Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
8-hydroxy-2-(di-n-propylamino)tetralin | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
ethylisopropylamiloride | Homo sapiens (human) | EC50 | 51.0195 | 2 | 0 |
tacrine | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
cgp 20712a | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
adtn | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
methergine | Homo sapiens (human) | EC50 | 92.4890 | 1 | 0 |
riluzole | Homo sapiens (human) | EC50 | 92.6270 | 1 | 0 |
suprofen | Homo sapiens (human) | EC50 | 92.5900 | 1 | 0 |
talipexole | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
racepinephrine hydrochloride | Homo sapiens (human) | EC50 | 92.5900 | 1 | 0 |
adrenalone | Homo sapiens (human) | EC50 | 92.3520 | 1 | 0 |
benzethonium chloride | Homo sapiens (human) | EC50 | 92.4610 | 1 | 0 |
lysergol | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
cetylpyridinium chloride | Homo sapiens (human) | EC50 | 92.4850 | 1 | 0 |
dobutamine | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
pergolide | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
pergolide mesylate | Homo sapiens (human) | EC50 | 92.4800 | 1 | 0 |
fenoldopam mesylate | Homo sapiens (human) | EC50 | 92.4800 | 1 | 0 |
quinpirole hydrochloride | Homo sapiens (human) | EC50 | 92.5810 | 1 | 0 |
aripiprazole | Homo sapiens (human) | EC50 | 92.4690 | 1 | 0 |
alfentanil hydrochloride | Homo sapiens (human) | EC50 | 0.4567 | 2 | 0 |
dobutamine hydrochloride | Homo sapiens (human) | EC50 | 92.5350 | 1 | 0 |
9-methoxyellipticine | Homo sapiens (human) | EC50 | 64.6640 | 1 | 0 |
ici 204448 | Homo sapiens (human) | EC50 | 53.9100 | 2 | 0 |
Serotonin hydrochloride | Homo sapiens (human) | EC50 | 92.3940 | 1 | 0 |
sk&f 75670 | Homo sapiens (human) | EC50 | 92.4520 | 1 | 0 |
piribedil mesylate | Homo sapiens (human) | EC50 | 92.4540 | 1 | 0 |
preclamol | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
chondocurine (1beta)-(+-)-isomer | Homo sapiens (human) | EC50 | 51.3280 | 2 | 0 |
n-methylserotonin oxalate salt | Homo sapiens (human) | EC50 | 92.4070 | 1 | 0 |
dironyl | Homo sapiens (human) | EC50 | 92.5070 | 1 | 0 |
dihydroergocristine monomesylate | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
calmidazolium | Homo sapiens (human) | EC50 | 47.9575 | 2 | 0 |
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanone | Homo sapiens (human) | EC50 | 64.5580 | 1 | 0 |
4-(3,4-dihydro-2H-quinolin-1-yl)-6-[(4-phenyl-1-piperazinyl)methyl]-1,3,5-triazin-2-amine | Homo sapiens (human) | EC50 | 92.4540 | 1 | 0 |
2-[4-[(3-fluorophenyl)methyl]-1-piperazinyl]pyrimidine | Homo sapiens (human) | EC50 | 92.4695 | 2 | 0 |
N-[5-(1,3-benzothiazol-2-yl)-2-chlorophenyl]-1,3-benzodioxole-5-carboxamide | Homo sapiens (human) | EC50 | 92.4500 | 1 | 0 |
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamide | Homo sapiens (human) | EC50 | 64.5720 | 1 | 0 |
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamine | Homo sapiens (human) | EC50 | 54.4430 | 2 | 0 |
N-[(3-benzamidoanilino)-sulfanylidenemethyl]-2-thiophenecarboxamide | Homo sapiens (human) | EC50 | 92.4730 | 1 | 0 |
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamide | Homo sapiens (human) | EC50 | 50.0220 | 1 | 0 |
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | Homo sapiens (human) | EC50 | 92.4980 | 2 | 0 |
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl ester | Homo sapiens (human) | EC50 | 92.4710 | 1 | 0 |
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thiourea | Homo sapiens (human) | EC50 | 2.5080 | 2 | 0 |
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamide | Homo sapiens (human) | EC50 | 92.4980 | 1 | 0 |
9,10-dihydrolysergol | Homo sapiens (human) | EC50 | 92.5260 | 1 | 0 |
n-oleoyldopamine | Homo sapiens (human) | EC50 | 92.3420 | 1 | 0 |
2-bromoergocryptine mesylate | Homo sapiens (human) | EC50 | 92.4520 | 1 | 0 |
phenylephrine hydrochloride | Homo sapiens (human) | EC50 | 92.4310 | 1 | 0 |
ethisterone | Homo sapiens (human) | EC50 | 92.6000 | 1 | 0 |
trimebutine maleate salt | Homo sapiens (human) | EC50 | 51.1495 | 2 | 0 |
hydrocotarnine hydrobromide | Homo sapiens (human) | EC50 | 92.4240 | 1 | 0 |
dihydroergotoxine | Homo sapiens (human) | EC50 | 92.4530 | 1 | 0 |
a 77636 | Homo sapiens (human) | EC50 | 92.4700 | 1 | 0 |
epinephrine bitartrate | Homo sapiens (human) | EC50 | 92.5070 | 1 | 0 |
8-hydroxy-2-(di-n-propylamino)tetralin hydrobromide | Homo sapiens (human) | EC50 | 92.5350 | 1 | 0 |
phencyclidine hydrochloride | Homo sapiens (human) | EC50 | 3.6255 | 2 | 0 |
a 77636 | Homo sapiens (human) | EC50 | 92.3760 | 1 | 0 |
cgp 20712a | Homo sapiens (human) | EC50 | 92.3860 | 1 | 0 |
dihydroxanthohumol | Homo sapiens (human) | EC50 | 64.5840 | 1 | 0 |
6-fluoronorepinephrine monohydrochloride, (+-)-isomer | Homo sapiens (human) | EC50 | 92.5540 | 1 | 0 |
adtn | Homo sapiens (human) | EC50 | 92.5440 | 1 | 0 |
2-hydroxyapomorphine, (r)-isomer | Homo sapiens (human) | EC50 | 92.3950 | 1 | 0 |
7-hydroxy-2-n,n-dipropylaminotetralin hydrobromide | Homo sapiens (human) | EC50 | 92.4470 | 1 | 0 |
2-(n-phenethyl-n-propyl)amino-5-hydroxytetralin hydrochloride | Homo sapiens (human) | EC50 | 92.6180 | 1 | 0 |
sk&f 77434 | Homo sapiens (human) | EC50 | 92.4680 | 1 | 0 |
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanol | Homo sapiens (human) | EC50 | 92.4810 | 1 | 0 |
[1-(2-benzofuranylmethyl)-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanol | Homo sapiens (human) | EC50 | 92.4795 | 2 | 0 |
cym51010 | Homo sapiens (human) | EC50 | 9.9552 | 4 | 0 |
norepinephrine bitartrate | Homo sapiens (human) | EC50 | 92.4680 | 1 | 0 |
demeclocycline hydrochloride | Homo sapiens (human) | EC50 | 92.4510 | 1 | 0 |