Proteins > recombinase A
Page last updated: 2024-08-07 19:24:54

recombinase A

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (218)

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
3-hydroxyanthranilic acidMycobacterium tuberculosis H37RvEC505.766020
4-aminophenolMycobacterium tuberculosis H37RvEC50205.710020
benzbromaroneMycobacterium tuberculosis H37RvEC5014.995020
fluspirileneMycobacterium tuberculosis H37RvEC5036.080020
hexachloropheneMycobacterium tuberculosis H37RvEC507.166020
edaravoneMycobacterium tuberculosis H37RvEC503.024520
papaverine hydrochlorideMycobacterium tuberculosis H37RvEC505.156520
methylene blueMycobacterium tuberculosis H37RvEC5078.650020
9,10-phenanthrenequinoneMycobacterium tuberculosis H37RvEC507.193520
n-isopropyl-n-phenyl-4-phenylenediamineMycobacterium tuberculosis H37RvEC50228.200020
1-amino-4-hydroxyanthraquinoneMycobacterium tuberculosis H37RvEC5047.935020
glaucineMycobacterium tuberculosis H37RvEC502.472020
1,2-naphthoquinoneMycobacterium tuberculosis H37RvEC509.135520
6-aminoquinolineMycobacterium tuberculosis H37RvEC5010.960020
diloxanide furoateMycobacterium tuberculosis H37RvEC50195.150020
nitroxolineMycobacterium tuberculosis H37RvEC5019.715020
cetyldimethylethylammonium bromideMycobacterium tuberculosis H37RvEC5015.160020
s-2678Mycobacterium tuberculosis H37RvEC50380.000020
sulconazole, mononitrate, (+-)-isomerMycobacterium tuberculosis H37RvEC5016.425020
physodic acidMycobacterium tuberculosis H37RvEC505.239020
toxoflavinMycobacterium tuberculosis H37RvEC500.054120
2,3-trimethylene-4-quinazoloneMycobacterium tuberculosis H37RvEC5065.100020
miconazole nitrateMycobacterium tuberculosis H37RvEC5016.620020
econazole nitrateMycobacterium tuberculosis H37RvEC5013.830020
epicatechinMycobacterium tuberculosis H37RvEC50380.000020
tosyllysine chloromethyl ketoneMycobacterium tuberculosis H37RvEC5037.630020
lobaric acidMycobacterium tuberculosis H37RvEC508.525020
5-hydroxyuracilMycobacterium tuberculosis H37RvEC5012.230020
tryptanthrineMycobacterium tuberculosis H37RvEC500.984020
6-aminoindazoleMycobacterium tuberculosis H37RvEC5015.310020
5-aminoindazoleMycobacterium tuberculosis H37RvEC5042.355020
9,10-phenanthrenequinone monoximeMycobacterium tuberculosis H37RvEC5023.735020
catechinMycobacterium tuberculosis H37RvEC50124.055020
dichloro-1,2-diaminocyclohexane platinum complexMycobacterium tuberculosis H37RvEC5040.845020
sch 45752Mycobacterium tuberculosis H37RvEC502.034520
17 alpha-hydroxyprogesterone caproateMycobacterium tuberculosis H37RvEC50192.440020
(R)-RoemerineMycobacterium tuberculosis H37RvEC500.474220
papaverinolMycobacterium tuberculosis H37RvEC5017.965020
nsc228155Mycobacterium tuberculosis H37RvEC5012.160020
dicentrineMycobacterium tuberculosis H37RvEC5011.006020
3-imino-1,5,5-trimethyl-2-oxabicyclo[2.2.1]heptane-4,7,7-tricarbonitrileMycobacterium tuberculosis H37RvEC5038.255020
tosylphenylalanyl chloromethyl ketoneMycobacterium tuberculosis H37RvEC501.287520
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneMycobacterium tuberculosis H37RvEC500.068820
menadione sodium bisulfite, trihydrateMycobacterium tuberculosis H37RvEC503.659020
1-phenyl-4-pyrazololMycobacterium tuberculosis H37RvEC5024.140020
2-furancarboxylic acid [4-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterMycobacterium tuberculosis H37RvEC5018.170020
N-[3,5-dimethyl-1-(1-oxopropyl)-4-pyrazolyl]propanamideMycobacterium tuberculosis H37RvEC50380.000020
