Page last updated: 2024-08-07 22:49:11

EWS/FLI fusion protein

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (1124)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
1-(2,4-dihydroxyphenyl)-3-(4-hydroxyphenyl)-2-propen-1-oneHomo sapiens (human)Potency18.965040
taxifolinHomo sapiens (human)Potency33.173430
aminocaproic acidHomo sapiens (human)Potency18.181030
acetylcysteineHomo sapiens (human)Potency0.001910
3-(4-hydroxy-3-methoxyphenyl)prop-2-enoic acidHomo sapiens (human)Potency11.063320
histamineHomo sapiens (human)Potency14.692120
melatoninHomo sapiens (human)Potency2.125040
spermidineHomo sapiens (human)Potency26.350610
taurineHomo sapiens (human)Potency0.935010
b 844-39Homo sapiens (human)Potency23.875640
huperzine aHomo sapiens (human)Potency15.032130
pk 11195Homo sapiens (human)Potency16.486930
pd 173074Homo sapiens (human)Potency18.209540
N-(4-hydroxyphenyl)-3,7-dimethyl-9-(2,6,6-trimethyl-1-cyclohexenyl)nona-2,4,6,8-tetraenamideHomo sapiens (human)Potency6.042540
nitrofurazoneHomo sapiens (human)Potency32.775240
tacrineHomo sapiens (human)Potency16.285540
abt 702Homo sapiens (human)Potency31.124840
acetaminophenHomo sapiens (human)Potency25.914120
tyrphostin ag 1024Homo sapiens (human)Potency33.491640
rtki cpdHomo sapiens (human)Potency13.523440
alfuzosinHomo sapiens (human)Potency4.176310
altretamineHomo sapiens (human)Potency1.049010
amantadineHomo sapiens (human)Potency25.625240
theophyllineHomo sapiens (human)Potency22.085830
amiodaroneHomo sapiens (human)Potency8.587040
dan 2163Homo sapiens (human)Potency10.466620
amlexanoxHomo sapiens (human)Potency25.011830
amoxapineHomo sapiens (human)Potency15.599440
aniracetamHomo sapiens (human)Potency33.173410
arecolineHomo sapiens (human)Potency17.543430
aspirinHomo sapiens (human)Potency14.922240
azathioprineHomo sapiens (human)Potency2.953840
azelastineHomo sapiens (human)Potency3.934840
benserazideHomo sapiens (human)Potency28.517240
berberineHomo sapiens (human)Potency8.357240
betaxololHomo sapiens (human)Potency18.654810
bicalutamideHomo sapiens (human)Potency2.323940
2-cyano-3-(3,4-dihydroxyphenyl)-N-(phenylmethyl)-2-propenamideHomo sapiens (human)Potency21.639040
ro 31-8425Homo sapiens (human)Potency18.209540
seratrodastHomo sapiens (human)Potency0.003710
bufexamacHomo sapiens (human)Potency7.448440
busulfanHomo sapiens (human)Potency8.316420
caffeic acidHomo sapiens (human)Potency17.850940
verapamilHomo sapiens (human)Potency0.005410
calmidazoliumHomo sapiens (human)Potency20.493340
N-[4-methyl-1-oxo-1-(1-oxohexan-2-ylamino)pentan-2-yl]carbamic acid (phenylmethyl) esterHomo sapiens (human)Potency9.194720
camostatHomo sapiens (human)Potency8.587040
capsaicinHomo sapiens (human)Potency10.990640
carbidopaHomo sapiens (human)Potency23.485010
carisoprodolHomo sapiens (human)Potency0.010510
carmofurHomo sapiens (human)Potency12.991240
carmustineHomo sapiens (human)Potency0.023510
carvedilolHomo sapiens (human)Potency15.401630
celecoxibHomo sapiens (human)Potency12.521140
chelerythrineHomo sapiens (human)Potency7.448740
chlorambucilHomo sapiens (human)Potency23.174840
chlorhexidineHomo sapiens (human)Potency5.977240
chlormezanoneHomo sapiens (human)Potency15.799130
chlorothiazideHomo sapiens (human)Potency0.014810
chloroxineHomo sapiens (human)Potency9.864140
ciclopiroxHomo sapiens (human)Potency5.971940
cilostazolHomo sapiens (human)Potency0.046910
ciprofibrateHomo sapiens (human)Potency29.892040
ciprofloxacinHomo sapiens (human)Potency0.078220
cisplatinHomo sapiens (human)Potency11.745120
citalopramHomo sapiens (human)Potency16.699630
N-[4-(4-morpholinyl)butyl]-2-benzofurancarboxamideHomo sapiens (human)Potency26.350610
clofibrateHomo sapiens (human)Potency23.485010
clomipheneHomo sapiens (human)Potency24.630140
clomipramineHomo sapiens (human)Potency1.829440
clotrimazoleHomo sapiens (human)Potency20.276940
cromoglycateHomo sapiens (human)Potency0.003010
crotamitonHomo sapiens (human)Potency29.683130
cyclobenzaprineHomo sapiens (human)Potency18.778640
cyclosporineHomo sapiens (human)Potency17.627720
cyproheptadineHomo sapiens (human)Potency17.028840
indibulinHomo sapiens (human)Potency0.132140
dacarbazineHomo sapiens (human)Potency18.654820
diclofenac sodiumHomo sapiens (human)Potency20.699930
dichlorphenamideHomo sapiens (human)Potency0.468610
dienestrolHomo sapiens (human)Potency28.309040
diethylstilbestrolHomo sapiens (human)Potency27.339940
3,3'-diindolylmethaneHomo sapiens (human)Potency6.451440
dilacor xrHomo sapiens (human)Potency18.654810
diphenhydramineHomo sapiens (human)Potency29.018930
dipyridamoleHomo sapiens (human)Potency24.995740
disulfiramHomo sapiens (human)Potency0.038940
domperidoneHomo sapiens (human)Potency18.654810
doxazosinHomo sapiens (human)Potency21.198730
dyphyllineHomo sapiens (human)Potency13.206610
econazoleHomo sapiens (human)Potency25.416040
efavirenzHomo sapiens (human)Potency24.917840
embelinHomo sapiens (human)Potency29.943930
emodinHomo sapiens (human)Potency29.565910
enoxacinHomo sapiens (human)Potency0.002610
ethosuximideHomo sapiens (human)Potency28.329220
etodolacHomo sapiens (human)Potency26.350610
famotidineHomo sapiens (human)Potency16.360030
felbamateHomo sapiens (human)Potency10.660230
fenbendazoleHomo sapiens (human)Potency1.455740
fenofibrateHomo sapiens (human)Potency8.313620
flecainideHomo sapiens (human)Potency33.320230
flucytosineHomo sapiens (human)Potency15.930720
fluphenazineHomo sapiens (human)Potency30.057640
flumazenilHomo sapiens (human)Potency18.345820
1-[bis(4-fluorophenyl)methyl]-4-(3-phenylprop-2-enyl)piperazineHomo sapiens (human)Potency20.543830
fluorouracilHomo sapiens (human)Potency6.983240
flurbiprofenHomo sapiens (human)Potency19.997030
flutamideHomo sapiens (human)Potency11.082640
luvoxHomo sapiens (human)Potency24.061040
fomepizoleHomo sapiens (human)Potency0.029440
furosemideHomo sapiens (human)Potency0.002610
gabapentinHomo sapiens (human)Potency34.185440
gabexateHomo sapiens (human)Potency6.619010
gbr 12935Homo sapiens (human)Potency24.270340
gemfibrozilHomo sapiens (human)Potency36.209340
gentian violetHomo sapiens (human)Potency0.272740
gliclazideHomo sapiens (human)Potency22.083040
glimepirideHomo sapiens (human)Potency37.221210
glipizideHomo sapiens (human)Potency21.069940
gö6983Homo sapiens (human)Potency0.028140
go 6976Homo sapiens (human)Potency3.782740
gossypolHomo sapiens (human)Potency13.530640
N-[2-(4-bromocinnamylamino)ethyl]isoquinoline-5-sulfonamideHomo sapiens (human)Potency3.020440
fasudilHomo sapiens (human)Potency13.181220
ha14-1Homo sapiens (human)Potency25.796240
haloperidolHomo sapiens (human)Potency23.159240
hexestrolHomo sapiens (human)Potency1.284840
hydroxychloroquineHomo sapiens (human)Potency24.314640
hydroxyureaHomo sapiens (human)Potency14.106440
atropine sulfateHomo sapiens (human)Potency18.068440
phenelzineHomo sapiens (human)Potency12.595940
idebenoneHomo sapiens (human)Potency32.479640
ifosfamideHomo sapiens (human)Potency22.831940
indapamideHomo sapiens (human)Potency28.064240
indomethacinHomo sapiens (human)Potency15.475430
ipriflavoneHomo sapiens (human)Potency33.173420
isoconazoleHomo sapiens (human)Potency28.850040
isoniazidHomo sapiens (human)Potency0.001010
isoproterenolHomo sapiens (human)Potency14.435440
isradipineHomo sapiens (human)Potency28.143740
whi p97Homo sapiens (human)Potency0.141340
ketanserinHomo sapiens (human)Potency2.232420
ketoprofenHomo sapiens (human)Potency16.026640
ketorolacHomo sapiens (human)Potency4.458740
ketotifenHomo sapiens (human)Potency17.792340
5-isoquinolinesulfonic acid [4-[2-[5-isoquinolinylsulfonyl(methyl)amino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl]phenyl] esterHomo sapiens (human)Potency17.757540
lamotrigineHomo sapiens (human)Potency34.295440
lansoprazoleHomo sapiens (human)Potency30.441930
beta-lapachoneHomo sapiens (human)Potency19.047640
