Page last updated: 2024-08-07 12:38:34

nuclear receptor ROR-gamma isoform 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (3856)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
9-xylosyladenineMus musculus (house mouse)Potency13.357410
chlordeconeMus musculus (house mouse)Potency27.005010
gallic acidMus musculus (house mouse)Potency13.891420
4-aminophenolMus musculus (house mouse)Potency17.782810
hydroquinoneMus musculus (house mouse)Potency19.468620
arabitolMus musculus (house mouse)Potency6.309610
kynurenineMus musculus (house mouse)Potency19.950620
thioctic acidMus musculus (house mouse)Potency17.782810
naringeninMus musculus (house mouse)Potency25.665110
pentachlorophenolMus musculus (house mouse)Potency22.259620
b 844-39Mus musculus (house mouse)Potency35.481320
1,10-phenanthrolineMus musculus (house mouse)Potency17.331120
1,3-dipropyl-8-cyclopentylxanthineMus musculus (house mouse)Potency35.481310
pd 173074Mus musculus (house mouse)Potency35.481310
hoe 33342Mus musculus (house mouse)Potency7.414020
2,4-dinitrophenolMus musculus (house mouse)Potency24.087420
2-aminoethoxydiphenyl borateMus musculus (house mouse)Potency21.818520
3-[(4-chlorophenyl)-phenylmethoxy]-8-methyl-8-azabicyclo[3.2.1]octaneMus musculus (house mouse)Potency11.904820
chlorocresolMus musculus (house mouse)Potency31.622810
phenytoinMus musculus (house mouse)Potency6.309610
5-(nonyloxy)tryptamineMus musculus (house mouse)Potency21.154620
2-(4-amino-5-iodo-7-pyrrolo[2,3-d]pyrimidinyl)-5-(hydroxymethyl)oxolane-3,4-diolMus musculus (house mouse)Potency4.802220
7,8-dihydroxyflavoneMus musculus (house mouse)Potency22.740620
7-nitroindazoleMus musculus (house mouse)Potency17.782810
oxyquinolineMus musculus (house mouse)Potency2.061020
tacrineMus musculus (house mouse)Potency28.183810
ro 48-8071Mus musculus (house mouse)Potency35.481310
acridoneMus musculus (house mouse)Potency11.557420
ag 127Mus musculus (house mouse)Potency24.035320
ag 1295Mus musculus (house mouse)Potency33.552020
tyrphostin a23Mus musculus (house mouse)Potency18.364420
tyrphostin 25Mus musculus (house mouse)Potency22.387210
methylglucosideMus musculus (house mouse)Potency0.707910
alprazolamMus musculus (house mouse)Potency2.253610
amiodaroneMus musculus (house mouse)Potency35.481310
amlexanoxMus musculus (house mouse)Potency7.308120
amlodipineMus musculus (house mouse)Potency12.589310
anethole trithioneMus musculus (house mouse)Potency11.220210
6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diolMus musculus (house mouse)Potency15.848910
aristolochic acid iMus musculus (house mouse)Potency14.721410
astemizoleMus musculus (house mouse)Potency21.997420
atrazineMus musculus (house mouse)Potency15.848910
azinphosmethylMus musculus (house mouse)Potency35.481310
benzethoniumMus musculus (house mouse)Potency9.053220
benzocaineMus musculus (house mouse)Potency7.079510
benzyl isothiocyanateMus musculus (house mouse)Potency14.005320
butylbenzyl phthalateMus musculus (house mouse)Potency22.387210
bicalutamideMus musculus (house mouse)Potency31.622810
bifemelaneMus musculus (house mouse)Potency35.481310
bay h 4502Mus musculus (house mouse)Potency14.484220
bithionolMus musculus (house mouse)Potency24.911520
bml 190Mus musculus (house mouse)Potency28.183810
bronopolMus musculus (house mouse)Potency35.481310
broxyquinolineMus musculus (house mouse)Potency0.281810
butambenMus musculus (house mouse)Potency11.220220
caffeineMus musculus (house mouse)Potency15.848910
calmidazoliumMus musculus (house mouse)Potency7.191220
candesartan cilexetilMus musculus (house mouse)Potency24.702820
cantharidinMus musculus (house mouse)Potency11.220210
carmustineMus musculus (house mouse)Potency31.622810
carvedilolMus musculus (house mouse)Potency10.899320
carbonyl cyanide m-chlorophenyl hydrazoneMus musculus (house mouse)Potency0.876520
cgs 15943Mus musculus (house mouse)Potency4.287110
chelerythrineMus musculus (house mouse)Potency6.657720
chloroxineMus musculus (house mouse)Potency746.360420
chlorprophamMus musculus (house mouse)Potency11.220210
ciglitazoneMus musculus (house mouse)Potency24.035320
cilostazolMus musculus (house mouse)Potency9.270620
clemizoleMus musculus (house mouse)Potency12.589310
clioquinolMus musculus (house mouse)Potency0.629420
clofoctolMus musculus (house mouse)Potency22.016420
clomipramineMus musculus (house mouse)Potency31.622810
clotrimazoleMus musculus (house mouse)Potency22.465420
cloxyquinMus musculus (house mouse)Potency2.484220
danthronMus musculus (house mouse)Potency10.000010
atenololMus musculus (house mouse)Potency12.589310
dequaliniumMus musculus (house mouse)Potency18.860020
diazoxideMus musculus (house mouse)Potency12.589310
dichlorophenMus musculus (house mouse)Potency17.450420
diflunisalMus musculus (house mouse)Potency0.063110
diphenyleneiodoniumMus musculus (house mouse)Potency1.000010
dipyridamoleMus musculus (house mouse)Potency1.412510
dipyrithioneMus musculus (house mouse)Potency0.623020
disulfiramMus musculus (house mouse)Potency0.526320
droperidolMus musculus (house mouse)Potency7.943310
dyclonineMus musculus (house mouse)Potency10.000010
ebastineMus musculus (house mouse)Potency11.220210
ebselenMus musculus (house mouse)Potency22.762820
efavirenzMus musculus (house mouse)Potency28.183810
ellipticineMus musculus (house mouse)Potency8.175720
emodinMus musculus (house mouse)Potency35.481310
epirizoleMus musculus (house mouse)Potency14.658760
ethacrynic acidMus musculus (house mouse)Potency28.362720
ethosuximideMus musculus (house mouse)Potency2.818410
ethoxyquinMus musculus (house mouse)Potency6.309610
carbonyl cyanide p-trifluoromethoxyphenylhydrazoneMus musculus (house mouse)Potency0.616820
fenbendazoleMus musculus (house mouse)Potency14.348420
fenofibrateMus musculus (house mouse)Potency23.350710
fipronilMus musculus (house mouse)Potency19.901620
flufenamic acidMus musculus (house mouse)Potency35.481310
flumazenilMus musculus (house mouse)Potency0.100010
fluspirileneMus musculus (house mouse)Potency19.610720
flutamideMus musculus (house mouse)Potency31.056720
fusaric acidMus musculus (house mouse)Potency12.319420
gaboxadolMus musculus (house mouse)Potency35.481310
vanoxerineMus musculus (house mouse)Potency31.762620
gbr 12935Mus musculus (house mouse)Potency33.552020
gemfibrozilMus musculus (house mouse)Potency19.952610
glimepirideMus musculus (house mouse)Potency10.000010
glyburideMus musculus (house mouse)Potency31.622810
gossypolMus musculus (house mouse)Potency19.191220
guaiazuleneMus musculus (house mouse)Potency3.548110
n-(2-aminoethyl)-5-isoquinolinesulfonamideMus musculus (house mouse)Potency22.387210
haloperidolMus musculus (house mouse)Potency35.481310
haloproginMus musculus (house mouse)Potency6.351420
harmalineMus musculus (house mouse)Potency12.589310
hexachloropheneMus musculus (house mouse)Potency8.572520
hexylresorcinolMus musculus (house mouse)Potency2.511910
beta-thujaplicinMus musculus (house mouse)Potency5.344620
ethidiumMus musculus (house mouse)Potency22.740620
hydralazineMus musculus (house mouse)Potency14.125410
ibudilastMus musculus (house mouse)Potency17.782810
idebenoneMus musculus (house mouse)Potency16.815820
amrinoneMus musculus (house mouse)Potency31.622810
indirubin-3'-monoximeMus musculus (house mouse)Potency20.811420
indomethacinMus musculus (house mouse)Potency12.589310
indoprofenMus musculus (house mouse)Potency4.920920
iodoquinolMus musculus (house mouse)Potency2.010420
ipriflavoneMus musculus (house mouse)Potency35.481310
isoniazidMus musculus (house mouse)Potency14.125410
1-(2-naphthalenyl)-3-[(phenylmethyl)-propan-2-ylamino]-1-propanoneMus musculus (house mouse)Potency2.665120
1-(2-naphthalenyl)-2-propen-1-oneMus musculus (house mouse)Potency0.669420
7-amino-4-chloro-3-methoxy-2-benzopyran-1-oneMus musculus (house mouse)Potency11.034420
jugloneMus musculus (house mouse)Potency11.220210
nsc 664704Mus musculus (house mouse)Potency25.118910
celanideMus musculus (house mouse)Potency7.079510
lansoprazoleMus musculus (house mouse)Potency20.850120
lapacholMus musculus (house mouse)Potency27.401520
beta-lapachoneMus musculus (house mouse)Potency4.067720
lauric acidMus musculus (house mouse)Potency31.622810
leflunomideMus musculus (house mouse)Potency35.481310
liranaftateMus musculus (house mouse)Potency17.782810
loperamideMus musculus (house mouse)Potency3.981110
loratadineMus musculus (house mouse)Potency35.481310
ly 171883Mus musculus (house mouse)Potency12.589320
6-anilino-5,8-quinolinedioneMus musculus (house mouse)Potency3.814620
manidipineMus musculus (house mouse)Potency12.589310
maprotilineMus musculus (house mouse)Potency19.091920
edaravoneMus musculus (house mouse)Potency21.951110
mechlorethamineMus musculus (house mouse)Potency11.220210
meclofenamic acid(1-)Mus musculus (house mouse)Potency28.183810
meclofenamate sodium anhydrousMus musculus (house mouse)Potency35.481320
mefenamic acidMus musculus (house mouse)Potency35.481310
vitamin k 3Mus musculus (house mouse)Potency11.354620
mequitazineMus musculus (house mouse)Potency21.421520
metaproterenolMus musculus (house mouse)Potency5.623410
nocodazoleMus musculus (house mouse)Potency5.008620
methyl parathionMus musculus (house mouse)Potency10.610120
miconazoleMus musculus (house mouse)Potency11.220210
ml 7Mus musculus (house mouse)Potency14.125410
myoseverinMus musculus (house mouse)Potency12.589310
1,3-dicyclohexylureaMus musculus (house mouse)Potency0.631010
clorgylineMus musculus (house mouse)Potency11.220210
etoposide phosphateMus musculus (house mouse)Potency22.387210
nabumetoneMus musculus (house mouse)Potency12.589310
nalidixic acidMus musculus (house mouse)Potency2.818410
niclosamideMus musculus (house mouse)Potency7.498920
nifedipineMus musculus (house mouse)Potency16.373020
niflumic acidMus musculus (house mouse)Potency35.481310
nilutamideMus musculus (house mouse)Potency18.430220
nimodipineMus musculus (house mouse)Potency22.874110
nisoldipineMus musculus (house mouse)Potency14.125410
omeprazoleMus musculus (house mouse)Potency11.879910
oxyphenbutazoneMus musculus (house mouse)Potency5.045120
quinoneMus musculus (house mouse)Potency11.220210
papaverineMus musculus (house mouse)Potency13.592020
patulinMus musculus (house mouse)Potency1.006620
pca 4248Mus musculus (house mouse)Potency23.753120
pd 153035Mus musculus (house mouse)Potency12.589310
pd 158780Mus musculus (house mouse)Potency12.589320
pd 98059Mus musculus (house mouse)Potency31.622810
5-hydroxy-4-methoxy-5-(1-methylethenyl)-2-furanoneMus musculus (house mouse)Potency10.166320
perphenazineMus musculus (house mouse)Potency15.848910
phenazopyridineMus musculus (house mouse)Potency0.631010
phloretinMus musculus (house mouse)Potency31.622810
pifithrinMus musculus (house mouse)Potency1.806420
pomiferinMus musculus (house mouse)Potency28.934220
prazosinMus musculus (house mouse)Potency18.175120
prochlorperazineMus musculus (house mouse)Potency12.589310
propachlorMus musculus (house mouse)Potency11.220210
propargiteMus musculus (house mouse)Potency14.125410
propidiumMus musculus (house mouse)Potency2.837120
protoporphyrin ixMus musculus (house mouse)Potency19.952610
1,2,5,8-tetrahydroxy anthraquinoneMus musculus (house mouse)Potency17.819920
resorcinolMus musculus (house mouse)Potency35.481310
pf 5901Mus musculus (house mouse)Potency35.481310
riluzoleMus musculus (house mouse)Potency5.380820
ritanserinMus musculus (house mouse)Potency25.118920
ro 31-8220Mus musculus (house mouse)Potency27.717020
aurinMus musculus (house mouse)Potency33.552020
salicylamideMus musculus (house mouse)Potency2.511910
salmeterol xinafoateMus musculus (house mouse)Potency18.256320
sanguinarineMus musculus (house mouse)Potency5.907720
sb 239063Mus musculus (house mouse)Potency22.387210
sc-10Mus musculus (house mouse)Potency25.118910
scriptaidMus musculus (house mouse)Potency1.584910
simazineMus musculus (house mouse)Potency39.810710
streptonigrinMus musculus (house mouse)Potency18.256320
sulfanitranMus musculus (house mouse)Potency22.387210
sulfinpyrazoneMus musculus (house mouse)Potency24.035320
2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanolMus musculus (house mouse)Potency11.220210
tegafurMus musculus (house mouse)Potency7.506020
temefosMus musculus (house mouse)Potency35.481310
terfenadineMus musculus (house mouse)Potency20.895410
thiramMus musculus (house mouse)Potency0.696120
tioconazoleMus musculus (house mouse)Potency14.219120
tizanidineMus musculus (house mouse)Potency35.481310
ici 136,753Mus musculus (house mouse)Potency33.552020
triamtereneMus musculus (house mouse)Potency14.976320
triazolamMus musculus (house mouse)Potency0.794310
octoxynolMus musculus (house mouse)Potency35.481310
troglitazoneMus musculus (house mouse)Potency15.848910
delavirdineMus musculus (house mouse)Potency14.125410
6,18,30-trimethyl-3,9,12,15,21,24,27,33,36-nona(propan-2-yl)-1,7,13,19,25,31-hexaoxa-4,10,16,22,28,34-hexazacyclohexatriacontane-2,5,8,11,14,17,20,23,26,29,32,35-dodeconeMus musculus (house mouse)Potency0.406820
xylazineMus musculus (house mouse)Potency10.000010
ici 204,219Mus musculus (house mouse)Potency11.220210
zm 336372Mus musculus (house mouse)Potency11.220210
3,3',5-triiodothyropropionic acidMus musculus (house mouse)Potency0.316210
norethindrone acetateMus musculus (house mouse)Potency7.943310
prednisoneMus musculus (house mouse)Potency3.548110
methyldimethylaminoazobenzeneMus musculus (house mouse)Potency10.266320
mechlorethamine hydrochlorideMus musculus (house mouse)Potency21.421520
cantharidinMus musculus (house mouse)Potency5.011910
cetrimonium bromideMus musculus (house mouse)Potency14.140620
9,10-dimethyl-1,2-benzanthraceneMus musculus (house mouse)Potency35.481310
apomorphineMus musculus (house mouse)Potency21.118320
carbostyrilMus musculus (house mouse)Potency9.449420
p-dimethylaminoazobenzeneMus musculus (house mouse)Potency12.589320
papaverine hydrochlorideMus musculus (house mouse)Potency8.731620
androstenedioneMus musculus (house mouse)Potency19.149810
desoxycorticosteroneMus musculus (house mouse)Potency35.481310
cycloheximideMus musculus (house mouse)Potency1.744920
gliotoxinMus musculus (house mouse)Potency0.044710
quinacrine monohydrochlorideMus musculus (house mouse)Potency23.350720
tubercidinMus musculus (house mouse)Potency0.876520
dinitrofluorobenzeneMus musculus (house mouse)Potency22.387210
mestranolMus musculus (house mouse)Potency7.079510
chlorquinaldolMus musculus (house mouse)Potency0.726820
4-chlorobenzoic acidMus musculus (house mouse)Potency0.005010
azovioletMus musculus (house mouse)Potency5.925620
triamcinolone acetonideMus musculus (house mouse)Potency12.589310
hexachlorocyclopentadieneMus musculus (house mouse)Potency26.632020
triparanolMus musculus (house mouse)Potency21.133520
chlorfenetholMus musculus (house mouse)Potency25.118910
cumene hydroperoxideMus musculus (house mouse)Potency35.481310
acenaphthenequinoneMus musculus (house mouse)Potency3.162310
cyclizineMus musculus (house mouse)Potency6.309610
quinophthaloneMus musculus (house mouse)Potency3.473720
pindoneMus musculus (house mouse)Potency24.803320
rotenoneMus musculus (house mouse)Potency5.993120
9,10-phenanthrenequinoneMus musculus (house mouse)Potency2.578820
1-(2-pyridylazo)-2-naphtholMus musculus (house mouse)Potency1.722020
acriflavine chlorideMus musculus (house mouse)Potency21.280420
dimoxylineMus musculus (house mouse)Potency2.115420
penicillin vMus musculus (house mouse)Potency25.118910
acetopyrrothineMus musculus (house mouse)Potency0.324620
2-phenylphenolMus musculus (house mouse)Potency35.481310
aminacrineMus musculus (house mouse)Potency11.220210
decalinMus musculus (house mouse)Potency10.000010
dehydrothio-4-toluidineMus musculus (house mouse)Potency7.233420
proflavineMus musculus (house mouse)Potency15.848910
phenothiazineMus musculus (house mouse)Potency12.589310
n,n-diethyl 4-phenylenediamineMus musculus (house mouse)Potency25.118910
thiohexamMus musculus (house mouse)Potency8.912510
2-dichlorobenzeneMus musculus (house mouse)Potency0.003210
2-amino-4-methylphenolMus musculus (house mouse)Potency12.967620
2,4,5-trichlorophenolMus musculus (house mouse)Potency35.481310
4,4'-thiobis(6-tert-butyl-3-cresol)Mus musculus (house mouse)Potency14.976320
fentichlorMus musculus (house mouse)Potency11.232220
fast red bMus musculus (house mouse)Potency10.000010
tetramethylthiuram monosulfideMus musculus (house mouse)Potency5.660820
benzenesulfonyl chlorideMus musculus (house mouse)Potency35.481310
p-tert-butyl catecholMus musculus (house mouse)Potency17.488220
dimethyl-4-phenylenediamineMus musculus (house mouse)Potency24.803320
tetramethylphenylenediamineMus musculus (house mouse)Potency33.552020
triclocarbanMus musculus (house mouse)Potency35.481310
pyridostigmine bromideMus musculus (house mouse)Potency5.623410
4-aminodiphenylamineMus musculus (house mouse)Potency8.912510
n-isopropyl-n-phenyl-4-phenylenediamineMus musculus (house mouse)Potency35.481320
1,3-diphenylureaMus musculus (house mouse)Potency3.548110
n-oxydiethylene-2-benzothiazole sulfenamideMus musculus (house mouse)Potency12.535420
succinonitrileMus musculus (house mouse)Potency0.141310
2-aminoanthraquinoneMus musculus (house mouse)Potency12.589310
chloranilMus musculus (house mouse)Potency22.710620
2-toluic acidMus musculus (house mouse)Potency22.874120
1-hydroxyphthalazineMus musculus (house mouse)Potency27.717020
dibenzoylmethaneMus musculus (house mouse)Potency5.962220
dibenzothiazyl disulfideMus musculus (house mouse)Potency14.929220
benzethonium chlorideMus musculus (house mouse)Potency28.652620
deserpidineMus musculus (house mouse)Potency7.079520
captanMus musculus (house mouse)Potency1.681020
menthyl anthranilateMus musculus (house mouse)Potency35.481310
phenazopyridine hydrochlorideMus musculus (house mouse)Potency12.589320
2-aminobenzothiazoleMus musculus (house mouse)Potency25.118910
ziramMus musculus (house mouse)Potency0.677420
4-nitrosodimethylanilineMus musculus (house mouse)Potency3.931020
4'-(chloroacetyl)acetanilideMus musculus (house mouse)Potency13.427020
4-tert-octylphenolMus musculus (house mouse)Potency22.387210
sterogenolMus musculus (house mouse)Potency8.813620
ditiocarbMus musculus (house mouse)Potency4.585820
5H-dibenzo[b,f]azepineMus musculus (house mouse)Potency35.481320
ethynodiol diacetateMus musculus (house mouse)Potency15.848910
nitroblue tetrazoliumMus musculus (house mouse)Potency19.702020
hydralazine hydrochlorideMus musculus (house mouse)Potency13.516020
fluorometholoneMus musculus (house mouse)Potency13.956130
cyproterone acetateMus musculus (house mouse)Potency1.412510
rheinMus musculus (house mouse)Potency31.832620
plumbaginMus musculus (house mouse)Potency8.712520
cepharanthineMus musculus (house mouse)Potency11.220210
menadiolMus musculus (house mouse)Potency28.183810
kainic acidMus musculus (house mouse)Potency35.481310
3,4-toluenediamineMus musculus (house mouse)Potency8.096920
hematoxylinMus musculus (house mouse)Potency14.219120
dequalinium chlorideMus musculus (house mouse)Potency5.011910
apioleMus musculus (house mouse)Potency2.818410
coumarin-3-carboxylic acidMus musculus (house mouse)Potency1.412510
dazometMus musculus (house mouse)Potency6.491820
4,6-dinitro-o-cresolMus musculus (house mouse)Potency11.232220
4,4'-diaminoazobenzeneMus musculus (house mouse)Potency3.981110
dicyclohexylcarbodiimideMus musculus (house mouse)Potency3.625320
8-hydroxy-7-iodo-5-quinolinesulfonic acidMus musculus (house mouse)Potency12.589310
gentian violetMus musculus (house mouse)Potency7.850920
1-naphthylisothiocyanateMus musculus (house mouse)Potency9.449420
3-hydroxyflavoneMus musculus (house mouse)Potency5.530320
aminacrineMus musculus (house mouse)Potency12.062720
toluene 2,4-diisocyanateMus musculus (house mouse)Potency10.000010
pentabromophenolMus musculus (house mouse)Potency22.387210
3,4,5-trichlorophenolMus musculus (house mouse)Potency35.481320
Berberine chloride (TN)Mus musculus (house mouse)Potency15.848910
2-phenylbenzimidazoleMus musculus (house mouse)Potency0.141310
n-(1,3-dimethylbutyl)-n'-phenyl-1,4-phenylenediamineMus musculus (house mouse)Potency11.703120
2,3,5-trichlorophenolMus musculus (house mouse)Potency10.000010
3-methoxycatecholMus musculus (house mouse)Potency23.350720
2-phenylindoleMus musculus (house mouse)Potency7.079510
demoxepamMus musculus (house mouse)Potency5.011910
cyproheptadine hydrochloride (anhydrous)Mus musculus (house mouse)Potency35.481310
dinobutonMus musculus (house mouse)Potency35.481320
estradiol valerateMus musculus (house mouse)Potency28.183810
pyrrolnitrinMus musculus (house mouse)Potency22.106020
bunamidineMus musculus (house mouse)Potency28.934220
c 137Mus musculus (house mouse)Potency11.220210
tetradecyltrimethylammoniumMus musculus (house mouse)Potency7.191220
2,2'-diaminodiphenyldisulfideMus musculus (house mouse)Potency35.481320
2-amino-4-phenylphenolMus musculus (house mouse)Potency22.740620
ethidium bromideMus musculus (house mouse)Potency19.307220
carmineMus musculus (house mouse)Potency14.620520
amylmetacresolMus musculus (house mouse)Potency35.481310
tribromsalanMus musculus (house mouse)Potency22.387210
antimycin aMus musculus (house mouse)Potency44.668410
flurandrenoloneMus musculus (house mouse)Potency28.183810
azacyclonolMus musculus (house mouse)Potency14.125410
tetrachloroisophthalonitrileMus musculus (house mouse)Potency2.145120
2-tert-butylhydroquinoneMus musculus (house mouse)Potency14.831720
amiloride hydrochloride, anhydrousMus musculus (house mouse)Potency35.481310
pimozideMus musculus (house mouse)Potency34.709620
pasiniazideMus musculus (house mouse)Potency23.350720
flumethasoneMus musculus (house mouse)Potency8.912510
2,4-diacetylphloroglucinolMus musculus (house mouse)Potency6.409220
dienochlorMus musculus (house mouse)Potency7.996020
ethoxazeneMus musculus (house mouse)Potency9.456220
didecyldimethylammoniumMus musculus (house mouse)Potency22.387210
quinomethionateMus musculus (house mouse)Potency8.764920
phenthoate, (+-)-isomerMus musculus (house mouse)Potency15.186120
1,2-benzisothiazoline-3-oneMus musculus (house mouse)Potency1.973120
1-myristylpicoliniumMus musculus (house mouse)Potency8.285220
dichloroacetonitrileMus musculus (house mouse)Potency5.865420
dibromoacetonitrileMus musculus (house mouse)Potency2.511910
pentaerythrityl triacrylateMus musculus (house mouse)Potency5.045120
nsc 3852Mus musculus (house mouse)Potency5.723820
diloxanide furoateMus musculus (house mouse)Potency35.481310
2-(alpha-thenoylamino)-2-nitro-5-thiazoleMus musculus (house mouse)Potency16.660420
nitroxolineMus musculus (house mouse)Potency0.499720
2,2',4'-trichloroacetophenoneMus musculus (house mouse)Potency15.649820
cladribineMus musculus (house mouse)Potency19.952610
beclomethasoneMus musculus (house mouse)Potency35.481310
fluoropheneMus musculus (house mouse)Potency4.739420
1,6-bismaleimidohexaneMus musculus (house mouse)Potency2.026820
2,3,4,5-tetrachlorophenateMus musculus (house mouse)Potency35.481320
benorilateMus musculus (house mouse)Potency14.125410
octocryleneMus musculus (house mouse)Potency35.481310
4-(4-dimethylaminophenylazo)benzoic acidMus musculus (house mouse)Potency0.956820
methylene bis(thiocyanate)Mus musculus (house mouse)Potency0.784420
helenalinMus musculus (house mouse)Potency3.162320
camptothecinMus musculus (house mouse)Potency0.831520
1,6-hexanediol diacrylateMus musculus (house mouse)Potency30.300120
pyrithione zincMus musculus (house mouse)Potency0.071320
diacereinMus musculus (house mouse)Potency10.000010
clioxanideMus musculus (house mouse)Potency22.535820
2,3,4-trichlorophenolMus musculus (house mouse)Potency12.589310
tetradecanoylphorbol acetateMus musculus (house mouse)Potency10.000010
metergolineMus musculus (house mouse)Potency16.803710
clonixinMus musculus (house mouse)Potency28.934210
n-(cyclohexylthio)phthalimideMus musculus (house mouse)Potency28.934220
tetraethylene glycol diacrylateMus musculus (house mouse)Potency23.688720
mecysteineMus musculus (house mouse)Potency0.707910
oryzalinMus musculus (house mouse)Potency35.481310
oxadiazonMus musculus (house mouse)Potency22.387210
2,5-dichloro-1,4-phenylenediamineMus musculus (house mouse)Potency2.818410
daunorubicinMus musculus (house mouse)Potency4.283620
cetylpyridinium chloride anhydrousMus musculus (house mouse)Potency2.403520
thymolphthaleinMus musculus (house mouse)Potency24.035320
butonateMus musculus (house mouse)Potency0.006310
2-methyl-1-nitroanthraquinoneMus musculus (house mouse)Potency35.481310
rafoxanideMus musculus (house mouse)Potency25.217120
triazophosMus musculus (house mouse)Potency19.952610
clobetasol propionateMus musculus (house mouse)Potency23.350720
(7S,9S)-7-[(4-amino-5-hydroxy-6-methyl-2-oxanyl)oxy]-6,9,11-trihydroxy-9-(2-hydroxy-1-oxoethyl)-4-methoxy-8,10-dihydro-7H-tetracene-5,12-dioneMus musculus (house mouse)Potency10.000010
cambendazoleMus musculus (house mouse)Potency35.481320
frentizoleMus musculus (house mouse)Potency10.000010
2-n-octyl-4-isothiazolin-3-oneMus musculus (house mouse)Potency0.538920
penfluridolMus musculus (house mouse)Potency11.294720
N-fluorenylacetamideMus musculus (house mouse)Potency4.466810
moricizine hydrochlorideMus musculus (house mouse)Potency35.481310
feprazoneMus musculus (house mouse)Potency31.622810
proroxanMus musculus (house mouse)Potency7.079520
etomidateMus musculus (house mouse)Potency3.162310
isovelleralMus musculus (house mouse)Potency1.267320
methyldopaMus musculus (house mouse)Potency35.481320
ciclopirox olamineMus musculus (house mouse)Potency1.536920
bifenoxMus musculus (house mouse)Potency22.387210
lonidamineMus musculus (house mouse)Potency31.622810
etofylline clofibrateMus musculus (house mouse)Potency35.481310
nicardipine hydrochlorideMus musculus (house mouse)Potency8.912510
nitazoxanideMus musculus (house mouse)Potency19.417420
closantelMus musculus (house mouse)Potency22.387210
s-2678Mus musculus (house mouse)Potency3.441220
idarubicinMus musculus (house mouse)Potency17.782810
propiconazoleMus musculus (house mouse)Potency21.450920
N-[4-(dimethylamino)phenyl]-3,4,5-trimethoxybenzamideMus musculus (house mouse)Potency12.589310
deltanitMus musculus (house mouse)Potency30.300120
cerm-1978Mus musculus (house mouse)Potency11.904820
triclabendazoleMus musculus (house mouse)Potency20.040920
mitoxantrone hydrochlorideMus musculus (house mouse)Potency7.506020
fenoxycarbMus musculus (house mouse)Potency27.717020
dazoxibenMus musculus (house mouse)Potency35.481310
lovastatinMus musculus (house mouse)Potency7.079510
chaetochrominMus musculus (house mouse)Potency5.530320
rimcazoleMus musculus (house mouse)Potency31.622810
3-chloro-4-(dichloromethyl)-5-hydroxy-2(5h)-furanoneMus musculus (house mouse)Potency2.528620
locerylMus musculus (house mouse)Potency31.622810
idazoxanMus musculus (house mouse)Potency15.848910
raloxifene hydrochlorideMus musculus (house mouse)Potency23.350720
mifepristoneMus musculus (house mouse)Potency8.912510
nitrogenase stabilizing-protective protein, bacteriaMus musculus (house mouse)Potency22.387210
finasterideMus musculus (house mouse)Potency3.981110
cy 208-243Mus musculus (house mouse)Potency11.220210
adapaleneMus musculus (house mouse)Potency35.481310
amlodipine besylateMus musculus (house mouse)Potency35.481310
niguldipineMus musculus (house mouse)Potency31.832620
mibefradil dihydrochlorideMus musculus (house mouse)Potency17.488220
mibefradilMus musculus (house mouse)Potency35.481310
topotecan hydrochlorideMus musculus (house mouse)Potency5.120920
aripiprazoleMus musculus (house mouse)Potency0.707910
ziprasidoneMus musculus (house mouse)Potency4.466810
relcovaptanMus musculus (house mouse)Potency35.481310
adenosineMus musculus (house mouse)Potency15.848910
phenelzine sulfateMus musculus (house mouse)Potency0.354810
tertiary-amyl methyl etherMus musculus (house mouse)Potency4.466810
Allyl nonanoateMus musculus (house mouse)Potency0.501210
Eugenyl benzoateMus musculus (house mouse)Potency35.481310
daunorubicin hydrochlorideMus musculus (house mouse)Potency3.723620
doxazosin mesylateMus musculus (house mouse)Potency12.589310
sertraline hydrochlorideMus musculus (house mouse)Potency24.803320
dexamethasone 17-valerateMus musculus (house mouse)Potency21.712320
efavirenzMus musculus (house mouse)Potency12.589310
nelfinavir mesylateMus musculus (house mouse)Potency7.079510
nelfinavirMus musculus (house mouse)Potency11.220210
meclizine monohydrochlorideMus musculus (house mouse)Potency25.118910
mevastatinMus musculus (house mouse)Potency14.125410
bts 54 524Mus musculus (house mouse)Potency10.000010
ursolic acidMus musculus (house mouse)Potency9.759130
arctigeninMus musculus (house mouse)Potency3.715820
diphenylcyclopropenoneMus musculus (house mouse)Potency19.554320
salvinMus musculus (house mouse)Potency25.665120
neocuproineMus musculus (house mouse)Potency0.406820
sulconazole, mononitrate, (+-)-isomerMus musculus (house mouse)Potency20.275620
ethefilMus musculus (house mouse)Potency0.100010
rutecarpineMus musculus (house mouse)Potency24.035320
indocateMus musculus (house mouse)Potency35.481310
lercanidipineMus musculus (house mouse)Potency17.488220
azelnidipineMus musculus (house mouse)Potency35.481320
repaglinideMus musculus (house mouse)Potency35.481310
thioridazine hydrochlorideMus musculus (house mouse)Potency17.488220
toxoflavinMus musculus (house mouse)Potency0.527940
xanthoxyletinMus musculus (house mouse)Potency14.125410
dibenzthioneMus musculus (house mouse)Potency15.257320
iodophthaleinMus musculus (house mouse)Potency35.481310
dictamnineMus musculus (house mouse)Potency22.387210
dimidium bromideMus musculus (house mouse)Potency17.488220
2,6-dimethoxy-1,4-benzoquinoneMus musculus (house mouse)Potency3.642620
1,2-dithiol-3-thioneMus musculus (house mouse)Potency18.854120
2-aminodiphenylamineMus musculus (house mouse)Potency12.589310
dyclonine hydrochlorideMus musculus (house mouse)Potency26.868820
nebularineMus musculus (house mouse)Potency5.120920
clomipramine hydrochlorideMus musculus (house mouse)Potency35.481310
prazosin hydrochlorideMus musculus (house mouse)Potency7.369720
miconazole nitrateMus musculus (house mouse)Potency20.283220
econazole nitrateMus musculus (house mouse)Potency13.808820
befuralineMus musculus (house mouse)Potency11.220210
quinocideMus musculus (house mouse)Potency16.930820
butinolineMus musculus (house mouse)Potency0.794310
1,3,5-trimethoxybenzeneMus musculus (house mouse)Potency31.622810
2-chloro-1,4-benzoquinoneMus musculus (house mouse)Potency23.350720
2,6-dihydroxyacetophenoneMus musculus (house mouse)Potency15.848910
2,6-di-tert-butyl-4-nitrophenolMus musculus (house mouse)Potency9.296120
2-(2'-pyridyl)benzimidazoleMus musculus (house mouse)Potency5.966520
2,2',2''-terpyridineMus musculus (house mouse)Potency12.589310
propipocaine monohydrochlorideMus musculus (house mouse)Potency18.256320
5-methyl-8-hydroxyquinolineMus musculus (house mouse)Potency6.962220
clobetasone butyrateMus musculus (house mouse)Potency10.000010
guanfacine hydrochlorideMus musculus (house mouse)Potency17.900820
loperamide hydrochlorideMus musculus (house mouse)Potency22.387210
maprotiline hydrochlorideMus musculus (house mouse)Potency27.394320
opipramol hydrochlorideMus musculus (house mouse)Potency11.220210
fluphenacurMus musculus (house mouse)Potency15.186120
chlormidazoleMus musculus (house mouse)Potency21.127720
hesperetinMus musculus (house mouse)Potency6.309610
magnololMus musculus (house mouse)Potency22.983310
honokiolMus musculus (house mouse)Potency24.454120
jatrorrhizineMus musculus (house mouse)Potency35.481310
nobiletinMus musculus (house mouse)Potency11.220210
nonoxynol-9Mus musculus (house mouse)Potency35.481320
9-aminocamptothecinMus musculus (house mouse)Potency0.187420
9-methoxyellipticineMus musculus (house mouse)Potency3.814620
3-hydroxy naphthoic acid hydrazideMus musculus (house mouse)Potency16.803720
methyl fluorone blackMus musculus (house mouse)Potency12.062720
2-phenyl-4,5-dichloro-3-pyridazinoneMus musculus (house mouse)Potency10.610120
tetrandrineMus musculus (house mouse)Potency26.751920
tosyllysine chloromethyl ketoneMus musculus (house mouse)Potency35.481310
fangchinolineMus musculus (house mouse)Potency24.035320
tryptanthrineMus musculus (house mouse)Potency11.220210
pramoxine hydrochlorideMus musculus (house mouse)Potency24.803310
n-benzylmaleimideMus musculus (house mouse)Potency26.632020
1,2,3,4,5,6-hexabromocyclohexaneMus musculus (house mouse)Potency6.477620
2,5-di-tert-butyl-4-hydroxyanisoleMus musculus (house mouse)Potency35.481310
atovaquoneMus musculus (house mouse)Potency5.750620
4-(2-thiazolylazo)resorcinolMus musculus (house mouse)Potency7.079510
4-methoxybenzohydrazideMus musculus (house mouse)Potency2.818410
3,5-di-tert-butyl-1,2-benzoquinoneMus musculus (house mouse)Potency11.294720
benzoyltyrosine ethyl esterMus musculus (house mouse)Potency1.825620
2-(4-Morpholinyl)benzothiazoleMus musculus (house mouse)Potency28.183810
2-methyl-4-nitroquinoline 1-oxideMus musculus (house mouse)Potency5.745720
dodecyltetraethylene glycol monoetherMus musculus (house mouse)Potency15.848910
n-benzyl-4-toluidineMus musculus (house mouse)Potency15.848910
2-amino-5-bromobenzoic acidMus musculus (house mouse)Potency2.115420
1-(2-phenanthrenyl)ethanoneMus musculus (house mouse)Potency28.183810
witisolMus musculus (house mouse)Potency1.935120
bexaroteneMus musculus (house mouse)Potency17.782810
8-(4-tolylsulfonylamino)quinolineMus musculus (house mouse)Potency1.667820
fentanyl isothiocyanateMus musculus (house mouse)Potency35.481320
isoamyl 4-n,n-dimethylaminobenzoateMus musculus (house mouse)Potency5.623410
prochlorperazine edisylate saltMus musculus (house mouse)Potency19.149820
azocyclotinMus musculus (house mouse)Potency28.934220
hydroxyflutamideMus musculus (house mouse)Potency35.481310
pyridabenMus musculus (house mouse)Potency0.014110
meclizine hydrochlorideMus musculus (house mouse)Potency8.912510
lopinavirMus musculus (house mouse)Potency12.589310
cycloadiphenine hydrochlorideMus musculus (house mouse)Potency22.387210
tyrphostin 8Mus musculus (house mouse)Potency31.056720
1-(2-thiazolylazo)-2-naphtholMus musculus (house mouse)Potency2.403520
cortisol octanoateMus musculus (house mouse)Potency11.220210
coumarin 7Mus musculus (house mouse)Potency5.581030
3-(n-salicyloyl)amino-1,2,4-triazoleMus musculus (house mouse)Potency35.481310
harmol hydrochlorideMus musculus (house mouse)Potency35.481310
5-MethoxyflavoneMus musculus (house mouse)Potency16.821520
diffractaic acidMus musculus (house mouse)Potency14.987210
osajinMus musculus (house mouse)Potency31.116620
4-methyl-N-(phenylmethyl)benzenesulfonamideMus musculus (house mouse)Potency15.848910
1,3,4,10-Tetrahydro-9(2H)-acridinoneMus musculus (house mouse)Potency33.552020
4',5,6,7-tetramethoxyflavoneMus musculus (house mouse)Potency10.000010
quercetin 5,7,3',4'-tetramethyl etherMus musculus (house mouse)Potency2.818420
10-hydroxycamptothecinMus musculus (house mouse)Potency6.012220
9-methoxyacridineMus musculus (house mouse)Potency18.256320
lecanoric acidMus musculus (house mouse)Potency11.220210
4-methoxydalbergioneMus musculus (house mouse)Potency25.665120
nortrachelogeninMus musculus (house mouse)Potency3.936920
diphyllinMus musculus (house mouse)Potency10.000010
EupatoriochromeneMus musculus (house mouse)Potency19.622220
3-chloro-6-hydrazino-pyridazineMus musculus (house mouse)Potency22.740620
5-(Ethylthio)-1,3,4-thiadiazol-2-amineMus musculus (house mouse)Potency1.000010
alexidine dihydrchlorideMus musculus (house mouse)Potency31.622810
sn 38Mus musculus (house mouse)Potency0.354810
bosentan anhydrousMus musculus (house mouse)Potency35.481310
beta-carboline-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency13.131120
sudan yellow 3gMus musculus (house mouse)Potency25.118910
dihydroergocristineMus musculus (house mouse)Potency2.818410
gr 127935Mus musculus (house mouse)Potency25.787720
deguelinMus musculus (house mouse)Potency561.291220
triptolideMus musculus (house mouse)Potency0.357120
ZearalanoneMus musculus (house mouse)Potency35.481310
desethylterbuthylazineMus musculus (house mouse)Potency12.589310
tanshinoneMus musculus (house mouse)Potency10.000010
3,4-dimethoxydalbergioneMus musculus (house mouse)Potency12.967620
pirlindole hydrochlorideMus musculus (house mouse)Potency1.995310
zk 93426Mus musculus (house mouse)Potency26.632020
1-[4-[2-hydroxy-3-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]propoxy]phenyl]-1-propanoneMus musculus (house mouse)Potency22.387210
3-(1-piperidinyl)-1-(4-propan-2-yloxyphenyl)-1-propanoneMus musculus (house mouse)Potency8.154820
n-(phenylthio)-epsilon-caprolactamMus musculus (house mouse)Potency28.934220
1-(6-hydroxy-2-isopropenyl-1-benzofuran-5-yl)-1-ethanoneMus musculus (house mouse)Potency0.446710
ak 2123Mus musculus (house mouse)Potency35.481310
piscidic acidMus musculus (house mouse)Potency3.981110
zk 93423Mus musculus (house mouse)Potency4.466810
pd 81723Mus musculus (house mouse)Potency31.622810
a 68930Mus musculus (house mouse)Potency26.651420
nsc 607097Mus musculus (house mouse)Potency8.539820
profenamine hydrochlorideMus musculus (house mouse)Potency11.220210
alpha-(n6-adenyl)styrene oxideMus musculus (house mouse)Potency14.125410
9-methoxy-n(2)-methylellipticiniumMus musculus (house mouse)Potency12.589310
lestaurtinibMus musculus (house mouse)Potency14.005320
sb 200646Mus musculus (house mouse)Potency12.589310
vb 20b7Mus musculus (house mouse)Potency7.079510
2-(3,4-dichlorophenyl)-n-methyl-n-(1-(3-isothiocyanatophenyl)-2-(1-pyrrolidinyl)ethyl)acetamideMus musculus (house mouse)Potency31.622820
n-butyl beta-carboline-3-carboxylateMus musculus (house mouse)Potency23.735820
1,3-dipropyl-8-phenylxanthineMus musculus (house mouse)Potency3.548110
2-(4-ethoxybenzyl)-1-diethylaminoethyl-5-isothiocyanatobenzimidazoleMus musculus (house mouse)Potency35.481320
3-(alpha,alpha-dimethylallyl)psoralenMus musculus (house mouse)Potency35.481310
n-(6-methoxy-8-quinolyl)-4-toluenesulfonamideMus musculus (house mouse)Potency0.716320
pyrophenMus musculus (house mouse)Potency23.350720
2-((5-chloro-2-methoxyphenyl)azo)-1h-imidazoleMus musculus (house mouse)Potency7.943310
3,5-bis(trifluoromethyl)benzyl n-acetyltryptophanMus musculus (house mouse)Potency28.183810
l 733060Mus musculus (house mouse)Potency25.118910
l 741742Mus musculus (house mouse)Potency35.481310
bts 54 505Mus musculus (house mouse)Potency10.000010
cd 437Mus musculus (house mouse)Potency19.731220
5-hydroxy-3,6,7,8,3',4'-hexamethoxyflavoneMus musculus (house mouse)Potency18.169620
1,3-bis(3-chlorophenyl)ureaMus musculus (house mouse)Potency15.848910
3',4'-dihydroxyflavoneMus musculus (house mouse)Potency3.162310
3,3',4'-trihydroxyflavoneMus musculus (house mouse)Potency31.622810
lexaproMus musculus (house mouse)Potency35.481310
1-(1,3-benzodioxol-5-yl)-3-(1-piperidinyl)-1-propanoneMus musculus (house mouse)Potency7.875820
nsc-141549Mus musculus (house mouse)Potency19.952610
proksifein hydrochlorideMus musculus (house mouse)Potency4.466810
ezetimibeMus musculus (house mouse)Potency13.516020
8-(methylsulfonylamino)quinolineMus musculus (house mouse)Potency7.126420
1,4-di(2'-thienyl)-1,4-butadioneMus musculus (house mouse)Potency35.481310
1,4-dimethyl-6-nitro-9H-carbazoleMus musculus (house mouse)Potency35.481310