7-nitro-5-indeno[1,2-b]pyridinoneMycobacterium tuberculosis H37RvEC5091.000020
xanthoangelolMycobacterium tuberculosis H37RvEC50234.200020
6-amino-4-(2-ethoxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5035.505020
6-amino-4-(2-methoxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5011.160020
6-amino-4-(2,3-dimethoxyphenyl)-3-methyl-1-phenyl-4H-pyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC509.785020
6-amino-4-(2,5-dimethoxyphenyl)-3-methyl-1-(4-methylphenyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5017.165020
2-[(3-chlorophenyl)-(3-oxo-5-propyl-1,2-dihydropyrazol-4-yl)methyl]propanedinitrileMycobacterium tuberculosis H37RvEC505.082020
6-amino-4-(2,4-dimethoxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5010.595020
6-amino-4-[3-ethoxy-4-[2-(4-morpholinyl)ethoxy]phenyl]-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5026.370020
6-amino-3-(methoxymethyl)-4-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5024.640020
2-[(3-oxo-5-phenyl-1,2-dihydropyrazol-4-yl)-(3-thiophenyl)methyl]propanedinitrileMycobacterium tuberculosis H37RvEC504.020520
4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl esterMycobacterium tuberculosis H37RvEC502.247020
cyclopropanecarboxylic acid [5-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)-2-ethoxyphenyl] esterMycobacterium tuberculosis H37RvEC5025.285020
2-(3-methylphenyl)sulfonyl-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetonitrileMycobacterium tuberculosis H37RvEC50380.000020
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterMycobacterium tuberculosis H37RvEC50192.330020
4-(1-benzotriazolyl)-5-(2-methoxyphenoxy)benzene-1,2-dicarbonitrileMycobacterium tuberculosis H37RvEC50145.685020
6-amino-3-(methoxymethyl)-5-spiro[2H-pyrano[2,3-c]pyrazole-4,4'-thiane]carbonitrileMycobacterium tuberculosis H37RvEC5011.125020
4-chloro-1-methyl-3-nitro-2-quinolinoneMycobacterium tuberculosis H37RvEC507.395020
5-(4-cyclohexylphenyl)-1,2-dihydropyrazol-3-oneMycobacterium tuberculosis H37RvEC501.449020
2-(3-oxo-2-phenyl-1H-pyrazol-5-yl)acetic acid methyl esterMycobacterium tuberculosis H37RvEC5041.915020
5-amino-3-(4-methoxyphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterMycobacterium tuberculosis H37RvEC5055.195020
2-(4-hydroxyanilino)-1,4-naphthoquinoneMycobacterium tuberculosis H37RvEC503.609520
acetic acid [2-(2-methylphenyl)-4-oxo-3,1-benzoxazin-7-yl] esterMycobacterium tuberculosis H37RvEC50208.900020
N-[4-(1-azepanyl)phenyl]-2-chloroacetamideMycobacterium tuberculosis H37RvEC5037.120020
3-chloro-1-(2-chlorophenyl)-4-(4-morpholinyl)pyrrole-2,5-dioneMycobacterium tuberculosis H37RvEC503.854520
4-[(4-chlorophenyl)thio]-5-methyl-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC5012.320020
[3-(4-chlorophenyl)-5-(methylthio)-1,2,4-triazol-1-yl]-(2-furanyl)methanoneMycobacterium tuberculosis H37RvEC50380.000020
2-[[4-(1-pyrrolidinylsulfonyl)phenyl]hydrazinylidene]propanedinitrileMycobacterium tuberculosis H37RvEC5032.485020
2-chloro-N-[5-ethyl-3-[(4-methylphenyl)-oxomethyl]-2-thiophenyl]acetamideMycobacterium tuberculosis H37RvEC507.670020
5-amino-3-(2-methylphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterMycobacterium tuberculosis H37RvEC50195.700020
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneMycobacterium tuberculosis H37RvEC500.214420
1-methyl-5-(1-naphthalenyloxy)-4-nitroimidazoleMycobacterium tuberculosis H37RvEC5033.790020
umi-77Mycobacterium tuberculosis H37RvEC500.461820