leflunomideHomo sapiens (human)Potency16.136240
letrozoleHomo sapiens (human)Potency20.041340
lg 100268Homo sapiens (human)Potency16.626110
linopirdineHomo sapiens (human)Potency15.722020
liranaftateHomo sapiens (human)Potency0.004210
lomefloxacinHomo sapiens (human)Potency0.742710
lomustineHomo sapiens (human)Potency0.016610
loperamideHomo sapiens (human)Potency19.285740
loratadineHomo sapiens (human)Potency25.634240
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-oneHomo sapiens (human)Potency16.785640
4-(dimethylamino)-n-(7-(hydroxyamino)-7-oxoheptyl)benzamideHomo sapiens (human)Potency0.518340
maprotilineHomo sapiens (human)Potency22.277440
mebendazoleHomo sapiens (human)Potency0.771840
mechlorethamineHomo sapiens (human)Potency34.522730
meclizineHomo sapiens (human)Potency18.999940
mefloquine hydrochlorideHomo sapiens (human)Potency25.346540
vitamin k 3Homo sapiens (human)Potency26.132440
metforminHomo sapiens (human)Potency0.001210
methocarbamolHomo sapiens (human)Potency0.037210
methoxsalenHomo sapiens (human)Potency3.317320
nocodazoleHomo sapiens (human)Potency0.023640
3,7-bis(dimethylamino)phenothiazin-5-iumHomo sapiens (human)Potency5.026540
metronidazoleHomo sapiens (human)Potency0.104910
mianserinHomo sapiens (human)Potency20.493340
miconazoleHomo sapiens (human)Potency22.993840
mirtazapineHomo sapiens (human)Potency5.257610
mitotaneHomo sapiens (human)Potency24.061140
mitoxantroneHomo sapiens (human)Potency0.106330
entinostatHomo sapiens (human)Potency3.927340
6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-isobenzofuran-5-yl)-4-methyl-4-hexenoic acid 2-(4-morpholinyl)ethyl esterHomo sapiens (human)Potency2.007040
6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-isobenzofuran-5-yl)-4-methyl-4-hexenoic acidHomo sapiens (human)Potency2.475240
nafamostatHomo sapiens (human)Potency37.221210
naftopidilHomo sapiens (human)Potency14.876830
naratriptanHomo sapiens (human)Potency1.181040
niclosamideHomo sapiens (human)Potency8.973440
nifekalantHomo sapiens (human)Potency21.000440
nilutamideHomo sapiens (human)Potency9.349510
nimesulideHomo sapiens (human)Potency12.846940
norfloxacinHomo sapiens (human)Potency23.485010
nu6102Homo sapiens (human)Potency13.999540
o(6)-benzylguanineHomo sapiens (human)Potency22.846440
ofloxacinHomo sapiens (human)Potency20.931020
olprinoneHomo sapiens (human)Potency0.018710
omeprazoleHomo sapiens (human)Potency26.455130
ondansetronHomo sapiens (human)Potency16.162530
5-[3-(benzenesulfonamido)phenyl]-N-hydroxypent-2-en-4-ynamideHomo sapiens (human)Potency1.238640
oxibendazoleHomo sapiens (human)Potency0.006340
oxymetazolineHomo sapiens (human)Potency34.185440
pantoprazoleHomo sapiens (human)Potency33.173410
papaverineHomo sapiens (human)Potency21.639040
pd 153035Homo sapiens (human)Potency0.759340
pd 98059Homo sapiens (human)Potency10.986020
pentamidineHomo sapiens (human)Potency11.190640
perhexilineHomo sapiens (human)Potency16.631140
phenoxybenzamineHomo sapiens (human)Potency0.033210
phenylmethylsulfonyl fluorideHomo sapiens (human)Potency2.232730
phloretinHomo sapiens (human)Potency1.806440
moxonidineHomo sapiens (human)Potency0.013210
3,3',4,5'-tetrahydroxystilbeneHomo sapiens (human)Potency18.716740
pimobendanHomo sapiens (human)Potency20.931010
pioglitazoneHomo sapiens (human)Potency0.155220
ono 1078Homo sapiens (human)Potency18.147640
praziquantelHomo sapiens (human)Potency33.393620
prazosinHomo sapiens (human)Potency26.132440
primidoneHomo sapiens (human)Potency13.648240
probucolHomo sapiens (human)Potency11.079030
procarbazineHomo sapiens (human)Potency0.001710
propafenoneHomo sapiens (human)Potency23.101840
pyrimethamineHomo sapiens (human)Potency5.352240
pyroxamideHomo sapiens (human)Potency4.026740
3-[(3,5-dibromo-4-hydroxyphenyl)methylidene]-5-iodo-1H-indol-2-oneHomo sapiens (human)Potency20.431440
raloxifeneHomo sapiens (human)Potency7.828640
opc 12759Homo sapiens (human)Potency35.197320
hydrochlorothiazideHomo sapiens (human)Potency2.643840
resveratrolHomo sapiens (human)Potency16.736440
riluzoleHomo sapiens (human)Potency24.366740
rimantadineHomo sapiens (human)Potency0.011810
risperidoneHomo sapiens (human)Potency33.173410
rofecoxibHomo sapiens (human)Potency25.602330
sb 206553Homo sapiens (human)Potency19.238040
sb 239063Homo sapiens (human)Potency24.323430
sb 202190Homo sapiens (human)Potency21.000440
sibutramineHomo sapiens (human)Potency27.121640
sotalolHomo sapiens (human)Potency19.093240
imatinibHomo sapiens (human)Potency29.849440
SU5402Homo sapiens (human)Potency31.467740
SU6656Homo sapiens (human)Potency5.468340
vorinostatHomo sapiens (human)Potency2.652540
sulfamethizoleHomo sapiens (human)Potency13.785340
sulfanilamideHomo sapiens (human)Potency26.350610
copal rosin varnishHomo sapiens (human)Potency10.300240
sulpirideHomo sapiens (human)Potency26.923620
sumatriptanHomo sapiens (human)Potency0.003310
suraminHomo sapiens (human)Potency10.476020
2-[4-(1,2-diphenylbut-1-enyl)phenoxy]-N,N-dimethylethanamineHomo sapiens (human)Potency20.133440
tazaroteneHomo sapiens (human)Potency0.014810
terazosinHomo sapiens (human)Potency33.173410
N,6,6-trimethyl-N-(1-naphthalenylmethyl)-1-hept-2-en-4-ynamineHomo sapiens (human)Potency37.221210
tetrahydropapaverineHomo sapiens (human)Potency24.917820
thalidomideHomo sapiens (human)Potency0.003710
theobromineHomo sapiens (human)Potency25.907140
thiotepaHomo sapiens (human)Potency10.626640
ticlopidineHomo sapiens (human)Potency0.083310
tioconazoleHomo sapiens (human)Potency26.132440
tioproninHomo sapiens (human)Potency37.221220
tizanidineHomo sapiens (human)Potency0.525810
2-[4-(4-chloro-1,2-diphenylbut-1-enyl)phenoxy]-N,N-dimethylethanamineHomo sapiens (human)Potency2.780430
tranexamic acidHomo sapiens (human)Potency11.278020
2-[[3-(3,4-dimethoxyphenyl)-1-oxoprop-2-enyl]amino]benzoic acidHomo sapiens (human)Potency23.485010
2-phenylcyclopropan-1-amineHomo sapiens (human)Potency23.485010
retinoic acidHomo sapiens (human)Potency14.796440
trifluoperazineHomo sapiens (human)Potency14.821040
trimetrexateHomo sapiens (human)Potency1.576240
trioxsalenHomo sapiens (human)Potency17.249140
2,3-bis[amino-[(2-aminophenyl)thio]methylidene]butanedinitrileHomo sapiens (human)Potency26.788840
venlafaxineHomo sapiens (human)Potency29.018930
xylometazolineHomo sapiens (human)Potency0.001210
3-(5'-hydroxymethyl-2'-furyl)-1-benzylindazoleHomo sapiens (human)Potency8.814040
ici 204,219Homo sapiens (human)Potency20.562740
zm 336372Homo sapiens (human)Potency0.685440
mitomycinHomo sapiens (human)Potency0.036240
phentolamineHomo sapiens (human)Potency15.722020
thyroxineHomo sapiens (human)Potency3.035320
chloramphenicolHomo sapiens (human)Potency0.020910
vincristineHomo sapiens (human)Potency0.002040
phenylephrineHomo sapiens (human)Potency0.026410
levodopaHomo sapiens (human)Potency0.372210
cytidineHomo sapiens (human)Potency0.038640
cycloheximideHomo sapiens (human)Potency0.233240
caffeine citrateHomo sapiens (human)Potency13.206610
cytarabineHomo sapiens (human)Potency0.468610
pantothenic acidHomo sapiens (human)Potency28.702640
rotenoneHomo sapiens (human)Potency2.619640
7,8-dimethyl-10-[(2R,3R,4S)-2,3,4,5-tetrahydroxypentyl]benzo[g]pteridine-2,4-dioneHomo sapiens (human)Potency29.762020
synephrineHomo sapiens (human)Potency0.001310
monobenzoneHomo sapiens (human)Potency5.012740
phenforminHomo sapiens (human)Potency16.995640
pyrazolanthroneHomo sapiens (human)Potency17.772440
rheinHomo sapiens (human)Potency34.042910
indirubinHomo sapiens (human)Potency15.571140
ostholHomo sapiens (human)Potency17.280930
cytisineHomo sapiens (human)Potency37.221210
podophyllotoxinHomo sapiens (human)Potency0.004210
physcioneHomo sapiens (human)Potency0.578720
azomycinHomo sapiens (human)Potency5.257610
docosanolHomo sapiens (human)Potency0.002610
antimycin aHomo sapiens (human)Potency0.070640
daminozideHomo sapiens (human)Potency30.057640
