Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
5-(n,n-hexamethylene)amiloride | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
3-(2'-aminobenzhydryloxy)tropane | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
amoxapine | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
brimonidine | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
nonivamide | Homo sapiens (human) | Potency | 0.0866 | 2 | 0 |
ebselen | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
haloperidol | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
perphenazine | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
promethazine hydrochloride | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
quinacrine monohydrochloride | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
imipramine hydrochloride | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
pargyline hydrochloride | Homo sapiens (human) | Potency | 3.5481 | 1 | 0 |
amitriptyline hydrochloride | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
cyproheptadine hydrochloride (anhydrous) | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
cyclobenzaprine hydrochloride | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
propionylpromazine hydrochloride | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
metergoline | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
captopril | Homo sapiens (human) | Potency | 5.0119 | 1 | 0 |
salmeterol xinafoate | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
propranolol hydrochloride | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
u 37883a | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
desipramine hydrochloride | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
siquil | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
ay-20694 | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
sanguinarine chloride | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
opipramol hydrochloride | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
5-(n-methyl-n-isobutyl)amiloride | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
amperozide hydrochloride | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
u 78517f | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
ml 9 | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
memantine hydrochloride | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
6-bromoindirubin-3'-oxime | Homo sapiens (human) | Potency | 4.4668 | 1 | 0 |
ketoconazole | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
4-Morpholinyl(4-pentylcyclohexyl)methanone | Homo sapiens (human) | Potency | 0.2864 | 2 | 0 |
2-(2-methoxyphenyl)-1H-indole | Homo sapiens (human) | Potency | 0.0129 | 1 | 0 |
5-bromo-N-(pyridin-4-ylmethyl)-2-thiophenesulfonamide | Homo sapiens (human) | Potency | 5.0807 | 1 | 0 |
4-[[[(2-methoxyphenyl)methylamino]-oxomethyl]amino]benzoic acid ethyl ester | Homo sapiens (human) | Potency | 40.5608 | 2 | 0 |
N-(4-methylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Homo sapiens (human) | Potency | 0.2400 | 2 | 0 |
N-(1,3-benzodioxol-5-yl)-6-methyl-2-(2-pyridinyl)-4-quinolinecarboxamide | Homo sapiens (human) | Potency | 0.4118 | 2 | 0 |
N-(4-methylphenyl)-4-benzofuro[3,2-d]pyrimidinamine | Homo sapiens (human) | Potency | 0.1131 | 2 | 0 |
3-[5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazol-2-yl]-1-(phenylmethyl)-2-pyridinone | Homo sapiens (human) | Potency | 22.6947 | 1 | 0 |
capsaicin | Homo sapiens (human) | Potency | 0.0433 | 3 | 0 |
4-(4-chlorophenoxy)-1-(1-piperidinyl)-1-butanone | Homo sapiens (human) | Potency | 1.8273 | 1 | 0 |
N-(3,4-dichlorophenyl)-2-[4-(4-methoxyphenyl)-1-oxo-2-phthalazinyl]acetamide | Homo sapiens (human) | Potency | 5.7785 | 1 | 0 |
1-(1,3-benzodioxol-5-ylmethylthio)-[1,2,4]triazolo[4,3-a]quinoline | Homo sapiens (human) | Potency | 102.7570 | 1 | 0 |
1-(4-acetyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-[[4-(difluoromethoxy)-3-methoxyphenyl]methyl-methylamino]ethanone | Homo sapiens (human) | Potency | 102.7570 | 1 | 0 |
N-[2-(4-tert-butylphenoxy)ethyl]-2-(4-fluorophenyl)acetamide | Homo sapiens (human) | Potency | 0.1352 | 2 | 0 |
3-(diethylsulfamoyl)benzoic acid [2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 18.0271 | 1 | 0 |
1-(4-tert-butylphenyl)-3-(3-pyridinylmethyl)thiourea | Homo sapiens (human) | Potency | 2.8482 | 2 | 0 |
5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamide | Homo sapiens (human) | Potency | 2.1754 | 2 | 0 |
N-(3,4-dimethylphenyl)-3-[(4-fluorophenyl)methyl]-1,3-diazinane-1-carboxamide | Homo sapiens (human) | Potency | 51.5007 | 1 | 0 |
2-methyl-1-phenyl-5-benzimidazolecarboxylic acid [2-(2-methoxyanilino)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 0.1028 | 1 | 0 |
N-(3-{[2-(2-fluorophenyl)quinazolin-4-yl]amino}phenyl)acetamide | Homo sapiens (human) | Potency | 4.4027 | 2 | 0 |
trimipramine maleate | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
5-hydroxy-7-(4-hydroxy-3-methoxyphenyl)-1-phenyl-3- heptanone | Homo sapiens (human) | Potency | 1.2184 | 2 | 0 |
ag 112 | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
semaxinib | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
bay 11-7085 | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
nylidrin hydrochloride | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
triprolidine hydrochloride anhydrous | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
sinequan | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
zimelidine hydrochloride | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
atomoxetine | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
4-chloro-N-(4-ethylphenyl)-3-methyl-5-isoxazolecarboxamide | Homo sapiens (human) | Potency | 2.0164 | 2 | 0 |
fluvoxamine maleate | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
octoclothepine maleate | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
2-(n-phenethyl-n-propyl)amino-5-hydroxytetralin hydrochloride | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
dafadine B | Homo sapiens (human) | Potency | 2.7436 | 2 | 0 |
3-(2-hydroxy-4,6-dimethoxyphenyl)-3-(4-methoxyphenyl)-1-(3-methyl-1-piperidinyl)-1-propanone | Homo sapiens (human) | Potency | 4.0908 | 1 | 0 |
mls002174161 | Homo sapiens (human) | Potency | 0.7135 | 2 | 0 |
clozapine | Homo sapiens (human) | Potency | 12.5893 | 1 | 0 |
1-hydroxyphenazine | Homo sapiens (human) | Potency | 2.8961 | 1 | 0 |