5]decaneBacillus subtilisPotency10.000010
N-cyclopropyl-3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolecarboxamideBacillus subtilisPotency15.848910
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-3-methylbenzamideBacillus subtilisPotency22.387210
2-[[(4-methyl-1-pyrazolyl)-oxomethyl]amino]benzoic acid methyl esterBacillus subtilisPotency31.622810
1-(1-pyrrolidinyl)-2-(8-quinolinylthio)ethanoneBacillus subtilisPotency31.622810
4-methyl-6-[2-(4-methyl-1-piperidinyl)-2-oxoethoxy]-1-benzopyran-2-oneBacillus subtilisPotency28.183810
N-[(1-ethyl-2-oxo-6-benzo[cd]indolyl)sulfonyl]-N-(4-methoxyphenyl)-3-pyridinecarboxamideBacillus subtilisPotency35.481310
N-[4-(1,3-benzothiazol-2-yl)phenyl]-2-[(4-tert-butylphenyl)sulfonylamino]acetamideBacillus subtilisPotency5.011910
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideBacillus subtilisPotency39.810710
umi-77Bacillus subtilisPotency31.622810
2-[[4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideBacillus subtilisPotency25.118910
4-[1-oxo-2-(1-piperidinyl)ethyl]-9-phenylmethoxy-2,3-dihydro-1H-[1]benzopyrano[3,4-b]pyridin-5-oneBacillus subtilisPotency31.622810
N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-(3-methyl-N-methylsulfonylanilino)acetamideBacillus subtilisPotency15.848910
6-(4-benzoyl-1-piperazinyl)-3,3-dimethyl-8-propan-2-yl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrileBacillus subtilisPotency28.183810
2-[(3-cyano-4-phenyl-6-thiophen-2-yl-2-pyridinyl)thio]-N-propan-2-ylacetamideBacillus subtilisPotency22.387210
5-(4-bromophenyl)-N-(2-methoxyphenyl)-2-furancarboxamideBacillus subtilisPotency39.810710
1-[[2-(4-chlorophenyl)-1-oxoethyl]amino]-3-(1-naphthalenyl)ureaBacillus subtilisPotency28.183810
2-chloro-N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-5-(1,2,4-triazol-4-yl)benzamideBacillus subtilisPotency25.118910
2-[3-(4-methoxyphenyl)-1-benzo[f]quinolinyl]acetic acid ethyl esterBacillus subtilisPotency8.912510
[5-phenyl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-(1-piperidinyl)methanoneBacillus subtilisPotency28.183810
1-methoxy-N-[4-(pyridin-4-ylmethyl)phenyl]-2-naphthalenecarboxamideBacillus subtilisPotency2.511910
N-(2-methoxyphenyl)-5-methyl-3-[(2-methylphenyl)methyl]-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideBacillus subtilisPotency22.216720
5-(3-chlorophenyl)-N-(2-propyl-5-tetrazolyl)-2-furancarboxamideBacillus subtilisPotency17.782810
2-[(4-ethoxyphenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideBacillus subtilisPotency25.118910
N-[2-(3-chlorophenyl)ethyl]-2-[[3-cyano-6-(3-methoxyphenyl)-2-pyridinyl]thio]acetamideBacillus subtilisPotency28.183810
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N,N-diethylacetamideBacillus subtilisPotency31.622810
[7-(difluoromethyl)-5-(4-methoxyphenyl)-3-pyrazolo[1,5-a]pyrimidinyl]-(1-piperidinyl)methanoneBacillus subtilisPotency15.848910
2-(4-methylphenoxy)-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]acetamideBacillus subtilisPotency2.511910
N-(2-furanylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideBacillus subtilisPotency15.848910
N-(2-furanylmethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideBacillus subtilisPotency35.481310
2-(2-methylphenoxy)-N-[2-(4-methylphenyl)-5-benzotriazolyl]acetamideBacillus subtilisPotency8.912510
N-(3-methoxyphenyl)-4-(1-oxopropylamino)benzamideBacillus subtilisPotency31.622810
2-[[3-cyano-6-(4-methoxyphenyl)-4-phenyl-2-pyridinyl]thio]-N-(5-methyl-2-thiazolyl)acetamideBacillus subtilisPotency7.943310
5-bromo-N-[3-(2-oxo-1-benzopyran-3-yl)phenyl]-2-furancarboxamideBacillus subtilisPotency35.481310
3-methyl-N'-(1-oxo-2-phenoxyethyl)-1-phenyl-5-thieno[2,3-c]pyrazolecarbohydrazideBacillus subtilisPotency22.387210
1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-methyl-1-(thiophen-2-ylmethyl)thioureaBacillus subtilisPotency25.118910
LSM-16774Bacillus subtilisPotency12.589310
2-(6-amino-2-methyl-4-oxo-3-quinazolinyl)-N-(2-methylphenyl)acetamideBacillus subtilisPotency28.183810
1-(2,3-dihydroindol-1-yl)-2-[[4-methyl-5-[4-(1-pyrrolidinylsulfonyl)phenyl]-1,2,4-triazol-3-yl]thio]ethanoneBacillus subtilisPotency31.622810
4-(4-ethoxycarbonylanilino)-2-quinazolinecarboxylic acid ethyl esterBacillus subtilisPotency39.810710
1-ethyl-2-oxo-N-(2-pyridinylmethyl)-6-benzo[cd]indolesulfonamideBacillus subtilisPotency25.118910
2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)acetamideBacillus subtilisPotency6.309610
3-methoxy-4-(2-methoxy-3-methoxycarbonyl-1-naphthalenyl)-2-naphthalenecarboxylic acid methyl esterBacillus subtilisPotency25.118910
N-(2-phenylethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideBacillus subtilisPotency1.995310
9-(dimethylamino)-3-(4-methoxyphenyl)-4-pyrido[1,2]thieno[3,4-d]pyrimidinoneBacillus subtilisPotency14.125410
1-benzimidazolyl-[2-(4-methoxyphenyl)-4-quinolinyl]methanoneBacillus subtilisPotency31.622810
2-(4-ethylphenyl)-N-(4-methyl-1-piperazinyl)-4-quinolinecarboxamideBacillus subtilisPotency31.622810
4-chloro-1-methyl-N-[1-[(4-methylphenyl)methyl]-3-pyrazolyl]-3-pyrazolecarboxamideBacillus subtilisPotency19.952610
2-(4-bromophenyl)-1-[4-(2-pyridinyl)-1-piperazinyl]ethanoneBacillus subtilisPotency22.387210
LSM-16526Bacillus subtilisPotency12.589310
2-benzamido-4,5-dihydrobenzo[g][1]benzothiole-3-carboxamideBacillus subtilisPotency31.622810
3-[[oxo-[3-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl]methoxy]methyl]benzoic acid ethyl esterBacillus subtilisPotency31.622810
N-[(3-methoxyphenyl)methyl]-1-propyl-5-benzimidazolamineBacillus subtilisPotency28.183810
3-[[[4-(4-methoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]methyl]benzoic acidBacillus subtilisPotency17.782810
N-(3,5-dichlorophenyl)-2-(methanesulfonamido)benzamideBacillus subtilisPotency14.125410
2-(4-propylphenyl)-N-[2-(4-sulfamoylphenyl)ethyl]-4-quinolinecarboxamideBacillus subtilisPotency31.622810
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamideBacillus subtilisPotency35.481310
1-oxo-3-(1-piperidinyl)-5,6,7,8-tetrahydropyrrolo[1,2-a]indole-2-carbonitrileBacillus subtilisPotency31.622810
3-thiophen-2-ylimidazo[1,5-a]pyridineBacillus subtilisPotency31.622810
6-thioxanthineBacillus subtilisPotency8.912510
N-(2-furanylmethyl)-2-imino-5-oxo-1-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideBacillus subtilisPotency28.183810
N-[3-[2-(1-azepanyl)-4,5-dicyanophenoxy]phenyl]acetamideBacillus subtilisPotency31.622810
2-[[5-[(2-methyl-8-quinolinyl)oxymethyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]acetamideBacillus subtilisPotency28.183810
4-[[2-[(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterBacillus subtilisPotency39.810710
N-[4-[4-(ethylsulfonylamino)-3-methoxyphenyl]-2-methoxyphenyl]ethanesulfonamideBacillus subtilisPotency11.220210
2-(4-methoxyphenyl)-N-[4-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideBacillus subtilisPotency1.412510
N-[6-(diethylsulfamoyl)-1,3-benzothiazol-2-yl]-2-thiophenecarboxamideBacillus subtilisPotency25.118910
4-[[2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterBacillus subtilisPotency39.810710
2-(4-bromophenoxy)-N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideBacillus subtilisPotency10.000010
2-(1-naphthalenyl)-N-(2-phenyl-1,3-benzoxazol-5-yl)acetamideBacillus subtilisPotency19.952610
N-cyclohexyl-2-[(8-methoxy-6-oxo-3-benzo[c][1]benzopyranyl)oxy]acetamideBacillus subtilisPotency8.912510
3-ethoxy-N-[3-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl]benzamideBacillus subtilisPotency35.481310
5-methyl-4-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxymethyl]-2-furancarboxylic acidBacillus subtilisPotency28.183810
LSM-24412Bacillus subtilisPotency4.466810
2-[[(4-bromo-1-ethyl-3-pyrazolyl)-oxomethyl]amino]-4-phenyl-3-thiophenecarboxylic acid ethyl esterBacillus subtilisPotency31.622810
N-(2-furanylmethyl)-2-[[[2-[(4-methylphenyl)sulfonyl-(phenylmethyl)amino]phenyl]-oxomethyl]amino]benzamideBacillus subtilisPotency25.118910
darunavir ethanolateBacillus subtilisPotency39.810710
N-(2-furanylmethyl)-2-[[oxo-(3,4,5-trimethoxyphenyl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideBacillus subtilisPotency39.810710
5-(3,3-dimethyl-2-oxobutoxy)-3,4,7-trimethyl-1-benzopyran-2-oneBacillus subtilisPotency31.622810
N-[[5-(1H-benzimidazol-2-yl)-2-methylanilino]-sulfanylidenemethyl]-5-chloro-2-methoxybenzamideBacillus subtilisPotency35.481310
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-(2-methoxyphenyl)acetamideBacillus subtilisPotency2.511910
2-(4-chlorophenyl)-N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideBacillus subtilisPotency31.622810
4-(dimethylsulfamoyl)-N-(4-thiophen-2-yl-2-thiazolyl)benzamideBacillus subtilisPotency31.622810