stavudineHomo sapiens (human)Potency34.042910
cladribineHomo sapiens (human)Potency0.318740
2,4,5-trimethoxybenzaldehydeHomo sapiens (human)Potency36.209340
buthionine sulfoximineHomo sapiens (human)Potency14.818010
vidarabineHomo sapiens (human)Potency9.208940
octocryleneHomo sapiens (human)Potency0.004210
zalcitabineHomo sapiens (human)Potency0.001210
usnic acidHomo sapiens (human)Potency0.004210
camptothecinHomo sapiens (human)Potency0.009540
chloropyramineHomo sapiens (human)Potency23.562940
parbendazoleHomo sapiens (human)Potency1.190340
thiamphenicolHomo sapiens (human)Potency16.278440
pizotylineHomo sapiens (human)Potency28.517240
(3R)-6,7-dimethoxy-3-[(5R)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]-3H-isobenzofuran-1-oneHomo sapiens (human)Potency0.127030
du-21220Homo sapiens (human)Potency20.931010
canadineHomo sapiens (human)Potency19.744730
flubendazoleHomo sapiens (human)Potency0.706440
dobutamineHomo sapiens (human)Potency26.623540
halofantrineHomo sapiens (human)Potency6.216220
lonidamineHomo sapiens (human)Potency0.003710
ng-nitroarginine methyl esterHomo sapiens (human)Potency0.014810
oxfendazoleHomo sapiens (human)Potency13.850640
nitazoxanideHomo sapiens (human)Potency20.895640
epirubicinHomo sapiens (human)Potency0.121040
s-2678Homo sapiens (human)Potency25.711540
clorsulonHomo sapiens (human)Potency23.485020
butoconazoleHomo sapiens (human)Potency35.197320
nicorandilHomo sapiens (human)Potency33.597730
fazarabineHomo sapiens (human)Potency5.727040
amonafideHomo sapiens (human)Potency9.931440
avobenzoneHomo sapiens (human)Potency1.616840
pramiracetamHomo sapiens (human)Potency16.626110
fenticonazoleHomo sapiens (human)Potency32.775240
lovastatinHomo sapiens (human)Potency15.457640
flupirtineHomo sapiens (human)Potency22.846540
2-[[1-(2-amino-4-thiazolyl)-2-[[(2S,3S)-2-methyl-4-oxo-1-sulfo-3-azetidinyl]amino]-2-oxoethylidene]amino]oxy-2-methylpropanoic acidHomo sapiens (human)Potency19.792920
simvastatinHomo sapiens (human)Potency14.408140
balsalazideHomo sapiens (human)Potency17.850040
pravastatinHomo sapiens (human)Potency27.052220
mifepristoneHomo sapiens (human)Potency0.282840
itraconazoleHomo sapiens (human)Potency0.833310
nitrogenase stabilizing-protective protein, bacteriaHomo sapiens (human)Potency4.043240
sarafloxacinHomo sapiens (human)Potency13.559630
imiquimodHomo sapiens (human)Potency15.340640
adapaleneHomo sapiens (human)Potency3.245230
sparfloxacinHomo sapiens (human)Potency10.223210
clopidogrelHomo sapiens (human)Potency35.197320
topotecanHomo sapiens (human)Potency0.026240
aripiprazoleHomo sapiens (human)Potency13.046440
sipatrigineHomo sapiens (human)Potency16.626110
monatepilHomo sapiens (human)Potency16.174140
duloxetineHomo sapiens (human)Potency4.417040
irinotecanHomo sapiens (human)Potency0.414440
ziprasidoneHomo sapiens (human)Potency22.846540
2-[11-[3-(dimethylamino)propylidene]-6H-benzo[c][1]benzoxepin-2-yl]acetic acidHomo sapiens (human)Potency19.548440
adefovir dipivoxilHomo sapiens (human)Potency0.357040
LSM-1535Homo sapiens (human)Potency0.001010
lincomycin monohydrochlorideHomo sapiens (human)Potency2.348510
plerixaforHomo sapiens (human)Potency4.685910
oseltamivirHomo sapiens (human)Potency0.007410
ginkgolide bHomo sapiens (human)Potency14.883630
secoisolariciresinolHomo sapiens (human)Potency0.424140
bendamustineHomo sapiens (human)Potency21.383840
mizolastineHomo sapiens (human)Potency24.552040
cgs 9343bHomo sapiens (human)Potency15.722040
prulifloxacinHomo sapiens (human)Potency11.770410
balofloxacinHomo sapiens (human)Potency18.833740
repaglinideHomo sapiens (human)Potency0.525810
telmisartanHomo sapiens (human)Potency34.185440
hordenineHomo sapiens (human)Potency18.654810
rilmenidineHomo sapiens (human)Potency1.865510
zoledronic acidHomo sapiens (human)Potency0.040020
mepivacaineHomo sapiens (human)Potency13.190120
diclofensineHomo sapiens (human)Potency30.353140
nefiracetamHomo sapiens (human)Potency2.956610
uk 68798Homo sapiens (human)Potency28.342840
dapoxetineHomo sapiens (human)Potency24.279340
bindaritHomo sapiens (human)Potency10.795230
hp 873Homo sapiens (human)Potency31.234840
dexrazoxaneHomo sapiens (human)Potency8.694830
masoprocolHomo sapiens (human)Potency15.423540
voriconazoleHomo sapiens (human)Potency23.485010
moroxydineHomo sapiens (human)Potency35.197340
Suplatast tosilateHomo sapiens (human)Potency0.009310
secnidazoleHomo sapiens (human)Potency32.642530
alibendolHomo sapiens (human)Potency17.302330
octyloniumHomo sapiens (human)Potency20.543830
nedaplatinHomo sapiens (human)Potency5.899210
thioxoloneHomo sapiens (human)Potency17.354640
ubenimexHomo sapiens (human)Potency26.623540
tetrahydropalmatineHomo sapiens (human)Potency14.381440
honokiolHomo sapiens (human)Potency29.762040
picropodophyllinHomo sapiens (human)Potency0.100740
tetrandrineHomo sapiens (human)Potency21.000440
LSM-4272Homo sapiens (human)Potency0.975940
rosiglitazoneHomo sapiens (human)Potency8.554720
bexaroteneHomo sapiens (human)Potency24.938230
s20098Homo sapiens (human)Potency19.536320
albendazole sulfoxideHomo sapiens (human)Potency22.208040
4-aminoquinazolineHomo sapiens (human)Potency35.197320
matrineHomo sapiens (human)Potency0.001010
hydroxyflutamideHomo sapiens (human)Potency22.034640
n-(4,4-diphenyl-3-butenyl)nipecotic acidHomo sapiens (human)Potency10.919040
nsc-87877Homo sapiens (human)Potency16.681340
mci 9038Homo sapiens (human)Potency12.286140
lopinavirHomo sapiens (human)Potency26.997040
10-hydroxycamptothecinHomo sapiens (human)Potency0.010440
fotemustineHomo sapiens (human)Potency0.014810
sn 38Homo sapiens (human)Potency0.106040
sr141716Homo sapiens (human)Potency28.351840
vanoxerineHomo sapiens (human)Potency23.875640
indolactam vHomo sapiens (human)Potency0.414120
(6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4,6-dimethyl-7-oxohepta-2,4-dienamideHomo sapiens (human)Potency0.446740
racecadotrilHomo sapiens (human)Potency0.803740
pyronaridineHomo sapiens (human)Potency22.742040
deguelinHomo sapiens (human)Potency20.052440
fingolimodHomo sapiens (human)Potency21.000440
tesmilifeneHomo sapiens (human)Potency24.679440
benzamilHomo sapiens (human)Potency27.330940
tamibaroteneHomo sapiens (human)Potency25.317940
carboxyamido-triazoleHomo sapiens (human)Potency21.716840
ci 988Homo sapiens (human)Potency1.343820
tanshinoneHomo sapiens (human)Potency11.770410
icrf 193Homo sapiens (human)Potency0.691830
sophocarpineHomo sapiens (human)Potency17.133340
nitisinoneHomo sapiens (human)Potency29.943930
sr 48692Homo sapiens (human)Potency4.176310
elacridarHomo sapiens (human)Potency23.540240
mosaprideHomo sapiens (human)Potency0.589420
ezogabineHomo sapiens (human)Potency25.887040
celastrolHomo sapiens (human)Potency1.066540
almotriptanHomo sapiens (human)Potency0.074310
gefitinibHomo sapiens (human)Potency30.540140
vadimezanHomo sapiens (human)Potency25.220440
gyki 53655Homo sapiens (human)Potency8.407340
methotrexateHomo sapiens (human)Potency0.027940
umifenovirHomo sapiens (human)Potency18.562240
safinamideHomo sapiens (human)Potency13.196740
ml-3000Homo sapiens (human)Potency23.927340
febuxostatHomo sapiens (human)Potency29.565910
(1R,3S)-5-[2-[(1R,3aS,7aR)-1-[(2R)-6-hydroxy-6-methylheptan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-4-methylenecyclohexane-1,3-diolHomo sapiens (human)Potency3.642840
aspartameHomo sapiens (human)Potency30.565840
pomalidomideHomo sapiens (human)Potency0.004210
cd 437Homo sapiens (human)Potency0.986440
tempolHomo sapiens (human)Potency0.372210
10-propargyl-10-deazaaminopterinHomo sapiens (human)Potency0.036240
atazanavirHomo sapiens (human)Potency4.685910
lonafarnibHomo sapiens (human)Potency13.638940
chs 828Homo sapiens (human)Potency0.002220
tariquidarHomo sapiens (human)Potency11.506840
levofloxacinHomo sapiens (human)Potency24.089720
nepafenacHomo sapiens (human)Potency20.200830