cinacalcetMus musculus (house mouse)Potency25.665120
sch 45752Mus musculus (house mouse)Potency8.800620
2-chloroacetoacetanilideMus musculus (house mouse)Potency35.481320
isosakuranetinMus musculus (house mouse)Potency12.589310
sulochrinMus musculus (house mouse)Potency35.481310
2-phenyl-4-oxohydroquinolineMus musculus (house mouse)Potency21.712310
8-(4-benzenesulfonylamino)quinolineMus musculus (house mouse)Potency2.110920
stephenanthrineMus musculus (house mouse)Potency1.258910
3,3-bis(4-hydroxy-3-methylphenyl)-1H-indol-2-oneMus musculus (house mouse)Potency15.848910
2,4-dinitropyrimidinyl-2-thiophenolMus musculus (house mouse)Potency15.165220
enniatin bMus musculus (house mouse)Potency27.005020
2-phenyl-1,2-benzisothiazol-3-(2h)-oneMus musculus (house mouse)Potency3.183220
histidinolMus musculus (house mouse)Potency35.481310
17 alpha-hydroxyprogesterone caproateMus musculus (house mouse)Potency35.481310
imazalil sulfateMus musculus (house mouse)Potency35.481310
nbi 27914Mus musculus (house mouse)Potency3.548110
sb 216763Mus musculus (house mouse)Potency35.481310
antalarminMus musculus (house mouse)Potency15.211320
chrysene-1,4-dioneMus musculus (house mouse)Potency14.125420
4',6-dihydroxyflavoneMus musculus (house mouse)Potency17.782810
6,7-dichloro-2,3-dimethylquinoxalineMus musculus (house mouse)Potency10.000010
tosifenMus musculus (house mouse)Potency35.481310
2-(4-morpholinoanilino)-6-cyclohexylaminopurineMus musculus (house mouse)Potency22.387210
4-(2-methyl-5-phenyl-1-pyrrolyl)benzoic acidMus musculus (house mouse)Potency25.118910
sorafenibMus musculus (house mouse)Potency10.750920
(7R)-7,15,17-trihydroxy-11-methyl-12-oxabicyclo[12.4.0]octadeca-1(14),15,17-trien-13-oneMus musculus (house mouse)Potency21.169920
nutlin 3Mus musculus (house mouse)Potency11.220210
N-(4-methoxyphenyl)-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency35.481310
brazilinMus musculus (house mouse)Potency3.165720
vacquinol-1Mus musculus (house mouse)Potency21.450920
gossypol acetic acidMus musculus (house mouse)Potency4.087120
ml 204Mus musculus (house mouse)Potency35.481310
(R)-RoemerineMus musculus (house mouse)Potency7.079510
benzatropine methanesulfonateMus musculus (house mouse)Potency1.995310
vincaleukoblastineMus musculus (house mouse)Potency11.220210
2-hydroxyestradiolMus musculus (house mouse)Potency12.589320
1,10-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,9-diolMus musculus (house mouse)Potency28.183810
chondocurine (1beta)-(+-)-isomerMus musculus (house mouse)Potency0.354810
n-acetyl-1-aminopyreneMus musculus (house mouse)Potency39.810710
coronopilinMus musculus (house mouse)Potency11.220210
1-(2,4-Dihydroxyphenyl)-2-(4-methoxyphenyl)ethanoneMus musculus (house mouse)Potency35.481320
nsc 95397Mus musculus (house mouse)Potency1.688920
2-cyano-2-cyclohexylideneacetamideMus musculus (house mouse)Potency35.481310
2-chloro-3-(4-methylanilino)naphthalene-1,4-dioneMus musculus (house mouse)Potency25.665120
dimethyl 2-(2-nitrobenzylidene)malonateMus musculus (house mouse)Potency17.782810
(RS)-coclaurineMus musculus (house mouse)Potency31.832620
aromaticinMus musculus (house mouse)Potency8.154820
homoharringtonineMus musculus (house mouse)Potency3.355220
1-(4-chlorophenyl)-3-(2-ethoxyphenyl)ureaMus musculus (house mouse)Potency8.116020
2-(4-aminophenyl)quinolineMus musculus (house mouse)Potency11.220210
pd 146176Mus musculus (house mouse)Potency7.233420
2-quinolinecarboxylic acid (4-nitrophenyl) esterMus musculus (house mouse)Potency10.000010
acetic acid (4-acetyloxy-6,7-dimethyl-5,8-dihydronaphthalen-1-yl) esterMus musculus (house mouse)Potency19.952610
N-(3-hydroxyphenyl)-2-(2,4,5-trichlorophenoxy)acetamideMus musculus (house mouse)Potency11.220210
4-[4-(3-methyl-4-nitrophenoxy)butoxy]benzonitrileMus musculus (house mouse)Potency25.118910
4-chloro-1H-indazol-3-amineMus musculus (house mouse)Potency35.481310
nsc228155Mus musculus (house mouse)Potency1.000020
1-(benzenesulfonyl)indoleMus musculus (house mouse)Potency28.183810
dicentrineMus musculus (house mouse)Potency24.035320
nsc-260594Mus musculus (house mouse)Potency2.511910
hematoxylinMus musculus (house mouse)Potency27.717010
N-[2-(1-azepanyl)-1,3-benzothiazol-6-yl]carbamic acid ethyl esterMus musculus (house mouse)Potency31.622810
2,2-bis(hydroxymethyl)-1-azabicyclo(2,2,2,)octan-3-oneMus musculus (house mouse)Potency15.211220
2-(1-adamantyl)imidazoleMus musculus (house mouse)Potency17.782810
pinafideMus musculus (house mouse)Potency10.610120
pifithrin muMus musculus (house mouse)Potency20.552320
3-(prop-2-enylthio)-5-thiophen-2-yl-1H-1,2,4-triazoleMus musculus (house mouse)Potency23.350720
[4-(4-hydroxyphenyl)phenyl]-phenylmethanoneMus musculus (house mouse)Potency10.665420
N-phenylcarbamic acid 2-phenoxyethyl esterMus musculus (house mouse)Potency1.258910
sakuranetinMus musculus (house mouse)Potency12.589310
5-[(4-chlorophenyl)methylthio]-1,3,4-thiadiazol-2-amineMus musculus (house mouse)Potency14.125410
3-(2-Methylpropanoyloxy)-8-(2-methylbutanoyloxy)-9,10-epoxy-p-mentha-1,3,5-trieneMus musculus (house mouse)Potency22.387210
7-Methoxy-2-methylisoflavoneMus musculus (house mouse)Potency10.000010
nsc606985Mus musculus (house mouse)Potency0.323120
1-phenyl-3-methyl-4-benzoyl-5-pyrazoloneMus musculus (house mouse)Potency22.387210
DubamineMus musculus (house mouse)Potency17.991220
4,5,7-trihydroxy-9,10-dioxo-2-anthracenecarboxylic acidMus musculus (house mouse)Potency8.764920
3-(1H-indol-3-yl)-1-phenylpyrrolidine-2,5-dioneMus musculus (house mouse)Potency22.387210
7-hydroxy-5-methyl-2-(2-oxopropyl)-8-[3,4,5-trihydroxy-6-(hydroxymethyl)-2-oxanyl]-1-benzopyran-4-oneMus musculus (house mouse)Potency0.199510
2,5-bis(5-hydroxymethyl-2-thienyl)furanMus musculus (house mouse)Potency1.108020
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneMus musculus (house mouse)Potency5.011920
7-benzoyl-3-chloroindolizine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency3.162310
nsc 663284Mus musculus (house mouse)Potency3.811820
2,2'-spirobi[3,6,7,8-tetrahydro-1H-cyclopenta[g]naphthalene]-5,5'-dioneMus musculus (house mouse)Potency33.552020
N2-phenyl-5-methyl-4,5-dihydro-1,3-thiazol-2-amineMus musculus (house mouse)Potency3.548110
3-imino-1,5,5-trimethyl-2-oxabicyclo[2.2.1]heptane-4,7,7-tricarbonitrileMus musculus (house mouse)Potency21.712320
ritonavirMus musculus (house mouse)Potency14.125410
nu 6027Mus musculus (house mouse)Potency16.487520
4-amino-2,6-dimethyl-5-[3-(4-methylphenyl)-1H-pyrazol-5-yl]-3-pyridazinoneMus musculus (house mouse)Potency35.481310
methylmercuric chlorideMus musculus (house mouse)Potency0.799620
1-methoxy-10H-acridin-9-oneMus musculus (house mouse)Potency3.162310
2H-pyrazolo[4,3-b]quinoxalin-3-amineMus musculus (house mouse)Potency14.721420
carnosineMus musculus (house mouse)Potency2.238710
5-hydroxytryptophanMus musculus (house mouse)Potency11.220210
tosylphenylalanyl chloromethyl ketoneMus musculus (house mouse)Potency25.665120
(R)-norlaudanosolineMus musculus (house mouse)Potency35.481310
digitoxinMus musculus (house mouse)Potency1.584910
amiodarone hydrochlorideMus musculus (house mouse)Potency28.934220
angustibalinMus musculus (house mouse)Potency1.258920
grosheiminMus musculus (house mouse)Potency24.035320
naringinMus musculus (house mouse)Potency0.707910
ochratoxin aMus musculus (house mouse)Potency19.118020
alpha bitter acidMus musculus (house mouse)Potency17.900820
acetylleucyl-leucyl-norleucinalMus musculus (house mouse)Potency2.238710
sb 228357Mus musculus (house mouse)Potency12.589310
carubicinMus musculus (house mouse)Potency5.313820
tolterodineMus musculus (house mouse)Potency5.623410
doxorubicin hydrochlorideMus musculus (house mouse)Potency3.788020
vinpocetineMus musculus (house mouse)Potency19.952610
amcinonideMus musculus (house mouse)Potency8.912510
flumethasone pivalateMus musculus (house mouse)Potency22.387210
dihydroergocristine monomesylateMus musculus (house mouse)Potency35.481310
tretinoinMus musculus (house mouse)Potency6.390310
arachidonic acidMus musculus (house mouse)Potency34.195120
resveratrolMus musculus (house mouse)Potency11.302640
retinolMus musculus (house mouse)Potency14.125410
tacrolimusMus musculus (house mouse)Potency11.220210
sr 12813Mus musculus (house mouse)Potency12.589310
gw 6471Mus musculus (house mouse)Potency22.387210
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolMus musculus (house mouse)Potency16.531120
gw 3965Mus musculus (house mouse)Potency35.481310
t0901317Mus musculus (house mouse)Potency1.995310
hts 466284Mus musculus (house mouse)Potency2.578820
epothilone bMus musculus (house mouse)Potency35.481310
diethylstilbestrolMus musculus (house mouse)Potency22.387210
6-bromoindirubin-3'-oximeMus musculus (house mouse)Potency10.000010
alitretinoinMus musculus (house mouse)Potency7.943310
afimoxifeneMus musculus (house mouse)Potency25.665120
(2R,3S,5S)-2-(6-aminopurin-9-yl)-5-(hydroxymethyl)-3-oxolanolMus musculus (house mouse)Potency6.045720
ketoconazoleMus musculus (house mouse)Potency7.079510
purvalanol aMus musculus (house mouse)Potency14.125410
dactinomycinMus musculus (house mouse)Potency18.206420
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneMus musculus (house mouse)Potency4.585820
rubitecanMus musculus (house mouse)Potency0.360020
(2S)-2-[[[4-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-1-oxo-3-phenylpropan-2-yl]amino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-3-phenylpropanoic acid tert-butyl esterMus musculus (house mouse)Potency15.165220
6,8-diprenylgenisteinMus musculus (house mouse)Potency16.010520
2-methyl-5-(4-methylanilino)-1,3-benzothiazole-4,7-dioneMus musculus (house mouse)Potency2.375320
4-(2-oxazolo[4,5-b]pyridinyl)anilineMus musculus (house mouse)Potency35.481310
3-Furan-3-yl-3a,7-dimethyl-3a,4,5,6-tetrahydro-3H-isobenzofuran-1-oneMus musculus (house mouse)Potency5.623410
menadione sodium bisulfite, trihydrateMus musculus (house mouse)Potency10.610120
N-bis(N-methylanilino)phosphoryl-N-methylanilineMus musculus (house mouse)Potency30.300120
jp-1302Mus musculus (house mouse)Potency10.000010
2-sulfanylidene-1,3-dithiole-4,5-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency19.622220
1-phenyl-4-pyrazololMus musculus (house mouse)Potency6.309610
1-[(4-fluoro-1-naphthalenyl)sulfonyl]piperidineMus musculus (house mouse)Potency35.481310
2-[[[2-methyl-1-(phenylmethyl)-5-benzimidazolyl]amino]methyl]phenolMus musculus (house mouse)Potency17.900820
1-(4-chloro-3-methoxyphenyl)sulfonylazepaneMus musculus (house mouse)Potency0.562310
2-chloro-N-(5-methyl-3-isoxazolyl)acetamideMus musculus (house mouse)Potency18.996620
2-(3-benzamidophenoxy)acetic acidMus musculus (house mouse)Potency35.481310
6-ethoxy-2-[(4-fluorophenyl)methylthio]-1,3-benzothiazoleMus musculus (house mouse)Potency11.220210
2-(2-phenoxyethylsulfonyl)-1H-benzimidazoleMus musculus (house mouse)Potency35.481310
3-(1-azepanylazo)benzoic acidMus musculus (house mouse)Potency12.589310
4-[[7-bicyclo[4.1.0]heptanyl(oxo)methyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency10.000010
3-(4-fluoroanilino)-1-(3-nitrophenyl)-1-propanoneMus musculus (house mouse)Potency20.386620
4-[2-(4-methoxycarbonylphenyl)iminohydrazinyl]benzoic acid methyl esterMus musculus (house mouse)Potency0.158510
LSM-22807Mus musculus (house mouse)Potency28.370820
3-pentyl-4,5,6,7-tetrahydro-1H-indazoleMus musculus (house mouse)Potency10.000010
2-[[(6-bromo-1H-benzimidazol-2-yl)thio]methyl]-1-methylbenzimidazoleMus musculus (house mouse)Potency35.481310
3-bromo-N-[2-(4-nitroanilino)ethyl]benzamideMus musculus (house mouse)Potency10.000010
5-[[[(5-tert-butyl-2-methyl-3-furanyl)-oxomethyl]amino]methyl]-2-furancarboxylic acid ethyl esterMus musculus (house mouse)Potency20.895420
6-propan-2-yl-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency5.011910
4-chloro-N-(4-chloro-2,5-dimethoxyphenyl)-5-dithiazolimineMus musculus (house mouse)Potency30.300120
5-methoxy-3-methyl-1H-indole-2-carboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
tolfenamic acidMus musculus (house mouse)Potency15.848910
N-benzylquinazolin-4-amineMus musculus (house mouse)Potency8.912510
7-amino-2-methyl-3-phenyl-6-pyrazolo[1,5-a]pyrimidinecarbonitrileMus musculus (house mouse)Potency35.481320
edulineMus musculus (house mouse)Potency12.589310
6-methyl-2-(methylthio)-N-phenyl-5-prop-2-enyl-4-pyrimidinamineMus musculus (house mouse)Potency14.005320
4-(2-pyridinylthio)benzofuro[3,2-d]pyrimidineMus musculus (house mouse)Potency10.000010
4-(4-hydroxy-3,5-dimethylphenyl)-2-methylphthalazin-1(2H)-oneMus musculus (house mouse)Potency0.177810
acetic acid (3-hydroxy-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl) esterMus musculus (house mouse)Potency11.220210
2,3-diphenyl-6-quinoxalinecarboxylic acidMus musculus (house mouse)Potency5.011910
3-[6-(4-aminophenyl)-2-phenyl-4-pyrimidinyl]anilineMus musculus (house mouse)Potency22.387210
pirarubicin hydrochlorideMus musculus (house mouse)Potency19.952610
cinnamaldehydeMus musculus (house mouse)Potency12.589310
piplartineMus musculus (house mouse)Potency5.745720
fumaronitrileMus musculus (house mouse)Potency13.516020
7-methoxyisoflavoneMus musculus (house mouse)Potency4.466810
retinaldehydeMus musculus (house mouse)Potency23.350720
piperineMus musculus (house mouse)Potency5.623410
2'-hydroxychalconeMus musculus (house mouse)Potency35.481310
isoliquiritigeninMus musculus (house mouse)Potency12.594120
dibenzylidene acetoneMus musculus (house mouse)Potency27.717020
cardamoninMus musculus (house mouse)Potency8.912510
4'-methoxychalconeMus musculus (house mouse)Potency35.481310
xanthoangelolMus musculus (house mouse)Potency35.481310
cgp 60474Mus musculus (house mouse)Potency1.389120
N-(2-fluorophenyl)-2-(3-methoxyphenyl)imino-3-methyl-4-oxo-1,3-thiazinane-6-carboxamideMus musculus (house mouse)Potency35.481310
2-(2,4-dichlorophenoxy)-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency14.125410
2-[[3-methyl-7-(3-methylbutyl)-2,6-dioxo-8-purinyl]thio]propanoic acid methyl esterMus musculus (house mouse)Potency10.000010
N-[2-(1-cyclohexenyl)ethyl]-4-(4-morpholinylmethyl)benzamideMus musculus (house mouse)Potency7.079510
2-(3-chloro-4-methylphenyl)isoindole-1,3-dioneMus musculus (house mouse)Potency11.220210
1-(2-furanyl)-N-[[1-[(4-methylphenyl)sulfonylmethyl]-5-tetrazolyl]methyl]-N-(thiophen-2-ylmethyl)methanamineMus musculus (house mouse)Potency14.125410
N-(3,5-dimethoxyphenyl)-2-thiophenecarboxamideMus musculus (house mouse)Potency18.966220
2-[5-(4-butoxyphenyl)-2-tetrazolyl]-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency8.912510
LSM-34798Mus musculus (house mouse)Potency35.481310
3-amino-N-cyclopentyl-6-thiophen-2-yl-2-thieno[2,3-b]pyridinecarboxamideMus musculus (house mouse)Potency11.220210
1-(1-benzimidazolyl)-3-(1-cyclohex-3-enylmethoxy)-2-propanolMus musculus (house mouse)Potency23.350720
3-[(2-fluorophenyl)methyl]-7-(1-imidazolyl)triazolo[4,5-d]pyrimidineMus musculus (house mouse)Potency35.481310
N-(2-pyridinylmethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-9-amineMus musculus (house mouse)Potency7.079510
N-(3H-benzimidazol-5-yl)-2-furancarboxamideMus musculus (house mouse)Potency3.548110
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency1.412510
4-[[2-(1-benzotriazolyl)-1-oxoethyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency0.199510
4-chloro-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)benzamideMus musculus (house mouse)Potency0.295220
N-[1-[(4-methylphenyl)methyl]-2-benzimidazolyl]-2-furancarboxamideMus musculus (house mouse)Potency0.933420
7,8-dimethyl-1-[2-oxo-2-(1-pyrrolidinyl)ethyl]-4-phenyl-3H-1,5-benzodiazepin-2-oneMus musculus (house mouse)Potency11.220210
4-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-2-methyl-5-thieno[3,2-b]pyrrolecarboxylic acid ethyl esterMus musculus (house mouse)Potency22.387210
3-[[2-(1-benzotriazolyl)-1-oxoethyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency0.251210
3-methyl-4-(7-methyl-2-indolizinyl)-1,2,5-oxadiazoleMus musculus (house mouse)Potency35.481310
N-(1,3-benzodioxol-5-ylmethyl)-1-(6-ethyl-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-3-piperidinecarboxamideMus musculus (house mouse)Potency20.552320
2-(2-ethyl-6-methyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(5-methyl-2-furanyl)methyl]-N-(3-pyridinylmethyl)acetamideMus musculus (house mouse)Potency15.954120
6-ethyl-N-[2-(4-methoxyphenyl)ethyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineMus musculus (house mouse)Potency17.782810
N4-cyclohexyl-N1-ethyl-N4-(2-pyridinylmethyl)benzene-1,4-disulfonamideMus musculus (house mouse)Potency26.632020
2-[cyclohexyl-(2,4,6-trimethylphenyl)sulfonylamino]-N-(3-pyridinylmethyl)acetamideMus musculus (house mouse)Potency35.481310
5-methyl-N-[4-(4-morpholinyl)phenyl]-2-pyrazinecarboxamideMus musculus (house mouse)Potency5.623410
N-[2-methyl-4-oxo-3-(phenylmethyl)-7-(1-piperidinyl)-6-quinazolinyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency22.387210
1-(3-chloro-4-methoxyphenyl)sulfonyl-N-(3-pyridinyl)-3-piperidinecarboxamideMus musculus (house mouse)Potency20.483920
2-(4-bromophenyl)-5-(2-methylphenyl)-1,3,4-oxadiazoleMus musculus (house mouse)Potency2.818410
3-[[[1-[1-(2-furanylmethyl)-5-tetrazolyl]-2-methylpropyl]-(2-oxolanylmethyl)amino]methyl]-8-methyl-1H-quinolin-2-oneMus musculus (house mouse)Potency15.848910
2,6-diamino-4-(1-phenylethyl)-4H-thiopyran-3,5-dicarbonitrileMus musculus (house mouse)Potency28.934220
N-(4-fluorophenyl)-3-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]propanamideMus musculus (house mouse)Potency35.481310
N-[4-[[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]sulfonyl]phenyl]acetamideMus musculus (house mouse)Potency11.220210
N-(1,3-benzothiazol-2-yl)-N-methylbenzamideMus musculus (house mouse)Potency13.357420
6-methyl-3-[[[1-(phenylmethyl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneMus musculus (house mouse)Potency14.125410
4-[2-[1-(4-methoxyphenyl)sulfonyl-2-benzimidazolyl]ethyl]morpholineMus musculus (house mouse)Potency25.118910
3-[(2-chlorophenyl)methyl]-N-phenyl-7-triazolo[4,5-d]pyrimidinamineMus musculus (house mouse)Potency12.589310
2-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-2-azaspiro[5.5]undecaneMus musculus (house mouse)Potency35.481310
2-(1-benzimidazolylmethyl)-5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazoleMus musculus (house mouse)Potency16.717130
6-ethoxy-3-[[2-oxolanylmethyl-[[1-(2-phenylethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneMus musculus (house mouse)Potency12.589310
N-[1-methyl-5-(4-methylphenyl)-2-imidazolyl]-4-oxo-4-(1-piperidinyl)butanamideMus musculus (house mouse)Potency5.745720
N-[2-[2,3-dihydroindol-1-yl(oxo)methyl]phenyl]acetamideMus musculus (house mouse)Potency0.125910
5-(1,3-benzodioxol-5-yl)-1-methyl-2-imidazolamineMus musculus (house mouse)Potency0.035510
N-[4-[1-(benzenesulfonyl)-2,3-dihydroindol-5-yl]-2-thiazolyl]-2-(4-morpholinyl)acetamideMus musculus (house mouse)Potency25.118910
5-[2-(3,4-dimethoxyphenyl)ethylamino]-2-[(2-fluorophenoxy)methyl]-4-oxazolecarbonitrileMus musculus (house mouse)Potency14.125410
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-N-[2-(4-morpholinyl)phenyl]acetamideMus musculus (house mouse)Potency15.848910
2-[[5-(1-benzotriazolylmethyl)-1,3,4-oxadiazol-2-yl]thio]-N-[(4-fluorophenyl)methyl]-N-phenylacetamideMus musculus (house mouse)Potency12.191220
[3-[3-(5-methyl-2-furanyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]-phenylmethanoneMus musculus (house mouse)Potency2.511910
3-[[[1-(2-furanylmethyl)-5-tetrazolyl]methyl-[(2-methoxyphenyl)methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneMus musculus (house mouse)Potency35.481310
bikininMus musculus (house mouse)Potency0.562310
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]propanoic acid ethyl esterMus musculus (house mouse)Potency22.445020
1-(1,3-benzodioxol-5-ylmethyl)-3-(4-methylphenyl)-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]ureaMus musculus (house mouse)Potency19.952610
N'-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]-N'-(3-fluorophenyl)-N-(3-pyridinyl)butanediamideMus musculus (house mouse)Potency1.995310
2-(3,4-diethoxyphenyl)-5-(2-furanyl)-1,3,4-oxadiazoleMus musculus (house mouse)Potency7.079510
haplamineMus musculus (house mouse)Potency26.850910
N-tert-butyl-2-(2-furanyl)-2-[[2-[5-(5-methyl-2-furanyl)-2-tetrazolyl]-1-oxoethyl]-(thiophen-2-ylmethyl)amino]acetamideMus musculus (house mouse)Potency35.481310
N-[2-(4-methoxyphenyl)-1,3-benzoxazol-5-yl]-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency0.891310
2-methoxy-N-(5-thiophen-2-yl-1,3,4-thiadiazol-2-yl)acetamideMus musculus (house mouse)Potency4.466810
3-[[[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl-(2-hydroxyethyl)amino]methyl]-7-methyl-1H-quinolin-2-oneMus musculus (house mouse)Potency35.481310
N-[1-[2-(2-chlorophenoxy)ethyl]-2-benzimidazolyl]acetamideMus musculus (house mouse)Potency1.026620
N-(4-chlorophenyl)-4-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinecarboxamideMus musculus (house mouse)Potency35.481320
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-1-(1-piperidinyl)ethanoneMus musculus (house mouse)Potency12.924420
N-(2,5-diethoxyphenyl)-2-[(3-methyl-2-imidazo[4,5-b]pyridinyl)thio]acetamideMus musculus (house mouse)Potency19.952610
N-(3-dibenzofuranyl)-4-morpholinecarboxamideMus musculus (house mouse)Potency0.707910
N-[1-(2-methoxyphenyl)-5-benzimidazolyl]benzenesulfonamideMus musculus (house mouse)Potency7.079510
N-[1-[4-(4-methylphenyl)-2-thiazolyl]-4-piperidinyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideMus musculus (house mouse)Potency25.118910
N-[2-methoxy-4-[(2-methyl-1-oxopropyl)amino]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency0.354810
6-bromo-N-tert-butyl-2-methyl-3-imidazo[1,2-a]pyridinamineMus musculus (house mouse)Potency21.154620
4-[[4-ethyl-5-[(2-methylphenoxy)methyl]-1,2,4-triazol-3-yl]thio]-N-(2-methoxyphenyl)-3-oxobutanamideMus musculus (house mouse)Potency11.294720
N-butyl-N-[5-(3,4,5-trimethoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-furancarboxamideMus musculus (house mouse)Potency0.631010
4-bromo-N-[(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-hydroxyethyl)benzamideMus musculus (house mouse)Potency27.717020
N-(4-methylphenyl)-2-(3-oxo-5,6-dihydroimidazo[2,1-b]thiazol-2-yl)acetamideMus musculus (house mouse)Potency15.586420
4-methyl-N-(pyridin-4-ylmethyl)benzenesulfonamideMus musculus (house mouse)Potency7.417730
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneMus musculus (house mouse)Potency14.125410
6-amino-4-(2,5-dimethoxyphenyl)-3-methyl-1-(4-methylphenyl)-4H-pyrano[2,3-c]pyrazole-5-carbonitrileMus musculus (house mouse)Potency10.000010
N-cyclopropyl-4-(2,3-dihydroindol-1-ylsulfonyl)benzenesulfonamideMus musculus (house mouse)Potency12.589320
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideMus musculus (house mouse)Potency1.778310
N-[2-(2-ethyl-5-tetrazolyl)phenyl]-4-(1-tetrazolyl)benzamideMus musculus (house mouse)Potency0.005010
2-[(4-fluorophenoxy)methyl]-5-[3-(1-imidazolyl)propylamino]-4-oxazolecarbonitrileMus musculus (house mouse)Potency12.589310
N-(1,3-benzodioxol-5-yl)-2-[4-(4-phenyl-2-thiazolyl)-1-piperazinyl]acetamideMus musculus (house mouse)Potency35.481310
3-[(2-fluorophenyl)methyl]-5-propyl-N-(pyridin-4-ylmethyl)-7-triazolo[4,5-d]pyrimidinamineMus musculus (house mouse)Potency19.952610
2-[(2-ethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)thio]-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency11.220210
3-fluoro-N-[1-[2-[(2-fluorophenyl)methylamino]-2-oxoethyl]-4-piperidinyl]benzamideMus musculus (house mouse)Potency35.481310
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-[(3-methyl-2-imidazo[4,5-b]pyridinyl)thio]acetamideMus musculus (house mouse)Potency35.481320
1-(4-chlorophenyl)-N-(2-furanylmethyl)-N-[[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]methanamineMus musculus (house mouse)Potency35.481310
(2,4-difluorophenyl)-[3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]methanoneMus musculus (house mouse)Potency35.481320
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-methoxyacetamideMus musculus (house mouse)Potency14.125410
[4-[5-tert-butyl-3-[(2-chlorophenyl)methyl]-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneMus musculus (house mouse)Potency17.796820
3-chloro-4-[4-(4-fluorophenyl)sulfonyl-1-piperazinyl]-N,N-dimethylbenzenesulfonamideMus musculus (house mouse)Potency35.481310
(6-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-yl)-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]methanoneMus musculus (house mouse)Potency5.011910
3-[[(1-tert-butyl-5-tetrazolyl)methyl-(thiophen-2-ylmethyl)amino]methyl]-6-ethoxy-1H-quinolin-2-oneMus musculus (house mouse)Potency17.776020
N-(2-furanylmethyl)-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]benzamideMus musculus (house mouse)Potency7.943310
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneMus musculus (house mouse)Potency35.481320
2-(3-oxo-1-(toluene-4-sulfonyl)-1,2,3,4-4h-quinoxalin-2-yl)-n-phenyl-acetamideMus musculus (house mouse)Potency22.387210
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2-pyrimidinyl)-3-piperidinecarboxamideMus musculus (house mouse)Potency22.387220
2-[(2-cyclohexyl-4-quinazolinyl)thio]-N-(4-methyl-1,2,5-oxadiazol-3-yl)acetamideMus musculus (house mouse)Potency8.285220
N-[2-[2-[2-(4-methoxyanilino)-2-oxoethyl]-5-tetrazolyl]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency35.481320
2-[(3-cyano-5,7-dimethyl-2-quinolinyl)thio]-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency24.035320
6-[(2-fluorophenyl)methyl]-2,4-dimethyl-5-thieno[3,4]pyrrolo[1,3-d]pyridazinoneMus musculus (house mouse)Potency25.118910
1-phenyl-4-[[1-(phenylmethyl)-5-tetrazolyl]-(3-pyridinyl)methyl]piperazineMus musculus (house mouse)Potency35.481310
3-[[1-[1-(2-furanylmethyl)-5-tetrazolyl]propyl-(2-phenylethyl)amino]methyl]-7-methoxy-1H-quinolin-2-oneMus musculus (house mouse)Potency11.220210
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[[5-[(3-methylphenoxy)methyl]-1,3,4-oxadiazol-2-yl]thio]acetamideMus musculus (house mouse)Potency35.481310
N-(2-furanylmethyl)-N-[(7-methyl-4-tetrazolo[1,5-a]quinolinyl)methyl]-2-phenoxyacetamideMus musculus (house mouse)Potency10.000010
5-amino-2-(4-methylphenyl)isoindole-1,3-dioneMus musculus (house mouse)Potency2.511910
9-oxo-N-(3-pyridinylmethyl)-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinoline-8-carboxamideMus musculus (house mouse)Potency25.118910
N-[4-(2-methyl-1-methylsulfonyl-2,3-dihydroindol-5-yl)-2-thiazolyl]-2-thiophen-2-ylacetamideMus musculus (house mouse)Potency30.300120
4-amino-N5-[1-(2-furanyl)-2-(3-methylbutylamino)-2-oxoethyl]-N5-(2-methoxyphenyl)isothiazole-3,5-dicarboxamideMus musculus (house mouse)Potency22.387210
N-[3-chloro-4-(4-morpholinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency0.811620
2-[[1-(4-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]thio]acetic acid ethyl esterMus musculus (house mouse)Potency35.481310
N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]butanamideMus musculus (house mouse)Potency35.481310
5-[(2-fluoroanilino)methyl]-8-quinolinolMus musculus (house mouse)Potency16.193620
2-(4,5-dihydrothiazol-2-ylthio)-N-(6-methoxy-1,3-benzothiazol-2-yl)acetamideMus musculus (house mouse)Potency15.848910
4-[[4-(1,3-benzothiazol-2-yl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-2-methoxyphenolMus musculus (house mouse)Potency35.481310
N,N-dimethyl-4-[[4-(5-methyl-1-benzotriazolyl)-1-piperidinyl]sulfonyl]benzamideMus musculus (house mouse)Potency11.220210
1-(4-chlorophenyl)-2-[[4-ethyl-5-(2-methyl-3-furanyl)-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency33.552020
polidocanolMus musculus (house mouse)Potency35.481310
(1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanolMus musculus (house mouse)Potency25.665120
dithizoneMus musculus (house mouse)Potency28.183810
phenytoin sodiumMus musculus (house mouse)Potency35.481310
r 59949Mus musculus (house mouse)Potency23.350720
2-(3,5-dimethyl-1-pyrazolyl)-N,6-dimethyl-4-pyrimidinamineMus musculus (house mouse)Potency1.571420
2-amino-7-cyclohexyl-6,8-dioxo-4,5,5a,8a-tetrahydrothieno[2,3-e]isoindole-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
5-ethyl-4,6-dimethyl-2-sulfanylidene-1H-pyridine-3-carbonitrileMus musculus (house mouse)Potency28.934220
3-(4-butyl-3,5-dimethyl-1-pyrazolyl)-5-methyl-[1,2,4]triazino[5,6-b]indoleMus musculus (house mouse)Potency3.936920
6-amino-4-(5-bromo-2-thiophenyl)-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMus musculus (house mouse)Potency23.350720
8-(2-furanyl)-6-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3,3-dimethyl-1,4-dihydrothiopyrano[3,4-c]pyridine-5-carbonitrileMus musculus (house mouse)Potency14.125410
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3,3,3-trifluoro-2-methyl-2-(trifluoromethyl)propanamideMus musculus (house mouse)Potency30.300120
5-bromo-3-[[2-(4-cyclohexyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterMus musculus (house mouse)Potency35.481310
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideMus musculus (house mouse)Potency2.129520
5-chloro-3-[[2-(4-ethoxycarbonyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterMus musculus (house mouse)Potency12.863120
3-(5-cycloheptylidene-4-oxo-2-sulfanylidene-3-thiazolidinyl)propanoic acidMus musculus (house mouse)Potency14.125410
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2,2-bis(trifluoromethyl)butanamideMus musculus (house mouse)Potency12.924420
(1-methyl-2-imidazolyl)-(4-phenylmethoxyphenyl)methanolMus musculus (house mouse)Potency35.481310
1-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaMus musculus (house mouse)Potency35.481310
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaMus musculus (house mouse)Potency4.280020
4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl esterMus musculus (house mouse)Potency35.481310
2-cyano-N-(2-furanylmethyl)-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetamideMus musculus (house mouse)Potency15.848910
2-[[3-cyano-4-(2-furanyl)-5,6,7,8-tetrahydroquinolin-2-yl]thio]-N-(2-methylphenyl)acetamideMus musculus (house mouse)Potency5.623410
3-[[2-[4-(3-chlorophenyl)-1-piperazinyl]-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterMus musculus (house mouse)Potency35.481310
8-methyl-6-(3-methyl-2-thiophenyl)-4-oxo-3,6-dihydro-2H-pyrimido[2,1-b][1,3]thiazine-7-carboxylic acid ethyl esterMus musculus (house mouse)Potency19.952610
N-cyano-N'-propan-2-ylcarbamimidothioic acid [2-(2-methoxyanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency35.481310
4-[1-(4-hydroxyphenyl)ethenyl]phenolMus musculus (house mouse)Potency35.481310
2-(2,4-dioxo-3-phenyl-5-thiazolidinyl)-N-phenylacetamideMus musculus (house mouse)Potency35.481320
2-ethyl-1-[(2-methoxyphenyl)methyl]benzimidazoleMus musculus (house mouse)Potency21.280420
N-[2-(1-cyclohexenyl)ethyl]-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineMus musculus (house mouse)Potency0.141310
2-(4-chlorophenyl)-5-(methylamino)-4-oxazolecarbonitrileMus musculus (house mouse)Potency0.354810
1-phenyl-N-(3-propan-2-yloxypropyl)-4-pyrazolo[3,4-d]pyrimidinamineMus musculus (house mouse)Potency12.863120
2-[2-[[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]amino]ethoxy]ethanolMus musculus (house mouse)Potency0.398110
3-(3,5-dimethoxyphenyl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency19.118020
N-[5-[[2-(4-methylanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-2-(4-morpholinyl)acetamideMus musculus (house mouse)Potency35.481310
2-(butylamino)-N-[4-[5-[[2-(butylamino)-1-oxoethyl]amino]-1,3-benzoxazol-2-yl]phenyl]acetamideMus musculus (house mouse)Potency3.162310
2-[[2-methyl-5-(3-methyl-4-oxo-1-phthalazinyl)phenyl]sulfonylamino]acetic acid ethyl esterMus musculus (house mouse)Potency0.354810
7-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxoethyl]amino]-5H-[1,3]dioxolo[4,5-f]indole-6-carboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
N-(3-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideMus musculus (house mouse)Potency30.300120
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenolMus musculus (house mouse)Potency17.782810
2-(4-chlorophenyl)-3-(2-furanylmethyl)imidazo[4,5-b]quinoxalineMus musculus (house mouse)Potency14.125410
2-[[4-amino-5-(4-tert-butylphenyl)-1,2,4-triazol-3-yl]thio]acetic acid propan-2-yl esterMus musculus (house mouse)Potency26.632020
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.738420
5-bromo-N-(2-pyridinylmethyl)-2-thiophenesulfonamideMus musculus (house mouse)Potency14.432620
2-[5-[(2-chlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineMus musculus (house mouse)Potency25.665120
2-[5-[(2,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineMus musculus (house mouse)Potency35.481320
2-(3,5-dimethyl-1-pyrazolyl)-4-(4-morpholinyl)-5-pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency11.220210
8-[4-(3-chlorophenyl)-1-piperazinyl]-3-methyl-7-pentylpurine-2,6-dioneMus musculus (house mouse)Potency35.481310
2-[5-[(4-bromophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineMus musculus (house mouse)Potency24.803320
5-[(2-chlorophenyl)methylamino]-2-(3,4-dimethoxyphenyl)-4-oxazolecarbonitrileMus musculus (house mouse)Potency8.912510
4-(1H-benzimidazol-2-ylmethylthio)-2-methylbenzofuro[3,2-d]pyrimidineMus musculus (house mouse)Potency24.803320
N-[3-(2-phenylethyl)-2,4-dihydro-1H-1,3,5-triazin-6-yl]-1,3-benzoxazol-2-amineMus musculus (house mouse)Potency3.548110
cp 84364Mus musculus (house mouse)Potency5.011910
LSM-28231Mus musculus (house mouse)Potency8.912510
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dioneMus musculus (house mouse)Potency25.665120
1-[(4-fluorophenyl)methyl]-3-(2-furanylmethyl)-4-imino-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-2-oneMus musculus (house mouse)Potency2.238710
N-(1-ethyl-6-methyl-3-pyrazolo[3,4-b]quinolinyl)-4-pyridinecarboxamideMus musculus (house mouse)Potency0.501210
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterMus musculus (house mouse)Potency14.733420
N-[5-(4-chlorophenyl)-7-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-furancarboxamideMus musculus (house mouse)Potency0.433220
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanolMus musculus (house mouse)Potency2.201620
LSM-32568Mus musculus (house mouse)Potency19.952610
3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpropanamideMus musculus (house mouse)Potency3.697820
N-(5-methyl-7-phenyl-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-2-thiophenecarboxamideMus musculus (house mouse)Potency18.256320
3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(3-methylphenyl)propanamideMus musculus (house mouse)Potency5.140920
2-[[2-(3,5-dimethyl-1-pyrazolyl)-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-4-yl]thio]-N-(2-thiazolyl)acetamideMus musculus (house mouse)Potency14.550020
2-amino-4-(2-furanyl)-6-(2-pyridinyl)-3-pyridinecarbonitrileMus musculus (house mouse)Potency10.610120
3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]-N-ethylpropanamideMus musculus (house mouse)Potency2.237260
2-[(2,5-dimethyl-3-phenyl-7-pyrazolo[1,5-a]pyrimidinyl)thio]acetonitrileMus musculus (house mouse)Potency1.885420
N-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-2-thiophenecarboxamideMus musculus (house mouse)Potency35.481310
[2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl]-(1-pyrrolidinyl)methanoneMus musculus (house mouse)Potency4.466810
N5,N5-dimethyl-2,1,3-benzoxadiazole-4,5-diamineMus musculus (house mouse)Potency31.622810
7-methyl-3-(3-methylbutylamino)-1-(1-pyrrolidinyl)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileMus musculus (house mouse)Potency13.534620
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-bis(phenylmethyl)-2,4-dihydro-1,3,5-triazin-6-amineMus musculus (house mouse)Potency20.386620
7-(3,4-dimethoxyphenyl)-4-methyl-2-[4-(phenylmethyl)-1-piperazinyl]-7,8-dihydro-6H-quinazolin-5-oneMus musculus (house mouse)Potency15.848910
N-[1-methyl-2-[2-(4-phenyl-1-piperazinyl)ethyl]-5-benzimidazolyl]-2-furancarboxamideMus musculus (house mouse)Potency7.943310
5-(3-methoxyphenyl)-N-(2-oxolanylmethyl)-7-(trifluoromethyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideMus musculus (house mouse)Potency22.387210
3-(1-benzotriazolylmethyl)-6-(2-phenylethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleMus musculus (house mouse)Potency14.125410
1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-2-phenyl-1-butanoneMus musculus (house mouse)Potency35.481310
N-[2-(2-benzamidoethyl)-1-methyl-5-benzimidazolyl]-2-furancarboxamideMus musculus (house mouse)Potency15.848910
2-methoxy-6-[[(1-propyl-5-benzimidazolyl)amino]methyl]phenolMus musculus (house mouse)Potency35.481320
8-methoxy-5-methyl-3-[2-(1-pyrrolidinyl)ethyl]-4-pyrimido[5,4-b]indoloneMus musculus (house mouse)Potency0.100010
5-[(2-chloro-6-fluorophenyl)methyl]-N-[2-[4-(4-methoxyphenyl)-1-piperazinyl]ethyl]-1,3,4-oxadiazole-2-carboxamideMus musculus (house mouse)Potency35.481310
1-(4-fluorophenyl)-2-[[4-(2-furanylmethyl)-5-(phenoxymethyl)-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency25.665120
3-(2,3-dihydro-1,4-benzodioxin-3-yl)-6-(4-fluorophenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleMus musculus (house mouse)Potency35.481310
ethoxydMus musculus (house mouse)Potency12.062710
methisazoneMus musculus (house mouse)Potency2.142220
dexketoprofenMus musculus (house mouse)Potency31.832620
4-cyclohexyl-3-[(3-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.026620
4-methoxy-N-(5-methyl-3-isoxazolyl)benzamideMus musculus (house mouse)Potency25.118910
2,4-difluoro-N-[[(5-methyl-1H-pyrazol-3-yl)amino]-oxomethyl]benzamideMus musculus (house mouse)Potency17.015720
4-amino-3-methyl-N-(phenylmethyl)-2-sulfanylidene-5-thiazolecarboxamideMus musculus (house mouse)Potency14.125410
5-[(1,3-benzothiazol-2-ylthio)methyl]-2-furancarboxylic acid methyl esterMus musculus (house mouse)Potency10.000010
dichloramine-tMus musculus (house mouse)Potency6.309610
N-[4-(diethylamino)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency15.848920
N-(2-furanylmethyl)-2-benzofurancarboxamideMus musculus (house mouse)Potency3.162310
1-[1-(4-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-(4-methyl-1-piperidinyl)ethanoneMus musculus (house mouse)Potency22.740620
4-ethyl-5-(4-fluorophenyl)-2,4-dihydro-3h-1,2,4-triazole-3-thioneMus musculus (house mouse)Potency1.558620
te 5Mus musculus (house mouse)Potency22.387210
4-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamideMus musculus (house mouse)Potency10.000010
(e)-3-(4-t-butylphenyl)-n-(2,3-dihydrobenzo(b)(1,4)dioxin-6-yl)acrylamideMus musculus (house mouse)Potency17.900820
2-[[anilino(oxo)methyl]amino]-4,5-dimethyl-3-thiophenecarboxamideMus musculus (house mouse)Potency1.122010
N-(4-fluorophenyl)-4-methyl-1-piperidinecarbothioamideMus musculus (house mouse)Potency25.665120
3-[[2-benzofuranyl(oxo)methyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency24.035320
2-(4-bromophenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency8.912510
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency3.548110
5-(1,3-benzodioxol-5-yl)-2-[(2-chloro-6-fluorophenyl)methyl]tetrazoleMus musculus (house mouse)Potency0.501210