3-(3-oxo-2-benzo[f][1]benzopyranyl)-1-phenyl-4-pyrazolecarboxaldehydeBacillus subtilisPotency5.623410
7-[4-(4-acetamidophenyl)sulfonyl-1-piperazinyl]-1-ethyl-6-fluoro-4-oxo-3-quinolinecarboxylic acidBacillus subtilisPotency39.810710
5-bromo-N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]-2-furancarboxamideBacillus subtilisPotency28.183810
N-(2-phenyl-5-benzotriazolyl)-2,3-dihydro-1,4-benzodioxin-6-carboxamideBacillus subtilisPotency8.912510
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzothiazoleBacillus subtilisPotency28.183810
2-(4-fluorophenoxy)-N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)acetamideBacillus subtilisPotency25.118910
3-bromo-5-[[4-[hydroxy(diphenyl)methyl]-1-piperidinyl]-oxomethyl]-2-pyranoneBacillus subtilisPotency31.622810
2-[[5-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-ethyl-1,3,4-thiadiazol-2-yl)acetamideBacillus subtilisPotency19.952610
2-[[5-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-[4-(1-pyrrolidinylsulfonyl)phenyl]acetamideBacillus subtilisPotency19.952610
2-[[[5-(5,6-dimethyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]methyl]benzonitrileBacillus subtilisPotency6.309610
4-[[3-[(2-chlorophenyl)methyl]-5-cyclopropyl-7-triazolo[4,5-d]pyrimidinyl]amino]-N,N-dimethylbenzenesulfonamideBacillus subtilisPotency31.622810
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidineBacillus subtilisPotency25.118910
2-(3-chlorophenyl)-9-[4-(2-pyrazinyl)-1-piperazinyl]-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolineBacillus subtilisPotency10.000010
4-cyano-N-methyl-N-[5-(2-pyridinyl)-1,3,4-thiadiazol-2-yl]benzamideBacillus subtilisPotency3.162310
1-[1-[(2-chloro-6-fluorophenyl)methyl]-2-oxo-3-pyridinyl]-3-(phenylmethyl)ureaBacillus subtilisPotency31.622810
7-methyl-2-[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]-3-quinolinecarbonitrileBacillus subtilisPotency25.118910
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-phenylethyl)acetamideBacillus subtilisPotency28.183810
(2,6-difluorophenyl)-[4-(5-fluoro-2-methyl-1-benzimidazolyl)-1-piperidinyl]methanoneBacillus subtilisPotency3.981110
7-(4-methoxyphenyl)-2-(1-pyrrolyl)-[1,2,4]triazolo[1,5-a]pyrimidineBacillus subtilisPotency28.183810
2-[benzenesulfonyl(2-pyridinyl)amino]acetic acidBacillus subtilisPotency28.183810
2-[(4-chlorophenyl)sulfonyl-(2-pyridinyl)amino]acetic acidBacillus subtilisPotency3.548110
1-[4-(2-fluorophenyl)-2-thiazolyl]-5-(trifluoromethyl)-4-pyrazolecarboxylic acid ethyl esterBacillus subtilisPotency35.481310
3-[5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazol-2-yl]-1-(phenylmethyl)-2-pyridinoneBacillus subtilisPotency39.810710
5-[1-(benzenesulfonyl)-3-pyrazolyl]-2-phenylthiazoleBacillus subtilisPotency14.125410
5-[1-(4-fluorophenyl)sulfonyl-3-pyrazolyl]-2-phenylthiazoleBacillus subtilisPotency19.952610
6-tert-butyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileBacillus subtilisPotency2.511910
7-(4-chlorophenyl)-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]-[1,2,4]triazolo[1,5-a]pyrimidineBacillus subtilisPotency39.810710
4-chloro-6-(4-methoxyphenyl)-2-phenyl-5-pyrimidinecarbonitrileBacillus subtilisPotency31.622810
3-phenyl-2H-1,4-benzoxazineBacillus subtilisPotency31.622810
2-(methylthio)-7-(4-phenylphenyl)-[1,2,4]triazolo[1,5-a]pyrimidineBacillus subtilisPotency28.183810
2-(2,4-dichlorophenyl)-5-[2-(methylthio)phenyl]-1,3,4-oxadiazoleBacillus subtilisPotency35.481310
r-7050Bacillus subtilisPotency39.810710
3-(5-chloro-1,3-benzoxazol-2-yl)-N-(phenylmethyl)-2-pyridinamineBacillus subtilisPotency2.818410
2-[(2,4-dichlorophenyl)methylthio]-6,7-dimethoxy-3-(thiophen-2-ylmethyl)-4-quinazolinimineBacillus subtilisPotency25.118910
2-(4-fluorophenyl)-1-indolizinecarboxylic acid ethyl esterBacillus subtilisPotency10.000010
1-[(4-methylphenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineBacillus subtilisPotency39.810710
4-(1-benzimidazolyl)-5-(4-methylphenyl)thieno[2,3-d]pyrimidineBacillus subtilisPotency28.183810
1-[(4-chlorophenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineBacillus subtilisPotency28.183810
3-(4-phenylphenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepineBacillus subtilisPotency8.912510
2-[[[4-(diethylsulfamoyl)phenyl]-oxomethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterBacillus subtilisPotency31.622810
6-(1,3-dioxo-2-isoindolyl)hexanoic acid (4-methyl-2-oxo-1-benzopyran-7-yl) esterBacillus subtilisPotency28.183810
1-ethyl-N-[3-(4-morpholinyl)propyl]-2-oxo-6-benzo[cd]indolesulfonamideBacillus subtilisPotency28.183810
2-[(7-methyl-4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-9-yl)oxy]acetic acid butyl esterBacillus subtilisPotency3.981110
N,N-diethylcarbamodithioic acid [2-(2-methyl-1H-indol-3-yl)-2-oxoethyl] esterBacillus subtilisPotency3.548110
N-(3-hydroxypropyl)-4-[(1-oxo-2,6,7,8-tetrahydrocyclopenta[2,3]thieno[2,4-b]pyrimidin-3-yl)thio]butanamideBacillus subtilisPotency31.622810
4-methoxy-2-(4-propoxyphenyl)quinazolineBacillus subtilisPotency31.622810
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-[(1,3-benzothiazol-2-ylthio)methyl]-4-triazolecarboxylic acid methyl esterBacillus subtilisPotency2.511910
2-chloro-4,6-diphenyl-5-pyrimidinamineBacillus subtilisPotency31.622810
4-(5-formyl-2-furanyl)benzoic acid propyl esterBacillus subtilisPotency31.622810
6-[4,6-bis(4-methoxyphenyl)-2-pyridinyl]-4H-1,4-benzoxazin-3-oneBacillus subtilisPotency3.162310
N-[3-(dimethylamino)propyl]-9H-carbazole-3-carboxamideBacillus subtilisPotency12.589310
3-chloro-N-[3-[[(3-chloro-4-nitrophenyl)-oxomethyl]amino]-2,2-dimethylpropyl]-4-nitrobenzamideBacillus subtilisPotency15.848910
5-[(4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl)oxymethyl]-2-furancarboxylic acidBacillus subtilisPotency2.511910
1-[[4-[(3,4-dichlorophenyl)thio]-3-pyridinyl]sulfonyl]-3-propylureaBacillus subtilisPotency22.387210
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(3,4-dimethoxyphenyl)-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency15.848910
3-chloro-6-(3,5-dimethyl-1h-pyrazol-1-yl)picolinic acidBacillus subtilisPotency28.183810
6-chloro-5,7-dimethyl-N-(thiophen-2-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineBacillus subtilisPotency12.589310
5-fluoro-3-[(4-methoxyphenyl)sulfonylamino]-1H-indole-2-carboxylic acid methyl esterBacillus subtilisPotency35.481310
tg 003Bacillus subtilisPotency0.707910
2-amino-1-[2-(4-morpholinyl)ethyl]-3-pyrrolo[3,2-b]quinoxalinecarboxylic acid ethyl esterBacillus subtilisPotency25.118910
2-amino-1-[2-(4-morpholinyl)ethyl]-N-prop-2-enyl-3-pyrrolo[3,2-b]quinoxalinecarboxamideBacillus subtilisPotency25.118910
N-(3,4-dichlorophenyl)-2-[4-(4-methoxyphenyl)-1-oxo-2-phthalazinyl]acetamideBacillus subtilisPotency28.183810
2-(2-furanyl)-3,5-dimethyl-4-oxido-6-phenylpyrazin-1-ium 1-oxideBacillus subtilisPotency28.183810
6-chloro-4-phenyl-2-(prop-2-enylthio)quinazolineBacillus subtilisPotency35.481310
1-[2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl]-3-phenylureaBacillus subtilisPotency15.848910
3-cyclohexyl-2-hydrazinyl-7-(phenylmethyl)-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-4-oneBacillus subtilisPotency39.810710
N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamideBacillus subtilisPotency10.000010
2-(2-furanyl)-5-methyl-6-(phenylmethyl)-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-oneBacillus subtilisPotency28.183810
4-chloro-N-(8-methyl-[1,3]dioxolo[4,5-g]quinazolin-6-yl)benzamideBacillus subtilisPotency35.481310
4-(4-chlorophenyl)-N-(3-pyridinylmethyl)-6-(trifluoromethyl)-2-pyrimidinamineBacillus subtilisPotency31.622810
3-amino-N-(2-fluorophenyl)-6-(2-furanyl)-2-thieno[2,3-b]pyridinecarboxamideBacillus subtilisPotency28.183810
N-(4,5-diphenyl-2-oxazolyl)-2-[(1-methyl-5-tetrazolyl)thio]acetamideBacillus subtilisPotency39.810710
2-amino-N-(3-ethoxypropyl)-1-(4-sulfamoylphenyl)-3-pyrrolo[3,2-b]quinoxalinecarboxamideBacillus subtilisPotency28.183810
N-[5-methyl-2-(4-methylphenyl)-3-pyrazolyl]-2-[(7-methyl-4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-9-yl)oxy]acetamideBacillus subtilisPotency25.118910
5-tert-butyl-2-methyl-3-phenyl-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineBacillus subtilisPotency2.238710
N-(1-ethyl-6-methyl-3-pyrazolo[3,4-b]quinolinyl)-2-(4-methoxyphenyl)acetamideBacillus subtilisPotency39.810710
3-methoxy-N-[[(2-oxo-1-benzopyran-6-yl)amino]-sulfanylidenemethyl]benzamideBacillus subtilisPotency19.952610
4,6-dimethyl-2-[3-(4-morpholinyl)propylamino]-3-pyridinecarbonitrileBacillus subtilisPotency14.125410
3,4,5-trimethoxy-N-(3-methyl-1,3-benzothiazol-2-ylidene)benzamideBacillus subtilisPotency28.183810
4-(3,4-dimethoxyphenyl)-1-(2-methoxyethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterBacillus subtilisPotency28.183810