conivaptanHomo sapiens (human)Potency24.816130
evodiamineHomo sapiens (human)Potency25.174730
varespladibHomo sapiens (human)Potency19.722440
canertinibHomo sapiens (human)Potency16.798340
cinacalcetHomo sapiens (human)Potency10.068320
birb 796Homo sapiens (human)Potency25.248440
nps-568Homo sapiens (human)Potency37.221220
telbivudineHomo sapiens (human)Potency9.309030
tipifarnibHomo sapiens (human)Potency5.817340
torcetrapibHomo sapiens (human)Potency27.800840
cryptotanshinoneHomo sapiens (human)Potency24.366740
cyc 202Homo sapiens (human)Potency22.013540
ampelopsinHomo sapiens (human)Potency31.791130
vincristineHomo sapiens (human)Potency19.496030
tanshinone ii aHomo sapiens (human)Potency0.003710
avasimibeHomo sapiens (human)Potency5.198630
sb 203580Homo sapiens (human)Potency44.307040
enzastaurinHomo sapiens (human)Potency8.697940
erlotinibHomo sapiens (human)Potency15.852640
piboserodHomo sapiens (human)Potency11.426740
l 163191Homo sapiens (human)Potency24.444640
cephalexin, (6r-(6alpha,7beta))-isomerHomo sapiens (human)Potency0.007410
latrepirdineHomo sapiens (human)Potency31.293230
orantinibHomo sapiens (human)Potency0.243640
dronedaroneHomo sapiens (human)Potency20.493340
ramelteonHomo sapiens (human)Potency2.348510
lapatinibHomo sapiens (human)Potency6.031240
2-(4-morpholinoanilino)-6-cyclohexylaminopurineHomo sapiens (human)Potency5.416840
dabigatran etexilateHomo sapiens (human)Potency17.466040
darunavirHomo sapiens (human)Potency1.992340
deferasiroxHomo sapiens (human)Potency17.112640
dabigatranHomo sapiens (human)Potency0.179520
sorafenibHomo sapiens (human)Potency6.716640
N-hydroxy-3-[4-[[2-hydroxyethyl-[2-(1H-indol-3-yl)ethyl]amino]methyl]phenyl]-2-propenamideHomo sapiens (human)Potency0.173040
lenalidomideHomo sapiens (human)Potency7.079020
N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamideHomo sapiens (human)Potency0.125340
sr 142806Homo sapiens (human)Potency24.279340
phenoxodiolHomo sapiens (human)Potency4.718840
1-methylpropyl-2-imidazolyl disulfideHomo sapiens (human)Potency22.793040
demecolcineHomo sapiens (human)Potency0.235640
nsc 74859Homo sapiens (human)Potency20.766240
gant58Homo sapiens (human)Potency23.875640
cyclovirobuxine dHomo sapiens (human)Potency13.206610
2,5-bis(5-hydroxymethyl-2-thienyl)furanHomo sapiens (human)Potency11.266440
nsc 663284Homo sapiens (human)Potency5.327240
bortezomibHomo sapiens (human)Potency0.032240
ritonavirHomo sapiens (human)Potency17.458430
nu 6027Homo sapiens (human)Potency14.862140
nsc 23766Homo sapiens (human)Potency27.052220
gant 61Homo sapiens (human)Potency20.431440
naringeninHomo sapiens (human)Potency17.068820
5-hydroxytryptophanHomo sapiens (human)Potency11.770410
amastatinHomo sapiens (human)Potency23.050630
tosylphenylalanyl chloromethyl ketoneHomo sapiens (human)Potency19.112440
mometasone furoateHomo sapiens (human)Potency7.987240
linezolidHomo sapiens (human)Potency9.425430
temocapril hydrochlorideHomo sapiens (human)Potency5.037840
vinpocetineHomo sapiens (human)Potency20.431440
estramustine phosphate sodiumHomo sapiens (human)Potency0.010510
fluticasone propionateHomo sapiens (human)Potency16.626110
pd 173955Homo sapiens (human)Potency0.114640
gw 3965Homo sapiens (human)Potency22.285940
y 27632Homo sapiens (human)Potency9.327920
rolipramHomo sapiens (human)Potency3.599240
6-bromoindirubin-3'-oximeHomo sapiens (human)Potency4.774140
purvalanol bHomo sapiens (human)Potency0.128140
repsoxHomo sapiens (human)Potency7.426610
roflumilastHomo sapiens (human)Potency17.684030
decitabineHomo sapiens (human)Potency10.221840
(2R,3S,5S)-2-(6-aminopurin-9-yl)-5-(hydroxymethyl)-3-oxolanolHomo sapiens (human)Potency20.347430
pa 824Homo sapiens (human)Potency6.180440
ketoconazoleHomo sapiens (human)Potency19.924240
purvalanol aHomo sapiens (human)Potency10.110640
diclazurilHomo sapiens (human)Potency29.696630
melphalanHomo sapiens (human)Potency3.585440
benzyloxycarbonylleucyl-leucyl-leucine aldehydeHomo sapiens (human)Potency0.440640
tenofovirHomo sapiens (human)Potency0.468610
terameprocolHomo sapiens (human)Potency1.104440
shikoninHomo sapiens (human)Potency2.283840
5-fluoro-2'-deoxycytidineHomo sapiens (human)Potency0.059040
IPA-3Homo sapiens (human)Potency29.045640
4-(4-chloro-2-methylphenoxy)-n-hydroxybutanamideHomo sapiens (human)Potency5.727940
mecarbinateHomo sapiens (human)Potency35.871930
pirarubicin hydrochlorideHomo sapiens (human)Potency0.502240
cgp 60474Homo sapiens (human)Potency0.149640
tram 34Homo sapiens (human)Potency1.020540
fludarabineHomo sapiens (human)Potency0.687840
propylthiouracilHomo sapiens (human)Potency35.197320
prothionamideHomo sapiens (human)Potency0.003710
etomidateHomo sapiens (human)Potency37.221210
mercaptopurineHomo sapiens (human)Potency2.477840
jrf 12Homo sapiens (human)Potency22.924440
rg108Homo sapiens (human)Potency0.003010
stf 62247Homo sapiens (human)Potency30.565840
stf 083010Homo sapiens (human)Potency2.391640
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-1-naphthalenecarboxamideHomo sapiens (human)Potency0.381240
paroxetine, cis-(+)-isomerHomo sapiens (human)Potency18.279930
eszopicloneHomo sapiens (human)Potency20.931010
cct018159Homo sapiens (human)Potency8.087340
secinh3Homo sapiens (human)Potency13.478330
2-[[benzamido(sulfanylidene)methyl]amino]-5,5-dimethyl-4,7-dihydrothieno[2,3-c]pyran-3-carboxylic acidHomo sapiens (human)Potency29.696630
jk184Homo sapiens (human)Potency0.002940
3-(1-azepanylsulfonyl)-n-(3-bromphenyl)benzamideHomo sapiens (human)Potency24.201440
xl147Homo sapiens (human)Potency13.843240
N-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)thio]acetamideHomo sapiens (human)Potency18.209540
3-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineHomo sapiens (human)Potency18.654810
thioguanine anhydrousHomo sapiens (human)Potency1.338140
hc-067047Homo sapiens (human)Potency11.196140
bi-78d3Homo sapiens (human)Potency4.989740
ethionamideHomo sapiens (human)Potency20.931020
kartogeninHomo sapiens (human)Potency29.565910
methyl-thiohydantoin-tryptophanHomo sapiens (human)Potency0.589910
10074-g5Homo sapiens (human)Potency33.173410
kl001Homo sapiens (human)Potency23.875640
2-[2-chloro-6-ethoxy-4-[(3-methyl-5-oxo-1-phenyl-4-pyrazolylidene)methyl]phenoxy]acetic acid methyl esterHomo sapiens (human)Potency10.695930
4-(5-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1h-pyrazol-1-yl)benzenesulfonamideHomo sapiens (human)Potency30.565840
monastrolHomo sapiens (human)Potency0.116340
maravirocHomo sapiens (human)Potency32.479640
rwj 67657Homo sapiens (human)Potency26.623540
nelarabineHomo sapiens (human)Potency20.931010
6-methyl-2-(phenylethynyl)pyridineHomo sapiens (human)Potency20.431440
bms 387032Homo sapiens (human)Potency0.153840
or 1259Homo sapiens (human)Potency24.444640
e 7010Homo sapiens (human)Potency0.097840
ly335979Homo sapiens (human)Potency25.985040
tandutinibHomo sapiens (human)Potency22.993940
vx-745Homo sapiens (human)Potency26.818330
corlanorHomo sapiens (human)Potency19.564440
prucaloprideHomo sapiens (human)Potency36.209340
dasatinibHomo sapiens (human)Potency15.990140
poly(2-fluoroadenylic acid)Homo sapiens (human)Potency14.508140
zd 6474Homo sapiens (human)Potency10.247440
N-methyl-2-[[3-[2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]thio]benzamideHomo sapiens (human)Potency8.417040
N-[2-(diethylamino)ethyl]-5-[(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamideHomo sapiens (human)Potency9.549640
compound 968Homo sapiens (human)Potency23.576830
gw 7647Homo sapiens (human)Potency12.719630
valproateHomo sapiens (human)Potency0.417610
brl 15572Homo sapiens (human)Potency20.050040
1-[6-(4-chlorophenyl)-5-imidazo[2,1-b]thiazolyl]-N-[(3,4-dichlorophenyl)methoxy]methanimineHomo sapiens (human)Potency14.830130
rose bengal(2-)Homo sapiens (human)Potency15.826440