N-(4-methoxyphenyl)-N-thiophen-2-ylsulfonyl-2-furancarboxamideMycobacterium tuberculosis H37RvEC50206.300020
1-(2,1,3-benzothiadiazol-5-yl)-3-[4-(4-morpholinyl)phenyl]ureaMycobacterium tuberculosis H37RvEC50380.000020
N-[2,2-dichloro-1-(4-chlorophenyl)sulfonylethenyl]benzamideMycobacterium tuberculosis H37RvEC50136.415020
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acidMycobacterium tuberculosis H37RvEC5031.095020
2-thiophenecarboxylic acid [3-(3,5-dimethylphenoxy)-4-oxo-1-benzopyran-7-yl] esterMycobacterium tuberculosis H37RvEC50199.400020
5-(4-fluorophenyl)sulfonyl-1-(2-methylpropyl)-4-nitro-2-propan-2-ylimidazoleMycobacterium tuberculosis H37RvEC50194.845020
5-bromo-2-furancarboxylic acid (3-benzamidophenyl) esterMycobacterium tuberculosis H37RvEC5070.600020
1-benzimidazolyl-[2-(4-methoxyphenyl)-4-quinolinyl]methanoneMycobacterium tuberculosis H37RvEC5026.675020
2-(4-hydroxyphenyl)-5-methyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC501.494020
3-chloro-1-(2,5-dimethoxyphenyl)-4-(1-piperidinyl)pyrrole-2,5-dioneMycobacterium tuberculosis H37RvEC5010.790020
(4-chlorophenyl)-(5-hydroxy-2-methyl-4,6-dinitro-3-benzofuranyl)methanoneMycobacterium tuberculosis H37RvEC5016.030020
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneMycobacterium tuberculosis H37RvEC5057.500020
2-(2-chloro-3-pyridinyl)-1-prop-2-enylbenzimidazoleMycobacterium tuberculosis H37RvEC50380.000020
1-(benzenesulfonyl)-3-pyrazolidinoneMycobacterium tuberculosis H37RvEC5018.245020
N-(4-methoxyphenyl)-2-(3-methylphenoxy)-N-(4-methylphenyl)sulfonylacetamideMycobacterium tuberculosis H37RvEC5080.615020
3-chloro-1-(2,4-dimethylphenyl)-4-(2-hydroxyethylamino)pyrrole-2,5-dioneMycobacterium tuberculosis H37RvEC5034.110020
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneMycobacterium tuberculosis H37RvEC5014.500020
4-(1-benzotriazolyl)-3,5-dinitrobenzonitrileMycobacterium tuberculosis H37RvEC50202.950020
[4-methoxy-6-(propan-2-ylamino)-1,3,5-triazin-2-yl]-[(1,1,3-trioxo-1,2-benzothiazol-2-yl)methyl]cyanamideMycobacterium tuberculosis H37RvEC5033.440020
4-(6-fluoro-3-methyl-4-oxo-1-benzopyran-2-yl)-2-methyl-1-phthalazinoneMycobacterium tuberculosis H37RvEC504.661020
N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamideMycobacterium tuberculosis H37RvEC5014.365020
1-[2-(5-fluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(4-fluorophenyl)-1-(3-pyridinylmethyl)thioureaMycobacterium tuberculosis H37RvEC50236.700020
2,2,2-trifluoro-N-(5-oxo-1-phenyl-4H-pyrazol-3-yl)acetamideMycobacterium tuberculosis H37RvEC5011.005020
3-[[(4-tert-butylphenyl)-oxomethyl]amino]-1H-1,2,4-triazole-5-carboxylic acid methyl esterMycobacterium tuberculosis H37RvEC5032.260020
5,6,7,8-tetrafluoro-2-(2,3,4,5,6-pentafluorophenyl)-4h-1-benzopyran-4-oneMycobacterium tuberculosis H37RvEC508.180020
N-[(1-adamantylamino)-oxomethyl]-2-chloroacetamideMycobacterium tuberculosis H37RvEC5017.090020
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideMycobacterium tuberculosis H37RvEC504.589020
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneMycobacterium tuberculosis H37RvEC5014.270020
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideMycobacterium tuberculosis H37RvEC504.030520
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideMycobacterium tuberculosis H37RvEC504.377520
2-chloro-1-[4-[(3-methylphenyl)methyl]-1-piperazinyl]ethanoneMycobacterium tuberculosis H37RvEC5080.300020