1-(1,3-benzodioxol-5-ylmethyl)-3-(4-methylphenyl)thioureaMus musculus (house mouse)Potency14.219120
1-ethyl-5-(phenylmethyl)-1,3,5-triazinane-2-thioneMus musculus (house mouse)Potency12.589320
levosulpirideMus musculus (house mouse)Potency35.481320
3,4'-dihydroxyflavoneMus musculus (house mouse)Potency7.943310
6-methylflavoneMus musculus (house mouse)Potency24.803320
caffeic acidMus musculus (house mouse)Potency12.589310
5-(4-chlorophenyl)-4h-1,2,4-triazole-3-thiolMus musculus (house mouse)Potency8.912510
5-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazole-3-thioneMus musculus (house mouse)Potency22.740620
isatin beta-thiosemicarbazoneMus musculus (house mouse)Potency19.952610
3-(4-methylbenzoyl)acrylic acidMus musculus (house mouse)Potency9.581820
N-[(2-phenylethylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency18.623120
2-chloro-N-(2-phenylethyl)benzamideMus musculus (house mouse)Potency8.427920
4-[4-[cyclohexyloxy(oxo)methyl]anilino]-4-oxobutanoic acidMus musculus (house mouse)Potency17.782820
2-(8-quinolinylthio)acetic acidMus musculus (house mouse)Potency17.782810
N-[2-(1-cyclohexenyl)ethyl]-4-fluorobenzamideMus musculus (house mouse)Potency11.220220
4-cyclohexyl-3-(3-pyridinyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency21.450920
4-cyclohexyl-3-(4-methoxyphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency5.120920
6-(2-methyl-3-benzofuranyl)-2,3-dihydroimidazo[2,1-b]thiazoleMus musculus (house mouse)Potency35.481320
N4-(3-chlorophenyl)-6-methyl-N2-(phenylmethyl)pyrimidine-2,4-diamineMus musculus (house mouse)Potency22.016420
N-(2-furanylmethyl)-4-(2-methyl-3-imidazo[1,2-a]pyridinyl)-2-thiazolamineMus musculus (house mouse)Potency23.350720
captaxMus musculus (house mouse)Potency6.482820
aeg 3482Mus musculus (house mouse)Potency33.552020
2-(4-ethylphenoxy)-N-(1H-1,2,4-triazol-5-yl)acetamideMus musculus (house mouse)Potency0.891310
iFSP1Mus musculus (house mouse)Potency13.516020
2-[(4-chloro-2-methylphenoxy)methyl]imidazo[1,2-a]pyrimidineMus musculus (house mouse)Potency1.778310
6-bromo-5-hydroxy-2-methyl-1H-indole-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency5.623410
5,6-diphenyl-1,2,4-triazine-3-thiolMus musculus (house mouse)Potency8.912510
diphenylthioureaMus musculus (house mouse)Potency14.987220
5-(5-chloro-2-methoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneMus musculus (house mouse)Potency35.481310
N-[(4-pyrimidinylthio)methyl]benzamideMus musculus (house mouse)Potency22.387210
4-chloro-1-methyl-3-nitro-2-quinolinoneMus musculus (house mouse)Potency11.294720
3,5,5-trimethyl-2-sulfanylidene-1,6-dihydrobenzo[h]quinazolin-4-oneMus musculus (house mouse)Potency0.398110
nitrofurylacrylic acidMus musculus (house mouse)Potency11.220210
5-(4-chlorophenyl)-3H-thieno[2,3-d]pyrimidine-4-thioneMus musculus (house mouse)Potency0.723320
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
ceefourin 1Mus musculus (house mouse)Potency7.079510
N-(4-hydroxy-2-methyl-5-propan-2-ylphenyl)-4-methoxybenzenesulfonamideMus musculus (house mouse)Potency25.665120
2-(3,4-dichlorophenyl)imidazo[1,2-a]pyrimidineMus musculus (house mouse)Potency1.584910
5-(2-phenyl-4-triazolyl)-2H-tetrazoleMus musculus (house mouse)Potency4.466810
1-(2-methoxyphenyl)-3-(2-pyridinyl)thioureaMus musculus (house mouse)Potency2.566520
4-(3-chlorophenyl)thiosemicarbazideMus musculus (house mouse)Potency15.165220
N-[2-(1H-benzimidazol-2-yl)ethyl]-4-chloro-3-nitrobenzamideMus musculus (house mouse)Potency5.011910
N-[(3-nitroanilino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency2.511910
4-(benzylsulfanyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency35.481310
5-methyl-6-phenyl-3H-thieno[2,3-d]pyrimidine-4-thioneMus musculus (house mouse)Potency0.750620
2-mercaptobenzoxazoleMus musculus (house mouse)Potency28.183810
3-[(2,4-dichlorophenyl)methylthio]-1,2,4-thiadiazol-5-amineMus musculus (house mouse)Potency11.220210
6-(chloromethyl)-N2-(2,5-dimethoxyphenyl)-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency35.481310
2-(3-oxo-2-phenyl-1H-pyrazol-5-yl)acetic acid methyl esterMus musculus (house mouse)Potency0.158510
1-(3,4-dihydroxyphenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)thio]ethanoneMus musculus (house mouse)Potency12.589310
4-(4-chlorophenyl)-3-(2-quinolinyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.267320
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileMus musculus (house mouse)Potency25.665120
4-chloro-N-(3,4,5-trimethoxyphenyl)-5-dithiazolimineMus musculus (house mouse)Potency25.665120
5-(2,3-dihydro-1H-inden-5-yloxymethyl)-2-furancarbohydrazideMus musculus (house mouse)Potency24.803320
5-[(4-ethylphenoxy)methyl]-N-(2-pyridinylmethyl)-2-furancarboxamideMus musculus (house mouse)Potency17.782810
N-(5-methyl-3-isoxazolyl)-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency12.589320
N-(2-chlorophenyl)hydrazine-1-carbothioamideMus musculus (house mouse)Potency9.581820
10-methyl-3-phenothiazinamineMus musculus (house mouse)Potency17.782810
4-[[[2-(4-fluorophenyl)ethylamino]-sulfanylidenemethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency17.559420
N-(2-furanylmethyl)-4-methyl-N-(phenylmethyl)benzenesulfonamideMus musculus (house mouse)Potency35.481310
1-ethyl-2-[[(1-methyl-2-benzimidazolyl)thio]methyl]benzimidazoleMus musculus (house mouse)Potency25.118910
vu0038882Mus musculus (house mouse)Potency10.217520
5-cyano-2-methyl-6-sulfanylidene-1H-pyridine-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency12.589310
3-cyclohexyl-1,1-bis(2-methylpropyl)thioureaMus musculus (house mouse)Potency4.949020
2-anilino-N-(4-fluorophenyl)acetamideMus musculus (house mouse)Potency0.891310
4-[[2-furanyl(oxo)methyl]amino]benzoic acid propan-2-yl esterMus musculus (house mouse)Potency1.995310
1-cyclohexyl-3-[[oxo(thiophen-2-yl)methyl]amino]thioureaMus musculus (house mouse)Potency1.412510
2-amino-4-(cyanomethyl)-6-(N-methylanilino)pyridine-3,5-dicarbonitrileMus musculus (house mouse)Potency11.220210
N-(4-anilinophenyl)cyclopropanecarboxamideMus musculus (house mouse)Potency35.481310
4-hydroxy-1-(4-methylphenyl)-3-pyrazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency3.981110
1-(2-furanyl)-2-([1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-ylthio)ethanoneMus musculus (house mouse)Potency14.125410
2-(thiophen-2-ylmethylidene)indene-1,3-dioneMus musculus (house mouse)Potency7.079510
1-(2,5-dimethoxyphenyl)-3-phenylthioureaMus musculus (house mouse)Potency19.952620
1-(4-chlorophenyl)-3-(4-sulfamoylphenyl)ureaMus musculus (house mouse)Potency18.854120
3-methyl-N-(2-phenylethyl)-2-butenamideMus musculus (house mouse)Potency11.220210
N-[4-(diethylamino)phenyl]-N'-phenylureaMus musculus (house mouse)Potency15.848910
4-bromo-N-phenacylbenzamideMus musculus (house mouse)Potency12.589310
4-bromo-2-phenyl-5-(1-piperidinyl)-3-pyridazinoneMus musculus (house mouse)Potency12.589310
N-[4-(4-ethylphenyl)-2-thiazolyl]carbamic acid phenyl esterMus musculus (house mouse)Potency11.557420
1-(2,3-dihydroindol-1-yl)-2-(phenylthio)ethanoneMus musculus (house mouse)Potency0.199510
krm iiiMus musculus (house mouse)Potency10.000020
N-[6-methyl-2-(4-methylphenyl)-5-benzotriazolyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency2.787120
1-(3-fluorophenyl)-3-(2-pyridinylmethyl)thioureaMus musculus (house mouse)Potency0.794310
N-[[(5-chloro-2-pyridinyl)amino]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency2.733420
N-[[(6-methyl-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency2.142220
2-(4-hydroxyanilino)-1,4-naphthoquinoneMus musculus (house mouse)Potency35.481310
N-(3,4,5,6-tetrahydro-2H-azepin-7-yl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency0.281810
2-(2-bromo-4-methylphenoxy)-N-(2-pyridinylmethyl)acetamideMus musculus (house mouse)Potency3.548110
1-(4-methoxyphenyl)-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ureaMus musculus (house mouse)Potency0.891310
1-cyclohexyl-3-(2-phenylethyl)ureaMus musculus (house mouse)Potency10.000020
1-(3,5-dichlorophenyl)-3-phenylureaMus musculus (house mouse)Potency27.717020
acetic acid [4-[oxo-(2-phenylethylamino)methyl]phenyl] esterMus musculus (house mouse)Potency27.717020
N-(3-methoxyphenyl)-2-benzo[cd]indolamineMus musculus (house mouse)Potency26.632020
4-[2-(1-methyl-2-benzimidazolyl)ethyl]anilineMus musculus (house mouse)Potency13.534620
3-pyridinecarboxylic acid (5-chloro-8-quinolinyl) esterMus musculus (house mouse)Potency0.945620
acetic acid (4-oxo-3-phenyl-1-benzopyran-7-yl) esterMus musculus (house mouse)Potency5.623410
N-phenyl-4-pyridin-4-yl-2-thiazolamineMus musculus (house mouse)Potency35.481310
N-(phenylmethyl)-4-(3-pyridinyl)-2-thiazolamineMus musculus (house mouse)Potency7.943310
N-(4-hydroxy-2-methyl-5-propan-2-ylphenyl)benzenesulfonamideMus musculus (house mouse)Potency35.481310
N-(3-chloro-4-hydroxy-2,5-dimethylphenyl)benzenesulfonamideMus musculus (house mouse)Potency25.665120
2-[[(4-chlorophenyl)thio]methyl]imidazo[1,2-a]pyridineMus musculus (house mouse)Potency8.912510
4-(2,5-dimethylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency10.000010
N-(4-methoxyphenyl)carbamic acid (9-fluorenylideneamino) esterMus musculus (house mouse)Potency6.309610
N2,N4-ditert-butyl-6-hydrazinyl-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency13.516020
N-(2,6-dimethoxy-4-pyrimidinyl)-3-phenylpropanamideMus musculus (house mouse)Potency3.981110
nsc185058Mus musculus (house mouse)Potency4.238020
2-[(2-fluorophenyl)methylthio]-5-(4-methylphenyl)-1,3,4-oxadiazoleMus musculus (house mouse)Potency22.106020
2-ethoxy-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.400020
2-furancarboxylic acid (7-methyl-4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-9-yl) esterMus musculus (house mouse)Potency22.387210
1-(2-methoxyphenyl)-5-(phenylmethyl)-1,3,5-triazinane-2-thioneMus musculus (house mouse)Potency18.738320
5-ethyl-1-(phenylmethyl)-1,3,5-triazinane-2-thioneMus musculus (house mouse)Potency19.118020
2-[(2-methoxyphenoxy)methyl]-1H-benzimidazoleMus musculus (house mouse)Potency11.220210
2,2,2-trifluoro-N-(2-methyl-8-quinolinyl)acetamideMus musculus (house mouse)Potency6.309610
3-(4-chlorophenyl)-2,5-dimethyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneMus musculus (house mouse)Potency11.464220
4-(4-(4-chloro-phenyl)thiazol-2-ylamino)phenolMus musculus (house mouse)Potency20.275620
N'-[(4-chlorophenyl)-oxomethyl]-2-pyrazinecarbohydrazideMus musculus (house mouse)Potency12.380720
cid755673Mus musculus (house mouse)Potency3.981110
2-fluoro-N-phenacylbenzamideMus musculus (house mouse)Potency23.350720
2-hydroxy-2,2-bis(4-methylphenyl)-N'-(2-pyridinyl)acetohydrazideMus musculus (house mouse)Potency22.740620
2-(4-chlorophenyl)-5-(4-fluorophenyl)-1,3,4-oxadiazoleMus musculus (house mouse)Potency0.446710
1-(3-pyridinylmethyl)-3-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]ureaMus musculus (house mouse)Potency22.740620
3-(2,3-dimethyl-1H-indol-5-yl)-4-methyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency16.803720
N-(4-anilinophenyl)-2,2,2-trichloroacetamideMus musculus (house mouse)Potency31.622810
3-(4-bromophenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneMus musculus (house mouse)Potency14.432620
2-(1,3-benzothiazol-2-ylmethoxy)phenolMus musculus (house mouse)Potency2.511910
3-(2-phenoxyethyl)-1H-benzimidazole-2-thioneMus musculus (house mouse)Potency2.818410
2,4,6-trimethyl-n-(meta-3-trifluoromethylphenyl)benzenesulfonamideMus musculus (house mouse)Potency22.874120
N-[4-[oxo(1-piperidinyl)methyl]phenyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency14.125410
5,7-dimethyl-2-(4-methylphenyl)pyrazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency7.079510
3-hydroxypyridine, sodium saltMus musculus (house mouse)Potency35.481310
3-(4-methylphenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneMus musculus (house mouse)Potency1.258910
2-(1H-benzimidazol-2-ylthio)-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamideMus musculus (house mouse)Potency28.934220
4-[(1H-benzimidazol-2-ylthio)methyl]-2-thiazolamineMus musculus (house mouse)Potency35.481320
N-[[(2-chloro-3-pyridinyl)amino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency22.387210
N-[2-(1-cyclohexenyl)ethyl]-2,5-dimethoxybenzenesulfonamideMus musculus (house mouse)Potency17.585520
3-[(4-methylphenoxy)methyl]-4-phenyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.648620
4-(4-chlorophenyl)-3-[(4-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency3.162310
1-(4,5-dihydrothiazol-2-yl)-3-phenylureaMus musculus (house mouse)Potency35.481320
3-[2-(4-methyl-2-propan-2-ylphenoxy)ethyl]-1H-benzimidazole-2-thioneMus musculus (house mouse)Potency3.764620
4-amino-N-(2-furanyl)benzamideMus musculus (house mouse)Potency0.398110
1-methyl-4-[(4-methylphenyl)thio]-3-nitro-2-quinolinoneMus musculus (house mouse)Potency9.149820
4-(6-methyl-4-phenyl-2-quinazolinyl)-1-piperazinecarboxaldehydeMus musculus (house mouse)Potency0.158510
3-(4-ethoxyphenyl)-1H-pyrazole-5-carbohydrazideMus musculus (house mouse)Potency1.000010
[3-fluoro-4-(4-morpholinyl)phenyl]-(4-methylphenyl)methanoneMus musculus (house mouse)Potency22.740620
1-[4-(1-azepanyl)-3-fluorophenyl]-1-propanoneMus musculus (house mouse)Potency28.183810
1-(1,3-benzodioxol-5-ylmethyl)-3-(2,1,3-benzothiadiazol-5-yl)thioureaMus musculus (house mouse)Potency35.481320
2-(8-quinolinylthio)acetic acid phenacyl esterMus musculus (house mouse)Potency35.481310
N-(4-methoxyphenyl)-3,4-dihydroquinolin-2-amineMus musculus (house mouse)Potency25.118910
4-methyl-N-[1-[2-(1-pyrrolidinyl)ethyl]-2-benzimidazolyl]benzamideMus musculus (house mouse)Potency4.795720
1-(3-nitrophenyl)-3-phenyl-2-propyn-1-oneMus musculus (house mouse)Potency5.966520
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazineMus musculus (house mouse)Potency5.629420
n-benzamidothioureaMus musculus (house mouse)Potency12.602820
1-spiro[2,4-dihydroisoquinoline-3,1'-cyclohexane]thioneMus musculus (house mouse)Potency10.537320
4-tert-butyl-N-[2-(2-methoxyphenyl)ethyl]-1-cyclohexanamineMus musculus (house mouse)Potency1.122010
6-(4-morpholinyl)naphthalene-2,3-dicarbonitrileMus musculus (house mouse)Potency28.183810
2-(1-methyl-2-phenyl-3-indolyl)ethanolMus musculus (house mouse)Potency25.118910
4-chloro-N-(4-methyl-2-thiazolyl)-2-nitrobenzamideMus musculus (house mouse)Potency35.481310
2-[[acetamido(sulfanylidene)methyl]amino]-5-ethyl-3-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency19.974020
5-[2-(5-methoxycarbonyl-2-thiophenyl)butan-2-yl]-2-thiophenecarboxylic acid methyl esterMus musculus (house mouse)Potency35.481310
2-(phenylmethylthio)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoleMus musculus (house mouse)Potency10.000020
5-methyl-N-(4,5,6-trimethyl-2-pyrimidinyl)-1,3-benzoxazol-2-amineMus musculus (house mouse)Potency1.258910
4-(4-morpholinyl)-N-(pyridin-4-ylmethyl)anilineMus musculus (house mouse)Potency25.118910
1-[[2-(3-methylanilino)-1-oxoethyl]amino]-3-phenylthioureaMus musculus (house mouse)Potency23.350720
N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-5-nitro-2-furancarboxamideMus musculus (house mouse)Potency35.481310
4-acetamido-N-(2-phenylethyl)benzamideMus musculus (house mouse)Potency3.981110
[5-(4-nitrophenyl)-2-furanyl]-(1-piperidinyl)methanoneMus musculus (house mouse)Potency25.665120
3-ethoxy-N-(2-thiazolyl)benzamideMus musculus (house mouse)Potency28.934220
1-[[3-(4-chlorophenoxy)phenyl]methyl]-4-ethylpiperazineMus musculus (house mouse)Potency19.952610
4-cyano-3-methyl-5-(4-methylphenyl)-2-thiophenecarbohydrazideMus musculus (house mouse)Potency5.773220
N4,N4-dimethyl-N1-(4-nitro-1,1-dioxo-2,5-dihydrothiophen-3-yl)benzene-1,4-diamineMus musculus (house mouse)Potency13.699620
3-(5-methoxy-2,2-dimethyl-1-benzopyran-8-yl)-3-oxopropanoic acidMus musculus (house mouse)Potency19.952610
N-[4-(1-azepanyl)phenyl]-2-chloroacetamideMus musculus (house mouse)Potency27.005020
2,4-dimethoxy-n-naphthalen-2-yl-benzamideMus musculus (house mouse)Potency35.481310
1-(1,3-benzodioxol-5-ylmethyl)-3-(2-methylphenyl)thioureaMus musculus (house mouse)Potency6.256020
N-(3-methoxyphenyl)-4-(phenylmethyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency19.952620
N-[[(4,6-dimethyl-2-pyrimidinyl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency29.903320
9-ethyl-1,2,4,5-tetrazaspiro[5.5]undecane-3-thioneMus musculus (house mouse)Potency24.035320
3-[[(2,5-dimethyl-3-furanyl)-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency35.481310
1-(4-ethoxyphenyl)-3-(6-quinoxalinyl)ureaMus musculus (house mouse)Potency11.220210
1,3-bis(2-phenylethyl)thioureaMus musculus (house mouse)Potency8.539820
5-ethyl-3-[[4-(2-methylpropoxy)phenyl]methylthio]-1H-1,2,4-triazoleMus musculus (house mouse)Potency9.505620
3-(2,3-dimethyl-1H-indol-5-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency9.106320
N-[4-(4-morpholinylazo)phenyl]acetamideMus musculus (house mouse)Potency12.589310
4-chloro-1-ethyl-3-nitro-2-quinolinoneMus musculus (house mouse)Potency8.427920
[4-[(2-fluorophenyl)methoxy]phenyl]-(1-pyrrolidinyl)methanethioneMus musculus (house mouse)Potency35.481310
3-(3-nitrophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency21.280420
1-(1,3-benzodioxol-5-ylmethyl)-3-(3-chloro-2-methylphenyl)thioureaMus musculus (house mouse)Potency9.149820
1-(1,3-benzodioxol-5-ylmethyl)-3-(2,5-dimethylphenyl)thioureaMus musculus (house mouse)Potency8.912510
1-ethyl-2-[(4-methylphenoxy)methyl]benzimidazoleMus musculus (house mouse)Potency22.196920
3-(4-methoxyphenyl)-1H-pyrazole-5-carbohydrazideMus musculus (house mouse)Potency0.794310
4-methyl-N-(3-nitrophenyl)-5-phenyl-3-thiophenecarboxamideMus musculus (house mouse)Potency1.258910
4-prop-2-enyl-3-(3,4,5-trimethoxyphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency35.481320
N-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-2,2,2-trichloroacetamideMus musculus (house mouse)Potency20.386620
N-(2-fluoro-5-methylphenyl)-3-phenylpropanamideMus musculus (house mouse)Potency2.665120
4,5-dimethoxy-2-[(1-oxo-2-thiophen-2-ylethyl)amino]benzoic acid methyl esterMus musculus (house mouse)Potency4.736020
4-tert-butyl-N-(1,4-dioxo-2,3-dihydrophthalazin-5-yl)benzamideMus musculus (house mouse)Potency4.928820
3-(4-chlorophenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneMus musculus (house mouse)Potency16.803720
2-[4-(4-fluorophenyl)-2-thiazolyl]-5-methyl-4H-pyrazol-3-oneMus musculus (house mouse)Potency12.589310
3-phenyl-5,6,7,8-tetrahydro-1H-pyrazolo[5,1-b]quinazolin-9-oneMus musculus (house mouse)Potency16.193620
N-[2-(2-methylpropyl)-1,3-dioxo-5-isoindolyl]-2-furancarboxamideMus musculus (house mouse)Potency6.729420
N-[[(2,4-dimethyl-8-quinolinyl)amino]-sulfanylidenemethyl]-4-methylbenzamideMus musculus (house mouse)Potency2.733420
N-(4-methoxyphenyl)-3,4-dihydro-1H-isoquinoline-2-carbothioamideMus musculus (house mouse)Potency28.934220
1-(4-bromophenyl)-3-(2-phenylethyl)thioureaMus musculus (house mouse)Potency4.087120
2-[2-[[benzamido(sulfanylidene)methyl]amino]-4-thiazolyl]acetic acid ethyl esterMus musculus (house mouse)Potency0.891310
5-bromo-N-[(2-pyridinylamino)-sulfanylidenemethyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency7.943320
5-(4-chlorophenyl)-2-furanpropionic acidMus musculus (house mouse)Potency35.481320
N'-[(2-chlorophenyl)-oxomethyl]-2-thiophenecarbohydrazideMus musculus (house mouse)Potency14.125410
6-(1,3-benzoxazol-2-yl)-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency17.811320
3-prop-2-enyl-2-sulfanylidene-5,6,7,8-tetrahydro-1H-[1]benzothiolo[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency0.553020
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneMus musculus (house mouse)Potency24.035320
3-methyl-7-(phenylmethyl)-8-(propan-2-ylthio)purine-2,6-dioneMus musculus (house mouse)Potency15.848910
2-methyl-5-(1-pyrrolidinyl)isoindole-1,3-dioneMus musculus (house mouse)Potency3.855220
N-(4-methylphenyl)carbamic acid (cyclopentylideneamino) esterMus musculus (house mouse)Potency31.622810
4-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency11.220220
2-methyl-N-(2-naphthalenyl)-3-furancarboxamideMus musculus (house mouse)Potency0.562310
N-[[(6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-4-phenylbenzamideMus musculus (house mouse)Potency14.550020
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideMus musculus (house mouse)Potency12.431220
N-(6-methyl-2-pyridinyl)-5-nitro-2-furancarboxamideMus musculus (house mouse)Potency23.350720
1-(3,4-dimethoxy-2-methylphenyl)-2-(3,4-dimethoxyphenyl)ethanoneMus musculus (house mouse)Potency18.867720
7-chloro 5-(2-chlorophenyl)-1,3-dihydro-2h-(1,4)-benzodiazepine-2-thioneMus musculus (house mouse)Potency7.511420
1-(3-chlorophenyl)-3-(phenylmethyl)thioureaMus musculus (house mouse)Potency9.106320
2-tert-butyl-N-(phenylmethyl)-4-pyridinecarboxamideMus musculus (house mouse)Potency6.581220
6-[amino(methyl)amino]-N2,N4-diethyl-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency21.280420
1-[3-(4-chlorophenyl)-5-(methylthio)-1,2,4-triazol-1-yl]-1-butanoneMus musculus (house mouse)Potency7.079510
4-methyl-N,5-diphenyl-3-thiophenecarboxamideMus musculus (house mouse)Potency24.068220
N-(2-pyridinyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideMus musculus (house mouse)Potency0.562310
5-[(2-chlorophenoxy)methyl]-3-pyridin-4-yl-1,2,4-oxadiazoleMus musculus (house mouse)Potency2.238710
N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamideMus musculus (house mouse)Potency19.118020
N-(3-phenyl-1,3-benzothiazol-2-ylidene)-2-propenamideMus musculus (house mouse)Potency22.740620
6-(1H-benzimidazol-2-yl)-2-methyl-1H-benzimidazoleMus musculus (house mouse)Potency35.481310
2-[[4-(1-pyrrolidinylsulfonyl)phenyl]hydrazinylidene]propanedinitrileMus musculus (house mouse)Potency14.432620
1-(2-fluoro-5-nitrophenyl)-3-phenylureaMus musculus (house mouse)Potency35.481310
N-[5-(methylthio)-1,3,4-thiadiazol-2-yl]-3-phenylpropanamideMus musculus (house mouse)Potency35.481310
3-ethoxy-N-[(3-pyridinylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency22.874120
2-phenyl-1H-quinazoline-4-thioneMus musculus (house mouse)Potency3.936920
N-(4-methoxyphenyl)-3-methyl-1,3-benzothiazol-2-imineMus musculus (house mouse)Potency0.398110
N-[4-(4-chlorophenyl)-3,5-dimethyl-2-thiazolylidene]-2-furancarboxamideMus musculus (house mouse)Potency25.118910
4-oxo-3-pyrimido[2,1-b][1,3]benzoxazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.199510
2-(4-nitro-2-pyridinyl)isoindole-1,3-dioneMus musculus (house mouse)Potency35.481310
3-[[(3-chloro-4-ethoxyphenyl)-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency8.154820
3-(2-furanyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency23.350720
N-(3-carbamoyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-4-chloro-2-methyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency8.912510
1-(4-chlorophenyl)-3-(2-furanylmethyl)thioureaMus musculus (house mouse)Potency14.501520
1-(3,4-dichlorophenyl)-3-(3-pyridinylmethyl)thioureaMus musculus (house mouse)Potency35.481320
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]acetamideMus musculus (house mouse)Potency24.035320
3,6-dichloro-N-(4-methyl-2-pyridinyl)-1-benzothiophene-2-carboxamideMus musculus (house mouse)Potency2.771720
2-methoxy-N-(4-methylphenyl)-4-(methylthio)benzamideMus musculus (house mouse)Potency15.586420
1-[[(1,3-dimethyl-4-pyrazolyl)-oxomethyl]amino]-3-(4-methylphenyl)thioureaMus musculus (house mouse)Potency11.220210
1-[[(1,5-dimethyl-3-pyrazolyl)-oxomethyl]amino]-3-(2-methoxyphenyl)thioureaMus musculus (house mouse)Potency35.481310
4-(2-methylphenyl)-3-(5-methyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency4.564020
1-(2-methylphenyl)-3-[[(5-methyl-3-thiophenyl)-oxomethyl]amino]thioureaMus musculus (house mouse)Potency3.981110
3-(4-ethyl-5-methyl-3-thiophenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency5.091020
1-(3-methylphenyl)-3-[[(5-methyl-3-thiophenyl)-oxomethyl]amino]thioureaMus musculus (house mouse)Potency9.568620
4-(3-methylphenyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency2.115420
1-(3-methylphenyl)-3-[[oxo-(5-propyl-3-thiophenyl)methyl]amino]thioureaMus musculus (house mouse)Potency3.931020
3-(1-benzothiophen-3-yl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.855620
4-(3-methylphenyl)-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency3.298420
3-(4,5-dimethyl-3-thiophenyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency4.564020
3-(2-methyl-3-furanyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency16.193620
4-(phenylmethyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency5.045120
N-(4-methyl-2-pyridinyl)-5-nitro-2-furancarboxamideMus musculus (house mouse)Potency35.481320
N-(2-chlorophenyl)-5-nitro-2-furancarboxamideMus musculus (house mouse)Potency12.924420
1-cyclohexyl-3-(2,3-dihydro-1,4-benzodioxin-6-yl)ureaMus musculus (house mouse)Potency12.589320
8-[(2-methyl-5-nitro-1,2,4-triazol-3-yl)thio]quinolineMus musculus (house mouse)Potency14.501520
4,5-dimethyl-2-[4-(3-nitrophenyl)-2-thiazolyl]-1H-pyrazol-3-oneMus musculus (house mouse)Potency35.481320
2-(4-fluoro-N-methylsulfonylanilino)-N-(3-methylphenyl)acetamideMus musculus (house mouse)Potency5.317720
2-[(1-ethyl-2,5-dimethyl-3-pyrrolyl)methylidene]indene-1,3-dioneMus musculus (house mouse)Potency11.220210
N-(6-ethoxy-1,3-benzothiazol-2-yl)butanamideMus musculus (house mouse)Potency35.481310
4-chloro-3-ethoxy-N-(4-ethylphenyl)benzenesulfonamideMus musculus (house mouse)Potency35.481320
N2,N4-bis(4-methoxyphenyl)pyrimidine-2,4-diamineMus musculus (house mouse)Potency35.481310
6-(2-phenylethyl)-3-(phenylmethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleMus musculus (house mouse)Potency35.481310
2-methoxy-3-methyl-N-[4-(4-morpholinylmethyl)phenyl]benzamideMus musculus (house mouse)Potency35.481310
4,4-dicarboxy-5-pyridoxylprolineMus musculus (house mouse)Potency0.398110
N-(2-phenyl-6-imidazo[1,2-a]pyridinyl)acetamideMus musculus (house mouse)Potency24.035320
N-(6-bromo-2,3-dihydro-1,4-benzodioxin-7-yl)-2-furancarboxamideMus musculus (house mouse)Potency0.562310
3-methyl-5-propyl-7-furo[3,2-g][1]benzopyranoneMus musculus (house mouse)Potency6.309610
3-(3,4-dimethylanilino)-1-thiophen-2-yl-1-propanoneMus musculus (house mouse)Potency3.162310
2-[(3-methyl-4-oxo-2-quinazolinyl)thio]-N-phenylacetamideMus musculus (house mouse)Potency15.586420
N-(4-methoxyphenyl)-2-(2-methylpropyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency35.481310
5-(4-fluorophenyl)-2-thiophen-2-yloxazoleMus musculus (house mouse)Potency22.387210
N-(2-chlorophenyl)-2-[[cyclopropyl(oxo)methyl]amino]-4-methyl-5-thiazolecarboxamideMus musculus (house mouse)Potency8.528020
4-[[[2-(3-methylphenyl)ethylamino]-sulfanylidenemethyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency1.258920
N-(4-fluorophenyl)-1-(3-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinamineMus musculus (house mouse)Potency11.220210
2-[[5-(4-ethoxyphenyl)-1,3,4-oxadiazol-2-yl]thio]-1-(4-morpholinyl)ethanoneMus musculus (house mouse)Potency31.622810
N,N-diethyl-4-[oxo-(2,4,6-trimethylphenyl)methyl]benzamideMus musculus (house mouse)Potency35.481310
N'-[(4-chlorophenyl)-oxomethyl]-2-hydroxy-3-methylbenzohydrazideMus musculus (house mouse)Potency7.079510
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-4-methylbenzamideMus musculus (house mouse)Potency11.590820
N-[[(6-methyl-4-pyrimidinyl)thio]methyl]benzamideMus musculus (house mouse)Potency25.118910
5-(1-methyl-2-benzimidazolyl)-2-thiophenecarboxaldehydeMus musculus (house mouse)Potency11.220210
N-(4-anilinophenyl)-2-methylpropanamideMus musculus (house mouse)Potency12.589310
N-[[(6-methoxy-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency3.715820
3-(4-bromoanilino)-1-(3-nitrophenyl)-1-propanoneMus musculus (house mouse)Potency25.118910
N-(3-hydroxyphenyl)-5-methyl-3-furancarboxamideMus musculus (house mouse)Potency35.481310
3-(4-methoxyphenyl)-5-(4-methylphenyl)-1,2,4-oxadiazoleMus musculus (house mouse)Potency21.450920
3-anilino-1-(3-nitrophenyl)-1-propanoneMus musculus (house mouse)Potency23.753120
2-[(2-chlorophenyl)methylthio]-6-nitro-1,3-benzothiazoleMus musculus (house mouse)Potency12.589310
4-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]benzoic acid ethyl esterMus musculus (house mouse)Potency31.622810
1-(4-chlorophenyl)-3-(2-phenylethyl)thioureaMus musculus (house mouse)Potency13.131120
4-sulfanylidene-1,6,7,8,9,10-hexahydropyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrileMus musculus (house mouse)Potency10.665420
3-acetyl-2-methylbenzo[f]benzofuran-4,9-dioneMus musculus (house mouse)Potency9.915020
7-methoxy-4,8-dimethyl-1-benzopyran-2-oneMus musculus (house mouse)Potency2.511910
3-bromo-N-[(tert-butylamino)-sulfanylidenemethyl]-4-methoxybenzamideMus musculus (house mouse)Potency4.969320
N-[(3-acetylanilino)-sulfanylidenemethyl]-3-chlorobenzamideMus musculus (house mouse)Potency6.409220
4-(3,4-dimethylphenyl)-5-phenyl-2-thiazolamineMus musculus (house mouse)Potency8.971620
2-(1H-benzimidazol-2-ylmethyl)benzene-1,4-diolMus musculus (house mouse)Potency15.848910
N-(2,4-dichlorophenyl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency28.934220
2-(4-chlorophenyl)-N-[(2-hydroxy-5-methylanilino)-sulfanylidenemethyl]acetamideMus musculus (house mouse)Potency11.904820
3,4-dimethoxybenzenecarbothioic acid S-(4-chlorophenyl) esterMus musculus (house mouse)Potency12.589310
1-[(3-methylphenyl)methyl]benzimidazoleMus musculus (house mouse)Potency7.943310
1-[(2,4-dichlorophenyl)methyl]-3-phenylthioureaMus musculus (house mouse)Potency6.694620
4-propan-2-yl-N-(3-pyridinyl)benzamideMus musculus (house mouse)Potency1.258910
1-(2-methylpropyl)-2-thiophen-2-ylbenzimidazoleMus musculus (house mouse)Potency35.481310
2-(2-phenylethylthio)-3-pyridinecarboxylic acidMus musculus (house mouse)Potency13.534620
N-[[2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency10.157820
lupitidineMus musculus (house mouse)Potency35.481310
2-[(3-ethyl-4-methyl-2-oxo-1-benzopyran-7-yl)oxy]acetic acid methyl esterMus musculus (house mouse)Potency35.481310
4-(2-furanylmethyl)-3-(phenylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency13.357420
2,4-dimethyl-6-oxo-3-pyrancarboxylic acid (3-nitrophenyl)methyl esterMus musculus (house mouse)Potency22.387210
1-(2-furanylmethyl)-3-(4-phenoxyphenyl)thioureaMus musculus (house mouse)Potency17.246720
N-[(2-methoxyphenyl)methyl]-4-(1-piperidinyl)anilineMus musculus (house mouse)Potency15.848910
1-(2-methylpropyl)-3-(4-phenoxyphenyl)thioureaMus musculus (house mouse)Potency3.764620
1-cyclopentyl-3-(4-phenoxyphenyl)thioureaMus musculus (house mouse)Potency5.011920
N-[3-[(1,3-dioxo-5-isoindolyl)oxy]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency0.891310
N-[anilino(sulfanylidene)methyl]-5-bromo-2-furancarboxamideMus musculus (house mouse)Potency3.162310
2-(2,3-dimethylphenoxy)-N-pyridin-4-ylacetamideMus musculus (house mouse)Potency1.978320
6-methoxy-4-methyl-2-[(2-methylphenyl)methylthio]quinazolineMus musculus (house mouse)Potency15.848910
2-[4-(pyridin-4-ylmethylsulfamoyl)phenoxy]acetic acid methyl esterMus musculus (house mouse)Potency5.865420
3-[1-(4-acetylphenyl)-5-thiophen-2-yl-2-pyrrolyl]propanoic acidMus musculus (house mouse)Potency35.481320
4-[methyl(methylsulfonyl)amino]-N-(2-phenylethyl)benzamideMus musculus (house mouse)Potency14.501520
N-[3-(methylthio)-1,2,4-thiadiazol-5-yl]-2-phenylacetamideMus musculus (house mouse)Potency21.280420
N-(4-phenylmethoxyphenyl)carbamic acid methyl esterMus musculus (house mouse)Potency5.623410
2-[[anilino(oxo)methyl]amino]-N-(phenylmethyl)benzamideMus musculus (house mouse)Potency35.481310
4-phenacyloxybenzoic acid methyl esterMus musculus (house mouse)Potency0.501210
2-(3-acetamidophenoxy)-N-phenylacetamideMus musculus (house mouse)Potency12.589310
N2-(4-methylphenyl)-6-[(2-pyrimidinylthio)methyl]-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency0.354810
N-(4-ethoxyphenyl)-1,2,5-thiadiazole-3-carboxamideMus musculus (house mouse)Potency18.169620
2-(2-methoxyphenyl)-1H-indoleMus musculus (house mouse)Potency2.818410
N-[5-(2-chlorophenyl)-1H-1,2,4-triazol-3-yl]-4,6-dimethyl-2-pyrimidinamineMus musculus (house mouse)Potency10.000010
2-(4-chloro-2-methylanilino)-3-pyridinecarboxamideMus musculus (house mouse)Potency12.589310
3-acetamidobenzoic acid [2-(2-chlorophenyl)-2-oxoethyl] esterMus musculus (house mouse)Potency0.398110
4-bromo-1-methyl-N-(2-thiazolyl)-3-pyrazolecarboxamideMus musculus (house mouse)Potency35.481310
N-(4,5-dimethyl-2-thiazolyl)cyclohexanecarboxamideMus musculus (house mouse)Potency6.309610
5-[(2-chlorophenoxy)methyl]-N-(2-thiazolyl)-2-furancarboxamideMus musculus (house mouse)Potency16.803720
N-(2,3-dihydro-1H-inden-5-yl)-2-methyl-3-nitrobenzamideMus musculus (house mouse)Potency11.220210
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneMus musculus (house mouse)Potency0.504520
2-methyl-4-phenyl-1H-pyrrole-3-carboxylic acid methyl esterMus musculus (house mouse)Potency28.183810
5-hydroxy-2-[[(4-methylphenyl)thio]methyl]-3-benzofurancarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
1-(2-methyl-1H-indol-3-yl)-2-(2-thiazolylamino)ethanoneMus musculus (house mouse)Potency4.152420
4-chloro-N-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]benzamideMus musculus (house mouse)Potency35.481310
1-ethyl-3-(4-methylphenyl)sulfonylthioureaMus musculus (house mouse)Potency24.803320
2-(2-imidazo[1,2-a]pyridinylmethylthio)-6-nitro-1H-benzimidazoleMus musculus (house mouse)Potency35.481310
N'-(1,3-benzoxazol-2-yl)benzohydrazideMus musculus (house mouse)Potency14.976320
N'-(1,3-benzothiazol-2-yl)-4-fluorobenzohydrazideMus musculus (house mouse)Potency0.910620
3-(4-ethoxyphenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency5.966520
1-(2,3-dimethyl-1-indolyl)-2-(4-methyl-1-piperidinyl)ethanoneMus musculus (house mouse)Potency12.589310
1-(cycloheptylideneamino)-3-(4-fluorophenyl)thioureaMus musculus (house mouse)Potency11.124820
4-methoxy-N-[[(phenylmethyl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency14.733420
N-(2-ethoxyphenyl)-1H-benzimidazol-2-amineMus musculus (house mouse)Potency35.481310
5-(5-ethyl-2-hydroxy-4-methoxyphenyl)-4-(4-methoxyphenyl)isoxazoleMus musculus (house mouse)Potency14.125420
2-[(3-chloro-1-benzothiophen-2-yl)methylideneamino]phenolMus musculus (house mouse)Potency5.623410
3-amino-2-(4-methylphenyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency0.112210
3-amino-4-methoxy-1H-indole-2-carbohydrazideMus musculus (house mouse)Potency14.125410
4-(4-methylphenyl)-3-(2-pyrazinyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency35.481310
N'-[1-oxo-2-(4-propan-2-ylphenoxy)ethyl]-2-pyrazinecarbohydrazideMus musculus (house mouse)Potency35.481310
N-(2-ethylphenyl)-2-methoxy-5-methylbenzenesulfonamideMus musculus (house mouse)Potency28.183810
4-ethoxy-N-(4-fluorophenyl)-2,3-dimethylbenzenesulfonamideMus musculus (house mouse)Potency18.867720
2-mercaptonaphth(2,3)imidazoleMus musculus (house mouse)Potency15.804820
3-[[[5-(phenylmethyl)-1,3,4-oxadiazol-2-yl]thio]methyl]benzoic acidMus musculus (house mouse)Potency0.501210
2-(2-fluorophenyl)-5-(4-methyl-1-piperidinyl)-4-oxazolecarbonitrileMus musculus (house mouse)Potency8.285220
1-(4-methyl-1-piperidinyl)-2-[(3-methyl-2-quinoxalinyl)thio]ethanoneMus musculus (house mouse)Potency17.900820
5-bromo-N-(pyridin-4-ylmethyl)-2-thiophenesulfonamideMus musculus (house mouse)Potency1.778310
6-(chloromethyl)-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency8.539820
3-[(2-chloro-6-fluorophenyl)methylthio]-4-ethyl-5-(2-furanyl)-1,2,4-triazoleMus musculus (house mouse)Potency12.589310
8-methyl-2-(3-methylbutyl)-1,2,4-triazaspiro[4.5]decane-3-thioneMus musculus (house mouse)Potency12.431220
8-(9-methyl-5H-pyrimido[5,4-b]indol-4-yl)-1,4-dioxa-8-azaspiro[4.5]decaneMus musculus (house mouse)Potency8.116020
thiothixeneMus musculus (house mouse)Potency20.207820
1-(phenylmethyl)-3-[4-(trifluoromethoxy)phenyl]thioureaMus musculus (house mouse)Potency9.149820
1-methyl-5-(1-naphthalenyloxy)-4-nitroimidazoleMus musculus (house mouse)Potency28.934220
4-chloro-N-(1,2-dimethyl-5-benzimidazolyl)benzamideMus musculus (house mouse)Potency28.183810
N-[2-(1-cyclohexenyl)ethyl]-4-[methyl(methylsulfonyl)amino]benzamideMus musculus (house mouse)Potency0.631010
4-(4-chlorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency5.889220
N-[[(phenylmethyl)amino]-sulfanylidenemethyl]-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency9.581820
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-3-methylbenzamideMus musculus (house mouse)Potency7.943320
4-phenyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency23.350720
terazosinMus musculus (house mouse)Potency35.481310
curcuminMus musculus (house mouse)Potency24.388820
4-(2-methylphenyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency12.589310
3-[[(3-acetylanilino)-oxomethyl]amino]-2-thiophenecarboxylic acid methyl esterMus musculus (house mouse)Potency7.943310
N-(1,3-benzodioxol-5-yl)-4-(2-furanylmethyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency11.220220
4-[[[(2-methoxyphenyl)methylamino]-oxomethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency35.481310
1-(4-methyl-3-nitrophenyl)-3-[(4-methylphenyl)methyl]thioureaMus musculus (house mouse)Potency4.928820
1-(4-methyl-2-oxo-1-benzopyran-7-yl)-3-(2-pyridinylmethyl)thioureaMus musculus (house mouse)Potency12.589310
1-(2,4-dichlorophenyl)-3-(1-methyl-3-pyrazolyl)ureaMus musculus (house mouse)Potency8.912510
1-(3,4-dimethoxyphenyl)-3-(2-methoxy-5-nitrophenyl)ureaMus musculus (house mouse)Potency25.665120
1-[[(2-methyl-3-furanyl)-oxomethyl]amino]-3-[2-(trifluoromethyl)phenyl]thioureaMus musculus (house mouse)Potency35.481310
1-cyclopentyl-3-(2-phenoxyphenyl)thioureaMus musculus (house mouse)Potency5.120920
1-(3-acetylphenyl)-3-(2-pyridinylmethyl)ureaMus musculus (house mouse)Potency19.149820
N-[4-[2-[(4-methyl-2-pyridinyl)amino]-4-thiazolyl]phenyl]acetamideMus musculus (house mouse)Potency2.238710
1-(2-chlorophenyl)-3-[(2-chlorophenyl)methyl]thioureaMus musculus (house mouse)Potency1.690420
2-[2-(4-methylphenoxy)ethyl]isoindole-1,3-dioneMus musculus (house mouse)Potency31.622810
1-(4-methoxyphenyl)-3-(6-quinoxalinyl)thioureaMus musculus (house mouse)Potency26.651420
4-mercapto-5-(4-methoxyphenyl)-2-oxo-1,5-diazaspiro[5.5]undec-3-ene-3-carbonitrileMus musculus (house mouse)Potency31.832620
1-(3-chloro-4-methoxyphenyl)-3-[2-(4-methyl-1-piperidinyl)ethyl]thioureaMus musculus (house mouse)Potency20.085020
4-(3,4-dimethoxyphenyl)-N-(3-methyl-2-pyridinyl)-2-thiazolamineMus musculus (house mouse)Potency3.548110
N-[3-[[(3,5-dimethoxyphenyl)-oxomethyl]amino]phenyl]carbamic acid ethyl esterMus musculus (house mouse)Potency19.952610
3-chloro-4-[(1-ethyl-2-benzimidazolyl)thio]anilineMus musculus (house mouse)Potency35.481310
1-(1-naphthalenylmethoxy)benzotriazoleMus musculus (house mouse)Potency0.983420
N-(4-methoxyphenyl)-4-(methylthio)benzenesulfonamideMus musculus (house mouse)Potency28.934220
2,2-dimethyl-N-[[2-(4-methyl-1-piperidinyl)anilino]-sulfanylidenemethyl]propanamideMus musculus (house mouse)Potency4.332220
N-cycloheptyl-2-[(6-nitro-1H-benzimidazol-2-yl)thio]acetamideMus musculus (house mouse)Potency12.967620