N4-ethyl-N6,1,2-trimethyl-N4-phenylpyrimidin-1-ium-4,6-diamineHomo sapiens (human)Potency12.026420
2-[[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]-1-oxo-5-isoquinolinyl]oxy]propanoic acid ethyl esterHomo sapiens (human)Potency7.526230
sb 415286Homo sapiens (human)Potency33.148740
4-methylene-2-octyl-5-oxo-3-oxolanecarboxylic acidHomo sapiens (human)Potency31.785940
stx-0119Homo sapiens (human)Potency17.486040
sch 79797Homo sapiens (human)Potency3.759140
LY-310762Homo sapiens (human)Potency20.931010
am 630Homo sapiens (human)Potency34.185440
sb 408124Homo sapiens (human)Potency27.958220
sitagliptinHomo sapiens (human)Potency19.924240
4-(5-benzo(1,3)dioxol-5-yl-4-pyridin-2-yl-1h-imidazol-2-yl)benzamideHomo sapiens (human)Potency15.722020
rabeprazole(1-)Homo sapiens (human)Potency14.631920
tolcaponeHomo sapiens (human)Potency36.209340
1-(4-Fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-oneHomo sapiens (human)Potency20.931010
eeyarestatin iHomo sapiens (human)Potency19.619640
imd 0354Homo sapiens (human)Potency1.437940
ex 527Homo sapiens (human)Potency11.426830
jtk-303Homo sapiens (human)Potency25.985040
ku 55933Homo sapiens (human)Potency20.493340
quercetinHomo sapiens (human)Potency15.820740
biochanin aHomo sapiens (human)Potency37.221210
apigeninHomo sapiens (human)Potency22.355440
luteolinHomo sapiens (human)Potency33.173410
hymecromoneHomo sapiens (human)Potency22.208020
daphnetinHomo sapiens (human)Potency15.826440
kaempferolHomo sapiens (human)Potency17.634140
genisteinHomo sapiens (human)Potency12.575730
baicaleinHomo sapiens (human)Potency25.268640
chrysinHomo sapiens (human)Potency31.293230
diosmetinHomo sapiens (human)Potency10.657940
fisetinHomo sapiens (human)Potency17.757540
morinHomo sapiens (human)Potency18.654810
myricetinHomo sapiens (human)Potency20.055620
daidzeinHomo sapiens (human)Potency17.970130
purmorphamineHomo sapiens (human)Potency0.001910
sag compoundHomo sapiens (human)Potency25.083140
levetiracetamHomo sapiens (human)Potency24.917820
blebbistatinHomo sapiens (human)Potency13.995840
ter 199Homo sapiens (human)Potency37.221220
acipimoxHomo sapiens (human)Potency30.090730
ly 320135Homo sapiens (human)Potency18.618020
n-(4-amino-2-methylquinolin-6-yl)-2-(4-ethylphenoxymethyl)benzamideHomo sapiens (human)Potency8.388040
pd 166285Homo sapiens (human)Potency2.013240
(3r)-((2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl))methanoneHomo sapiens (human)Potency28.056340
3-[6-[4-(trifluoromethoxy)anilino]-4-pyrimidinyl]benzamideHomo sapiens (human)Potency26.150340
icaritinHomo sapiens (human)Potency22.532840
bosutinibHomo sapiens (human)Potency19.462040
palbociclibHomo sapiens (human)Potency14.915440
jnj-7706621Homo sapiens (human)Potency7.337440
benazeprilHomo sapiens (human)Potency22.846540
verteporfinHomo sapiens (human)Potency0.079340
batimastatHomo sapiens (human)Potency16.124920
sinomenineHomo sapiens (human)Potency6.444440
pepstatinHomo sapiens (human)Potency2.093110
norbinaltorphimineHomo sapiens (human)Potency33.173410
pregabalinHomo sapiens (human)Potency16.626110
2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz(h)imidazo(4,5-f)isoquinoline-7-oneHomo sapiens (human)Potency4.734440
vx680Homo sapiens (human)Potency2.953440
cgp 3466Homo sapiens (human)Potency0.074310
d 4476Homo sapiens (human)Potency24.630140
cyc 116Homo sapiens (human)Potency12.733040
bay 19-8004Homo sapiens (human)Potency17.751140
indiplonHomo sapiens (human)Potency21.209740
pai 039Homo sapiens (human)Potency20.931010
tubacinHomo sapiens (human)Potency9.631440
(13S)-3-hydroxy-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-oneHomo sapiens (human)Potency6.119940
ispinesibHomo sapiens (human)Potency2.338640
nps2143Homo sapiens (human)Potency15.722040
pd 184352Homo sapiens (human)Potency22.915440
prasugrelHomo sapiens (human)Potency3.187340
fesoterodineHomo sapiens (human)Potency33.173410
hdac-42Homo sapiens (human)Potency0.636740
3-tritylthio-l-alanine, (d)-isomerHomo sapiens (human)Potency24.993840
posaconazoleHomo sapiens (human)Potency14.128640
a 770041Homo sapiens (human)Potency3.790840
tws 119Homo sapiens (human)Potency3.199740
[4-[[4-(1-benzothiophen-2-yl)-2-pyrimidinyl]amino]phenyl]-[4-(1-pyrrolidinyl)-1-piperidinyl]methanoneHomo sapiens (human)Potency19.792940
pnu-282987Homo sapiens (human)Potency17.039140
iniparibHomo sapiens (human)Potency8.332810
nepicastatHomo sapiens (human)Potency24.366740
[4-(2-amino-4-bromoanilino)-2-chlorophenyl]-(2-methylphenyl)methanoneHomo sapiens (human)Potency17.553840
mk 0752Homo sapiens (human)Potency12.934340
nt 702Homo sapiens (human)Potency13.596740
gw 501516Homo sapiens (human)Potency12.836630
az 11645373Homo sapiens (human)Potency6.867040
av 412Homo sapiens (human)Potency2.042440
ag-041rHomo sapiens (human)Potency34.522730
telatinibHomo sapiens (human)Potency11.750820
y-39983Homo sapiens (human)Potency24.713240
cp 547632Homo sapiens (human)Potency14.862140
bms345541Homo sapiens (human)Potency6.207740
vidofludimusHomo sapiens (human)Potency13.141040
spc-839Homo sapiens (human)Potency1.508440
lenvatinibHomo sapiens (human)Potency0.850040
andarineHomo sapiens (human)Potency3.722110
adw 742Homo sapiens (human)Potency12.656640
gw843682xHomo sapiens (human)Potency2.074940
pd 0325901Homo sapiens (human)Potency32.775240
gsk 256066Homo sapiens (human)Potency0.002310
midostaurinHomo sapiens (human)Potency1.802440
ly 404039Homo sapiens (human)Potency19.958140
ag 14361Homo sapiens (human)Potency19.792940
sb 265610Homo sapiens (human)Potency31.567640
ly 450139Homo sapiens (human)Potency20.055620
cp 91149Homo sapiens (human)Potency22.083040
gw791343Homo sapiens (human)Potency12.858540
cabazitaxelHomo sapiens (human)Potency0.239620
sb-505124Homo sapiens (human)Potency9.951040
sb 242235Homo sapiens (human)Potency8.034640
mocetinostatHomo sapiens (human)Potency1.088440
sd 0006Homo sapiens (human)Potency0.028420
osi 930Homo sapiens (human)Potency18.147640
carbobenzoxy-leucyl-leucyl-norvalinalHomo sapiens (human)Potency1.072440
ki 20227Homo sapiens (human)Potency29.210940
scio-469Homo sapiens (human)Potency22.083040
ssr 69071Homo sapiens (human)Potency19.106740
sb 3ct compoundHomo sapiens (human)Potency21.131840
orteronelHomo sapiens (human)Potency18.912430
pi103Homo sapiens (human)Potency0.404140
l 084Homo sapiens (human)Potency33.173420
2-((aminocarbonyl)amino)-5-(4-fluorophenyl)-3-thiophenecarboxamideHomo sapiens (human)Potency1.978940
tgx 221Homo sapiens (human)Potency30.353140
sa 4503Homo sapiens (human)Potency17.874520
ic 87114Homo sapiens (human)Potency2.283440
zibotentanHomo sapiens (human)Potency18.654810
sb 705498Homo sapiens (human)Potency25.083140
tivozanibHomo sapiens (human)Potency3.156540
zm 447439Homo sapiens (human)Potency11.119440
avn 944Homo sapiens (human)Potency0.482940
n-(6-chloro-7-methoxy-9h-beta-carbolin-8-yl)-2-methylnicotinamideHomo sapiens (human)Potency3.877540
rucaparibHomo sapiens (human)Potency17.126940
cediranibHomo sapiens (human)Potency21.770340
tae226Homo sapiens (human)Potency3.808740
gw0742Homo sapiens (human)Potency28.143740
sb 743921Homo sapiens (human)Potency11.296820
ps1145Homo sapiens (human)Potency25.416040
l-779,450Homo sapiens (human)Potency21.786340
tak-715Homo sapiens (human)Potency18.833740
aq4nHomo sapiens (human)Potency14.711840
chir 99021Homo sapiens (human)Potency12.124940
ym 201636Homo sapiens (human)Potency17.640440
sb 525334Homo sapiens (human)Potency21.848240
osu 03012Homo sapiens (human)Potency16.173340
sb-612111Homo sapiens (human)Potency9.436340
masitinibHomo sapiens (human)Potency24.917840
bx795Homo sapiens (human)Potency8.511740
linagliptinHomo sapiens (human)Potency28.860140
as 601245Homo sapiens (human)Potency17.436840
pazopanibHomo sapiens (human)Potency20.668220
sepantroniumHomo sapiens (human)Potency0.007240
azd 6244Homo sapiens (human)Potency14.711840
odanacatibHomo sapiens (human)Potency18.716740
