Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
1-(2,4-dihydroxyphenyl)-3-(4-hydroxyphenyl)-2-propen-1-one | Homo sapiens (human) | Potency | 18.9650 | 4 | 0 |
taxifolin | Homo sapiens (human) | Potency | 33.1734 | 3 | 0 |
aminocaproic acid | Homo sapiens (human) | Potency | 18.1810 | 3 | 0 |
acetylcysteine | Homo sapiens (human) | Potency | 0.0019 | 1 | 0 |
3-(4-hydroxy-3-methoxyphenyl)prop-2-enoic acid | Homo sapiens (human) | Potency | 11.0633 | 2 | 0 |
histamine | Homo sapiens (human) | Potency | 14.6921 | 2 | 0 |
melatonin | Homo sapiens (human) | Potency | 2.1250 | 4 | 0 |
spermidine | Homo sapiens (human) | Potency | 26.3506 | 1 | 0 |
taurine | Homo sapiens (human) | Potency | 0.9350 | 1 | 0 |
b 844-39 | Homo sapiens (human) | Potency | 23.8756 | 4 | 0 |
huperzine a | Homo sapiens (human) | Potency | 15.0321 | 3 | 0 |
pk 11195 | Homo sapiens (human) | Potency | 16.4869 | 3 | 0 |
pd 173074 | Homo sapiens (human) | Potency | 18.2095 | 4 | 0 |
N-(4-hydroxyphenyl)-3,7-dimethyl-9-(2,6,6-trimethyl-1-cyclohexenyl)nona-2,4,6,8-tetraenamide | Homo sapiens (human) | Potency | 6.0425 | 4 | 0 |
nitrofurazone | Homo sapiens (human) | Potency | 32.7752 | 4 | 0 |
tacrine | Homo sapiens (human) | Potency | 16.2855 | 4 | 0 |
abt 702 | Homo sapiens (human) | Potency | 31.1248 | 4 | 0 |
acetaminophen | Homo sapiens (human) | Potency | 25.9141 | 2 | 0 |
tyrphostin ag 1024 | Homo sapiens (human) | Potency | 33.4916 | 4 | 0 |
rtki cpd | Homo sapiens (human) | Potency | 13.5234 | 4 | 0 |
alfuzosin | Homo sapiens (human) | Potency | 4.1763 | 1 | 0 |
altretamine | Homo sapiens (human) | Potency | 1.0490 | 1 | 0 |
amantadine | Homo sapiens (human) | Potency | 25.6252 | 4 | 0 |
theophylline | Homo sapiens (human) | Potency | 22.0858 | 3 | 0 |
amiodarone | Homo sapiens (human) | Potency | 8.5870 | 4 | 0 |
dan 2163 | Homo sapiens (human) | Potency | 10.4666 | 2 | 0 |
amlexanox | Homo sapiens (human) | Potency | 25.0118 | 3 | 0 |
amoxapine | Homo sapiens (human) | Potency | 15.5994 | 4 | 0 |
aniracetam | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
arecoline | Homo sapiens (human) | Potency | 17.5434 | 3 | 0 |
aspirin | Homo sapiens (human) | Potency | 14.9222 | 4 | 0 |
azathioprine | Homo sapiens (human) | Potency | 2.9538 | 4 | 0 |
azelastine | Homo sapiens (human) | Potency | 3.9348 | 4 | 0 |
benserazide | Homo sapiens (human) | Potency | 28.5172 | 4 | 0 |
berberine | Homo sapiens (human) | Potency | 8.3572 | 4 | 0 |
betaxolol | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
bicalutamide | Homo sapiens (human) | Potency | 2.3239 | 4 | 0 |
2-cyano-3-(3,4-dihydroxyphenyl)-N-(phenylmethyl)-2-propenamide | Homo sapiens (human) | Potency | 21.6390 | 4 | 0 |
ro 31-8425 | Homo sapiens (human) | Potency | 18.2095 | 4 | 0 |
seratrodast | Homo sapiens (human) | Potency | 0.0037 | 1 | 0 |
bufexamac | Homo sapiens (human) | Potency | 7.4484 | 4 | 0 |
busulfan | Homo sapiens (human) | Potency | 8.3164 | 2 | 0 |
caffeic acid | Homo sapiens (human) | Potency | 17.8509 | 4 | 0 |
verapamil | Homo sapiens (human) | Potency | 0.0054 | 1 | 0 |
calmidazolium | Homo sapiens (human) | Potency | 20.4933 | 4 | 0 |
N-[4-methyl-1-oxo-1-(1-oxohexan-2-ylamino)pentan-2-yl]carbamic acid (phenylmethyl) ester | Homo sapiens (human) | Potency | 9.1947 | 2 | 0 |
camostat | Homo sapiens (human) | Potency | 8.5870 | 4 | 0 |
capsaicin | Homo sapiens (human) | Potency | 10.9906 | 4 | 0 |
carbidopa | Homo sapiens (human) | Potency | 23.4850 | 1 | 0 |
carisoprodol | Homo sapiens (human) | Potency | 0.0105 | 1 | 0 |
carmofur | Homo sapiens (human) | Potency | 12.9912 | 4 | 0 |
carmustine | Homo sapiens (human) | Potency | 0.0235 | 1 | 0 |
carvedilol | Homo sapiens (human) | Potency | 15.4016 | 3 | 0 |
celecoxib | Homo sapiens (human) | Potency | 12.5211 | 4 | 0 |
chelerythrine | Homo sapiens (human) | Potency | 7.4487 | 4 | 0 |
chlorambucil | Homo sapiens (human) | Potency | 23.1748 | 4 | 0 |
chlorhexidine | Homo sapiens (human) | Potency | 5.9772 | 4 | 0 |
chlormezanone | Homo sapiens (human) | Potency | 15.7991 | 3 | 0 |
chlorothiazide | Homo sapiens (human) | Potency | 0.0148 | 1 | 0 |
chloroxine | Homo sapiens (human) | Potency | 9.8641 | 4 | 0 |
ciclopirox | Homo sapiens (human) | Potency | 5.9719 | 4 | 0 |
cilostazol | Homo sapiens (human) | Potency | 0.0469 | 1 | 0 |
ciprofibrate | Homo sapiens (human) | Potency | 29.8920 | 4 | 0 |
ciprofloxacin | Homo sapiens (human) | Potency | 0.0782 | 2 | 0 |
cisplatin | Homo sapiens (human) | Potency | 11.7451 | 2 | 0 |
citalopram | Homo sapiens (human) | Potency | 16.6996 | 3 | 0 |
N-[4-(4-morpholinyl)butyl]-2-benzofurancarboxamide | Homo sapiens (human) | Potency | 26.3506 | 1 | 0 |
clofibrate | Homo sapiens (human) | Potency | 23.4850 | 1 | 0 |
clomiphene | Homo sapiens (human) | Potency | 24.6301 | 4 | 0 |
clomipramine | Homo sapiens (human) | Potency | 1.8294 | 4 | 0 |
clotrimazole | Homo sapiens (human) | Potency | 20.2769 | 4 | 0 |
cromoglycate | Homo sapiens (human) | Potency | 0.0030 | 1 | 0 |
crotamiton | Homo sapiens (human) | Potency | 29.6831 | 3 | 0 |
cyclobenzaprine | Homo sapiens (human) | Potency | 18.7786 | 4 | 0 |
cyclosporine | Homo sapiens (human) | Potency | 17.6277 | 2 | 0 |
cyproheptadine | Homo sapiens (human) | Potency | 17.0288 | 4 | 0 |
indibulin | Homo sapiens (human) | Potency | 0.1321 | 4 | 0 |
dacarbazine | Homo sapiens (human) | Potency | 18.6548 | 2 | 0 |
diclofenac sodium | Homo sapiens (human) | Potency | 20.6999 | 3 | 0 |
dichlorphenamide | Homo sapiens (human) | Potency | 0.4686 | 1 | 0 |
dienestrol | Homo sapiens (human) | Potency | 28.3090 | 4 | 0 |
diethylstilbestrol | Homo sapiens (human) | Potency | 27.3399 | 4 | 0 |
3,3'-diindolylmethane | Homo sapiens (human) | Potency | 6.4514 | 4 | 0 |
dilacor xr | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
diphenhydramine | Homo sapiens (human) | Potency | 29.0189 | 3 | 0 |
dipyridamole | Homo sapiens (human) | Potency | 24.9957 | 4 | 0 |
disulfiram | Homo sapiens (human) | Potency | 0.0389 | 4 | 0 |
domperidone | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
doxazosin | Homo sapiens (human) | Potency | 21.1987 | 3 | 0 |
dyphylline | Homo sapiens (human) | Potency | 13.2066 | 1 | 0 |
econazole | Homo sapiens (human) | Potency | 25.4160 | 4 | 0 |
efavirenz | Homo sapiens (human) | Potency | 24.9178 | 4 | 0 |
embelin | Homo sapiens (human) | Potency | 29.9439 | 3 | 0 |
emodin | Homo sapiens (human) | Potency | 29.5659 | 1 | 0 |
enoxacin | Homo sapiens (human) | Potency | 0.0026 | 1 | 0 |
ethosuximide | Homo sapiens (human) | Potency | 28.3292 | 2 | 0 |
etodolac | Homo sapiens (human) | Potency | 26.3506 | 1 | 0 |
famotidine | Homo sapiens (human) | Potency | 16.3600 | 3 | 0 |
felbamate | Homo sapiens (human) | Potency | 10.6602 | 3 | 0 |
fenbendazole | Homo sapiens (human) | Potency | 1.4557 | 4 | 0 |
fenofibrate | Homo sapiens (human) | Potency | 8.3136 | 2 | 0 |
flecainide | Homo sapiens (human) | Potency | 33.3202 | 3 | 0 |
flucytosine | Homo sapiens (human) | Potency | 15.9307 | 2 | 0 |
fluphenazine | Homo sapiens (human) | Potency | 30.0576 | 4 | 0 |
flumazenil | Homo sapiens (human) | Potency | 18.3458 | 2 | 0 |
1-[bis(4-fluorophenyl)methyl]-4-(3-phenylprop-2-enyl)piperazine | Homo sapiens (human) | Potency | 20.5438 | 3 | 0 |
fluorouracil | Homo sapiens (human) | Potency | 6.9832 | 4 | 0 |
flurbiprofen | Homo sapiens (human) | Potency | 19.9970 | 3 | 0 |
flutamide | Homo sapiens (human) | Potency | 11.0826 | 4 | 0 |
luvox | Homo sapiens (human) | Potency | 24.0610 | 4 | 0 |
fomepizole | Homo sapiens (human) | Potency | 0.0294 | 4 | 0 |
furosemide | Homo sapiens (human) | Potency | 0.0026 | 1 | 0 |
gabapentin | Homo sapiens (human) | Potency | 34.1854 | 4 | 0 |
gabexate | Homo sapiens (human) | Potency | 6.6190 | 1 | 0 |
gbr 12935 | Homo sapiens (human) | Potency | 24.2703 | 4 | 0 |
gemfibrozil | Homo sapiens (human) | Potency | 36.2093 | 4 | 0 |
gentian violet | Homo sapiens (human) | Potency | 0.2727 | 4 | 0 |
gliclazide | Homo sapiens (human) | Potency | 22.0830 | 4 | 0 |
glimepiride | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
glipizide | Homo sapiens (human) | Potency | 21.0699 | 4 | 0 |
gö6983 | Homo sapiens (human) | Potency | 0.0281 | 4 | 0 |
go 6976 | Homo sapiens (human) | Potency | 3.7827 | 4 | 0 |
gossypol | Homo sapiens (human) | Potency | 13.5306 | 4 | 0 |
N-[2-(4-bromocinnamylamino)ethyl]isoquinoline-5-sulfonamide | Homo sapiens (human) | Potency | 3.0204 | 4 | 0 |
fasudil | Homo sapiens (human) | Potency | 13.1812 | 2 | 0 |
ha14-1 | Homo sapiens (human) | Potency | 25.7962 | 4 | 0 |
haloperidol | Homo sapiens (human) | Potency | 23.1592 | 4 | 0 |
hexestrol | Homo sapiens (human) | Potency | 1.2848 | 4 | 0 |
hydroxychloroquine | Homo sapiens (human) | Potency | 24.3146 | 4 | 0 |
hydroxyurea | Homo sapiens (human) | Potency | 14.1064 | 4 | 0 |
atropine sulfate | Homo sapiens (human) | Potency | 18.0684 | 4 | 0 |
phenelzine | Homo sapiens (human) | Potency | 12.5959 | 4 | 0 |
idebenone | Homo sapiens (human) | Potency | 32.4796 | 4 | 0 |
ifosfamide | Homo sapiens (human) | Potency | 22.8319 | 4 | 0 |
indapamide | Homo sapiens (human) | Potency | 28.0642 | 4 | 0 |
indomethacin | Homo sapiens (human) | Potency | 15.4754 | 3 | 0 |
ipriflavone | Homo sapiens (human) | Potency | 33.1734 | 2 | 0 |
isoconazole | Homo sapiens (human) | Potency | 28.8500 | 4 | 0 |
isoniazid | Homo sapiens (human) | Potency | 0.0010 | 1 | 0 |
isoproterenol | Homo sapiens (human) | Potency | 14.4354 | 4 | 0 |
isradipine | Homo sapiens (human) | Potency | 28.1437 | 4 | 0 |
whi p97 | Homo sapiens (human) | Potency | 0.1413 | 4 | 0 |
ketanserin | Homo sapiens (human) | Potency | 2.2324 | 2 | 0 |
ketoprofen | Homo sapiens (human) | Potency | 16.0266 | 4 | 0 |
ketorolac | Homo sapiens (human) | Potency | 4.4587 | 4 | 0 |
ketotifen | Homo sapiens (human) | Potency | 17.7923 | 4 | 0 |
5-isoquinolinesulfonic acid [4-[2-[5-isoquinolinylsulfonyl(methyl)amino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl]phenyl] ester | Homo sapiens (human) | Potency | 17.7575 | 4 | 0 |
lamotrigine | Homo sapiens (human) | Potency | 34.2954 | 4 | 0 |
lansoprazole | Homo sapiens (human) | Potency | 30.4419 | 3 | 0 |
