Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
aminooxyacetic acid | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
catechol | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
3,4-dihydroxyphenylacetic acid | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
diacetyl | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
hydroquinone | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
spermidine | Homo sapiens (human) | Potency | 6.3096 | 2 | 0 |
spermine | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
1,10-phenanthroline | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
1,3-diethyl-8-phenylxanthine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
1-(3-chlorophenyl)biguanide | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
1-aminobenzotriazole | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
3,4-dichloroisocoumarin | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
4,5,6,7-tetrabromo-2-azabenzimidazole | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
cgp 52411 | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
4-aminobenzamidine | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
p-chloromercuribenzoic acid | Homo sapiens (human) | Potency | 6.3096 | 2 | 0 |
4-phenyl-3-furoxancarbonitrile | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
5-(n,n-hexamethylene)amiloride | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
ethylisopropylamiloride | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
6,7-dichloroquinoxaline-2,3-dione | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
6-chloromelatonin | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
6-nitroso-1,2-benzopyrone | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
tyrphostin a23 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
tyrphostin 25 | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
amiodarone | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
amoxapine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
amsacrine | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid prop-2-ynyl ester | Homo sapiens (human) | Potency | 1.2589 | 2 | 0 |
aurintricarboxylic acid | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
bmy 7378 | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
3-(1-methyl-4-piperidinyl)-1H-indol-5-ol | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
cgs 12066 | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
cgs 15943 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
chelerythrine | Homo sapiens (human) | Potency | 1.9953 | 2 | 0 |
chlorambucil | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
chlorpromazine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
chlorzoxazone | Homo sapiens (human) | Potency | 0.1259 | 2 | 0 |
cilostazol | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
cirazoline | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
clomipramine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
clotrimazole | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
cyclobenzaprine | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
cystamine | Homo sapiens (human) | Potency | 31.6228 | 2 | 0 |
dephostatin | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
dequalinium | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
desipramine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
dicyclomine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
diphenhydramine | Homo sapiens (human) | Potency | 0.0631 | 2 | 0 |
diphenyleneiodonium | Homo sapiens (human) | Potency | 0.0398 | 2 | 0 |
dipyridamole | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
disulfiram | Homo sapiens (human) | Potency | 0.3981 | 2 | 0 |
2,3-dimethoxy-1,4-naphthoquinone | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
ebselen | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
ellipticine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
emodin | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
fluphenazine | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
fluorouracil | Homo sapiens (human) | Potency | 0.0126 | 2 | 0 |
fluspirilene | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
fusaric acid | Homo sapiens (human) | Potency | 1.9953 | 2 | 0 |
vanoxerine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
gbr 12935 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
n-(2-aminoethyl)-5-isoquinolinesulfonamide | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
haloperidol | Homo sapiens (human) | Potency | 6.3096 | 2 | 0 |
hydralazine | Homo sapiens (human) | Potency | 0.0398 | 2 | 0 |
imetit | Homo sapiens (human) | Potency | 0.7943 | 2 | 0 |
indirubin-3'-monoxime | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
iodoacetamide | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
1-(2-naphthalenyl)-3-[(phenylmethyl)-propan-2-ylamino]-1-propanone | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
nsc 664704 | Homo sapiens (human) | Potency | 0.1585 | 2 | 0 |
beta-lapachone | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
leflunomide | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
linopirdine | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
loperamide | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
loratadine | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-one | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
maprotiline | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
methoctramine | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
nocodazole | Homo sapiens (human) | Potency | 0.0126 | 2 | 0 |
mitoxantrone | Homo sapiens (human) | Potency | 0.0251 | 2 | 0 |
ethylmaleimide | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
fg 7142 | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
clorgyline | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
deoxyepinephrine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
n 0840 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
niclosamide | Homo sapiens (human) | Potency | 0.1000 | 2 | 0 |
nifedipine | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
nortriptyline | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
5-nitro-2-(3-phenylpropylamino)benzoic acid | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
papaverine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
pd 169316 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
pd 98059 | Homo sapiens (human) | Potency | 0.3981 | 2 | 0 |
perphenazine | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
pirenperone | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
prochlorperazine | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
promazine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
protriptyline | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
6-nitroquipazine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
n-methylquipazine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
raloxifene | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
ro 41-1049 | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
sanguinarine | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
sb 206553 | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
sb 202190 | Homo sapiens (human) | Potency | 31.6228 | 2 | 0 |
carbamylhydrazine | Homo sapiens (human) | Potency | 0.1259 | 2 | 0 |
sk&f 97541 | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
sobuzoxane | Homo sapiens (human) | Potency | 0.2512 | 2 | 0 |
sulfaphenazole | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
terfenadine | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
8-(n,n-diethylamino)octyl-3,4,5-trimethoxybenzoate | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
ici 136,753 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
trequinsin | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
trifluoperazine | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
trifluperidol | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
triflupromazine | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