2-chloro-N-[(5-chloro-2-thiophenyl)methyl]-N-methylacetamideMycobacterium tuberculosis H37RvEC5038.595020
5-(3-fluorophenoxy)-8-nitroisoquinolineMycobacterium tuberculosis H37RvEC5024.453020
4,5-dichloro-2-[2-[2,5-dimethyl-1-(2,2,2-trifluoroethyl)-3-pyrrolyl]-2-oxoethyl]-3-pyridazinoneMycobacterium tuberculosis H37RvEC504.347020
4-amino-5-hydrazino-1,2,4-triazole-3-thiolMycobacterium tuberculosis H37RvEC50233.200020
3-(tert-butyl)-1-methyl-4,5-dihydro-1H-pyrazol-5-oneMycobacterium tuberculosis H37RvEC5010.530020
1-[4-[(2-bromophenyl)-oxomethyl]-1H-pyrrol-2-yl]-2,2,2-trichloroethanoneMycobacterium tuberculosis H37RvEC5016.215020
2-[4-[[4-[bis(2-hydroxyethyl)amino]-2-chlorophenyl]-(2-chlorophenyl)methyl]-3-chloro-N-(2-hydroxyethyl)anilino]ethanolMycobacterium tuberculosis H37RvEC50124.900010
4b,9b-dihydroxy-7,8-dihydro-6H-indeno[1,2-b]benzofuran-9,10-dioneMycobacterium tuberculosis H37RvEC5010.860020
1-hexadecyl-3-methylimidazolium bromideMycobacterium tuberculosis H37RvEC5010.770020
6-amino-4-(3-chlorophenyl)-3-methyl-1-(phenylmethyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5017.870020
6-amino-4-(2-methylpropyl)-3-phenyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC507.480020
6-amino-4-[3-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-4-methoxyphenyl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5014.795020
4-[[3-methoxy-4-[(4-nitrophenyl)methoxy]phenyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneMycobacterium tuberculosis H37RvEC500.263520
2-(2-hydroxyethylamino)-3-(4-methoxyanilino)naphthalene-1,4-dioneMycobacterium tuberculosis H37RvEC5026.430020
4-methylbenzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-methoxyphenyl] esterMycobacterium tuberculosis H37RvEC500.318620
4-methylbenzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-ethoxyphenyl] esterMycobacterium tuberculosis H37RvEC500.322820
benzenesulfonic acid [4-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-methoxyphenyl] esterMycobacterium tuberculosis H37RvEC500.326720
N-[3-(4-chlorophenyl)-5-oxo-4-pyrazolidinyl]-3-methylbenzamideMycobacterium tuberculosis H37RvEC5032.290020
4-(5-methyl-3-oxo-1H-pyrazol-2-yl)benzoic acidMycobacterium tuberculosis H37RvEC502.375020
6-amino-4-(2-furanyl)-3-propan-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5015.935020
2-[[4-(4-fluorophenyl)-6-(trifluoromethyl)-2-pyrimidinyl]sulfonyl]acetic acid ethyl esterMycobacterium tuberculosis H37RvEC504.669520
zuclomifene citrateMycobacterium tuberculosis H37RvEC5014.950020
2-[[3-methyl-5-oxo-1-(phenylmethyl)-4H-pyrazol-4-yl]-phenylmethyl]propanedinitrileMycobacterium tuberculosis H37RvEC505.462020
2-[(prop-2-enylthio)-(4,5,6,7-tetrahydro-1H-indol-2-yl)methylidene]propanedinitrileMycobacterium tuberculosis H37RvEC5011.595020
acetic acid [1-[(3-nitrophenyl)-(1-oxopentylamino)methyl]-2-naphthalenyl] esterMycobacterium tuberculosis H37RvEC50202.700020
3-[5-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl esterMycobacterium tuberculosis H37RvEC500.355320
2-[6-amino-5-cyano-4-(4-ethylphenyl)-2,4-dihydropyrano[2,3-c]pyrazol-3-yl]acetic acid methyl esterMycobacterium tuberculosis H37RvEC5022.335020
6-amino-4-(3-furanyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC502.603520
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[4-(methylthio)phenyl]methyl]-1,2-dihydropyrazol-3-oneMycobacterium tuberculosis H37RvEC500.404820