beta-lapachone | Homo sapiens (human) | Potency | 19.0476 | 4 | 0 |
leflunomide | Homo sapiens (human) | Potency | 16.1362 | 4 | 0 |
letrozole | Homo sapiens (human) | Potency | 20.0413 | 4 | 0 |
lg 100268 | Homo sapiens (human) | Potency | 16.6261 | 1 | 0 |
linopirdine | Homo sapiens (human) | Potency | 15.7220 | 2 | 0 |
liranaftate | Homo sapiens (human) | Potency | 0.0042 | 1 | 0 |
lomefloxacin | Homo sapiens (human) | Potency | 0.7427 | 1 | 0 |
lomustine | Homo sapiens (human) | Potency | 0.0166 | 1 | 0 |
loperamide | Homo sapiens (human) | Potency | 19.2857 | 4 | 0 |
loratadine | Homo sapiens (human) | Potency | 25.6342 | 4 | 0 |
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-one | Homo sapiens (human) | Potency | 16.7856 | 4 | 0 |
4-(dimethylamino)-n-(7-(hydroxyamino)-7-oxoheptyl)benzamide | Homo sapiens (human) | Potency | 0.5183 | 4 | 0 |
maprotiline | Homo sapiens (human) | Potency | 22.2774 | 4 | 0 |
mebendazole | Homo sapiens (human) | Potency | 0.7718 | 4 | 0 |
mechlorethamine | Homo sapiens (human) | Potency | 34.5227 | 3 | 0 |
meclizine | Homo sapiens (human) | Potency | 18.9999 | 4 | 0 |
mefloquine hydrochloride | Homo sapiens (human) | Potency | 25.3465 | 4 | 0 |
vitamin k 3 | Homo sapiens (human) | Potency | 26.1324 | 4 | 0 |
metformin | Homo sapiens (human) | Potency | 0.0012 | 1 | 0 |
methocarbamol | Homo sapiens (human) | Potency | 0.0372 | 1 | 0 |
methoxsalen | Homo sapiens (human) | Potency | 3.3173 | 2 | 0 |
nocodazole | Homo sapiens (human) | Potency | 0.0236 | 4 | 0 |
3,7-bis(dimethylamino)phenothiazin-5-ium | Homo sapiens (human) | Potency | 5.0265 | 4 | 0 |
metronidazole | Homo sapiens (human) | Potency | 0.1049 | 1 | 0 |
mianserin | Homo sapiens (human) | Potency | 20.4933 | 4 | 0 |
miconazole | Homo sapiens (human) | Potency | 22.9938 | 4 | 0 |
mirtazapine | Homo sapiens (human) | Potency | 5.2576 | 1 | 0 |
mitotane | Homo sapiens (human) | Potency | 24.0611 | 4 | 0 |
mitoxantrone | Homo sapiens (human) | Potency | 0.1063 | 3 | 0 |
entinostat | Homo sapiens (human) | Potency | 3.9273 | 4 | 0 |
6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-isobenzofuran-5-yl)-4-methyl-4-hexenoic acid 2-(4-morpholinyl)ethyl ester | Homo sapiens (human) | Potency | 2.0070 | 4 | 0 |
6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-isobenzofuran-5-yl)-4-methyl-4-hexenoic acid | Homo sapiens (human) | Potency | 2.4752 | 4 | 0 |
nafamostat | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
naftopidil | Homo sapiens (human) | Potency | 14.8768 | 3 | 0 |
naratriptan | Homo sapiens (human) | Potency | 1.1810 | 4 | 0 |
niclosamide | Homo sapiens (human) | Potency | 8.9734 | 4 | 0 |
nifekalant | Homo sapiens (human) | Potency | 21.0004 | 4 | 0 |
nilutamide | Homo sapiens (human) | Potency | 9.3495 | 1 | 0 |
nimesulide | Homo sapiens (human) | Potency | 12.8469 | 4 | 0 |
norfloxacin | Homo sapiens (human) | Potency | 23.4850 | 1 | 0 |
nu6102 | Homo sapiens (human) | Potency | 13.9995 | 4 | 0 |
o(6)-benzylguanine | Homo sapiens (human) | Potency | 22.8464 | 4 | 0 |
ofloxacin | Homo sapiens (human) | Potency | 20.9310 | 2 | 0 |
olprinone | Homo sapiens (human) | Potency | 0.0187 | 1 | 0 |
omeprazole | Homo sapiens (human) | Potency | 26.4551 | 3 | 0 |
ondansetron | Homo sapiens (human) | Potency | 16.1625 | 3 | 0 |
5-[3-(benzenesulfonamido)phenyl]-N-hydroxypent-2-en-4-ynamide | Homo sapiens (human) | Potency | 1.2386 | 4 | 0 |
oxibendazole | Homo sapiens (human) | Potency | 0.0063 | 4 | 0 |
oxymetazoline | Homo sapiens (human) | Potency | 34.1854 | 4 | 0 |
pantoprazole | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
papaverine | Homo sapiens (human) | Potency | 21.6390 | 4 | 0 |
pd 153035 | Homo sapiens (human) | Potency | 0.7593 | 4 | 0 |
pd 98059 | Homo sapiens (human) | Potency | 10.9860 | 2 | 0 |
pentamidine | Homo sapiens (human) | Potency | 11.1906 | 4 | 0 |
perhexiline | Homo sapiens (human) | Potency | 16.6311 | 4 | 0 |
phenoxybenzamine | Homo sapiens (human) | Potency | 0.0332 | 1 | 0 |
phenylmethylsulfonyl fluoride | Homo sapiens (human) | Potency | 2.2327 | 3 | 0 |
phloretin | Homo sapiens (human) | Potency | 1.8064 | 4 | 0 |
moxonidine | Homo sapiens (human) | Potency | 0.0132 | 1 | 0 |
3,3',4,5'-tetrahydroxystilbene | Homo sapiens (human) | Potency | 18.7167 | 4 | 0 |
pimobendan | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
pioglitazone | Homo sapiens (human) | Potency | 0.1552 | 2 | 0 |
ono 1078 | Homo sapiens (human) | Potency | 18.1476 | 4 | 0 |
praziquantel | Homo sapiens (human) | Potency | 33.3936 | 2 | 0 |
prazosin | Homo sapiens (human) | Potency | 26.1324 | 4 | 0 |
primidone | Homo sapiens (human) | Potency | 13.6482 | 4 | 0 |
probucol | Homo sapiens (human) | Potency | 11.0790 | 3 | 0 |
procarbazine | Homo sapiens (human) | Potency | 0.0017 | 1 | 0 |
propafenone | Homo sapiens (human) | Potency | 23.1018 | 4 | 0 |
pyrimethamine | Homo sapiens (human) | Potency | 5.3522 | 4 | 0 |
pyroxamide | Homo sapiens (human) | Potency | 4.0267 | 4 | 0 |
3-[(3,5-dibromo-4-hydroxyphenyl)methylidene]-5-iodo-1H-indol-2-one | Homo sapiens (human) | Potency | 20.4314 | 4 | 0 |
raloxifene | Homo sapiens (human) | Potency | 7.8286 | 4 | 0 |
opc 12759 | Homo sapiens (human) | Potency | 35.1973 | 2 | 0 |
hydrochlorothiazide | Homo sapiens (human) | Potency | 2.6438 | 4 | 0 |
resveratrol | Homo sapiens (human) | Potency | 16.7364 | 4 | 0 |
riluzole | Homo sapiens (human) | Potency | 24.3667 | 4 | 0 |
rimantadine | Homo sapiens (human) | Potency | 0.0118 | 1 | 0 |
risperidone | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
rofecoxib | Homo sapiens (human) | Potency | 25.6023 | 3 | 0 |
sb 206553 | Homo sapiens (human) | Potency | 19.2380 | 4 | 0 |
sb 239063 | Homo sapiens (human) | Potency | 24.3234 | 3 | 0 |
sb 202190 | Homo sapiens (human) | Potency | 21.0004 | 4 | 0 |
sibutramine | Homo sapiens (human) | Potency | 27.1216 | 4 | 0 |
sotalol | Homo sapiens (human) | Potency | 19.0932 | 4 | 0 |
imatinib | Homo sapiens (human) | Potency | 29.8494 | 4 | 0 |
SU5402 | Homo sapiens (human) | Potency | 31.4677 | 4 | 0 |
SU6656 | Homo sapiens (human) | Potency | 5.4683 | 4 | 0 |
vorinostat | Homo sapiens (human) | Potency | 2.6525 | 4 | 0 |
sulfamethizole | Homo sapiens (human) | Potency | 13.7853 | 4 | 0 |
sulfanilamide | Homo sapiens (human) | Potency | 26.3506 | 1 | 0 |
copal rosin varnish | Homo sapiens (human) | Potency | 10.3002 | 4 | 0 |
sulpiride | Homo sapiens (human) | Potency | 26.9236 | 2 | 0 |
sumatriptan | Homo sapiens (human) | Potency | 0.0033 | 1 | 0 |
suramin | Homo sapiens (human) | Potency | 10.4760 | 2 | 0 |
2-[4-(1,2-diphenylbut-1-enyl)phenoxy]-N,N-dimethylethanamine | Homo sapiens (human) | Potency | 20.1334 | 4 | 0 |
tazarotene | Homo sapiens (human) | Potency | 0.0148 | 1 | 0 |
terazosin | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
N,6,6-trimethyl-N-(1-naphthalenylmethyl)-1-hept-2-en-4-ynamine | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
tetrahydropapaverine | Homo sapiens (human) | Potency | 24.9178 | 2 | 0 |
thalidomide | Homo sapiens (human) | Potency | 0.0037 | 1 | 0 |
theobromine | Homo sapiens (human) | Potency | 25.9071 | 4 | 0 |
thiotepa | Homo sapiens (human) | Potency | 10.6266 | 4 | 0 |
ticlopidine | Homo sapiens (human) | Potency | 0.0833 | 1 | 0 |
tioconazole | Homo sapiens (human) | Potency | 26.1324 | 4 | 0 |
tiopronin | Homo sapiens (human) | Potency | 37.2212 | 2 | 0 |
tizanidine | Homo sapiens (human) | Potency | 0.5258 | 1 | 0 |
2-[4-(4-chloro-1,2-diphenylbut-1-enyl)phenoxy]-N,N-dimethylethanamine | Homo sapiens (human) | Potency | 2.7804 | 3 | 0 |
tranexamic acid | Homo sapiens (human) | Potency | 11.2780 | 2 | 0 |
2-[[3-(3,4-dimethoxyphenyl)-1-oxoprop-2-enyl]amino]benzoic acid | Homo sapiens (human) | Potency | 23.4850 | 1 | 0 |
2-phenylcyclopropan-1-amine | Homo sapiens (human) | Potency | 23.4850 | 1 | 0 |
retinoic acid | Homo sapiens (human) | Potency | 14.7964 | 4 | 0 |
trifluoperazine | Homo sapiens (human) | Potency | 14.8210 | 4 | 0 |
trimetrexate | Homo sapiens (human) | Potency | 1.5762 | 4 | 0 |
trioxsalen | Homo sapiens (human) | Potency | 17.2491 | 4 | 0 |
2,3-bis[amino-[(2-aminophenyl)thio]methylidene]butanedinitrile | Homo sapiens (human) | Potency | 26.7888 | 4 | 0 |
venlafaxine | Homo sapiens (human) | Potency | 29.0189 | 3 | 0 |
xylometazoline | Homo sapiens (human) | Potency | 0.0012 | 1 | 0 |
3-(5'-hydroxymethyl-2'-furyl)-1-benzylindazole | Homo sapiens (human) | Potency | 8.8140 | 4 | 0 |
ici 204,219 | Homo sapiens (human) | Potency | 20.5627 | 4 | 0 |
zm 336372 | Homo sapiens (human) | Potency | 0.6854 | 4 | 0 |
mitomycin | Homo sapiens (human) | Potency | 0.0362 | 4 | 0 |
phentolamine | Homo sapiens (human) | Potency | 15.7220 | 2 | 0 |
thyroxine | Homo sapiens (human) | Potency | 3.0353 | 2 | 0 |
chloramphenicol | Homo sapiens (human) | Potency | 0.0209 | 1 | 0 |
vincristine | Homo sapiens (human) | Potency | 0.0020 | 4 | 0 |
phenylephrine | Homo sapiens (human) | Potency | 0.0264 | 1 | 0 |
levodopa | Homo sapiens (human) | Potency | 0.3722 | 1 | 0 |
cytidine | Homo sapiens (human) | Potency | 0.0386 | 4 | 0 |
cycloheximide | Homo sapiens (human) | Potency | 0.2332 | 4 | 0 |
caffeine citrate | Homo sapiens (human) | Potency | 13.2066 | 1 | 0 |
cytarabine | Homo sapiens (human) | Potency | 0.4686 | 1 | 0 |
pantothenic acid | Homo sapiens (human) | Potency | 28.7026 | 4 | 0 |
rotenone | Homo sapiens (human) | Potency | 2.6196 | 4 | 0 |
7,8-dimethyl-10-[(2R,3R,4S)-2,3,4,5-tetrahydroxypentyl]benzo[g]pteridine-2,4-dione | Homo sapiens (human) | Potency | 29.7620 | 2 | 0 |
synephrine | Homo sapiens (human) | Potency | 0.0013 | 1 | 0 |
monobenzone | Homo sapiens (human) | Potency | 5.0127 | 4 | 0 |
phenformin | Homo sapiens (human) | Potency | 16.9956 | 4 | 0 |
pyrazolanthrone | Homo sapiens (human) | Potency | 17.7724 | 4 | 0 |
rhein | Homo sapiens (human) | Potency | 34.0429 | 1 | 0 |
indirubin | Homo sapiens (human) | Potency | 15.5711 | 4 | 0 |
osthol | Homo sapiens (human) | Potency | 17.2809 | 3 | 0 |
cytisine | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
podophyllotoxin | Homo sapiens (human) | Potency | 0.0042 | 1 | 0 |