acetic acid 2-[[oxo-(2-oxo-1-benzopyran-3-yl)methyl]amino]ethyl esterBacillus subtilisPotency25.118910
2-[[(4-bromo-1-ethyl-3-pyrazolyl)-oxomethyl]amino]-4,5-dimethyl-3-thiophenecarboxylic acid ethyl esterBacillus subtilisPotency39.810710
2-(1,3-benzoxazol-2-ylthio)-N-(4-phenyl-2-thiazolyl)acetamideBacillus subtilisPotency39.810710
3-methyl-2-benzo[g]benzofurancarboxylic acid [2-[N-(2-cyanoethyl)anilino]-2-oxoethyl] esterBacillus subtilisPotency25.118910
2-hydroxybenzoic acid [2-[[(1-methyl-2-pyrrolyl)-oxomethyl]amino]-2-oxoethyl] esterBacillus subtilisPotency39.810710
N-(1,3-benzodioxol-5-ylmethyl)-2-[(3-methyl-4-oxo-5-thiophen-2-yl-2-thieno[2,3-d]pyrimidinyl)thio]acetamideBacillus subtilisPotency39.810710
1-(4-fluorophenyl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxylic acid [2-(methylamino)-2-oxoethyl] esterBacillus subtilisPotency35.481310
2-[7-chloro-2,3-dioxo-4-(phenylmethyl)-1-quinoxalinyl]-N-(3-fluorophenyl)acetamideBacillus subtilisPotency39.810710
5-methyl-7-(trifluoromethyl)-2-thiazolo[4,5-b]pyridinamineBacillus subtilisPotency28.183810
3-methyl-1-[2-(2H-tetrazol-5-yl)ethyl]-4,6-bis(trifluoromethyl)pyrazolo[3,4-b]pyridineBacillus subtilisPotency10.000010
(3,4-dimethoxyphenyl)-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]methanoneBacillus subtilisPotency17.782810
1-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]-2-(2-methyl-4-thiazolyl)ethanoneBacillus subtilisPotency28.183810
2-[[2-furanyl(oxo)methyl]amino]benzoic acid [2-(cyclohexylmethylamino)-2-oxoethyl] esterBacillus subtilisPotency31.622810
2-[[2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]-1-oxoethyl]amino]-5-phenyl-3-thiophenecarboxamideBacillus subtilisPotency31.622810
(2S)-2-[[(2-chlorophenyl)-oxomethyl]amino]-3-methylbutanoic acid (6-nitro-4H-1,3-benzodioxin-8-yl)methyl esterBacillus subtilisPotency22.387210
3-[[[5-[3-(1-piperidinylsulfonyl)phenyl]-1,3,4-oxadiazol-2-yl]thio]methyl]-1,2,3-benzotriazin-4-oneBacillus subtilisPotency39.810710
3-methyl-6-thiophen-2-yl-4-isoxazolo[5,4-b]pyridinecarboxylic acid ethyl esterBacillus subtilisPotency31.622810
4-[[oxo-(1-phenyl-3-pyridin-4-yl-4-pyrazolyl)methyl]amino]benzoic acid methyl esterBacillus subtilisPotency39.810710
N-(4-fluorophenyl)-2-(5-methoxy-1-oxo-2-isoquinolinyl)acetamideBacillus subtilisPotency11.220210
4-fluoro-3-methoxy-N-(2-pyridinyl)benzenesulfonamideBacillus subtilisPotency28.183810
[9-(4-ethoxyphenyl)sulfonyl-2,3-dihydro-[1,4]dioxino[2,3-g]quinolin-8-yl]-(4-methylphenyl)methanoneBacillus subtilisPotency15.848910
(4-tert-butylphenyl)-[2-(4-fluorophenyl)-8-methyl-3-sulfanylidene-1,4,8-triazaspiro[4.5]dec-1-en-4-yl]methanoneBacillus subtilisPotency22.387210
2-[[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-oxomethyl]imino-1-(2-methylpropyl)-5-oxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterBacillus subtilisPotency6.309610
2-oxo-N-[2-[(2-phenyl-1H-indol-3-yl)thio]ethyl]-1-benzopyran-3-carboxamideBacillus subtilisPotency2.511910
3-[[(2,3-dimethylanilino)-sulfanylidenemethyl]amino]-1H-indole-2-carboxylic acid ethyl esterBacillus subtilisPotency14.125410
LSM-26967Bacillus subtilisPotency25.118910
3-(1H-indol-3-yl)-N-[4-(2-pyrimidinylsulfamoyl)phenyl]propanamideBacillus subtilisPotency31.622810
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterBacillus subtilisPotency39.810710
N-(2-methoxyphenyl)-5-methyl-3-(1-naphthalenylmethyl)-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideBacillus subtilisPotency31.622810
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-2-benzofurancarboxamideBacillus subtilisPotency31.622810
4-(benzenesulfonamido)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)benzamideBacillus subtilisPotency28.183810
N-[2-(1-naphthalenyl)-1,3-benzoxazol-5-yl]-1H-1,2,4-triazole-5-carboxamideBacillus subtilisPotency31.622810
3-[[[3-[(3-nitrophenyl)sulfamoyl]phenyl]-oxomethyl]amino]benzoic acidBacillus subtilisPotency3.162310
3-[1-(3-methoxypropyl)-5-thiophen-2-yl-2-pyrrolyl]propanoic acidBacillus subtilisPotency7.943310
N-[3-[(cyclopropylamino)-oxomethyl]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophen-2-yl]-2-furancarboxamideBacillus subtilisPotency31.622810
2-(3,5-dimethylphenoxy)-N-[3-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideBacillus subtilisPotency31.622810
4-chloro-3-[(2,5-dimethylphenyl)sulfamoyl]-N-(2-phenylphenyl)benzamideBacillus subtilisPotency28.183810
2-(5-bromo-2-furanyl)-6-methyl-3,1-benzoxazin-4-oneBacillus subtilisPotency39.810710
2-fluoro-N-[2-(2-methylpropyl)-1,3-dioxo-5-isoindolyl]benzamideBacillus subtilisPotency31.622810
5-(2-ethoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneBacillus subtilisPotency31.622810
N-(3-acetylphenyl)-5,7-dimethyl-2-pyrazolo[1,5-a]pyrimidinecarboxamideBacillus subtilisPotency28.183810
2-[[5-(2-benzofuranyl)-4-(phenylmethyl)-1,2,4-triazol-3-yl]thio]acetamideBacillus subtilisPotency35.481310
1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(5,7-diphenyl-2-pyrazolo[1,5-a]pyrimidinyl)methanoneBacillus subtilisPotency35.481310
2-[(3,4-dimethyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid prop-2-enyl esterBacillus subtilisPotency12.589310
2-[(3,4,8-trimethyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid prop-2-enyl esterBacillus subtilisPotency15.848910
2-[[[5-(3-chlorophenyl)-2-furanyl]-oxomethyl]amino]benzoic acid methyl esterBacillus subtilisPotency2.818410
4-[benzenesulfonyl(methyl)amino]-N-[2-[(4-chlorophenyl)methylthio]ethyl]benzamideBacillus subtilisPotency28.183810
2-[[5-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]-4-oxo-2-phenyl-1-benzopyran-7-yl]oxy]acetic acid tert-butyl esterBacillus subtilisPotency28.183810
4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-[4-(1-piperidinylsulfonyl)phenyl]benzamideBacillus subtilisPotency22.387210
8-[2-(4-chloro-2,5-dimethylphenoxy)ethoxy]quinolineBacillus subtilisPotency35.481310
4-chloro-N-[(phenacylamino)-sulfanylidenemethyl]benzamideBacillus subtilisPotency28.183810
N-(3-dibenzofuranyl)-2-[2-oxo-2-(2,4,6-trimethylanilino)ethoxy]benzamideBacillus subtilisPotency1.584910
reversanBacillus subtilisPotency15.848910
2-(4-methoxyphenyl)-N-[2-(4-morpholinyl)ethyl]-4-quinolinecarboxamideBacillus subtilisPotency35.481310
3-[2-(4-fluorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineBacillus subtilisPotency31.622810
4-(difluoromethoxy)-N-[5-[[4-(difluoromethylthio)phenyl]methyl]-2-thiazolyl]benzamideBacillus subtilisPotency14.125410
1-(2-chlorophenyl)-3-[[(1-ethyl-2-methyl-5-benzimidazolyl)-oxomethyl]amino]thioureaBacillus subtilisPotency28.183810
2-[(2,5-dimethylphenyl)sulfonylamino]-N-[4-(2-pyrimidinylsulfamoyl)phenyl]benzamideBacillus subtilisPotency25.118910
3-methoxy-2-naphthalenecarboxylic acid [2-(4-morpholinyl)-2-oxoethyl] esterBacillus subtilisPotency2.511910
LSM-19724Bacillus subtilisPotency35.481310
4-(diethylsulfamoyl)benzoic acid [2-[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]-2-oxoethyl] esterBacillus subtilisPotency25.118910
5-[(2-hydroxy-5-methylphenyl)-oxomethyl]-N,1-bis[2-(4-methoxyphenyl)ethyl]-2-oxo-3-pyridinecarboxamideBacillus subtilisPotency2.511910
3-[3-oxo-4-(2-phenylethyl)-2-quinoxalinyl]propanoic acidBacillus subtilisPotency28.183810
4-chloro-3-[(4-chlorophenyl)sulfamoyl]-N-(1H-1,2,4-triazol-5-yl)benzamideBacillus subtilisPotency31.622810
3-[2-(4-chlorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineBacillus subtilisPotency31.622810
2-(2-phenylanilino)-N-(phenylmethyl)acetamideBacillus subtilisPotency31.622810
1-(2-fluorophenyl)-1-cyclopentanecarboxylic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterBacillus subtilisPotency25.118910
3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolecarboxylic acid [2-(butylamino)-2-oxoethyl] esterBacillus subtilisPotency7.943310
2-(2-furanylmethylamino)benzoic acid [2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl] esterBacillus subtilisPotency25.118910
2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]-N-(2-pyridinylmethyl)acetamideBacillus subtilisPotency25.118910
1-(4-fluorophenyl)-1-cyclopentanecarboxylic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterBacillus subtilisPotency28.183810
1-(2-cyanoethyl)-6-(2-fluoro-4-methoxyphenyl)-3-methyl-4-pyrazolo[3,4-b]pyridinecarboxylic acid ethyl esterBacillus subtilisPotency25.118910
3-(1,3-benzodioxol-5-yl)-4-phenyl-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency28.183810
5-bromo-2-furancarboxylic acid [2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterBacillus subtilisPotency39.810710
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4,5-diphenyl-2-thiazolyl)acetamideBacillus subtilisPotency28.183810
