Page last updated: 2024-08-07 12:35:43

prostaglandin E2 receptor EP2 subtype

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (19)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
bardoxolone methylHomo sapiens (human)Potency16.626110
3-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineHomo sapiens (human)Potency1.905020
[1-(3-methylphenyl)-5-benzimidazolyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency0.543320
2-[[(6-bromo-1H-imidazo[4,5-b]pyridin-2-yl)thio]methyl]benzonitrileHomo sapiens (human)Potency28.300920
dinoprostoneHomo sapiens (human)Potency0.148210
15-deoxy-delta(12,14)-prostaglandin j2Homo sapiens (human)Potency41.762910

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
pk 11195Homo sapiens (human)Active Concentration20.000010
celecoxibHomo sapiens (human)Active Concentration20.000010
chlorpyrifosHomo sapiens (human)Active Concentration20.000010
nitroarginineHomo sapiens (human)Active Concentration20.000010
2-[[2-furanyl(oxo)methyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid ethyl esterHomo sapiens (human)Active Concentration20.000010
2-[[oxo(thiophen-2-yl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid propan-2-yl esterHomo sapiens (human)Active Concentration20.000010
5-ethyl-2-[[oxo-(3,4,5-trimethoxyphenyl)methyl]amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Active Concentration20.000010
2,2-diphenylacetic acid (2,6-dimethylphenyl) esterHomo sapiens (human)Active Concentration20.000010
5-bromo-N-(2-phenylphenyl)-2-furancarboxamideHomo sapiens (human)Active Concentration20.000010
4-(3,4-dimethoxyphenyl)-2-(1-piperidinyl)-6-(trifluoromethyl)pyrimidineHomo sapiens (human)Active Concentration20.000010
4-(1-phenylethyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Active Concentration20.000010
5-methoxy-3,6-diphenyl-1,2,4-triazineHomo sapiens (human)Active Concentration20.000010
LSM-34734Homo sapiens (human)Active Concentration20.000010