physcione | Homo sapiens (human) | Potency | 0.5787 | 2 | 0 |
azomycin | Homo sapiens (human) | Potency | 5.2576 | 1 | 0 |
docosanol | Homo sapiens (human) | Potency | 0.0026 | 1 | 0 |
antimycin a | Homo sapiens (human) | Potency | 0.0706 | 4 | 0 |
daminozide | Homo sapiens (human) | Potency | 30.0576 | 4 | 0 |
stavudine | Homo sapiens (human) | Potency | 34.0429 | 1 | 0 |
cladribine | Homo sapiens (human) | Potency | 0.3187 | 4 | 0 |
2,4,5-trimethoxybenzaldehyde | Homo sapiens (human) | Potency | 36.2093 | 4 | 0 |
buthionine sulfoximine | Homo sapiens (human) | Potency | 14.8180 | 1 | 0 |
vidarabine | Homo sapiens (human) | Potency | 9.2089 | 4 | 0 |
octocrylene | Homo sapiens (human) | Potency | 0.0042 | 1 | 0 |
zalcitabine | Homo sapiens (human) | Potency | 0.0012 | 1 | 0 |
usnic acid | Homo sapiens (human) | Potency | 0.0042 | 1 | 0 |
camptothecin | Homo sapiens (human) | Potency | 0.0095 | 4 | 0 |
chloropyramine | Homo sapiens (human) | Potency | 23.5629 | 4 | 0 |
parbendazole | Homo sapiens (human) | Potency | 1.1903 | 4 | 0 |
thiamphenicol | Homo sapiens (human) | Potency | 16.2784 | 4 | 0 |
pizotyline | Homo sapiens (human) | Potency | 28.5172 | 4 | 0 |
(3R)-6,7-dimethoxy-3-[(5R)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]-3H-isobenzofuran-1-one | Homo sapiens (human) | Potency | 0.1270 | 3 | 0 |
du-21220 | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
canadine | Homo sapiens (human) | Potency | 19.7447 | 3 | 0 |
flubendazole | Homo sapiens (human) | Potency | 0.7064 | 4 | 0 |
dobutamine | Homo sapiens (human) | Potency | 26.6235 | 4 | 0 |
halofantrine | Homo sapiens (human) | Potency | 6.2162 | 2 | 0 |
lonidamine | Homo sapiens (human) | Potency | 0.0037 | 1 | 0 |
ng-nitroarginine methyl ester | Homo sapiens (human) | Potency | 0.0148 | 1 | 0 |
oxfendazole | Homo sapiens (human) | Potency | 13.8506 | 4 | 0 |
nitazoxanide | Homo sapiens (human) | Potency | 20.8956 | 4 | 0 |
epirubicin | Homo sapiens (human) | Potency | 0.1210 | 4 | 0 |
s-2678 | Homo sapiens (human) | Potency | 25.7115 | 4 | 0 |
clorsulon | Homo sapiens (human) | Potency | 23.4850 | 2 | 0 |
butoconazole | Homo sapiens (human) | Potency | 35.1973 | 2 | 0 |
nicorandil | Homo sapiens (human) | Potency | 33.5977 | 3 | 0 |
fazarabine | Homo sapiens (human) | Potency | 5.7270 | 4 | 0 |
amonafide | Homo sapiens (human) | Potency | 9.9314 | 4 | 0 |
avobenzone | Homo sapiens (human) | Potency | 1.6168 | 4 | 0 |
pramiracetam | Homo sapiens (human) | Potency | 16.6261 | 1 | 0 |
fenticonazole | Homo sapiens (human) | Potency | 32.7752 | 4 | 0 |
lovastatin | Homo sapiens (human) | Potency | 15.4576 | 4 | 0 |
flupirtine | Homo sapiens (human) | Potency | 22.8465 | 4 | 0 |
2-[[1-(2-amino-4-thiazolyl)-2-[[(2S,3S)-2-methyl-4-oxo-1-sulfo-3-azetidinyl]amino]-2-oxoethylidene]amino]oxy-2-methylpropanoic acid | Homo sapiens (human) | Potency | 19.7929 | 2 | 0 |
simvastatin | Homo sapiens (human) | Potency | 14.4081 | 4 | 0 |
balsalazide | Homo sapiens (human) | Potency | 17.8500 | 4 | 0 |
pravastatin | Homo sapiens (human) | Potency | 27.0522 | 2 | 0 |
mifepristone | Homo sapiens (human) | Potency | 0.2828 | 4 | 0 |
itraconazole | Homo sapiens (human) | Potency | 0.8333 | 1 | 0 |
nitrogenase stabilizing-protective protein, bacteria | Homo sapiens (human) | Potency | 4.0432 | 4 | 0 |
sarafloxacin | Homo sapiens (human) | Potency | 13.5596 | 3 | 0 |
imiquimod | Homo sapiens (human) | Potency | 15.3406 | 4 | 0 |
adapalene | Homo sapiens (human) | Potency | 3.2452 | 3 | 0 |
sparfloxacin | Homo sapiens (human) | Potency | 10.2232 | 1 | 0 |
clopidogrel | Homo sapiens (human) | Potency | 35.1973 | 2 | 0 |
topotecan | Homo sapiens (human) | Potency | 0.0262 | 4 | 0 |
aripiprazole | Homo sapiens (human) | Potency | 13.0464 | 4 | 0 |
sipatrigine | Homo sapiens (human) | Potency | 16.6261 | 1 | 0 |
monatepil | Homo sapiens (human) | Potency | 16.1741 | 4 | 0 |
duloxetine | Homo sapiens (human) | Potency | 4.4170 | 4 | 0 |
irinotecan | Homo sapiens (human) | Potency | 0.4144 | 4 | 0 |
ziprasidone | Homo sapiens (human) | Potency | 22.8465 | 4 | 0 |
2-[11-[3-(dimethylamino)propylidene]-6H-benzo[c][1]benzoxepin-2-yl]acetic acid | Homo sapiens (human) | Potency | 19.5484 | 4 | 0 |
adefovir dipivoxil | Homo sapiens (human) | Potency | 0.3570 | 4 | 0 |
LSM-1535 | Homo sapiens (human) | Potency | 0.0010 | 1 | 0 |
lincomycin monohydrochloride | Homo sapiens (human) | Potency | 2.3485 | 1 | 0 |
plerixafor | Homo sapiens (human) | Potency | 4.6859 | 1 | 0 |
oseltamivir | Homo sapiens (human) | Potency | 0.0074 | 1 | 0 |
ginkgolide b | Homo sapiens (human) | Potency | 14.8836 | 3 | 0 |
secoisolariciresinol | Homo sapiens (human) | Potency | 0.4241 | 4 | 0 |
bendamustine | Homo sapiens (human) | Potency | 21.3838 | 4 | 0 |
mizolastine | Homo sapiens (human) | Potency | 24.5520 | 4 | 0 |
cgs 9343b | Homo sapiens (human) | Potency | 15.7220 | 4 | 0 |
prulifloxacin | Homo sapiens (human) | Potency | 11.7704 | 1 | 0 |
balofloxacin | Homo sapiens (human) | Potency | 18.8337 | 4 | 0 |
repaglinide | Homo sapiens (human) | Potency | 0.5258 | 1 | 0 |
telmisartan | Homo sapiens (human) | Potency | 34.1854 | 4 | 0 |
hordenine | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
rilmenidine | Homo sapiens (human) | Potency | 1.8655 | 1 | 0 |
zoledronic acid | Homo sapiens (human) | Potency | 0.0400 | 2 | 0 |
mepivacaine | Homo sapiens (human) | Potency | 13.1901 | 2 | 0 |
diclofensine | Homo sapiens (human) | Potency | 30.3531 | 4 | 0 |
nefiracetam | Homo sapiens (human) | Potency | 2.9566 | 1 | 0 |
uk 68798 | Homo sapiens (human) | Potency | 28.3428 | 4 | 0 |
dapoxetine | Homo sapiens (human) | Potency | 24.2793 | 4 | 0 |
bindarit | Homo sapiens (human) | Potency | 10.7952 | 3 | 0 |
hp 873 | Homo sapiens (human) | Potency | 31.2348 | 4 | 0 |
dexrazoxane | Homo sapiens (human) | Potency | 8.6948 | 3 | 0 |
masoprocol | Homo sapiens (human) | Potency | 15.4235 | 4 | 0 |
voriconazole | Homo sapiens (human) | Potency | 23.4850 | 1 | 0 |
moroxydine | Homo sapiens (human) | Potency | 35.1973 | 4 | 0 |
Suplatast tosilate | Homo sapiens (human) | Potency | 0.0093 | 1 | 0 |
secnidazole | Homo sapiens (human) | Potency | 32.6425 | 3 | 0 |
alibendol | Homo sapiens (human) | Potency | 17.3023 | 3 | 0 |
octylonium | Homo sapiens (human) | Potency | 20.5438 | 3 | 0 |
nedaplatin | Homo sapiens (human) | Potency | 5.8992 | 1 | 0 |
thioxolone | Homo sapiens (human) | Potency | 17.3546 | 4 | 0 |
ubenimex | Homo sapiens (human) | Potency | 26.6235 | 4 | 0 |
tetrahydropalmatine | Homo sapiens (human) | Potency | 14.3814 | 4 | 0 |
honokiol | Homo sapiens (human) | Potency | 29.7620 | 4 | 0 |
picropodophyllin | Homo sapiens (human) | Potency | 0.1007 | 4 | 0 |
tetrandrine | Homo sapiens (human) | Potency | 21.0004 | 4 | 0 |
LSM-4272 | Homo sapiens (human) | Potency | 0.9759 | 4 | 0 |
rosiglitazone | Homo sapiens (human) | Potency | 8.5547 | 2 | 0 |
bexarotene | Homo sapiens (human) | Potency | 24.9382 | 3 | 0 |
s20098 | Homo sapiens (human) | Potency | 19.5363 | 2 | 0 |
albendazole sulfoxide | Homo sapiens (human) | Potency | 22.2080 | 4 | 0 |
4-aminoquinazoline | Homo sapiens (human) | Potency | 35.1973 | 2 | 0 |
matrine | Homo sapiens (human) | Potency | 0.0010 | 1 | 0 |
hydroxyflutamide | Homo sapiens (human) | Potency | 22.0346 | 4 | 0 |
n-(4,4-diphenyl-3-butenyl)nipecotic acid | Homo sapiens (human) | Potency | 10.9190 | 4 | 0 |
nsc-87877 | Homo sapiens (human) | Potency | 16.6813 | 4 | 0 |
mci 9038 | Homo sapiens (human) | Potency | 12.2861 | 4 | 0 |
lopinavir | Homo sapiens (human) | Potency | 26.9970 | 4 | 0 |
10-hydroxycamptothecin | Homo sapiens (human) | Potency | 0.0104 | 4 | 0 |
fotemustine | Homo sapiens (human) | Potency | 0.0148 | 1 | 0 |
sn 38 | Homo sapiens (human) | Potency | 0.1060 | 4 | 0 |
sr141716 | Homo sapiens (human) | Potency | 28.3518 | 4 | 0 |
vanoxerine | Homo sapiens (human) | Potency | 23.8756 | 4 | 0 |
indolactam v | Homo sapiens (human) | Potency | 0.4141 | 2 | 0 |
(6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4,6-dimethyl-7-oxohepta-2,4-dienamide | Homo sapiens (human) | Potency | 0.4467 | 4 | 0 |
racecadotril | Homo sapiens (human) | Potency | 0.8037 | 4 | 0 |
pyronaridine | Homo sapiens (human) | Potency | 22.7420 | 4 | 0 |
deguelin | Homo sapiens (human) | Potency | 20.0524 | 4 | 0 |
fingolimod | Homo sapiens (human) | Potency | 21.0004 | 4 | 0 |
tesmilifene | Homo sapiens (human) | Potency | 24.6794 | 4 | 0 |
benzamil | Homo sapiens (human) | Potency | 27.3309 | 4 | 0 |
tamibarotene | Homo sapiens (human) | Potency | 25.3179 | 4 | 0 |
carboxyamido-triazole | Homo sapiens (human) | Potency | 21.7168 | 4 | 0 |
ci 988 | Homo sapiens (human) | Potency | 1.3438 | 2 | 0 |
tanshinone | Homo sapiens (human) | Potency | 11.7704 | 1 | 0 |
icrf 193 | Homo sapiens (human) | Potency | 0.6918 | 3 | 0 |
sophocarpine | Homo sapiens (human) | Potency | 17.1333 | 4 | 0 |
nitisinone | Homo sapiens (human) | Potency | 29.9439 | 3 | 0 |
sr 48692 | Homo sapiens (human) | Potency | 4.1763 | 1 | 0 |
elacridar | Homo sapiens (human) | Potency | 23.5402 | 4 | 0 |
mosapride | Homo sapiens (human) | Potency | 0.5894 | 2 | 0 |
ezogabine | Homo sapiens (human) | Potency | 25.8870 | 4 | 0 |
celastrol | Homo sapiens (human) | Potency | 1.0665 | 4 | 0 |
almotriptan | Homo sapiens (human) | Potency | 0.0743 | 1 | 0 |
gefitinib | Homo sapiens (human) | Potency | 30.5401 | 4 | 0 |
vadimezan | Homo sapiens (human) | Potency | 25.2204 | 4 | 0 |
gyki 53655 | Homo sapiens (human) | Potency | 8.4073 | 4 | 0 |
methotrexate | Homo sapiens (human) | Potency | 0.0279 | 4 | 0 |
umifenovir | Homo sapiens (human) | Potency | 18.5622 | 4 | 0 |
safinamide | Homo sapiens (human) | Potency | 13.1967 | 4 | 0 |
ml-3000 | Homo sapiens (human) | Potency | 23.9273 | 4 | 0 |
febuxostat | Homo sapiens (human) | Potency | 29.5659 | 1 | 0 |
(1R,3S)-5-[2-[(1R,3aS,7aR)-1-[(2R)-6-hydroxy-6-methylheptan-2-yl]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-4-ylidene]ethylidene]-4-methylenecyclohexane-1,3-diol | Homo sapiens (human) | Potency | 3.6428 | 4 | 0 |
aspartame | Homo sapiens (human) | Potency | 30.5658 | 4 | 0 |
pomalidomide | Homo sapiens (human) | Potency | 0.0042 | 1 | 0 |