N-methyl-N-phenylcarbamic acid (4-tert-butylphenyl) esterMus musculus (house mouse)Potency35.481310
(2,3-dimethoxyphenyl)-(1-pyrrolidinyl)methanethioneMus musculus (house mouse)Potency2.545620
1-(4-bromophenyl)-3-(2-fluorophenyl)thioureaMus musculus (house mouse)Potency23.350720
1-(3,4-dichlorophenyl)-3-(3,5-dimethylphenyl)thioureaMus musculus (house mouse)Potency22.740620
1-[[(2-chlorophenyl)-oxomethyl]amino]-3-(2-methoxy-5-methylphenyl)thioureaMus musculus (house mouse)Potency7.079510
4-[[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]methylamino]benzenesulfonamideMus musculus (house mouse)Potency22.387210
4-[5-(2-phenylethyl)-2-sulfanylidene-1,3,5-triazinan-1-yl]benzoic acid ethyl esterMus musculus (house mouse)Potency35.481320
N-[(1-ethyl-2-oxo-6-benzo[cd]indolyl)sulfonyl]-N-(4-methoxyphenyl)-3-pyridinecarboxamideMus musculus (house mouse)Potency35.481310
2,3,5,6-tetramethyl-N-(2-methyl-1,3-benzothiazol-5-yl)benzenesulfonamideMus musculus (house mouse)Potency8.116020
cct018159Mus musculus (house mouse)Potency24.035320
N-[4-(1,3-benzothiazol-2-yl)phenyl]-2-[(4-tert-butylphenyl)sulfonylamino]acetamideMus musculus (house mouse)Potency35.481310
5-chloro-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-3-methyl-2-benzofurancarboxamideMus musculus (house mouse)Potency15.848910
1-[tert-butyl-[(3,5-dimethylphenyl)-oxomethyl]amino]-3-(4-chlorophenyl)ureaMus musculus (house mouse)Potency35.481320
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideMus musculus (house mouse)Potency3.981110
N-[3-cyano-4-(4-methoxyphenyl)-5-methyl-2-thiophenyl]-2-methyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency35.481310
4-[(2-bromophenoxy)methyl]-N-[4-[(3,5-dimethyl-1-pyrazolyl)methyl]phenyl]benzamideMus musculus (house mouse)Potency22.387210
1-[[(5-bromo-2-furanyl)-oxomethyl]amino]-3-(2,5-dimethylphenyl)thioureaMus musculus (house mouse)Potency0.089110
1-[[[2-(difluoromethoxy)phenyl]-oxomethyl]amino]-3-(4-fluorophenyl)thioureaMus musculus (house mouse)Potency2.818410
1-[[[2-(difluoromethoxy)phenyl]-oxomethyl]amino]-3-(3-methylphenyl)thioureaMus musculus (house mouse)Potency18.186320
N-(1-ethyl-2-benzimidazolyl)-5-[(4-methyl-2-nitrophenoxy)methyl]-2-furancarboxamideMus musculus (house mouse)Potency3.625320
N-(5-bromo-8-quinolinyl)-5-[(4-chloro-1-pyrazolyl)methyl]-2-furancarboxamideMus musculus (house mouse)Potency5.623410
1-[[[2-(2,4-dichlorophenyl)-4-quinolinyl]-oxomethyl]amino]-3-phenylureaMus musculus (house mouse)Potency11.220210
[3-amino-6-(4-methoxyphenyl)-2-thieno[2,3-b]pyridinyl]-(3,4-dimethoxyphenyl)methanoneMus musculus (house mouse)Potency22.387210
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamideMus musculus (house mouse)Potency31.622810
5-(4-bromophenyl)-N-[[(2-propyl-5-tetrazolyl)amino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency1.653120
2-[(5-bromo-2-thiophenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideMus musculus (house mouse)Potency14.125410
3-chloro-4,5-dimethoxy-N-(1-naphthalenylmethyl)benzamideMus musculus (house mouse)Potency12.589310
2-(3-bromophenyl)-N-(4,5-dihydrothiazol-2-yl)-4-quinolinecarboxamideMus musculus (house mouse)Potency14.733420
N-[4-[oxo-[(1-oxo-2,2-diphenylethyl)hydrazo]methyl]phenyl]propanamideMus musculus (house mouse)Potency2.511910
1-[[2-(2,4-dichlorophenoxy)-1-oxoethyl]amino]-3-(4-fluorophenyl)thioureaMus musculus (house mouse)Potency8.836820
tenovin-1Mus musculus (house mouse)Potency35.481310
N-[4-[[[2-(2,5-dimethylphenoxy)-1-oxoethyl]hydrazo]-oxomethyl]phenyl]propanamideMus musculus (house mouse)Potency5.623410
2-bromo-N-[2,3-dihydroindol-1-yl(sulfanylidene)methyl]benzamideMus musculus (house mouse)Potency0.495620
N-[[3-(hydroxymethyl)anilino]-sulfanylidenemethyl]-4-phenylbenzamideMus musculus (house mouse)Potency2.201620
5-bromo-N-[[4-[(3,5-dimethylphenyl)sulfamoyl]anilino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency5.745720
N-[[methyl-(phenylmethyl)amino]-sulfanylidenemethyl]-4-phenylbenzamideMus musculus (house mouse)Potency0.185420
N-[(3-acetylanilino)-sulfanylidenemethyl]-5-bromo-3-pyridinecarboxamideMus musculus (house mouse)Potency13.891420
5-bromo-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency15.848910
2-(1,3-dimethyl-2,6-dioxo-9-purinyl)-N-[2-(4-morpholinyl)-5-(trifluoromethyl)phenyl]acetamideMus musculus (house mouse)Potency12.589310
2-chloro-N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-5-(1,2,4-triazol-4-yl)benzamideMus musculus (house mouse)Potency26.632020
5-[(3,5-dimethyl-4-nitro-1-pyrazolyl)methyl]-N-[(4-methoxyphenyl)methyl]-2-furancarboxamideMus musculus (house mouse)Potency5.317720
N-[3-chloro-2-(4-morpholinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideMus musculus (house mouse)Potency14.125410
N-[4,6-bis(4-morpholinyl)-1,3,5-triazin-2-yl]-2-(methylthio)-1,3-benzothiazol-6-amineMus musculus (house mouse)Potency0.100010
3,4-dimethoxy-N-[[4-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency0.669020
4-[[4-bromo-5-(4-morpholinyl)-2-furanyl]methylideneamino]phenolMus musculus (house mouse)Potency35.481310
N-(4-chlorophenyl)-7,8-dimethoxy-1-oxo-2-benzothiopyran-3-carboxamideMus musculus (house mouse)Potency35.481310
4-(4-fluorophenyl)sulfonyl-2-(2-furanyl)-N-phenyl-5-oxazolamineMus musculus (house mouse)Potency14.125410
4-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-3-quinolinecarboxylic acid ethyl esterMus musculus (house mouse)Potency23.350720
4-bromo-N'-[(4-bromophenyl)-oxomethyl]-1-methyl-3-pyrazolecarbohydrazideMus musculus (house mouse)Potency22.387210
N-[[(5-methyl-1H-pyrazol-3-yl)amino]-oxomethyl]-3-(1,1,2,2-tetrafluoroethoxy)benzamideMus musculus (house mouse)Potency1.995310
N-[[3-chloro-4-(4-morpholinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency9.053220
N-[[3-chloro-4-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideMus musculus (house mouse)Potency4.736020
pyridine-2-carboxylic acid thiazol-2-ylamideMus musculus (house mouse)Potency7.550620
3-chloro-N-[3-nitro-5-(2-pyridinylthio)phenyl]benzamideMus musculus (house mouse)Potency35.481310
2-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]thio]-N-(4-methyl-2-thiazolyl)acetamideMus musculus (house mouse)Potency35.481310
1-methoxy-N-[4-(pyridin-4-ylmethyl)phenyl]-2-naphthalenecarboxamideMus musculus (house mouse)Potency25.665120
1-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-2-[(4-chlorophenyl)methylthio]ethanoneMus musculus (house mouse)Potency27.717020
N-(3,5-dimethylphenyl)-4-(3-methoxyphenyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency3.981110
N-(1-tert-butyl-5-benzimidazolyl)-3,4,5-trimethoxybenzamideMus musculus (house mouse)Potency3.981110
N-(4-acetamidophenyl)-2-[[1-(4-ethylphenyl)-5-tetrazolyl]thio]acetamideMus musculus (house mouse)Potency12.589310
2-[acetyl(2-furanylmethyl)amino]-N-(4-chlorophenyl)-5-methyl-4-thiazolecarboxamideMus musculus (house mouse)Potency12.589310
3-(4-chlorophenyl)-5-propyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneMus musculus (house mouse)Potency3.814620
4-[[[3-(4-morpholinylsulfonyl)phenyl]-oxomethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency11.220210
5-(3,4-dimethoxyphenyl)-2-phenyl-4-thieno[2,3-d][1,3]oxazinoneMus musculus (house mouse)Potency35.481310
N-[2-(2-pyridinyl)-3H-benzimidazol-5-yl]cyclohexanecarboxamideMus musculus (house mouse)Potency35.481310
2-fluoro-N-[2-(3-pyridinyl)-3H-benzimidazol-5-yl]benzamideMus musculus (house mouse)Potency11.220210
2-[(4-ethoxyphenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideMus musculus (house mouse)Potency18.256320
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N,N-diethylacetamideMus musculus (house mouse)Potency6.309610
1-(4-methylphenyl)sulfonyl-2-benzimidazolamineMus musculus (house mouse)Potency31.622810
2-(3-acetyl-1-indolyl)-N-(2,4-dimethylphenyl)acetamideMus musculus (house mouse)Potency18.169620
2-(4-chlorophenoxy)-N-[4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]phenyl]acetamideMus musculus (house mouse)Potency35.481310
1-(4-morpholinyl)-2-[2-(phenylmethylthio)-1-benzimidazolyl]ethanoneMus musculus (house mouse)Potency10.000010
N-[4-[[2-furanyl(oxo)methyl]amino]phenyl]-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency28.934220
2-ethyl-N-[1-[2-(1-piperidinyl)ethyl]-2-benzimidazolyl]-3-pyrazolecarboxamideMus musculus (house mouse)Potency25.665120
N-[4-[2-[(6-methyl-2-pyridinyl)amino]-4-thiazolyl]phenyl]acetamideMus musculus (house mouse)Potency19.952610
N-(1,3-benzothiazol-2-yl)-2-[methyl-(4-methylphenyl)sulfonylamino]acetamideMus musculus (house mouse)Potency2.511910
4-[(3-methyl-2-oxo-1,3-benzoxazol-6-yl)sulfonylamino]benzoic acid ethyl esterMus musculus (house mouse)Potency22.387210
[7-(difluoromethyl)-5-(4-methoxyphenyl)-3-pyrazolo[1,5-a]pyrimidinyl]-(1-piperidinyl)methanoneMus musculus (house mouse)Potency11.220210
1-methyl-2-oxo-N-(2-pyridinyl)-6-benzo[cd]indolesulfonamideMus musculus (house mouse)Potency17.782810
2,5-dichloro-4-ethoxy-N-(2-pyridinylmethyl)benzenesulfonamideMus musculus (house mouse)Potency16.271020
N'-methyl-N-[1-methyl-5-(4-methylphenyl)-2-imidazolyl]-N'-(phenylmethyl)butanediamideMus musculus (house mouse)Potency3.352820
N-[2,2-dichloro-1-(4-chlorophenyl)sulfonylethenyl]benzamideMus musculus (house mouse)Potency25.665120
N2,N7-bis(2,5-dimethylphenyl)-9H-fluorene-2,7-disulfonamideMus musculus (house mouse)Potency1.000010
3-(1-piperidinylsulfonyl)-N-(2-thiazolyl)benzamideMus musculus (house mouse)Potency35.481320
4-chloro-3-(1-piperidinylsulfonyl)-N-(2-thiazolyl)benzamideMus musculus (house mouse)Potency22.740620
LSM-16285Mus musculus (house mouse)Potency10.537320
ym-90709Mus musculus (house mouse)Potency31.832620
5-nitro-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency0.562310
2-[[[3-[2-(4-methylphenyl)sulfonylethylthio]phenyl]-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency31.622810
2-(3,4-dimethoxyphenyl)-8-methoxy-4,4-dimethyl-5H-isothiazolo[5,4-c]quinoline-1-thioneMus musculus (house mouse)Potency10.000010
3-methoxy-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)benzamideMus musculus (house mouse)Potency7.943310
N'-[2,6-bis(4-morpholinyl)-4-pyrimidinyl]-3,4-dichlorobenzohydrazideMus musculus (house mouse)Potency21.154620
[4-(diphenylmethyl)-1-piperazinyl]-[5-thiophen-2-yl-7-(trifluoromethyl)-3-pyrazolo[1,5-a]pyrimidinyl]methanoneMus musculus (house mouse)Potency3.981110
6-(4,5-dihydrothiazol-2-ylthio)-N2,N4-bis(2-methylphenyl)-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency6.694620
4-(4-bromophenyl)-3-[(4-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency3.931020
2-[2-oxo-2-(2,2,4,6-tetramethyl-1-quinolinyl)ethyl]isoindole-1,3-dioneMus musculus (house mouse)Potency11.750420
3-(2-chloro-6-fluorophenyl)-N-(3-fluoro-4-methylphenyl)-5-methyl-4-isoxazolecarboxamideMus musculus (house mouse)Potency7.079510
1-[4-(2-pyridinyl)-1-piperazinyl]-2-(9H-xanthen-9-yl)ethanoneMus musculus (house mouse)Potency35.481310
2-(1,3-benzodioxol-5-yl)-N-[(2-ethoxyphenyl)methyl]-N-(2-pyridinylmethyl)ethanamineMus musculus (house mouse)Potency19.118020
N-[4-[[[[oxo(thiophen-2-yl)methyl]amino]-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency11.220210
5-bromo-N-[3-(2-oxo-1-benzopyran-3-yl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency0.089110
3-methyl-N'-(1-oxo-2-phenoxyethyl)-1-phenyl-5-thieno[2,3-c]pyrazolecarbohydrazideMus musculus (house mouse)Potency8.539820
N-(1,3-benzodioxol-5-yl)-2-[[4-(4-methoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]acetamideMus musculus (house mouse)Potency35.481310
Silica aerogelMus musculus (house mouse)Potency5.623410
2-(4-methoxyphenyl)-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]acetamideMus musculus (house mouse)Potency6.309610
1,4-bis[(4-methoxy-2-methylphenyl)sulfonyl]-1,4-diazepaneMus musculus (house mouse)Potency12.589310
4-[(3,5-dichloro-2-hydroxyphenyl)methylamino]-1,5-dimethyl-2-phenyl-3-pyrazoloneMus musculus (house mouse)Potency35.481310
LSM-16774Mus musculus (house mouse)Potency11.220210
2-[(3-cyano-6-methoxy-2-quinolinyl)thio]-N-(2-methyl-1,3-benzothiazol-5-yl)acetamideMus musculus (house mouse)Potency11.220210
4-[4-(benzenesulfonyl)-1-piperazinyl]-2-methylquinolineMus musculus (house mouse)Potency33.552020
N-[3-chloro-4-[[2-furanyl(oxo)methyl]amino]phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideMus musculus (house mouse)Potency11.904820
2-[[5-(1-benzotriazolylmethyl)-4-methyl-1,2,4-triazol-3-yl]thio]-1-(2-fluorophenyl)ethanoneMus musculus (house mouse)Potency7.079510
N-[2,5-diethoxy-4-[[(3-methoxyanilino)-sulfanylidenemethyl]amino]phenyl]-4-methylbenzamideMus musculus (house mouse)Potency11.896120
N-[4-[[anilino(sulfanylidene)methyl]amino]-2,5-diethoxyphenyl]-4-methoxybenzamideMus musculus (house mouse)Potency7.600620
N-[2,5-diethoxy-4-[[(2-methylpropylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency6.477620
N-[4-[[anilino(sulfanylidene)methyl]amino]-2,5-diethoxyphenyl]benzamideMus musculus (house mouse)Potency5.889220
N-[2,5-diethoxy-4-[[ethylamino(sulfanylidene)methyl]amino]phenyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency16.803720
1-[(7,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-furanylmethyl)-3-(2-methoxyphenyl)thioureaMus musculus (house mouse)Potency35.481310
N-[2,5-diethoxy-4-[[(2-furanylmethylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency18.301620
4,5-dimethoxy-2-[[1-oxo-2-[(3,5,8-trimethyl-2-quinolinyl)thio]ethyl]amino]benzoic acidMus musculus (house mouse)Potency5.623410
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acidMus musculus (house mouse)Potency11.294720
5-chloro-4-(4-methylphenyl)sulfonyl-N-phenyl-2-thiazolamineMus musculus (house mouse)Potency31.622810
3-pyridinecarboxylic acid [2-(2-furanyl)-4-oxo-1-benzopyran-3-yl] esterMus musculus (house mouse)Potency30.300120
5-[2-[(4-chlorophenyl)thio]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
1-[2,5-dimethyl-1-(4-methylphenyl)-3-pyrrolyl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneMus musculus (house mouse)Potency35.481310
4-[[7-methoxy-4-oxo-2-(trifluoromethyl)-1-benzopyran-3-yl]oxy]benzoic acidMus musculus (house mouse)Potency9.106320
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterMus musculus (house mouse)Potency4.466820
N-(2,5-dimethylphenyl)-2-[[3-(4-ethylphenoxy)-4-oxo-1-benzopyran-7-yl]oxy]acetamideMus musculus (house mouse)Potency16.531120
2-(3-methylphenyl)-N-[4-(4-morpholinyl)phenyl]-4-quinazolinamineMus musculus (house mouse)Potency17.782810
4-(5,6-dimethyl-1-benzimidazolyl)-5-phenylthieno[2,3-d]pyrimidineMus musculus (house mouse)Potency5.623410
3-chloro-4-[2-(3,4-dimethoxyphenyl)ethylamino]-1-(2-phenylethyl)pyrrole-2,5-dioneMus musculus (house mouse)Potency12.589310
2-(3-chlorophenoxy)acetic acid [4-[(4-methylanilino)-oxomethyl]phenyl] esterMus musculus (house mouse)Potency3.162310
2-[[cyclohexyl(oxo)methyl]amino]-4-(3-nitrophenyl)-3-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency6.990620
2-methyl-N-(4-oxo-2-sulfanylidene-3-thiazolidinyl)benzamideMus musculus (house mouse)Potency35.481310
5-(3,4-dimethoxyphenyl)-2-(4-methylphenyl)-4-thieno[2,3-d][1,3]oxazinoneMus musculus (house mouse)Potency5.623410
3-imino-2-benzo[f][1]benzopyrancarbothioamideMus musculus (house mouse)Potency20.895420
N-(4-chlorophenyl)carbamic acid 2-pyridinylmethyl esterMus musculus (house mouse)Potency6.581220
4-bromo-N'-(3,4-dihydro-2H-pyrrol-5-yl)benzohydrazideMus musculus (house mouse)Potency5.966520
2-[(4,6-dimethyl-2-pyrimidinyl)thio]-N-(4,5-diphenyl-2-oxazolyl)acetamideMus musculus (house mouse)Potency15.586420
5-(2,4-dichlorophenyl)-N-(4-methyl-2-thiazolyl)-2-furancarboxamideMus musculus (house mouse)Potency25.665120
5-(4-fluorophenyl)sulfonyl-1-(2-methylpropyl)-4-nitro-2-propan-2-ylimidazoleMus musculus (house mouse)Potency23.350720
1-(4-bromophenyl)-4-[1-naphthalenyl(oxo)methyl]-3-pyrazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency1.995310
4-(3-bromophenyl)-2-(4-bromophenyl)-7-methylpyrazolo[3,4-d]pyridazineMus musculus (house mouse)Potency11.220210
N-(4-methylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideMus musculus (house mouse)Potency11.220210
2-amino-4-[(4-bromophenyl)methylthio]-3-azaspiro[5.5]undeca-1,4-diene-1,5-dicarbonitrileMus musculus (house mouse)Potency25.118910
(4-phenyl-1-piperazinyl)-(9H-xanthen-9-yl)methanoneMus musculus (house mouse)Potency1.122010
1-benzimidazolyl-[2-(4-methoxyphenyl)-4-quinolinyl]methanoneMus musculus (house mouse)Potency22.387220
N-(1,3-benzothiazol-2-yl)-2-(3-methoxyphenyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency4.466810
N'-[2-(4-bromo-2-methylphenoxy)-1-oxoethyl]-2-pyrazinecarbohydrazideMus musculus (house mouse)Potency18.548220
N-[(4-ethylanilino)-sulfanylidenemethyl]-3-methylbutanamideMus musculus (house mouse)Potency1.061020
N-[(2-fluoroanilino)-sulfanylidenemethyl]-2-(4-methoxyphenoxy)acetamideMus musculus (house mouse)Potency22.387210
3-[(4-bromophenoxy)methyl]-N-(5-methyl-3-isoxazolyl)benzamideMus musculus (house mouse)Potency11.464220
1-(3-methoxy-5-nitrophenyl)-3-(4-methylphenyl)ureaMus musculus (house mouse)Potency19.952610
N-(5-chloro-2-pyridinyl)-2-(3,5-dimethyl-4-nitro-1-pyrazolyl)acetamideMus musculus (house mouse)Potency4.466810
N-[4-[methyl(phenyl)sulfamoyl]phenyl]benzamideMus musculus (house mouse)Potency5.011910
3-[[(2-cyclohexyl-1,3-dioxo-5-isoindolyl)-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency0.707910
1-[[2-(3-bromo-4-methoxyphenyl)-1-oxoethyl]amino]-3-phenylthioureaMus musculus (house mouse)Potency24.035320
2-(1,3-dioxo-2-isoindolyl)-N-(4-methyl-1,3-benzothiazol-2-yl)acetamideMus musculus (house mouse)Potency25.118910
3,5-dimethoxy-N-[(2-phenylethylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency0.669420
2-(phenylmethyl)-5-[4-(phenylmethyl)-1-piperidinyl]-4-oxazolecarbonitrileMus musculus (house mouse)Potency10.000010
5-bromo-N-[3-chloro-2-(1-pyrrolidinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency0.056210
2-(2-fluorophenyl)-4-(4-fluorophenyl)sulfonyl-5-(1-piperidinyl)oxazoleMus musculus (house mouse)Potency28.183810
N-(3-carbamoyl-5-propyl-2-thiophenyl)-2-methyl-3-furancarboxamideMus musculus (house mouse)Potency0.707910
4-(2,4-dichlorophenyl)-2-[(1-oxo-2-phenylethyl)amino]-3-thiophenecarboxamideMus musculus (house mouse)Potency5.120920
N-(5-tert-butyl-3-isoxazolyl)-3-nitrobenzamideMus musculus (house mouse)Potency0.005610
4-ethyl-5-methyl-N-[1-[(3-methylphenyl)methyl]-1,2,4-triazol-3-yl]-3-thiophenecarboxamideMus musculus (house mouse)Potency8.285220
N-[5-(4-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-5-methyl-3-isoxazolecarboxamideMus musculus (house mouse)Potency35.481310
5-bromo-N-[2-(4-chlorophenyl)ethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency3.162310
N-[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]-3-pyridinecarboxamideMus musculus (house mouse)Potency1.075120
2-benzamido-4,5-dihydrobenzo[g][1]benzothiole-3-carboxamideMus musculus (house mouse)Potency0.562310
N2,N2-dimethyl-6-[[(1-phenyl-5-tetrazolyl)thio]methyl]-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency14.125410
N-(1,3-benzodioxol-5-yl)-2-[[4-(4-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]thio]acetamideMus musculus (house mouse)Potency35.481310
5-[[[4-(4-fluorophenyl)-5-(phenylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-3-thiophen-2-yl-1,2,4-oxadiazoleMus musculus (house mouse)Potency17.918020
N-(3-hydroxyphenyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideMus musculus (house mouse)Potency1.412510
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency22.387210
6-(2,3-dihydroindol-1-ylmethyl)-3-phenylthiazolo[2,3-c][1,2,4]triazoleMus musculus (house mouse)Potency11.220210
(4-chlorophenyl)-[4-(7-chloro-4-quinolinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency14.140620
3-[[[3-(1-azepanylsulfonyl)-4-chlorophenyl]-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency5.623410
2-[2-nitro-4-(trifluoromethyl)phenoxy]-N-phenylbenzamideMus musculus (house mouse)Potency5.623410
5-(2,3-dihydroindol-1-ylsulfonyl)-1,3-diethyl-2-benzimidazoloneMus musculus (house mouse)Potency18.137820
4-chloro-N-[2-(4-methylsulfonyl-1-piperazinyl)phenyl]benzamideMus musculus (house mouse)Potency22.387210
N-[[3-chloro-2-(4-morpholinyl)anilino]-sulfanylidenemethyl]-4-methoxy-3-nitrobenzamideMus musculus (house mouse)Potency3.395120
N-[[3-chloro-2-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency8.278420
1-[[4-(dimethylamino)phenyl]methyl]-1-(2-furanylmethyl)-3-(4-methoxyphenyl)thioureaMus musculus (house mouse)Potency16.271020
8-chloro-N-(4-fluorophenyl)-2-(2-pyridinyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency12.589310
N-(5-bromo-6-methyl-2-pyridinyl)-3-(2-oxo-1-benzopyran-3-yl)benzamideMus musculus (house mouse)Potency3.162310
N-(3,5-dichlorophenyl)-2-(methanesulfonamido)benzamideMus musculus (house mouse)Potency25.118910
[2-(4-propylphenyl)-4-quinolinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency12.672820
2-(3-bromophenyl)-6-methyl-N-(1,2,4-triazol-4-yl)-4-quinolinecarboxamideMus musculus (house mouse)Potency17.782810
[4-[(2-chlorophenyl)methyl]-1-piperazinyl]-(6,8-dimethyl-2-pyridin-4-yl-4-quinolinyl)methanoneMus musculus (house mouse)Potency35.481310
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(2-pyridinyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency12.589310
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency16.271020
1-(3,4-dimethoxyphenyl)sulfonyl-4-(2,6-dimethylphenyl)piperazineMus musculus (house mouse)Potency31.622810
2-[[5-(7-methoxy-2-benzofuranyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-1-(4-methoxyphenyl)ethanoneMus musculus (house mouse)Potency7.911310
[4-(2,3-dimethylphenyl)-1-piperazinyl]-(3,4,5-trimethoxyphenyl)methanoneMus musculus (house mouse)Potency31.622810
N-(4-hydroxy-3,5-dimethylphenyl)-2,5-dimethyl-3-thiophenesulfonamideMus musculus (house mouse)Potency22.535820
N-(4-methyl-2-thiazolyl)-2-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]acetamideMus musculus (house mouse)Potency35.481310
2-[[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(1,3,4-thiadiazol-2-yl)acetamideMus musculus (house mouse)Potency20.386620
2-(1-imidazolyl)-4-phenyl-6-(4-phenyl-1-piperazinyl)-1,3,5-triazineMus musculus (house mouse)Potency14.219120
N-(5-chloro-2-methylphenyl)-4-[(4-chloro-1-pyrazolyl)methyl]benzamideMus musculus (house mouse)Potency5.011910
2-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]thio]-3-phenyl-4-quinazolinoneMus musculus (house mouse)Potency6.783420
2-furanyl-[4-(4-phenoxyphenyl)sulfonyl-1-piperazinyl]methanoneMus musculus (house mouse)Potency26.632020
4-(2-methoxyphenoxy)-N-(3-pyridinyl)benzenesulfonamideMus musculus (house mouse)Potency17.782810
1-(1,2,3-benzothiadiazol-5-yl)-3-(1-naphthalenyl)ureaMus musculus (house mouse)Potency35.481310
2,4-dimethyl-N-[[4-(4-morpholinyl)anilino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency13.815420
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamineMus musculus (house mouse)Potency35.481320
1-(3-chlorophenyl)-3-(2-phenoxyphenyl)thioureaMus musculus (house mouse)Potency22.740620
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamineMus musculus (house mouse)Potency22.196920
2-(4-chlorophenyl)-N-[[2-(4-morpholinyl)anilino]-sulfanylidenemethyl]acetamideMus musculus (house mouse)Potency5.011920
3-(4-oxo-3-quinazolinyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)propanamideMus musculus (house mouse)Potency11.220210
3-(2-chlorophenyl)-5-methyl-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-isoxazolecarboxamideMus musculus (house mouse)Potency25.665120
2-phenyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-4-quinolinecarboxamideMus musculus (house mouse)Potency22.196920
4-methoxy-N-[2-[(4-nitrophenyl)methylthio]-4-oxo-3-quinazolinyl]benzamideMus musculus (house mouse)Potency35.481310
N-[[2-(4-morpholinyl)anilino]-sulfanylidenemethyl]-4-nitrobenzamideMus musculus (house mouse)Potency14.432620
N-[4-[4-(ethylsulfonylamino)-3-methoxyphenyl]-2-methoxyphenyl]ethanesulfonamideMus musculus (house mouse)Potency35.481310
3-(2,3-dimethyl-1H-indol-5-yl)-4-(3-methoxyphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency12.589310
2-[[4-(4-methoxyphenyl)-5-(2-phenylethyl)-1,2,4-triazol-3-yl]thio]-N-(phenylmethyl)acetamideMus musculus (house mouse)Potency35.481320
2,5-dimethoxy-N-(4-phenoxyphenyl)benzenesulfonamideMus musculus (house mouse)Potency11.079220
7-chloro-4-[4-(3,4-dimethylphenyl)sulfonyl-1-piperazinyl]quinolineMus musculus (house mouse)Potency35.481310
N-[(3,5-dimethoxyanilino)-sulfanylidenemethyl]-3-phenylpropanamideMus musculus (house mouse)Potency3.820920
4-(5-amino-4-phenyl-1-pyrazolyl)benzoic acidMus musculus (house mouse)Potency17.559420
5-bromo-N-[[(3-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency20.246620
3-methoxy-N-[[2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency8.285220
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-5-methyl-3-phenyl-4-isoxazolecarboxamideMus musculus (house mouse)Potency25.118910
2-methoxy-N-[[2-(1-piperidinyl)anilino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency6.990620
LSM-32435Mus musculus (house mouse)Potency28.934220
2,4,5-trimethoxy-N-(2-phenylphenyl)benzamideMus musculus (house mouse)Potency11.220210
2-imino-10-methyl-N-[2-(4-morpholinyl)ethyl]-5-oxo-1-(3-pyridinylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideMus musculus (house mouse)Potency12.589310
1-[4-[[4-(2-chloro-6-nitrophenoxy)phenyl]methoxy]phenyl]ethanoneMus musculus (house mouse)Potency27.717020
5-(2,5-dichlorophenyl)-N-(2-propyl-5-tetrazolyl)-2-furancarboxamideMus musculus (house mouse)Potency2.511910
2-[[5-(3-aminophenyl)-4-methyl-1,2,4-triazol-3-yl]thio]-1-(9H-fluoren-2-yl)ethanoneMus musculus (house mouse)Potency12.589310
4-[[(4-bromo-2-ethyl-3-pyrazolyl)-oxomethyl]amino]benzoic acid propan-2-yl esterMus musculus (house mouse)Potency35.481310
1-(4-bromophenyl)-3-(3-methylbutyl)thioureaMus musculus (house mouse)Potency6.774020
5-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxymethyl]-2-furancarboxylic acid methyl esterMus musculus (house mouse)Potency12.589310
2-(4-bromophenyl)-N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)acetamideMus musculus (house mouse)Potency35.481310
5-[2-methyl-1-(phenylmethyl)-6-(trifluoromethyl)-4-pyridinylidene]-2-sulfanylidene-1,3-diazinane-4,6-dioneMus musculus (house mouse)Potency15.848920
N-[4-[[[[(4-tert-butylphenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-2-methoxyphenyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency3.355220
[1-(2-phenoxyethyl)-3-indolyl]-(1-pyrrolidinyl)methanethioneMus musculus (house mouse)Potency21.571730
4-bromo-3-nitrobenzoic acid [2-[anilino(oxo)methyl]phenyl] esterMus musculus (house mouse)Potency22.387210
N-(9,9-dimethyl-7-oxo-8,10-dihydronaphtho[1,2-b]benzofuran-5-yl)-4-methoxybenzenesulfonamideMus musculus (house mouse)Potency8.912510
2-(4-chlorophenyl)-N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideMus musculus (house mouse)Potency27.005020
2-(4-bromophenoxy)-N-[(2-hydroxy-5-methylanilino)-sulfanylidenemethyl]acetamideMus musculus (house mouse)Potency35.481320
N-[[4-(4-chlorophenoxy)anilino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency5.745720
N-[[5-(5,7-dimethyl-1,3-benzoxazol-2-yl)-2-methylanilino]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency4.152420
N-[(3-benzamidoanilino)-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency7.811720
methimazoleMus musculus (house mouse)Potency11.220210
N-[2-(2-benzoyl-4-bromoanilino)-2-oxoethyl]-2-chlorobenzamideMus musculus (house mouse)Potency17.782810
N-cycloheptyl-2-[[2-(1,3-dioxo-2-isoindolyl)-1-oxoethyl]amino]benzamideMus musculus (house mouse)Potency7.943310
N-[[3-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency3.548110
2-[(3-bromo-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzothiazoleMus musculus (house mouse)Potency0.281810
4-(2-chlorophenyl)-3-(5-methyl-3-phenyl-4-isoxazolyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency10.157820
3-[(1,3-benzothiazol-2-ylthio)methyl]-4-cyclohexyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency0.729220
1-ethyl-3-sulfanylidene-5,6,7,8-tetrahydro-2H-isoquinoline-4-carbonitrileMus musculus (house mouse)Potency27.717020
2-(8-methoxy-2-methyl-4-oxo-1-quinolinyl)-N-(2-methoxyphenyl)acetamideMus musculus (house mouse)Potency28.183810
N-(4-methoxyphenyl)-2-(3-nitrophenyl)-4-quinazolinamineMus musculus (house mouse)Potency35.481310
2-(3,5-dinitrophenyl)-3-(2-phenylethyl)imidazo[4,5-b]quinoxalineMus musculus (house mouse)Potency3.162310
2-(5-bromo-3-nitro-1,2,4-triazol-1-yl)-N-(diphenylmethyl)acetamideMus musculus (house mouse)Potency7.600620
4-(4-methoxyphenyl)-3-(4-methylphenyl)-5-[(4-nitrophenyl)methylthio]-1,2,4-triazoleMus musculus (house mouse)Potency4.466810
2-[1-(4-tert-butylphenyl)sulfonyl-4-piperidinyl]-6-chloro-1H-benzimidazoleMus musculus (house mouse)Potency31.622810
2-[[5-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-ethyl-1,3,4-thiadiazol-2-yl)acetamideMus musculus (house mouse)Potency2.511910
4-[[3-[(2-chlorophenyl)methyl]-5-cyclopropyl-7-triazolo[4,5-d]pyrimidinyl]amino]-N,N-dimethylbenzenesulfonamideMus musculus (house mouse)Potency3.981110
1-(3,4-dimethylphenyl)-2-[[5-[[2-(4-ethoxyanilino)-4-thiazolyl]methyl]-1,3,4-oxadiazol-2-yl]thio]ethanoneMus musculus (house mouse)Potency35.481310
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[[2-(phenylmethyl)-4-quinazolinyl]thio]ethanoneMus musculus (house mouse)Potency8.154820
1-(4-fluorophenyl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneMus musculus (house mouse)Potency21.169920
N-(5-methyl-3-isoxazolyl)-2-[(2-propan-2-yl-4-quinazolinyl)thio]acetamideMus musculus (house mouse)Potency1.584910
(5-chloro-2-hydroxyphenyl)-[2-ethyl-3-(4-fluorophenyl)-6-pyrazolo[1,5-a]pyrimidinyl]methanoneMus musculus (house mouse)Potency19.952610
N-[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]-2-methoxyacetamideMus musculus (house mouse)Potency30.300120
N-[5-[(2,2-dimethyl-1-oxopropyl)amino]-2-pyridinyl]-2-furancarboxamideMus musculus (house mouse)Potency0.380920
1-[2-(5,6-dimethyl-1H-benzimidazol-2-yl)ethyl]-3-(2,5-dimethylphenyl)-1-(3-pyridinylmethyl)thioureaMus musculus (house mouse)Potency15.848910
5-tert-butyl-N-[2-(cyclopentylamino)-2-oxoethyl]-N-(2,5-dimethylphenyl)-3-methyl-2-furancarboxamideMus musculus (house mouse)Potency22.387210
N-[(4-fluorophenyl)methyl]-N-[(8-methyl-2-oxo-1H-quinolin-3-yl)methyl]-4-morpholinecarboxamideMus musculus (house mouse)Potency0.251210
2-[4-(4-chlorophenyl)sulfonyl-1-piperazinyl]-1-ethylbenzimidazoleMus musculus (house mouse)Potency35.481320
N-(2-methoxyphenyl)-2-[5-[2-[(4-methoxyphenyl)sulfonylamino]phenyl]-2-tetrazolyl]acetamideMus musculus (house mouse)Potency1.000010
4-[(2,6-dichlorophenyl)thio]-5-methoxy-2-(2-pyridinyl)pyrimidineMus musculus (house mouse)Potency6.581220
4-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]oxy]-N-propan-2-ylbenzenesulfonamideMus musculus (house mouse)Potency5.623410
4-chloro-N-(4-chloro-2-methylphenyl)-5-dithiazolimineMus musculus (house mouse)Potency23.350720
7-(4-methoxyphenyl)-2-(1-pyrrolyl)-[1,2,4]triazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency0.112210
2-[(4-chlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinoneMus musculus (house mouse)Potency19.952610
6-(4-fluorophenyl)-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileMus musculus (house mouse)Potency35.481310
1-[2-(1H-indol-3-yl)ethyl]-5,6,7,8-tetrahydroquinolin-4-oneMus musculus (house mouse)Potency1.584910
4-methyl-2-(4-nitrophenyl)-5-thiazolecarboxylic acidMus musculus (house mouse)Potency7.943310
4-[(4-chloro-1-naphthalenyl)oxy]-5-methoxy-2-(2-pyridinyl)pyrimidineMus musculus (house mouse)Potency4.601120
4-(2,6-dimethylphenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidineMus musculus (house mouse)Potency13.516020
6,7-dimethoxy-N-[(4-methylphenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency3.981110
2-[2-(2,4-dichloro-5-propan-2-yloxyanilino)-2-oxoethyl]sulfinyl-N-[3-(trifluoromethyl)phenyl]acetamideMus musculus (house mouse)Potency35.481310
4-[2-[(3,4-dichlorophenyl)methylthio]-6-[(methylthio)methyl]-4-pyrimidinyl]morpholineMus musculus (house mouse)Potency30.300120
N-[(4-chlorophenyl)methyl]-6-(3,5-dimethyl-1-pyrazolyl)-1,2,4,5-tetrazin-3-amineMus musculus (house mouse)Potency2.818410
5-[1-[(4-fluorophenyl)methyl]-3-pyrazolyl]-2-phenylthiazoleMus musculus (house mouse)Potency3.981110
4-(4-chlorophenyl)sulfinyl-6-(methoxymethyl)-2-methylpyrimidineMus musculus (house mouse)Potency5.388220
6-(4-methyl-1-piperazinyl)-2-(3,4,5-trimethoxyphenyl)-1H-benzimidazoleMus musculus (house mouse)Potency21.280420
4-(4-chlorophenyl)-1-(6-fluoro-2-pyridinyl)-3-pyrazolamineMus musculus (house mouse)Potency0.004510
4-(2-chlorophenoxy)-2-(2-pyridinyl)-6-(trifluoromethyl)pyrimidineMus musculus (house mouse)Potency17.782810
3-[2-(4-chlorophenyl)-4-thiazolyl]-4-ethyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency0.910620
N-(4-bromophenyl)-1-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-2-pyrrolecarboxamideMus musculus (house mouse)Potency31.622810
4-chloro-5-(dimethylamino)-2-(4-methylphenyl)-3-pyridazinoneMus musculus (house mouse)Potency11.904820
7-(4-chlorophenyl)-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]-[1,2,4]triazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency25.665120
3-phenyl-6-(trifluoromethyl)-1H-pyrazolo[4,3-b]pyridineMus musculus (house mouse)Potency35.481310
N-phenylcarbamic acid [5-(2-chlorophenyl)-3-isoxazolyl]methyl esterMus musculus (house mouse)Potency3.981110
1-[[2-(1,2-benzoxazol-3-yl)-1-oxoethyl]amino]-3-(4-chlorophenyl)thioureaMus musculus (house mouse)Potency11.220210
3-(4-morpholinyl)-4-(2-pyridinyl)-N-[3-(trifluoromethyl)phenyl]-1-pyrazolecarboxamideMus musculus (house mouse)Potency19.149820
2-(2,4-dichlorophenyl)-5-[2-(methylthio)phenyl]-1,3,4-oxadiazoleMus musculus (house mouse)Potency22.387210
N,N-dimethylcarbamic acid [4-[2-(benzenesulfonyl)-1-oxoethyl]-2,6-dimethylphenyl] esterMus musculus (house mouse)Potency35.481310
1,1-bis(4-chlorophenyl)-2-[(3-methoxyphenyl)methylamino]ethanolMus musculus (house mouse)Potency35.481320
N,N-dimethylcarbamic acid [4-[2-(4-fluorophenyl)sulfonyl-1-oxoethyl]-2,6-dimethylphenyl] esterMus musculus (house mouse)Potency1.122010
4-(3-chloro-2-thiophenyl)-2-(3-pyridinyl)thiazoleMus musculus (house mouse)Potency11.220210
3,4-dichloro-N-(4-chloro-3-methyl-5-isoxazolyl)benzamideMus musculus (house mouse)Potency12.431220
2-(4-chlorophenoxy)-4-(dimethylamino)-3-pyridinecarbonitrileMus musculus (house mouse)Potency11.220210
N-[1-methyl-3-(trifluoromethyl)-5-thieno[2,3-c]pyrazolyl]carbamic acid (4-fluorophenyl)methyl esterMus musculus (house mouse)Potency17.782810
2-[(2,4-dichlorophenyl)methylthio]-6,7-dimethoxy-3-(thiophen-2-ylmethyl)-4-quinazolinimineMus musculus (house mouse)Potency25.665120
7-chloro-N-(2-furanylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency24.035320
(2-methylanilino)thioureaMus musculus (house mouse)Potency10.665420
2-(4-fluorophenyl)-1-indolizinecarboxylic acid ethyl esterMus musculus (house mouse)Potency6.309610
5-(4-chlorophenyl)-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency15.848910
4-methyl-N-[(2-methyl-4-quinolinyl)methyl]-3-nitrobenzamideMus musculus (house mouse)Potency35.481310
6-methyl-5-[2-(2-methylphenoxy)ethyl]-2-sulfanylidene-1H-pyrimidin-4-oneMus musculus (house mouse)Potency19.952610
3-methyl-N-[oxo-[(2,4,6-trimethyl-3-pyridinyl)amino]methyl]benzamideMus musculus (house mouse)Potency11.220210
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-oneMus musculus (house mouse)Potency2.990420
4-chloro-N-(3,4-dimethoxyphenyl)-1-ethyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency35.481310
N2,N2-dimethyl-6-[[[1-(1-naphthalenyl)-5-tetrazolyl]thio]methyl]-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency6.309610
5-[(4-methyl-1-piperidinyl)methyl]-1-[4-(1-pyrrolyl)-1,2,5-oxadiazol-3-yl]-4-triazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
1-isonicotinoyl-4-(2-tolyl)thiosemicarbazideMus musculus (house mouse)Potency10.000010
4-(1-benzimidazolyl)-5-(4-methylphenyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency21.169920
2-chloro-1-[1-(2-furanylmethyl)-2,5-dimethyl-3-pyrrolyl]ethanoneMus musculus (house mouse)Potency12.863120
N-[2-[(phenylmethyl)amino]-1,3-benzodioxol-2-yl]carbamic acid ethyl esterMus musculus (house mouse)Potency19.952610
LSM-19448Mus musculus (house mouse)Potency3.981110
1-[[2-[[4-(4-chlorophenyl)-5-phenyl-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-3-phenylthioureaMus musculus (house mouse)Potency12.924420
2-[(3,4-dichlorophenyl)methylthio]-6-(3-pyridinyl)-3-pyridinecarbonitrileMus musculus (house mouse)Potency23.350720
N-(4-methoxyphenyl)-2-(3-methylphenoxy)-N-(4-methylphenyl)sulfonylacetamideMus musculus (house mouse)Potency28.183810
3-(4-phenylphenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepineMus musculus (house mouse)Potency8.764920
2-[[[4-(diethylsulfamoyl)phenyl]-oxomethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.125910
sulindacMus musculus (house mouse)Potency35.481310
cis-resveratrolMus musculus (house mouse)Potency7.834720
capsaicinMus musculus (house mouse)Potency35.481310
enclomipheneMus musculus (house mouse)Potency19.952610
fluoxetineMus musculus (house mouse)Potency3.548110
terbinafineMus musculus (house mouse)Potency14.125410
1,4-benzoquinone guanylhydrazone thiosemicarbazoneMus musculus (house mouse)Potency17.803610
auraptenMus musculus (house mouse)Potency7.079510
1-[[2-(1,3-benzothiazol-2-ylthio)-1-oxoethyl]amino]-3-phenylthioureaMus musculus (house mouse)Potency2.733420
N-[2-(1H-benzimidazol-2-yl)ethyl]-3,5-dinitrobenzamideMus musculus (house mouse)Potency2.238710
N-[4-(4-morpholinyl)phenyl]carbamic acid butyl esterMus musculus (house mouse)Potency0.177810
4-[[(3,6-dichloro-2-methoxyphenyl)-oxomethyl]amino]benzoic acid propyl esterMus musculus (house mouse)Potency20.552320
1-[[1-oxo-2-[[5-(phenylmethylthio)-1,3,4-thiadiazol-2-yl]thio]ethyl]amino]-3-phenylthioureaMus musculus (house mouse)Potency13.357420
N-[(phenacylamino)-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency17.782810
2-[[2-(2-methylphenoxy)ethylthio]methyl]-1H-benzimidazoleMus musculus (house mouse)Potency35.481310
2-[2-[[1-oxo-2-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]ethyl]amino]-4-thiazolyl]acetic acid ethyl esterMus musculus (house mouse)Potency11.220210
N-[(2-adamantylamino)-sulfanylidenemethyl]hexanamideMus musculus (house mouse)Potency5.091020
1-(4-fluorophenyl)-7-(4-methylphenyl)-5,5-bis(trifluoromethyl)-8H-pyrimido[4,5-d]pyrimidine-2,4-dioneMus musculus (house mouse)Potency11.220210
4-cyano-5-[[2-[[5-(2,4-dichlorophenyl)-1H-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-3-methyl-2-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency15.586420
2-chloro-N-heptyl-N-(3-methylphenyl)acetamideMus musculus (house mouse)Potency22.387220
1-[[3-(9-carbazolyl)-1-oxopropyl]amino]-3-(2-methylprop-2-enyl)thioureaMus musculus (house mouse)Potency14.733420
4-(4-methylphenyl)-2-[[oxo-(2-oxo-1-benzopyran-3-yl)methyl]amino]-3-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481320
4-(5-formyl-2-furanyl)benzoic acid propyl esterMus musculus (house mouse)Potency24.035320
