Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
pomiferin | Mus musculus (house mouse) | AC50 | 0.8090 | 1 | 0 |
sirodesmin a | Mus musculus (house mouse) | AC50 | 5.6110 | 1 | 0 |
2-[cyclohexyl-[2-[5-(3,4-dimethoxyphenyl)-2-tetrazolyl]-1-oxoethyl]amino]-N-cyclopentylpropanamide | Mus musculus (house mouse) | AbsAC40_uM | 0.4370 | 1 | 0 |
2-[cyclohexyl-[2-[5-(3,4-dimethoxyphenyl)-2-tetrazolyl]-1-oxoethyl]amino]-N-cyclopentylpropanamide | Mus musculus (house mouse) | AC50 | 87.6399 | 4 | 0 |
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrile | Mus musculus (house mouse) | AC50 | 11.2270 | 2 | 0 |
2-[(7-ethyl-[1,3]dioxolo[4,5-g]quinolin-6-yl)thio]acetic acid propan-2-yl ester | Mus musculus (house mouse) | AC50 | 0.9230 | 2 | 0 |
N-[3-[[(3,5-dimethoxyphenyl)-oxomethyl]amino]phenyl]carbamic acid ethyl ester | Mus musculus (house mouse) | AC50 | 176.1350 | 2 | 0 |
2-[[5-[(2,6-dimethylphenoxy)methyl]-4-ethyl-1,2,4-triazol-3-yl]thio]-1-(4-phenyl-1-piperazinyl)ethanone | Mus musculus (house mouse) | AC50 | 14.4650 | 2 | 0 |
2-chloro-N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-5-(1,2,4-triazol-4-yl)benzamide | Mus musculus (house mouse) | AbsAC40_uM | 80.0000 | 1 | 0 |
2-chloro-N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-5-(1,2,4-triazol-4-yl)benzamide | Mus musculus (house mouse) | AC50 | 16.1167 | 6 | 0 |
2-(3,4-dimethoxyphenyl)-8-methoxy-4,4-dimethyl-5H-isothiazolo[5,4-c]quinoline-1-thione | Mus musculus (house mouse) | AC50 | 3.0800 | 1 | 0 |
1-[1-naphthalenyl(oxo)methyl]-3-indolecarboxylic acid methyl ester | Mus musculus (house mouse) | AC50 | 24.0290 | 2 | 0 |
1-(3-fluorophenyl)-4-(4-hydroxy-3-methoxy-5-nitrophenyl)-4H-pyridine-3,5-dicarboxylic acid diethyl ester | Mus musculus (house mouse) | AC50 | 7.7200 | 1 | 0 |
N-tert-butyl-4-[3-(trifluoromethyl)-2-pyridinyl]-1-piperazinecarboxamide | Mus musculus (house mouse) | AC50 | 7.6100 | 1 | 0 |
3-(methanesulfonamido)benzoic acid [1-[4-(4-morpholinyl)anilino]-1-oxopropan-2-yl] ester | Mus musculus (house mouse) | AC50 | 3.0160 | 2 | 0 |
4-(6-bromo-1,3-benzodioxol-5-yl)-7,9-dimethyl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline | Mus musculus (house mouse) | AC50 | 13.6270 | 2 | 0 |
4-[3-(2-furanylmethyl)-4-oxo-2-thiazolidinyl]-N-(3-propan-2-yloxypropyl)benzamide | Mus musculus (house mouse) | AC50 | 8.7320 | 2 | 0 |
N-(3-chlorophenyl)-4-[4-(3-methoxyphenyl)-2-thiazolyl]-1-piperazinecarbothioamide | Mus musculus (house mouse) | AC50 | 12.0200 | 1 | 0 |
1-(2-methylphenyl)-3-[[1-[4-(4-morpholinylsulfonyl)phenyl]-4-piperidinyl]methyl]urea | Mus musculus (house mouse) | AC50 | 88.6580 | 3 | 0 |
2-[4-[2-(3,5-dimethoxyanilino)-2-oxoethyl]-1-piperazinyl]-N-(4-ethoxyphenyl)acetamide | Mus musculus (house mouse) | AC50 | 68.8813 | 3 | 0 |
N-(3,5-dichloro-2-pyridinyl)-2-[(4-methyl-2-quinolinyl)thio]propanamide | Mus musculus (house mouse) | AC50 | 3.7365 | 2 | 0 |
6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylic acid [1-[1-[4-(difluoromethoxy)phenyl]-2,5-dimethyl-3-pyrrolyl]-1-oxopropan-2-yl] ester | Mus musculus (house mouse) | AC50 | 107.6840 | 4 | 0 |
ly 367265 | Mus musculus (house mouse) | AC50 | 87.8300 | 1 | 0 |
LSM-4844 | Mus musculus (house mouse) | AC50 | 0.5380 | 2 | 0 |
cyclosporine | Mus musculus (house mouse) | AbsAC40_uM | 35.0000 | 1 | 0 |
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazine | Mus musculus (house mouse) | AC50 | 72.7977 | 3 | 0 |
N3,N6-bis(2,5-dimethoxyphenyl)pyridazine-3,6-diamine | Mus musculus (house mouse) | AC50 | 12.4205 | 2 | 0 |
4-[[[4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazin-6-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl ester | Mus musculus (house mouse) | AC50 | 2.4000 | 1 | 0 |
N-[3-[2-(4-chloroanilino)-4-thiazolyl]phenyl]-3-(trifluoromethyl)benzamide | Mus musculus (house mouse) | AC50 | 2.1000 | 1 | 0 |
3-(trifluoromethyl)-N-[4-[2-[3-(trifluoromethyl)anilino]-4-thiazolyl]phenyl]benzamide | Mus musculus (house mouse) | AC50 | 0.4350 | 1 | 0 |
N-[2-(2,5-dimethoxyphenyl)ethyl]-4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazine-6-carboxamide | Mus musculus (house mouse) | AC50 | 4.1080 | 2 | 0 |
N-[4-[1-(1-oxopropyl)-2,3-dihydroindol-5-yl]-2-thiazolyl]-2-furancarboxamide | Mus musculus (house mouse) | AbsAC40_uM | 1.2910 | 1 | 0 |
N-[4-[1-(1-oxopropyl)-2,3-dihydroindol-5-yl]-2-thiazolyl]-2-furancarboxamide | Mus musculus (house mouse) | AC50 | 0.2070 | 5 | 0 |
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2-(3,5-dimethyl-1-pyrazolyl)acetamide | Mus musculus (house mouse) | AC50 | 0.4342 | 2 | 0 |
(5R)-3-(4-dibenzothiophenyl)-5-(3,4-dimethoxyphenyl)-1-cyclohex-2-enone | Mus musculus (house mouse) | AC50 | 2.2800 | 1 | 0 |
1-[(2S,3S)-2-[[benzenesulfonyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-[4-(trifluoromethyl)phenyl]urea | Mus musculus (house mouse) | AbsAC40_uM | 34.6000 | 1 | 0 |
N-[(2R,3R)-2-[[(4-fluorophenyl)sulfonyl-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-2-(1-methyl-3-indolyl)acetamide | Mus musculus (house mouse) | AC50 | 1.0573 | 3 | 0 |