cd 437 | Homo sapiens (human) | Potency | 0.9864 | 4 | 0 |
tempol | Homo sapiens (human) | Potency | 0.3722 | 1 | 0 |
10-propargyl-10-deazaaminopterin | Homo sapiens (human) | Potency | 0.0362 | 4 | 0 |
atazanavir | Homo sapiens (human) | Potency | 4.6859 | 1 | 0 |
lonafarnib | Homo sapiens (human) | Potency | 13.6389 | 4 | 0 |
chs 828 | Homo sapiens (human) | Potency | 0.0022 | 2 | 0 |
tariquidar | Homo sapiens (human) | Potency | 11.5068 | 4 | 0 |
levofloxacin | Homo sapiens (human) | Potency | 24.0897 | 2 | 0 |
nepafenac | Homo sapiens (human) | Potency | 20.2008 | 3 | 0 |
conivaptan | Homo sapiens (human) | Potency | 24.8161 | 3 | 0 |
evodiamine | Homo sapiens (human) | Potency | 25.1747 | 3 | 0 |
varespladib | Homo sapiens (human) | Potency | 19.7224 | 4 | 0 |
canertinib | Homo sapiens (human) | Potency | 16.7983 | 4 | 0 |
cinacalcet | Homo sapiens (human) | Potency | 10.0683 | 2 | 0 |
birb 796 | Homo sapiens (human) | Potency | 25.2484 | 4 | 0 |
nps-568 | Homo sapiens (human) | Potency | 37.2212 | 2 | 0 |
telbivudine | Homo sapiens (human) | Potency | 9.3090 | 3 | 0 |
tipifarnib | Homo sapiens (human) | Potency | 5.8173 | 4 | 0 |
torcetrapib | Homo sapiens (human) | Potency | 27.8008 | 4 | 0 |
cryptotanshinone | Homo sapiens (human) | Potency | 24.3667 | 4 | 0 |
cyc 202 | Homo sapiens (human) | Potency | 22.0135 | 4 | 0 |
ampelopsin | Homo sapiens (human) | Potency | 31.7911 | 3 | 0 |
vincristine | Homo sapiens (human) | Potency | 19.4960 | 3 | 0 |
tanshinone ii a | Homo sapiens (human) | Potency | 0.0037 | 1 | 0 |
avasimibe | Homo sapiens (human) | Potency | 5.1986 | 3 | 0 |
sb 203580 | Homo sapiens (human) | Potency | 44.3070 | 4 | 0 |
enzastaurin | Homo sapiens (human) | Potency | 8.6979 | 4 | 0 |
erlotinib | Homo sapiens (human) | Potency | 15.8526 | 4 | 0 |
piboserod | Homo sapiens (human) | Potency | 11.4267 | 4 | 0 |
l 163191 | Homo sapiens (human) | Potency | 24.4446 | 4 | 0 |
cephalexin, (6r-(6alpha,7beta))-isomer | Homo sapiens (human) | Potency | 0.0074 | 1 | 0 |
latrepirdine | Homo sapiens (human) | Potency | 31.2932 | 3 | 0 |
orantinib | Homo sapiens (human) | Potency | 0.2436 | 4 | 0 |
dronedarone | Homo sapiens (human) | Potency | 20.4933 | 4 | 0 |
ramelteon | Homo sapiens (human) | Potency | 2.3485 | 1 | 0 |
lapatinib | Homo sapiens (human) | Potency | 6.0312 | 4 | 0 |
2-(4-morpholinoanilino)-6-cyclohexylaminopurine | Homo sapiens (human) | Potency | 5.4168 | 4 | 0 |
dabigatran etexilate | Homo sapiens (human) | Potency | 17.4660 | 4 | 0 |
darunavir | Homo sapiens (human) | Potency | 1.9923 | 4 | 0 |
deferasirox | Homo sapiens (human) | Potency | 17.1126 | 4 | 0 |
dabigatran | Homo sapiens (human) | Potency | 0.1795 | 2 | 0 |
sorafenib | Homo sapiens (human) | Potency | 6.7166 | 4 | 0 |
N-hydroxy-3-[4-[[2-hydroxyethyl-[2-(1H-indol-3-yl)ethyl]amino]methyl]phenyl]-2-propenamide | Homo sapiens (human) | Potency | 0.1730 | 4 | 0 |
lenalidomide | Homo sapiens (human) | Potency | 7.0790 | 2 | 0 |
N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide | Homo sapiens (human) | Potency | 0.1253 | 4 | 0 |
sr 142806 | Homo sapiens (human) | Potency | 24.2793 | 4 | 0 |
phenoxodiol | Homo sapiens (human) | Potency | 4.7188 | 4 | 0 |
1-methylpropyl-2-imidazolyl disulfide | Homo sapiens (human) | Potency | 22.7930 | 4 | 0 |
demecolcine | Homo sapiens (human) | Potency | 0.2356 | 4 | 0 |
nsc 74859 | Homo sapiens (human) | Potency | 20.7662 | 4 | 0 |
gant58 | Homo sapiens (human) | Potency | 23.8756 | 4 | 0 |
cyclovirobuxine d | Homo sapiens (human) | Potency | 13.2066 | 1 | 0 |
2,5-bis(5-hydroxymethyl-2-thienyl)furan | Homo sapiens (human) | Potency | 11.2664 | 4 | 0 |
nsc 663284 | Homo sapiens (human) | Potency | 5.3272 | 4 | 0 |
bortezomib | Homo sapiens (human) | Potency | 0.0322 | 4 | 0 |
ritonavir | Homo sapiens (human) | Potency | 17.4584 | 3 | 0 |
nu 6027 | Homo sapiens (human) | Potency | 14.8621 | 4 | 0 |
nsc 23766 | Homo sapiens (human) | Potency | 27.0522 | 2 | 0 |
gant 61 | Homo sapiens (human) | Potency | 20.4314 | 4 | 0 |
naringenin | Homo sapiens (human) | Potency | 17.0688 | 2 | 0 |
5-hydroxytryptophan | Homo sapiens (human) | Potency | 11.7704 | 1 | 0 |
amastatin | Homo sapiens (human) | Potency | 23.0506 | 3 | 0 |
tosylphenylalanyl chloromethyl ketone | Homo sapiens (human) | Potency | 19.1124 | 4 | 0 |
mometasone furoate | Homo sapiens (human) | Potency | 7.9872 | 4 | 0 |
linezolid | Homo sapiens (human) | Potency | 9.4254 | 3 | 0 |
temocapril hydrochloride | Homo sapiens (human) | Potency | 5.0378 | 4 | 0 |
vinpocetine | Homo sapiens (human) | Potency | 20.4314 | 4 | 0 |
estramustine phosphate sodium | Homo sapiens (human) | Potency | 0.0105 | 1 | 0 |
fluticasone propionate | Homo sapiens (human) | Potency | 16.6261 | 1 | 0 |
pd 173955 | Homo sapiens (human) | Potency | 0.1146 | 4 | 0 |
gw 3965 | Homo sapiens (human) | Potency | 22.2859 | 4 | 0 |
y 27632 | Homo sapiens (human) | Potency | 9.3279 | 2 | 0 |
rolipram | Homo sapiens (human) | Potency | 3.5992 | 4 | 0 |
6-bromoindirubin-3'-oxime | Homo sapiens (human) | Potency | 4.7741 | 4 | 0 |
purvalanol b | Homo sapiens (human) | Potency | 0.1281 | 4 | 0 |
repsox | Homo sapiens (human) | Potency | 7.4266 | 1 | 0 |
roflumilast | Homo sapiens (human) | Potency | 17.6840 | 3 | 0 |
decitabine | Homo sapiens (human) | Potency | 10.2218 | 4 | 0 |
(2R,3S,5S)-2-(6-aminopurin-9-yl)-5-(hydroxymethyl)-3-oxolanol | Homo sapiens (human) | Potency | 20.3474 | 3 | 0 |
pa 824 | Homo sapiens (human) | Potency | 6.1804 | 4 | 0 |
ketoconazole | Homo sapiens (human) | Potency | 19.9242 | 4 | 0 |
purvalanol a | Homo sapiens (human) | Potency | 10.1106 | 4 | 0 |
diclazuril | Homo sapiens (human) | Potency | 29.6966 | 3 | 0 |
melphalan | Homo sapiens (human) | Potency | 3.5854 | 4 | 0 |
benzyloxycarbonylleucyl-leucyl-leucine aldehyde | Homo sapiens (human) | Potency | 0.4406 | 4 | 0 |
tenofovir | Homo sapiens (human) | Potency | 0.4686 | 1 | 0 |
terameprocol | Homo sapiens (human) | Potency | 1.1044 | 4 | 0 |
shikonin | Homo sapiens (human) | Potency | 2.2838 | 4 | 0 |
5-fluoro-2'-deoxycytidine | Homo sapiens (human) | Potency | 0.0590 | 4 | 0 |
IPA-3 | Homo sapiens (human) | Potency | 29.0456 | 4 | 0 |
4-(4-chloro-2-methylphenoxy)-n-hydroxybutanamide | Homo sapiens (human) | Potency | 5.7279 | 4 | 0 |
mecarbinate | Homo sapiens (human) | Potency | 35.8719 | 3 | 0 |
pirarubicin hydrochloride | Homo sapiens (human) | Potency | 0.5022 | 4 | 0 |
cgp 60474 | Homo sapiens (human) | Potency | 0.1496 | 4 | 0 |
tram 34 | Homo sapiens (human) | Potency | 1.0205 | 4 | 0 |
fludarabine | Homo sapiens (human) | Potency | 0.6878 | 4 | 0 |
propylthiouracil | Homo sapiens (human) | Potency | 35.1973 | 2 | 0 |
prothionamide | Homo sapiens (human) | Potency | 0.0037 | 1 | 0 |
etomidate | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
mercaptopurine | Homo sapiens (human) | Potency | 2.4778 | 4 | 0 |
jrf 12 | Homo sapiens (human) | Potency | 22.9244 | 4 | 0 |
rg108 | Homo sapiens (human) | Potency | 0.0030 | 1 | 0 |
stf 62247 | Homo sapiens (human) | Potency | 30.5658 | 4 | 0 |
stf 083010 | Homo sapiens (human) | Potency | 2.3916 | 4 | 0 |
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-1-naphthalenecarboxamide | Homo sapiens (human) | Potency | 0.3812 | 4 | 0 |
paroxetine, cis-(+)-isomer | Homo sapiens (human) | Potency | 18.2799 | 3 | 0 |
eszopiclone | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
cct018159 | Homo sapiens (human) | Potency | 8.0873 | 4 | 0 |
secinh3 | Homo sapiens (human) | Potency | 13.4783 | 3 | 0 |
2-[[benzamido(sulfanylidene)methyl]amino]-5,5-dimethyl-4,7-dihydrothieno[2,3-c]pyran-3-carboxylic acid | Homo sapiens (human) | Potency | 29.6966 | 3 | 0 |
jk184 | Homo sapiens (human) | Potency | 0.0029 | 4 | 0 |
3-(1-azepanylsulfonyl)-n-(3-bromphenyl)benzamide | Homo sapiens (human) | Potency | 24.2014 | 4 | 0 |
xl147 | Homo sapiens (human) | Potency | 13.8432 | 4 | 0 |
N-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)thio]acetamide | Homo sapiens (human) | Potency | 18.2095 | 4 | 0 |
3-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
thioguanine anhydrous | Homo sapiens (human) | Potency | 1.3381 | 4 | 0 |
hc-067047 | Homo sapiens (human) | Potency | 11.1961 | 4 | 0 |
bi-78d3 | Homo sapiens (human) | Potency | 4.9897 | 4 | 0 |
ethionamide | Homo sapiens (human) | Potency | 20.9310 | 2 | 0 |
kartogenin | Homo sapiens (human) | Potency | 29.5659 | 1 | 0 |
methyl-thiohydantoin-tryptophan | Homo sapiens (human) | Potency | 0.5899 | 1 | 0 |
10074-g5 | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
kl001 | Homo sapiens (human) | Potency | 23.8756 | 4 | 0 |
2-[2-chloro-6-ethoxy-4-[(3-methyl-5-oxo-1-phenyl-4-pyrazolylidene)methyl]phenoxy]acetic acid methyl ester | Homo sapiens (human) | Potency | 10.6959 | 3 | 0 |
4-(5-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1h-pyrazol-1-yl)benzenesulfonamide | Homo sapiens (human) | Potency | 30.5658 | 4 | 0 |
monastrol | Homo sapiens (human) | Potency | 0.1163 | 4 | 0 |
maraviroc | Homo sapiens (human) | Potency | 32.4796 | 4 | 0 |
rwj 67657 | Homo sapiens (human) | Potency | 26.6235 | 4 | 0 |
nelarabine | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
6-methyl-2-(phenylethynyl)pyridine | Homo sapiens (human) | Potency | 20.4314 | 4 | 0 |
bms 387032 | Homo sapiens (human) | Potency | 0.1538 | 4 | 0 |
or 1259 | Homo sapiens (human) | Potency | 24.4446 | 4 | 0 |
e 7010 | Homo sapiens (human) | Potency | 0.0978 | 4 | 0 |
ly335979 | Homo sapiens (human) | Potency | 25.9850 | 4 | 0 |
tandutinib | Homo sapiens (human) | Potency | 22.9939 | 4 | 0 |
vx-745 | Homo sapiens (human) | Potency | 26.8183 | 3 | 0 |
corlanor | Homo sapiens (human) | Potency | 19.5644 | 4 | 0 |
prucalopride | Homo sapiens (human) | Potency | 36.2093 | 4 | 0 |
dasatinib | Homo sapiens (human) | Potency | 15.9901 | 4 | 0 |
poly(2-fluoroadenylic acid) | Homo sapiens (human) | Potency | 14.5081 | 4 | 0 |
zd 6474 | Homo sapiens (human) | Potency | 10.2474 | 4 | 0 |
N-methyl-2-[[3-[2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]thio]benzamide | Homo sapiens (human) | Potency | 8.4170 | 4 | 0 |
N-[2-(diethylamino)ethyl]-5-[(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide | Homo sapiens (human) | Potency | 9.5496 | 4 | 0 |