4-methoxy-N-[[(1-oxo-2-phenoxyethyl)hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency21.280420
3-propoxy-N-[sulfanylidene-[3-(trifluoromethyl)anilino]methyl]benzamideMus musculus (house mouse)Potency16.193620
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneMus musculus (house mouse)Potency17.488220
N-[4-[[(1-oxohexylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency22.740620
N-[[3-chloro-4-(1-piperidinyl)anilino]-sulfanylidenemethyl]hexanamideMus musculus (house mouse)Potency4.332220
3-(5,8-dinitro-1,3-dioxo-2-benzo[de]isoquinolinyl)benzoic acidMus musculus (house mouse)Potency13.534620
2-(benzenesulfonamido)acetic acid [2-(4-nitrophenyl)-2-oxoethyl] esterMus musculus (house mouse)Potency5.623410
4-methyl-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency11.124820
N-[(benzenesulfonylhydrazo)-sulfanylidenemethyl]-4-methylbenzamideMus musculus (house mouse)Potency8.643820
3-chloro-N-[3-[[(3-chloro-4-nitrophenyl)-oxomethyl]amino]-2,2-dimethylpropyl]-4-nitrobenzamideMus musculus (house mouse)Potency5.317720
N-[[[2-(2-methoxyphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency15.848910
4-butyl-3-(5-ethyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.103420
4-butyl-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.990620
1-ethyl-3-[[[2-(2-methylpropyl)-4-quinolinyl]-oxomethyl]amino]thioureaMus musculus (house mouse)Potency7.261820
4-butyl-3-(3-methyl-2-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency8.116020
1-(3-methoxyphenyl)-3-[[3-(4-nitro-1-pyrazolyl)-1-oxopropyl]amino]thioureaMus musculus (house mouse)Potency2.511910
N-cyano-N'-(2-fluorophenyl)carbamimidothioic acid [2-(tert-butylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency25.665120
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency1.806420
2-methyl-N-[[[oxo-(3,4,5-trimethoxyphenyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency12.589310
4-chloro-N-[[[oxo-(3,4,5-trimethoxyphenyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency31.832620
3-bromo-4-methoxy-N-[(propan-2-ylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency6.499220
2-[[[(3-methyl-1-oxobutyl)amino]-sulfanylidenemethyl]amino]-N-phenylbenzamideMus musculus (house mouse)Potency35.481310
4-phenyl-N-[sulfanylidene-(2,4,6-trimethylanilino)methyl]benzamideMus musculus (house mouse)Potency5.045120
1-[2-(2-methylphenoxy)ethyl]-3-phenylthioureaMus musculus (house mouse)Potency4.392820
2-butoxy-3-phenyl-4-quinazolinoneMus musculus (house mouse)Potency35.481310
1-ethyl-3-[(1-oxo-2-phenylethyl)amino]thioureaMus musculus (house mouse)Potency35.481310
N4-ethyl-6-[2-(4-methylphenoxy)ethylthio]-N2-propan-2-yl-1,3,5-triazine-2,4-diamineMus musculus (house mouse)Potency35.481310
1-ethyl-3-[[[(phenylmethyl)amino]-sulfanylidenemethyl]amino]thioureaMus musculus (house mouse)Potency21.280420
5-bromo-N-(2-fluorophenyl)-6-oxo-3-pyrancarboxamideMus musculus (house mouse)Potency35.481310
4-(2-bromo-4-methylphenyl)-3-[5-(2-furanyl)-1H-pyrazol-3-yl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency8.912510
4-(2,5-dimethoxyphenyl)-3-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency8.912510
5-tert-butyl-3-(4-chlorophenyl)-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineMus musculus (house mouse)Potency0.531720
3-(1,3-benzodioxol-5-yl)-4-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency26.632020
N-[[(5-chloro-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency27.717020
2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylamino]phenolMus musculus (house mouse)Potency7.079510
1-[[oxo(3-pyridinyl)methyl]amino]-3-(4-propan-2-ylphenyl)thioureaMus musculus (house mouse)Potency18.860020
LSM-20639Mus musculus (house mouse)Potency3.548110
3-phenyl-2-propan-2-yl[1]benzopyrano[2,3-d]pyrimidine-4,5-dioneMus musculus (house mouse)Potency19.952610
N-[[(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-5-methyl-3-phenyl-4-isoxazolecarboxamideMus musculus (house mouse)Potency3.548110
1-[2-[(3-chloro-4-methoxyphenyl)methylthio]ethyl]-3-phenylthioureaMus musculus (house mouse)Potency11.124820
2-[[2-(3,5-dimethyl-1-pyrazolyl)-6-methyl-4-pyrimidinyl]amino]ethanolMus musculus (house mouse)Potency13.131120
N'-(4-phenyl-2-thiazolyl)-N-(2-pyridinylmethyl)oxamideMus musculus (house mouse)Potency16.193620
4-[[1,2-dioxo-2-(pyridin-4-ylmethylamino)ethyl]amino]benzoic acid butyl esterMus musculus (house mouse)Potency26.632020
amn082Mus musculus (house mouse)Potency25.333720
2-amino-4-[[2-(4-bromophenyl)-2-oxoethyl]thio]-3-azaspiro[5.5]undeca-1,4-diene-1,5-dicarbonitrileMus musculus (house mouse)Potency15.848910
1-[(3,4-dichlorophenyl)methyl]indole-2,3-dioneMus musculus (house mouse)Potency35.481320
4-(phenylmethyl)-3-[2-(4-propoxyphenyl)ethyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.627120
1-[[1-oxo-3-(4-propan-2-yloxyphenyl)propyl]amino]-3-(phenylmethyl)thioureaMus musculus (house mouse)Potency10.472620
N-[3-(3-methylphenoxy)-5-nitrophenyl]-2-(3-nitro-1,2,4-triazol-1-yl)acetamideMus musculus (house mouse)Potency28.934220
N-bis(2-fluorophenoxy)phosphoryl-3,4-dimethylanilineMus musculus (house mouse)Potency19.952610
1-[[(2-chlorophenyl)-oxomethyl]amino]-3-[3-(trifluoromethyl)phenyl]thioureaMus musculus (house mouse)Potency11.294720
2-[[[2-amino-1-(3-methoxypropyl)-3-pyrrolo[3,2-b]quinoxalinyl]-oxomethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency27.717020
4-(2,4-dichlorophenoxy)-N-(3-pyridinyl)butanamideMus musculus (house mouse)Potency17.782810
1-[[(4-ethoxyanilino)-sulfanylidenemethyl]amino]-3-[3-(trifluoromethyl)phenyl]thioureaMus musculus (house mouse)Potency12.589310
2-(2-furanyl)-5-methyl-6-(phenylmethyl)-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-oneMus musculus (house mouse)Potency35.481310
7-amino-9-(phenacylthio)-8-azaspiro[4.5]deca-6,9-diene-6,10-dicarbonitrileMus musculus (house mouse)Potency3.981110
4-[[(4-tert-butylphenyl)-oxomethyl]amino]-3-methyl-2-sulfanylidene-5-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency28.183810
3-(1H-benzimidazol-2-yl)-N-(3-pyridinylmethyl)anilineMus musculus (house mouse)Potency1.258910
1-(6-methyl-2-pyridinyl)-3-(2-phenylethyl)thioureaMus musculus (house mouse)Potency1.862320
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-methoxyphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency19.149820
N-(4,5-diphenyl-2-oxazolyl)-3-methoxybenzamideMus musculus (house mouse)Potency2.837120
4,5-dichloro-1-[2-(4-chlorophenoxy)ethyl]imidazoleMus musculus (house mouse)Potency6.309610
[4-methoxy-6-(propan-2-ylamino)-1,3,5-triazin-2-yl]-[(1,1,3-trioxo-1,2-benzothiazol-2-yl)methyl]cyanamideMus musculus (house mouse)Potency35.481320
2-[5-(4-chlorophenyl)-1,3,5-dithiazinan-2-ylidene]-2-diethoxyphosphorylacetonitrileMus musculus (house mouse)Potency24.803320
3-(1-benzotriazolylmethyl)-6-thiophen-2-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleMus musculus (house mouse)Potency0.707910
2-[[[[(1-ethyl-4-pyrazolyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylic acid methyl esterMus musculus (house mouse)Potency18.446920
N-(4,5-diphenyl-2-oxazolyl)-2-[(1-methyl-5-tetrazolyl)thio]acetamideMus musculus (house mouse)Potency16.193620
4-(2,5-dimethoxyphenyl)-3-(3-phenyl-1H-pyrazol-5-yl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency21.712320
1-butyl-3-(4-phenoxyphenyl)thioureaMus musculus (house mouse)Potency3.518020
1-(3,5-dimethoxyphenyl)-3-(3-pyridinyl)thioureaMus musculus (house mouse)Potency22.740620
N-[5-methyl-2-(4-methylphenyl)-3-pyrazolyl]-2-[(7-methyl-4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-9-yl)oxy]acetamideMus musculus (house mouse)Potency35.481320
5-tert-butyl-2-methyl-3-phenyl-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineMus musculus (house mouse)Potency1.245020
2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]thio]-N-(9-ethyl-3-carbazolyl)acetamideMus musculus (house mouse)Potency16.271020
N-(4-butylphenyl)-4-(2-pyrimidinyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency14.792820
1-[2-(diethylamino)ethyl]-7,7-dimethyl-2-(4-methylphenyl)-5,8-dihydropyrano[4,3-d]pyrimidine-4-thioneMus musculus (house mouse)Potency19.952610
3-methoxy-N-[[(2-oxo-1-benzopyran-6-yl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency11.319220
2-[[1-oxo-2-(2-pyrimidinylthio)ethyl]amino]-6-(phenylmethyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency8.971620
6-(4-hydroxyphenyl)-5-(4-methoxyphenyl)-1,3-dimethylpyrrolo[3,4-d]pyrimidine-2,4-dioneMus musculus (house mouse)Potency10.000010
1-[2-[(4-chlorophenyl)thio]ethyl]-3-(2-methoxyphenyl)thioureaMus musculus (house mouse)Potency20.085020
1-(2-methoxyphenyl)-3-[2-[(4-methylphenyl)thio]ethyl]thioureaMus musculus (house mouse)Potency11.904820
N-(4-bromophenyl)-5-tert-butyl-2-methyl-4-nitro-3-pyrazolecarboxamideMus musculus (house mouse)Potency35.481310
2-tert-butyl-4-[(4-chlorophenyl)thio]-5-methyl-1H-pyrazol-3-oneMus musculus (house mouse)Potency10.000010
(4,7-dichloro-1,3-benzothiazol-2-yl)hydrazineMus musculus (house mouse)Potency14.501520
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(4-methyl-1-piperidinyl)sulfonyl]benzamideMus musculus (house mouse)Potency0.335520
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[methyl-(phenylmethyl)sulfamoyl]benzamideMus musculus (house mouse)Potency0.422020
N-(1,3-benzodioxol-5-yl)-2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideMus musculus (house mouse)Potency11.220210
3-(4-bromophenyl)-4-(4-methoxyphenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency2.375320
4-(4-morpholinylsulfonyl)-N-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)benzamideMus musculus (house mouse)Potency1.146420
1-(3-chlorophenyl)-3-(thiophen-2-ylmethyl)thioureaMus musculus (house mouse)Potency24.068220
5,6-dimethyl-N-(thiophen-2-ylmethyl)-4-thieno[2,3-d]pyrimidinamineMus musculus (house mouse)Potency10.000010
4-propan-2-ylbenzenecarbothioamideMus musculus (house mouse)Potency10.882020
N-(5-tert-butyl-2-phenyl-3-pyrazolyl)-2-[(6-methyl-1H-benzimidazol-2-yl)thio]acetamideMus musculus (house mouse)Potency7.268020
benzoic acid [2-oxo-2-[2-(phenylthio)anilino]ethyl] esterMus musculus (house mouse)Potency17.782810
N-[4-[[2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]thio]phenyl]acetamideMus musculus (house mouse)Potency25.118910
1-(2,4-dimethylphenyl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneMus musculus (house mouse)Potency10.000010
1-[(2-chlorophenyl)methyl]-3-methyl-N-(4-methyl-2-thiazolyl)-5-thieno[2,3-c]pyrazolecarboxamideMus musculus (house mouse)Potency26.632020
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-(3,4,5-trimethoxyphenyl)acetamideMus musculus (house mouse)Potency14.125410
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)thio]ethanoneMus musculus (house mouse)Potency28.183810
N-[4-[[2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]thio]phenyl]acetamideMus musculus (house mouse)Potency26.632020
2-[[6-(butylsulfamoyl)-1H-benzimidazol-2-yl]thio]-N-(2-chlorophenyl)acetamideMus musculus (house mouse)Potency19.952610
3-methyl-2-benzofurancarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] esterMus musculus (house mouse)Potency7.079510
1H-indazole-3-carboxylic acid 4-(1,3-dioxo-2-isoindolyl)butyl esterMus musculus (house mouse)Potency31.622810
N-[(2-furanylmethylamino)-oxomethyl]-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideMus musculus (house mouse)Potency35.481310
N-[(tert-butylamino)-oxomethyl]-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideMus musculus (house mouse)Potency22.387210
N-(3-cyano-2-thiophenyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]acetamideMus musculus (house mouse)Potency1.258910
2-(1,4-dioxo-3H-phthalazin-2-yl)-N-(5-methyl-4-phenyl-2-thiazolyl)acetamideMus musculus (house mouse)Potency0.794310
4-(1,3-benzothiazol-2-ylthio)butanoic acid [2-[(3-cyano-2-thiophenyl)amino]-2-oxoethyl] esterMus musculus (house mouse)Potency12.482220
N-(1,3-benzothiazol-2-yl)-3-(2,3-dihydroindol-1-ylsulfonyl)benzamideMus musculus (house mouse)Potency5.011910
N-(1H-benzimidazol-2-yl)-3-[phenyl(prop-2-enyl)sulfamoyl]benzamideMus musculus (house mouse)Potency3.642620
N-(4,5-dihydrothiazol-2-yl)-2-thiophen-2-yl-4-quinolinecarboxamideMus musculus (house mouse)Potency30.300120
N-[(tert-butylamino)-oxomethyl]-2-[4-(3-chlorophenyl)-1-piperazinyl]acetamideMus musculus (house mouse)Potency17.246720
2-(4-methoxyphenyl)-4-quinolinecarboxylic acid [2-oxo-2-(propan-2-ylamino)ethyl] esterMus musculus (house mouse)Potency0.891310
2-(2-bromophenyl)-5-[(2-chlorophenoxy)methyl]-1,3,4-oxadiazoleMus musculus (house mouse)Potency3.548110
1-(4-ethylphenyl)-3-(phenylmethyl)thioureaMus musculus (house mouse)Potency16.930820
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(cyclopropylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency18.094620
1-[1-(phenylmethyl)-4-piperidinyl]-3-(2,4,4-trimethylpentan-2-yl)thioureaMus musculus (house mouse)Potency12.062720
4-[4-(phenylmethyl)-1-piperidinyl]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency6.990620
N-[4-(4-methyl-2-thiazolyl)-2-phenyl-3-pyrazolyl]-3-(trifluoromethyl)benzamideMus musculus (house mouse)Potency35.481310
6-(4-bromophenyl)-3-methyl-1-[2-(2H-tetrazol-5-yl)ethyl]-4-(trifluoromethyl)pyrazolo[3,4-b]pyridineMus musculus (house mouse)Potency35.481320
2-[[5-[(1,3-benzothiazol-2-ylthio)methyl]-4-ethyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanoneMus musculus (house mouse)Potency14.125410
2-chloro-1-[2,5-dimethyl-1-(5-methyl-3-isoxazolyl)-3-pyrrolyl]ethanoneMus musculus (house mouse)Potency20.895420
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3-[methyl-(4-methylphenyl)sulfamoyl]benzamideMus musculus (house mouse)Potency19.118020
N-(2-methyl-1,3-benzothiazol-6-yl)-2,3-dihydro-1,4-benzodioxin-6-sulfonamideMus musculus (house mouse)Potency6.230320
4-acetyl-3,5-dimethyl-1H-pyrrole-2-carboxylic acid (5-methoxycarbonyl-2-furanyl)methyl esterMus musculus (house mouse)Potency21.712320
4-(4-chloro-2-methylphenoxy)-N-[3-(methylthio)phenyl]butanamideMus musculus (house mouse)Potency31.622810
1-(4-acetyl-3,5-dimethyl-1H-pyrrol-2-yl)-2-[[4-(difluoromethoxy)-3-methoxyphenyl]methyl-methylamino]ethanoneMus musculus (house mouse)Potency2.818410
2-ethoxy-3-pyridinecarboxylic acid [2-[1-(2-furanylmethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterMus musculus (house mouse)Potency19.952610
1-[2-[2,5-dimethyl-1-(phenylmethyl)-3-pyrrolyl]-2-oxoethyl]pyrrolidine-2,5-dioneMus musculus (house mouse)Potency17.782810
N-[4-(2,5-dimethoxyphenyl)-2-thiazolyl]-2-[(4-nitrophenyl)thio]acetamideMus musculus (house mouse)Potency5.623410
2-(1H-benzimidazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneMus musculus (house mouse)Potency11.294720
1-(4-bromo-2-fluorophenyl)-3-(3-chlorophenyl)ureaMus musculus (house mouse)Potency22.387210
(3,4-dimethoxyphenyl)-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]methanoneMus musculus (house mouse)Potency19.952610
1-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]-2-(2-methyl-4-thiazolyl)ethanoneMus musculus (house mouse)Potency22.387210
3-[(4-acetyl-1-piperazinyl)sulfonyl]-N-(1H-benzimidazol-2-yl)benzamideMus musculus (house mouse)Potency35.481310
3-(phenylmethyl)-2-sulfanylidene-1H-thieno[3,2-d]pyrimidin-4-oneMus musculus (house mouse)Potency2.298420
2-phenylacetic acid [2-[4-[(4-ethoxyanilino)-oxomethyl]anilino]-2-oxoethyl] esterMus musculus (house mouse)Potency5.623410
2-chloro-N-(2-phenyl-5-propyl-3-pyrazolyl)acetamideMus musculus (house mouse)Potency27.717020
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-quinolinecarboxamideMus musculus (house mouse)Potency0.854020
N-(3,4-dihydro-2H-pyrrol-5-yl)-5-phenyl-1,3,4-oxadiazol-2-amineMus musculus (house mouse)Potency7.079510
N-(3,4-dihydro-2H-pyrrol-5-yl)-5-(2-furanyl)-1,3,4-oxadiazol-2-amineMus musculus (house mouse)Potency12.589310
4-(4-tert-butylphenoxy)-N-(4,5-dihydrothiazol-2-yl)butanamideMus musculus (house mouse)Potency27.717020
N-(1H-benzimidazol-2-yl)-3-[methyl-(4-methylphenyl)sulfamoyl]benzamideMus musculus (house mouse)Potency1.190420
N-[(2S)-1-(1H-benzimidazol-2-ylamino)-3-methyl-1-oxobutan-2-yl]-3,5-dimethoxybenzamideMus musculus (house mouse)Potency35.481320
5-(3,4-dimethoxyphenyl)-3-(4-methoxyphenyl)-1H-imidazole-2-thioneMus musculus (house mouse)Potency5.997620
5-(3,4-dimethoxyphenyl)-3-(4-ethoxyphenyl)-1H-imidazole-2-thioneMus musculus (house mouse)Potency2.620020
4-[2-[[3-(4-methylphenyl)-5-triazolo[1,5-a]quinazolinyl]amino]ethyl]benzenesulfonamideMus musculus (house mouse)Potency0.631010
5-[(4-fluorophenyl)methyl]-7-(4-methylphenyl)sulfonyl-[1,3]dioxolo[4,5-g]quinolin-8-oneMus musculus (house mouse)Potency35.481310
N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency10.736220
N-(4-acetylphenyl)-5-[(phenylthio)methyl]-2-furancarboxamideMus musculus (house mouse)Potency14.125410
3-cyclohexyl-N-(1,3-dimethyl-2,6-dioxo-4-pyrimidinyl)propanamideMus musculus (house mouse)Potency3.981110
3-phenyl-2-sulfanylidene-1H-benzofuro[3,2-d]pyrimidin-4-oneMus musculus (house mouse)Potency6.477620
N-(3,5-dimethylphenyl)-2-[(4-oxo-3-phenyl-2-benzofuro[3,2-d]pyrimidinyl)thio]acetamideMus musculus (house mouse)Potency0.446710
(4-tert-butylphenyl)-[2-(4-fluorophenyl)-8-methyl-3-sulfanylidene-1,4,8-triazaspiro[4.5]dec-1-en-4-yl]methanoneMus musculus (house mouse)Potency24.035320
5-[[2-[(3-methylphenyl)methyl]-1-oxo-3,4-dihydroisoquinolin-5-yl]oxymethyl]-2-furancarboxylic acid methyl esterMus musculus (house mouse)Potency28.183810
5-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethoxy]-2-[(3-methylphenyl)methyl]-3,4-dihydroisoquinolin-1-oneMus musculus (house mouse)Potency35.481310
2-[[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-oxomethyl]imino-1-(2-methylpropyl)-5-oxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency4.466810
2-[[3-(4-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetic acid ethyl esterMus musculus (house mouse)Potency12.589310
N-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[methyl(phenyl)sulfamoyl]benzamideMus musculus (house mouse)Potency0.504520
4-[bis(2-methoxyethyl)sulfamoyl]-N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)benzamideMus musculus (house mouse)Potency4.007520
4-(dipropylsulfamoyl)-N-[5-[(methylthio)methyl]-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency1.075120
4-[butyl(methyl)sulfamoyl]-N-[5-[(methylthio)methyl]-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.958220
4-[ethyl-(phenylmethyl)sulfamoyl]-N-(5-methyl-1,3,4-oxadiazol-2-yl)benzamideMus musculus (house mouse)Potency0.562320
3-[[(2,3-dimethylanilino)-sulfanylidenemethyl]amino]-1H-indole-2-carboxylic acid ethyl esterMus musculus (house mouse)Potency33.552020
1-[2-(2,5-dimethyl-1H-indol-3-yl)ethyl]-3-methyl-1-(thiophen-2-ylmethyl)thioureaMus musculus (house mouse)Potency23.350720
1-[2-(5-fluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)thioureaMus musculus (house mouse)Potency11.220210
4-[ethyl-(phenylmethyl)sulfamoyl]-N-[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.277220
4-[bis(2-methylpropyl)sulfamoyl]-N-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.318320
1-[4-(benzenesulfonyl)-1-piperazinyl]-2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]ethanoneMus musculus (house mouse)Potency19.952610
N-[2-(methylthio)-1,3-benzothiazol-6-yl]-2-furancarboxamideMus musculus (house mouse)Potency19.952610
N-[(2S)-1-(1H-benzimidazol-2-ylamino)-3-methyl-1-oxobutan-2-yl]-3-methylbenzamideMus musculus (house mouse)Potency20.386620
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterMus musculus (house mouse)Potency1.584910
2-[[oxo-(2,3,4,5,6-pentafluorophenyl)methyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency7.943310
1-ethyl-3-[(1-oxo-2,2-diphenylethyl)amino]thioureaMus musculus (house mouse)Potency7.191220
1-[2-[(4-chlorophenyl)thio]ethyl]-3-(2,4-dimethylphenyl)thioureaMus musculus (house mouse)Potency0.897220
1-(3,5-dimethylphenyl)-3-(3-ethoxypropyl)thioureaMus musculus (house mouse)Potency8.154820
1-(2,4-dimethylphenyl)-3-[2-[(4-methylphenyl)thio]ethyl]thioureaMus musculus (house mouse)Potency5.745720
1-[2,3-bis(2-pyridinyl)-6-quinoxalinyl]-3-propylthioureaMus musculus (house mouse)Potency10.000010
1-[2-[(2-methylphenyl)methylthio]ethyl]-3-phenylthioureaMus musculus (house mouse)Potency4.659120
thiocyanic acid [2-(1-naphthalenyl)-2-oxoethyl] esterMus musculus (house mouse)Potency23.350720
mcb-613Mus musculus (house mouse)Potency3.700820
2-[2-(1-naphthalenyloxy)ethylthio]pyrimidineMus musculus (house mouse)Potency10.665420
2-[2-(4-chlorophenoxy)ethylthio]pyrimidineMus musculus (house mouse)Potency4.220920
N-(4-cyclohexylphenyl)-2-(2-hydroxyethylthio)acetamideMus musculus (house mouse)Potency16.973930
5-bromo-N-[[(4-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency4.392820
6-bromo-3-[4-nitro-3-(trifluoromethyl)phenyl]-2-propyl-4-quinazolinoneMus musculus (house mouse)Potency29.903320
2-bromo-N-(9-fluorenylideneamino)benzamideMus musculus (house mouse)Potency8.539820
3-methoxy-N-[2-(3-methoxyphenoxy)ethyl]benzamideMus musculus (house mouse)Potency22.387210
1-[3-(4-phenylphenoxy)propyl]-1,2,4-triazoleMus musculus (house mouse)Potency3.162310
2,5-dimethoxybenzenesulfonic acid (1,3-dioxo-2-isoindolyl) esterMus musculus (house mouse)Potency6.783420
2-(2-bromo-4-tert-butylphenoxy)-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency35.481310
2-[2-nitro-4-(trifluoromethyl)phenyl]sulfinylacetic acid (4-chlorophenyl) esterMus musculus (house mouse)Potency24.803320
1-[[(4-ethyl-5-methyl-3-thiophenyl)-oxomethyl]amino]-3-(2-phenylethyl)thioureaMus musculus (house mouse)Potency35.481320
1-(4-bromo-2-chlorophenyl)-3-[[oxo(pyridin-4-yl)methyl]amino]thioureaMus musculus (house mouse)Potency19.952610
N-[4-(diethylsulfamoyl)phenyl]-4-(4-morpholinylmethyl)benzamideMus musculus (house mouse)Potency5.623410
N-[[(cyclohexylamino)-sulfanylidenemethyl]amino]carbamic acid tert-butyl esterMus musculus (house mouse)Potency11.220210
4-butyl-3-(phenylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency35.481310
1-[[(4-bromo-2-methyl-3-pyrazolyl)-oxomethyl]amino]-3-(2-methoxy-5-methylphenyl)thioureaMus musculus (house mouse)Potency1.995310
4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-[4-(1-pyrrolidinylsulfonyl)phenyl]benzamideMus musculus (house mouse)Potency3.518020
1-(4-bromo-2-chlorophenyl)-3-(3-methyl-2-pyridinyl)thioureaMus musculus (house mouse)Potency4.795720
2-[4-[2-(1-cyclohexenyl)ethylsulfamoyl]-2-methylphenoxy]acetic acid methyl esterMus musculus (house mouse)Potency35.481320
[5-[(4-methoxyphenyl)methylamino]-3-phenyl-1,2,4-triazol-1-yl]-(4-nitrophenyl)methanoneMus musculus (house mouse)Potency1.122010
2-[[5-[3-(2,4-dichlorophenoxy)propyl]-4-methyl-1,2,4-triazol-3-yl]thio]-N-(2-ethyl-6-methylphenyl)acetamideMus musculus (house mouse)Potency31.622810
N-[(3-ethoxy-2-prop-2-enoxyphenyl)methyl]-2-thiazolamineMus musculus (house mouse)Potency16.803720
2-[[1-oxo-2-(1H-1,2,4-triazol-5-ylthio)ethyl]amino]-4-thiophen-2-yl-3-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency19.321820
N-[[[2-(2-bromo-4-propan-2-ylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency6.309620
N-[5-(2-methoxyethylthio)-1,3,4-thiadiazol-2-yl]-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency5.623410
2-butoxy-7-hydroxy-9-fluorenoneMus musculus (house mouse)Potency14.432620
6-bromo-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-pyridinyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency21.169920
5-bromo-N-[2-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency1.000010
1-(4-bromophenyl)-3-[2-(2-methoxyphenoxy)ethyl]ureaMus musculus (house mouse)Potency8.912510
3-(3-bromoanilino)-1-(5-methyl-2-furanyl)-1-propanoneMus musculus (house mouse)Potency35.481310
3-[1-(3-methoxypropyl)-5-thiophen-2-yl-2-pyrrolyl]propanoic acidMus musculus (house mouse)Potency35.481310
1-(3-chlorophenyl)-3-[3-[methyl(methylsulfonyl)amino]phenyl]ureaMus musculus (house mouse)Potency11.220210
N-[[[[4-[(2-methyl-1-oxopropyl)amino]phenyl]-oxomethyl]hydrazo]-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency11.220210
3-chloro-N-[3-(4-morpholinyl)propyl]-6-nitro-1-benzothiophene-2-carboxamideMus musculus (house mouse)Potency8.912510
N-[(3-bromoanilino)-sulfanylidenemethyl]-3-phenylpropanamideMus musculus (house mouse)Potency23.350720
N-[4-(cyanomethyl)phenyl]-4-cyclohexylbenzenesulfonamideMus musculus (house mouse)Potency25.118910
8-quinolinecarboxylic acid phenyl esterMus musculus (house mouse)Potency3.246520
N-[[3-chloro-2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]butanamideMus musculus (house mouse)Potency4.169220
N-(4-ethoxyphenyl)-4-[[4-(methylthio)phenyl]sulfonylamino]benzenesulfonamideMus musculus (house mouse)Potency3.162310
N-(4-chlorophenyl)-4-methyl-2-thiazolamineMus musculus (house mouse)Potency19.952610
1-(3-fluorophenyl)-4-(4-hydroxy-3-methoxy-5-nitrophenyl)-4H-pyridine-3,5-dicarboxylic acid diethyl esterMus musculus (house mouse)Potency12.589310
3-bromo-N-[(2-hydroxyethylamino)-sulfanylidenemethyl]-4-methoxybenzamideMus musculus (house mouse)Potency0.958220
2-[[5-(2-benzofuranyl)-4-(phenylmethyl)-1,2,4-triazol-3-yl]thio]acetamideMus musculus (house mouse)Potency35.481310
N-[[[(2,4-dichlorophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2,2-dimethylpropanamideMus musculus (house mouse)Potency12.191220
4-phenyl-3-[2-(phenylmethylthio)ethyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency2.818410
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneMus musculus (house mouse)Potency16.271020
[3,5-bis[(phenylmethyl)amino]-1,2,4-triazol-1-yl]-thiophen-2-ylmethanoneMus musculus (house mouse)Potency5.623410
4-chloro-N-[(2-methylpropylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency19.731220
5-[2-(2-methoxyphenoxy)ethylthio]-1-(4-methylphenyl)tetrazoleMus musculus (house mouse)Potency15.848910
1,3-dimethyl-5-[[5-(phenylthio)-2-furanyl]methylidene]-1,3-diazinane-2,4,6-trioneMus musculus (house mouse)Potency35.481310
N-(2,1,3-benzothiadiazol-4-yl)-5-(3-chlorophenyl)-2-furancarboxamideMus musculus (house mouse)Potency24.803320
N-(3-acetylphenyl)-2-naphthalenecarboxamideMus musculus (house mouse)Potency13.534620
2-(2,4-dichloro-6-methylphenoxy)-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency33.552020
4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-[4-(1-piperidinylsulfonyl)phenyl]benzamideMus musculus (house mouse)Potency19.974020
3,4-dimethyl-N-[sulfanylidene-[2-(trifluoromethyl)anilino]methyl]benzamideMus musculus (house mouse)Potency7.550620
8-[2-(4-chloro-3,5-dimethylphenoxy)ethoxy]quinolineMus musculus (house mouse)Potency19.952610
3,4-dimethoxy-N-[4-(2,2,3,3-tetrafluoropropoxy)-3-(trifluoromethyl)phenyl]benzamideMus musculus (house mouse)Potency25.118910
5-[[2-methoxy-4-(4-morpholinyl)phenyl]methylidene]-1,3-diazinane-2,4,6-trioneMus musculus (house mouse)Potency0.891310
8-[3-(3,4-dimethylphenoxy)propoxy]quinolineMus musculus (house mouse)Potency24.803320
N-[2-(4-tert-butylphenoxy)ethyl]-2-(4-fluorophenyl)acetamideMus musculus (house mouse)Potency25.118910
4-chloro-N-[(phenacylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency11.294720
2-chloro-N-[(2-pyrimidinylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency9.043820
N-[(phenacylamino)-sulfanylidenemethyl]cyclohexanecarboxamideMus musculus (house mouse)Potency21.712320
N-[[(1-oxo-3-phenylpropyl)hydrazo]-sulfanylidenemethyl]pentanamideMus musculus (house mouse)Potency11.220210
N1-phenethylhydrazine-1-carbothioamideMus musculus (house mouse)Potency6.774020
N-[4-[(4,6-dimethyl-2-pyrimidinyl)sulfamoyl]phenyl]-2-phenyl-4-quinolinecarboxamideMus musculus (house mouse)Potency12.589310
1-[2-[3-(1-methylethenyl)phenyl]propan-2-yl]-3-(4-methyl-2-pyridinyl)ureaMus musculus (house mouse)Potency11.220220
N-(1H-benzimidazol-2-yl)-4-(dimethylsulfamoyl)benzamideMus musculus (house mouse)Potency23.350720
4-amino-N-(2-methoxyphenyl)benzamideMus musculus (house mouse)Potency7.943310
N'-(3,4-dihydro-2H-pyrrol-5-yl)-2-(2-naphthalenylamino)acetohydrazideMus musculus (house mouse)Potency3.399820
N-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethenyl]-4-morpholinecarboxamideMus musculus (house mouse)Potency12.313020
3-[2-(4-fluorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineMus musculus (house mouse)Potency7.191220
4-(difluoromethoxy)-N-[5-[[4-(difluoromethylthio)phenyl]methyl]-2-thiazolyl]benzamideMus musculus (house mouse)Potency12.589310
2-(4,6-dimethyl-2-pyrimidinyl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamineMus musculus (house mouse)Potency3.109920
5-chloro-N-(3,4-dimethylphenyl)-2,1-benzothiazole-3-carboxamideMus musculus (house mouse)Potency3.162310
N-[[2-(diethylamino)ethylamino]-sulfanylidenemethyl]-3-(4-methoxyphenyl)-1-phenyl-4-pyrazolecarboxamideMus musculus (house mouse)Potency9.834420
3-(4-methoxyphenyl)-N-[[[oxo(pyridin-4-yl)methyl]hydrazo]-sulfanylidenemethyl]-1-phenyl-4-pyrazolecarboxamideMus musculus (house mouse)Potency6.309610
[[2-[[4-(4-bromophenyl)-2-thiazolyl]amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esterMus musculus (house mouse)Potency5.660820
3-methyl-N,1-diphenyl-4-pyrazolecarbothioamideMus musculus (house mouse)Potency11.220210
N-[2-[5-(1,3-benzothiazol-2-yl)-3-ethyl-1-phenyl-2-benzimidazol-3-iumyl]ethenyl]-N-methylanilineMus musculus (house mouse)Potency126.483620
N-[5-(1,3-benzodioxol-5-ylmethyl)-4-methyl-2-thiazolyl]-4-chlorobenzamideMus musculus (house mouse)Potency27.717020
1-(2-chlorophenyl)-3-[[(1-ethyl-2-methyl-5-benzimidazolyl)-oxomethyl]amino]thioureaMus musculus (house mouse)Potency15.586420
N2-(4-methylphenyl)benzene-1,2-diamineMus musculus (house mouse)Potency11.220210
6-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]-2-[3-(trifluoromethyl)phenyl]benzo[de]isoquinoline-1,3-dioneMus musculus (house mouse)Potency19.321820
1-[4-(difluoromethylthio)phenyl]-3-(phenylmethyl)thioureaMus musculus (house mouse)Potency14.501520
2-[(4-ethoxyphenyl)sulfonylamino]-N-[2-(4-morpholinyl)phenyl]benzamideMus musculus (house mouse)Potency6.309610
3-[(2-adamantylamino)-oxomethyl]-1-methylsulfonyl-1-pentylureaMus musculus (house mouse)Potency0.794310
2-(methylthio)-3-pyridinecarboxylic acid [2-[2-(4-morpholinyl)-5-(trifluoromethyl)anilino]-2-oxoethyl] esterMus musculus (house mouse)Potency35.481310
5,6,7,8-tetrafluoro-2-(2,3,4,5,6-pentafluorophenyl)-4h-1-benzopyran-4-oneMus musculus (house mouse)Potency2.837120
4-(4-chlorophenyl)-4-oxobutanoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency35.481310
3-methyl-5-[[1-oxo-2-(2-pyridinylmethylamino)ethyl]amino]thiophene-2,4-dicarboxylic acid diethyl esterMus musculus (house mouse)Potency11.896120
N-[[2-(1-cyclohexenyl)ethylamino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency19.974020
12-oxo-N-(4-phenyl-2-thiazolyl)-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazoline-3-carboxamideMus musculus (house mouse)Potency5.158120
2-[(4-cyanophenyl)methylthio]-N-(2-methoxyphenyl)-1,3-benzoxazole-5-sulfonamideMus musculus (house mouse)Potency12.672820
1-(2-tert-butylphenyl)-3-cyclohexylthioureaMus musculus (house mouse)Potency4.044020
1-(5-isoquinolinyl)-3-(2-phenylethyl)thioureaMus musculus (house mouse)Potency4.739420
2-[4-(4-chlorophenyl)-2-thiazolyl]ethanethioamideMus musculus (house mouse)Potency7.506020
N-(2-cyanophenyl)-2-[(5,7-dibromo-8-quinolinyl)oxy]acetamideMus musculus (house mouse)Potency16.271020
2-[[5-(4-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-N-[4-(4-morpholinylsulfonyl)phenyl]acetamideMus musculus (house mouse)Potency35.481310
N-(3,5-dichloro-2-pyridinyl)-2-methoxy-4-(methylthio)benzamideMus musculus (house mouse)Potency6.309610
4-(diethylsulfamoyl)benzoic acid [2-[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]-2-oxoethyl] esterMus musculus (house mouse)Potency1.455020
2,3-dihydro-1,4-dioxin-5-carboxylic acid [2-[4-[4-(2-methylbutan-2-yl)phenoxy]anilino]-2-oxoethyl] esterMus musculus (house mouse)Potency12.589310
2-[(4-methylphenyl)-oxomethyl]benzoic acid [2-(3-nitroanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency35.481320
4-(dimethylamino)benzoic acid [2-(2-methoxyphenyl)-2-oxoethyl] esterMus musculus (house mouse)Potency1.584910
3-(1-azepanylsulfonyl)-4-chloro-N-(1H-1,2,4-triazol-5-yl)benzamideMus musculus (house mouse)Potency1.412510
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-methoxy-5-methylphenyl)benzamideMus musculus (house mouse)Potency35.481310
1-[1-(2-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-(4-methyl-1-piperidinyl)ethanoneMus musculus (house mouse)Potency5.045120
2-[2-(4-fluoroanilino)-4-thiophen-2-yl-5-thiazolyl]acetic acidMus musculus (house mouse)Potency35.481310
2-(1H-benzimidazol-2-ylthio)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamideMus musculus (house mouse)Potency3.162310
2-ethoxy-3-pyridinecarboxylic acid (4-methoxycarbonylphenyl)methyl esterMus musculus (house mouse)Potency5.623410
4-hexyl-3-thiophen-2-yl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency4.537420
N,N-diethyl-2-[(4-fluorophenyl)methylthio]-1,3-benzoxazole-5-sulfonamideMus musculus (house mouse)Potency6.783420
1-(4-ethoxyphenyl)-3-(5-isoquinolinyl)thioureaMus musculus (house mouse)Potency26.632020
1-[1-(phenylmethyl)-4-piperidinyl]-3-(2-propan-2-ylphenyl)thioureaMus musculus (house mouse)Potency14.987220
1-(2,6-dimethylphenyl)-3-[3-(2-oxo-1-pyrrolidinyl)propyl]thioureaMus musculus (house mouse)Potency20.483920
2-[(1-oxido-2-pyridin-1-iumyl)thio]-1-(4-phenylphenyl)ethanoneMus musculus (house mouse)Potency35.481310
N-[(1-adamantylamino)-oxomethyl]-2-chloroacetamideMus musculus (house mouse)Potency22.387220
n-benzyl-n,1-dimethyl-2-propynylamineMus musculus (house mouse)Potency2.818410
4-chloro-3-[(4-chlorophenyl)sulfamoyl]-N-(1H-1,2,4-triazol-5-yl)benzamideMus musculus (house mouse)Potency24.068220
3-[2-(4-chlorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineMus musculus (house mouse)Potency19.321820
1-[[2-(1H-benzimidazol-2-ylthio)-1-oxoethyl]amino]-3-ethylthioureaMus musculus (house mouse)Potency8.285220
5-methyl-N-(4-propan-2-ylphenyl)-2-pyrazinecarboxamideMus musculus (house mouse)Potency5.011910
3-[2-(cyclohexylamino)-4-(4-methoxyphenyl)-5-thiazolyl]propanoic acid methyl esterMus musculus (house mouse)Potency19.952610
2-(thiophen-2-ylsulfonylamino)benzoic acid [2-(cyclohexylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency0.177810
1-(2-fluorophenyl)-1-cyclopentanecarboxylic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterMus musculus (house mouse)Potency4.466810
N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)-4-oxo-4-thiophen-2-ylbutanamideMus musculus (house mouse)Potency14.125410
3-(4-tert-butylphenoxy)-N-(4,5-dihydrothiazol-2-yl)propanamideMus musculus (house mouse)Potency6.230320
2-(4-methoxyphenyl)-5-(2-methylpropylthio)-1,3,4-oxadiazoleMus musculus (house mouse)Potency15.848910
4-(1H-benzimidazol-2-ylthio)butanoic acid [2-oxo-2-(4-phenoxyanilino)ethyl] esterMus musculus (house mouse)Potency22.387210
N-(2-methoxyphenyl)-2-(2-oxopropylthio)-1,3-benzoxazole-5-sulfonamideMus musculus (house mouse)Potency24.035320
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideMus musculus (house mouse)Potency28.934220
N-(2-phenylethyl)-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency20.483920
thiocyanic acid [4-[(2-chloro-1-oxoethyl)amino]-3,5-dimethylphenyl] esterMus musculus (house mouse)Potency4.280020
N-(3-chloro-2-quinoxalinyl)-2-naphthalenesulfonamideMus musculus (house mouse)Potency35.481310
2-(4-chlorophenyl)-N-[4-(difluoromethylthio)phenyl]acetamideMus musculus (house mouse)Potency14.125410
2-[[[[(4-fluorophenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-4-(5-methyl-2-furanyl)-3-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency2.470320
5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylic acid [2-[2-(3,4-diethoxyphenyl)ethylamino]-2-oxoethyl] esterMus musculus (house mouse)Potency5.623410
N-[4-(1-piperidinyl)phenyl]-2-quinolinecarboxamideMus musculus (house mouse)Potency0.707910
2-[[5-(1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]thio]-N-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]acetamideMus musculus (house mouse)Potency19.731220
2-chloro-N-[3-[(2-chlorophenyl)methyl]-2-thiazolylidene]acetamideMus musculus (house mouse)Potency24.803320
4-[4-(2,3,5,6-Tetramethylphenyl)sulfonylpiperazine-1-carbonyl]-1H-quinolin-2-oneMus musculus (house mouse)Potency35.481310
2-[4-[benzenesulfonyl(methyl)amino]phenoxy]-N-(1,3-benzothiazol-2-yl)acetamideMus musculus (house mouse)Potency5.120920
N-[4-bromo-3-(trifluoromethyl)phenyl]-2,4,6-trimethylbenzamideMus musculus (house mouse)Potency35.481320
2-(2-methyl-1-benzimidazolyl)acetic acid [2-(2-methyl-1H-indol-3-yl)-2-oxoethyl] esterMus musculus (house mouse)Potency19.952610
2-[(2-hydroxy-1-naphthalenyl)methyl-methylamino]-N-[4-(4-morpholinyl)phenyl]acetamideMus musculus (house mouse)Potency1.778310
3-(1,3-benzodioxol-5-yl)-4-phenyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency10.066420
2-[[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]thio]-1-(2-methoxyphenyl)ethanoneMus musculus (house mouse)Potency24.803320
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4-methyl-5-phenyl-2-thiazolyl)-N-prop-2-enylacetamideMus musculus (house mouse)Potency24.035320
1-(2,6-diethylphenyl)-3-[2-(3,4-dihydroxyphenyl)ethyl]thioureaMus musculus (house mouse)Potency12.589310
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4,5-diphenyl-2-thiazolyl)acetamideMus musculus (house mouse)Potency7.511420
4-[(1-methyl-5-tetrazolyl)thio]-5-phenylthieno[2,3-d]pyrimidineMus musculus (house mouse)Potency11.220210
N-[4-(difluoromethylthio)phenyl]-5-[(2-hydroxy-5-methoxyphenyl)-oxomethyl]-2-imino-3-pyrancarboxamideMus musculus (house mouse)Potency35.481310
N-(4-acetamidophenyl)-2-[5-(1-piperidinylsulfonyl)-2-thiophenyl]acetamideMus musculus (house mouse)Potency11.220210
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-quinolinecarboxamideMus musculus (house mouse)Potency4.949020
1-(2-chlorophenyl)-3-(3-phenylpropyl)thioureaMus musculus (house mouse)Potency5.623410
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneMus musculus (house mouse)Potency8.285220
4,6,8-trimethyl-1H-quinoline-2-thioneMus musculus (house mouse)Potency35.481310
N-[5-[(2,6-dichlorophenyl)methylthio]-1,3,4-thiadiazol-2-yl]-5-methyl-2-pyrazinecarboxamideMus musculus (house mouse)Potency3.503620
N-(4,5,6-trifluoro-1,3-benzothiazol-2-yl)-2-furancarboxamideMus musculus (house mouse)Potency1.258910
7-[[[1-(2-methylphenyl)-5-tetrazolyl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneMus musculus (house mouse)Potency19.952610
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideMus musculus (house mouse)Potency14.976320
2-phenyl-5-thiophen-2-yl-3-pyrazolecarboxylic acid [2-(4-chloro-3-nitroanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency14.125410
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideMus musculus (house mouse)Potency27.717020
N-[[(4-oxo-1-phenyl-5-pyrazolo[3,4-d]pyrimidinyl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency31.832620
2-phenyl-5-sulfanylidene-3,7,8,9,10,11-hexahydropyrazolo[4,5]pyrimido[3,5-a]azepin-1-oneMus musculus (house mouse)Potency18.854120
2-[(6-chloro-1H-benzimidazol-2-yl)thio]-N-(2,3-dihydro-1H-inden-5-yl)acetamideMus musculus (house mouse)Potency35.481320
5-(3,4-dimethoxyphenyl)-2-methyl-4-(4-methyl-1-piperidinyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency7.079510