N-[2-(tert-butylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2-oxolanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideMycobacterium tuberculosis H37RvEC50274.300020
CID 3192987Mycobacterium tuberculosis H37RvEC501.652020
N-tert-butyl-2-[(2-chloro-1-oxoethyl)-(2-furanylmethyl)amino]-2-(4-chlorophenyl)acetamideMycobacterium tuberculosis H37RvEC5011.950020
2-[[3-(4-fluorophenyl)-7-triazolo[4,5-d]pyrimidinyl]thio]butanoic acid ethyl esterMycobacterium tuberculosis H37RvEC50203.350020
5-(4-piperidinyl)-1,2-dihydropyrazol-3-oneMycobacterium tuberculosis H37RvEC503.400020
4-morpholinecarboxylic acid [4-[6-amino-5-cyano-3-(4-methylphenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]phenyl] esterMycobacterium tuberculosis H37RvEC505.845020
2-[[4-cyano-3-[(2-methoxy-2-oxoethyl)thio]-5-isothiazolyl]thio]acetic acid ethenyl esterMycobacterium tuberculosis H37RvEC5062.920020
N-(1,3-benzodioxol-5-yl)-2-[4-(4-chlorophenyl)sulfonyl-1-piperazinyl]acetamideMycobacterium tuberculosis H37RvEC50380.000020
2-furancarboxylic acid [4-(6-amino-5-cyano-3-propan-2-yl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterMycobacterium tuberculosis H37RvEC5011.555020
4-morpholinecarboxylic acid [3-(6-amino-5-cyano-3-propan-2-yl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterMycobacterium tuberculosis H37RvEC5028.675020
4-morpholinecarboxylic acid [3-(6-amino-5-cyano-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterMycobacterium tuberculosis H37RvEC5028.785020
6-amino-4-(2-ethoxy-4-hydroxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5031.020020
benzoic acid [4-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)-2-methoxyphenyl] esterMycobacterium tuberculosis H37RvEC5032.980020
5-amino-2-(3-nitrophenyl)-1-phenyl-2H-pyrrole-3,3,4-tricarbonitrileMycobacterium tuberculosis H37RvEC5018.420020
2-chloro-N-[2-(2,2-dimethyl-4-phenyl-4-oxanyl)ethyl]acetamideMycobacterium tuberculosis H37RvEC5083.200020
2-(6-amino-5-cyano-3-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)benzoic acidMycobacterium tuberculosis H37RvEC506.890020
6-amino-4-methyl-3-(4-methylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC500.506920
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinolMycobacterium tuberculosis H37RvEC5083.550020
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olMycobacterium tuberculosis H37RvEC501.424520
4-[1-(4-bromophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC5011.470020
ML162Mycobacterium tuberculosis H37RvEC500.597620
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideMycobacterium tuberculosis H37RvEC501.801520
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideMycobacterium tuberculosis H37RvEC501.018520
6-amino-4-(3-furanyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5010.610020
2-[1-(2-methylphenyl)-3-oxo-3-thiophen-2-ylpropyl]propanedinitrileMycobacterium tuberculosis H37RvEC501.676020
5-[(4-chlorophenyl)-oxomethyl]-4-hydroxy-6-[5-(2-nitrophenyl)-2-furanyl]-4-(trifluoromethyl)-1,3-diazinan-2-oneMycobacterium tuberculosis H37RvEC5025.190010
6-amino-3-methyl-4-(2-methylpropyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5012.190020
6-amino-3-(3-methoxyphenyl)-4-(3-thiophenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC504.118520
2-chloro-N-(2-methyl-6-oxo-5H-benzo[b][1,4]benzoxazepin-8-yl)acetamideMycobacterium tuberculosis H37RvEC5036.730020
4-[(4-ethoxy-3-methoxyphenyl)-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneMycobacterium tuberculosis H37RvEC500.375220