compound 968 | Homo sapiens (human) | Potency | 23.5768 | 3 | 0 |
gw 7647 | Homo sapiens (human) | Potency | 12.7196 | 3 | 0 |
valproate | Homo sapiens (human) | Potency | 0.4176 | 1 | 0 |
brl 15572 | Homo sapiens (human) | Potency | 20.0500 | 4 | 0 |
1-[6-(4-chlorophenyl)-5-imidazo[2,1-b]thiazolyl]-N-[(3,4-dichlorophenyl)methoxy]methanimine | Homo sapiens (human) | Potency | 14.8301 | 3 | 0 |
rose bengal(2-) | Homo sapiens (human) | Potency | 15.8264 | 4 | 0 |
N4-ethyl-N6,1,2-trimethyl-N4-phenylpyrimidin-1-ium-4,6-diamine | Homo sapiens (human) | Potency | 12.0264 | 2 | 0 |
2-[[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]-1-oxo-5-isoquinolinyl]oxy]propanoic acid ethyl ester | Homo sapiens (human) | Potency | 7.5262 | 3 | 0 |
sb 415286 | Homo sapiens (human) | Potency | 33.1487 | 4 | 0 |
4-methylene-2-octyl-5-oxo-3-oxolanecarboxylic acid | Homo sapiens (human) | Potency | 31.7859 | 4 | 0 |
stx-0119 | Homo sapiens (human) | Potency | 17.4860 | 4 | 0 |
sch 79797 | Homo sapiens (human) | Potency | 3.7591 | 4 | 0 |
LY-310762 | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
am 630 | Homo sapiens (human) | Potency | 34.1854 | 4 | 0 |
sb 408124 | Homo sapiens (human) | Potency | 27.9582 | 2 | 0 |
sitagliptin | Homo sapiens (human) | Potency | 19.9242 | 4 | 0 |
4-(5-benzo(1,3)dioxol-5-yl-4-pyridin-2-yl-1h-imidazol-2-yl)benzamide | Homo sapiens (human) | Potency | 15.7220 | 2 | 0 |
rabeprazole(1-) | Homo sapiens (human) | Potency | 14.6319 | 2 | 0 |
tolcapone | Homo sapiens (human) | Potency | 36.2093 | 4 | 0 |
1-(4-Fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-one | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
eeyarestatin i | Homo sapiens (human) | Potency | 19.6196 | 4 | 0 |
imd 0354 | Homo sapiens (human) | Potency | 1.4379 | 4 | 0 |
ex 527 | Homo sapiens (human) | Potency | 11.4268 | 3 | 0 |
jtk-303 | Homo sapiens (human) | Potency | 25.9850 | 4 | 0 |
ku 55933 | Homo sapiens (human) | Potency | 20.4933 | 4 | 0 |
quercetin | Homo sapiens (human) | Potency | 15.8207 | 4 | 0 |
biochanin a | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
apigenin | Homo sapiens (human) | Potency | 22.3554 | 4 | 0 |
luteolin | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
hymecromone | Homo sapiens (human) | Potency | 22.2080 | 2 | 0 |
daphnetin | Homo sapiens (human) | Potency | 15.8264 | 4 | 0 |
kaempferol | Homo sapiens (human) | Potency | 17.6341 | 4 | 0 |
genistein | Homo sapiens (human) | Potency | 12.5757 | 3 | 0 |
baicalein | Homo sapiens (human) | Potency | 25.2686 | 4 | 0 |
chrysin | Homo sapiens (human) | Potency | 31.2932 | 3 | 0 |
diosmetin | Homo sapiens (human) | Potency | 10.6579 | 4 | 0 |
fisetin | Homo sapiens (human) | Potency | 17.7575 | 4 | 0 |
morin | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
myricetin | Homo sapiens (human) | Potency | 20.0556 | 2 | 0 |
daidzein | Homo sapiens (human) | Potency | 17.9701 | 3 | 0 |
purmorphamine | Homo sapiens (human) | Potency | 0.0019 | 1 | 0 |
sag compound | Homo sapiens (human) | Potency | 25.0831 | 4 | 0 |
levetiracetam | Homo sapiens (human) | Potency | 24.9178 | 2 | 0 |
blebbistatin | Homo sapiens (human) | Potency | 13.9958 | 4 | 0 |
ter 199 | Homo sapiens (human) | Potency | 37.2212 | 2 | 0 |
acipimox | Homo sapiens (human) | Potency | 30.0907 | 3 | 0 |
ly 320135 | Homo sapiens (human) | Potency | 18.6180 | 2 | 0 |
n-(4-amino-2-methylquinolin-6-yl)-2-(4-ethylphenoxymethyl)benzamide | Homo sapiens (human) | Potency | 8.3880 | 4 | 0 |
pd 166285 | Homo sapiens (human) | Potency | 2.0132 | 4 | 0 |
(3r)-((2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl))methanone | Homo sapiens (human) | Potency | 28.0563 | 4 | 0 |
3-[6-[4-(trifluoromethoxy)anilino]-4-pyrimidinyl]benzamide | Homo sapiens (human) | Potency | 26.1503 | 4 | 0 |
icaritin | Homo sapiens (human) | Potency | 22.5328 | 4 | 0 |
bosutinib | Homo sapiens (human) | Potency | 19.4620 | 4 | 0 |
palbociclib | Homo sapiens (human) | Potency | 14.9154 | 4 | 0 |
jnj-7706621 | Homo sapiens (human) | Potency | 7.3374 | 4 | 0 |
benazepril | Homo sapiens (human) | Potency | 22.8465 | 4 | 0 |
verteporfin | Homo sapiens (human) | Potency | 0.0793 | 4 | 0 |
batimastat | Homo sapiens (human) | Potency | 16.1249 | 2 | 0 |
sinomenine | Homo sapiens (human) | Potency | 6.4444 | 4 | 0 |
pepstatin | Homo sapiens (human) | Potency | 2.0931 | 1 | 0 |
norbinaltorphimine | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
pregabalin | Homo sapiens (human) | Potency | 16.6261 | 1 | 0 |
2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz(h)imidazo(4,5-f)isoquinoline-7-one | Homo sapiens (human) | Potency | 4.7344 | 4 | 0 |
vx680 | Homo sapiens (human) | Potency | 2.9534 | 4 | 0 |
cgp 3466 | Homo sapiens (human) | Potency | 0.0743 | 1 | 0 |
d 4476 | Homo sapiens (human) | Potency | 24.6301 | 4 | 0 |
cyc 116 | Homo sapiens (human) | Potency | 12.7330 | 4 | 0 |
bay 19-8004 | Homo sapiens (human) | Potency | 17.7511 | 4 | 0 |
indiplon | Homo sapiens (human) | Potency | 21.2097 | 4 | 0 |
pai 039 | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
tubacin | Homo sapiens (human) | Potency | 9.6314 | 4 | 0 |
(13S)-3-hydroxy-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthren-17-one | Homo sapiens (human) | Potency | 6.1199 | 4 | 0 |
ispinesib | Homo sapiens (human) | Potency | 2.3386 | 4 | 0 |
nps2143 | Homo sapiens (human) | Potency | 15.7220 | 4 | 0 |
pd 184352 | Homo sapiens (human) | Potency | 22.9154 | 4 | 0 |
prasugrel | Homo sapiens (human) | Potency | 3.1873 | 4 | 0 |
fesoterodine | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
hdac-42 | Homo sapiens (human) | Potency | 0.6367 | 4 | 0 |
3-tritylthio-l-alanine, (d)-isomer | Homo sapiens (human) | Potency | 24.9938 | 4 | 0 |
posaconazole | Homo sapiens (human) | Potency | 14.1286 | 4 | 0 |
a 770041 | Homo sapiens (human) | Potency | 3.7908 | 4 | 0 |
tws 119 | Homo sapiens (human) | Potency | 3.1997 | 4 | 0 |
[4-[[4-(1-benzothiophen-2-yl)-2-pyrimidinyl]amino]phenyl]-[4-(1-pyrrolidinyl)-1-piperidinyl]methanone | Homo sapiens (human) | Potency | 19.7929 | 4 | 0 |
pnu-282987 | Homo sapiens (human) | Potency | 17.0391 | 4 | 0 |
iniparib | Homo sapiens (human) | Potency | 8.3328 | 1 | 0 |
nepicastat | Homo sapiens (human) | Potency | 24.3667 | 4 | 0 |
[4-(2-amino-4-bromoanilino)-2-chlorophenyl]-(2-methylphenyl)methanone | Homo sapiens (human) | Potency | 17.5538 | 4 | 0 |
mk 0752 | Homo sapiens (human) | Potency | 12.9343 | 4 | 0 |
nt 702 | Homo sapiens (human) | Potency | 13.5967 | 4 | 0 |
gw 501516 | Homo sapiens (human) | Potency | 12.8366 | 3 | 0 |
az 11645373 | Homo sapiens (human) | Potency | 6.8670 | 4 | 0 |
av 412 | Homo sapiens (human) | Potency | 2.0424 | 4 | 0 |
ag-041r | Homo sapiens (human) | Potency | 34.5227 | 3 | 0 |
telatinib | Homo sapiens (human) | Potency | 11.7508 | 2 | 0 |
y-39983 | Homo sapiens (human) | Potency | 24.7132 | 4 | 0 |
cp 547632 | Homo sapiens (human) | Potency | 14.8621 | 4 | 0 |
bms345541 | Homo sapiens (human) | Potency | 6.2077 | 4 | 0 |
vidofludimus | Homo sapiens (human) | Potency | 13.1410 | 4 | 0 |
spc-839 | Homo sapiens (human) | Potency | 1.5084 | 4 | 0 |
lenvatinib | Homo sapiens (human) | Potency | 0.8500 | 4 | 0 |
andarine | Homo sapiens (human) | Potency | 3.7221 | 1 | 0 |
adw 742 | Homo sapiens (human) | Potency | 12.6566 | 4 | 0 |
gw843682x | Homo sapiens (human) | Potency | 2.0749 | 4 | 0 |
pd 0325901 | Homo sapiens (human) | Potency | 32.7752 | 4 | 0 |
gsk 256066 | Homo sapiens (human) | Potency | 0.0023 | 1 | 0 |
midostaurin | Homo sapiens (human) | Potency | 1.8024 | 4 | 0 |
ly 404039 | Homo sapiens (human) | Potency | 19.9581 | 4 | 0 |
ag 14361 | Homo sapiens (human) | Potency | 19.7929 | 4 | 0 |
sb 265610 | Homo sapiens (human) | Potency | 31.5676 | 4 | 0 |
ly 450139 | Homo sapiens (human) | Potency | 20.0556 | 2 | 0 |
cp 91149 | Homo sapiens (human) | Potency | 22.0830 | 4 | 0 |
gw791343 | Homo sapiens (human) | Potency | 12.8585 | 4 | 0 |
cabazitaxel | Homo sapiens (human) | Potency | 0.2396 | 2 | 0 |
sb-505124 | Homo sapiens (human) | Potency | 9.9510 | 4 | 0 |
sb 242235 | Homo sapiens (human) | Potency | 8.0346 | 4 | 0 |
mocetinostat | Homo sapiens (human) | Potency | 1.0884 | 4 | 0 |
sd 0006 | Homo sapiens (human) | Potency | 0.0284 | 2 | 0 |
osi 930 | Homo sapiens (human) | Potency | 18.1476 | 4 | 0 |
carbobenzoxy-leucyl-leucyl-norvalinal | Homo sapiens (human) | Potency | 1.0724 | 4 | 0 |
ki 20227 | Homo sapiens (human) | Potency | 29.2109 | 4 | 0 |
scio-469 | Homo sapiens (human) | Potency | 22.0830 | 4 | 0 |
ssr 69071 | Homo sapiens (human) | Potency | 19.1067 | 4 | 0 |
sb 3ct compound | Homo sapiens (human) | Potency | 21.1318 | 4 | 0 |
orteronel | Homo sapiens (human) | Potency | 18.9124 | 3 | 0 |
pi103 | Homo sapiens (human) | Potency | 0.4041 | 4 | 0 |
l 084 | Homo sapiens (human) | Potency | 33.1734 | 2 | 0 |
2-((aminocarbonyl)amino)-5-(4-fluorophenyl)-3-thiophenecarboxamide | Homo sapiens (human) | Potency | 1.9789 | 4 | 0 |
tgx 221 | Homo sapiens (human) | Potency | 30.3531 | 4 | 0 |
sa 4503 | Homo sapiens (human) | Potency | 17.8745 | 2 | 0 |
ic 87114 | Homo sapiens (human) | Potency | 2.2834 | 4 | 0 |
zibotentan | Homo sapiens (human) | Potency | 18.6548 | 1 | 0 |
sb 705498 | Homo sapiens (human) | Potency | 25.0831 | 4 | 0 |
tivozanib | Homo sapiens (human) | Potency | 3.1565 | 4 | 0 |
zm 447439 | Homo sapiens (human) | Potency | 11.1194 | 4 | 0 |
avn 944 | Homo sapiens (human) | Potency | 0.4829 | 4 | 0 |
n-(6-chloro-7-methoxy-9h-beta-carbolin-8-yl)-2-methylnicotinamide | Homo sapiens (human) | Potency | 3.8775 | 4 | 0 |
rucaparib | Homo sapiens (human) | Potency | 17.1269 | 4 | 0 |
cediranib | Homo sapiens (human) | Potency | 21.7703 | 4 | 0 |
tae226 | Homo sapiens (human) | Potency | 3.8087 | 4 | 0 |
gw0742 | Homo sapiens (human) | Potency | 28.1437 | 4 | 0 |
sb 743921 | Homo sapiens (human) | Potency | 11.2968 | 2 | 0 |
ps1145 | Homo sapiens (human) | Potency | 25.4160 | 4 | 0 |
l-779,450 | Homo sapiens (human) | Potency | 21.7863 | 4 | 0 |
tak-715 | Homo sapiens (human) | Potency | 18.8337 | 4 | 0 |
aq4n | Homo sapiens (human) | Potency | 14.7118 | 4 | 0 |