3-[2-(2-furanylmethylamino)-2-oxoethoxy]-N-(2-methoxy-5-methylphenyl)-2-naphthalenecarboxamideBacillus subtilisPotency35.481310
2-phenyl-5-thiophen-2-yl-3-pyrazolecarboxylic acid [2-(4-chloro-3-nitroanilino)-2-oxoethyl] esterBacillus subtilisPotency22.387210
2-anilinobenzoic acid [2-(4-acetylanilino)-2-oxoethyl] esterBacillus subtilisPotency31.622810
4-[2-(4-fluoroanilino)-2-oxoethoxy]-3-methoxy-N-[4-(4-methoxyphenyl)-5-methyl-2-thiazolyl]benzamideBacillus subtilisPotency13.197020
3-(benzenesulfonyl)propanoic acid [2-[(3,5-dichloro-4-methyl-2-pyridinyl)amino]-2-oxoethyl] esterBacillus subtilisPotency31.622810
2-(butylamino)benzoic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterBacillus subtilisPotency28.183810
N-(3,4-dimethoxyphenyl)-6-phenyl-4-thieno[2,3-d]pyrimidinamineBacillus subtilisPotency31.622810
4-methyl-N-[4-(2-methyl-4-thiazolyl)phenyl]benzamideBacillus subtilisPotency14.125410
7-(4-quinazolinyloxymethyl)-5-thiazolo[3,2-a]pyrimidinoneBacillus subtilisPotency31.622810
N-cyclohexyl-2-[(4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl)oxy]acetamideBacillus subtilisPotency14.125410
N-(4-chloro-2-fluorophenyl)-3-(methoxymethyl)-2-benzofurancarboxamideBacillus subtilisPotency39.810710
2-[2-(2,3-dimethoxyphenyl)-4-thiazolyl]acetic acidBacillus subtilisPotency12.589310
2-[(3-chlorophenyl)methoxy]-3-methylquinoxalineBacillus subtilisPotency28.183810
5-[2-[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterBacillus subtilisPotency8.912510
5-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acidBacillus subtilisPotency10.000010
2-[[(3-methylphenyl)-oxomethyl]amino]benzoic acid (3,5-dimethyl-4-isoxazolyl)methyl esterBacillus subtilisPotency28.183810
2-[[[2-[(5-methoxycarbonyl-2-furanyl)methoxy]-2-oxoethyl]thio]methyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylic acid ethyl esterBacillus subtilisPotency28.183810
4-(4-methyl-1-piperidinyl)-5-phenyl-2-(3-pyridinyl)thieno[2,3-d]pyrimidineBacillus subtilisPotency3.162310
N-[2-[(1,3-benzodioxol-5-ylmethylamino)-oxomethyl]phenyl]-2-ethoxy-3-pyridinecarboxamideBacillus subtilisPotency39.810710
2-[(2,4-dimethoxyphenyl)methyl-methylamino]-N-(2-methoxy-3-dibenzofuranyl)acetamideBacillus subtilisPotency35.481310
tacrine hydrochlorideBacillus subtilisPotency31.622810
2-oxo-6-phenyl-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileBacillus subtilisPotency3.162310
3-(4-methylphenyl)-2,1-benzoxazole-5-carboxaldehydeBacillus subtilisPotency25.118910
2-(3,4-dichlorophenoxy)-6-(4-fluorophenyl)-3-pyridinecarbonitrileBacillus subtilisPotency39.810710
2-(4-chloro-2-methylphenoxy)-6-(4-fluorophenyl)-3-pyridinecarbonitrileBacillus subtilisPotency28.682620
2-chloro-N-(7-methyl-9-oxo-2-thioxanthenyl)benzamideBacillus subtilisPotency3.981110
2,6-dichlorobenzoic acid [3-cyano-6-(3-methoxyphenyl)-2-pyridinyl] esterBacillus subtilisPotency15.848910
2-chloro-N-[3-cyano-4-[(4-methoxyphenyl)thio]phenyl]benzamideBacillus subtilisPotency39.810710
2-[1-(1H-imidazol-1-yl)vinyl]phenolBacillus subtilisPotency12.589310
(3,5-dichlorophenyl)-[4-[2-(trifluoromethyl)-4-quinolinyl]-1-piperazinyl]methanoneBacillus subtilisPotency31.622810
LSM-28486Bacillus subtilisPotency2.818410
4-(9H-fluoren-9-yl)-N-phenyl-1-piperazinecarboxamideBacillus subtilisPotency31.622810
4-[4-(3-bromophenyl)sulfonyl-1-piperazinyl]-7-chloroquinolineBacillus subtilisPotency28.183810
2-fluoro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]acetamideBacillus subtilisPotency3.981110
2-[[sulfanylidene-[[2,2,2-trichloro-1-[(1-oxo-2-phenoxyethyl)amino]ethyl]amino]methyl]amino]benzoic acidBacillus subtilisPotency35.481310
3-(4-ethyl-1-piperazinyl)-5-methylpyridazino[3,4-b][1,4]benzoxazineBacillus subtilisPotency28.183810
dihydrosamidineBacillus subtilisPotency15.848910
1-(9-anthracenylmethyl)-3-piperidinolBacillus subtilisPotency19.952610
2-(difluoromethyl)-4-benzo[h][1]benzopyranoneBacillus subtilisPotency35.481310
3,7-dimethyl-2-[4-(2-pyridinyl)-1-piperazinyl]quinolineBacillus subtilisPotency31.622810
2-(4,6,7-Trimethyl-2-quinazolinyl)guanidineBacillus subtilisPotency17.782810
3-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) esterBacillus subtilisPotency15.848910
4-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) esterBacillus subtilisPotency31.622810
2-[[oxo(thiophen-2-yl)methyl]amino]-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideBacillus subtilisPotency39.810710
LSM-19241Bacillus subtilisPotency28.183810
N-[(2-chlorophenyl)-(2-hydroxy-1-naphthalenyl)methyl]butanamideBacillus subtilisPotency31.622810
2-methoxy-N-(2-pyridinylmethyl)-3-dibenzofuranamineBacillus subtilisPotency28.183810
LSM-19663Bacillus subtilisPotency28.183810
3-phenyl-1-[4-(2-pyridinyl)-1-piperazinyl]-1-propanoneBacillus subtilisPotency31.622810
2-(2,4-dichlorophenyl)-3-(phenylmethyl)-1,2-dihydroquinazolin-4-oneBacillus subtilisPotency31.622810
2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)-4-oxobutyl]benzo[de]isoquinoline-1,3-dioneBacillus subtilisPotency35.481310
2-(4-fluorophenyl)-4-(4-methoxyanilino)-1-(4-methoxyphenyl)-2H-pyrrol-5-oneBacillus subtilisPotency20.811920
3-(2-furanylmethyl)-2-phenyl-1,2-dihydroquinazolin-4-oneBacillus subtilisPotency28.183810
N-(3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-9H-xanthene-9-carboxamideBacillus subtilisPotency39.810710
9-[2-hydroxy-3-(2-methyl-1-benzimidazolyl)propyl]-6-methyl-3,4-dihydro-2H-carbazol-1-oneBacillus subtilisPotency14.125410
N-(2-adamantyl)-4-(4-ethylsulfonyl-1-piperazinyl)-3-nitrobenzamideBacillus subtilisPotency25.118910
LSM-19894Bacillus subtilisPotency31.622810
2-(2-oxo-1-benzo[cd]indolyl)-N-(2-oxolanylmethyl)acetamideBacillus subtilisPotency25.118910
1-(4-fluorophenyl)-3-(2-methoxy-3-dibenzofuranyl)ureaBacillus subtilisPotency39.810710
N-([biphenyl]-2-yl)-3-cyclopentylpropanamideBacillus subtilisPotency5.011910
importazoleBacillus subtilisPotency17.782810
N,4-dimethyl-N-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}benzenesulfonamideBacillus subtilisPotency12.589310
N-[2-[(2-furanylmethylamino)-oxomethyl]phenyl]-4-methyl-3-(1-piperidinylsulfonyl)benzamideBacillus subtilisPotency35.481310
2-[[(3-ethoxycarbonyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-oxomethyl]-3-methyl-3-bicyclo[2.2.1]hept-5-enecarboxylic acidBacillus subtilisPotency25.118910
2-[[(2-methoxy-4-nitroanilino)-sulfanylidenemethyl]amino]benzene-1,4-dicarboxylic acid diethyl esterBacillus subtilisPotency25.118910
2-(1,3-benzothiazol-2-ylamino)-5-spiro[1,6,7,8-tetrahydroquinazoline-4,1'-cyclopentane]oneBacillus subtilisPotency28.183810
N-[[(5-bromo-6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-2-(2-chlorophenoxy)acetamideBacillus subtilisPotency28.183810
4-methoxy-N-[4-[1-[(4-methoxyanilino)-oxomethyl]cyclopentyl]phenyl]benzamideBacillus subtilisPotency28.183810
1-(4-morpholinyl)-2-(4-phenylphenoxy)-1-propanoneBacillus subtilisPotency25.118910
N-(2-methoxy-3-dibenzofuranyl)-2-oxolanecarboxamideBacillus subtilisPotency31.622810
1-[(4-tert-butylphenyl)methyl]-4-(4-nitrophenyl)imidazoleBacillus subtilisPotency10.000010
3-[5-(4-methylphenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acidBacillus subtilisPotency25.118910
4H-[1,3]thiazino[3,2-a]benzimidazol-4-olBacillus subtilisPotency28.183810
2-[[4-(4-fluorophenyl)-6-(trifluoromethyl)-2-pyrimidinyl]sulfonyl]acetic acid ethyl esterBacillus subtilisPotency22.387210
3-[5-(4-fluorophenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acidBacillus subtilisPotency22.387210
N-[4-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-oxolanecarboxamideBacillus subtilisPotency28.183810
N-(3-cyano-2-thiophenyl)-2-[(1-methyl-2-imidazolyl)thio]acetamideBacillus subtilisPotency3.548110
2-[(4-methylphenyl)sulfonylamino]acetic acid (2-oxo-3-oxolanyl) esterBacillus subtilisPotency28.183810
4-[[2-(dimethylamino)-2-thiophen-2-ylethyl]amino]-5-methyl-6-thieno[2,3-d]pyrimidinecarboxylic acid ethyl esterBacillus subtilisPotency17.782810
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideBacillus subtilisPotency28.183810
5-[[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]methyl]-3-methyl-1H-pyrrole-2,4-dicarboxylic acid diethyl esterBacillus subtilisPotency39.810710
7-(3-methoxypropyl)-3-(phenylmethyl)-8-(3-thiophenyl)purine-2,6-dioneBacillus subtilisPotency31.622810
2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)benzoic acid thiophen-2-ylmethyl esterBacillus subtilisPotency28.183810
7-[3-[4-(2-ethoxyphenyl)-1-piperazinyl]-2-hydroxypropoxy]-4-methyl-1-benzopyran-2-oneBacillus subtilisPotency11.220210
2-amino-4-chlorobenzoic acid [2-oxo-2-(3,3,5-trimethyl-7-azabicyclo[3.2.1]octan-7-yl)ethyl] esterBacillus subtilisPotency28.183810
3-fluoro-6a,7,8,9,10,11-hexahydro-6H-azepino[2,1-c][1,2,4]benzothiadiazine 5,5-dioxideBacillus subtilisPotency28.183810