N-[4-(4-methylphenyl)-2-thiazolyl]-1-thiophen-2-ylsulfonyl-4-piperidinecarboxamideMus musculus (house mouse)Potency35.481310
4-acetyl-N-[4-(4-chlorophenyl)-2-thiazolyl]-3,5-dimethyl-1H-pyrrole-2-carboxamideMus musculus (house mouse)Potency5.125620
3-(4-acetylphenyl)-1-(phenylmethyl)-1-propylthioureaMus musculus (house mouse)Potency7.233420
2-anilinobenzoic acid [2-(4-acetylanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency35.481310
2-chloro-N-[(5-chloro-2-thiophenyl)methyl]-N-methylacetamideMus musculus (house mouse)Potency10.000010
N-[6-amino-2,4-dioxo-1-(phenylmethyl)-5-pyrimidinyl]-2-[(5-amino-1,3,4-thiadiazol-2-yl)thio]-N-methylacetamideMus musculus (house mouse)Potency1.000010
4-[2-(4-fluoroanilino)-2-oxoethoxy]-3-methoxy-N-[4-(4-methoxyphenyl)-5-methyl-2-thiazolyl]benzamideMus musculus (house mouse)Potency27.717020
N-(1H-benzimidazol-2-yl)-4-(3-methylphenoxy)butanamideMus musculus (house mouse)Potency14.125410
N-[[2-cyanoethyl(methyl)amino]-sulfanylidenemethyl]-4-(4-morpholinylsulfonyl)benzamideMus musculus (house mouse)Potency13.699620
5-methyl-2-(2-phenylethylamino)-4-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
4-ethyl-3-[2-(4-methylphenyl)-4-quinolinyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.122010
3-[3-[2-(2-carbamoylphenoxy)-1-oxoethyl]-2,5-dimethyl-1-pyrrolyl]propanoic acid methyl esterMus musculus (house mouse)Potency11.220210
2-hydroxy-4-methoxybenzoic acid (2-methyl-4-thiazolyl)methyl esterMus musculus (house mouse)Potency17.782810
5-bromo-N-(4-methyl-2-thiazolyl)-3-pyridinecarboxamideMus musculus (house mouse)Potency35.481310
1-(4-ethylphenyl)-3-[1-(phenylmethyl)-4-piperidinyl]thioureaMus musculus (house mouse)Potency16.193620
2-[[3-[(4-fluorophenyl)methyl]-4-oxo-2-quinazolinyl]thio]-N-(thiophen-2-ylmethyl)acetamideMus musculus (house mouse)Potency3.915220
5-(2-chlorophenyl)-2-(2-pyridinylmethyl)-3H-thieno[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency8.764920
4-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]-7-ethyl-1-benzopyran-2-oneMus musculus (house mouse)Potency5.011910
2-[[(6-chloro-4-oxo-3-prop-2-enyl-2-quinazolinyl)thio]methyl]isoindole-1,3-dioneMus musculus (house mouse)Potency8.427920
4-[[2-[[5-(3-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-1-oxoethyl]amino]benzoic acidMus musculus (house mouse)Potency14.125410
3-[(3,4-difluorophenyl)sulfonylamino]benzoic acid [2-[[(2-methylpropylamino)-oxomethyl]amino]-2-oxoethyl] esterMus musculus (house mouse)Potency19.952610
2-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]thio]-3-ethyl-5,6-dimethyl-4-thieno[2,3-d]pyrimidinoneMus musculus (house mouse)Potency11.220210
2-(2,4-dioxo-1,3-diazaspiro[4.4]nonan-3-yl)acetic acid (7-bromo-4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl esterMus musculus (house mouse)Potency3.162310
1-(2-benzofuranyl)-2-[(4-methyl-2-quinolinyl)thio]ethanoneMus musculus (house mouse)Potency12.672820
2-(2,4-dichlorophenoxy)-N-[2-(methylthio)phenyl]acetamideMus musculus (house mouse)Potency35.481310
2-(4-chlorophenyl)-5-[[(4-methyl-2-thiazolyl)thio]methyl]-1,3,4-oxadiazoleMus musculus (house mouse)Potency0.501210
4-(3,4-dimethoxyphenyl)-2-thiophen-2-ylthiazoleMus musculus (house mouse)Potency3.548110
[4-(4-bromo-2-chlorophenyl)sulfonyl-1-piperazinyl]-(2-sulfanylidene-1H-pyridin-3-yl)methanoneMus musculus (house mouse)Potency22.387210
3-(2-furanylmethyl)-4-oxo-N,N-dipropyl-2-sulfanylidene-1H-quinazoline-7-carboxamideMus musculus (house mouse)Potency15.673020
3-[5-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-1,3,4-oxadiazol-2-yl]-1-benzopyran-2-oneMus musculus (house mouse)Potency35.481310
2-oxo-1H-pyridine-3-carboxylic acid [2-(2,5-dimethyl-1-propyl-3-pyrrolyl)-2-oxoethyl] esterMus musculus (house mouse)Potency5.145420
2-Chloro-1-[2,5-dimethyl-1-(3-nitrophenyl)-1H-pyrrol-3-yl]ethan-1-oneMus musculus (house mouse)Potency22.196920
2-[4-(2-hydroxyphenyl)-1-piperazinyl]-N-(5-methyl-3-isoxazolyl)acetamideMus musculus (house mouse)Potency11.220210
1-[2,5-dimethyl-1-(phenylmethyl)-3-pyrrolyl]-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]ethanoneMus musculus (house mouse)Potency35.481310
4-hydroxybenzoic acid [2-[1-(2-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterMus musculus (house mouse)Potency5.011910
N-[4-(2-pyridinyl)-2-thiazolyl]cyclopentanecarboxamideMus musculus (house mouse)Potency22.196920
4-methyl-N'-(4-quinazolinyl)benzohydrazideMus musculus (house mouse)Potency35.481310
N-(3-pyridinylmethyl)-1,3-benzodioxol-5-amineMus musculus (house mouse)Potency19.952610
2-[[[5-methyl-4-(2-methylphenyl)-1,2,4-triazol-3-yl]thio]methyl]-1,3-benzothiazoleMus musculus (house mouse)Potency7.079510
N-ethyl-3-(1H-indol-3-yl)-N-[2-oxo-2-(thiophen-2-ylmethylamino)ethyl]propanamideMus musculus (house mouse)Potency35.481310
2,4-dithiophen-2-ylthiazoleMus musculus (house mouse)Potency19.952610
5-(3-fluorophenoxy)-8-nitroisoquinolineMus musculus (house mouse)Potency8.912510
2-chloro-N-(2-chloro-5-methylsulfonylphenyl)acetamideMus musculus (house mouse)Potency14.125410
5,6-dimethyl-N-[2-methyl-2-(4-morpholinyl)propyl]-4-thieno[2,3-d]pyrimidinamineMus musculus (house mouse)Potency26.632020
4-(4-methyl-1-piperidinyl)-5-phenyl-2-(3-pyridinyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency35.481310
N-(5-methyl-2-thiazolyl)cyclopentanecarboxamideMus musculus (house mouse)Potency25.665120
4,5-dichloro-2-[2-[2,5-dimethyl-1-(2,2,2-trifluoroethyl)-3-pyrrolyl]-2-oxoethyl]-3-pyridazinoneMus musculus (house mouse)Potency24.035320
3-(1H-indol-3-yl)propanoic acid [2-[tert-butyl-(phenylmethyl)amino]-2-oxoethyl] esterMus musculus (house mouse)Potency19.952610
2-(2,3-dihydro-1H-inden-5-yloxy)-1-(2,3-dihydroindol-1-yl)ethanoneMus musculus (house mouse)Potency12.589310
5-[[(5,6-dimethyl-4-thieno[2,3-d]pyrimidinyl)thio]methyl]-2-furancarboxylic acid methyl esterMus musculus (house mouse)Potency26.632020
2-[[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)thio]methyl]-1,3-benzothiazoleMus musculus (house mouse)Potency5.623410
4-chloro-N-[3-[(3,5-dimethyl-4-isoxazolyl)methylthio]-2-quinoxalinyl]benzenesulfonamideMus musculus (house mouse)Potency11.220210
2-(1,3-benzoxazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneMus musculus (house mouse)Potency31.622810
3-[[2-(6-methoxy-3-benzofuranyl)-1-oxoethyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency22.387210
3-(difluoromethoxy)-N-(4,5-dihydrothiazol-2-yl)benzamideMus musculus (house mouse)Potency11.220210
3-methoxy-N-(4-methyl-2-thiazolyl)benzamideMus musculus (house mouse)Potency35.481310
2-(4-methyl-1-piperidinyl)-N-[2-(phenylthio)phenyl]acetamideMus musculus (house mouse)Potency5.623410
2-[(2,4-dimethoxyphenyl)methyl-methylamino]-N-(2-methoxy-3-dibenzofuranyl)acetamideMus musculus (house mouse)Potency7.079510
thiosemicarbazideMus musculus (house mouse)Potency14.125410
5-chloro-2-mercaptobenzothiazoleMus musculus (house mouse)Potency22.106020
4-amino-5-hydrazino-1,2,4-triazole-3-thiolMus musculus (house mouse)Potency35.481320
brij-58Mus musculus (house mouse)Potency27.717020
digoxinMus musculus (house mouse)Potency1.990710
malachite greenMus musculus (house mouse)Potency0.577320
2-(1-adamantylcarbonyl)hydrazine-1-carbothioamideMus musculus (house mouse)Potency13.347720
5-anilino-3-oxo-4-isothiazolecarbonitrileMus musculus (house mouse)Potency23.350720
5-(4-chloroanilino)-3-oxo-4-isothiazolecarbonitrileMus musculus (house mouse)Potency26.632020
5-(2-chloroanilino)-3-oxo-4-isothiazolecarbonitrileMus musculus (house mouse)Potency2.210620
5-Methyl-6-(2-thienyl)-2,3,4,5-tetrahydropyridazin-3-oneMus musculus (house mouse)Potency0.631010
N-(4-bromophenyl)-4-(2-methoxyphenyl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency16.597820
3-(9-carbazolylmethyl)-4-methyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency8.068720
1-(4-tert-butylphenyl)-3-(3-pyridinylmethyl)thioureaMus musculus (house mouse)Potency25.787720
1-[[2-[5-[3,5-bis(trifluoromethyl)phenyl]-2-tetrazolyl]-1-oxoethyl]amino]-3-(4-chlorophenyl)thioureaMus musculus (house mouse)Potency16.803720
1-(4-methoxyphenyl)-3-(6-methyl-2-pyridinyl)thioureaMus musculus (house mouse)Potency2.484020
1-(3-methylphenyl)-3-(2-pyridinyl)thioureaMus musculus (house mouse)Potency3.405420
1-anilino-3-ethylthioureaMus musculus (house mouse)Potency2.344520
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency22.740620
capsazepineMus musculus (house mouse)Potency28.183810
tamoxifen citrateMus musculus (house mouse)Potency25.228820
tamoxifenMus musculus (house mouse)Potency23.735820
tetraoctylammonium bromideMus musculus (house mouse)Potency3.231120
1-butyl-3-methylimidazoliumMus musculus (house mouse)Potency22.387210
(2-bromophenyl)thioureaMus musculus (house mouse)Potency22.196920
2-[1-[2-oxo-2-[(4-thiophen-2-ylphenyl)methylamino]ethyl]cyclohexyl]acetic acidMus musculus (house mouse)Potency30.300120
5-(4-methoxyphenyl)-N-[(5-methyl-2-phenyl-4-triazolyl)methyl]-4-oxazolecarboxamideMus musculus (house mouse)Potency22.387210
2-(1,3,4-oxadiazol-2-yl)phenyl 4-chlorobenzoateMus musculus (house mouse)Potency35.481310
4-(2-fluorophenyl)-N-(2-methylbut-3-yn-2-yl)benzamideMus musculus (house mouse)Potency5.623410
N-(4-chlorophenyl)-2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolecarboxamideMus musculus (house mouse)Potency35.481310
N'-[(4-chlorophenyl)-oxomethyl]-2-methyl-4-thiazolecarbohydrazideMus musculus (house mouse)Potency19.731220
N'-benzoyl-5-(3,5-dichlorophenoxy)-2-furancarbohydrazideMus musculus (house mouse)Potency35.481310
1-[2-[(4-chlorophenoxy)methyl]-4-thiazolyl]ethanoneMus musculus (house mouse)Potency17.782810
5-cyano-2-(methoxymethyl)-6-sulfanylidene-1H-pyridine-3-carboxylic acid methyl esterMus musculus (house mouse)Potency12.589310
6-(2-methyl-3-imidazo[1,2-a]pyridinyl)-1H-pyrimidine-2-thioneMus musculus (house mouse)Potency35.481310
N-(3-chlorophenyl)-2-[[2-(2-pyridinyl)-2,3-dihydro-1,3,4-thiadiazol-5-yl]thio]acetamideMus musculus (house mouse)Potency8.068720
3-[[(2,4-dichlorophenyl)methylthio]methyl]-4-propan-2-yl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency2.287420
2-amino-6-[4-(6-chloro-2-pyridinyl)-1-piperazinyl]pyridine-3,5-dicarbonitrileMus musculus (house mouse)Potency20.552320
3-[5-[anilino(oxo)methyl]-2-furanyl]-2-thiophenecarboxylic acid methyl esterMus musculus (house mouse)Potency11.220210
[5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-yl]hydrazineMus musculus (house mouse)Potency12.589310
4-(benzenesulfonyl)-1-[(4-chlorophenyl)methyl]-4-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
3-[5-[oxo-(3-pyridinylamino)methyl]-2-furanyl]-2-thiophenecarboxylic acid methyl esterMus musculus (house mouse)Potency10.610120
1-[4-[(2-bromophenyl)-oxomethyl]-1H-pyrrol-2-yl]-2,2,2-trichloroethanoneMus musculus (house mouse)Potency22.387210
2-chloro-N-[(methylcarbamoylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency12.589310
2-chloro-N-[3-cyano-4-[(4-methoxyphenyl)thio]phenyl]benzamideMus musculus (house mouse)Potency12.589310
1H-benzimidazole-5,6-diamineMus musculus (house mouse)Potency19.952610
2-(4-fluorophenyl)-2-[4-[(4-fluorophenyl)-oxomethyl]phenyl]acetonitrileMus musculus (house mouse)Potency35.481310
t 0070907Mus musculus (house mouse)Potency22.196920
statticMus musculus (house mouse)Potency10.291820
3-chloro-1-(4-methoxyphenyl)-4-(3-methyl-1-piperidinyl)pyrrole-2,5-dioneMus musculus (house mouse)Potency35.481310
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineMus musculus (house mouse)Potency3.761920
2-[3-(4-pyridyl)-1H-1,2,4-triazol-5-yl]pyridineMus musculus (house mouse)Potency8.800620
2-[1-(1H-imidazol-1-yl)vinyl]phenolMus musculus (house mouse)Potency4.466810
3-[1-(2,4-dichlorophenyl)sulfonyl-2-pyrrolidinyl]pyridineMus musculus (house mouse)Potency12.589310
N1-{3-[2-(2-pyridyl)ethyl]phenyl}-4-chlorobenzene-1-sulfonamideMus musculus (house mouse)Potency35.481310
2-({[2-acetyl-5-(tert-butyl)-3-thienyl]amino}carbonyl)benzoic acidMus musculus (house mouse)Potency35.481310
ethyl 1-[4-(4-chlorobenzenesulfonamido)phenyl]-5-(trifluoromethyl)pyrazole-4-carboxylateMus musculus (house mouse)Potency35.481310
5-methyl-N-[1-(phenylmethyl)-4-piperidinyl]-4-thieno[2,3-d]pyrimidinamineMus musculus (house mouse)Potency2.665120
5-(4-morpholinylsulfonyl)-N-[4-(trifluoromethoxy)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency35.481310
5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamideMus musculus (house mouse)Potency23.350720
N-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-2-furancarboxamideMus musculus (house mouse)Potency4.466810
5-[[[5-(4-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esterMus musculus (house mouse)Potency35.481310
N'-(4-tert-butyl-2-thiazolyl)-4-chlorobenzohydrazideMus musculus (house mouse)Potency3.763120
1-(4-fluorophenyl)-3-[4-(4-fluorophenyl)-2-methyl-5-(trifluoromethyl)-3-pyrazolyl]ureaMus musculus (house mouse)Potency35.481310
[4-(2-methoxyphenyl)-1-piperidinyl]-(5-methyl-1-phenyl-4-pyrazolyl)methanoneMus musculus (house mouse)Potency35.481310
5-(tert-butyl)-2-methyl-N-(5-methyl-3-isoxazolyl)-3-furamideMus musculus (house mouse)Potency12.589310
4-acetamidobenzenesulfonic acid [2-(1-piperidinyl)phenyl] esterMus musculus (house mouse)Potency33.552020
2-[(7-chloro-4-quinazolinyl)oxy]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethanoneMus musculus (house mouse)Potency0.707910
N-(3-chlorophenyl)-4-(9H-fluoren-9-yl)-1-piperazinecarboxamideMus musculus (house mouse)Potency19.952610
4-[[5-ethyl-3-[(4-methoxyphenyl)-oxomethyl]-2-thiophenyl]amino]-4-oxobutanoic acidMus musculus (house mouse)Potency35.481310
2-[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazoleMus musculus (house mouse)Potency6.309610
N-[(2-hydroxyphenyl)-oxomethyl]-2,3-dihydrobenzofuran-5-carboxamideMus musculus (house mouse)Potency8.116020
4-(2-furanylmethyl)-3-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency3.548110
3-oxo-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)thio]butanoic acid ethyl esterMus musculus (house mouse)Potency1.724720
3-(2,4-dimethoxyphenyl)-6-phenyl-2-sulfanylidene-1H-thieno[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency5.313820
N'-[4-(3-methoxyphenyl)-2-thiazolyl]-2-thiophenecarbohydrazideMus musculus (house mouse)Potency6.119420
2-amino-4-(2-chlorophenyl)-6-[(4-chlorophenyl)thio]pyridine-3,5-dicarbonitrileMus musculus (house mouse)Potency25.118910
5-(4-Chloro-benzenesulfonyl)-pyrimidine-2,4-diamineMus musculus (house mouse)Potency15.848910
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileMus musculus (house mouse)Potency35.481310
3-chloro-4-propan-2-ylsulfonyl-2-thiophenecarbohydrazideMus musculus (house mouse)Potency10.000010
1-(3-chloro-4-propan-2-ylsulfonyl-2-thiophenyl)-3-(3-nitrophenyl)ureaMus musculus (house mouse)Potency3.162310
6-(2,3-dihydrobenzofuran-5-yl)-1H-pyrimidine-2-thioneMus musculus (house mouse)Potency4.736020
1-(5-tert-butyl-2-methyl-3-pyrazolyl)-3-(3,5-dichlorophenyl)ureaMus musculus (house mouse)Potency19.952610
1-(3,5-dichlorophenyl)-3-[2-(2-furanylmethylthio)ethyl]ureaMus musculus (house mouse)Potency17.782810
4-[4-(3-bromophenyl)sulfonyl-1-piperazinyl]-7-chloroquinolineMus musculus (house mouse)Potency35.481310
2-[(4-chlorophenyl)methoxy]-6-methoxybenzonitrileMus musculus (house mouse)Potency24.803320
N,N'-di[4-(2,6-dimethylmorpholino)phenyl]thioureaMus musculus (house mouse)Potency5.712220
1-tert-butyl-3-[(4-methylphenyl)sulfonylamino]thioureaMus musculus (house mouse)Potency22.196920
N-phenyl-2-benzo[g][1]benzothiolecarboxamideMus musculus (house mouse)Potency6.402620
(4-chloro-2-methylanilino)thioureaMus musculus (house mouse)Potency26.632020
2-[4-[[4-[bis(2-hydroxyethyl)amino]-2-chlorophenyl]-(2-chlorophenyl)methyl]-3-chloro-N-(2-hydroxyethyl)anilino]ethanolMus musculus (house mouse)Potency24.803320
methyl-thiohydantoin-tryptophanMus musculus (house mouse)Potency9.962520
2-[4-(2-methylpropyl)phenyl]propanoic acid [2-(1H-indol-3-yl)-2-oxoethyl] esterMus musculus (house mouse)Potency16.815820
2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-phenylacetamideMus musculus (house mouse)Potency20.246620
2-fluoro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]acetamideMus musculus (house mouse)Potency4.466810
2,4-dichloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamideMus musculus (house mouse)Potency5.623410
2-(1-naphthalenyl)-N-[2,2,2-trichloro-1-[[(2-chloroanilino)-sulfanylidenemethyl]amino]ethyl]acetamideMus musculus (house mouse)Potency25.118910
N-[(2-chloroanilino)-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency24.035320
acetic acid [4-[acetyl-(4-chlorophenyl)sulfonylamino]-1-naphthalenyl] esterMus musculus (house mouse)Potency1.739220
4-[[4-(3-methylanilino)-3,5-dinitrophenyl]-oxomethyl]-1,3-dihydroquinoxalin-2-oneMus musculus (house mouse)Potency17.782810
2-[2-[bis(4-methoxyphenyl)methylidene]hydrazinyl]benzoic acidMus musculus (house mouse)Potency24.803320
N'-[3-bicyclo[2.2.1]heptanyl(oxo)methyl]-3-chloro-1-benzothiophene-2-carbohydrazideMus musculus (house mouse)Potency23.753120
1-(4-ethoxyphenyl)-3-[methyl-(phenylmethyl)amino]pyrrolidine-2,5-dioneMus musculus (house mouse)Potency12.924420
1-(4-fluorophenyl)-3-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]pyrrolidine-2,5-dioneMus musculus (house mouse)Potency25.118910
1-(4-bromophenyl)-3-(diethylamino)pyrrolidine-2,5-dioneMus musculus (house mouse)Potency15.186120
dihydrosamidineMus musculus (house mouse)Potency10.300620
4-(5,6-diphenyl-1,2,4-triazin-3-yl)morpholineMus musculus (house mouse)Potency0.089110
3-benzylbenzothiazoliumMus musculus (house mouse)Potency23.350720
1-(4-tert-butylphenoxy)-3-(1H-1,2,4-triazol-5-ylthio)-2-propanolMus musculus (house mouse)Potency7.811720
2,2-dibromo-1-methyl-N-(2-naphthalenyl)-1-cyclopropanecarboxamideMus musculus (house mouse)Potency23.350720
5-cyclopentylidene-2-sulfanylidene-4-thiazolidinoneMus musculus (house mouse)Potency22.387210
1-(9-anthracenylmethyl)-3-piperidinolMus musculus (house mouse)Potency6.309610
1-hexadecyl-3-methylimidazolium bromideMus musculus (house mouse)Potency10.087620
1,3-bis(butylsulfonyl)-3a,4,6,6a-tetrahydro-2H-imidazo[4,5-d]imidazol-5-oneMus musculus (house mouse)Potency0.251210
N-[2-(4-chlorophenoxy)ethyl]-5-(3,5-dimethyl-1-piperazinyl)-2-nitroanilineMus musculus (house mouse)Potency17.782820
N-(2-methoxycyclohexyl)-2,5-dimethylanilineMus musculus (house mouse)Potency0.003510
3,5,7-trimethyl-N-[4-morpholinyl(sulfanylidene)methyl]-1-adamantanecarboxamideMus musculus (house mouse)Potency11.639220
1-anilino-3-[4-(3-anilino-2-hydroxypropoxy)phenoxy]-2-propanolMus musculus (house mouse)Potency31.622810
N-[2-(3-methylphenoxy)ethyl]-5-(4-morpholinyl)-2-nitroanilineMus musculus (house mouse)Potency15.848910
4-chloro-N-[2-(4-nitroanilino)ethyl]benzamideMus musculus (house mouse)Potency12.774820
N-(4-methylphenyl)-5-nitro-4-spiro[benzimidazole-2,1'-cyclohexane]amineMus musculus (house mouse)Potency7.943310
3-hydroxy-7-methyl-3-(4-morpholinyl)-5-nitro-1H-indol-2-oneMus musculus (house mouse)Potency19.702020
1-[(4-chlorophenyl)-oxomethyl]-5-hydroxy-5-phenyl-4H-pyrazole-3-carboxylic acid methyl esterMus musculus (house mouse)Potency23.350720
6-amino-4-(1,3-benzodioxol-5-yl)-5-cyano-2-methyl-4H-pyran-3-carboxylic acid 2-methoxyethyl esterMus musculus (house mouse)Potency0.281810
2,4-dichloro-6-[1-(4-morpholinyl)-3-phenylprop-2-ynyl]phenolMus musculus (house mouse)Potency12.589310
2-[[1-(4-ethoxyphenyl)-2,5-dioxo-3-pyrrolidinyl]amino]acetonitrileMus musculus (house mouse)Potency21.712320
N-(3-acetyl-2-methyl-5-benzofuranyl)-N-(4-chloro-3-nitrophenyl)sulfonylacetamideMus musculus (house mouse)Potency27.717020
N'-[(4-methoxyphenyl)methyl]-N-phenylcarbamimidothioic acid (2,5-dioxo-3-pyrrolidinyl) esterMus musculus (house mouse)Potency12.589310
1-ethoxy-3-(2-methoxy-4-prop-2-enylphenoxy)-2-propanolMus musculus (house mouse)Potency0.316210
(2-chlorophenyl)-(5-hydroxy-3-methyl-5-phenyl-4H-pyrazol-1-yl)methanoneMus musculus (house mouse)Potency6.694620
4-[3-[[(2,5-dichloroanilino)-methyliminomethyl]thio]-2,5-dioxo-1-pyrrolidinyl]benzoic acid methyl esterMus musculus (house mouse)Potency35.481310
N-[4-bromo-2-[[(2-hydrazinyl-2-oxoethyl)amino]-phenylmethyl]phenyl]-3-(4-morpholinyl)propanamideMus musculus (house mouse)Potency3.162310
N'-[4-(1-adamantyl)-2-thiazolyl]-N-[(4-fluorophenyl)methyl]oxamideMus musculus (house mouse)Potency4.802220
N-(3-chloro-4-methylphenyl)-2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)acetamideMus musculus (house mouse)Potency5.623410
2-[[2-methyl-5-nitro-3-(phenylmethyl)-4-imidazolyl]thio]-6-nitro-1H-benzimidazoleMus musculus (house mouse)Potency25.665120
1-(2-chlorophenoxy)-3-(2-methyl-1-benzimidazolyl)-2-propanolMus musculus (house mouse)Potency10.147420
N-[2-furanyl-(8-hydroxy-7-quinolinyl)methyl]-2-methylpropanamideMus musculus (house mouse)Potency3.915220
1-(3-nitrophenyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneMus musculus (house mouse)Potency35.481320
1-[1-(2,3-dihydro-1,4-benzodioxin-3-yl)ethyl]-3-phenylthioureaMus musculus (house mouse)Potency5.660820
[(2S)-1,3-dimethyl-3'-nitro-1'-spiro[cyclohepta[d]imidazol-3-ium-2,4'-cyclohexa-2,5-diene]ylidene]-dioxidoammoniumMus musculus (house mouse)Potency11.220210
1-(4-methylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneMus musculus (house mouse)Potency35.481320
1-[8-chloro-4-(1-naphthalenyl)-3,3a,4,9b-tetrahydrocyclopenta[c]quinolin-5-yl]ethanoneMus musculus (house mouse)Potency23.753120
N-(5-bromo-2-pyridinyl)-2,2-dimethyl-3-(2-methylprop-1-enyl)-1-cyclopropanecarboxamideMus musculus (house mouse)Potency35.481310
3-(4-methoxyphenyl)-3-(4-methylphenyl)sulfonyl-1-phenyl-1-propanoneMus musculus (house mouse)Potency22.387210
3-[[[1,3-dioxo-2-(2-oxolanylmethyl)-5-isoindolyl]-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency0.562310
1-(3,5-dimethylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneMus musculus (house mouse)Potency35.481320
N-(2-methoxyphenyl)-2-phenyl-2-(phenylthio)acetamideMus musculus (house mouse)Potency35.481310
N-[2,2,2-trichloro-1-[[sulfanylidene-(2,4,6-trimethylanilino)methyl]amino]ethyl]benzamideMus musculus (house mouse)Potency27.717020
3-phenyl-1-[4-(2-pyridinyl)-1-piperazinyl]-1-propanoneMus musculus (house mouse)Potency0.002810
N-[5-[(4-methylphenyl)methyl]-2-thiazolyl]-2-oxolanecarboxamideMus musculus (house mouse)Potency35.481310
4-(3-methoxyphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazoline-2-thioneMus musculus (house mouse)Potency0.281810
2-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]-1-phenylethanoneMus musculus (house mouse)Potency12.589310
N-[1-[[anilino(sulfanylidene)methyl]amino]-2,2,2-trichloroethyl]-2-(4-ethylphenoxy)acetamideMus musculus (house mouse)Potency24.035320
4-[5-(3-chloro-2-methylphenyl)-2-furanyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterMus musculus (house mouse)Potency6.446820
N-[[4-(4-nitrophenyl)-1-piperazinyl]-sulfanylidenemethyl]butanamideMus musculus (house mouse)Potency12.774820
2-[[(1-butyl-2-benzimidazolyl)amino]methyl]phenolMus musculus (house mouse)Potency12.589310
2-chloro-N-[(2-hydroxy-5-methylanilino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency8.068720
5-methyl-2-phenyl-5-(2-phenylethyl)-1,2,4-triazolidine-3-thioneMus musculus (house mouse)Potency21.169920
N-cyclohexyl-4-(4-nitrophenyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency35.481310
2,2'-[3-(2-methoxyphenyl)-1,2-propanediyl]bis(1H-benzimidazole)Mus musculus (house mouse)Potency9.844420
N-[(2-ethyl-1-piperidinyl)-sulfanylidenemethyl]-4-nitrobenzamideMus musculus (house mouse)Potency0.266520
N-(1-butyl-2-benzimidazolyl)cyclohexanecarboxamideMus musculus (house mouse)Potency2.038620
N-[3-(3,5-dimethyl-1-pyrazolyl)-2-hydroxypropyl]-N-(4-methylphenyl)-2-naphthalenesulfonamideMus musculus (house mouse)Potency35.481320
N-(4-fluorophenyl)-4-(4-nitrophenyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency26.632020
4-chloro-3-(diethylsulfamoyl)-N-(2-nitrophenyl)benzamideMus musculus (house mouse)Potency11.220210
N-[(2-ethyl-1-piperidinyl)-sulfanylidenemethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency0.915020
2-[(4-chlorophenyl)thio]-N-[4-[(2,4-dimethylphenyl)sulfamoyl]phenyl]propanamideMus musculus (house mouse)Potency35.481320
4-[[3-methoxy-4-[(4-nitrophenyl)methoxy]phenyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneMus musculus (house mouse)Potency13.131120
eskazineMus musculus (house mouse)Potency17.039020
N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-2-phenyl-4-quinolinecarboxamideMus musculus (house mouse)Potency7.811720
N-(4-chloro-3-nitrophenyl)-3-phenylbutanamideMus musculus (house mouse)Potency15.848910
1-[2-(4-chlorophenyl)ethyl]-3-(4-fluorophenyl)thioureaMus musculus (house mouse)Potency2.142220
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(4-methoxyphenyl)methyl]acetamideMus musculus (house mouse)Potency1.790120
2-(3,5-diphenyl-3,4-dihydropyrazol-2-yl)-2-(4-hydroxy-3-methoxyphenyl)acetonitrileMus musculus (house mouse)Potency13.980230
3-acetamidobenzoic acid [2-(4-methylphenyl)-2-oxo-1-phenylethyl] esterMus musculus (house mouse)Potency35.481320
4-[[3-[2-(1-cyclohexenyl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazolin-7-yl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency14.125410
5-[[(1-cyclohexyl-5-tetrazolyl)thio]methyl]-3-phenyl-1,2,4-oxadiazoleMus musculus (house mouse)Potency18.629820
2-(3-nitrophenyl)-N-(phenylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency12.589310
1-azepanyl-[2-(phenylmethyl)-1-benzimidazolyl]methanoneMus musculus (house mouse)Potency35.481310
1-cyclopentyl-2-imino-10-methyl-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideMus musculus (house mouse)Potency0.025110
4-[[1-[(3,4-dichlorophenyl)methyl]-3-indolyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-oneMus musculus (house mouse)Potency19.952610
1-adamantyl-[4-(2-fluorophenyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency22.387210
N,N'-bis(3-phenylpropyl)butanediamideMus musculus (house mouse)Potency0.631010
1-(3,4-dimethylphenyl)-3-(2-pyrimidinylthio)pyrrolidine-2,5-dioneMus musculus (house mouse)Potency16.271020
2-[4-(4-nitrophenyl)-1-piperazinyl]-N-(2-pyridinyl)acetamideMus musculus (house mouse)Potency17.782810
4-ethoxy-N-(3-quinolinyl)benzenesulfonamideMus musculus (house mouse)Potency5.145420
N-(4-ethoxyphenyl)-4-[hydroxy(diphenyl)methyl]-1-piperidinecarbothioamideMus musculus (house mouse)Potency24.035320
2-(3,4-dimethylphenyl)-5-ethyl-5-phenyl-1,2,4-triazolidine-3-thioneMus musculus (house mouse)Potency12.602820
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dioneMus musculus (house mouse)Potency20.386620
N-[4-(butylsulfamoyl)phenyl]-2-phenyl-2-(phenylthio)acetamideMus musculus (house mouse)Potency24.035320
N-[2,6-dimethyl-3-[(4-methyl-1-piperazinyl)sulfonyl]phenyl]-N,4-dimethylbenzenesulfonamideMus musculus (house mouse)Potency5.623410
1-(4-methoxyphenyl)-N,N-dipropyl-4-pyrazolo[3,4-d]pyrimidinamineMus musculus (house mouse)Potency22.387210
N-(2-adamantyl)-4-(4-ethylsulfonyl-1-piperazinyl)-3-nitrobenzamideMus musculus (house mouse)Potency14.125410
5-(2-oxolanylmethylamino)-2-thiophen-2-yl-4-oxazolecarbonitrileMus musculus (house mouse)Potency4.466810
2-[(4,7-dimethyl-2-quinazolinyl)thio]-1,2-diphenylethanoneMus musculus (house mouse)Potency27.717020
2-[[1-(4-methoxy-2-nitrophenyl)-2,5-dioxo-3-pyrrolidinyl]thio]benzoic acidMus musculus (house mouse)Potency35.481310
2-methyl-3-phenyl-3H-1,5-benzodiazepin-4-amineMus musculus (house mouse)Potency5.722020
4-phenoxy-1-[4-(2-pyridinyl)-1-piperazinyl]-1-butanoneMus musculus (house mouse)Potency12.924420
LSM-19894Mus musculus (house mouse)Potency6.309610
N-(4-anilinophenyl)-3-(hydroxymethyl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency7.511420
4-(1-phenylethyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency22.740620
N-(4-chloro-2,5-dimethoxyphenyl)-3-methyl-1-piperidinecarbothioamideMus musculus (house mouse)Potency15.186120
4-[hydroxy(diphenyl)methyl]-N-(2-phenylethyl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency24.035320
N4-(4-fluorophenyl)-N5-(2-nitrophenyl)-1H-imidazole-4,5-dicarboxamideMus musculus (house mouse)Potency11.220210
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[(4-methylphenyl)thio]propanamideMus musculus (house mouse)Potency5.623410
1-(4-fluorophenyl)-3-(2-methoxy-3-dibenzofuranyl)ureaMus musculus (house mouse)Potency5.011910
5-bromo-N-(2-oxolanylmethyl)-2-thiophenesulfonamideMus musculus (house mouse)Potency35.481310
1-(2,4-dimethoxyphenyl)-3-[4-(4-morpholinyl)anilino]pyrrolidine-2,5-dioneMus musculus (house mouse)Potency12.589310
N-([biphenyl]-2-yl)-3-cyclopentylpropanamideMus musculus (house mouse)Potency5.011910
5-(4-methoxyanilino)-2-[(3-methylphenoxy)methyl]-4-oxazolecarbonitrileMus musculus (house mouse)Potency22.387210
importazoleMus musculus (house mouse)Potency35.481310
3-nitro-N-[[4-[4-(1-oxopropyl)-1-piperazinyl]anilino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency4.564020
3-(2-pyrimidinylthio)-1-[2-(trifluoromethyl)phenyl]pyrrolidine-2,5-dioneMus musculus (house mouse)Potency5.773220
N-[amino-[2-(1H-indol-3-yl)ethylimino]methyl]-4-chlorobenzamideMus musculus (house mouse)Potency11.220210
2-[[[4-[[2-(4-chloro-2-methylphenoxy)-1-oxopropyl]amino]phenyl]-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency15.848910
3-(4-methoxyphenyl)-N-methyl-5-(4-methylphenyl)-3,4-dihydropyrazole-2-carbothioamideMus musculus (house mouse)Potency11.220210
N-(5-chloro-2-hydroxyphenyl)-2-ethoxybenzamideMus musculus (house mouse)Potency28.183810
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-phenoxybutanamideMus musculus (house mouse)Potency13.534620
N-[2-[(2-furanylmethylamino)-oxomethyl]phenyl]-4-methyl-3-(1-piperidinylsulfonyl)benzamideMus musculus (house mouse)Potency35.481310
1-[[2-(2,4-difluorophenoxy)-1-oxopropyl]amino]-3-(2-oxolanylmethyl)thioureaMus musculus (house mouse)Potency13.534620
2-[[(4-fluoro-2-nitroanilino)-sulfanylidenemethyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid methyl esterMus musculus (house mouse)Potency6.309620
4-[[2-(4-ethyl-3-oxo-2-morpholinyl)-1-oxoethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency27.717020
3-[2-(2,4-dimethyl-3-furanyl)-2-oxoethyl]-3-hydroxy-1-(2-phenylethyl)-2-indoloneMus musculus (house mouse)Potency35.481310
4-(4-nitrophenyl)-N-prop-2-enyl-1-piperazinecarbothioamideMus musculus (house mouse)Potency31.622810
2-[[(3-ethoxycarbonyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-oxomethyl]-3-methyl-3-bicyclo[2.2.1]hept-5-enecarboxylic acidMus musculus (house mouse)Potency14.125410
2-chloro-5-[[2,3-dihydro-1,4-benzodioxin-3-yl(oxo)methyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency14.125410
N-(4,5-dihydrothiazol-2-yl)-3,5-dimethyl-1-adamantanecarboxamideMus musculus (house mouse)Potency5.380820
2-[[(2-methoxy-4-nitroanilino)-sulfanylidenemethyl]amino]benzene-1,4-dicarboxylic acid diethyl esterMus musculus (house mouse)Potency2.528620
1-[1-(1-adamantyl)butyl]-3-(2-oxolanylmethyl)thioureaMus musculus (house mouse)Potency1.804520
N-[5-(2-oxolanyl)-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamideMus musculus (house mouse)Potency3.548110
N-[(4-sulfamoylanilino)-sulfanylidenemethyl]-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency7.811720
N-[[(5-bromo-6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]-2-(2-chlorophenoxy)acetamideMus musculus (house mouse)Potency7.079520
4-fluoro-N-[3-[2-nitro-4-(trifluoromethyl)anilino]propyl]benzamideMus musculus (house mouse)Potency5.623410
1-(4-fluorophenyl)-3-hydroxy-6,6-dimethyl-3-(trifluoromethyl)-5,7-dihydroindole-2,4-dioneMus musculus (house mouse)Potency11.220210
N'-(9-acridinyl)-2-(3-methylphenoxy)acetohydrazideMus musculus (house mouse)Potency4.280020
2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-N-(2-methoxy-3-dibenzofuranyl)acetamideMus musculus (house mouse)Potency17.782810
5-(3,5-dimethyl-1-piperidinyl)-2-(2-furanyl)-4-oxazolecarbonitrileMus musculus (house mouse)Potency0.112210
1-(3-chloro-4-methylphenyl)-5-oxo-N-(2-thiazolyl)-3-pyrrolidinecarboxamideMus musculus (house mouse)Potency8.912510
3-(5-chloro-2-hydroxyphenyl)-3-phenyl-N-[(4-propan-2-yloxyphenyl)methyl]propanamideMus musculus (house mouse)Potency19.952610
[2-(3-chlorophenyl)-4-quinolinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency17.782810
4-oxido-3-(4-phenoxyphenyl)-4a,5,6,7,8,8a-hexahydroquinoxalin-1-ium 1-oxideMus musculus (house mouse)Potency22.387210
5-chloro-7-[3-pyridinyl-(2-pyridinylamino)methyl]-8-quinolinolMus musculus (house mouse)Potency4.224020
N-[4-cyano-5-methyl-2-oxo-3-(trifluoromethyl)-1H-pyrrol-3-yl]cyclopropanecarboxamideMus musculus (house mouse)Potency3.548110
LSM-16248Mus musculus (house mouse)Potency23.350720
1-[2-(hydroxymethyl)-1-benzimidazolyl]-3-(1-indolyl)-2-propanolMus musculus (house mouse)Potency19.118020
2-[[(4-chlorophenyl)thio]methyl]-5-methylimidazo[1,2-a]pyridineMus musculus (house mouse)Potency8.971620
3-[(1-methyl-5-tetrazolyl)thio]-1-phenylpyrrolidine-2,5-dioneMus musculus (house mouse)Potency21.712320
4-[cyclohexyl(methyl)amino]-N-(6-methyl-2-pyridinyl)-3-nitrobenzamideMus musculus (house mouse)Potency35.481310
N-(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-3-isoxazolecarboxamideMus musculus (house mouse)Potency19.952620
5-bromo-N-[1-(2,5-dimethylphenyl)ethyl]-2-furancarboxamideMus musculus (house mouse)Potency18.256320
[3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-phenylmethanoneMus musculus (house mouse)Potency4.224020
1-[(4-tert-butylphenyl)methyl]-4-(4-nitrophenyl)imidazoleMus musculus (house mouse)Potency18.446920
4-[[3-[(4-chlorophenyl)sulfonylamino]-2-quinoxalinyl]amino]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.631010
6,7-dimethoxy-3-(2-oxolanylmethyl)-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency35.481320
1-(4-methoxy-2-nitrophenyl)-4-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonyl)piperazineMus musculus (house mouse)Potency14.987220
N-[3-chloro-4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]phenyl]-2-(4-chlorophenyl)acetamideMus musculus (house mouse)Potency1.584910
N-(1,3-dioxo-5-isoindolyl)-3-methoxybenzamideMus musculus (house mouse)Potency22.387210
cb 7969312Mus musculus (house mouse)Potency5.045120
2-[(4-methylphenyl)thio]-N-(1H-1,2,4-triazol-5-yl)propanamideMus musculus (house mouse)Potency25.118910
2-[1-[[[(3-chloro-1-benzothiophen-2-yl)-oxomethyl]amino]-sulfanylidenemethyl]-3-oxo-2-piperazinyl]acetic acid methyl esterMus musculus (house mouse)Potency3.855220
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methoxy-4-propan-2-yloxybenzamideMus musculus (house mouse)Potency3.981110
2-[[4-(4-fluorophenyl)-6-(trifluoromethyl)-2-pyrimidinyl]sulfonyl]acetic acid ethyl esterMus musculus (house mouse)Potency5.317720
2-[1-(4-chlorophenyl)-5-oxo-3-(2-pyridin-4-ylethyl)-2-sulfanylidene-4-imidazolidinyl]-N-(4-fluorophenyl)acetamideMus musculus (house mouse)Potency35.481310
N-[4-[(3-acetylphenyl)sulfamoyl]phenyl]-1-piperidinecarboxamideMus musculus (house mouse)Potency10.000010
4-[1-(4-fluorophenyl)ethyl]-3-thiophen-2-yl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.409220
4-(4-bromophenyl)-2-(3,5-dimethyl-1-pyrazolyl)-4-oxobutanoic acid methyl esterMus musculus (house mouse)Potency17.743420
2-[3-oxo-1-[[[oxo(thiophen-2-yl)methyl]amino]-sulfanylidenemethyl]-2-piperazinyl]acetic acid propan-2-yl esterMus musculus (house mouse)Potency6.866020
2-[1-[[[(4-methoxyphenyl)-oxomethyl]amino]-sulfanylidenemethyl]-3-oxo-2-piperazinyl]acetic acid propan-2-yl esterMus musculus (house mouse)Potency7.233420
N-[4-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-oxolanecarboxamideMus musculus (house mouse)Potency31.622810
N-[4-(4-acetyl-1-piperazinyl)-3-chlorophenyl]-2-furancarboxamideMus musculus (house mouse)Potency7.079510
5-(2-nitrophenyl)-N-(2-thiazolyl)-2-furancarboxamideMus musculus (house mouse)Potency28.934220
2,2-dimethyl-N-[[4-(pyridin-4-ylmethyl)anilino]-sulfanylidenemethyl]propanamideMus musculus (house mouse)Potency12.589320
3-methyl-N-[[(2-methyl-5-quinolinyl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency8.539820
1-(2-furanyl)-3-(phenylthio)-3-thiophen-2-yl-1-propanoneMus musculus (house mouse)Potency35.481310
2-[(2-furanylmethylthio)methyl]-5-methylimidazo[1,2-a]pyridineMus musculus (house mouse)Potency17.782810
3-[5-(dimethylsulfamoyl)-1-ethyl-2-benzimidazolyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)propanamideMus musculus (house mouse)Potency14.125410
N-(1,1-dioxo-3-thiolanyl)-N-methyl-2-[[1-(2-phenylethyl)-2-benzimidazolyl]thio]acetamideMus musculus (house mouse)Potency25.665120
N-(5-chloro-2-pyridinyl)-2-[(1-phenyl-5-tetrazolyl)thio]propanamideMus musculus (house mouse)Potency6.309620
1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)-2-(1-phthalazinyloxy)ethanoneMus musculus (house mouse)Potency6.309610
7-[[[1-(3-methylphenyl)-2-benzimidazolyl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneMus musculus (house mouse)Potency0.354810
5-[[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]methyl]-2-furancarboxylic acid methyl esterMus musculus (house mouse)Potency15.186120
N-[1-(4-chlorophenyl)sulfonyl-2-pyrrolidinyl]-4-methyl-1-piperazinecarboxamideMus musculus (house mouse)Potency35.481310
4-[[2-(dimethylamino)-2-thiophen-2-ylethyl]amino]-5-methyl-6-thieno[2,3-d]pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency22.535820
N-(3-methyl-1,3-benzothiazol-2-ylidene)-2-pyrazinecarboxamideMus musculus (house mouse)Potency24.035320
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamideMus musculus (house mouse)Potency4.466810
3-hydroxy-1-adamantanecarboxylic acid [2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterMus musculus (house mouse)Potency7.769020
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideMus musculus (house mouse)Potency2.566520
5-[[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]methyl]-3-methyl-1H-pyrrole-2,4-dicarboxylic acid diethyl esterMus musculus (house mouse)Potency12.589310
2-[2-[2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolyl]-2-oxoethyl]isoindole-1,3-dioneMus musculus (house mouse)Potency3.162310
1-(2-furanyl)-2-[(1-methyl-5-tetrazolyl)thio]ethanoneMus musculus (house mouse)Potency2.511910
2-(1,3-diphenyl-4-pyrazolyl)-3-(2-furanylmethyl)-4-thiazolidinoneMus musculus (house mouse)Potency17.782810
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-4-thiophen-2-ylbutanamideMus musculus (house mouse)Potency35.481320
N-(1,3-benzodioxol-5-ylmethyl)-4-benzofuro[3,2-d]pyrimidinamineMus musculus (house mouse)Potency35.481310
4,5-dimethyl-3-(2-oxolanylmethyl)-1H-imidazole-2-thioneMus musculus (house mouse)Potency0.631010
benzoic acid [5-(6-benzamido-9-purinyl)-3-fluoro-4-hydroxy-2-oxolanyl]methyl esterMus musculus (house mouse)Potency10.610120
2-benzoyl-N-(6-methoxy-3-pyridinyl)-3,4-dihydro-1H-isoquinoline-3-carboxamideMus musculus (house mouse)Potency10.000010
bis(1-ethenyl-2-imidazolyl)-(9-ethyl-3-carbazolyl)-sulfanylidenephosphoraneMus musculus (house mouse)Potency12.875020
3,5-dimethyl-1-phenyl-4-pyrazolecarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] esterMus musculus (house mouse)Potency14.125410
2-(4-chloro-2-methylphenoxy)-N-[2-(4-morpholinyl)phenyl]propanamideMus musculus (house mouse)Potency25.665120
