Page last updated: 2024-08-07 15:59:47

Peptidylglycine alpha-amidating monooxygenase

A peptidyl-glycine alpha-amidating monooxygenase that is encoded in the genome of rat. [OMA:P14925, PRO:DNx]

Synonyms

PAM

Research

Bioassay Publications (2)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (24)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
cyclosporineRattus norvegicus (Norway rat)Ki0.006011

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
p-aminohippuric acidRattus norvegicus (Norway rat)Km2,600.000011
iodohippuric acidRattus norvegicus (Norway rat)Km3,400.000011
salicylurateRattus norvegicus (Norway rat)Km860.000011
aceturic acidRattus norvegicus (Norway rat)Km9,300.000011
n-benzyloxycarbonylglycineRattus norvegicus (Norway rat)Km590.000011
4-nitrohippuric acidRattus norvegicus (Norway rat)Km470.000011
furoylglycineRattus norvegicus (Norway rat)Km2,700.000011
4-chlorohippuric acidRattus norvegicus (Norway rat)Km620.000011
thiophenoxyacetic acidRattus norvegicus (Norway rat)Kis380.000011
salicylhydroxamic acidRattus norvegicus (Norway rat)Kis300.000011
phenylacetylglycineRattus norvegicus (Norway rat)Km160.000011
nicotinuric acidRattus norvegicus (Norway rat)Km1,900.000011
benzoylpropionic acidRattus norvegicus (Norway rat)Kis2,900.000011
boc-glycineRattus norvegicus (Norway rat)Km3,700.000011
n-benzylglycineRattus norvegicus (Norway rat)Kis18,000.000011
2-methylhippuric acidRattus norvegicus (Norway rat)Km4,300.000011
hippuryl-glycyl-glycineRattus norvegicus (Norway rat)Km310.000011
4-methylhippuric acidRattus norvegicus (Norway rat)Km1,800.000011
3-methylhippuric acidRattus norvegicus (Norway rat)Km1,400.000011
4-methyoxybenzoyl-n-glycineRattus norvegicus (Norway rat)Km820.000011
4-hydroxyhippuric acidRattus norvegicus (Norway rat)Km1,700.000011
cinnamoylglycineRattus norvegicus (Norway rat)Km230.000011
2-aminohippuric acidRattus norvegicus (Norway rat)Km1,400.000011