2-(2-amino-4H-[1,3,5]triazino[2,1-b][1,3]benzoxazol-4-yl)propanedioic acid diethyl esterBacillus subtilisPotency25.118910
2-(2-furanyl)-N-(2-oxolanylmethyl)-4-quinolinecarboxamideBacillus subtilisPotency1.258910
3-(4-methylphenyl)sulfonyl-1-(3-oxolanylmethyl)-2-pyrrolo[3,2-b]quinoxalinamineBacillus subtilisPotency12.589310
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideBacillus subtilisPotency35.481310
n-methylnandigerineBacillus subtilisPotency31.622810
2-(2,4-dioxo-3-phenyl-5-thiazolidinyl)-N-(3-methylphenyl)acetamideBacillus subtilisPotency35.481310
N-[(2-hydroxy-1-naphthalenyl)-(4-methylphenyl)methyl]cyclohexanecarboxamideBacillus subtilisPotency31.622810
1-[4-(6-bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]ethanoneBacillus subtilisPotency12.589310
N-[2-[5-[(4-tert-butylphenyl)methylthio]-1,3,4-oxadiazol-2-yl]phenyl]benzamideBacillus subtilisPotency28.183810
N-(4-fluorophenyl)-5-nitro-2-pyridinamineBacillus subtilisPotency3.981110
yl-109Bacillus subtilisPotency8.912510
3-ethyl-1-(2-furanylmethyl)-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]thioureaBacillus subtilisPotency28.183810
3-butan-2-yl-1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-phenylethyl)thioureaBacillus subtilisPotency19.952610
4-ethoxy-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-[(4-methoxyphenyl)methyl]benzamideBacillus subtilisPotency31.622810
3-(4-fluorophenyl)-1-[(6-oxo-5H-[1,3]dioxolo[4,5-g]quinolin-7-yl)methyl]-1-(thiophen-2-ylmethyl)ureaBacillus subtilisPotency31.622810
4-[3-(1,3-benzodioxol-5-ylmethylamino)-7-methyl-2-imidazo[1,2-a]pyridinyl]phenolBacillus subtilisPotency28.183810
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid [1-(cyclohexylamino)-1-oxopropan-2-yl] esterBacillus subtilisPotency3.548110
1-[3-[(7-cyano-[1,3]dioxolo[4,5-g]quinolin-6-yl)amino]propyl]-3-(3-methoxypropyl)thioureaBacillus subtilisPotency8.912510
1-[3-[(7-cyano-[1,3]dioxolo[4,5-g]quinolin-6-yl)amino]propyl]-3-(3-ethoxypropyl)thioureaBacillus subtilisPotency10.000010
[4-[5-tert-butyl-3-(phenylmethyl)-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneBacillus subtilisPotency31.622810
3-[(2-chlorophenyl)methyl]-7-[4-[4-(trifluoromethyl)phenyl]-1-piperazinyl]triazolo[4,5-d]pyrimidineBacillus subtilisPotency3.981110
7-(2-ethyl-1-piperidinyl)-5-methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidineBacillus subtilisPotency28.183810
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(4-methyl-2-thiazolyl)acetamideBacillus subtilisPotency7.943310
1-methyl-4-[2-oxo-2-(N-(phenylmethyl)anilino)ethyl]-5-pyrrolo[3,2-b]pyrrolecarboxylic acid propan-2-yl esterBacillus subtilisPotency28.183810
N-(2,4-dimethoxyphenyl)-2-[1-(3,4-dimethylphenyl)-4-oxo-5-pyrazolo[3,4-d]pyrimidinyl]acetamideBacillus subtilisPotency31.622810
2-[5-[[2-(3-methoxypropylamino)-2-oxoethyl]thio]-3-oxo-2H-imidazo[1,2-c]quinazolin-2-yl]-N-(phenylmethyl)acetamideBacillus subtilisPotency28.183810
3-(3,4-dimethoxyphenyl)-6,7-dimethoxy-2-methyl-N-(6-methyl-2-pyridinyl)-1-oxo-3,4-dihydroisoquinoline-4-carboxamideBacillus subtilisPotency7.079510
N-(4-methyl-5-oxo-2-[1]benzopyrano[4,3-b]pyridinyl)-4-(1-pyrrolidinylsulfonyl)benzamideBacillus subtilisPotency31.622810
N-(2,4-dimethoxyphenyl)-3-[[2-(2-methoxyphenoxy)-1-oxoethyl]amino]-2-benzofurancarboxamideBacillus subtilisPotency3.981110
N-[2-(2,4-dimethylphenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-1,3-benzodioxole-5-carboxamideBacillus subtilisPotency39.810710
N-(1,3-benzodioxol-5-yl)-3-methyl-6-phenyl-2-imidazo[2,1-b]thiazolecarboxamideBacillus subtilisPotency35.481310
2-[(2-methoxycarbonylanilino)-oxomethyl]-1-cyclohexanecarboxylic acidBacillus subtilisPotency28.183810
3-[[2-(4-fluorophenoxy)-1-oxoethyl]amino]-2-benzofurancarboxylic acid ethyl esterBacillus subtilisPotency39.810710
N-(2,4-dimethoxyphenyl)-3-[[2-furanyl(oxo)methyl]amino]-2-benzofurancarboxamideBacillus subtilisPotency29.732820
7-(4-methoxyphenyl)-5-methyl-2-(methylthio)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidineBacillus subtilisPotency2.511910
2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-(1-phenylethyl)acetamideBacillus subtilisPotency28.183810
N-[1-[(4-chlorophenyl)methyl]-5-methyl-3-pyrazolyl]-5-(3,4-dimethoxyphenyl)-3-isoxazolecarboxamideBacillus subtilisPotency25.118910
3-[2,4-dioxo-1-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl]-3-quinazolinyl]-N-(2-furanylmethyl)propanamideBacillus subtilisPotency14.125410
2-[[2-(4-ethoxyphenyl)-5-methyl-4-oxazolyl]methylthio]-N-(2-furanylmethyl)acetamideBacillus subtilisPotency15.848910
2-(2-methoxyphenyl)-1-oxo-N-[2-oxo-2-[4-(2-pyridinyl)-1-piperazinyl]ethyl]-4-isoquinolinecarboxamideBacillus subtilisPotency28.183810
N-(3-chlorophenyl)-2-[6,7-dimethoxy-2,4-dioxo-3-(2-oxolanylmethyl)-1-quinazolinyl]acetamideBacillus subtilisPotency31.622810
2,4-dioxo-3-pentyl-N-[3-(1-piperidinyl)propyl]-1H-quinazoline-7-carboxamideBacillus subtilisPotency28.183810
2-(2-methoxyethyl)-9-methyl-N-[3-(4-methyl-1-piperidinyl)propyl]-1-oxo-4-pyrido[3,4-b]indolecarboxamideBacillus subtilisPotency31.622810
1-(1-naphthalenyl)-3-[3-(1-pyrrolidinyl)propyl]ureaBacillus subtilisPotency11.220210
1-oxo-N-(3-pyridinyl)-2-benzopyran-4-carboxamideBacillus subtilisPotency25.118910
N-[2-(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)ethyl]-1-propanesulfonamideBacillus subtilisPotency28.183810
4-(1-methyl-3-indolyl)-N-propan-2-ylbutanamideBacillus subtilisPotency31.622810
4-[2-[(1'-acetyl-4-oxo-6-spiro[3,4-dihydro-2H-1-benzopyran-2,4'-piperidine]yl)oxy]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterBacillus subtilisPotency15.848910
N-[4-[5-[(2-methylphenoxy)methyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideBacillus subtilisPotency28.183810
2-[(3-oxo-2-propan-2-yl-2H-imidazo[1,2-c]quinazolin-5-yl)thio]-N-[2-(4-sulfamoylphenyl)ethyl]acetamideBacillus subtilisPotency31.622810
3-(4-bromophenyl)-4-(2-furanylmethyl)-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency19.952610
N-(3-chlorophenyl)-2-[1-(3,4-dimethylphenyl)-4-oxo-5-pyrazolo[3,4-d]pyrimidinyl]acetamideBacillus subtilisPotency25.118910
2-[[5-methyl-2-[4-(methylthio)phenyl]-4-oxazolyl]methylthio]-1-(4-morpholinyl)ethanoneBacillus subtilisPotency31.622810
2-(6-benzimidazolo[1,2-c]quinazolinylthio)-N-(2-furanylmethyl)acetamideBacillus subtilisPotency39.810710
1-[5-amino-3-(4-methoxyphenyl)-1,2,4-triazol-1-yl]-1-propanoneBacillus subtilisPotency35.481310
1,7,7-trimethyl-9-oxo-N-(2-oxolanylmethyl)-8H-furo[3,2-f][1]benzopyran-2-carboxamideBacillus subtilisPotency25.118910
2-(3-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneBacillus subtilisPotency31.622810
2-(pyridin-4-ylmethylamino)benzoic acidBacillus subtilisPotency14.125410
N-[2-(2,3-dimethylphenyl)-5,5-dioxo-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-2-methoxybenzamideBacillus subtilisPotency25.118910
5-(3,4-dimethoxyphenyl)-N-[1-[(2-methylphenyl)methyl]-4-pyrazolyl]-3-isoxazolecarboxamideBacillus subtilisPotency3.981110
4-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-6-(trifluoromethyl)pyrimidineBacillus subtilisPotency35.481310
5a,6,7,8,9,10-hexahydro-5H-azepino[2,1-b]quinazolin-12-oneBacillus subtilisPotency12.589310
2-cyclopentyl-4-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-9-methyl-1-pyrido[3,4-b]indoloneBacillus subtilisPotency3.162310
5-(dimethylamino)-2-phenyl-4-oxazolecarbonitrileBacillus subtilisPotency0.631010
3-pyridinecarboxylic acid 2-[[oxo-(2-oxo-1-benzopyran-3-yl)methyl]amino]ethyl esterBacillus subtilisPotency15.848910
N-[4-[[4-(2-fluorophenyl)-1-piperazinyl]-oxomethyl]-1-oxo-2-isoquinolinyl]-2-pyrazinecarboxamideBacillus subtilisPotency22.387210
2-(4-ethoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acidBacillus subtilisPotency28.183810
2-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methylthio]-3-pyridinecarboxylic acid propan-2-yl esterBacillus subtilisPotency14.125410
2,4-dioxo-3-(2-oxolanylmethyl)-N-pentyl-1H-quinazoline-7-carboxamideBacillus subtilisPotency17.782810
2-[[2-(3,4-dimethoxyphenyl)-5-methyl-4-oxazolyl]methylsulfinyl]-N-[3-(1-pyrrolidinyl)propyl]acetamideBacillus subtilisPotency15.848910
3-[[(3-methoxyphenyl)-oxomethyl]amino]-2-benzofurancarboxylic acid ethyl esterBacillus subtilisPotency31.622810
2-[(3-bromo-5,7-dimethyl-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzoxazoleBacillus subtilisPotency28.183810
N-ethyl-3-[4-morpholinyl(oxo)methyl]-4-oxo-N-phenyl-1H-quinoline-6-sulfonamideBacillus subtilisPotency31.622810
2-(2-methoxyethyl)-9-methyl-4-[(4-methyl-1-piperidinyl)-oxomethyl]-1-pyrido[3,4-b]indoloneBacillus subtilisPotency15.848910
2-(4-methyl-1-oxo-[1]benzothiolo[2,3-d]pyridazin-2-yl)propanoic acidBacillus subtilisPotency28.183810
