Page last updated: 2024-08-07 15:15:37

mu-type opioid receptor isoform MOR-1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (71)

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
8-hydroxy-2-(di-n-propylamino)tetralinHomo sapiens (human)EC5092.470010
ethylisopropylamilorideHomo sapiens (human)EC5051.019520
tacrineHomo sapiens (human)EC5092.470010
cgp 20712aHomo sapiens (human)EC5092.470010
adtnHomo sapiens (human)EC5092.470010
methergineHomo sapiens (human)EC5092.489010
riluzoleHomo sapiens (human)EC5092.627010
suprofenHomo sapiens (human)EC5092.590010
talipexoleHomo sapiens (human)EC5092.470010
racepinephrine hydrochlorideHomo sapiens (human)EC5092.590010
adrenaloneHomo sapiens (human)EC5092.352010
benzethonium chlorideHomo sapiens (human)EC5092.461010
lysergolHomo sapiens (human)EC5092.470010
cetylpyridinium chlorideHomo sapiens (human)EC5092.485010
dobutamineHomo sapiens (human)EC5092.470010
pergolideHomo sapiens (human)EC5092.470010
pergolide mesylateHomo sapiens (human)EC5092.480010
fenoldopam mesylateHomo sapiens (human)EC5092.480010
quinpirole hydrochlorideHomo sapiens (human)EC5092.581010
aripiprazoleHomo sapiens (human)EC5092.469010
alfentanil hydrochlorideHomo sapiens (human)EC500.456720
dobutamine hydrochlorideHomo sapiens (human)EC5092.535010
9-methoxyellipticineHomo sapiens (human)EC5064.664010
ici 204448Homo sapiens (human)EC5053.910020
Serotonin hydrochlorideHomo sapiens (human)EC5092.394010
sk&f 75670Homo sapiens (human)EC5092.452010
piribedil mesylateHomo sapiens (human)EC5092.454010
preclamolHomo sapiens (human)EC5092.470010
chondocurine (1beta)-(+-)-isomerHomo sapiens (human)EC5051.328020
n-methylserotonin oxalate saltHomo sapiens (human)EC5092.407010
dironylHomo sapiens (human)EC5092.507010
dihydroergocristine monomesylateHomo sapiens (human)EC5092.470010
calmidazoliumHomo sapiens (human)EC5047.957520
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)EC5064.558010
4-(3,4-dihydro-2H-quinolin-1-yl)-6-[(4-phenyl-1-piperazinyl)methyl]-1,3,5-triazin-2-amineHomo sapiens (human)EC5092.454010
2-[4-[(3-fluorophenyl)methyl]-1-piperazinyl]pyrimidineHomo sapiens (human)EC5092.469520
N-[5-(1,3-benzothiazol-2-yl)-2-chlorophenyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)EC5092.450010
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamideHomo sapiens (human)EC5064.572010
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamineHomo sapiens (human)EC5054.443020
N-[(3-benzamidoanilino)-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)EC5092.473010
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideHomo sapiens (human)EC5050.022010
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)EC5092.498020
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterHomo sapiens (human)EC5092.471010
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thioureaHomo sapiens (human)EC502.508020
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideHomo sapiens (human)EC5092.498010
9,10-dihydrolysergolHomo sapiens (human)EC5092.526010
n-oleoyldopamineHomo sapiens (human)EC5092.342010
2-bromoergocryptine mesylateHomo sapiens (human)EC5092.452010
phenylephrine hydrochlorideHomo sapiens (human)EC5092.431010
ethisteroneHomo sapiens (human)EC5092.600010
trimebutine maleate saltHomo sapiens (human)EC5051.149520
hydrocotarnine hydrobromideHomo sapiens (human)EC5092.424010
dihydroergotoxineHomo sapiens (human)EC5092.453010
a 77636Homo sapiens (human)EC5092.470010
epinephrine bitartrateHomo sapiens (human)EC5092.507010
8-hydroxy-2-(di-n-propylamino)tetralin hydrobromideHomo sapiens (human)EC5092.535010
phencyclidine hydrochlorideHomo sapiens (human)EC503.625520
a 77636Homo sapiens (human)EC5092.376010
cgp 20712aHomo sapiens (human)EC5092.386010
dihydroxanthohumolHomo sapiens (human)EC5064.584010
6-fluoronorepinephrine monohydrochloride, (+-)-isomerHomo sapiens (human)EC5092.554010
adtnHomo sapiens (human)EC5092.544010
2-hydroxyapomorphine, (r)-isomerHomo sapiens (human)EC5092.395010
7-hydroxy-2-n,n-dipropylaminotetralin hydrobromideHomo sapiens (human)EC5092.447010
2-(n-phenethyl-n-propyl)amino-5-hydroxytetralin hydrochlorideHomo sapiens (human)EC5092.618010
sk&f 77434Homo sapiens (human)EC5092.468010
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)EC5092.481010
[1-(2-benzofuranylmethyl)-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolHomo sapiens (human)EC5092.479520
cym51010Homo sapiens (human)EC509.955240
norepinephrine bitartrateHomo sapiens (human)EC5092.468010
demeclocycline hydrochlorideHomo sapiens (human)EC5092.451010