N-[1-oxo-1-[[4-(2-pyridinyl)-2-thiazolyl]amino]propan-2-yl]-2-furancarboxamideMus musculus (house mouse)Potency11.220210
3-[(4-phenyl-1-piperazinyl)sulfonyl]benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency9.456220
zeranolMus musculus (house mouse)Potency35.481320
2-(1,3-benzodioxol-5-yl)-5-[[2-(4-methoxyphenyl)-4,5-dihydrothiazol-5-yl]methylthio]-1,3,4-oxadiazoleMus musculus (house mouse)Potency15.848910
1-butyl-2-[(5-phenyl-2-oxazolyl)methylthio]-5-benzimidazolesulfonamideMus musculus (house mouse)Potency22.387210
2-(2-amino-4H-[1,3,5]triazino[2,1-b][1,3]benzoxazol-4-yl)propanedioic acid diethyl esterMus musculus (house mouse)Potency15.714220
6-methyl-2-[[2-(4-morpholinyl)-1-oxoethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterMus musculus (house mouse)Potency15.848910
2-(4-butyl-4-methyl-2,5-dioxo-1-imidazolidinyl)-N-[4-(4-morpholinylsulfonyl)phenyl]acetamideMus musculus (house mouse)Potency7.079510
cyclopropanecarboxylic acid [2-oxo-2-(4-phenoxyanilino)ethyl] esterMus musculus (house mouse)Potency0.281810
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideMus musculus (house mouse)Potency4.564020
2-[2-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-2-oxoethyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dioneMus musculus (house mouse)Potency7.875820
4-phenyl-3H-thiazole-2-thioneMus musculus (house mouse)Potency21.280420
LSM-1318Mus musculus (house mouse)Potency23.350720
2-amino-9-pentyl-3H-purine-6-thioneMus musculus (house mouse)Potency19.149820
(4As,6aS,6bR,10S,12aR)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylic acidMus musculus (house mouse)Potency6.309610
l 783281Mus musculus (house mouse)Potency15.848910
zephiranMus musculus (house mouse)Potency22.196920
AvocadyneMus musculus (house mouse)Potency23.350720
6-methyl-2-(phenylethynyl)pyridineMus musculus (house mouse)Potency24.803320
prosultiamineMus musculus (house mouse)Potency35.481320
p-201-1Mus musculus (house mouse)Potency11.294720
thiophanateMus musculus (house mouse)Potency35.481310
altanserinMus musculus (house mouse)Potency11.034420
9-cyclopentyl-3H-purine-6-thioneMus musculus (house mouse)Potency10.000010
1,3-dimethyl-8-[2-(1-pyrrolidinyl)ethylthio]-6-sulfanylidene-7H-purin-2-oneMus musculus (house mouse)Potency2.490620
12-deoxyphorbolphenylacetate-20-acetateMus musculus (house mouse)Potency19.952610
erysolinMus musculus (house mouse)Potency12.589310
asterric acidMus musculus (house mouse)Potency7.079510
1-(3-chloro-2,6-dihydroxy-4-methoxyphenyl)-1-hexanoneMus musculus (house mouse)Potency35.481310
zd 6474Mus musculus (house mouse)Potency35.481320
2,2-dimethyl-N-[2,2,2-trichloro-1-(2-pyrimidinylthio)ethyl]propanamideMus musculus (house mouse)Potency31.622810
N-(2-hydroxy-5-nitrophenyl)-3-nitrobenzamideMus musculus (house mouse)Potency2.818410
N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) esterMus musculus (house mouse)Potency1.000010
3,4-dimethyl-6-phenyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylic acid propan-2-yl esterMus musculus (house mouse)Potency24.803320
3-chloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamideMus musculus (house mouse)Potency23.735820
3-O-AcetylepisamarcandinMus musculus (house mouse)Potency25.118910
N-methyl-5-nitro-N-(phenylmethyl)-2-furancarboxamideMus musculus (house mouse)Potency4.466810
N-[[2-(4-chlorophenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]benzenesulfonamideMus musculus (house mouse)Potency22.387210
2-[[2,2,2-trichloro-1-[(2-methyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency15.848910
2-[[2,2,2-trichloro-1-[(2,2-dimethyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterMus musculus (house mouse)Potency10.000010
2-(2,3,3-trichloro-1-nitroprop-2-enylidene)-1,3-dihydrobenzimidazoleMus musculus (house mouse)Potency23.350720
2-(2,4-dioxo-3-phenyl-5-thiazolidinyl)-N-(3-methylphenyl)acetamideMus musculus (house mouse)Potency20.483920
2-(2,2-dimethyl-4-oxanyl)-4-(4-nitrophenyl)thiazoleMus musculus (house mouse)Potency35.481310
2-[[2-(4-chlorophenoxy)-1-oxoethyl]hydrazo]-N-(2-methoxy-5-methylphenyl)-2-oxoacetamideMus musculus (house mouse)Potency25.118910
4-methyl-2-[3-methyl-4-(3-methylphenyl)azo-5-oxo-4H-pyrazol-1-yl]-5-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency16.803720
N-[4-(1H-benzimidazol-2-yl)phenyl]-4-ethoxy-3-nitrobenzamideMus musculus (house mouse)Potency22.387210
1-(4-bromophenyl)-N-(3,4-dichlorophenyl)-5-oxo-3-pyrrolidinecarboxamideMus musculus (house mouse)Potency35.481320
2-[(4-chlorophenyl)-[2-[5-(4-chlorophenyl)-2-thiazolyl]-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]propanedinitrileMus musculus (house mouse)Potency24.803320
2-[[2-(2,4-dichlorophenoxy)-1-oxopropyl]hydrazo]-N-(4-methoxyphenyl)-2-oxoacetamideMus musculus (house mouse)Potency20.246620
2-[(3-cyano-4,6-diphenyl-2-pyridinyl)thio]-3-methylbutanoic acidMus musculus (house mouse)Potency3.162310
6-amino-5-cyano-2-phenyl-4-pyridin-4-yl-4H-pyran-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency35.481320
5-methyl-N-(3-methylphenyl)-4-nitro-1H-pyrazol-3-amineMus musculus (house mouse)Potency4.466810
1-[5-hydroxy-3-methyl-5-(3-pyridinyl)-4H-pyrazol-1-yl]-2-(4-methylphenyl)ethanoneMus musculus (house mouse)Potency22.196920
2-[(prop-2-enylthio)-(4,5,6,7-tetrahydro-1H-indol-2-yl)methylidene]propanedinitrileMus musculus (house mouse)Potency28.934220
2-[[2-furanyl(oxo)methyl]hydrazo]-N-(2-methoxy-5-methylphenyl)-2-oxoacetamideMus musculus (house mouse)Potency35.481310
2-[[5-(dimethylsulfamoyl)-1H-indol-3-yl]methylidene]propanedioic acid diethyl esterMus musculus (house mouse)Potency22.387210
acetic acid [1-[(3-nitrophenyl)-(1-oxopentylamino)methyl]-2-naphthalenyl] esterMus musculus (house mouse)Potency31.622810
N-[[5-[(4-chlorophenyl)methylthio]-4-phenyl-1,2,4-triazol-3-yl]methyl]-4-ethoxyanilineMus musculus (house mouse)Potency5.623410
3-nitro-N-(pyridin-4-ylmethyl)benzenesulfonamideMus musculus (house mouse)Potency10.000010
2-(3,4-dimethoxyphenyl)-1-[5-hydroxy-3-methyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneMus musculus (house mouse)Potency17.015720
3-nitro-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency0.945620
4-amino-2-(butylthio)-5-pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.794310
3,4-dimethoxy-N-[(2-methyl-4-nitroanilino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency25.665120
N'-[2-[(6-methoxy-2-methyl-4-quinolinyl)thio]-1-oxoethyl]-2-(1-naphthalenyloxy)acetohydrazideMus musculus (house mouse)Potency22.196920
2-[(2-ethyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-3-yl)oxy]acetic acid methyl esterMus musculus (house mouse)Potency17.782810
N-(4-fluorophenyl)-5-nitro-2-pyridinamineMus musculus (house mouse)Potency5.623410
N-[4-(1H-benzimidazol-2-yl)phenyl]-2-methyl-4-nitro-3-pyrazolecarboxamideMus musculus (house mouse)Potency6.205020
2-(4-chlorophenoxy)-N-(5-nitro-2-thiazolyl)acetamideMus musculus (house mouse)Potency12.736820
2-furanyl-[3-hydroxy-3-(trifluoromethyl)-3a,4,5,6,7,8-hexahydrocyclohepta[c]pyrazol-2-yl]methanoneMus musculus (house mouse)Potency0.815520
2-[7-oxo-7-(3-phenyl-1-pyrrolidinyl)heptyl]isoindole-1,3-dioneMus musculus (house mouse)Potency17.782810
1-(3-hydroxy-2,4,4-trimethyl-1-oxido-5-thiophen-2-yl-2-imidazol-1-iumyl)ethanoneMus musculus (house mouse)Potency7.233420
5-hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazole-1-carboxylic acid ethyl esterMus musculus (house mouse)Potency6.309620
3-[5-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl esterMus musculus (house mouse)Potency11.220210
6-amino-5,7,7-tricyano-8-pyridin-4-yl-1,3,8,8a-tetrahydroisoquinoline-2-carboxylic acid (phenylmethyl) esterMus musculus (house mouse)Potency0.112210
6-amino-2-ethyl-8-[2-(trifluoromethyl)phenyl]-1,6,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrileMus musculus (house mouse)Potency5.623410
6-amino-4-(3-furanyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMus musculus (house mouse)Potency35.481310
6-amino-4-(5-chloro-2-thiophenyl)-5-cyano-2-phenyl-4H-pyran-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency33.552020
2-methyl-N-[1-(4-prop-2-enyl-5-sulfanylidene-1H-1,2,4-triazol-3-yl)ethyl]benzamideMus musculus (house mouse)Potency15.848910
N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideMus musculus (house mouse)Potency22.387210
2-chloro-N-(3-ethyl-2-oxo-1,3-benzoxazol-6-yl)acetamideMus musculus (house mouse)Potency23.350720
6-(3,4-dimethoxyphenyl)-4-oxo-3-phenyl-1,5,6,7-tetrahydroindole-2-carboxylic acid ethyl esterMus musculus (house mouse)Potency19.952610
9-(2-ethoxy-3-methoxyphenyl)-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneMus musculus (house mouse)Potency30.300120
4-(dimethylsulfamoyl)-N-(6,7,8,9-tetrahydro-5H-carbazol-3-ylmethyl)benzamideMus musculus (house mouse)Potency14.125410
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneMus musculus (house mouse)Potency2.115420
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[4-(methylthio)phenyl]methyl]-1,2-dihydropyrazol-3-oneMus musculus (house mouse)Potency1.122010
2-[[5-(phenoxymethyl)-4-phenyl-1,2,4-triazol-3-yl]thio]acetonitrileMus musculus (house mouse)Potency30.300120
N'-[2-[(4-amino-5-cyano-2-pyrimidinyl)thio]-1-oxoethyl]-2-(4-methylphenoxy)acetohydrazideMus musculus (house mouse)Potency0.604520
2-[[5-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-1,2,4-triazol-3-yl]thio]acetonitrileMus musculus (house mouse)Potency18.256320
7'-hydroxy-4'-(4-methoxyphenyl)-4,4,5'-trimethyl-2-spiro[1,3-diazinane-6,2'-3,4-dihydro-2H-1-benzopyran]thioneMus musculus (house mouse)Potency28.934220
4-amino-N5-(4-butoxyphenyl)-N5-[2-(cyclohexylamino)-2-oxoethyl]isothiazole-3,5-dicarboxamideMus musculus (house mouse)Potency35.481310
2-(2-furanyl)-2-[(4-methoxyphenyl)methyl-[2-[5-(5-methyl-2-furanyl)-2-tetrazolyl]-1-oxoethyl]amino]-N-(2-oxolanylmethyl)acetamideMus musculus (house mouse)Potency6.045720
3-ethyl-1-(2-furanylmethyl)-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]thioureaMus musculus (house mouse)Potency10.000010
1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-[2-(3-methylphenyl)ethyl]-3-[3-(4-morpholinyl)propyl]thioureaMus musculus (house mouse)Potency16.099220
N-[2-(tert-butylamino)-2-oxo-1-pyridin-4-ylethyl]-N-(2-furanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideMus musculus (house mouse)Potency12.431220
3-butan-2-yl-1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-phenylethyl)thioureaMus musculus (house mouse)Potency5.623410
N1-butan-2-yl-N4-[2-(3,4-dimethoxyphenyl)ethyl]-N4-(thiophen-2-ylmethyl)benzene-1,4-disulfonamideMus musculus (house mouse)Potency10.000010
4-(2-azaspiro[5.5]undecan-2-ylsulfonyl)-N-butan-2-ylbenzenesulfonamideMus musculus (house mouse)Potency24.035320
N-tert-butyl-2-(N-[2-[5-(4-fluorophenyl)-2-tetrazolyl]-1-oxoethyl]-3-hydroxyanilino)-2-(1H-indol-3-yl)acetamideMus musculus (house mouse)Potency22.387210
4-[[(2,3-dihydro-1H-inden-1-ylamino)-sulfanylidenemethyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency18.063620
1-(4-chlorophenyl)sulfonyl-N'-[oxo-[4-(1-piperidinylsulfonyl)phenyl]methyl]-4-piperidinecarbohydrazideMus musculus (house mouse)Potency5.623410
CID 3192987Mus musculus (house mouse)Potency25.665120
[4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-(2-furanyl)methanoneMus musculus (house mouse)Potency23.350720
4-ethoxy-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-[(4-methoxyphenyl)methyl]benzamideMus musculus (house mouse)Potency35.481310
3-(4-fluorophenyl)-1-[(6-oxo-5H-[1,3]dioxolo[4,5-g]quinolin-7-yl)methyl]-1-(thiophen-2-ylmethyl)ureaMus musculus (house mouse)Potency17.782810
2-[2-[[2-[[1-(2,4-dimethylphenyl)-5-tetrazolyl]thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esterMus musculus (house mouse)Potency9.698520
N-(4-Butan-2-ylphenyl)-N-[2-(cyclopentylamino)-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamideMus musculus (house mouse)Potency13.534620
2-[2-methoxyethyl-(1-oxo-2-thiophen-2-ylethyl)amino]-N-[(4-methoxyphenyl)methyl]-2-(4-propan-2-ylphenyl)acetamideMus musculus (house mouse)Potency35.481310
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[[3-(phenylmethyl)-2-imidazo[4,5-b]pyridinyl]thio]acetamideMus musculus (house mouse)Potency17.488220
1-(9-cyclopentyl-9-azabicyclo[3.3.1]nonan-3-yl)-3-(3,5-dimethylphenyl)thioureaMus musculus (house mouse)Potency35.481310
2-furancarboxylic acid [2-(cyclohexylamino)-2-oxo-1-phenylethyl] esterMus musculus (house mouse)Potency35.481310
1-[2-[(3-cyano-5,7-dimethyl-2-quinolinyl)amino]ethyl]-3-(3-methoxypropyl)thioureaMus musculus (house mouse)Potency22.196920
1-[3-[(7-cyano-[1,3]dioxolo[4,5-g]quinolin-6-yl)amino]propyl]-3-(3-ethoxypropyl)thioureaMus musculus (house mouse)Potency35.481310
1-[2-[(3-cyano-7-methyl-2-quinolinyl)amino]ethyl]-3-[3-(4-morpholinyl)propyl]thioureaMus musculus (house mouse)Potency35.481310
2-[4-[4-(4-fluorophenyl)-2-thiazolyl]-1-piperazinyl]-1-[4-(4-methoxyphenyl)-1-piperazinyl]ethanoneMus musculus (house mouse)Potency3.981110
N-(3-chlorophenyl)-4-[4-(3-methoxyphenyl)-2-thiazolyl]-1-piperazinecarbothioamideMus musculus (house mouse)Potency10.300620
N-(2,4-dimethoxyphenyl)-3-(6-methyl-1H-benzimidazol-2-yl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency35.481310
1-cyclopentyl-1-[2-(5,6-dimethyl-1H-benzimidazol-2-yl)ethyl]-3-(2-oxolanylmethyl)thioureaMus musculus (house mouse)Potency18.854120
N-[2-(cyclopentylamino)-2-oxoethyl]-4,7-dimethyl-N-(2-methylphenyl)-2-oxo-3H-pyrido[1,2-a]pyrimidine-4-carboxamideMus musculus (house mouse)Potency1.000010
[4-[5-tert-butyl-3-(phenylmethyl)-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneMus musculus (house mouse)Potency35.481310
2,4-dimethyl-5-furo[3,2-b]pyrrolecarboxylic acid [3-methyl-1-oxo-1-(2-oxolanylmethylamino)butan-2-yl] esterMus musculus (house mouse)Potency10.865520
3-[(2-chlorophenyl)methyl]-7-[4-[4-(trifluoromethyl)phenyl]-1-piperazinyl]triazolo[4,5-d]pyrimidineMus musculus (house mouse)Potency4.736020
1-(2-methyl-2,3-dihydroindol-1-yl)-2-[4-[5-(trifluoromethyl)-1-benzotriazolyl]-1-piperidinyl]ethanoneMus musculus (house mouse)Potency3.981110
1-(1-tert-butyl-5-tetrazolyl)-N-(2-furanylmethyl)-N-(phenylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamineMus musculus (house mouse)Potency5.145420
1-(1-tert-butyl-5-tetrazolyl)-N-(phenylmethyl)-1-(3-pyridinyl)-N-(thiophen-2-ylmethyl)methanamineMus musculus (house mouse)Potency35.481320
1-(1-tert-butyl-5-tetrazolyl)-N-[(4-fluorophenyl)methyl]-N-(2-furanylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamineMus musculus (house mouse)Potency5.966520
N-(1,3-benzothiazol-2-yl)-2-methoxy-N-[2-(1-methyl-2-pyrrolidinyl)ethyl]benzamideMus musculus (house mouse)Potency11.464220
7-(2-ethyl-1-piperidinyl)-5-methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency10.000010
N-[2-(3-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-N',N'-dimethylpropane-1,3-diamineMus musculus (house mouse)Potency25.665120
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(4-methyl-2-thiazolyl)acetamideMus musculus (house mouse)Potency1.258910
N-[4-[1-(benzenesulfonyl)-2,3-dihydroindol-5-yl]-5-methyl-2-thiazolyl]-2-(4-morpholinyl)acetamideMus musculus (house mouse)Potency6.351420
1-methyl-4-[2-oxo-2-(N-(phenylmethyl)anilino)ethyl]-5-pyrrolo[3,2-b]pyrrolecarboxylic acid propan-2-yl esterMus musculus (house mouse)Potency21.169920
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency15.848910
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency11.220210
6-(3-pyridinyl)-N-(3-pyridinylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency2.238710
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency35.481320
N-(1,3-benzodioxol-5-yl)-2-(5-methyl-2-furanyl)-3-imidazo[1,2-a]pyrimidinamineMus musculus (house mouse)Potency6.309610
2-[[3-(4-methoxyphenyl)-1,2,4-thiadiazol-5-yl]thio]acetic acid ethyl esterMus musculus (house mouse)Potency10.000010
2-(3-ethoxycarbonyl-2-methyl-5-phenyl-1-pyrrolyl)acetic acidMus musculus (house mouse)Potency6.309610
4-[[2-(4-methyl-1-piperidinyl)-1,3-benzothiazol-6-yl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
4-[butan-2-yl-[(3,4-dichloroanilino)-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
3-[6-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-6-oxohexyl]-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency19.091920
3-[2-[butyl(methyl)amino]ethyl]-6-(4-morpholinyl)-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency35.481320
2-[(6-fluoro-1,3-benzothiazol-2-yl)amino]-4-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency21.712320
3-(1,3-benzodioxol-5-ylmethyl)-7-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency18.854120
6-bromo-3-[4-oxo-4-[4-(2-pyridinyl)-1-piperazinyl]butyl]-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency21.280420
3-[[2-(4-fluorophenoxy)-1-oxoethyl]amino]-2-benzofurancarboxylic acid ethyl esterMus musculus (house mouse)Potency0.251210
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[[1-(3-methylphenyl)-2-imidazolyl]thio]acetamideMus musculus (house mouse)Potency15.586420
1-[cyclopropyl(oxo)methyl]-N-(2-hydroxyethyl)-N-(phenylmethyl)-2,3-dihydroindole-5-sulfonamideMus musculus (house mouse)Potency22.106020
N-[1-[(4-chlorophenyl)methyl]-5-methyl-3-pyrazolyl]-5-(3,4-dimethoxyphenyl)-3-isoxazolecarboxamideMus musculus (house mouse)Potency35.481310
5-bromo-1-(1-oxopropyl)-N,N-dipropyl-2,3-dihydroindole-7-sulfonamideMus musculus (house mouse)Potency28.934220
2-[[2-(4-ethoxyphenyl)-5-methyl-4-oxazolyl]methylthio]-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency25.118910
3-chloro-N-(5-chloro-2-pyridinyl)-4-ethoxybenzamideMus musculus (house mouse)Potency22.387210
2-(2-methoxyphenyl)-1-oxo-N-[2-oxo-2-[4-(2-pyridinyl)-1-piperazinyl]ethyl]-4-isoquinolinecarboxamideMus musculus (house mouse)Potency7.703820
N-(1,3-benzodioxol-5-yl)-3-(1-ethyl-5-methyl-4-pyrazolyl)-4,5-dihydroisoxazole-5-carboxamideMus musculus (house mouse)Potency15.848910
2-[(3,5-dimethyl-4-isoxazolyl)methylthio]-4-ethyl-7,7-dimethyl-5-oxo-6,8-dihydroquinoline-3-carbonitrileMus musculus (house mouse)Potency15.848920
1-(4-bromophenyl)sulfonyl-4-[(3-methoxyphenyl)methyl]-1,4-diazepaneMus musculus (house mouse)Potency17.782810
N-(1,3-benzodioxol-5-ylmethyl)-2-[[2-(2-fluorophenyl)-5-methyl-4-oxazolyl]methylthio]acetamideMus musculus (house mouse)Potency14.125410
4-[(1-methyl-2-oxo-4-quinolinyl)oxy]-N-(4-methyl-2-pyridinyl)butanamideMus musculus (house mouse)Potency12.589310
1-(4-chlorophenyl)sulfonyl-N-(2-thiazolyl)-1-cyclopropanecarboxamideMus musculus (house mouse)Potency21.280420
3-(4-bromophenyl)-4-(2-furanylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.962220
5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinolMus musculus (house mouse)Potency0.162620
1-(2-methoxyethyl)-2-[(4-methylphenoxy)methyl]benzimidazoleMus musculus (house mouse)Potency11.220210
3,4-dihydro-2H-quinolin-1-yl-(7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl)methanoneMus musculus (house mouse)Potency35.481310
2-(6-benzimidazolo[1,2-c]quinazolinylthio)-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency3.162310
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideMus musculus (house mouse)Potency35.481310
3-[[oxo(2-quinoxalinyl)methyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency8.764920
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamideMus musculus (house mouse)Potency1.831820
N-(2-furanylmethyl)-2-[(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)thio]acetamideMus musculus (house mouse)Potency1.995310
LSM-28383Mus musculus (house mouse)Potency6.309610
5-ethyl-N-[2-(2-phenyl-4-thiazolyl)ethyl]-2-thiophenesulfonamideMus musculus (house mouse)Potency25.118910
N-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-2-[[1-oxo-2-(1-oxo-2-isoquinolinyl)ethyl]amino]acetamideMus musculus (house mouse)Potency2.511910
3-[4-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-4-oxobutyl]-6,7-diethoxy-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency24.068220
3,7-dimethyl-2-(methylthio)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency35.481310
5a,6,7,8,9,10-hexahydro-5H-azepino[2,1-b]quinazolin-12-oneMus musculus (house mouse)Potency35.481310
3-(4-bromophenyl)-1H-pyrazole-5-carboxylic acid methyl esterMus musculus (house mouse)Potency7.079510
LSM-18934Mus musculus (house mouse)Potency22.387210
4-[2-[[2-[[4-(1,3-benzodioxol-5-yl)-2-thiazolyl]amino]-2-oxoethyl]thio]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency12.589310
1-[4-[4-[[1-(4-chlorophenyl)sulfonylcyclopropyl]-oxomethyl]-1-piperazinyl]phenyl]ethanoneMus musculus (house mouse)Potency0.005010
2-[(5-bromo-2-thiophenyl)sulfonyl-methylamino]-N-(6-methyl-1,3-benzothiazol-2-yl)acetamideMus musculus (house mouse)Potency35.481310
5-amino-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-triazolecarboxamideMus musculus (house mouse)Potency11.220210
N-(1,3-benzodioxol-5-ylmethyl)-3-cyclopentyl-2,4-dioxo-1H-quinazoline-7-carboxamideMus musculus (house mouse)Potency0.079410
N-[4-[[4-(2-fluorophenyl)-1-piperazinyl]-oxomethyl]-1-oxo-2-isoquinolinyl]-2-pyrazinecarboxamideMus musculus (house mouse)Potency19.622220
2-(4-ethoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acidMus musculus (house mouse)Potency12.589310
1-[4-[(4-ethyl-1-piperazinyl)methyl]phenyl]-3-thiophen-2-ylureaMus musculus (house mouse)Potency17.039020
1-[[5-bromo-1-[cyclopropyl(oxo)methyl]-2,3-dihydroindol-7-yl]sulfonyl]-4-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency12.589310
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-piperidinecarboxamideMus musculus (house mouse)Potency8.912510
2-(1,3-benzodioxol-5-yl)-3-hydroxy-1,2-dihydroquinazolin-4-oneMus musculus (house mouse)Potency17.782810
6-(1,3-benzodioxol-5-ylmethylamino)-3-(2-methylphenyl)-1H-pyrimidine-2,4-dioneMus musculus (house mouse)Potency35.481310
2-(4-methoxyphenyl)-N-[4-[5-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]acetamideMus musculus (house mouse)Potency5.158120
6-chloro-3-[2-(diethylamino)ethyl]-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency4.564020
N-(5-chloro-2,4-dimethoxyphenyl)-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideMus musculus (house mouse)Potency14.125410
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-methyl-4-oxo-1-phthalazinyl)acetamideMus musculus (house mouse)Potency7.943310
N-ethyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(phenylmethyl)propanamideMus musculus (house mouse)Potency35.481310
N-(3,4-dimethoxyphenyl)-7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamideMus musculus (house mouse)Potency3.212220
4-[[2-[4-(4-chlorophenyl)-1-piperazinyl]-1-oxoethyl]amino]benzoic acid methyl esterMus musculus (house mouse)Potency11.220210
N-[2-(2-methyl-1-indolyl)ethyl]benzamideMus musculus (house mouse)Potency3.489420
3-(2-furanylmethyl)-5-(2-methoxyethyl)-1,3,5-thiadiazinane-2-thioneMus musculus (house mouse)Potency7.079510
2-[[2-(2-ethyl-1-piperidinyl)-2-oxoethyl]thio]-3-methyl-5H-pyrimido[5,4-b]indol-4-oneMus musculus (house mouse)Potency15.848910
7-[(4-methyl-1-piperazinyl)methyl]-5-(phenylmethoxymethyl)-8-quinolinolMus musculus (house mouse)Potency1.627120
N-butyl-2-[[6-(4-morpholinyl)-4-oxo-3-(2-phenylethyl)-2-quinazolinyl]thio]acetamideMus musculus (house mouse)Potency7.943320
6,7-diethoxy-3-(3-methoxypropyl)-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency23.350720
N-(1,3-benzodioxol-5-yl)-2-[(1-ethyl-2-oxo-4-quinolinyl)thio]acetamideMus musculus (house mouse)Potency10.000010
1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-ethylphenyl)ureaMus musculus (house mouse)Potency35.481310
6-(1-azepanylsulfonyl)-1-ethyl-N-(2-furanylmethyl)-4-oxo-3-quinolinecarboxamideMus musculus (house mouse)Potency22.387210
1-[2-(1-oxo-2-thiophen-2-ylethoxy)ethyl]-5-[(1-oxo-2-thiophen-2-ylethyl)amino]-4-pyrazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency15.848910
6-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-5-thieno[2,3-b]pyrrolecarboxylic acid methyl esterMus musculus (house mouse)Potency35.481320
5-(4-methoxyphenyl)-N-propan-2-yl-3-isoxazolecarboxamideMus musculus (house mouse)Potency0.562310
5-amino-1-(3,5-dimethylphenyl)-N-(phenylmethyl)-4-triazolecarboxamideMus musculus (house mouse)Potency25.118910
[1-(3-methylphenyl)-5-benzimidazolyl]-(1-piperidinyl)methanoneMus musculus (house mouse)Potency35.481310
N-(4-ethylphenyl)-5-(2-furanyl)-3-isoxazolecarboxamideMus musculus (house mouse)Potency35.481310
2-furancarboxylic acid [4-(6-amino-5-cyano-3-propan-2-yl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterMus musculus (house mouse)Potency0.112210
2-[3-[3-(2-furanylmethylamino)-3-oxopropyl]-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]acetic acid (phenylmethyl) esterMus musculus (house mouse)Potency14.125410
N4,N5-bis(2-ethoxyphenyl)-1H-imidazole-4,5-dicarboxamideMus musculus (house mouse)Potency2.988220
N-[2-(1-cyclohexenyl)ethyl]-1-[cyclopropyl(oxo)methyl]-2,3-dihydroindole-5-sulfonamideMus musculus (house mouse)Potency12.589310
N-(4-acetylphenyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideMus musculus (house mouse)Potency0.281810
N-(2-furanylmethyl)-5-(3-methoxyphenyl)-3-isoxazolecarboxamideMus musculus (house mouse)Potency0.562310
2-(1-ethyl-4-oxo-3-furo[3,4]pyrrolo[3,5-c][1,2,4]triazinyl)-N-[4-(2-furanyl)butan-2-yl]propanamideMus musculus (house mouse)Potency35.481310
3,4-dimethoxy-N-[3-(methylthio)phenyl]benzenesulfonamideMus musculus (house mouse)Potency16.271020
N-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideMus musculus (house mouse)Potency17.782810
N-[(2-methyl-4-thiazolyl)methyl]-4-phenoxybenzenesulfonamideMus musculus (house mouse)Potency25.118910
N-ethyl-N-(2-ethylphenyl)-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideMus musculus (house mouse)Potency21.280420
2-[2,4-dioxo-3-(phenylmethyl)-1-quinazolinyl]-N-(5-methyl-3-isoxazolyl)acetamideMus musculus (house mouse)Potency26.632020
7-[4-[4-(2-fluorophenyl)-1-piperazinyl]-4-oxobutyl]-6-sulfanylidene-5H-[1,3]dioxolo[4,5-g]quinazolin-8-oneMus musculus (house mouse)Potency10.266320
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamideMus musculus (house mouse)Potency35.481310
4-[[3-[(2-furanylmethylamino)-oxomethyl]-7-methoxy-1-benzopyran-2-ylidene]amino]benzoic acidMus musculus (house mouse)Potency1.970220
N-(3-methoxyphenyl)-2-(1-methyl-3-indolyl)acetamideMus musculus (house mouse)Potency15.848910
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-3-piperidinecarboxamideMus musculus (house mouse)Potency12.589310
N-[3-(cyclohexylthio)propyl]-1-[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]-3-piperidinecarboxamideMus musculus (house mouse)Potency35.481310
6-methoxy-N-(thiophen-2-ylmethyl)-2-furo[2,3-b]quinolinecarboxamideMus musculus (house mouse)Potency6.309610
N-[4-[(2,3-dihydro-1,4-benzodioxin-6-ylamino)-oxomethyl]phenyl]-2-oxolanecarboxamideMus musculus (house mouse)Potency5.056120
2-[[3-(4-methoxyphenyl)-7-triazolo[4,5-d]pyrimidinyl]thio]-N-(2-oxolanylmethyl)acetamideMus musculus (house mouse)Potency25.665120
2-[(1-acetyl-2-benzimidazolyl)thio]-N-(2-methoxyphenyl)acetamideMus musculus (house mouse)Potency28.183810
8-(2-propoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-oneMus musculus (house mouse)Potency14.125410
N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-[(5-methyl-2-furanyl)methylamino]-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]carbamic acid (phenylmethyl) esterMus musculus (house mouse)Potency33.552020
2,5-dimethyl-N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-(2-naphthalenylamino)-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]-3-pyrazolecarboxamideMus musculus (house mouse)Potency31.622810
3-[(3-fluorophenyl)methyl]-8-[4-(4-fluorophenyl)-4-oxobutyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-oneMus musculus (house mouse)Potency35.481310
N-[(4-chlorophenyl)methyl]-4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinamineMus musculus (house mouse)Potency31.622810
[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency26.632020
n-(1-methyl-5-indolyl)-n'-(3-methyl-5-isothiazolyl)ureaMus musculus (house mouse)Potency19.952610
5-bromo-N-(cycloheptylideneamino)-2-furancarboxamideMus musculus (house mouse)Potency22.387210
3-[3-(N-ethylanilino)propyl]-6-(4-morpholinyl)-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency3.571720
8-[(1-ethyl-3-piperidinyl)thio]-1,3-dimethyl-6-sulfanylidene-7H-purin-2-oneMus musculus (house mouse)Potency5.145420
3-methyl-4-nitro-N-(1H-1,2,4-triazol-5-yl)benzamideMus musculus (house mouse)Potency35.481320
4-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-3-nitrobenzenesulfonamideMus musculus (house mouse)Potency20.386620
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-(1-phenylethylamino)ethyl] esterMus musculus (house mouse)Potency11.220210
2-[(5-amino-1H-1,2,4-triazol-3-yl)thio]-N-(2-bromo-4-nitrophenyl)acetamideMus musculus (house mouse)Potency12.589310
5-hydroxy-2-methyl-4-[1-piperidinyl(3-pyridinyl)methyl]-3-benzo[g]benzofurancarboxylic acid ethyl esterMus musculus (house mouse)Potency22.387210
4-(1-azepanyl)-6-hydrazinyl-N-(4-nitrophenyl)-1,3,5-triazin-2-amineMus musculus (house mouse)Potency14.219120
3-(5-ethyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency7.414020
N-(5-acetyl-2-phenyl-4-sulfanylidene-1H-pyrimidin-6-yl)benzamideMus musculus (house mouse)Potency6.037420
4-butyl-3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.581220
2-[(1-oxo-3-phenylpropyl)amino]-3-thiophenecarboxylic acid methyl esterMus musculus (house mouse)Potency35.481310
1-(6-methyl-2-pyridinyl)-3-[3-(trifluoromethyl)phenyl]thioureaMus musculus (house mouse)Potency1.129420
N-(3,4-dimethylphenyl)-2-[(1-phenyl-1,2,4-triazol-3-yl)thio]acetamideMus musculus (house mouse)Potency6.309610
3-amino-4-(1,3-benzothiazol-2-yl)-N-(3-chloro-2-methylphenyl)-5-phenylimino-2H-thiophene-2-carboxamideMus musculus (house mouse)Potency3.915220
N'-[5-(phenylmethyl)-4,5-dihydrothiazol-2-yl]hexanehydrazideMus musculus (house mouse)Potency18.446920
N-[4-(difluoromethoxy)phenyl]-4-(phenylmethyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency35.481310
1-(4-fluorophenyl)-N-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbothioamideMus musculus (house mouse)Potency35.481310
1-(2-furanylmethyl)-3-(2-methylphenyl)-1-(3-pyridinylmethyl)thioureaMus musculus (house mouse)Potency3.981110
3-(1-methyl-2-benzimidazolyl)-1-phenyl-2-pyrrolo[3,2-b]quinoxalinamineMus musculus (house mouse)Potency2.335020
2-phenoxy-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamideMus musculus (house mouse)Potency4.585820
sb-224289Mus musculus (house mouse)Potency29.903320
1,8-dinitro-4,5-dihydroxyanthraquinoneMus musculus (house mouse)Potency8.764920
6-amino-5-cyano-2-(4-methoxyphenyl)-4-(3-pyridinyl)-4H-pyran-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency15.848910
5-methyl-2-(2-phenoxyethyl)-4-phenyl-1,2,4-triazol-3-oneMus musculus (house mouse)Potency5.011910
2-(dichloromethyl)-4-(4-methylphenyl)-6-(methylthio)-1,3,5-triazineMus musculus (house mouse)Potency2.511910
4-[[7-[(4-fluorophenyl)methyl]-1,3-dimethyl-2,6-dioxo-8-purinyl]methyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency15.848910
4-[[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholineMus musculus (house mouse)Potency23.350720
1-[2-(dimethylamino)ethyl]-3-(2,4-dimethylphenyl)-1-(thiophen-2-ylmethyl)thioureaMus musculus (house mouse)Potency10.000010
LSM-19878Mus musculus (house mouse)Potency1.518620
2-[(5-chloro-1,3-benzothiazol-2-yl)thio]-N-[3-(4-morpholinylsulfonyl)phenyl]propanamideMus musculus (house mouse)Potency31.622810
2-(1-naphthalenyl)acetic acid [2-[4-chloro-3-(dimethylsulfamoyl)anilino]-2-oxoethyl] esterMus musculus (house mouse)Potency14.976320
3-(6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.962220
N,N,1-triethyl-2-sulfanylidene-3H-benzimidazole-5-sulfonamideMus musculus (house mouse)Potency6.309610
2-(2-methoxyphenyl)-1-methyl-3,5-dinitro-2H-pyridineMus musculus (house mouse)Potency23.350720
N-[(4-methoxyphenyl)methyl]-2-(phenylmethyl)-4-thiazolecarboxamideMus musculus (house mouse)Potency8.912510
4-butyl-3-(6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency1.653120
2-phenoxyacetic acid (2-oxo-1,2-diphenylethyl) esterMus musculus (house mouse)Potency11.220210
N-[2-(4-morpholinyl)ethyl]-2-(4-propan-2-yloxyphenyl)-4-quinolinecarboxamideMus musculus (house mouse)Potency22.740620
5-[[(3,4-dichloroanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterMus musculus (house mouse)Potency9.053220
5-(diethylsulfamoyl)-2-hydroxybenzoic acid [2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] esterMus musculus (house mouse)Potency35.481310
(4-methylphenyl)-[4-[4-nitro-3-(3-pyridinylmethylamino)phenyl]-1-piperazinyl]methanoneMus musculus (house mouse)Potency15.848910
2-methyl-N'-[2-[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]benzohydrazideMus musculus (house mouse)Potency4.466810
1-(2,5-dimethoxyphenyl)-3-[5-(2-methyl-1-piperidinyl)-1,3,4-thiadiazol-2-yl]ureaMus musculus (house mouse)Potency35.481310
1-(3-methoxyphenyl)-3-[5-(2-methyl-1-piperidinyl)-1,3,4-thiadiazol-2-yl]ureaMus musculus (house mouse)Potency11.220210
2-[(5-chloro-2-thiophenyl)-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.562310
2-fluoro-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)benzamideMus musculus (house mouse)Potency8.539820
sto 609Mus musculus (house mouse)Potency10.602520
5-(3-nitrophenyl)-3-phenyl-1H-imidazole-2-thioneMus musculus (house mouse)Potency6.607820
1-(3,4-dichlorophenyl)-3-[1-(4-morpholinyl)-1-phenylpropan-2-yl]ureaMus musculus (house mouse)Potency35.481310
N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-[4-methyl-4-(4-methylphenyl)-2,5-dioxo-1-imidazolidinyl]acetamideMus musculus (house mouse)Potency3.981110
N,N-dimethylcarbamodithioic acid (1-acetamido-2,2,2-trichloroethyl) esterMus musculus (house mouse)Potency24.035320
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinolMus musculus (house mouse)Potency4.220920
4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)-N-(5-ethyl-1,3,4-oxadiazol-2-yl)benzamideMus musculus (house mouse)Potency0.458620
3-(3-chloro-2-methylphenyl)-1-[(4-methylphenyl)methyl]-1-(3-pyridinylmethyl)thioureaMus musculus (house mouse)Potency19.731220
1-[4-chloro-3-[(2-methoxyphenyl)sulfamoyl]phenyl]-3-(2-methoxyphenyl)ureaMus musculus (house mouse)Potency11.220210
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinolMus musculus (house mouse)Potency3.915220
6-amino-5-cyano-4-(2-fluorophenyl)-2-sulfanylidene-3,4-dihydro-1H-pyridine-3-carboxamideMus musculus (house mouse)Potency16.517620
N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-methyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency2.238710
2-(2,4-dibromophenoxy)-N-[[3-(hydroxymethyl)anilino]-sulfanylidenemethyl]acetamideMus musculus (house mouse)Potency5.162520
N-[2-(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)ethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency8.912510
2-[[1-(phenylmethyl)-3-indolyl]thio]-N-(2-thiazolyl)acetamideMus musculus (house mouse)Potency3.981110
N-(4-bromophenyl)-2-[(5,6-dimethyl-4-thieno[2,3-d]pyrimidinyl)thio]benzamideMus musculus (house mouse)Potency9.456220
N-(4-ethoxyphenyl)sulfonyl-N-(2-oxo-5-benzo[g][1,3]benzoxathiolyl)-2-furancarboxamideMus musculus (house mouse)Potency24.035320
2-(thiophen-2-ylsulfonylamino)benzoic acid [2-(3-acetylanilino)-2-oxo-1-phenylethyl] esterMus musculus (house mouse)Potency5.623410
3-(4-benzoyl-1-piperazinyl)-1-(2-methylpropyl)-6,7-dihydro-5H-cyclopenta[c]pyridine-4-carbonitrileMus musculus (house mouse)Potency37.646020
[1-[2-(2-methylphenoxy)ethyl]-3-indolyl]-(4-methyl-1-piperazinyl)methanethioneMus musculus (house mouse)Potency12.589310
1-butyl-3-[[(4,5-dimethyl-3-thiophenyl)-oxomethyl]amino]thioureaMus musculus (house mouse)Potency7.562720
1-(Chloroacetyl)-3-(1H-indol-3-yl)-5-(4-methoxyphenyl)-4,5-dihydro-1H-pyrazol-4-olMus musculus (house mouse)Potency11.294720
1-(4-methoxyphenyl)-3-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)pyrrolidine-2,5-dioneMus musculus (house mouse)Potency35.481310
1-(4-butylphenyl)-3-[4-chloro-3-(dimethylsulfamoyl)phenyl]thioureaMus musculus (house mouse)Potency23.350720
N-(6-acetamido-3-prop-2-enyl-1,3-benzothiazol-2-ylidene)cyclohexanecarboxamideMus musculus (house mouse)Potency25.118910
N4-(2-furanylmethyl)-N2-(3-methoxyphenyl)-5-nitropyrimidine-2,4,6-triamineMus musculus (house mouse)Potency15.848910
6-bromo-2-(4-methylphenyl)-N-[(1-methyl-4-pyrazolyl)methyl]-4-quinolinecarboxamideMus musculus (house mouse)Potency35.481310
4-[1-(4-bromophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMus musculus (house mouse)Potency19.952610
1-[2-[(4-chlorophenyl)thio]ethyl]-3-(4-methylphenyl)thioureaMus musculus (house mouse)Potency0.842820
nsc 105827Mus musculus (house mouse)Potency4.795720
AngolensinMus musculus (house mouse)Potency35.481310
7-(2-chloro-6-fluorophenyl)-5-methyl-6,7-dihydro-1H-1,4-diazepine-2,3-dicarbonitrileMus musculus (house mouse)Potency27.717020
N-(5-chloro-2-methoxyphenyl)-2-pyridin-4-yl-4,5-dihydrothiazole-4-carboxamideMus musculus (house mouse)Potency11.220210
4-chloro-N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.631010
2-[[2-[(2,5-dimethylphenyl)sulfonylamino]-1-oxoethyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideMus musculus (house mouse)Potency35.481310
4-(4-chlorophenyl)-N-[3-[(4-methoxyphenyl)sulfamoyl]phenyl]-4-oxobutanamideMus musculus (house mouse)Potency25.665120
2-amino-4-nitrophenolMus musculus (house mouse)Potency12.589310
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-morpholinecarboxamideMus musculus (house mouse)Potency0.125910
2-phenylbutanoic acid [2-(3,5-dichloroanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency31.832620
7-(5-bromo-2-fluorophenyl)-5-(4-bromophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency14.348420
N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]-5-nitro-2-thiophenecarboxamideMus musculus (house mouse)Potency2.990420
2-[[7-(4-methoxyphenyl)-5-phenyl-4-pyrrolo[2,3-d]pyrimidinyl]thio]propanoic acid ethyl esterMus musculus (house mouse)Potency10.000010
N-[[4-[[4-(4-fluorophenyl)-1-piperazinyl]-oxomethyl]cyclohexyl]methyl]-2-thiophenesulfonamideMus musculus (house mouse)Potency10.000010
l 663536Mus musculus (house mouse)Potency17.039020
N'-[(3-nitrophenyl)-oxomethyl]-2-pyridinecarbohydrazideMus musculus (house mouse)Potency22.740620
2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-5-methyl-4-(4-methylphenyl)-1,2,4-triazol-3-oneMus musculus (house mouse)Potency35.481310
6,8-dibromo-2-thiophen-2-ylquinolineMus musculus (house mouse)Potency3.981110
N-[2-[(3-nitrophenyl)methylthio]-4-oxo-3-quinazolinyl]benzamideMus musculus (house mouse)Potency5.317720
1-[4,6-bis(ethylamino)-1,3,5-triazin-2-yl]-1-ethylthioureaMus musculus (house mouse)Potency20.246620
4-[1-oxo-6-(4-oxo-2-sulfanylidene-1H-thieno[3,2-d]pyrimidin-3-yl)hexyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency23.350720
N-[3-[(3-chlorophenyl)sulfamoyl]-4-methylphenyl]-3-(4-nitrophenyl)-3-oxopropanamideMus musculus (house mouse)Potency35.481310
2-chloro-N-(3-methyl-1,3-benzothiazol-2-ylidene)acetamideMus musculus (house mouse)Potency16.193620
3-[(4-ethylphenoxy)methyl]-4-(6-methylheptan-2-yl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.309610