1-(2-(1-adamantyl)ethyl)-1-pentyl-3-(3-(4-pyridyl)propyl)ureaHomo sapiens (human)Potency17.188440
cp-673,451Homo sapiens (human)Potency18.903240
a 443654Homo sapiens (human)Potency1.840140
apixabanHomo sapiens (human)Potency0.020910
bay 61-3606Homo sapiens (human)Potency8.300340
gw 799388Homo sapiens (human)Potency19.384830
ar c155858Homo sapiens (human)Potency0.135620
gw 842166xHomo sapiens (human)Potency30.565840
akt-i-1 compoundHomo sapiens (human)Potency0.601040
erteberelHomo sapiens (human)Potency16.211340
aee 788Homo sapiens (human)Potency0.017830
saracatinibHomo sapiens (human)Potency20.788740
az10606120Homo sapiens (human)Potency15.450440
sd-208Homo sapiens (human)Potency3.409730
osi-420Homo sapiens (human)Potency9.318040
gm 1489Homo sapiens (human)Potency34.185440
[4-(3-chlorophenyl)-1-piperazinyl]-(5-methyl-2-phenyl-3-pyrazolyl)methanoneHomo sapiens (human)Potency2.846230
vx 702Homo sapiens (human)Potency26.350610
crenolanibHomo sapiens (human)Potency0.013210
ki16425Homo sapiens (human)Potency0.016610
tg100-115Homo sapiens (human)Potency22.208040
cc 401Homo sapiens (human)Potency19.597840
ly 411575Homo sapiens (human)Potency20.931010
bms 599626Homo sapiens (human)Potency0.908040
e 5555Homo sapiens (human)Potency10.344840
volasertibHomo sapiens (human)Potency0.090840
PB28Homo sapiens (human)Potency19.854840
azd 7762Homo sapiens (human)Potency0.319540
krp-203Homo sapiens (human)Potency30.565840
regorafenibHomo sapiens (human)Potency20.931040
at 7867Homo sapiens (human)Potency20.041340
acetic acid 2-[4-methyl-8-(4-morpholinylsulfonyl)-1,3-dioxo-2-pyrrolo[3,4-c]quinolinyl]ethyl esterHomo sapiens (human)Potency0.018710
6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-oneHomo sapiens (human)Potency0.844940
ptc 124Homo sapiens (human)Potency19.496030
abt-737Homo sapiens (human)Potency11.440340
brivanibHomo sapiens (human)Potency14.354340
icg 001Homo sapiens (human)Potency2.908440
pha 680632Homo sapiens (human)Potency2.836040
4-(2-((1r)-1-(((4-chlorophenyl)sulfonyl)-2,5-difluoroanilino)ethyl)-5-fluorophenyl)butanoic acidHomo sapiens (human)Potency21.270140
fg-4592Homo sapiens (human)Potency5.899210
mp470Homo sapiens (human)Potency6.605840
jnj16259685Homo sapiens (human)Potency14.459240
ki 8751Homo sapiens (human)Potency14.748540
mk 2866Homo sapiens (human)Potency33.173410
nu 7441Homo sapiens (human)Potency7.334640
at 7519Homo sapiens (human)Potency0.269240
cyt997Homo sapiens (human)Potency1.482440
bi 2536Homo sapiens (human)Potency0.056240
N-(6-fluoro-1H-indazol-5-yl)-6-methyl-2-oxo-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyridine-5-carboxamideHomo sapiens (human)Potency4.454220
compound 26Homo sapiens (human)Potency11.640430
r 1487Homo sapiens (human)Potency1.902720
adl 5859Homo sapiens (human)Potency10.490410
danusertibHomo sapiens (human)Potency0.261540
N-[4-(2-tert-butylphenyl)sulfonylphenyl]-2,3,4-trihydroxy-5-[(2-propan-2-ylphenyl)methyl]benzamideHomo sapiens (human)Potency7.879740
N-[5-[[5-[(4-acetyl-1-piperazinyl)-oxomethyl]-4-methoxy-2-methylphenyl]thio]-2-thiazolyl]-4-[(3,3-dimethylbutan-2-ylamino)methyl]benzamideHomo sapiens (human)Potency8.970640
nvp-aew541Homo sapiens (human)Potency11.299940
abt 869Homo sapiens (human)Potency33.283540
azd 8931Homo sapiens (human)Potency0.056240
fr 180204Homo sapiens (human)Potency10.657140
dorsomorphinHomo sapiens (human)Potency18.833740
ac 261066Homo sapiens (human)Potency25.642040
quisinostatHomo sapiens (human)Potency0.030140
anacetrapibHomo sapiens (human)Potency20.055620
carfilzomibHomo sapiens (human)Potency0.021040
hcv 796Homo sapiens (human)Potency17.978630
pf-2545920Homo sapiens (human)Potency17.702340
jnj 26854165Homo sapiens (human)Potency10.489840
pf 573228Homo sapiens (human)Potency15.633540
tak 285Homo sapiens (human)Potency22.714440
idelalisibHomo sapiens (human)Potency2.724240
nebivolol hydrochlorideHomo sapiens (human)Potency22.208040
crizotinibHomo sapiens (human)Potency11.527740
5-(5,6-dimethoxy-1-benzimidazolyl)-3-[(2-methylsulfonylphenyl)methoxy]-2-thiophenecarbonitrileHomo sapiens (human)Potency14.476130
4-[2-(2-chloro-4-fluoroanilino)-5-methyl-4-pyrimidinyl]-N-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-1H-pyrrole-2-carboxamideHomo sapiens (human)Potency21.000440
osi 906Homo sapiens (human)Potency10.027840
zstk474Homo sapiens (human)Potency1.166140
4-cyano-N-[4-(4-methyl-1-piperazinyl)-2-(4-methyl-1-piperidinyl)phenyl]-1H-pyrrole-2-carboxamideHomo sapiens (human)Potency29.083640
ly2109761Homo sapiens (human)Potency23.650240
chir-265Homo sapiens (human)Potency7.398840
motesanibHomo sapiens (human)Potency8.035040
fostamatinibHomo sapiens (human)Potency9.785140
az-628Homo sapiens (human)Potency16.798340
jnj 28312141Homo sapiens (human)Potency17.354640
omecamtiv mecarbilHomo sapiens (human)Potency6.661030
trametinibHomo sapiens (human)Potency13.192140
mln8054Homo sapiens (human)Potency0.692040
pf-562,271Homo sapiens (human)Potency9.123240
pha 767491Homo sapiens (human)Potency3.631840
abexinostatHomo sapiens (human)Potency0.966640
N-[3-[[5-bromo-4-[2-(1H-imidazol-5-yl)ethylamino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamideHomo sapiens (human)Potency3.644040
N-(2,4-dimethoxyphenyl)-N-[2-[4-(4-methyl-1-piperazinyl)anilino]-4-pyrimidinyl]carbamic acid (2,6-dimethylphenyl) esterHomo sapiens (human)Potency2.371140
at 13387Homo sapiens (human)Potency0.321240
ly2603618Homo sapiens (human)Potency1.090440
veliparibHomo sapiens (human)Potency22.502720
ku-0060648Homo sapiens (human)Potency8.224640
Glycyl-H-1152Homo sapiens (human)Potency6.740740
dactolisibHomo sapiens (human)Potency0.042240
bgt226Homo sapiens (human)Potency0.017040
palomid 529Homo sapiens (human)Potency19.638440
sc1 compoundHomo sapiens (human)Potency0.510240
bilobalideHomo sapiens (human)Potency20.931010
(7R,9S)-9-acetyl-7-[[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-methyl-2-oxanyl]oxy]-6,9,11-trihydroxy-4-methoxy-8,10-dihydro-7H-tetracene-5,12-dioneHomo sapiens (human)Potency0.051940
4-[(1,4-dioxo-2-naphthalenyl)amino]benzenesulfonamideHomo sapiens (human)Potency10.629340
doxifluridineHomo sapiens (human)Potency14.007240
3'',4''-DiacetylafzelinHomo sapiens (human)Potency26.923620
tosedostatHomo sapiens (human)Potency20.578840
novobiocinHomo sapiens (human)Potency4.644440
ku 60019Homo sapiens (human)Potency21.639040
gsk 461364Homo sapiens (human)Potency0.079140
azd 1152-hqpaHomo sapiens (human)Potency3.019740
nvp-tae684Homo sapiens (human)Potency6.993540
a 803467Homo sapiens (human)Potency35.197340
4-methyl-3-(2-(2-morpholinoethylamino)quinazolin-6-yl)-n-(3-(trifluoromethyl)phenyl)benzamideHomo sapiens (human)Potency14.056140
gsk 269962aHomo sapiens (human)Potency9.193940
tak-901Homo sapiens (human)Potency1.103140
cct129202Homo sapiens (human)Potency22.346340
a-83-01Homo sapiens (human)Potency13.294220
3-[(1-methyl-3-indolyl)methylidene]-1H-pyrrolo[3,2-b]pyridin-2-oneHomo sapiens (human)Potency33.393620
buparlisibHomo sapiens (human)Potency0.568640
azd 1480Homo sapiens (human)Potency15.021540
azd8330Homo sapiens (human)Potency0.001910
lumacaftorHomo sapiens (human)Potency0.047340
pha 848125Homo sapiens (human)Potency2.208340
tg101209Homo sapiens (human)Potency2.428040
fedratinibHomo sapiens (human)Potency0.235620
gsk690693Homo sapiens (human)Potency21.069940
cnf 2024Homo sapiens (human)Potency0.163340
ku 0063794Homo sapiens (human)Potency0.652740
azd 7545Homo sapiens (human)Potency21.023630
nvp-bhg712Homo sapiens (human)Potency14.971540
azd5438Homo sapiens (human)Potency4.045840
nutlin-3bHomo sapiens (human)Potency14.291240
amg 1Homo sapiens (human)Potency26.276040
cct 128930Homo sapiens (human)Potency17.133340
gdc 0941Homo sapiens (human)Potency2.289140
sm 164Homo sapiens (human)Potency28.850040
N-[5-[[5-[(4-acetyl-1-piperazinyl)-oxomethyl]-4-methoxy-2-methylphenyl]thio]-2-thiazolyl]-4-[(3-methylbutan-2-ylamino)methyl]benzamideHomo sapiens (human)Potency10.773540
