Proteins > Chain A, BCL-2-RELATED PROTEIN A1
Page last updated: 2024-08-07 15:08:50

Chain A, BCL-2-RELATED PROTEIN A1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (76)

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
fluconazoleHomo sapiens (human)EC50350.000010
isoconazoleHomo sapiens (human)EC50350.000010
phenprobamateHomo sapiens (human)EC50350.000010
2-fluoroadenosineHomo sapiens (human)EC50350.000010
acetylsalicylsalicylic acidHomo sapiens (human)EC50350.000010
cladribineHomo sapiens (human)EC50350.000010
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazineHomo sapiens (human)EC50350.000010
dv 1006Homo sapiens (human)EC50350.000010
imidazolidinyl ureaHomo sapiens (human)EC50350.000010
closantelHomo sapiens (human)EC50350.000010
sotalol hydrochlorideHomo sapiens (human)EC50350.000010
anisomycinHomo sapiens (human)EC50350.000010
aromaticinHomo sapiens (human)EC50350.000010
angustibalinHomo sapiens (human)EC50350.000010
oleic acidHomo sapiens (human)EC50350.000010
idarubicin hydrochlorideHomo sapiens (human)EC50350.000010
isoliquiritigeninHomo sapiens (human)EC50350.000010
3-[[2-(4-methyl-1-piperazinyl)-1-oxoethyl]amino]-2-benzofurancarboxylic acid ethyl esterHomo sapiens (human)EC50350.000010
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterHomo sapiens (human)EC50350.000010
1-methyl-4-[(4-methylphenyl)thio]-3-nitro-2-quinolinoneHomo sapiens (human)EC50188.600010
4-[[4-(2,5-dimethylphenyl)-1-piperazinyl]methyl]-2-methoxyphenolHomo sapiens (human)EC5098.590010
2,5-dimethyl-1-(phenylmethyl)pyrrole-3,4-dicarboxaldehydeHomo sapiens (human)EC50286.800010
2-[[anilino(oxo)methyl]amino]-4,5-dimethoxybenzoic acidHomo sapiens (human)EC50350.000010
3,4-dimethoxybenzenecarbothioic acid S-(4-chlorophenyl) esterHomo sapiens (human)EC50350.000010
N-(2,5-dimethylphenyl)-2-[[3-(4-ethylphenoxy)-4-oxo-1-benzopyran-7-yl]oxy]acetamideHomo sapiens (human)EC5037.360010
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)EC50350.000010
4-[(3,5-dimethylphenyl)-oxomethyl]-1,3-dihydroquinoxalin-2-oneHomo sapiens (human)EC50350.000010
N-[2-(4-methoxyphenyl)ethyl]-2,3-dihydro-1,4-dioxin-5-carboxamideHomo sapiens (human)EC50350.000010
2-chloro-N-[3-[(2-chlorophenyl)methyl]-2-thiazolylidene]acetamideHomo sapiens (human)EC50350.000010
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)EC50350.000010
N1-(2,6-dimorpholino-3-pyridyl)-4-methylbenzamideHomo sapiens (human)EC50350.000010
3,3-dimethyl-2-morpholino-2,3-dihydrobenzo[b]furan-5-olHomo sapiens (human)EC50350.000010
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)EC50350.000010
4-chloro-3-(diethylsulfamoyl)-N-(2-nitrophenyl)benzamideHomo sapiens (human)EC50350.000010
4-fluoro-N-[3-[2-nitro-4-(trifluoromethyl)anilino]propyl]benzamideHomo sapiens (human)EC50350.000010
2-[(4-methylphenyl)sulfonylamino]acetic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)EC50350.000010
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[4-(methylthio)phenyl]methyl]-1,2-dihydropyrazol-3-oneHomo sapiens (human)EC50350.000010
4-[[2-(4-methyl-1-piperidinyl)-1,3-benzothiazol-6-yl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)EC50350.000010
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideHomo sapiens (human)EC5041.050010
N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-2-(3-oxo-1,4-benzoxazin-4-yl)acetamideHomo sapiens (human)EC50350.000010
6,7-diethoxy-3-(3-methoxypropyl)-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)EC50350.000010
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olHomo sapiens (human)EC5068.270010
nsc 105827Homo sapiens (human)EC50145.900010
2-[[2-[(2,5-dimethylphenyl)sulfonylamino]-1-oxoethyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)EC50110.800010
N-(3-methylbutyl)-6-(4-morpholinylsulfonyl)-2-pyridin-4-yl-4-quinolinecarboxamideHomo sapiens (human)EC50350.000010
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideHomo sapiens (human)EC50214.000010
ML162Homo sapiens (human)EC5070.600010
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleHomo sapiens (human)EC5050.550010
digitoxigeninHomo sapiens (human)EC50350.000010
2-chloro-N-(2,6-dimethylphenyl)-3-oxo-3-phenylpropanamideHomo sapiens (human)EC50350.000010
4-[2-[[1-(2-methoxyethyl)-2-benzimidazolyl]thio]-1-oxoethyl]-2,5-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterHomo sapiens (human)EC50350.000010
harmanHomo sapiens (human)EC50350.000010
astragalinHomo sapiens (human)EC50350.000010
n-oleoyldopamineHomo sapiens (human)EC508.057010
2-(5-methyl-4,5,6,7-tetrahydroindazol-2-yl)-N-[3-(2-oxo-1-pyrrolidinyl)propyl]acetamideHomo sapiens (human)EC50350.000010
3-(3-bromophenyl)-2-(4-fluorophenyl)-5,6,7,7a-tetrahydro-3H-pyrrolo[1,2-c]imidazol-1-oneHomo sapiens (human)EC50350.000010
mdl 105519Homo sapiens (human)EC50350.000010
chaetoglobosin AHomo sapiens (human)EC50216.400010
emetine hydrochlorideHomo sapiens (human)EC50350.000010
3-hydroxy-2-methyl-1-(phenylmethyl)-4-pyridinoneHomo sapiens (human)EC50350.000010
chlorhexidineHomo sapiens (human)EC50350.000010
benalfocin hydrochlorideHomo sapiens (human)EC50350.000010
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)EC50338.000010
5-chloro-2-[(3-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)EC50163.700010
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideHomo sapiens (human)EC5058.100010
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideHomo sapiens (human)EC5047.250010
amphidinolide bHomo sapiens (human)EC50350.000010
lisinoprilHomo sapiens (human)EC50350.000010
1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-(2-nitrophenyl)sulfonylpiperazineHomo sapiens (human)EC50350.000010
5-(4-dibenzothiophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineHomo sapiens (human)EC50350.000010
4-chloro-N-[(2R,3R)-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl(pyridin-4-ylmethyl)amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]benzenesulfonamideHomo sapiens (human)EC50350.000010
kf38789Homo sapiens (human)EC50350.000010