2-Chloro-1-[5-(3,4-dimethoxyphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneMycobacterium tuberculosis H37RvEC502.931020
4-[(2-hydroxy-3-nitrophenyl)-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)methyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC501.120520
5-[[(4-chlorophenyl)thio]methyl]-2-methyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC5018.560020
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleMycobacterium tuberculosis H37RvEC501.464020
4-chloro-5-(2,3-dihydro-1,4-benzodioxin-3-yl)thieno[2,3-d]pyrimidineMycobacterium tuberculosis H37RvEC5012.130020
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-1-nitro-9,10-dioxo-2-anthracenecarboxamideMycobacterium tuberculosis H37RvEC5017.190020
[4-(butan-2-ylamino)-6-chloro-1,3,5-triazin-2-yl]-[(1,1,3-trioxo-1,2-benzothiazol-2-yl)methyl]cyanamideMycobacterium tuberculosis H37RvEC5030.945020
1,8-dimethoxyphenazineMycobacterium tuberculosis H37RvEC5022.475020
N-[3-(1-azepanylsulfonyl)-4-methylphenyl]-2-(4-quinazolinylthio)acetamideMycobacterium tuberculosis H37RvEC50191.330020
2-(4-methoxyphenyl)sulfonylquinoxalineMycobacterium tuberculosis H37RvEC5079.200020
5-methyl-4-[(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-(3-nitrophenyl)methyl]-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC502.800520
4-(3-chlorophenyl)sulfonyl-N-cyclohexyl-N-methyl-3-nitrobenzamideMycobacterium tuberculosis H37RvEC50135.665020
2-(N-(2-chloro-1-oxoethyl)-4-fluoroanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMycobacterium tuberculosis H37RvEC506.158020
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMycobacterium tuberculosis H37RvEC505.804520
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMycobacterium tuberculosis H37RvEC503.177020
4-[1-(4-fluorophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvEC5013.300020
6-amino-4-(3,5-dimethyl-1-phenyl-4-pyrazolyl)-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5034.060020
2-Chloro-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneMycobacterium tuberculosis H37RvEC502.379020
N-(1-dibutoxyphosphoryl-4-oxo-1-naphthalenyl)benzenesulfonamideMycobacterium tuberculosis H37RvEC503.402520
3-pyridinecarboxylic acid [4-[heptoxy(oxo)methyl]phenyl] esterMycobacterium tuberculosis H37RvEC50237.070020
4-(1-imidazolyl)-3,5-dinitrobenzoic acid methyl esterMycobacterium tuberculosis H37RvEC507.700020
4-chloro-N-[3-(N-methylanilino)-1,4-dioxo-2-naphthalenyl]benzamideMycobacterium tuberculosis H37RvEC5038.370020
8-nitro-5-[3-(trifluoromethyl)-1-piperidinyl]isoquinolineMycobacterium tuberculosis H37RvEC50195.400020
2-(Chloroacetyl)-N,2-diphenylhydrazinecarboxamideMycobacterium tuberculosis H37RvEC508.005520
2-Chloro-1-[5-(furan-2-yl)-3-(5-methylfuran-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneMycobacterium tuberculosis H37RvEC5022.630020
5-methyl-2-phenyl-4-propan-2-ylidene-3-pyrazoloneMycobacterium tuberculosis H37RvEC505.455520
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazoleMycobacterium tuberculosis H37RvEC50110.590020
4-(3,4-dimethoxyphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazoline-2-thioneMycobacterium tuberculosis H37RvEC5016.940020
6-amino-1,3-diphenyl-4-(3,4,5-trimethoxyphenyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrileMycobacterium tuberculosis H37RvEC5045.515020
prostaglandin f2 methyl esterMycobacterium tuberculosis H37RvEC5052.755020
2-bromoergocryptine mesylateMycobacterium tuberculosis H37RvEC50380.000020