3-(3,4-dihydroxyphenyl)lactateHomo sapiens (human)Potency30.768430
ph 797804Homo sapiens (human)Potency30.353140
pha 408Homo sapiens (human)Potency10.237240
kw-2478Homo sapiens (human)Potency1.146340
cefpodoximeHomo sapiens (human)Potency26.701440
gsk 1016790aHomo sapiens (human)Potency22.846540
kx-01Homo sapiens (human)Potency0.026940
mesnaHomo sapiens (human)Potency0.002110
olaparibHomo sapiens (human)Potency10.300040
srt1720Homo sapiens (human)Potency28.351840
plx 4720Homo sapiens (human)Potency17.188440
ast 1306Homo sapiens (human)Potency1.062940
mk 5108Homo sapiens (human)Potency1.865940
cx 4945Homo sapiens (human)Potency5.547040
pci 34051Homo sapiens (human)Potency11.263240
cudc 101Homo sapiens (human)Potency0.047840
purfalcamineHomo sapiens (human)Potency0.001710
amg 458Homo sapiens (human)Potency28.133640
cpi 613Homo sapiens (human)Potency1.659220
mln 8237Homo sapiens (human)Potency0.532740
snx 2112Homo sapiens (human)Potency0.104640
lde225Homo sapiens (human)Potency15.292240
gdc 0449Homo sapiens (human)Potency1.421630
sgx 523Homo sapiens (human)Potency25.248420
bms 754807Homo sapiens (human)Potency1.142640
gdc-0068Homo sapiens (human)Potency5.188540
bms 777607Homo sapiens (human)Potency29.341240
sgi 1776Homo sapiens (human)Potency14.237340
lomibuvirHomo sapiens (human)Potency27.422430
1-(1-(1-methylcyclooctyl)-4-piperidinyl)-2-((3r)-3-piperidinyl)-1h-benzimidazoleHomo sapiens (human)Potency15.494940
delanzomibHomo sapiens (human)Potency0.059240
pci 32765Homo sapiens (human)Potency23.159240
cink4Homo sapiens (human)Potency27.635440
ponatinibHomo sapiens (human)Potency5.435540
amg 900Homo sapiens (human)Potency0.010640
mk-1775Homo sapiens (human)Potency0.262740
tak-875Homo sapiens (human)Potency20.931020
cgi 1746Homo sapiens (human)Potency22.520740
apalutamideHomo sapiens (human)Potency5.199840
bag956Homo sapiens (human)Potency0.121740
N-[[3-fluoro-4-[[2-(1-methyl-4-imidazolyl)-7-thieno[3,2-b]pyridinyl]oxy]anilino]-sulfanylidenemethyl]-2-phenylacetamideHomo sapiens (human)Potency21.639040
PP121Homo sapiens (human)Potency1.068240
as 605240Homo sapiens (human)Potency11.033540
SL-327Homo sapiens (human)Potency6.241140
N-[4-[3-[[[7-(hydroxyamino)-7-oxoheptyl]amino]-oxomethyl]-5-isoxazolyl]phenyl]carbamic acid tert-butyl esterHomo sapiens (human)Potency2.008240
niraparibHomo sapiens (human)Potency3.840740
tak 733Homo sapiens (human)Potency37.221210
mk 2206Homo sapiens (human)Potency15.577140
navitoclaxHomo sapiens (human)Potency19.957240
mk 8245Homo sapiens (human)Potency0.004710
sns 314Homo sapiens (human)Potency0.519940
mk 3207Homo sapiens (human)Potency0.020910
jzl 184Homo sapiens (human)Potency26.923620
at 406Homo sapiens (human)Potency34.522730
gsk 650394Homo sapiens (human)Potency8.100430
pf-04691502Homo sapiens (human)Potency0.071240
n-(cyanomethyl)-4-(2-((4-(4-morpholinyl)phenyl)amino)-4-pyrimidinyl)benzamideHomo sapiens (human)Potency11.572240
dcc-2036Homo sapiens (human)Potency19.285740
oprozomibHomo sapiens (human)Potency0.170240
az 960Homo sapiens (human)Potency4.309740
cabozantinibHomo sapiens (human)Potency1.595240
N-(2,6-difluorophenyl)-5-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonyl-1-piperazinyl)-1-piperidinyl]anilino]-4-pyrimidinyl]-2-imidazo[1,2-a]pyridinyl]-2-methoxybenzamideHomo sapiens (human)Potency20.071640
bs 194Homo sapiens (human)Potency0.350040
incb-018424Homo sapiens (human)Potency23.358340
asp3026Homo sapiens (human)Potency17.757540
bix 01294Homo sapiens (human)Potency7.876840
cct 137690Homo sapiens (human)Potency8.896240
pf 3845Homo sapiens (human)Potency18.147640
TAK-580Homo sapiens (human)Potency24.201440
gsk 2126458Homo sapiens (human)Potency0.045640
emd1214063Homo sapiens (human)Potency16.262340
gsk 1838705aHomo sapiens (human)Potency12.652340
ixazomibHomo sapiens (human)Potency0.303040
ldn 193189Homo sapiens (human)Potency12.460740
gne 477Homo sapiens (human)Potency0.057140
nvp-bep800Homo sapiens (human)Potency1.066240
1-[4-[[4-amino-5-chloro-6-(2-propan-2-ylsulfonylanilino)-2-pyrimidinyl]amino]-3-methoxyphenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency11.306340
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamideHomo sapiens (human)Potency2.900140
pf 3758309Homo sapiens (human)Potency3.674940
telotristat etiprateHomo sapiens (human)Potency24.279340
cx 5461Homo sapiens (human)Potency5.253930
wye 125132Homo sapiens (human)Potency0.020240
plx4032Homo sapiens (human)Potency18.110240
(2S)-2-[[2-(2,3-dihydro-1H-inden-5-yloxy)-9-[(4-phenylphenyl)methyl]-6-purinyl]amino]-3-phenyl-1-propanolHomo sapiens (human)Potency11.283540
N-[3-[[2-[[4-(dimethylamino)cyclohexyl]amino]-9-propan-2-yl-6-purinyl]amino]phenyl]-2-propenamideHomo sapiens (human)Potency0.356740
4-[(9-cyclopentyl-6-oxo-5-propan-2-yl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidinyl)benzamideHomo sapiens (human)Potency2.220840
gsk 1363089Homo sapiens (human)Potency5.731740
arry-334543Homo sapiens (human)Potency9.444740
kin-193Homo sapiens (human)Potency28.494440
mk 2461Homo sapiens (human)Potency10.149040
N-(2-chlorophenyl)-4-[[2-[4-[2-(4-ethyl-1-piperazinyl)-2-oxoethyl]anilino]-5-fluoro-4-pyrimidinyl]amino]benzamideHomo sapiens (human)Potency5.341240
8-chloro-4-(3-chloro-4-fluoroanilino)-6-[[1-(1-ethyl-4-piperidinyl)-4-triazolyl]methylamino]-3-quinolinecarbonitrileHomo sapiens (human)Potency18.716740
bay 869766Homo sapiens (human)Potency18.203140
as 703026Homo sapiens (human)Potency19.106740
pki 402Homo sapiens (human)Potency0.017640
pf 04929113Homo sapiens (human)Potency0.168540
baricitinibHomo sapiens (human)Potency3.720240
nvp bvu972Homo sapiens (human)Potency0.046910
4-[6-[4-(methoxycarbonylamino)phenyl]-4-(4-morpholinyl)-1-pyrazolo[3,4-d]pyrimidinyl]-1-piperidinecarboxylic acid methyl esterHomo sapiens (human)Potency0.096640
ly2811376Homo sapiens (human)Potency37.221210
dabrafenibHomo sapiens (human)Potency10.255440
as1949490Homo sapiens (human)Potency17.923740
3-[2-[2-chloro-4-[[3-(2,6-dichlorophenyl)-5-propan-2-yl-4-isoxazolyl]methoxy]phenyl]ethenyl]benzoic acidHomo sapiens (human)Potency18.654820
3-[[4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-1,4-diazepan-1-yl]sulfonyl]anilineHomo sapiens (human)Potency15.722020
cp 466722Homo sapiens (human)Potency14.223140
an2728Homo sapiens (human)Potency31.785920
CAY10626Homo sapiens (human)Potency0.033740
N-[3-[[5-chloro-2-[4-(4-methyl-1-piperazinyl)anilino]-4-pyrimidinyl]oxy]phenyl]-2-propenamideHomo sapiens (human)Potency5.609240
thiopental sodiumHomo sapiens (human)Potency0.015440
yk 4-279Homo sapiens (human)Potency2.202640
5-(4-amino-1-propan-2-yl-3-pyrazolo[3,4-d]pyrimidinyl)-1,3-benzoxazol-2-amineHomo sapiens (human)Potency0.009340
pha 793887Homo sapiens (human)Potency0.798140
stemregenin 1Homo sapiens (human)Potency5.976940
thiazovivinHomo sapiens (human)Potency26.483240
ly2784544Homo sapiens (human)Potency9.620940
unc 0638Homo sapiens (human)Potency6.502540
jzl195Homo sapiens (human)Potency29.565910
mk-8776Homo sapiens (human)Potency0.196040
nvp-bsk805Homo sapiens (human)Potency20.362040
xmd 8-92Homo sapiens (human)Potency19.417140
lrrk2-in1Homo sapiens (human)Potency7.854640
bms 708163Homo sapiens (human)Potency14.473240
gsk 1070916Homo sapiens (human)Potency2.810640
gsk923295Homo sapiens (human)Potency0.211540
jq1 compoundHomo sapiens (human)Potency5.227640
jnj38877605Homo sapiens (human)Potency15.468840
N-[3-(1,3-benzothiazol-2-yl)-5,6-dihydro-4H-thieno[2,3-c]pyrrol-2-yl]acetamideHomo sapiens (human)Potency15.319240
lgk974Homo sapiens (human)Potency19.924240
gsk525762aHomo sapiens (human)Potency4.355640
1-[(3,4-difluorophenyl)methyl]-2-oxo-N-[(1R)-2-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)oxy]-1-phenylethyl]-3-pyridinecarboxamideHomo sapiens (human)Potency24.061140
ch 5132799Homo sapiens (human)Potency0.577840