7-methoxy-4,5-dihydro-2H-benzo[g]indazole-3-carboxylic acidBacillus subtilisPotency19.952610
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-(7-methoxy-2-furo[2,3-b]quinolinyl)methanoneBacillus subtilisPotency31.622810
2-ethyl-N-[2-(7-methoxy-2-oxo-1H-quinolin-3-yl)ethyl]butanamideBacillus subtilisPotency15.848910
3-methyl-N-[2-(4-morpholinyl)ethyl]-1-phenyl-5-thieno[2,3-c]pyrazolecarboxamideBacillus subtilisPotency28.183810
3-(2-chlorophenyl)-5-methyl-N-[3-(3-methyl-2-imidazo[1,2-a]pyrimidinyl)phenyl]-4-isoxazolecarboxamideBacillus subtilisPotency2.511910
N-[2-(7-methoxy-2-oxo-1H-quinolin-3-yl)ethyl]cyclopropanecarboxamideBacillus subtilisPotency17.782810
savirinBacillus subtilisPotency25.118910
4-[(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)methyl]-N-(3-methoxypropyl)-1-cyclohexanecarboxamideBacillus subtilisPotency8.912510
2-(2-methoxyethyl)-9-methyl-1-oxo-N-(thiophen-2-ylmethyl)-4-pyrido[3,4-b]indolecarboxamideBacillus subtilisPotency19.952610
2-chloro-6-[4-morpholinyl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneBacillus subtilisPotency17.782810
4-[[9-methyl-2-(2-methylpropyl)-1-oxo-4-pyrido[3,4-b]indolyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterBacillus subtilisPotency25.118910
5-(4-methoxyphenyl)-N-propan-2-yl-3-isoxazolecarboxamideBacillus subtilisPotency31.622810
N-(4-ethylphenyl)-5-(2-furanyl)-3-isoxazolecarboxamideBacillus subtilisPotency31.622810
N-(4-fluorophenyl)-6-methyl-1-propyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carboxamideBacillus subtilisPotency25.118910
N-(2-chlorophenyl)-5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-methyl-2-benzofurancarboxamideBacillus subtilisPotency39.810710
3-acetyl-6-methyl-1H-quinolin-4-oneBacillus subtilisPotency25.118910
N-[3-cyano-4-[4-(4-methoxyphenyl)-1-piperazinyl]phenyl]cyclohexanecarboxamideBacillus subtilisPotency28.183810
2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-(3-pyridinylmethyl)acetamideBacillus subtilisPotency19.952610
acetic acid [2-(1-acetyl-6-indolyl)-2-oxoethyl] esterBacillus subtilisPotency35.481310
1-[(5,7-dimethyl-3-pyrazolo[1,5-a]pyrimidinyl)-oxomethyl]-4-piperidinecarboxylic acid ethyl esterBacillus subtilisPotency31.622810
N-(2-furanylmethyl)-N'-[4-methyl-2-(4-methyl-1-piperazinyl)-6-quinolinyl]butanediamideBacillus subtilisPotency22.387210
3-[5-(4-fluorophenyl)-7-phenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-1-propanolBacillus subtilisPotency10.000010
N-(2,3-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideBacillus subtilisPotency39.810710
N-(3,4-dimethylphenyl)-5-(2-furanyl)-3-isoxazolecarboxamideBacillus subtilisPotency39.810710
3-(4-chlorophenyl)-2-(1-pyrrolidinyl)-4-quinazolinoneBacillus subtilisPotency22.387210
1-[(6-methoxy-2-furo[2,3-b]quinolinyl)-oxomethyl]-4-piperidinecarboxylic acid ethyl esterBacillus subtilisPotency17.782810
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamideBacillus subtilisPotency31.622810
N-cyclopentyl-4-(3,4-dimethoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinamineBacillus subtilisPotency35.481310
N-(3,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideBacillus subtilisPotency28.183810
3-[4-[2-(3,4-dimethoxyphenyl)-2-oxoethyl]-3-oxo-[1,2,4]triazino[2,3-a]benzimidazol-2-yl]propanoic acidBacillus subtilisPotency22.387210
N-[2-(dipropylamino)ethyl]-4-methyl-2-furo[3,2-c]quinolinecarboxamideBacillus subtilisPotency35.481310
N-(2-fluorophenyl)-3-[4-(2-fluorophenyl)-1-piperazinyl]propanamideBacillus subtilisPotency15.848910
4-[[3-[(2-furanylmethylamino)-oxomethyl]-7-methoxy-1-benzopyran-2-ylidene]amino]benzoic acidBacillus subtilisPotency19.952610
cyclopentanecarboxylic acid [4-(benzenesulfonyl)-2-tert-butyl-5-methyl-3-pyrazolyl] esterBacillus subtilisPotency11.220210
6-methoxy-N-(thiophen-2-ylmethyl)-2-furo[2,3-b]quinolinecarboxamideBacillus subtilisPotency3.981110
2-cyclohexyl-9-methyl-1-oxo-N-[3-(2-oxo-1-pyrrolidinyl)propyl]-4-pyrido[3,4-b]indolecarboxamideBacillus subtilisPotency14.125410
N-[2-(3,4-diethoxyphenyl)ethyl]-1-[6-(4-morpholinyl)-3-pyridazinyl]-4-piperidinecarboxamideBacillus subtilisPotency15.848910
N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamineBacillus subtilisPotency28.183810
LSM-28187Bacillus subtilisPotency15.848910
2,6-dimethyl-4-(4-phenyl-2-quinolinyl)morpholineBacillus subtilisPotency25.118910
8-[(1-ethyl-3-piperidinyl)thio]-1,3-dimethyl-6-sulfanylidene-7H-purin-2-oneBacillus subtilisPotency0.707910
3-(2-benzofuranyl)-N-(4-nitrophenyl)-1-phenyl-4-pyrazolecarboxamideBacillus subtilisPotency28.183810
2-[(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)thio]-N-(1,1-dioxo-3-thiolanyl)-N-ethylacetamideBacillus subtilisPotency15.848910
N-[4-(difluoromethoxy)phenyl]-4-(phenylmethyl)-1-piperazinecarbothioamideBacillus subtilisPotency8.912510
2-(trifluoromethyl)-3-imidazo[1,2-a]pyrimidinecarboxylic acid ethyl esterBacillus subtilisPotency25.118910
4-[3-(1,3-diphenyl-4-pyrazolyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-oxobutanoic acidBacillus subtilisPotency14.125410
N-[4-(methoxymethyl)-6-methyl-2-oxo-1H-quinolin-7-yl]cyclopropanecarboxamideBacillus subtilisPotency19.952610
3,3,3-trifluoro-2-[[(4-hydroxyanilino)-oxomethyl]amino]-2-phenylpropanoic acid ethyl esterBacillus subtilisPotency25.118910
2-[[[3-(2,5-dioxo-1-pyrrolidinyl)phenyl]-oxomethyl]amino]-4-(4-phenylphenyl)-3-thiophenecarboxylic acid ethyl esterBacillus subtilisPotency15.848910
N-[2-(4-morpholinyl)ethyl]-2-(4-propan-2-yloxyphenyl)-4-quinolinecarboxamideBacillus subtilisPotency22.387210
2-(4-benzofuro[3,2-d]pyrimidinylthio)-N-(3-methylphenyl)acetamideBacillus subtilisPotency31.622810
5-[3-[3-(4-methoxyphenyl)-1-phenyl-4-pyrazolyl]-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acidBacillus subtilisPotency28.183810
N-[2-(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)ethyl]-2-thiophenecarboxamideBacillus subtilisPotency19.952610
6-[4-oxo-2-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methylthio]-3-thieno[3,2-d]pyrimidinyl]hexanoic acidBacillus subtilisPotency31.622810
3-(4-benzoyl-1-piperazinyl)-1-(2-methylpropyl)-6,7-dihydro-5H-cyclopenta[c]pyridine-4-carbonitrileBacillus subtilisPotency31.622810
2-chloro-8-[4-morpholinyl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneBacillus subtilisPotency15.848910
2-[[2-[(2,5-dimethylphenyl)sulfonylamino]-1-oxoethyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideBacillus subtilisPotency31.622810
2-[2-[(5-chloro-2-thiophenyl)-oxomethyl]imino-6-fluoro-1,3-benzothiazol-3-yl]acetic acid methyl esterBacillus subtilisPotency28.183810
5-chloro-N-(1,3-dioxo-5-isoindolyl)-2-thiophenecarboxamideBacillus subtilisPotency3.981110
2-[[2-[3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]thio]acetic acid butyl esterBacillus subtilisPotency14.125410
6-[2-(1-azepanyl)-2-oxoethoxy]-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-oneBacillus subtilisPotency28.183810
2-[[7-(4-methoxyphenyl)-5-phenyl-4-pyrrolo[2,3-d]pyrimidinyl]thio]propanoic acid ethyl esterBacillus subtilisPotency25.118910
1-[(2,6-dichlorophenyl)methyl]-5-(4-methylphenyl)-2-oxo-3-pyridinecarbonitrileBacillus subtilisPotency7.079510
5-[2-[3-(4-fluorophenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]-2-(phenylmethyl)-3,4-dihydroisoquinolin-1-oneBacillus subtilisPotency15.848910
5-(4-ethoxyphenyl)-1,3-diphenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-4,6-dioneBacillus subtilisPotency11.220210
2-(4-methoxyphenyl)-N-[2-(4-morpholinyl)-5-(4-morpholinylsulfonyl)phenyl]-4-quinolinecarboxamideBacillus subtilisPotency28.183810
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideBacillus subtilisPotency31.622810
2-[(2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)oxy]-N-heptylacetamideBacillus subtilisPotency28.183810
N-(3-chlorophenyl)-5-oxo-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindole-1-carboxamideBacillus subtilisPotency15.848910
LSM-24581Bacillus subtilisPotency19.952610
1-bromo-3-(5,5-dimethyl-3-phenyl-4H-pyrazolo[4,3-a]carbazol-10-yl)-2-propanolBacillus subtilisPotency14.125410
N-methyl-5-phenyl-2-thiophenecarboxamideBacillus subtilisPotency15.415220
AnthraniloyllycoctonineBacillus subtilisPotency15.848910
5-tert-butyl-7-(4-ethyl-1-piperazinyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidineBacillus subtilisPotency35.481310
LSM-31277Bacillus subtilisPotency31.622810
4-(2-methylphenoxy)-6-phenylfuro[2,3-d]pyrimidineBacillus subtilisPotency31.622810
N-(2,2,2-trichloro-1-diethoxyphosphorylethyl)-1-naphthalenecarboxamideBacillus subtilisPotency25.118910
4-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-3-oxobutanoic acid ethyl esterBacillus subtilisPotency14.125410