chir 99021 | Homo sapiens (human) | Potency | 12.1249 | 4 | 0 |
ym 201636 | Homo sapiens (human) | Potency | 17.6404 | 4 | 0 |
sb 525334 | Homo sapiens (human) | Potency | 21.8482 | 4 | 0 |
osu 03012 | Homo sapiens (human) | Potency | 16.1733 | 4 | 0 |
sb-612111 | Homo sapiens (human) | Potency | 9.4363 | 4 | 0 |
masitinib | Homo sapiens (human) | Potency | 24.9178 | 4 | 0 |
bx795 | Homo sapiens (human) | Potency | 8.5117 | 4 | 0 |
linagliptin | Homo sapiens (human) | Potency | 28.8601 | 4 | 0 |
as 601245 | Homo sapiens (human) | Potency | 17.4368 | 4 | 0 |
pazopanib | Homo sapiens (human) | Potency | 20.6682 | 2 | 0 |
sepantronium | Homo sapiens (human) | Potency | 0.0072 | 4 | 0 |
azd 6244 | Homo sapiens (human) | Potency | 14.7118 | 4 | 0 |
odanacatib | Homo sapiens (human) | Potency | 18.7167 | 4 | 0 |
1-(2-(1-adamantyl)ethyl)-1-pentyl-3-(3-(4-pyridyl)propyl)urea | Homo sapiens (human) | Potency | 17.1884 | 4 | 0 |
cp-673,451 | Homo sapiens (human) | Potency | 18.9032 | 4 | 0 |
a 443654 | Homo sapiens (human) | Potency | 1.8401 | 4 | 0 |
apixaban | Homo sapiens (human) | Potency | 0.0209 | 1 | 0 |
bay 61-3606 | Homo sapiens (human) | Potency | 8.3003 | 4 | 0 |
gw 799388 | Homo sapiens (human) | Potency | 19.3848 | 3 | 0 |
ar c155858 | Homo sapiens (human) | Potency | 0.1356 | 2 | 0 |
gw 842166x | Homo sapiens (human) | Potency | 30.5658 | 4 | 0 |
akt-i-1 compound | Homo sapiens (human) | Potency | 0.6010 | 4 | 0 |
erteberel | Homo sapiens (human) | Potency | 16.2113 | 4 | 0 |
aee 788 | Homo sapiens (human) | Potency | 0.0178 | 3 | 0 |
saracatinib | Homo sapiens (human) | Potency | 20.7887 | 4 | 0 |
az10606120 | Homo sapiens (human) | Potency | 15.4504 | 4 | 0 |
sd-208 | Homo sapiens (human) | Potency | 3.4097 | 3 | 0 |
osi-420 | Homo sapiens (human) | Potency | 9.3180 | 4 | 0 |
gm 1489 | Homo sapiens (human) | Potency | 34.1854 | 4 | 0 |
[4-(3-chlorophenyl)-1-piperazinyl]-(5-methyl-2-phenyl-3-pyrazolyl)methanone | Homo sapiens (human) | Potency | 2.8462 | 3 | 0 |
vx 702 | Homo sapiens (human) | Potency | 26.3506 | 1 | 0 |
crenolanib | Homo sapiens (human) | Potency | 0.0132 | 1 | 0 |
ki16425 | Homo sapiens (human) | Potency | 0.0166 | 1 | 0 |
tg100-115 | Homo sapiens (human) | Potency | 22.2080 | 4 | 0 |
cc 401 | Homo sapiens (human) | Potency | 19.5978 | 4 | 0 |
ly 411575 | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
bms 599626 | Homo sapiens (human) | Potency | 0.9080 | 4 | 0 |
e 5555 | Homo sapiens (human) | Potency | 10.3448 | 4 | 0 |
volasertib | Homo sapiens (human) | Potency | 0.0908 | 4 | 0 |
PB28 | Homo sapiens (human) | Potency | 19.8548 | 4 | 0 |
azd 7762 | Homo sapiens (human) | Potency | 0.3195 | 4 | 0 |
krp-203 | Homo sapiens (human) | Potency | 30.5658 | 4 | 0 |
regorafenib | Homo sapiens (human) | Potency | 20.9310 | 4 | 0 |
at 7867 | Homo sapiens (human) | Potency | 20.0413 | 4 | 0 |
acetic acid 2-[4-methyl-8-(4-morpholinylsulfonyl)-1,3-dioxo-2-pyrrolo[3,4-c]quinolinyl]ethyl ester | Homo sapiens (human) | Potency | 0.0187 | 1 | 0 |
6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one | Homo sapiens (human) | Potency | 0.8449 | 4 | 0 |
ptc 124 | Homo sapiens (human) | Potency | 19.4960 | 3 | 0 |
abt-737 | Homo sapiens (human) | Potency | 11.4403 | 4 | 0 |
brivanib | Homo sapiens (human) | Potency | 14.3543 | 4 | 0 |
icg 001 | Homo sapiens (human) | Potency | 2.9084 | 4 | 0 |
pha 680632 | Homo sapiens (human) | Potency | 2.8360 | 4 | 0 |
4-(2-((1r)-1-(((4-chlorophenyl)sulfonyl)-2,5-difluoroanilino)ethyl)-5-fluorophenyl)butanoic acid | Homo sapiens (human) | Potency | 21.2701 | 4 | 0 |
fg-4592 | Homo sapiens (human) | Potency | 5.8992 | 1 | 0 |
mp470 | Homo sapiens (human) | Potency | 6.6058 | 4 | 0 |
jnj16259685 | Homo sapiens (human) | Potency | 14.4592 | 4 | 0 |
ki 8751 | Homo sapiens (human) | Potency | 14.7485 | 4 | 0 |
mk 2866 | Homo sapiens (human) | Potency | 33.1734 | 1 | 0 |
nu 7441 | Homo sapiens (human) | Potency | 7.3346 | 4 | 0 |
at 7519 | Homo sapiens (human) | Potency | 0.2692 | 4 | 0 |
cyt997 | Homo sapiens (human) | Potency | 1.4824 | 4 | 0 |
bi 2536 | Homo sapiens (human) | Potency | 0.0562 | 4 | 0 |
N-(6-fluoro-1H-indazol-5-yl)-6-methyl-2-oxo-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyridine-5-carboxamide | Homo sapiens (human) | Potency | 4.4542 | 2 | 0 |
compound 26 | Homo sapiens (human) | Potency | 11.6404 | 3 | 0 |
r 1487 | Homo sapiens (human) | Potency | 1.9027 | 2 | 0 |
adl 5859 | Homo sapiens (human) | Potency | 10.4904 | 1 | 0 |
danusertib | Homo sapiens (human) | Potency | 0.2615 | 4 | 0 |
N-[4-(2-tert-butylphenyl)sulfonylphenyl]-2,3,4-trihydroxy-5-[(2-propan-2-ylphenyl)methyl]benzamide | Homo sapiens (human) | Potency | 7.8797 | 4 | 0 |
N-[5-[[5-[(4-acetyl-1-piperazinyl)-oxomethyl]-4-methoxy-2-methylphenyl]thio]-2-thiazolyl]-4-[(3,3-dimethylbutan-2-ylamino)methyl]benzamide | Homo sapiens (human) | Potency | 8.9706 | 4 | 0 |
nvp-aew541 | Homo sapiens (human) | Potency | 11.2999 | 4 | 0 |
abt 869 | Homo sapiens (human) | Potency | 33.2835 | 4 | 0 |
azd 8931 | Homo sapiens (human) | Potency | 0.0562 | 4 | 0 |
fr 180204 | Homo sapiens (human) | Potency | 10.6571 | 4 | 0 |
dorsomorphin | Homo sapiens (human) | Potency | 18.8337 | 4 | 0 |
ac 261066 | Homo sapiens (human) | Potency | 25.6420 | 4 | 0 |
quisinostat | Homo sapiens (human) | Potency | 0.0301 | 4 | 0 |
anacetrapib | Homo sapiens (human) | Potency | 20.0556 | 2 | 0 |
carfilzomib | Homo sapiens (human) | Potency | 0.0210 | 4 | 0 |
hcv 796 | Homo sapiens (human) | Potency | 17.9786 | 3 | 0 |
pf-2545920 | Homo sapiens (human) | Potency | 17.7023 | 4 | 0 |
jnj 26854165 | Homo sapiens (human) | Potency | 10.4898 | 4 | 0 |
pf 573228 | Homo sapiens (human) | Potency | 15.6335 | 4 | 0 |
tak 285 | Homo sapiens (human) | Potency | 22.7144 | 4 | 0 |
idelalisib | Homo sapiens (human) | Potency | 2.7242 | 4 | 0 |
nebivolol hydrochloride | Homo sapiens (human) | Potency | 22.2080 | 4 | 0 |
crizotinib | Homo sapiens (human) | Potency | 11.5277 | 4 | 0 |
5-(5,6-dimethoxy-1-benzimidazolyl)-3-[(2-methylsulfonylphenyl)methoxy]-2-thiophenecarbonitrile | Homo sapiens (human) | Potency | 14.4761 | 3 | 0 |
4-[2-(2-chloro-4-fluoroanilino)-5-methyl-4-pyrimidinyl]-N-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-1H-pyrrole-2-carboxamide | Homo sapiens (human) | Potency | 21.0004 | 4 | 0 |
osi 906 | Homo sapiens (human) | Potency | 10.0278 | 4 | 0 |
zstk474 | Homo sapiens (human) | Potency | 1.1661 | 4 | 0 |
4-cyano-N-[4-(4-methyl-1-piperazinyl)-2-(4-methyl-1-piperidinyl)phenyl]-1H-pyrrole-2-carboxamide | Homo sapiens (human) | Potency | 29.0836 | 4 | 0 |
ly2109761 | Homo sapiens (human) | Potency | 23.6502 | 4 | 0 |
chir-265 | Homo sapiens (human) | Potency | 7.3988 | 4 | 0 |
motesanib | Homo sapiens (human) | Potency | 8.0350 | 4 | 0 |
fostamatinib | Homo sapiens (human) | Potency | 9.7851 | 4 | 0 |
az-628 | Homo sapiens (human) | Potency | 16.7983 | 4 | 0 |
jnj 28312141 | Homo sapiens (human) | Potency | 17.3546 | 4 | 0 |
omecamtiv mecarbil | Homo sapiens (human) | Potency | 6.6610 | 3 | 0 |
trametinib | Homo sapiens (human) | Potency | 13.1921 | 4 | 0 |
mln8054 | Homo sapiens (human) | Potency | 0.6920 | 4 | 0 |
pf-562,271 | Homo sapiens (human) | Potency | 9.1232 | 4 | 0 |
pha 767491 | Homo sapiens (human) | Potency | 3.6318 | 4 | 0 |
abexinostat | Homo sapiens (human) | Potency | 0.9666 | 4 | 0 |
N-[3-[[5-bromo-4-[2-(1H-imidazol-5-yl)ethylamino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide | Homo sapiens (human) | Potency | 3.6440 | 4 | 0 |
N-(2,4-dimethoxyphenyl)-N-[2-[4-(4-methyl-1-piperazinyl)anilino]-4-pyrimidinyl]carbamic acid (2,6-dimethylphenyl) ester | Homo sapiens (human) | Potency | 2.3711 | 4 | 0 |
at 13387 | Homo sapiens (human) | Potency | 0.3212 | 4 | 0 |
ly2603618 | Homo sapiens (human) | Potency | 1.0904 | 4 | 0 |
veliparib | Homo sapiens (human) | Potency | 22.5027 | 2 | 0 |
ku-0060648 | Homo sapiens (human) | Potency | 8.2246 | 4 | 0 |
Glycyl-H-1152 | Homo sapiens (human) | Potency | 6.7407 | 4 | 0 |
dactolisib | Homo sapiens (human) | Potency | 0.0422 | 4 | 0 |
bgt226 | Homo sapiens (human) | Potency | 0.0170 | 4 | 0 |
palomid 529 | Homo sapiens (human) | Potency | 19.6384 | 4 | 0 |
sc1 compound | Homo sapiens (human) | Potency | 0.5102 | 4 | 0 |
bilobalide | Homo sapiens (human) | Potency | 20.9310 | 1 | 0 |
(7R,9S)-9-acetyl-7-[[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-methyl-2-oxanyl]oxy]-6,9,11-trihydroxy-4-methoxy-8,10-dihydro-7H-tetracene-5,12-dione | Homo sapiens (human) | Potency | 0.0519 | 4 | 0 |
4-[(1,4-dioxo-2-naphthalenyl)amino]benzenesulfonamide | Homo sapiens (human) | Potency | 10.6293 | 4 | 0 |
doxifluridine | Homo sapiens (human) | Potency | 14.0072 | 4 | 0 |
3'',4''-Diacetylafzelin | Homo sapiens (human) | Potency | 26.9236 | 2 | 0 |
tosedostat | Homo sapiens (human) | Potency | 20.5788 | 4 | 0 |
novobiocin | Homo sapiens (human) | Potency | 4.6444 | 4 | 0 |
ku 60019 | Homo sapiens (human) | Potency | 21.6390 | 4 | 0 |
gsk 461364 | Homo sapiens (human) | Potency | 0.0791 | 4 | 0 |
azd 1152-hqpa | Homo sapiens (human) | Potency | 3.0197 | 4 | 0 |
nvp-tae684 | Homo sapiens (human) | Potency | 6.9935 | 4 | 0 |
a 803467 | Homo sapiens (human) | Potency | 35.1973 | 4 | 0 |
4-methyl-3-(2-(2-morpholinoethylamino)quinazolin-6-yl)-n-(3-(trifluoromethyl)phenyl)benzamide | Homo sapiens (human) | Potency | 14.0561 | 4 | 0 |
gsk 269962a | Homo sapiens (human) | Potency | 9.1939 | 4 | 0 |
tak-901 | Homo sapiens (human) | Potency | 1.1031 | 4 | 0 |
cct129202 | Homo sapiens (human) | Potency | 22.3463 | 4 | 0 |
a-83-01 | Homo sapiens (human) | Potency | 13.2942 | 2 | 0 |
3-[(1-methyl-3-indolyl)methylidene]-1H-pyrrolo[3,2-b]pyridin-2-one | Homo sapiens (human) | Potency | 33.3936 | 2 | 0 |
buparlisib | Homo sapiens (human) | Potency | 0.5686 | 4 | 0 |
azd 1480 | Homo sapiens (human) | Potency | 15.0215 | 4 | 0 |
azd8330 | Homo sapiens (human) | Potency | 0.0019 | 1 | 0 |
lumacaftor | Homo sapiens (human) | Potency | 0.0473 | 4 | 0 |
pha 848125 | Homo sapiens (human) | Potency | 2.2083 | 4 | 0 |
tg101209 | Homo sapiens (human) | Potency | 2.4280 | 4 | 0 |
fedratinib | Homo sapiens (human) | Potency | 0.2356 | 2 | 0 |