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ag 1879Homo sapiens (human)AC50697.450020
2-fluoroadenosineHomo sapiens (human)AC50234.938030
anisomycinHomo sapiens (human)AC50150.339730
idarubicin hydrochlorideHomo sapiens (human)AC50233.630230
4-chloro-1-methyl-3-nitro-2-quinolinoneHomo sapiens (human)AbsAC10_uM1.106010
1-methyl-4-[(4-methylphenyl)thio]-3-nitro-2-quinolinoneHomo sapiens (human)AbsAC10_uM5.093010
1-methyl-4-[(4-methylphenyl)thio]-3-nitro-2-quinolinoneHomo sapiens (human)AC50227.300050
4-[[4-(2,5-dimethylphenyl)-1-piperazinyl]methyl]-2-methoxyphenolHomo sapiens (human)AC50308.612570
4-chloro-3-nitro-1-(phenylmethyl)-2-quinolinoneHomo sapiens (human)AbsAC10_uM22.735020
2,5-dimethyl-1-(phenylmethyl)pyrrole-3,4-dicarboxaldehydeHomo sapiens (human)AC50494.600050
N-(2,5-dimethylphenyl)-2-[[3-(4-ethylphenoxy)-4-oxo-1-benzopyran-7-yl]oxy]acetamideHomo sapiens (human)AC50155.203330
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)AC50350.000030
2-chloro-N-[3-[(2-chlorophenyl)methyl]-2-thiazolylidene]acetamideHomo sapiens (human)AC50350.000030
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)AC50145.621760
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)AC50262.730040
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideHomo sapiens (human)AC50155.953330
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olHomo sapiens (human)AC5046.300330
nsc 105827Homo sapiens (human)AC50212.778730
2-[[2-[(2,5-dimethylphenyl)sulfonylamino]-1-oxoethyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)AC50350.000030
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideHomo sapiens (human)AC50342.200030
ML162Homo sapiens (human)AC5082.453360
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleHomo sapiens (human)AC50107.863330
2-chloro-N-(2,6-dimethylphenyl)-3-oxo-3-phenylpropanamideHomo sapiens (human)AC50256.013330
n-oleoyldopamineHomo sapiens (human)AC5035.253330
chaetoglobosin AHomo sapiens (human)AC50133.330330
emetine hydrochlorideHomo sapiens (human)AC50233.729030
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)AC50283.090030
5-chloro-2-[(3-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)AC50282.800030
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideHomo sapiens (human)AC50278.307530
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideHomo sapiens (human)AC50260.480030
amphidinolide bHomo sapiens (human)AC50350.000030
navitoclaxHomo sapiens (human)AbsAC10_uM3.090010
kf38789Homo sapiens (human)AC50350.000030