1-[3-[(2-methoxyphenyl)sulfamoyl]-4-(1-piperidinyl)phenyl]-3-(3-methylphenyl)ureaBacillus subtilisPotency11.220210
N-[2-(2-chlorophenoxy)ethyl]-2-(1H-indol-3-yl)-2-oxoacetamideBacillus subtilisPotency25.118910
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(2-methoxy-4-methylphenyl)-2-thiophenecarboxamideBacillus subtilisPotency28.183810
N-(3,5-dichloro-2-pyridinyl)-2-[[1-(2-methoxyethyl)-2-benzimidazolyl]thio]propanamideBacillus subtilisPotency31.622810
6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylic acid [1-[1-[4-(difluoromethoxy)phenyl]-2,5-dimethyl-3-pyrrolyl]-1-oxopropan-2-yl] esterBacillus subtilisPotency19.952610
N-[4-[[(4-tert-butylphenyl)-oxomethyl]amino]phenyl]-2-furancarboxamideBacillus subtilisPotency31.622810
2-hydroxybenzoic acid [2-(2-ethoxyanilino)-2-oxo-1-phenylethyl] esterBacillus subtilisPotency39.810710
N-(2,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamideBacillus subtilisPotency3.981110
2-(1,3-benzoxazol-2-ylthio)-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneBacillus subtilisPotency14.125410
2-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-6,7,8,8a-tetrahydro-5H-imidazo[1,5-a]pyridine-1,3-dioneBacillus subtilisPotency31.622810
N-[3-[3-(1-piperidinylsulfonyl)anilino]-2-quinoxalinyl]benzenesulfonamideBacillus subtilisPotency25.118910
3-(4-methylphenyl)-N-[3-(4-morpholinylsulfonyl)phenyl]-1-phenyl-4-pyrazolecarboxamideBacillus subtilisPotency25.118910
4-(4-ethoxyphenyl)-1-(4-methoxyphenyl)-2-(methylthio)imidazoleBacillus subtilisPotency28.183810
N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)-2,3-dihydro-1,4-benzodioxin-6-carboxamideBacillus subtilisPotency12.589310
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneBacillus subtilisPotency28.183810
3-(2-methoxyphenyl)-2,5-dimethyl-7-[4-(phenylmethyl)-1-piperazinyl]pyrazolo[1,5-a]pyrimidineBacillus subtilisPotency35.481310
3-(1,5-dimethyl-3-pyrazolyl)-4-phenyl-1H-1,2,4-triazole-5-thioneBacillus subtilisPotency31.622810
2-(2-bromophenyl)-3-[3-(4-morpholinyl)propyl]-1,2-dihydroquinazolin-4-oneBacillus subtilisPotency35.481310
2-(2-furanylmethylamino)benzoic acid [2-[(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-2-oxoethyl] esterBacillus subtilisPotency12.589310
N-[4-(1H-benzimidazol-2-yl)phenyl]-3-(2,5-dioxo-1-pyrrolidinyl)benzamideBacillus subtilisPotency39.810710
6-benzoyl-2-phenyl-5-(trifluoromethyl)-3-pyridazinoneBacillus subtilisPotency31.622810
1-(4-methylphenyl)-2-[(1-phenyl-2-imidazolyl)thio]ethanoneBacillus subtilisPotency28.183810
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterBacillus subtilisPotency25.118910
1-(4-methoxyphenyl)-N-(2-oxolanylmethyl)-4-pyrazolo[3,4-d]pyrimidinamineBacillus subtilisPotency31.622810
1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)-2-[(6-methyl-2-nitro-3-pyridinyl)oxy]ethanoneBacillus subtilisPotency3.981110
4-[(7-methyl-2-phenyl-3-imidazo[1,2-a]pyridinyl)methyl]morpholineBacillus subtilisPotency22.387210
4-(2,5-dioxo-1-pyrrolidinyl)-N-[4-(4-methoxyphenyl)-2-thiazolyl]benzamideBacillus subtilisPotency28.183810
2-[[[5-(2-fluoroanilino)-1,3,4-thiadiazol-2-yl]thio]methyl]isoindole-1,3-dioneBacillus subtilisPotency28.183810
1-(2-methoxy-3-dibenzofuranyl)-3-(3-methylphenyl)thioureaBacillus subtilisPotency11.220210
2-(3-oxo-4H-1,4-benzothiazin-2-yl)acetic acid (7-methoxy-2-oxo-1-benzopyran-4-yl)methyl esterBacillus subtilisPotency19.952610
1-[(7-chloro-4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl]-3-(3-fluoro-4-methylphenyl)thieno[3,2-d]pyrimidine-2,4-dioneBacillus subtilisPotency11.220210
4-(1,3-dioxo-2-benzo[de]isoquinolinyl)butanoic acid [2-(2-acetylanilino)-2-oxoethyl] esterBacillus subtilisPotency39.810710
2-(4-chlorophenoxy)-N-(2-thiophen-2-yl-3-imidazo[1,2-a]pyridinyl)acetamideBacillus subtilisPotency28.183810
5-(2-chlorophenyl)-N-(4-methoxyphenyl)-2-furancarboxamideBacillus subtilisPotency39.810710
3-chloro-N-[3-(2-methoxyethyl)-6-sulfamoyl-1,3-benzothiazol-2-ylidene]-1-benzothiophene-2-carboxamideBacillus subtilisPotency22.387210
3-amino-4-[(4-chlorophenyl)thio]benzoic acid methyl esterBacillus subtilisPotency25.118910
N-[2,5-diethoxy-4-(4-morpholinyl)phenyl]-4-[(3,5-dimethyl-4-isoxazolyl)methoxy]-3-methoxybenzamideBacillus subtilisPotency11.220210
4-(4-propan-2-ylphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazolin-2-oneBacillus subtilisPotency28.183810
LSM-31434Bacillus subtilisPotency31.622810
2-bromo-6-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-11-pyrido[2,1-b]quinazolinoneBacillus subtilisPotency8.912510
LSM-16483Bacillus subtilisPotency7.079510
2-[2-[(3-chloro-1-benzothiophen-2-yl)-oxomethyl]imino-6-sulfamoyl-1,3-benzothiazol-3-yl]acetic acid ethyl esterBacillus subtilisPotency14.125410
2-(4-bromophenyl)-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterBacillus subtilisPotency31.622810
2-[[2-(4-ethoxy-3-methoxyphenyl)-4-thiazolyl]methylthio]-5-methyl-1,3,4-thiadiazoleBacillus subtilisPotency25.118910
8-(4-methoxyphenyl)-7-methyl-3-(phenylmethyl)purine-2,6-dioneBacillus subtilisPotency35.481310
N-(4,5-dithiophen-2-yl-2-thiazolyl)-2-methyl-1-cyclopropanecarboxamideBacillus subtilisPotency19.952610
N-(3-chloro-4-fluorophenyl)-2-[5-(dimethylsulfamoyl)-2-(ethylamino)anilino]acetamideBacillus subtilisPotency39.810710
3-methoxy-N-[2-(4-methoxyphenyl)-2-(1-pyrrolidinyl)ethyl]-2-naphthalenecarboxamideBacillus subtilisPotency10.000010
2-[[oxo-(1-oxo-3,4-dihydro-1H-2-benzopyran-3-yl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterBacillus subtilisPotency39.810710
5-(4-methylphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acidBacillus subtilisPotency3.162310
1-(4-carbamoyl-2-nitrophenyl)-4-piperidinecarboxylic acid methyl esterBacillus subtilisPotency35.481310
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(4-methoxyphenyl)-2-thiophenecarboxamideBacillus subtilisPotency31.622810
N-[2-(4-methoxyphenyl)-4-oxo-1,2-dihydroquinazolin-3-yl]carbamic acid ethyl esterBacillus subtilisPotency31.622810
N-(3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(2-chlorophenyl)-5-methyl-4-isoxazolecarboxamideBacillus subtilisPotency31.622810
2-(3-methyl-1-oxo-2-isoquinolinyl)-N-(3,4,5-trimethoxyphenyl)acetamideBacillus subtilisPotency16.082510
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideBacillus subtilisPotency39.810710
4-(3,4-dimethoxyphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazoline-2-thioneBacillus subtilisPotency15.848910
N-[bis(methylthio)methylideneamino]-4-hydroxybenzamideBacillus subtilisPotency28.183810
N-(5,5-dimethyl-7-oxo-4,6-dihydro-1,3-benzothiazol-2-yl)-2-(2,5-dioxo-1-pyrrolidinyl)acetamideBacillus subtilisPotency31.622810
2-[3-(1-benzotriazolylmethyl)-4-methoxyphenyl]-3-(4-methoxyphenyl)-1,2-dihydroquinazolin-4-oneBacillus subtilisPotency31.622810
trans-2,3',4,5'-tetrahydroxystilbeneBacillus subtilisPotency25.118910
3-(4-chlorophenyl)-N-cyclopropyl-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideBacillus subtilisPotency14.125410
2-[[oxo-(5-propyl-3-isoxazolyl)methyl]amino]benzoic acid methyl esterBacillus subtilisPotency39.810710
N-(6-acetyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenyl-3-pyrazolecarboxamideBacillus subtilisPotency2.511910
3-(4-fluorophenyl)-6-(1-pyrrolidinyl)-[1,2,4]triazolo[4,3-b]pyridazineBacillus subtilisPotency39.810710
N-(6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamideBacillus subtilisPotency35.481310
N-(2-ethoxyphenyl)-[1,2,4]triazolo[4,3-a]quinoxalin-4-amineBacillus subtilisPotency12.589310
N-[2-(2-imidazo[1,2-a]pyridinyl)ethyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideBacillus subtilisPotency14.125410
7-hydroxy-8-(4-morpholinylmethyl)-3-phenyl-1-benzopyran-4-oneBacillus subtilisPotency3.162310
3-[6-[4-(trifluoromethoxy)anilino]-4-pyrimidinyl]benzamideBacillus subtilisPotency35.481310
bornyl ferulateBacillus subtilisPotency31.622810
thunberginol aBacillus subtilisPotency31.622810
3,5-dimethoxycinnamic acidBacillus subtilisPotency31.622810
erbstatinBacillus subtilisPotency22.387210
4-methyl-2,7-diphenyl-8H-pyrido[2,3-d]pyrimidin-5-oneBacillus subtilisPotency39.810710
5-deazaflavinBacillus subtilisPotency3.548110
urolithin bBacillus subtilisPotency39.810710
2-(5,7-dihydroxy-4-methyl-2-oxo-1-benzopyran-3-yl)acetic acid ethyl esterBacillus subtilisPotency25.118910
6-ethyl-7-hydroxy-4-[[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-1-benzopyran-2-oneBacillus subtilisPotency14.125410
6-bromo-5-methyl-1,3-dihydroimidazo[4,5-b]pyridine-2-thioneBacillus subtilisPotency10.000010
8-(diethylaminomethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-7-hydroxy-1-benzopyran-4-oneBacillus subtilisPotency28.183810
b 43Bacillus subtilisPotency28.183810
(8R)-7-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triolBacillus subtilisPotency28.183810