gsk690693 | Homo sapiens (human) | Potency | 21.0699 | 4 | 0 |
cnf 2024 | Homo sapiens (human) | Potency | 0.1633 | 4 | 0 |
ku 0063794 | Homo sapiens (human) | Potency | 0.6527 | 4 | 0 |
azd 7545 | Homo sapiens (human) | Potency | 21.0236 | 3 | 0 |
nvp-bhg712 | Homo sapiens (human) | Potency | 14.9715 | 4 | 0 |
azd5438 | Homo sapiens (human) | Potency | 4.0458 | 4 | 0 |
nutlin-3b | Homo sapiens (human) | Potency | 14.2912 | 4 | 0 |
amg 1 | Homo sapiens (human) | Potency | 26.2760 | 4 | 0 |
cct 128930 | Homo sapiens (human) | Potency | 17.1333 | 4 | 0 |
gdc 0941 | Homo sapiens (human) | Potency | 2.2891 | 4 | 0 |
sm 164 | Homo sapiens (human) | Potency | 28.8500 | 4 | 0 |
N-[5-[[5-[(4-acetyl-1-piperazinyl)-oxomethyl]-4-methoxy-2-methylphenyl]thio]-2-thiazolyl]-4-[(3-methylbutan-2-ylamino)methyl]benzamide | Homo sapiens (human) | Potency | 10.7735 | 4 | 0 |
3-(3,4-dihydroxyphenyl)lactate | Homo sapiens (human) | Potency | 30.7684 | 3 | 0 |
ph 797804 | Homo sapiens (human) | Potency | 30.3531 | 4 | 0 |
pha 408 | Homo sapiens (human) | Potency | 10.2372 | 4 | 0 |
kw-2478 | Homo sapiens (human) | Potency | 1.1463 | 4 | 0 |
cefpodoxime | Homo sapiens (human) | Potency | 26.7014 | 4 | 0 |
gsk 1016790a | Homo sapiens (human) | Potency | 22.8465 | 4 | 0 |
kx-01 | Homo sapiens (human) | Potency | 0.0269 | 4 | 0 |
mesna | Homo sapiens (human) | Potency | 0.0021 | 1 | 0 |
olaparib | Homo sapiens (human) | Potency | 10.3000 | 4 | 0 |
srt1720 | Homo sapiens (human) | Potency | 28.3518 | 4 | 0 |
plx 4720 | Homo sapiens (human) | Potency | 17.1884 | 4 | 0 |
ast 1306 | Homo sapiens (human) | Potency | 1.0629 | 4 | 0 |
mk 5108 | Homo sapiens (human) | Potency | 1.8659 | 4 | 0 |
cx 4945 | Homo sapiens (human) | Potency | 5.5470 | 4 | 0 |
pci 34051 | Homo sapiens (human) | Potency | 11.2632 | 4 | 0 |
cudc 101 | Homo sapiens (human) | Potency | 0.0478 | 4 | 0 |
purfalcamine | Homo sapiens (human) | Potency | 0.0017 | 1 | 0 |
amg 458 | Homo sapiens (human) | Potency | 28.1336 | 4 | 0 |
cpi 613 | Homo sapiens (human) | Potency | 1.6592 | 2 | 0 |
mln 8237 | Homo sapiens (human) | Potency | 0.5327 | 4 | 0 |
snx 2112 | Homo sapiens (human) | Potency | 0.1046 | 4 | 0 |
lde225 | Homo sapiens (human) | Potency | 15.2922 | 4 | 0 |
gdc 0449 | Homo sapiens (human) | Potency | 1.4216 | 3 | 0 |
sgx 523 | Homo sapiens (human) | Potency | 25.2484 | 2 | 0 |
bms 754807 | Homo sapiens (human) | Potency | 1.1426 | 4 | 0 |
gdc-0068 | Homo sapiens (human) | Potency | 5.1885 | 4 | 0 |
bms 777607 | Homo sapiens (human) | Potency | 29.3412 | 4 | 0 |
sgi 1776 | Homo sapiens (human) | Potency | 14.2373 | 4 | 0 |
lomibuvir | Homo sapiens (human) | Potency | 27.4224 | 3 | 0 |
1-(1-(1-methylcyclooctyl)-4-piperidinyl)-2-((3r)-3-piperidinyl)-1h-benzimidazole | Homo sapiens (human) | Potency | 15.4949 | 4 | 0 |
delanzomib | Homo sapiens (human) | Potency | 0.0592 | 4 | 0 |
pci 32765 | Homo sapiens (human) | Potency | 23.1592 | 4 | 0 |
cink4 | Homo sapiens (human) | Potency | 27.6354 | 4 | 0 |
ponatinib | Homo sapiens (human) | Potency | 5.4355 | 4 | 0 |
amg 900 | Homo sapiens (human) | Potency | 0.0106 | 4 | 0 |
mk-1775 | Homo sapiens (human) | Potency | 0.2627 | 4 | 0 |
tak-875 | Homo sapiens (human) | Potency | 20.9310 | 2 | 0 |
cgi 1746 | Homo sapiens (human) | Potency | 22.5207 | 4 | 0 |
apalutamide | Homo sapiens (human) | Potency | 5.1998 | 4 | 0 |
bag956 | Homo sapiens (human) | Potency | 0.1217 | 4 | 0 |
N-[[3-fluoro-4-[[2-(1-methyl-4-imidazolyl)-7-thieno[3,2-b]pyridinyl]oxy]anilino]-sulfanylidenemethyl]-2-phenylacetamide | Homo sapiens (human) | Potency | 21.6390 | 4 | 0 |
PP121 | Homo sapiens (human) | Potency | 1.0682 | 4 | 0 |
as 605240 | Homo sapiens (human) | Potency | 11.0335 | 4 | 0 |
SL-327 | Homo sapiens (human) | Potency | 6.2411 | 4 | 0 |
N-[4-[3-[[[7-(hydroxyamino)-7-oxoheptyl]amino]-oxomethyl]-5-isoxazolyl]phenyl]carbamic acid tert-butyl ester | Homo sapiens (human) | Potency | 2.0082 | 4 | 0 |
niraparib | Homo sapiens (human) | Potency | 3.8407 | 4 | 0 |
tak 733 | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
mk 2206 | Homo sapiens (human) | Potency | 15.5771 | 4 | 0 |
navitoclax | Homo sapiens (human) | Potency | 19.9572 | 4 | 0 |
mk 8245 | Homo sapiens (human) | Potency | 0.0047 | 1 | 0 |
sns 314 | Homo sapiens (human) | Potency | 0.5199 | 4 | 0 |
mk 3207 | Homo sapiens (human) | Potency | 0.0209 | 1 | 0 |
jzl 184 | Homo sapiens (human) | Potency | 26.9236 | 2 | 0 |
at 406 | Homo sapiens (human) | Potency | 34.5227 | 3 | 0 |
gsk 650394 | Homo sapiens (human) | Potency | 8.1004 | 3 | 0 |
pf-04691502 | Homo sapiens (human) | Potency | 0.0712 | 4 | 0 |
n-(cyanomethyl)-4-(2-((4-(4-morpholinyl)phenyl)amino)-4-pyrimidinyl)benzamide | Homo sapiens (human) | Potency | 11.5722 | 4 | 0 |
dcc-2036 | Homo sapiens (human) | Potency | 19.2857 | 4 | 0 |
oprozomib | Homo sapiens (human) | Potency | 0.1702 | 4 | 0 |
az 960 | Homo sapiens (human) | Potency | 4.3097 | 4 | 0 |
cabozantinib | Homo sapiens (human) | Potency | 1.5952 | 4 | 0 |
N-(2,6-difluorophenyl)-5-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonyl-1-piperazinyl)-1-piperidinyl]anilino]-4-pyrimidinyl]-2-imidazo[1,2-a]pyridinyl]-2-methoxybenzamide | Homo sapiens (human) | Potency | 20.0716 | 4 | 0 |
bs 194 | Homo sapiens (human) | Potency | 0.3500 | 4 | 0 |
incb-018424 | Homo sapiens (human) | Potency | 23.3583 | 4 | 0 |
asp3026 | Homo sapiens (human) | Potency | 17.7575 | 4 | 0 |
bix 01294 | Homo sapiens (human) | Potency | 7.8768 | 4 | 0 |
cct 137690 | Homo sapiens (human) | Potency | 8.8962 | 4 | 0 |
pf 3845 | Homo sapiens (human) | Potency | 18.1476 | 4 | 0 |
TAK-580 | Homo sapiens (human) | Potency | 24.2014 | 4 | 0 |
gsk 2126458 | Homo sapiens (human) | Potency | 0.0456 | 4 | 0 |
emd1214063 | Homo sapiens (human) | Potency | 16.2623 | 4 | 0 |
gsk 1838705a | Homo sapiens (human) | Potency | 12.6523 | 4 | 0 |
ixazomib | Homo sapiens (human) | Potency | 0.3030 | 4 | 0 |
ldn 193189 | Homo sapiens (human) | Potency | 12.4607 | 4 | 0 |
gne 477 | Homo sapiens (human) | Potency | 0.0571 | 4 | 0 |
nvp-bep800 | Homo sapiens (human) | Potency | 1.0662 | 4 | 0 |
1-[4-[[4-amino-5-chloro-6-(2-propan-2-ylsulfonylanilino)-2-pyrimidinyl]amino]-3-methoxyphenyl]-4-piperidinecarboxamide | Homo sapiens (human) | Potency | 11.3063 | 4 | 0 |
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamide | Homo sapiens (human) | Potency | 2.9001 | 4 | 0 |
pf 3758309 | Homo sapiens (human) | Potency | 3.6749 | 4 | 0 |
telotristat etiprate | Homo sapiens (human) | Potency | 24.2793 | 4 | 0 |
cx 5461 | Homo sapiens (human) | Potency | 5.2539 | 3 | 0 |
wye 125132 | Homo sapiens (human) | Potency | 0.0202 | 4 | 0 |
plx4032 | Homo sapiens (human) | Potency | 18.1102 | 4 | 0 |
(2S)-2-[[2-(2,3-dihydro-1H-inden-5-yloxy)-9-[(4-phenylphenyl)methyl]-6-purinyl]amino]-3-phenyl-1-propanol | Homo sapiens (human) | Potency | 11.2835 | 4 | 0 |
N-[3-[[2-[[4-(dimethylamino)cyclohexyl]amino]-9-propan-2-yl-6-purinyl]amino]phenyl]-2-propenamide | Homo sapiens (human) | Potency | 0.3567 | 4 | 0 |
4-[(9-cyclopentyl-6-oxo-5-propan-2-yl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidinyl)benzamide | Homo sapiens (human) | Potency | 2.2208 | 4 | 0 |
gsk 1363089 | Homo sapiens (human) | Potency | 5.7317 | 4 | 0 |
arry-334543 | Homo sapiens (human) | Potency | 9.4447 | 4 | 0 |
kin-193 | Homo sapiens (human) | Potency | 28.4944 | 4 | 0 |
mk 2461 | Homo sapiens (human) | Potency | 10.1490 | 4 | 0 |
N-(2-chlorophenyl)-4-[[2-[4-[2-(4-ethyl-1-piperazinyl)-2-oxoethyl]anilino]-5-fluoro-4-pyrimidinyl]amino]benzamide | Homo sapiens (human) | Potency | 5.3412 | 4 | 0 |
8-chloro-4-(3-chloro-4-fluoroanilino)-6-[[1-(1-ethyl-4-piperidinyl)-4-triazolyl]methylamino]-3-quinolinecarbonitrile | Homo sapiens (human) | Potency | 18.7167 | 4 | 0 |
bay 869766 | Homo sapiens (human) | Potency | 18.2031 | 4 | 0 |
as 703026 | Homo sapiens (human) | Potency | 19.1067 | 4 | 0 |
pki 402 | Homo sapiens (human) | Potency | 0.0176 | 4 | 0 |
pf 04929113 | Homo sapiens (human) | Potency | 0.1685 | 4 | 0 |
baricitinib | Homo sapiens (human) | Potency | 3.7202 | 4 | 0 |
nvp bvu972 | Homo sapiens (human) | Potency | 0.0469 | 1 | 0 |
4-[6-[4-(methoxycarbonylamino)phenyl]-4-(4-morpholinyl)-1-pyrazolo[3,4-d]pyrimidinyl]-1-piperidinecarboxylic acid methyl ester | Homo sapiens (human) | Potency | 0.0966 | 4 | 0 |
ly2811376 | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
dabrafenib | Homo sapiens (human) | Potency | 10.2554 | 4 | 0 |
as1949490 | Homo sapiens (human) | Potency | 17.9237 | 4 | 0 |
3-[2-[2-chloro-4-[[3-(2,6-dichlorophenyl)-5-propan-2-yl-4-isoxazolyl]methoxy]phenyl]ethenyl]benzoic acid | Homo sapiens (human) | Potency | 18.6548 | 2 | 0 |
3-[[4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-1,4-diazepan-1-yl]sulfonyl]aniline | Homo sapiens (human) | Potency | 15.7220 | 2 | 0 |
cp 466722 | Homo sapiens (human) | Potency | 14.2231 | 4 | 0 |
an2728 | Homo sapiens (human) | Potency | 31.7859 | 2 | 0 |
CAY10626 | Homo sapiens (human) | Potency | 0.0337 | 4 | 0 |
N-[3-[[5-chloro-2-[4-(4-methyl-1-piperazinyl)anilino]-4-pyrimidinyl]oxy]phenyl]-2-propenamide | Homo sapiens (human) | Potency | 5.6092 | 4 | 0 |
thiopental sodium | Homo sapiens (human) | Potency | 0.0154 | 4 | 0 |
yk 4-279 | Homo sapiens (human) | Potency | 2.2026 | 4 | 0 |
5-(4-amino-1-propan-2-yl-3-pyrazolo[3,4-d]pyrimidinyl)-1,3-benzoxazol-2-amine | Homo sapiens (human) | Potency | 0.0093 | 4 | 0 |
pha 793887 | Homo sapiens (human) | Potency | 0.7981 | 4 | 0 |
stemregenin 1 | Homo sapiens (human) | Potency | 5.9769 | 4 | 0 |
thiazovivin | Homo sapiens (human) | Potency | 26.4832 | 4 | 0 |
ly2784544 | Homo sapiens (human) | Potency | 9.6209 | 4 | 0 |
unc 0638 | Homo sapiens (human) | Potency | 6.5025 | 4 | 0 |
jzl195 | Homo sapiens (human) | Potency | 29.5659 | 1 | 0 |
mk-8776 | Homo sapiens (human) | Potency | 0.1960 | 4 | 0 |
nvp-bsk805 | Homo sapiens (human) | Potency | 20.3620 | 4 | 0 |
xmd 8-92 | Homo sapiens (human) | Potency | 19.4171 | 4 | 0 |
lrrk2-in1 | Homo sapiens (human) | Potency | 7.8546 | 4 | 0 |
bms 708163 | Homo sapiens (human) | Potency | 14.4732 | 4 | 0 |
gsk 1070916 | Homo sapiens (human) | Potency | 2.8106 | 4 | 0 |
gsk923295 | Homo sapiens (human) | Potency | 0.2115 | 4 | 0 |