alectinibHomo sapiens (human)Potency0.013040
ML240Homo sapiens (human)Potency8.872240
glpg0634Homo sapiens (human)Potency10.914540
torin 1Homo sapiens (human)Potency0.023540
abt-199Homo sapiens (human)Potency22.522640
ly2940680Homo sapiens (human)Potency25.003640
tubastatin aHomo sapiens (human)Potency15.423540
1-[4-fluoro-3-(trifluoromethyl)phenyl]-3-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ureaHomo sapiens (human)Potency34.295440
xl765Homo sapiens (human)Potency19.223940
bs-181Homo sapiens (human)Potency10.067440
ro 4929097Homo sapiens (human)Potency17.691940
mln 9708Homo sapiens (human)Potency0.229840
gsk4112Homo sapiens (human)Potency3.141630
bms-911543Homo sapiens (human)Potency24.208440
ve 821Homo sapiens (human)Potency9.291130
spautin-1Homo sapiens (human)Potency13.500040
azd4547Homo sapiens (human)Potency16.278440
torin 2Homo sapiens (human)Potency0.010440
pf-4708671Homo sapiens (human)Potency18.209540
gsk1210151aHomo sapiens (human)Potency8.661440
apr-246Homo sapiens (human)Potency2.356340
3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-(4-(4-ethylpiperazin-1-yl)-phenylamino)pyrimidin-4-yl)-1-methylureaHomo sapiens (human)Potency37.221210
acy-1215Homo sapiens (human)Potency5.308140
bp-1-102Homo sapiens (human)Potency10.739040
as 604850Homo sapiens (human)Potency32.381640
chir 98014Homo sapiens (human)Potency3.406730
N-(3-chlorophenyl)-3-[[3,5-dimethyl-4-[(4-methyl-1-piperazinyl)-oxomethyl]-1H-pyrrol-2-yl]methylidene]-N-methyl-2-oxo-1H-indole-5-sulfonamideHomo sapiens (human)Potency29.068240
N-[4-(1-benzoyl-4-piperidinyl)butyl]-3-(3-pyridinyl)-2-propenamideHomo sapiens (human)Potency0.005040
N-[4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamideHomo sapiens (human)Potency3.010440
2-methoxy-N-[3-[4-[3-methyl-4-[(6-methyl-3-pyridinyl)oxy]anilino]-6-quinazolinyl]prop-2-enyl]acetamideHomo sapiens (human)Potency27.690740
belinostatHomo sapiens (human)Potency2.071840
bibr 1532Homo sapiens (human)Potency9.305740
cudc-907Homo sapiens (human)Potency0.006040
tetracyclineHomo sapiens (human)Potency10.760640
minocyclineHomo sapiens (human)Potency5.994740
piroxicamHomo sapiens (human)Potency36.209340
mobiflexHomo sapiens (human)Potency13.415120
ethyl 1-benzyl-3-hydroxy-2(5h)-oxopyrrole-4-carboxylateHomo sapiens (human)Potency11.770410
warfarinHomo sapiens (human)Potency0.003020
2-[[[4-hydroxy-2-oxo-1-(phenylmethyl)-3-quinolinyl]-oxomethyl]amino]acetic acidHomo sapiens (human)Potency20.468040
lornoxicamHomo sapiens (human)Potency8.307040
a 769662Homo sapiens (human)Potency19.472240
dolutegravirHomo sapiens (human)Potency19.069440
agi-5198Homo sapiens (human)Potency11.575420
pf-5274857Homo sapiens (human)Potency9.328420
3-[[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)-4-pyrimidinyl]amino]propanoic acidHomo sapiens (human)Potency20.344730
pik 75Homo sapiens (human)Potency0.033640
5-[[5-(4-fluoro-2-hydroxyphenyl)-2-furanyl]methylidene]thiazolidine-2,4-dioneHomo sapiens (human)Potency22.277440
LimKi 3Homo sapiens (human)Potency35.197340
1-[4-amino-7-[3-(2-methoxyethylamino)propyl]-5-(4-methylphenyl)-6-pyrrolo[2,3-d]pyrimidinyl]-2-fluoroethanoneHomo sapiens (human)Potency9.388530
cep 33779Homo sapiens (human)Potency3.731640
entecavirHomo sapiens (human)Potency12.900740
2-[5-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxy-2-pyrrolylidene]indoleHomo sapiens (human)Potency1.464940
sr9011Homo sapiens (human)Potency19.924240
4-[[9-[(3R)-3-oxolanyl]-8-(2,4,6-trifluoroanilino)-2-purinyl]amino]-1-cyclohexanolHomo sapiens (human)Potency11.961040
N-hydroxy-3-[4-[[2-(2-methyl-1H-indol-3-yl)ethylamino]methyl]phenyl]-2-propenamideHomo sapiens (human)Potency0.079340
3-[(5-tert-butyl-1H-imidazol-4-yl)methylidene]-6-(phenylmethylene)piperazine-2,5-dioneHomo sapiens (human)Potency35.314320
gsk837149aHomo sapiens (human)Potency21.848240
N-[4-(3-chloro-4-fluoroanilino)-7-[[(3S)-3-oxolanyl]oxy]-6-quinazolinyl]-4-(dimethylamino)-2-butenamideHomo sapiens (human)Potency18.209540
N-[4-(3-chloro-4-fluoroanilino)-7-methoxy-6-quinazolinyl]-4-(1-piperidinyl)-2-butenamideHomo sapiens (human)Potency6.590440
wnt-c59Homo sapiens (human)Potency16.136240
5-[1-(2-hydroxyethyl)-3-pyridin-4-yl-4-pyrazolyl]-2,3-dihydroinden-1-one oximeHomo sapiens (human)Potency29.974130
d159687Homo sapiens (human)Potency23.159240
HG-10-102-01Homo sapiens (human)Potency6.662920
N-[(5-methyl-2-furanyl)methylideneamino]-2-phenoxybenzamideHomo sapiens (human)Potency22.161730
N-[5-[[6-[3-(1,3-dioxo-2-isoindolyl)phenyl]-4-pyrimidinyl]amino]-2-methylphenyl]methanesulfonamideHomo sapiens (human)Potency23.492040
[4-[2-(1H-indazol-3-yl)ethenyl]phenyl]-(1-piperazinyl)methanoneHomo sapiens (human)Potency1.938340
gsk-2816126Homo sapiens (human)Potency20.869040
N-cyclopropyl-3-[3-[[cyclopropyl(oxo)methyl]amino]-1H-indazol-6-yl]benzamideHomo sapiens (human)Potency1.921040
1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-[4-methyl-3-[[2-oxo-3-(1H-pyrrol-2-ylmethylidene)-1H-indol-6-yl]amino]phenyl]ureaHomo sapiens (human)Potency26.438040
9-(3,5-dimethoxyphenyl)-1-[4-(1-piperazinyl)-3-(trifluoromethyl)phenyl]-2-benzo[h][1,6]naphthyridinoneHomo sapiens (human)Potency3.271340
agi-6780Homo sapiens (human)Potency23.422640
khs101Homo sapiens (human)Potency14.862140
GSK1059615Homo sapiens (human)Potency0.139840
3-[4-[3-(3-fluorophenyl)-3-oxoprop-1-enyl]-1-methyl-2-pyrrolyl]-N-hydroxy-2-propenamideHomo sapiens (human)Potency19.924240
9-(1-methyl-4-pyrazolyl)-1-[1-(1-oxoprop-2-enyl)-2,3-dihydroindol-6-yl]-2-benzo[h][1,6]naphthyridinoneHomo sapiens (human)Potency4.142740
[4-amino-2-[2-methoxy-4-(4-methyl-1-piperazinyl)anilino]-5-thiazolyl]-(2,6-dichlorophenyl)methanoneHomo sapiens (human)Potency11.252240
N-[2-methyl-5-[oxo-[3-(1-oxoprop-2-enylamino)-5-(trifluoromethyl)anilino]methyl]phenyl]-5-isoxazolecarboxamideHomo sapiens (human)Potency22.208040
3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-[4-(diethylamino)butylamino]-1-methyl-4H-pyrimido[4,5-d]pyrimidin-2-oneHomo sapiens (human)Potency20.362040
(8R,9S,13S,14R,17R)-17-ethynyl-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diolHomo sapiens (human)Potency19.285740
at 9283Homo sapiens (human)Potency2.812040
akt-i-1,2 compoundHomo sapiens (human)Potency21.000440
chir 258Homo sapiens (human)Potency11.826440
acyclovirHomo sapiens (human)Potency0.295710
osi 027Homo sapiens (human)Potency0.636740
3-methyladenineHomo sapiens (human)Potency0.218040
clozapineHomo sapiens (human)Potency34.669430
didanosineHomo sapiens (human)Potency34.295440
ganciclovirHomo sapiens (human)Potency15.882440
valacyclovirHomo sapiens (human)Potency17.247120
sildenafilHomo sapiens (human)Potency12.025040
chir-124Homo sapiens (human)Potency0.465540
raltitrexedHomo sapiens (human)Potency0.024340
vardenafilHomo sapiens (human)Potency7.207840
hli 373Homo sapiens (human)Potency4.314840
bl 4162aHomo sapiens (human)Potency22.846540
pemetrexedHomo sapiens (human)Potency0.390340
xav939Homo sapiens (human)Potency24.366740
hesperadinHomo sapiens (human)Potency0.240240
nintedanibHomo sapiens (human)Potency1.422540
heliomycinHomo sapiens (human)Potency31.970930
bms 536924Homo sapiens (human)Potency5.876040
amg531Homo sapiens (human)Potency13.924840
ver 52296Homo sapiens (human)Potency0.089040
sb-590885Homo sapiens (human)Potency29.045640
sta 9090Homo sapiens (human)Potency0.072540
pf-477736Homo sapiens (human)Potency0.541940
bay 80-6946Homo sapiens (human)Potency0.764040
bix 02189Homo sapiens (human)Potency22.924440
carbazochrome sodium sulfonateHomo sapiens (human)Potency0.005320
s-1530Homo sapiens (human)Potency30.356230
6-bromoindirubin-3'-acetoximeHomo sapiens (human)Potency6.789840

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
curcuminHomo sapiens (human)AbsAC35_uM40.250010
3-(2-fluorophenyl)-6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineHomo sapiens (human)AbsAC35_uM137.490010