(8R)-7-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triolBacillus subtilisPotency25.118910
mrs 1754Bacillus subtilisPotency12.589310
N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-8-methyl-4-oxo-2-thieno[3,2-c][1]benzopyrancarboxamideBacillus subtilisPotency15.848910
2-(2-furanyl)-N-phenyl-3-imidazo[1,2-a]pyridinamineBacillus subtilisPotency25.118910
4-[3-[(3-chloro-4-fluoroanilino)-oxomethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid tert-butyl esterBacillus subtilisPotency8.912510
N-(4-ethoxyphenyl)-1,5-dimethyl-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamideBacillus subtilisPotency39.810710
LSM-32377Bacillus subtilisPotency3.162310
6-fluoro-N-phenyl-1,3-benzothiazol-2-amineBacillus subtilisPotency11.220210
4-fluoro-N-(4-fluoro-1,3-benzothiazol-2-yl)-1,3-benzothiazol-2-amineBacillus subtilisPotency8.912510
N-(6-fluoro-1,3-benzothiazol-2-yl)-6,7-dihydro-[1,4]dioxino[2,3-f][1,3]benzothiazol-2-amineBacillus subtilisPotency5.081620
N-[5-[(2-methylphenyl)methylthio]-1,3,4-thiadiazol-2-yl]-2-thiophen-2-ylacetamideBacillus subtilisPotency39.810710
2-[[6-(2-furanyl)-3-pyridazinyl]thio]-N-(3-methylphenyl)acetamideBacillus subtilisPotency28.183810
3-butyl-10-phenylpyrimido[4,5-b]quinoline-2,4-dioneBacillus subtilisPotency25.118910
N-[2-(3-methoxyphenyl)-4-[(4-methoxyphenyl)methoxy]-6-quinolinyl]-3-pyridinecarboxamideBacillus subtilisPotency28.183810
N-ethyl-8-methyl-4-oxo-N-(phenylmethyl)-2-thieno[3,2-c][1]benzopyrancarboxamideBacillus subtilisPotency17.782810
N-[3-(4-morpholinyl)propyl]-2,4-dioxo-3-(2-phenylethyl)-1H-quinazoline-7-carboxamideBacillus subtilisPotency14.125410
N-[2-methyl-5-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-phenoxyacetamideBacillus subtilisPotency31.622810
8-methyl-N-[(4-methylphenyl)methyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-amineBacillus subtilisPotency31.622810
1-(3,4-dimethylphenyl)-2,5-dioxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarbonitrileBacillus subtilisPotency2.511910
6-[(2-fluorophenyl)methyl]-5-methyl-N-(3-methylbutyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamideBacillus subtilisPotency28.183810
1'-acetyl-6-[2-(4-ethyl-1-piperazinyl)-2-oxoethoxy]-4-spiro[3,4-dihydro-2H-1-benzopyran-2,4'-piperidine]oneBacillus subtilisPotency31.622810
3-(2-methoxyethyl)-2,4-dioxo-N-pentyl-1H-quinazoline-7-carboxamideBacillus subtilisPotency31.622810
3-methoxy-5-pyridin-2-ylethynylpyridineBacillus subtilisPotency17.782810
calcimycinBacillus subtilisPotency27.282410
N-[5-[2-(2-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]heptanamideBacillus subtilisPotency14.125410
N-butyl-N-methyl-4-[(2-methyl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)hydrazo]-4-oxobutanamideBacillus subtilisPotency25.118910
2-[6,7-dimethoxy-3-(3-methoxyphenyl)-2,4-dioxo-1-quinazolinyl]-N-(5-methyl-1H-pyrazol-3-yl)acetamideBacillus subtilisPotency28.183810
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamideBacillus subtilisPotency3.981110
4-[3-(3-fluorophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamideBacillus subtilisPotency3.162310
N-[2-methyl-5-(2-thiazolo[5,4-b]pyridinyl)phenyl]-5,6,7,8-tetrahydronaphthalene-2-sulfonamideBacillus subtilisPotency22.387210
2-[[5-(2-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-N-(2-nitrophenyl)acetamideBacillus subtilisPotency31.622810
1-[(4-methylphenyl)methyl]-2,4-dioxo-N-(phenylmethyl)-3-prop-2-enyl-7-quinazolinecarboxamideBacillus subtilisPotency39.810710
2-(8-methoxy-4-methyl-1-oxo-[1,2,4]triazino[4,5-a]indol-2-yl)-N-(3-propan-2-yloxypropyl)acetamideBacillus subtilisPotency2.818410
N-(4-ethyl-1,2,5-oxadiazol-3-yl)-3,5,6-trimethyl-2-benzofurancarboxamideBacillus subtilisPotency22.387210
1-(1,5-dimethyl-3-pyrazolyl)-N-[[5-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl]methanamineBacillus subtilisPotency14.125410
N-[5-[[2-(2-furanylmethylamino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-1,3-benzodioxole-5-carboxamideBacillus subtilisPotency4.466810
2-[[6-(4-ethylphenyl)-3-pyridazinyl]thio]-N-(2-oxolanylmethyl)acetamideBacillus subtilisPotency39.810710
3-chloro-N-propan-2-yl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideBacillus subtilisPotency25.118910
5-[2-(4-chlorophenyl)-4-methyl-5-thiazolyl]-3-(3-fluorophenyl)-5-methyl-4H-isoxazoleBacillus subtilisPotency15.848910
3-(4-bromophenyl)-N-[5-[[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)anilino]-oxomethyl]-2-methylphenyl]-1H-pyrazole-5-carboxamideBacillus subtilisPotency31.622810
8-[1-(1,3-benzodioxol-5-yl)-3-(4-phenyl-1-piperazinyl)propyl]-5,7-dimethoxy-4-methyl-1-benzopyran-2-oneBacillus subtilisPotency31.622810
5,7-dimethoxy-8-[1-(4-methoxyphenyl)-3-(3-methyl-1-piperidinyl)-3-oxopropyl]-4-phenyl-1-benzopyran-2-oneBacillus subtilisPotency35.481310
8-{1-[4-(dimethylamino)phenyl]-3-(pyrrolidin-1-yl)propyl}-5,7-dimethoxy-4-pentyl-2H-chromen-2-oneBacillus subtilisPotency17.782810
3-(2-hydroxy-4,6-dimethoxyphenyl)-3-(4-methoxyphenyl)-1-(3-methyl-1-piperidinyl)-1-propanoneBacillus subtilisPotency3.981110
(3R,3aS,7R,7aS)-3-[5-(1-benzothiophen-2-yl)-2-methoxyphenyl]-7-methyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneBacillus subtilisPotency10.000010
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esterBacillus subtilisPotency25.118910
(2S)-2-[[[4-[(3-methylanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-3-phenylpropanoic acid (phenylmethyl) esterBacillus subtilisPotency25.118910
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterBacillus subtilisPotency39.810710
reserpic acid, hydrochloride salt, (3beta,16beta,17alpha,18beta,20alpha)-isomerBacillus subtilisPotency28.183810
amorfrutin aBacillus subtilisPotency25.118910
sri 62320Bacillus subtilisPotency11.220210
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl esterBacillus subtilisPotency39.810710
[2-(2-methoxyethyl)-1-piperidinyl]-[5-[[4-(1,2,4-triazol-1-yl)phenoxy]methyl]-3-isoxazolyl]methanoneBacillus subtilisPotency44.668410
4-[(6-chloro-1H-benzimidazol-2-yl)amino]benzoic acidBacillus subtilisPotency31.622810
4-(4-acetyloxyphenyl)benzoic acid [2-[[2-(2-chloroanilino)-2-oxoethyl]-methylamino]-2-oxoethyl] esterBacillus subtilisPotency11.220210
3-cyclohexyl-1-[[(2S,3R)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-10-[[oxo-(propan-2-ylamino)methyl]amino]-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methylureaBacillus subtilisPotency28.183810
N-[(2R,3S)-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[(1-naphthalenylamino)-oxomethyl]amino]methyl]-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-2-phenylacetamideBacillus subtilisPotency25.118910
5-(2,5-dichlorophenyl)-N-(2,6-diethylphenyl)-2-furancarboxamideBacillus subtilisPotency50.118710
4-hydroxy-1-methyl-3-(phenylthio)-1,2-dihydroquinolin-2-oneBacillus subtilisPotency19.952610
N-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-1-prop-2-enyl-3-quinolinecarboxamideBacillus subtilisPotency28.183810
LSM-23565Bacillus subtilisPotency31.622810
chlortetracycline hydrochlorideBacillus subtilisPotency15.848910
N-(4-hydroxy-2-oxo-1H-quinolin-3-yl)heptanamideBacillus subtilisPotency25.118910
2-(4-hydroxy-2-oxo-1H-quinolin-3-yl)acetic acid propyl esterBacillus subtilisPotency25.118910
N-(4-hydroxy-2-oxo-1H-quinolin-3-yl)pentanamideBacillus subtilisPotency28.183810
2-(4-hydroxy-2-oxo-1H-quinolin-3-yl)acetic acid pentyl esterBacillus subtilisPotency15.848910
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-[4-oxo-2-(phenylmethyl)-3-quinazolinyl]-5,6,7,8-tetrahydroquinoline-3-carboxamideBacillus subtilisPotency3.548110
4-hydroxy-2-oxo-1-pentyl-N-(2-pyridinylmethyl)-3-quinolinecarboxamideBacillus subtilisPotency28.183810
N-[2-(4-chlorophenyl)ethyl]-4-hydroxy-2-oxo-1-propyl-3-quinolinecarboxamideBacillus subtilisPotency28.183810
ganciclovirBacillus subtilisPotency0.707910
suptopin 2Bacillus subtilisPotency28.183810
ImidazosagatriazinoneBacillus subtilisPotency19.952610
1-[amino-[(6-methoxy-4-methyl-2-quinazolinyl)amino]methylidene]-3-phenylureaBacillus subtilisPotency14.125410
4-oxo-2-(trifluoromethyl)-1H-quinazoline-6-carboxylic acid ethyl esterBacillus subtilisPotency3.981110
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-6-methyl-1H-pyrimidin-4-oneBacillus subtilisPotency28.183810
1-cyclopentyl-1-[(4-oxo-1H-quinazolin-2-yl)methyl]-3-(phenylmethyl)ureaBacillus subtilisPotency14.125410
pyridoxal 4-methoxybenzoyl hydrazoneBacillus subtilisPotency8.912510
4-methyl-3-phenyl-1,2-dihydropyrazolo[3,4-b]pyridin-6-oneBacillus subtilisPotency25.118910
LSM-20825Bacillus subtilisPotency28.183810
5,5-diethyl-2-(2-hydroxyethylamino)-1,6-dihydrobenzo[h]quinazolin-4-oneBacillus subtilisPotency6.309610