jq1 compound | Homo sapiens (human) | Potency | 5.2276 | 4 | 0 |
jnj38877605 | Homo sapiens (human) | Potency | 15.4688 | 4 | 0 |
N-[3-(1,3-benzothiazol-2-yl)-5,6-dihydro-4H-thieno[2,3-c]pyrrol-2-yl]acetamide | Homo sapiens (human) | Potency | 15.3192 | 4 | 0 |
lgk974 | Homo sapiens (human) | Potency | 19.9242 | 4 | 0 |
gsk525762a | Homo sapiens (human) | Potency | 4.3556 | 4 | 0 |
1-[(3,4-difluorophenyl)methyl]-2-oxo-N-[(1R)-2-[(2-oxo-1,3-dihydrobenzimidazol-5-yl)oxy]-1-phenylethyl]-3-pyridinecarboxamide | Homo sapiens (human) | Potency | 24.0611 | 4 | 0 |
ch 5132799 | Homo sapiens (human) | Potency | 0.5778 | 4 | 0 |
alectinib | Homo sapiens (human) | Potency | 0.0130 | 4 | 0 |
ML240 | Homo sapiens (human) | Potency | 8.8722 | 4 | 0 |
glpg0634 | Homo sapiens (human) | Potency | 10.9145 | 4 | 0 |
torin 1 | Homo sapiens (human) | Potency | 0.0235 | 4 | 0 |
abt-199 | Homo sapiens (human) | Potency | 22.5226 | 4 | 0 |
ly2940680 | Homo sapiens (human) | Potency | 25.0036 | 4 | 0 |
tubastatin a | Homo sapiens (human) | Potency | 15.4235 | 4 | 0 |
1-[4-fluoro-3-(trifluoromethyl)phenyl]-3-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)urea | Homo sapiens (human) | Potency | 34.2954 | 4 | 0 |
xl765 | Homo sapiens (human) | Potency | 19.2239 | 4 | 0 |
bs-181 | Homo sapiens (human) | Potency | 10.0674 | 4 | 0 |
ro 4929097 | Homo sapiens (human) | Potency | 17.6919 | 4 | 0 |
mln 9708 | Homo sapiens (human) | Potency | 0.2298 | 4 | 0 |
gsk4112 | Homo sapiens (human) | Potency | 3.1416 | 3 | 0 |
bms-911543 | Homo sapiens (human) | Potency | 24.2084 | 4 | 0 |
ve 821 | Homo sapiens (human) | Potency | 9.2911 | 3 | 0 |
spautin-1 | Homo sapiens (human) | Potency | 13.5000 | 4 | 0 |
azd4547 | Homo sapiens (human) | Potency | 16.2784 | 4 | 0 |
torin 2 | Homo sapiens (human) | Potency | 0.0104 | 4 | 0 |
pf-4708671 | Homo sapiens (human) | Potency | 18.2095 | 4 | 0 |
gsk1210151a | Homo sapiens (human) | Potency | 8.6614 | 4 | 0 |
apr-246 | Homo sapiens (human) | Potency | 2.3563 | 4 | 0 |
3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-(4-(4-ethylpiperazin-1-yl)-phenylamino)pyrimidin-4-yl)-1-methylurea | Homo sapiens (human) | Potency | 37.2212 | 1 | 0 |
acy-1215 | Homo sapiens (human) | Potency | 5.3081 | 4 | 0 |
bp-1-102 | Homo sapiens (human) | Potency | 10.7390 | 4 | 0 |
as 604850 | Homo sapiens (human) | Potency | 32.3816 | 4 | 0 |
chir 98014 | Homo sapiens (human) | Potency | 3.4067 | 3 | 0 |
N-(3-chlorophenyl)-3-[[3,5-dimethyl-4-[(4-methyl-1-piperazinyl)-oxomethyl]-1H-pyrrol-2-yl]methylidene]-N-methyl-2-oxo-1H-indole-5-sulfonamide | Homo sapiens (human) | Potency | 29.0682 | 4 | 0 |
N-[4-(1-benzoyl-4-piperidinyl)butyl]-3-(3-pyridinyl)-2-propenamide | Homo sapiens (human) | Potency | 0.0050 | 4 | 0 |
N-[4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide | Homo sapiens (human) | Potency | 3.0104 | 4 | 0 |
2-methoxy-N-[3-[4-[3-methyl-4-[(6-methyl-3-pyridinyl)oxy]anilino]-6-quinazolinyl]prop-2-enyl]acetamide | Homo sapiens (human) | Potency | 27.6907 | 4 | 0 |
belinostat | Homo sapiens (human) | Potency | 2.0718 | 4 | 0 |
bibr 1532 | Homo sapiens (human) | Potency | 9.3057 | 4 | 0 |
cudc-907 | Homo sapiens (human) | Potency | 0.0060 | 4 | 0 |
tetracycline | Homo sapiens (human) | Potency | 10.7606 | 4 | 0 |
minocycline | Homo sapiens (human) | Potency | 5.9947 | 4 | 0 |
piroxicam | Homo sapiens (human) | Potency | 36.2093 | 4 | 0 |
mobiflex | Homo sapiens (human) | Potency | 13.4151 | 2 | 0 |
ethyl 1-benzyl-3-hydroxy-2(5h)-oxopyrrole-4-carboxylate | Homo sapiens (human) | Potency | 11.7704 | 1 | 0 |
warfarin | Homo sapiens (human) | Potency | 0.0030 | 2 | 0 |
2-[[[4-hydroxy-2-oxo-1-(phenylmethyl)-3-quinolinyl]-oxomethyl]amino]acetic acid | Homo sapiens (human) | Potency | 20.4680 | 4 | 0 |
lornoxicam | Homo sapiens (human) | Potency | 8.3070 | 4 | 0 |
a 769662 | Homo sapiens (human) | Potency | 19.4722 | 4 | 0 |
dolutegravir | Homo sapiens (human) | Potency | 19.0694 | 4 | 0 |
agi-5198 | Homo sapiens (human) | Potency | 11.5754 | 2 | 0 |
pf-5274857 | Homo sapiens (human) | Potency | 9.3284 | 2 | 0 |
3-[[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)-4-pyrimidinyl]amino]propanoic acid | Homo sapiens (human) | Potency | 20.3447 | 3 | 0 |
pik 75 | Homo sapiens (human) | Potency | 0.0336 | 4 | 0 |
5-[[5-(4-fluoro-2-hydroxyphenyl)-2-furanyl]methylidene]thiazolidine-2,4-dione | Homo sapiens (human) | Potency | 22.2774 | 4 | 0 |
LimKi 3 | Homo sapiens (human) | Potency | 35.1973 | 4 | 0 |
1-[4-amino-7-[3-(2-methoxyethylamino)propyl]-5-(4-methylphenyl)-6-pyrrolo[2,3-d]pyrimidinyl]-2-fluoroethanone | Homo sapiens (human) | Potency | 9.3885 | 3 | 0 |
cep 33779 | Homo sapiens (human) | Potency | 3.7316 | 4 | 0 |
entecavir | Homo sapiens (human) | Potency | 12.9007 | 4 | 0 |
2-[5-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxy-2-pyrrolylidene]indole | Homo sapiens (human) | Potency | 1.4649 | 4 | 0 |
sr9011 | Homo sapiens (human) | Potency | 19.9242 | 4 | 0 |
4-[[9-[(3R)-3-oxolanyl]-8-(2,4,6-trifluoroanilino)-2-purinyl]amino]-1-cyclohexanol | Homo sapiens (human) | Potency | 11.9610 | 4 | 0 |
N-hydroxy-3-[4-[[2-(2-methyl-1H-indol-3-yl)ethylamino]methyl]phenyl]-2-propenamide | Homo sapiens (human) | Potency | 0.0793 | 4 | 0 |
3-[(5-tert-butyl-1H-imidazol-4-yl)methylidene]-6-(phenylmethylene)piperazine-2,5-dione | Homo sapiens (human) | Potency | 35.3143 | 2 | 0 |
gsk837149a | Homo sapiens (human) | Potency | 21.8482 | 4 | 0 |
N-[4-(3-chloro-4-fluoroanilino)-7-[[(3S)-3-oxolanyl]oxy]-6-quinazolinyl]-4-(dimethylamino)-2-butenamide | Homo sapiens (human) | Potency | 18.2095 | 4 | 0 |
N-[4-(3-chloro-4-fluoroanilino)-7-methoxy-6-quinazolinyl]-4-(1-piperidinyl)-2-butenamide | Homo sapiens (human) | Potency | 6.5904 | 4 | 0 |
wnt-c59 | Homo sapiens (human) | Potency | 16.1362 | 4 | 0 |
5-[1-(2-hydroxyethyl)-3-pyridin-4-yl-4-pyrazolyl]-2,3-dihydroinden-1-one oxime | Homo sapiens (human) | Potency | 29.9741 | 3 | 0 |
d159687 | Homo sapiens (human) | Potency | 23.1592 | 4 | 0 |
HG-10-102-01 | Homo sapiens (human) | Potency | 6.6629 | 2 | 0 |
N-[(5-methyl-2-furanyl)methylideneamino]-2-phenoxybenzamide | Homo sapiens (human) | Potency | 22.1617 | 3 | 0 |
N-[5-[[6-[3-(1,3-dioxo-2-isoindolyl)phenyl]-4-pyrimidinyl]amino]-2-methylphenyl]methanesulfonamide | Homo sapiens (human) | Potency | 23.4920 | 4 | 0 |
[4-[2-(1H-indazol-3-yl)ethenyl]phenyl]-(1-piperazinyl)methanone | Homo sapiens (human) | Potency | 1.9383 | 4 | 0 |
gsk-2816126 | Homo sapiens (human) | Potency | 20.8690 | 4 | 0 |
N-cyclopropyl-3-[3-[[cyclopropyl(oxo)methyl]amino]-1H-indazol-6-yl]benzamide | Homo sapiens (human) | Potency | 1.9210 | 4 | 0 |
1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-[4-methyl-3-[[2-oxo-3-(1H-pyrrol-2-ylmethylidene)-1H-indol-6-yl]amino]phenyl]urea | Homo sapiens (human) | Potency | 26.4380 | 4 | 0 |
9-(3,5-dimethoxyphenyl)-1-[4-(1-piperazinyl)-3-(trifluoromethyl)phenyl]-2-benzo[h][1,6]naphthyridinone | Homo sapiens (human) | Potency | 3.2713 | 4 | 0 |
agi-6780 | Homo sapiens (human) | Potency | 23.4226 | 4 | 0 |
khs101 | Homo sapiens (human) | Potency | 14.8621 | 4 | 0 |
GSK1059615 | Homo sapiens (human) | Potency | 0.1398 | 4 | 0 |
3-[4-[3-(3-fluorophenyl)-3-oxoprop-1-enyl]-1-methyl-2-pyrrolyl]-N-hydroxy-2-propenamide | Homo sapiens (human) | Potency | 19.9242 | 4 | 0 |
9-(1-methyl-4-pyrazolyl)-1-[1-(1-oxoprop-2-enyl)-2,3-dihydroindol-6-yl]-2-benzo[h][1,6]naphthyridinone | Homo sapiens (human) | Potency | 4.1427 | 4 | 0 |
[4-amino-2-[2-methoxy-4-(4-methyl-1-piperazinyl)anilino]-5-thiazolyl]-(2,6-dichlorophenyl)methanone | Homo sapiens (human) | Potency | 11.2522 | 4 | 0 |
N-[2-methyl-5-[oxo-[3-(1-oxoprop-2-enylamino)-5-(trifluoromethyl)anilino]methyl]phenyl]-5-isoxazolecarboxamide | Homo sapiens (human) | Potency | 22.2080 | 4 | 0 |
3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-[4-(diethylamino)butylamino]-1-methyl-4H-pyrimido[4,5-d]pyrimidin-2-one | Homo sapiens (human) | Potency | 20.3620 | 4 | 0 |
(8R,9S,13S,14R,17R)-17-ethynyl-13-methyl-7,8,9,11,12,14,15,16-octahydro-6H-cyclopenta[a]phenanthrene-3,17-diol | Homo sapiens (human) | Potency | 19.2857 | 4 | 0 |
at 9283 | Homo sapiens (human) | Potency | 2.8120 | 4 | 0 |
akt-i-1,2 compound | Homo sapiens (human) | Potency | 21.0004 | 4 | 0 |
chir 258 | Homo sapiens (human) | Potency | 11.8264 | 4 | 0 |
acyclovir | Homo sapiens (human) | Potency | 0.2957 | 1 | 0 |
osi 027 | Homo sapiens (human) | Potency | 0.6367 | 4 | 0 |
3-methyladenine | Homo sapiens (human) | Potency | 0.2180 | 4 | 0 |
clozapine | Homo sapiens (human) | Potency | 34.6694 | 3 | 0 |
didanosine | Homo sapiens (human) | Potency | 34.2954 | 4 | 0 |
ganciclovir | Homo sapiens (human) | Potency | 15.8824 | 4 | 0 |
valacyclovir | Homo sapiens (human) | Potency | 17.2471 | 2 | 0 |
sildenafil | Homo sapiens (human) | Potency | 12.0250 | 4 | 0 |
chir-124 | Homo sapiens (human) | Potency | 0.4655 | 4 | 0 |
raltitrexed | Homo sapiens (human) | Potency | 0.0243 | 4 | 0 |
vardenafil | Homo sapiens (human) | Potency | 7.2078 | 4 | 0 |
hli 373 | Homo sapiens (human) | Potency | 4.3148 | 4 | 0 |
bl 4162a | Homo sapiens (human) | Potency | 22.8465 | 4 | 0 |
pemetrexed | Homo sapiens (human) | Potency | 0.3903 | 4 | 0 |
xav939 | Homo sapiens (human) | Potency | 24.3667 | 4 | 0 |
hesperadin | Homo sapiens (human) | Potency | 0.2402 | 4 | 0 |
nintedanib | Homo sapiens (human) | Potency | 1.4225 | 4 | 0 |
heliomycin | Homo sapiens (human) | Potency | 31.9709 | 3 | 0 |
bms 536924 | Homo sapiens (human) | Potency | 5.8760 | 4 | 0 |
amg531 | Homo sapiens (human) | Potency | 13.9248 | 4 | 0 |
ver 52296 | Homo sapiens (human) | Potency | 0.0890 | 4 | 0 |
sb-590885 | Homo sapiens (human) | Potency | 29.0456 | 4 | 0 |
sta 9090 | Homo sapiens (human) | Potency | 0.0725 | 4 | 0 |
pf-477736 | Homo sapiens (human) | Potency | 0.5419 | 4 | 0 |
bay 80-6946 | Homo sapiens (human) | Potency | 0.7640 | 4 | 0 |
bix 02189 | Homo sapiens (human) | Potency | 22.9244 | 4 | 0 |
carbazochrome sodium sulfonate | Homo sapiens (human) | Potency | 0.0053 | 2 | 0 |
s-1530 | Homo sapiens (human) | Potency | 30.3562 | 3 | 0 |
6-bromoindirubin-3'-acetoxime | Homo sapiens (human) | Potency | 6.7898 | 4 | 0 |