Page last updated: 2024-08-07 19:41:56

DNA dC->dU-editing enzyme APOBEC-3A isoform a

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (45)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
dimethylphenylpiperazinium iodideHomo sapiens (human)IC501.930010
c 137Homo sapiens (human)IC5018.000010
cefotetanHomo sapiens (human)IC5029.600010
2,2'-dipyridyl disulfideHomo sapiens (human)IC50100.000010
N-(4-ethoxyphenyl)-3-hydroxy-2-naphthalenecarboxamideHomo sapiens (human)IC5012.900010
trimethylphenylammonium iodideHomo sapiens (human)IC502.160010
2-phenyl-1,2-benzisothiazol-3-(2h)-oneHomo sapiens (human)IC50100.000010
4-chloro-N-(4-chloro-2,5-dimethoxyphenyl)-5-dithiazolimineHomo sapiens (human)IC50100.000010
N,N-diethyl-2-[(3-thiophen-2-yl-7-isothiazolo[4,5-d]pyrimidinyl)thio]acetamideHomo sapiens (human)IC5061.200010
5-ethyl-4,6-dimethyl-2-sulfanylidene-1H-pyridine-3-carbonitrileHomo sapiens (human)IC50100.000010
3-pyridinecarboxylic acid (3-acetyl-4-oxido-2-quinoxalin-4-iumyl)methyl esterHomo sapiens (human)IC501.480010
5-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazole-3-thioneHomo sapiens (human)IC5099.333330
ceefourin 1Homo sapiens (human)IC50100.000010
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileHomo sapiens (human)IC50100.000010
4-chloro-N-(3,4,5-trimethoxyphenyl)-5-dithiazolimineHomo sapiens (human)IC50100.000010
4-pyridin-4-yl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-quinoline-3-carbonitrileHomo sapiens (human)IC50100.000010
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3,4,5-trimethoxybenzamideHomo sapiens (human)IC502.240010
4-phenyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)IC50100.000010
2-[[2-[4-(4-chlorophenyl)-1-piperazinyl]-2-oxoethyl]thio]-3-ethyl-4-quinazolinoneHomo sapiens (human)IC502.830010
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-propan-2-yl-2-furancarboxamideHomo sapiens (human)IC506.260010
4-chloro-N-(4-chloro-2-methylphenyl)-5-dithiazolimineHomo sapiens (human)IC50100.000010
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC50100.000010
5-chloro-1h-benzimidazole-2-thiolHomo sapiens (human)IC50100.000010
N-(3-dibenzofuranyl)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)thio]acetamideHomo sapiens (human)IC505.400010
3-chloro-N-[3-(4-morpholinyl)propyl]-6-nitro-1-benzothiophene-2-carboxamideHomo sapiens (human)IC50100.000010
N-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)-2-furancarboxamideHomo sapiens (human)IC50100.000010
(2S)-3-methyl-2-[[(3-methylphenyl)-oxomethyl]amino]butanoic acid (4-oxo-2-pyrimido[2,1-b][1,3]benzothiazolyl)methyl esterHomo sapiens (human)IC5014.700010
5-[[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]methyl]-2-furancarboxylic acid methyl esterHomo sapiens (human)IC50100.000010
2-methoxy-4-[3-(2-methoxyphenyl)-5,6-dihydro-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]phenolHomo sapiens (human)IC50100.000010
ssya10-001Homo sapiens (human)IC5038.900010
5-cyclopentylidene-2-sulfanylidene-4-thiazolidinoneHomo sapiens (human)IC505.610010
2-[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]propanoic acid methyl esterHomo sapiens (human)IC50100.000010
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidHomo sapiens (human)IC50100.000010
4-(3,4-dimethylphenyl)-3-(5-methyl-3-isoxazolyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)IC50100.000010
N-(3,4-dimethylphenyl)-2-[[5-[3-(4-methoxyphenyl)propyl]-1,3,4-oxadiazol-2-yl]thio]acetamideHomo sapiens (human)IC502.180010
2-(3-oxo-4H-1,4-benzothiazin-2-yl)acetic acid (7-acetamido-2-oxo-1-benzopyran-4-yl)methyl esterHomo sapiens (human)IC5019.300010
myricetinHomo sapiens (human)IC5017.500010
6-bromo-5-methyl-1,3-dihydroimidazo[4,5-b]pyridine-2-thioneHomo sapiens (human)IC50100.000010
mg 624Homo sapiens (human)IC502.330010
trimetazidine dihydrochlorideHomo sapiens (human)IC508.260010
enisamium iodideHomo sapiens (human)IC502.980010
2-[6-[(2-fluorophenyl)methyl]-5,7-dimethyl-4-oxo-3-pyrrolo[3,4-d]pyridazinyl]-N-(2,3,5,6-tetrafluorophenyl)acetamideHomo sapiens (human)IC5049.300010
5-fluoro-2-phenyl-1,2-benzothiazol-3-oneHomo sapiens (human)IC50100.000010
2-(4-fluorophenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)IC50100.000010
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimineHomo sapiens (human)IC50100.000010