nifuroxazideMycobacterium tuberculosis H37RvEC50380.000020
HTS 01037Mycobacterium tuberculosis H37RvEC5054.480020
enclomiphene citrateMycobacterium tuberculosis H37RvEC5016.240020
N-[1-(5,6-dicyano-3-methyl-2-pyrazinyl)ethyl]-N-phenylacetamideMycobacterium tuberculosis H37RvEC5021.400020
geduninMycobacterium tuberculosis H37RvEC5087.100020
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideMycobacterium tuberculosis H37RvEC500.176820
2-(4-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideMycobacterium tuberculosis H37RvEC500.322620
2-[(2-chloro-1-oxoethyl)-(2,2-dimethoxyethyl)amino]-2-(4-chlorophenyl)-N-cyclohexylacetamideMycobacterium tuberculosis H37RvEC5017.910020
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideMycobacterium tuberculosis H37RvEC502.207020
5-chloro-2-[(3-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideMycobacterium tuberculosis H37RvEC500.584120
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideMycobacterium tuberculosis H37RvEC5020.980020
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideMycobacterium tuberculosis H37RvEC5010.885020
N-[5-Ethyl-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chlorideMycobacterium tuberculosis H37RvEC50198.400020
N-[5-Bromo-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chlorideMycobacterium tuberculosis H37RvEC5074.450020
N-[5-Fluoro-1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-3-yl]acetamide;hydron;chlorideMycobacterium tuberculosis H37RvEC5034.425020
(3R)-3-(4-chlorophenyl)-4-oxo-3-propan-2-yldiazetidine-1,2-dicarboxylic acid diethyl esterMycobacterium tuberculosis H37RvEC503.419520
2-[[3-[(2-ethoxy-2-oxoethyl)thio]-5-oxo-2H-1,2,4-triazin-6-yl]amino]acetic acid butyl esterMycobacterium tuberculosis H37RvEC507.905020

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
glaucineMycobacterium tuberculosis H37RvIC9040.200010
toxoflavinMycobacterium tuberculosis H37RvIC902.870010
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneMycobacterium tuberculosis H37RvIC904.190010
2-chloro-N-[5-ethyl-3-[(4-methylphenyl)-oxomethyl]-2-thiophenyl]acetamideMycobacterium tuberculosis H37RvIC9051.850010
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneMycobacterium tuberculosis H37RvAC500.095020
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneMycobacterium tuberculosis H37RvIC9022.290010
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideMycobacterium tuberculosis H37RvIC909.100010
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideMycobacterium tuberculosis H37RvIC9052.360010
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideMycobacterium tuberculosis H37RvIC908.420010
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideMycobacterium tuberculosis H37RvIC9031.960010
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideMycobacterium tuberculosis H37RvIC9022.940010
5-methyl-4-[(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)-(3-nitrophenyl)methyl]-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvIC90100.000010
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMycobacterium tuberculosis H37RvIC9028.000010
4-[1-(4-fluorophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMycobacterium tuberculosis H37RvIC9032.770010
4-chloro-N-[3-(N-methylanilino)-1,4-dioxo-2-naphthalenyl]benzamideMycobacterium tuberculosis H37RvIC9016.700010
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideMycobacterium tuberculosis H37RvIC90100.000010