Proteins > 5-hydroxytryptamine receptor 3A
Page last updated: 2024-08-07 12:45:32

5-hydroxytryptamine receptor 3A

[no definition available]

Synonyms

5-HT3-A;
5-HT3A;
5-hydroxytryptamine receptor 3;
5-HT-3;
5-HT3R;
Serotonin receptor 3A;
Serotonin-gated ion channel receptor

Research

Bioassay Publications (9)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (44.44)29.6817
2010's3 (33.33)24.3611
2020's2 (22.22)2.80

Compounds (12)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
granisetronCavia porcellus (domestic guinea pig)Ki0.004011
quipazineCavia porcellus (domestic guinea pig)Ki6.667023
aripiprazoleCavia porcellus (domestic guinea pig)IC50630.000011
3-(1-methyl-1,2,3,6-tetrahydropyrid-4-yl)indoleCavia porcellus (domestic guinea pig)IC500.690011
trichostatin aCavia porcellus (domestic guinea pig)IC507.690011
2-(1-(2-allylphenoxy)ethyl)-4,5-dihydro-1h-imidazoleCavia porcellus (domestic guinea pig)Ki0.085111
clozapineCavia porcellus (domestic guinea pig)IC50110.000011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
clonidineCavia porcellus (domestic guinea pig)EC500.008311
ondansetronCavia porcellus (domestic guinea pig)Kd0.077611
benziodaroneCavia porcellus (domestic guinea pig)Kd8.000011
3-cyano-4-phenyl-6-(3-bromo-6-hydroxyphenyl)-2-pyridoneCavia porcellus (domestic guinea pig)Kd5.000011
3-methoxy-n-p-tolylquinoxalin-2-carboxamideCavia porcellus (domestic guinea pig)Kd0.050111