Page last updated: 2024-08-07 16:34:21
Nociceptin receptor
A nociceptin receptor that is encoded in the genome of mouse. [OMA:P35377, PRO:DNx]
Synonyms
K3 opiate receptor;
Kappa-type 3 opioid receptor;
KOR-3;
ORGC;
Orphanin FQ receptor
Research
Bioassay Publications (6)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (16.67) | 18.2507 |
2000's | 4 (66.67) | 29.6817 |
2010's | 1 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (6)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
melatonin | Mus musculus (house mouse) | Ki | 0.0003 | 1 | 1 |
phosphoric acid | Mus musculus (house mouse) | Ki | 20,000.0000 | 1 | 1 |
diphosphoric acid | Mus musculus (house mouse) | Ki | 240.0000 | 1 | 1 |
methylene diphosphonate | Mus musculus (house mouse) | Ki | 20,000.0000 | 1 | 1 |
n(delta)-(phosphonoacetyl)-l-ornithine | Mus musculus (house mouse) | Ki | 0.1300 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
nociceptin | Mus musculus (house mouse) | EC50 | 0.0061 | 4 | 6 |