tyrphostin a9 | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
w 7 | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
corticosterone | Homo sapiens (human) | Potency | 1.2589 | 2 | 0 |
reserpine | Homo sapiens (human) | Potency | 31.6228 | 2 | 0 |
bretylium tosylate | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
colchicine | Homo sapiens (human) | Potency | 0.5012 | 2 | 0 |
pseudoephedrine | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
synephrine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
suramin sodium | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
pyrazolanthrone | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
azacitidine | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
acetylcysteine | Homo sapiens (human) | Potency | 31.6228 | 2 | 0 |
pimozide | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
dexpropranolol | Homo sapiens (human) | Potency | 0.3162 | 2 | 0 |
levodopa methyl ester | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
propionylpromazine | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
camptothecin | Homo sapiens (human) | Potency | 0.1259 | 2 | 0 |
clemastine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
metergoline | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
carbidopa | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
ribavirin | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
captopril | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
salmeterol xinafoate | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
mibefradil | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
eliprodil | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
aptiganel | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
3-iodobenzylguanidine | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
paroxetine hydrochloride | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
u 37883a | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
rutecarpine | Homo sapiens (human) | Potency | 0.3162 | 2 | 0 |
masoprocol | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
5-(n-methyl-n-isobutyl)amiloride | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
sk&f 95282 | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
zpck | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
gr 127935 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
benzamil | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
3',4'-dichlorobenzamil | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
1-(2-(4-aminophenyl)ethyl)-4-(3-trifluoromethylphenyl)piperazine | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
1-(1-(2-benzo(b)thienyl)cyclohexyl)piperidine | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
indatraline | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
sr 2640 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
n-(2-chloroethyl)-4-piperidinyl diphenylacetate | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
n,n-di-n-hexyl-2-(4-fluorophenyl)indole-3-acetamide | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
3,5-bis(trifluoromethyl)benzyl n-acetyltryptophan | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
l 741626 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
corbadrine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
esatenolol | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
sb 216763 | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
ketoprofen | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
dexefaroxan | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
nsc 95397 | Homo sapiens (human) | Potency | 1.2589 | 2 | 0 |
tosylphenylalanyl chloromethyl ketone | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
hydrastine hydrochloride, (s-(r*,s*))-isomer | Homo sapiens (human) | Potency | 6.3096 | 2 | 0 |
sb 228357 | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
6-bromoindirubin-3'-oxime | Homo sapiens (human) | Potency | 0.2512 | 2 | 0 |
ketoconazole | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
gw9662 | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
sch-202676 | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
4-bromotetramisole, (s)-isomer | Homo sapiens (human) | Potency | 25.1189 | 2 | 0 |
dexchlorpheniramine | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
phenylthiazolylthiourea | Homo sapiens (human) | Potency | 19.9526 | 2 | 0 |
cis-resveratrol | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
fluoxetine | Homo sapiens (human) | Potency | 14.1806 | 2 | 0 |
tg 003 | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
capsazepine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
tamoxifen citrate | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
6-methyl-2-(phenylethynyl)pyridine | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
thioperamide | Homo sapiens (human) | Potency | 3.9811 | 2 | 0 |
bp 897 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
sb 203186 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
n-(1-methyl-5-indolyl)-n'-(3-methyl-5-isothiazolyl)urea | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
sb-224289 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
pd 168,077 | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
sb 415286 | Homo sapiens (human) | Potency | 0.1995 | 2 | 0 |
LY-310762 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
sc 560 | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
sc-19220 | Homo sapiens (human) | Potency | 6.3096 | 2 | 0 |
ly 367265 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazole | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
sib 1757 | Homo sapiens (human) | Potency | 0.0794 | 2 | 0 |
apigenin | Homo sapiens (human) | Potency | 0.5012 | 2 | 0 |
daphnetin | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
genistein | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
pulmicort | Homo sapiens (human) | Potency | 0.0100 | 2 | 0 |
morin | Homo sapiens (human) | Potency | 3.1623 | 2 | 0 |
myricetin | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
daidzein | Homo sapiens (human) | Potency | 2.5119 | 2 | 0 |
n-oleoyldopamine | Homo sapiens (human) | Potency | 0.5012 | 2 | 0 |
tranilast | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
fenretinide | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
ic 261 | Homo sapiens (human) | Potency | 7.9433 | 2 | 0 |
su 9516 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acid | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
k 185 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
casein kinase ii | Homo sapiens (human) | Potency | 1.2589 | 2 | 0 |
ag 538 | Homo sapiens (human) | Potency | 31.6228 | 2 | 0 |
tyrphostin ag 555 | Homo sapiens (human) | Potency | 1.5849 | 2 | 0 |
tyrphostin b44 | Homo sapiens (human) | Potency | 6.3096 | 2 | 0 |
ag-490 | Homo sapiens (human) | Potency | 1.0000 | 2 | 0 |
cisplatin | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
a 77636 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
b 43 | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
(8R)-7-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triol | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
(8R)-7-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,13,14-triol | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
dilazep(2+) | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
dihydrexidine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
erythro-dihydrosphingosine | Homo sapiens (human) | Potency | 12.5893 | 2 | 0 |
gw2974 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
(2S)-1-(1H-imidazol-5-yl)-2-propanamine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
l 750667 | Homo sapiens (human) | Potency | 1.9953 | 2 | 0 |
l 162313 | Homo sapiens (human) | Potency | 5.0119 | 2 | 0 |
s-nitroso-n-acetylpenicillamine | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |
pd 404182 | Homo sapiens (human) | Potency | 15.8489 | 2 | 0 |
ag-879 | Homo sapiens (human) | Potency | 10.0000 | 2 | 0 |