Page last updated: 2024-08-07 21:31:07
Histone deacetylase
[no definition available]
Synonyms
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 2 (66.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
entinostat | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.9400 | 1 | 1 |
fenofibrate | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 10.0000 | 1 | 1 |
vorinostat | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.0945 | 2 | 2 |
trichostatin a | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.0006 | 1 | 1 |
(3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.0010 | 1 | 1 |
belinostat | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.2147 | 1 | 1 |
panobinostat | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.0026 | 2 | 2 |