Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
bithionol | Homo sapiens (human) | IC50 | 58.6741 | 2 | 0 |
hexachlorophene | Homo sapiens (human) | IC50 | 0.0983 | 1 | 0 |
phentolamine | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
metoclopramide hydrochloride | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
benserazide hydrochloride | Homo sapiens (human) | IC50 | 3.0540 | 1 | 0 |
methyldopa | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-benzoylanthranilic acid | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
gossypol acetic acid | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
2-[[5-[[2-(3-chloroanilino)-4-thiazolyl]methyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]thio]acetic acid methyl ester | Homo sapiens (human) | IC50 | 16.9870 | 1 | 0 |
Thieno[3,2-b]thiophene-2-carboxylic acid | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
(3aR,6aS)-3-(2-chlorophenyl)-5-(2,5-dimethoxyphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dione | Homo sapiens (human) | IC50 | 26.2452 | 2 | 0 |
2-(2,3-dihydroindol-1-yl)-N,N-dimethylethanamine | Homo sapiens (human) | IC50 | 0.0579 | 1 | 0 |
N-[4-(4-morpholinyl)phenyl]-2-thiophenesulfonamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
4-[(4-chlorophenyl)thio]-5-methyl-2-phenyl-1H-pyrazol-3-one | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
1-(2-methylpropyl)-2-thiophen-2-ylbenzimidazole | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-(1,3-benzodioxol-5-yl)-6-bromo-2-pyrazolo[1,5-a]pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 0.0230 | 1 | 0 |
N-(2-furanylmethyl)-2-imino-5-oxo-1-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 50.0000 | 2 | 0 |
N-cyclohexyl-2-[(8-methoxy-6-oxo-3-benzo[c][1]benzopyranyl)oxy]acetamide | Homo sapiens (human) | IC50 | 28.7540 | 2 | 0 |
cinnarizine | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
2-[3-(2-furanylmethyl)-2,4-dioxo-6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-b]pyrimidin-1-yl]acetamide | Homo sapiens (human) | IC50 | 0.0230 | 1 | 0 |
2-(2-furanyl)-4-quinolinecarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-[4-(dibutylsulfamoyl)phenyl]-2-thiophen-2-ylacetamide | Homo sapiens (human) | IC50 | 9.9232 | 2 | 0 |
benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 2.9453 | 2 | 0 |
2-[[5-(2-fluoroanilino)-1,3,4-thiadiazol-2-yl]thio]-N-(2-furanylmethyl)acetamide | Homo sapiens (human) | IC50 | 6.9080 | 2 | 0 |
5-cyclopentylidene-2-sulfanylidene-4-thiazolidinone | Homo sapiens (human) | IC50 | 25.1202 | 2 | 0 |
2-[[2-(4-ethyl-4-methyl-2,5-dioxo-1-imidazolidinyl)-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamide | Homo sapiens (human) | IC50 | 0.0325 | 1 | 0 |
2-[[5-[(2-fluorophenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-N-[(2-furanylmethylamino)-oxomethyl]acetamide | Homo sapiens (human) | IC50 | 34.4232 | 2 | 0 |
5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylic acid [2-[(1,1-dioxo-3-thiolanyl)-(2-methylpropyl)amino]-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 1.9230 | 2 | 0 |
2-(2-furanyl)-N-(2-oxolanylmethyl)-4-quinolinecarboxamide | Homo sapiens (human) | IC50 | 26.4051 | 1 | 0 |
1-[4-[(4-ethyl-1-piperazinyl)methyl]phenyl]-3-thiophen-2-ylurea | Homo sapiens (human) | IC50 | 0.4104 | 1 | 0 |
5-(1-ethyl-3-methyl-4-pyrazolyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxylic acid | Homo sapiens (human) | IC50 | 3.4145 | 1 | 0 |
5-hydroxy-2-methyl-4-[1-piperidinyl(3-pyridinyl)methyl]-3-benzo[g]benzofurancarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinol | Homo sapiens (human) | IC50 | 2.3924 | 1 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-3-yl)-3-(phenoxymethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole | Homo sapiens (human) | IC50 | 25.0115 | 2 | 0 |
morin | Homo sapiens (human) | IC50 | 2.9272 | 1 | 0 |
4-[[[2-(4-methoxyphenyl)-3-oxo-1H-isoindol-4-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-[4-[(4-methyl-1-piperidinyl)methyl]phenyl]-1-[5-(1-pyrrolyl)-1,3,4-thiadiazol-2-yl]-4-piperidinecarboxamide | Homo sapiens (human) | IC50 | 1.1036 | 1 | 0 |
2-methyl-5-[(2-oxo-1H-benzo[cd]indol-6-yl)sulfonylamino]-3-benzofurancarboxylic acid butyl ester | Homo sapiens (human) | IC50 | 13.5106 | 1 | 0 |
tetracycline | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
demeclocycline hydrochloride | Homo sapiens (human) | IC50 | 0.0614 | 1 | 0 |
4-[[2-[(6-methyl-4-oxo-1H-pyrimidin-2-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl ester | Homo sapiens (human) | IC50 | 0.0230 | 1 | 0 |