Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
citric acid, anhydrous | Homo sapiens (human) | IC50 | 4.5885 | 2 | 0 |
benzbromarone | Homo sapiens (human) | IC50 | 18.8080 | 1 | 0 |
disulfiram | Homo sapiens (human) | IC50 | 1.6220 | 1 | 0 |
ebselen | Homo sapiens (human) | IC50 | 1.1010 | 1 | 0 |
ethacrynic acid | Homo sapiens (human) | IC50 | 4.8320 | 1 | 0 |
amrinone | Homo sapiens (human) | IC50 | 78.8160 | 1 | 0 |
ketotifen | Homo sapiens (human) | IC50 | 39.8410 | 2 | 0 |
vitamin k 3 | Homo sapiens (human) | IC50 | 9.4680 | 1 | 0 |
nifedipine | Homo sapiens (human) | IC50 | 7.1330 | 1 | 0 |
9,10-phenanthrenequinone | Homo sapiens (human) | IC50 | 6.4430 | 1 | 0 |
phosmet | Homo sapiens (human) | IC50 | 11.9110 | 1 | 0 |
alverine citrate | Homo sapiens (human) | IC50 | 2.6350 | 2 | 0 |
sufentanil citrate | Homo sapiens (human) | IC50 | 2.6340 | 2 | 0 |
carbetapentane citrate | Homo sapiens (human) | IC50 | 1.6103 | 4 | 0 |
butethamate citrate | Homo sapiens (human) | IC50 | 2.6075 | 2 | 0 |
mosapride | Homo sapiens (human) | IC50 | 2.2130 | 2 | 0 |
mosapride | Homo sapiens (human) | IC50 | 1.3150 | 2 | 0 |
1,5-bis(2-methoxyphenyl)penta-1,4-dien-3-one | Homo sapiens (human) | IC50 | 5.7115 | 2 | 0 |
tosylphenylalanyl chloromethyl ketone | Homo sapiens (human) | IC50 | 1.9010 | 1 | 0 |
[(1S,2R,3S,4S,6R,7R,8R)-4-ethenyl-3-hydroxy-2,4,7,14-tetramethyl-9-oxo-6-tricyclo[5.4.3.01,8]tetradecanyl] 2-[2-(diethylamino)ethylsulfanyl]acetate | Homo sapiens (human) | IC50 | 6.2360 | 2 | 0 |
chalcone | Homo sapiens (human) | IC50 | 4.2450 | 1 | 0 |
dibenzylidene acetone | Homo sapiens (human) | IC50 | 1.4840 | 1 | 0 |
curcumin | Homo sapiens (human) | IC50 | 10.2320 | 1 | 0 |
mecysteine hydrochloride | Homo sapiens (human) | IC50 | 4.6410 | 1 | 0 |
toremifene citrate | Homo sapiens (human) | IC50 | 1.2915 | 2 | 0 |
zuclomifene citrate | Homo sapiens (human) | IC50 | 2.4255 | 2 | 0 |
ketotifen fumarate | Homo sapiens (human) | IC50 | 8.8080 | 2 | 0 |
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-N-(3-methylphenyl)acetamide | Homo sapiens (human) | IC50 | 2.6505 | 2 | 0 |
enclomiphene citrate | Homo sapiens (human) | IC50 | 1.2165 | 2 | 0 |
dibenzheptropine citrate | Homo sapiens (human) | IC50 | 2.4345 | 2 | 0 |
chlorhexidine | Homo sapiens (human) | IC50 | 4.0045 | 4 | 0 |
tiamulin fumarate (1:1), (3as-(3aalpha,4beta,5alpha,6alpha,8beta,9alpha,9abeta,10s*))-isomer | Homo sapiens (human) | IC50 | 6.3260 | 2 | 0 |
chlorhexidine hydrochloride | Homo sapiens (human) | IC50 | 4.9115 | 2 | 0 |
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 14.3458 | 4 | 0 |
1-butyl-3-(5-methyl-6-oxo-3-benzo[b][1,4]benzothiazepinyl)urea | Homo sapiens (human) | IC50 | 6.6856 | 5 | 0 |
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 4.6620 | 2 | 0 |
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 3.0700 | 2 | 0 |