Proteins > Peptidylglycine alpha-amidating monooxygenase
Page last updated: 2024-08-07 15:59:47
Peptidylglycine alpha-amidating monooxygenase
A peptidyl-glycine alpha-amidating monooxygenase that is encoded in the genome of rat. [OMA:P14925, PRO:DNx]
Synonyms
PAM
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (24)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
cyclosporine | Rattus norvegicus (Norway rat) | Ki | 0.0060 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
p-aminohippuric acid | Rattus norvegicus (Norway rat) | Km | 2,600.0000 | 1 | 1 |
iodohippuric acid | Rattus norvegicus (Norway rat) | Km | 3,400.0000 | 1 | 1 |
salicylurate | Rattus norvegicus (Norway rat) | Km | 860.0000 | 1 | 1 |
aceturic acid | Rattus norvegicus (Norway rat) | Km | 9,300.0000 | 1 | 1 |
n-benzyloxycarbonylglycine | Rattus norvegicus (Norway rat) | Km | 590.0000 | 1 | 1 |
4-nitrohippuric acid | Rattus norvegicus (Norway rat) | Km | 470.0000 | 1 | 1 |
furoylglycine | Rattus norvegicus (Norway rat) | Km | 2,700.0000 | 1 | 1 |
4-chlorohippuric acid | Rattus norvegicus (Norway rat) | Km | 620.0000 | 1 | 1 |
thiophenoxyacetic acid | Rattus norvegicus (Norway rat) | Kis | 380.0000 | 1 | 1 |
salicylhydroxamic acid | Rattus norvegicus (Norway rat) | Kis | 300.0000 | 1 | 1 |
phenylacetylglycine | Rattus norvegicus (Norway rat) | Km | 160.0000 | 1 | 1 |
nicotinuric acid | Rattus norvegicus (Norway rat) | Km | 1,900.0000 | 1 | 1 |
benzoylpropionic acid | Rattus norvegicus (Norway rat) | Kis | 2,900.0000 | 1 | 1 |
boc-glycine | Rattus norvegicus (Norway rat) | Km | 3,700.0000 | 1 | 1 |
n-benzylglycine | Rattus norvegicus (Norway rat) | Kis | 18,000.0000 | 1 | 1 |
2-methylhippuric acid | Rattus norvegicus (Norway rat) | Km | 4,300.0000 | 1 | 1 |
hippuryl-glycyl-glycine | Rattus norvegicus (Norway rat) | Km | 310.0000 | 1 | 1 |
4-methylhippuric acid | Rattus norvegicus (Norway rat) | Km | 1,800.0000 | 1 | 1 |
3-methylhippuric acid | Rattus norvegicus (Norway rat) | Km | 1,400.0000 | 1 | 1 |
4-methyoxybenzoyl-n-glycine | Rattus norvegicus (Norway rat) | Km | 820.0000 | 1 | 1 |
4-hydroxyhippuric acid | Rattus norvegicus (Norway rat) | Km | 1,700.0000 | 1 | 1 |
cinnamoylglycine | Rattus norvegicus (Norway rat) | Km | 230.0000 | 1 | 1 |
2-aminohippuric acid | Rattus norvegicus (Norway rat) | Km | 1,400.0000 | 1 | 1 |