1-(4-chlorophenyl)-3-[[1-(4-methoxyphenyl)-3-pyrrolidinyl]methyl]ureaMus musculus (house mouse)Potency31.622810
1-[[1-(4-methoxyphenyl)-3-pyrrolidinyl]methyl]-3-(2,4,6-trimethylphenyl)thioureaMus musculus (house mouse)Potency4.246020
ML162Mus musculus (house mouse)Potency11.220210
2-(N-(2-chloro-1-oxoethyl)-3-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideMus musculus (house mouse)Potency12.589310
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideMus musculus (house mouse)Potency23.350720
1-(phenylmethyl)-3-(1,2,3,4-tetrahydronaphthalen-1-yl)thioureaMus musculus (house mouse)Potency6.866020
N-decyl-N'-(2-pyridinyl)oxamideMus musculus (house mouse)Potency24.803320
1-phenyl-2-[[4-(trifluoromethyl)phenyl]methylthio]imidazoleMus musculus (house mouse)Potency14.125410
6-amino-4-(3-furanyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileMus musculus (house mouse)Potency14.125410
1-(2-ethyl-6-methylphenyl)-3-[(1-methyl-2-pyrrolyl)methyl]thioureaMus musculus (house mouse)Potency14.125410
3-methyl-2-methylene-1,5-diphenylpentane-1,5-dioneMus musculus (house mouse)Potency15.954120
2-[(4-amino-7-tert-butyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)thio]acetic acidMus musculus (house mouse)Potency10.000010
2-[(4-chlorophenyl)methylthio]-N-(2-hydroxy-5-nitrophenyl)acetamideMus musculus (house mouse)Potency9.505620
3-ethyl-2-sulfanylidene-5-thiophen-2-yl-1H-thieno[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency1.935120
LSM-1924Mus musculus (house mouse)Potency12.589310
2-(4-chlorophenyl)sulfonylquinoxalineMus musculus (house mouse)Potency35.481310
2-[1-(2-methylphenyl)-3-oxo-3-thiophen-2-ylpropyl]propanedinitrileMus musculus (house mouse)Potency1.584910
1-[(4-chlorophenyl)methyl]-3-(3-fluorophenyl)-1-(3,3,3-trifluoro-2-hydroxypropyl)ureaMus musculus (house mouse)Potency23.350720
5-[(4-chlorophenyl)-oxomethyl]-4-hydroxy-6-[5-(2-nitrophenyl)-2-furanyl]-4-(trifluoromethyl)-1,3-diazinan-2-oneMus musculus (house mouse)Potency25.118910
N-(3-chlorophenyl)-5-oxo-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindole-1-carboxamideMus musculus (house mouse)Potency14.125410
2-(4-chlorophenyl)-5-methyl-4-oxo-2,3-dihydro-1H-thieno[3,4-d]pyrimidine-7-carboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
4-[[anilino-(4-methylphenyl)methyl]-propoxyphosphoryl]-N,N-dimethylanilineMus musculus (house mouse)Potency35.481320
1-butyl-4,6-dimethyl-3-(2-methylphenyl)sulfonyl-2-pyridinoneMus musculus (house mouse)Potency14.125410
2-(4-nitrophenyl)-4-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.891310
2-chloro-N-(2-methyl-6-oxo-5H-benzo[b][1,4]benzoxazepin-8-yl)acetamideMus musculus (house mouse)Potency13.891420
5-methyl-3-phenyl-7-(prop-2-enylthio)pyrazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency20.811420
1-ethyl-3-[[2-[(1-methyl-2-benzimidazolyl)thio]-1-oxoethyl]amino]thioureaMus musculus (house mouse)Potency0.465920
4-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitrobenzoic acid methyl esterMus musculus (house mouse)Potency35.481310
2-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitropyridineMus musculus (house mouse)Potency6.309610
benzoic acid [[1-(4-nitrophenyl)-4-piperidinylidene]amino] esterMus musculus (house mouse)Potency19.952610
4-(4-methylphenyl)sulfonyl-3-phenyl-2,3-dihydro-1,4-benzoxazineMus musculus (house mouse)Potency35.481310
N-[3-(4-methyl-1-piperazinyl)-1,4-dioxo-2-naphthalenyl]benzenesulfonamideMus musculus (house mouse)Potency11.904820
5-(benzenesulfonyl)-4-(2,6-dimethylphenoxy)-2-phenylpyrimidineMus musculus (house mouse)Potency11.220210
4-(2-methylcyclohexyl)-3-(3-pyridinyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency11.294720
(4-chlorophenyl)-(7-methyl-3-imidazo[1,2-a]pyridinyl)methanoneMus musculus (house mouse)Potency0.281810
3-methyl-N-[[[(4-nitrophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]butanamideMus musculus (house mouse)Potency4.802220
7-chloro-3-hydroxy-2-[3-(trifluoromethyl)phenyl]-4-quinazolinoneMus musculus (house mouse)Potency5.313820
4-[[[2-(4-methoxyphenyl)-3-thiazolidinyl]-sulfanylidenemethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency23.753120
4-fluoro-N-[[2-(3-pyridinyl)-1-piperidinyl]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency1.701620
N-[(5-quinolinylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency13.948020
2-Chloro-1-[5-(3,4-dimethoxyphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneMus musculus (house mouse)Potency27.717020
LSM-31277Mus musculus (house mouse)Potency25.118910
5-methyl-2-[[(4-nitrophenyl)-oxomethyl]hydrazo]-4-thiazolecarboxylic acid ethyl esterMus musculus (house mouse)Potency3.378220
2-[2-[5-amino-4-(3-thiophenyl)-1-pyrazolyl]-4-phenyl-5-thiazolyl]acetic acidMus musculus (house mouse)Potency3.162310
(2,5-dimethylanilino)thioureaMus musculus (house mouse)Potency20.085020
N-(4-phenylmethoxyphenyl)-3-[4-(phenylmethyl)-1-piperazinyl]propanamideMus musculus (house mouse)Potency17.782810
N-(4-methoxyphenyl)-5-oxo-6,7-dihydro-[1,2,4]triazolo[3,4-b][1,3]thiazine-7-carboxamideMus musculus (house mouse)Potency28.934220
3-(2,4-dichloro-5-methoxyphenyl)-2-sulfanyl-4(3h)-quinazolinoneMus musculus (house mouse)Potency4.220920
2-amino-7,7-dimethyl-4-(4-methylphenyl)-5-oxo-6,8-dihydro-4H-1-benzopyran-3-carbothioamideMus musculus (house mouse)Potency35.481320
1-(4-chlorophenyl)-3-[2-(2-furanylmethyl)cyclohexyl]ureaMus musculus (house mouse)Potency35.481310
4-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-3-oxobutanoic acid ethyl esterMus musculus (house mouse)Potency21.169920
4-[(2-hydroxy-3-nitrophenyl)-(5-methyl-3-oxo-2-phenyl-1H-pyrazol-4-yl)methyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMus musculus (house mouse)Potency35.481320
2-furanyl-[4-(4-propan-2-ylphenyl)sulfonyl-1-piperazinyl]methanoneMus musculus (house mouse)Potency19.952610
4-(2-chlorophenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidineMus musculus (house mouse)Potency7.414020
N-(3,5-dimethylphenyl)-2-(2-nitroethyl)benzamideMus musculus (house mouse)Potency3.981110
4-(2-fluorophenyl)-5-methyl-2-(2-phenoxyethyl)-1,2,4-triazol-3-oneMus musculus (house mouse)Potency33.552020
rose bengal(2-)Mus musculus (house mouse)Potency12.750320
1-(Chloroacetyl)-5-[4-(difluoromethoxy)-3-methoxyphenyl]-3-thien-2-yl-4,5-dihydro-1H-pyrazoleMus musculus (house mouse)Potency15.848920
1-(1-adamantyl)-3-(3,4-dimethoxyphenyl)thioureaMus musculus (house mouse)Potency2.403520
6-nitro-3-phenyl-1H-benzimidazole-2-thioneMus musculus (house mouse)Potency5.011910
or486Mus musculus (house mouse)Potency23.753110
N-(4-fluorophenyl)-5-methyl-1H-indole-2-carboxamideMus musculus (house mouse)Potency10.000010
5-nitro-2-thiophenecarboxylic acid [1-[(3,5-dichloro-2-pyridinyl)amino]-1-oxopropan-2-yl] esterMus musculus (house mouse)Potency19.952610
LSM-22738Mus musculus (house mouse)Potency3.981110
rs 17053Mus musculus (house mouse)Potency14.219120
2-[(4-chloro-3-nitrophenyl)-oxomethyl]benzoic acid [2-[di(propan-2-yl)amino]-2-oxoethyl] esterMus musculus (house mouse)Potency31.622810
ro 106-9920Mus musculus (house mouse)Potency0.610820
4-chloro-5-(2,3-dihydro-1,4-benzodioxin-3-yl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency10.605820
2-(1H-benzimidazol-2-ylthio)-1-[2,5-dimethyl-1-(2-oxolanylmethyl)-3-pyrrolyl]ethanoneMus musculus (house mouse)Potency19.702020
1-(2-fluorophenyl)-3-(N-(phenylmethyl)anilino)thioureaMus musculus (house mouse)Potency7.233420
N-[2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl]-4-nitroanilineMus musculus (house mouse)Potency6.351420
2,5-dihydroxy-4-methoxybenzophenoneMus musculus (house mouse)Potency14.219120
N-[5-(diethylsulfamoyl)-2-methoxyphenyl]-2-[(2,5-dimethylphenyl)thio]acetamideMus musculus (house mouse)Potency17.782810
N-(1,3-benzothiazol-2-yl)-2-ethylsulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxamideMus musculus (house mouse)Potency4.007520
2-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamideMus musculus (house mouse)Potency20.811420
4-oxo-4-thiophen-2-ylbutanoic acid [2-(ethylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency3.981110
3-(5-bromo-2-furanyl)-5-(4-methoxyphenyl)-1,2,4-oxadiazoleMus musculus (house mouse)Potency8.912510
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-1-nitro-9,10-dioxo-2-anthracenecarboxamideMus musculus (house mouse)Potency10.610120
6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylic acid [1-[1-[4-(difluoromethoxy)phenyl]-2,5-dimethyl-3-pyrrolyl]-1-oxopropan-2-yl] esterMus musculus (house mouse)Potency22.387210
N-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-2-quinolinecarboxamideMus musculus (house mouse)Potency21.280420
4-benzoyl-2-heptyl-5-methyl-4H-pyrazol-3-oneMus musculus (house mouse)Potency35.481320
3-bromo-4-methyl-N-[(2-oxolanylmethylamino)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency10.430420
2-hydroxybenzoic acid [2-(2-ethoxyanilino)-2-oxo-1-phenylethyl] esterMus musculus (house mouse)Potency10.000010
vu0155094Mus musculus (house mouse)Potency22.387210
N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]cyclohexanecarboxamideMus musculus (house mouse)Potency3.548110
3-[[(3-methoxyphenyl)-oxomethyl]amino]-2-benzofurancarboxamideMus musculus (house mouse)Potency22.387210
1-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-3-ethyl-1-(2-furanylmethyl)thioureaMus musculus (house mouse)Potency35.481320
[4-[(2-chlorophenyl)methylsulfonyl]-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency12.589310
3-(2-chlorophenyl)-N-[5-(2,4-dichlorophenyl)-1,3,4-thiadiazol-2-yl]-5-methyl-4-isoxazolecarboxamideMus musculus (house mouse)Potency18.256320
1-butyl-3-[[2-furanyl(oxo)methyl]amino]thioureaMus musculus (house mouse)Potency24.035320
N-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]acetamideMus musculus (house mouse)Potency8.912520
2-(1,3-benzothiazol-2-ylmethylthio)-1-butyl-5-benzimidazolesulfonamideMus musculus (house mouse)Potency12.589310
4-chloro-N-[(4-ethoxy-2-nitroanilino)-sulfanylidenemethyl]-2,5-dimethyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency22.740620
4-(6-methyl-4-phenyl-2-quinazolinyl)-1,3-dihydroquinoxalin-2-oneMus musculus (house mouse)Potency19.731220
N-[4-(phenoxymethyl)-2-thiazolyl]-1-adamantanecarboxamideMus musculus (house mouse)Potency33.552020
1-[(1,2-dimethyl-5-indolyl)methyl]-3-(phenylmethyl)thioureaMus musculus (house mouse)Potency26.632020
N-[2-(1-cyclohexenyl)ethyl]-3-[(4-methylphenyl)methylthio]propanamideMus musculus (house mouse)Potency12.589310
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidMus musculus (house mouse)Potency10.000010
5-[2-furanyl(4-morpholinyl)methyl]-6-thiazolo[3,2-b][1,2,4]triazololMus musculus (house mouse)Potency35.481310
N-[3-[3-(1-piperidinylsulfonyl)anilino]-2-quinoxalinyl]benzenesulfonamideMus musculus (house mouse)Potency24.035320
[4-(2,3-dimethylphenyl)-1-piperazinyl]-[5-[(4-methoxyphenyl)sulfonylmethyl]-2-furanyl]methanoneMus musculus (house mouse)Potency35.481310
6-(4-morpholinyl)-3-(2-phenylethyl)-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency2.578820
N-(5-chloro-2-methoxyphenyl)-2-[[3-(2-methoxyethyl)-6-methyl-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideMus musculus (house mouse)Potency20.386620
N-[3-[(4-ethoxyphenyl)-[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-4,5-dimethyl-2-thiophenyl]benzamideMus musculus (house mouse)Potency35.481310
3,5-bis(4-methoxyphenyl)-1H-imidazole-2-thioneMus musculus (house mouse)Potency0.905320
4-(1-phenylethyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency7.079520
2-bromo-N-[[(2-methylcyclohexyl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency3.915220
4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dioneMus musculus (house mouse)Potency4.736020
1-[[2-(2,4-dichlorophenoxy)-1-oxoethyl]amino]-3-(4-methoxyphenyl)thioureaMus musculus (house mouse)Potency17.782810
3-methoxy-N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)benzamideMus musculus (house mouse)Potency14.125410
2-[(1-methyl-2-imidazolyl)thio]-1-(2-naphthalenyl)ethanoneMus musculus (house mouse)Potency23.350720
1,8-dimethoxyphenazineMus musculus (house mouse)Potency27.005020
N-[5-(2-chlorophenyl)-1,3,4-thiadiazol-2-yl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]butanamideMus musculus (house mouse)Potency2.511910
N-(1,3-diphenylpropan-2-ylideneamino)-2-hydroxybenzamideMus musculus (house mouse)Potency4.928820
N-[3-(1-azepanylsulfonyl)-4-methylphenyl]-2-(4-quinazolinylthio)acetamideMus musculus (house mouse)Potency35.481320
3-(2-fluorophenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxylic acid methyl esterMus musculus (house mouse)Potency4.392820
2-[[[[[5-[(4-chloro-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]-sulfanylidenemethyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency1.122010
2-[3-(2-methylphenyl)-4-oxo-2-thiazolidinylidene]propanedinitrileMus musculus (house mouse)Potency3.981110
1-(3,3-dimethylbutan-2-yl)-3-[3-(trifluoromethyl)phenyl]thioureaMus musculus (house mouse)Potency6.581220
1-(1H-benzimidazol-2-yl)-3-cyclohexylureaMus musculus (house mouse)Potency13.534620
N-[3-(2-methoxyethyl)-6-methylsulfonyl-1,3-benzothiazol-2-ylidene]-2-nitrobenzamideMus musculus (house mouse)Potency1.000010
2-(1-naphthalenyl)-4-quinolinecarboxylic acid [1-[(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)amino]-1-oxopropan-2-yl] esterMus musculus (house mouse)Potency22.387210
2-(4-ethoxyphenyl)-1-[5-hydroxy-3-methyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneMus musculus (house mouse)Potency3.298420
1-(1-adamantyl)-2-[(1-oxido-2-pyridin-1-iumyl)thio]ethanoneMus musculus (house mouse)Potency35.481310
N-cyclopropyl-2-[[2-(4-ethoxyphenyl)-5-methyl-4-oxazolyl]methylthio]acetamideMus musculus (house mouse)Potency13.347720
1-(2-methylphenyl)-3-(6,7,8,9-tetrahydro-5H-carbazol-3-ylmethyl)thioureaMus musculus (house mouse)Potency2.566520
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneMus musculus (house mouse)Potency22.387210
1-[[4-anilino-6-(1-piperidinyl)-1,3,5-triazin-2-yl]amino]-3-cyclohexylthioureaMus musculus (house mouse)Potency8.528020
7-(1-azepanyl)-3-(2-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidineMus musculus (house mouse)Potency17.900820
2-[[(3-methoxyanilino)-oxomethyl]-[(3-methyl-2-thiophenyl)methyl]amino]acetic acid ethyl esterMus musculus (house mouse)Potency11.220210
N-[5-[[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-1-naphthalenecarboxamideMus musculus (house mouse)Potency14.125410
2-[[[4-[bis(2-methoxyethyl)sulfamoyl]phenyl]-oxomethyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxamideMus musculus (house mouse)Potency2.879720
2-cyclopentylacetic acid [2-[(3-chloro-9,10-dioxo-2-anthracenyl)amino]-2-oxoethyl] esterMus musculus (house mouse)Potency19.952610
3-[3-[4-(4-methoxyphenyl)-1-piperazinyl]propyl]-2-sulfanylidene-1H-pyrido[2,3-d]pyrimidin-4-oneMus musculus (house mouse)Potency11.220210
5-[[2-[2-[[cyclohexyl(oxo)methyl]amino]-1-oxoethoxy]-1-oxoethyl]amino]-3-methylthiophene-2,4-dicarboxylic acid diethyl esterMus musculus (house mouse)Potency35.481310
LSM-19765Mus musculus (house mouse)Potency35.481310
2-[1-[4-(diethylamino)phenyl]-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-N-phenylacetamideMus musculus (house mouse)Potency28.183810
2-(4-methoxyphenyl)sulfonylquinoxalineMus musculus (house mouse)Potency12.672820
sb 415286Mus musculus (house mouse)Potency18.854110
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[4-(2-methoxyphenyl)-1-piperazinyl]acetamideMus musculus (house mouse)Potency26.632020
1-(2,6-dimethylphenyl)-3-[[1-(4-methoxyphenyl)-3-pyrrolidinyl]methyl]thioureaMus musculus (house mouse)Potency1.565020
2-[4-(9H-fluoren-9-yl)-1-piperazinyl]-N-(4-methoxyphenyl)acetamideMus musculus (house mouse)Potency31.622810
3-chloro-N-[5-(3-pyridinyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.604520
1-(5-methyl-2-furanyl)-2-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-1H-[1]benzopyrano[2,3-c]pyrrole-3,9-dioneMus musculus (house mouse)Potency28.183810
N-(3-chlorophenyl)-4-fluoro-3-(thiophen-2-ylmethylsulfamoyl)benzamideMus musculus (house mouse)Potency19.952610
5-[[(2-methylanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterMus musculus (house mouse)Potency16.903620
N-[[4-(2-ethoxyphenyl)-1-piperazinyl]-sulfanylidenemethyl]-1-adamantanecarboxamideMus musculus (house mouse)Potency3.548120
N'-(4,6-difluoro-1,3-benzothiazol-2-yl)benzohydrazideMus musculus (house mouse)Potency20.246620
N-(2,5-dimethoxyphenyl)-4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1H-quinazoline-7-carboxamideMus musculus (house mouse)Potency0.842820
3-acetamido-N-[(4-ethoxy-3-methoxyphenyl)methyl]-4-[(4-methylphenyl)thio]benzamideMus musculus (house mouse)Potency11.220210
N-[3-(N-(2-chloro-1-oxoethyl)-4-nitroanilino)propyl]-2,2,2-trifluoroacetamideMus musculus (house mouse)Potency35.481310
sch 79797Mus musculus (house mouse)Potency23.735820
N-[[(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-5-methyl-3-phenyl-4-isoxazolecarboxamideMus musculus (house mouse)Potency17.220620
2-[[4-phenyl-5-(propylthio)-1,2,4-triazol-3-yl]methylthio]-1,3-benzothiazoleMus musculus (house mouse)Potency35.481310
4-(3-chlorophenyl)sulfonyl-N-cyclohexyl-N-methyl-3-nitrobenzamideMus musculus (house mouse)Potency35.481310
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(3-methyl-1-piperidinyl)sulfonyl]benzamideMus musculus (house mouse)Potency0.612020
1-(4-methylphenyl)-2-[(1-phenyl-2-imidazolyl)thio]ethanoneMus musculus (house mouse)Potency22.740620
3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-4-(4-fluorophenyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency12.589310
[2-(3,4-dimethylphenyl)-4-quinolinyl]-(1-piperidinyl)methanoneMus musculus (house mouse)Potency22.387210
2-(4-chlorophenyl)-3-methyl-N-(2-thiazolyl)butanamideMus musculus (house mouse)Potency17.039020
5-(4-methylphenyl)-2-methylsulfonyl-3-thiophen-2-yl-3,4-dihydropyrazoleMus musculus (house mouse)Potency0.891310
4-(4-morpholinyl)-3-nitro-N-(2-thiazolyl)benzamideMus musculus (house mouse)Potency35.481320
2-[(5-methyl-4-phenyl-2-thiazolyl)methyl]-4-thiazololMus musculus (house mouse)Potency11.220210
LSM-16826Mus musculus (house mouse)Potency35.481310
N-[2-(2,4,6-trinitrophenyl)ethyl]anilineMus musculus (house mouse)Potency10.000010
N-(1,3-benzodioxol-5-yl)-6-chloro-2-(2-pyridinyl)-3-imidazo[1,2-a]pyridinamineMus musculus (house mouse)Potency9.581820
3-[(4-bromophenoxy)methyl]benzohydrazideMus musculus (house mouse)Potency17.782810
5H-phenanthridine-6-thioneMus musculus (house mouse)Potency13.347720
2-[[5-(cyclohexylamino)-1,3,4-thiadiazol-2-yl]thio]-N-(9,10-dioxo-2-anthracenyl)acetamideMus musculus (house mouse)Potency12.589310
sb 408124Mus musculus (house mouse)Potency10.000010
2-(2-fluoroanilino)-3-pyridinecarboxylic acid [2-[(1,1-dioxo-3-thiolanyl)-methylamino]-2-oxoethyl] esterMus musculus (house mouse)Potency8.912510
2,4-dichloro-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency0.586620
1,3-benzodioxol-5-yl-[2-(phenylmethylthio)-4,5-dihydroimidazol-1-yl]methanoneMus musculus (house mouse)Potency3.548110
1-benzoyl-5-hydroxy-5-(4-methylphenyl)-4H-pyrazole-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency19.091920
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterMus musculus (house mouse)Potency15.848910
N-(3-methoxyphenyl)-1,3-dioxo-2-(2-oxolanylmethyl)-5-isoindolecarboxamideMus musculus (house mouse)Potency14.125410
1-(4-methoxyphenyl)-N-(2-oxolanylmethyl)-4-pyrazolo[3,4-d]pyrimidinamineMus musculus (house mouse)Potency35.481310
2-[4-[[[[(2,4-dichlorophenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-3-methylphenyl]-3,3,3-trifluoro-2-hydroxypropanoic acid ethyl esterMus musculus (house mouse)Potency24.035320
pd 407824Mus musculus (house mouse)Potency35.481310
2-(N-(2-chloro-1-oxoethyl)-4-fluoroanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMus musculus (house mouse)Potency23.350720
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMus musculus (house mouse)Potency15.848910
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideMus musculus (house mouse)Potency18.854120
2-(3-oxo-2,4-dihydroquinoxalin-1-yl)-2-phenyl-N-(4-propan-2-ylphenyl)acetamideMus musculus (house mouse)Potency22.387210
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thioureaMus musculus (house mouse)Potency8.285220
2-chloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency1.026620
2-furanyl-[4-[(6-hydroxy-2-methyl-5-thiazolo[3,2-b][1,2,4]triazolyl)-thiophen-2-ylmethyl]-1-piperazinyl]methanoneMus musculus (house mouse)Potency0.631010
3-(2-methylphenyl)-2-(2-thiazolyl)-5,6,7,7a-tetrahydro-3H-pyrrolo[1,2-c]imidazol-1-oneMus musculus (house mouse)Potency27.717020
1-tert-butyl-3-[[(2-chlorophenyl)-oxomethyl]amino]thioureaMus musculus (house mouse)Potency0.929620
5-nitro-2-furancarboxylic acid [2-oxo-2-[3-(1-piperidinylsulfonyl)anilino]ethyl] esterMus musculus (house mouse)Potency19.952610
2-[[4-(4-chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]thio]-N-(3-methoxyphenyl)-2-phenylacetamideMus musculus (house mouse)Potency25.118910
5-methyl-4-(3-phenoxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-6-carboxylic acid ethyl esterMus musculus (house mouse)Potency12.431220
N-(1-adamantyl)-6-(3,5-dimethyl-1-pyrazolyl)-1,2,4,5-tetrazin-3-amineMus musculus (house mouse)Potency21.450920
N2,N6-bis[4-(dimethylamino)phenyl]pyridine-2,6-dicarboxamideMus musculus (house mouse)Potency19.952610
N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-4-propan-2-yloxybenzamideMus musculus (house mouse)Potency20.811420
4-bromo-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency0.112210
N-(3-chlorophenyl)-2-[4-oxo-2-phenylimino-3-(2-pyridinylmethyl)-5-thiazolidinyl]acetamideMus musculus (house mouse)Potency6.309610
4-[1-(4-fluorophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-oneMus musculus (house mouse)Potency35.481320
1-(2-methoxy-3-dibenzofuranyl)-3-(3-methylphenyl)thioureaMus musculus (house mouse)Potency28.934220
2-Chloro-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneMus musculus (house mouse)Potency26.632020
2-(3-oxo-4H-1,4-benzothiazin-2-yl)acetic acid (7-methoxy-2-oxo-1-benzopyran-4-yl)methyl esterMus musculus (house mouse)Potency17.782810
N-[5-(phenylmethyl)-2-thiazolyl]-4,5-dihydro-1H-imidazole-2-carboxamideMus musculus (house mouse)Potency14.236640
2-(4-chlorophenoxy)-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamideMus musculus (house mouse)Potency22.387210
N-(4-ethylphenyl)-2-[[3-[3-(4-methyl-1-piperidinyl)propyl]-4-oxo-2-quinazolinyl]thio]acetamideMus musculus (house mouse)Potency25.118910
2,6-difluoro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency2.484020
4-(1,3-dioxo-2-benzo[de]isoquinolinyl)butanoic acid [2-(2-acetylanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency5.623410
1-methyl-3-(6,7,8,9-tetrahydro-5H-carbazol-3-ylmethyl)thioureaMus musculus (house mouse)Potency17.782810
2,6-diphenyl-7-pyrazolo[1,5-a]pyrimidinamineMus musculus (house mouse)Potency3.399820
2,5-dichloro-N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-3-thiophenecarboxamideMus musculus (house mouse)Potency2.837120
N-[4-[5-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-4-pyridinecarboxamideMus musculus (house mouse)Potency0.005010
2-chloro-N-(2,6-dimethylphenyl)-3-oxo-3-phenylpropanamideMus musculus (house mouse)Potency23.753120
N-[4-chloro-3-(dimethylsulfamoyl)phenyl]-2-[(phenylmethyl)amino]acetamideMus musculus (house mouse)Potency11.220210
2-thiophen-2-yl-N-[5-[[4-(trifluoromethyl)phenyl]methylthio]-1,3,4-thiadiazol-2-yl]acetamideMus musculus (house mouse)Potency10.000010
3-chloro-N-[3-(2-methoxyethyl)-6-sulfamoyl-1,3-benzothiazol-2-ylidene]-1-benzothiophene-2-carboxamideMus musculus (house mouse)Potency15.848910
N-[1-(1H-benzimidazol-2-yl)-3-(methylthio)propyl]-3,5-dinitrobenzamideMus musculus (house mouse)Potency25.118910
2-hydroxy-5-[(4-methoxyphenyl)sulfamoyl]benzoic acid [2-[1-(3-bicyclo[2.2.1]heptanyl)ethylamino]-2-oxoethyl] esterMus musculus (house mouse)Potency7.943310
8-[4-(4-fluorophenoxy)-3-nitrophenyl]-7-(2-hydroxyethyl)-3-(phenylmethyl)purine-2,6-dioneMus musculus (house mouse)Potency17.782810
1-cyclohexyl-3-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)thioureaMus musculus (house mouse)Potency15.848910
N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]-4-[(2-methyl-1-piperidinyl)sulfonyl]benzamideMus musculus (house mouse)Potency0.669420
N-[3-[(2-bromo-5-methylphenyl)sulfamoyl]-4-methoxyphenyl]-4-fluorobenzamideMus musculus (house mouse)Potency12.589310
N-[3-(1-azepanylsulfonyl)phenyl]-2-[4-(1H-indol-3-ylmethyl)-2,5-dioxo-1-imidazolidinyl]acetamideMus musculus (house mouse)Potency5.011910
N-(1H-benzimidazol-2-yl)-3-phenylbutanamideMus musculus (house mouse)Potency12.209720
N-(7-methyl-2-thiazolo[4,5-g][1,3]benzothiazolyl)propanamideMus musculus (house mouse)Potency3.642620
6-chloro-2-[(phenylmethylthio)methyl]imidazo[1,2-a]pyridineMus musculus (house mouse)Potency35.481310
1-(4-methoxyphenyl)-3-(1-thiophen-2-ylpropan-2-yl)thioureaMus musculus (house mouse)Potency8.471920
5-[(4-phenyl-1-piperazinyl)-thiophen-2-ylmethyl]-6-thiazolo[3,2-b][1,2,4]triazololMus musculus (house mouse)Potency0.112210
N-[(3,5-dimethyl-1-piperidinyl)-sulfanylidenemethyl]-2-methyl-5-(4-morpholinylsulfonyl)benzamideMus musculus (house mouse)Potency3.298420
3-(4-ethoxyphenyl)-N-[(1-methyl-4-piperidinylidene)amino]-1H-pyrazole-5-carboxamideMus musculus (house mouse)Potency17.782820
4-(1-imidazolyl)-3,5-dinitrobenzoic acid methyl esterMus musculus (house mouse)Potency10.000010
4-methyl-N-[2-[(5-oxo-2,3-dihydrothiazolo[2,3-b]quinazolin-3-yl)methylthio]phenyl]benzamideMus musculus (house mouse)Potency22.387210
4-[4-[(5-chloro-2-hydroxyphenyl)-oxomethyl]-1-pyrazolyl]-N-(4-methoxyphenyl)-3-nitrobenzenesulfonamideMus musculus (house mouse)Potency11.220210
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-4-(4-methyl-1-piperidinyl)-3-nitrobenzamideMus musculus (house mouse)Potency17.782810
[5-(2-furanyl)-3-isoxazolyl]-(4-methyl-1-piperidinyl)methanoneMus musculus (house mouse)Potency1.995310
1-(3,4-dihydro-2H-quinolin-1-yl)-2-[[1-(4-ethoxyphenyl)-2-imidazolyl]thio]ethanoneMus musculus (house mouse)Potency21.280420
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-2-oxolanecarboxamideMus musculus (house mouse)Potency1.412510
1-amino-3-(4-chloro-2-methoxy-5-methylphenyl)thioureaMus musculus (house mouse)Potency18.996620
2,4-dichloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency1.584920
2-[2-[(3-chloro-1-benzothiophen-2-yl)-oxomethyl]imino-6-sulfamoyl-1,3-benzothiazol-3-yl]acetic acid ethyl esterMus musculus (house mouse)Potency22.387210
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(6-methyl-2-nitro-3-pyridinyl)oxy]ethanoneMus musculus (house mouse)Potency26.632020
4-[bis(2-methoxyethyl)sulfamoyl]-N-[5-(methoxymethyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency22.387210
2-(2-furanyl)-4-mercapto-3-(4-methylphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileMus musculus (house mouse)Potency15.848910
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[(phenylmethyl)amino]ethyl] esterMus musculus (house mouse)Potency11.220210
4-dimethoxyphosphoryl-2-(1-naphthalenyl)-N-(phenylmethyl)-5-oxazolamineMus musculus (house mouse)Potency35.481310
1-[4-[[4-[[(2-methoxyanilino)-sulfanylidenemethyl]amino]cyclohexyl]methyl]cyclohexyl]-3-(2-methoxyphenyl)thioureaMus musculus (house mouse)Potency3.355220
4-[2-[[1-(2-methoxyethyl)-2-benzimidazolyl]thio]-1-oxoethyl]-2,5-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency21.169920
4-cyano-N-[4-thiophen-2-yl-5-(2,2,2-trifluoro-1-oxoethyl)-2-thiazolyl]benzamideMus musculus (house mouse)Potency17.392620
2-methyl-1-phenyl-5-benzimidazolecarboxylic acid [2-(3-methylbutan-2-ylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency28.183810
5-bromo-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)-2-thiophenecarboxamideMus musculus (house mouse)Potency1.006620
4-(1-azepanylsulfonyl)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-hydroxyphenyl]benzamideMus musculus (house mouse)Potency26.632020
1-[4-(2-fluorophenyl)-1-piperazinyl]-4-(4,4,6-trimethyl-2-sulfanylidene-1,3-diazinan-1-yl)-1-butanoneMus musculus (house mouse)Potency18.256320
4-chloro-N-[3-(N-methylanilino)-1,4-dioxo-2-naphthalenyl]benzamideMus musculus (house mouse)Potency11.220220
2-[(2-nitrophenyl)thio]-1-cyclooctanoneMus musculus (house mouse)Potency14.976320
4-chloro-N-[3-(4-fluorophenyl)-5-[2-(4-methoxyanilino)-2-oxoethyl]-4-oxo-2-sulfanylidene-1-imidazolidinyl]benzamideMus musculus (house mouse)Potency15.586420
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-2-(2-fluorophenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxamideMus musculus (house mouse)Potency15.649820
4-(5-methyl-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)benzoic acid 8-quinolinyl esterMus musculus (house mouse)Potency4.736020
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency5.623410
3-(2,6-dimethyl-3-oxo-1,4-benzoxazin-4-yl)-N-(thiophen-2-ylmethyl)propanamideMus musculus (house mouse)Potency35.481310
5-(4-nitrophenyl)-3-phenyl-1H-imidazole-2-thioneMus musculus (house mouse)Potency2.391520
4-(4-chlorophenyl)-3-[2-(4-methylphenyl)cyclopropyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency6.409220
[4-[(4-bromo-3,5-dimethyl-1-pyrazolyl)methyl]phenyl]-[5-hydroxy-3-methyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]methanoneMus musculus (house mouse)Potency15.186120
3-[(4-methoxyphenoxy)methyl]-N-(4-nitro-1-pyrazolyl)benzamideMus musculus (house mouse)Potency0.891310
8-nitro-5-[3-(trifluoromethyl)-1-piperidinyl]isoquinolineMus musculus (house mouse)Potency28.934220
3-[2-(2,4-dichlorophenoxy)ethoxy]-6-methyl-2-nitropyridineMus musculus (house mouse)Potency19.952610
2-(3,4-dichlorophenyl)-N-[3-(dimethylsulfamoyl)-4-methylphenyl]acetamideMus musculus (house mouse)Potency17.782810
2-(4-benzoylphenoxy)-N-(4-methylcyclohexyl)acetamideMus musculus (house mouse)Potency35.481320
1-(2,4-difluorophenyl)-3-[4-(2-pyridinyl)-2-thiazolyl]ureaMus musculus (house mouse)Potency3.183220
1-(4-methoxyphenyl)-3-[3-(1-piperidinylsulfonyl)phenyl]thioureaMus musculus (house mouse)Potency26.632020
1-[2-(trifluoromethyl)phenyl]sulfonyl-4-piperidinecarboxylic acid [2-[(4-fluorophenyl)methylamino]-2-oxoethyl] esterMus musculus (house mouse)Potency22.387210
N-[4-(4-fluorophenyl)-2-thiazolyl]-3-methoxy-4-[2-(4-morpholinyl)-2-oxoethoxy]benzamideMus musculus (house mouse)Potency5.011910
6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid [2-[4-methyl-3-(1-piperidinylsulfonyl)anilino]-2-oxoethyl] esterMus musculus (house mouse)Potency35.481310
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[[oxo-[(phenylmethyl)amino]methyl]amino]ethyl] esterMus musculus (house mouse)Potency17.782810
[[2-[(4,5-dimethyl-2-thiazolyl)amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esterMus musculus (house mouse)Potency24.035320
2-[(2,6-dichlorophenyl)sulfonylamino]-3-methylbutanoic acid [2-(1H-indol-3-yl)-2-oxoethyl] esterMus musculus (house mouse)Potency12.589310
N-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxolanylmethoxy)benzamideMus musculus (house mouse)Potency35.481310
1-[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-[3-(dimethylamino)propyl]thioureaMus musculus (house mouse)Potency16.803720
4-[4-(4-acetylphenyl)-1-piperazinyl]-N-[3-(dimethylamino)propyl]-3-nitrobenzenesulfonamideMus musculus (house mouse)Potency35.481310
LSM-28572Mus musculus (house mouse)Potency19.952610
2-(Chloroacetyl)-N,2-diphenylhydrazinecarboxamideMus musculus (house mouse)Potency20.085020
2-chloro-1-[1-(3-isoxazolyl)-2,5-dimethyl-3-pyrrolyl]ethanoneMus musculus (house mouse)Potency15.649820
4-(4-chlorophenyl)-3-(phenylmethyl)-1H-imidazole-2-thioneMus musculus (house mouse)Potency2.665120
2,5-dimethyl-3-furancarboxylic acid [2-(2-ethoxyanilino)-2-oxo-1-phenylethyl] esterMus musculus (house mouse)Potency35.481310
N-[2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]benzamideMus musculus (house mouse)Potency19.952610
6-chloro-N-[3-[(2-chlorophenyl)sulfamoyl]phenyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency6.309620
N-(1H-benzimidazol-2-yl)-2-nitrobenzamideMus musculus (house mouse)Potency15.649820
4-methyl-7-[[4-[[4-(4-nitrophenyl)-1-piperazinyl]-oxomethyl]phenyl]methoxy]-1-benzopyran-2-oneMus musculus (house mouse)Potency5.623410
2-[(2-chlorophenyl)methoxy]-N-(4,5-dihydrothiazol-2-yl)benzamideMus musculus (house mouse)Potency22.740620
N-[4-methoxy-3-(4-morpholinylsulfonyl)phenyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideMus musculus (house mouse)Potency10.000010
3'-[2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]spiro[6,7-dihydro-5H-1-benzothiophene-4,5'-imidazolidine]-2',4'-dioneMus musculus (house mouse)Potency28.934220
N-(4-tert-butylphenyl)-2-[4-(1-imidazolyl)phenoxy]acetamideMus musculus (house mouse)Potency10.000010
5'-bromo-2'-spiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3'-1H-indole]oneMus musculus (house mouse)Potency14.501520
2-(4-benzoylphenoxy)-N-[4-(propan-2-ylsulfamoyl)phenyl]propanamideMus musculus (house mouse)Potency21.280420
3-[(2,5,6-trimethyl-4-thieno[2,3-d]pyrimidinyl)thio]-2-oxolanoneMus musculus (house mouse)Potency13.534620
2-(2-chloro-4-methylanilino)-N-[3-(dimethylsulfamoyl)phenyl]acetamideMus musculus (house mouse)Potency8.205620
N-[2-[1-(3,5-dimethyl-1-piperidinyl)-1-oxopropan-2-yl]oxyphenyl]acetamideMus musculus (house mouse)Potency12.589310
N-(4,5-dithiophen-2-yl-2-thiazolyl)-2-methyl-1-cyclopropanecarboxamideMus musculus (house mouse)Potency10.000010
2-[[4-(3,4-dimethylphenyl)-1-phenyl-2-imidazolyl]thio]-N-(1,1-dioxo-3-thiolanyl)acetamideMus musculus (house mouse)Potency12.589320
2-[2,5-diethoxy-4-(4-morpholinyl)anilino]-1-(4-methyl-1-piperidinyl)-1-propanoneMus musculus (house mouse)Potency11.220210
N-(3-chloro-4-fluorophenyl)-2-[5-(dimethylsulfamoyl)-2-(ethylamino)anilino]acetamideMus musculus (house mouse)Potency16.815820
2-(4-benzoyl-1-piperazinyl)-N-(2-phenylphenyl)propanamideMus musculus (house mouse)Potency14.125410
N-[[[2-(2-naphthalenyloxy)-1-oxopropyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency22.740620
N-[[1-(2-phenoxyethyl)-2-benzimidazolyl]methyl]anilineMus musculus (house mouse)Potency24.035320
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[[2-(2-pyridinyl)-1-benzimidazolyl]methyl]-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency17.488220
1-(4-bromophenyl)-1'-methyl-6'-nitro-2'-phenylspiro[1,3-diazinane-5,3'-2,4-dihydroquinoline]-2,4,6-trioneMus musculus (house mouse)Potency22.387210
N-[3-(1-imidazolyl)propyl]-2-methyl-3-phenyl-5-propyl-7-pyrazolo[1,5-a]pyrimidinamineMus musculus (house mouse)Potency1.584910
LSM-24595Mus musculus (house mouse)Potency27.717020
3-(1-methyl-2-benzimidazolyl)-1-(3-methylphenyl)-2-pyrrolo[3,2-b]quinoxalinamineMus musculus (house mouse)Potency3.915220
N-(4-Nitro-1,2,5-oxadiazol-3-yl)-2-pyridin-2-ylsulfanylacetamideMus musculus (house mouse)Potency5.317720
[5-(4-fluorophenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[2-(3-pyridinyl)-1-piperidinyl]methanoneMus musculus (house mouse)Potency35.481320
6-(4-methoxyphenyl)-8-methyl-4-oxo-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylic acid O7-ethyl ester O2-methyl esterMus musculus (house mouse)Potency4.044020
N-(4-ethoxyphenyl)-2-[5-oxo-1-phenyl-3-(2-pyridinylmethyl)-2-sulfanylidene-4-imidazolidinyl]acetamideMus musculus (house mouse)Potency12.589310
2-Chloro-1-[5-(furan-2-yl)-3-(5-methylfuran-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneMus musculus (house mouse)Potency14.501520
5-(4-methylphenyl)-2-(1-piperidinyl)-7-thiazolo[4,5-b]pyridinecarboxylic acidMus musculus (house mouse)Potency11.220210
3-(2-methoxyphenyl)-4-phenyl-1H-imidazole-2-thioneMus musculus (house mouse)Potency4.220920
4-(4-methylphenyl)-3-phenyl-1H-imidazole-2-thioneMus musculus (house mouse)Potency3.135420
2-(4-oxo-3-quinazolinyl)-N-[3-(1-piperidinylsulfonyl)phenyl]acetamideMus musculus (house mouse)Potency5.388220
1-(4-carbamoyl-2-nitrophenyl)-4-piperidinecarboxylic acid methyl esterMus musculus (house mouse)Potency35.481310
3-[5-(diethylsulfamoyl)-1-methyl-2-benzimidazolyl]propanoic acid [2-(3,5-dichloroanilino)-2-oxoethyl] esterMus musculus (house mouse)Potency15.848910
2-[8-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-1,3-dimethyl-2,6-dioxo-7-purinyl]acetic acid methyl esterMus musculus (house mouse)Potency5.634250
N2-(2-furanylmethyl)-6-(3-methyl-1-piperidinyl)-5-nitropyrimidine-2,4-diamineMus musculus (house mouse)Potency19.952610
2-amino-5-nitrophenolMus musculus (house mouse)Potency19.952610
N-[(4-chlorophenyl)methyl]-2-[[[(2-fluorophenyl)methyl-(phenylmethyl)amino]-sulfanylidenemethyl]amino]acetamideMus musculus (house mouse)Potency1.995310
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(4-methoxyphenyl)-2-thiophenecarboxamideMus musculus (house mouse)Potency5.623410
3-amino-N-(2-chlorophenyl)-4-(1-pyrrolidinyl)benzenesulfonamideMus musculus (house mouse)Potency35.481310
1-(7-methyloctyl)-3-[4-(4-morpholinylsulfonyl)phenyl]thioureaMus musculus (house mouse)Potency22.387220
7-chloro-3-[2-(1-cyclohexenyl)ethyl]-2-sulfanylidene-1H-quinazolin-4-oneMus musculus (house mouse)Potency1.885420
4-bromo-N-[(4-ethoxy-2-nitroanilino)-sulfanylidenemethyl]-2-methyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency22.387210
N-(3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(2-chlorophenyl)-5-methyl-4-isoxazolecarboxamideMus musculus (house mouse)Potency5.623410
3-[4-(dimethylamino)phenyl]-1-[1-(3-methylphenyl)-2,5-dioxo-3-pyrrolidinyl]-1-[(1,3,5-trimethyl-4-pyrazolyl)methyl]thioureaMus musculus (house mouse)Potency0.069920
5-[(5-bromo-2-hydroxyphenyl)-oxomethyl]-1-cyclohexyl-2-oxo-3-pyridinecarbonitrileMus musculus (house mouse)Potency19.952610
cgp 7930Mus musculus (house mouse)Potency22.874120
[3-(2-hydroxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-thiophen-2-ylmethanoneMus musculus (house mouse)Potency12.589310
1-(5-chloro-2,4-dimethoxyphenyl)-3-(phenylmethyl)thioureaMus musculus (house mouse)Potency16.803720
N,N-dimethyl-3-(3-oxo-1,2-benzothiazol-2-yl)benzenesulfonamideMus musculus (house mouse)Potency27.717020
N-(1,3-benzodioxol-5-yl)-4-(4-methyl-1-piperidinyl)-3-nitrobenzamideMus musculus (house mouse)Potency11.220210
(4-chloro-1-ethyl-3-pyrazolyl)-[3-(2-hydroxyphenyl)-5-(2-naphthalenyl)-3,4-dihydropyrazol-2-yl]methanoneMus musculus (house mouse)Potency23.735820
2-(4,5-dihydrothiazol-2-ylthio)-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]acetamideMus musculus (house mouse)Potency35.481310
5-[2-furanyl-[4-(phenylmethyl)-1-piperidinyl]methyl]-6-thiazolo[3,2-b][1,2,4]triazololMus musculus (house mouse)Potency12.774820
1-butyl-3-[[oxo-(5-propan-2-yl-3-thiophenyl)methyl]amino]thioureaMus musculus (house mouse)Potency12.863120
1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-3-(4,4,6-trimethyl-2-sulfanylidene-1,3-diazinan-1-yl)-1-propanoneMus musculus (house mouse)Potency13.427020
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideMus musculus (house mouse)Potency1.995310
1-(2-furanylmethyl)-3-(3-methoxyphenyl)-1-[2-(2-methyl-1H-indol-3-yl)ethyl]thioureaMus musculus (house mouse)Potency23.350720
imd 0354Mus musculus (house mouse)Potency0.880620
4-(dimethylsulfamoyl)-N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency2.081220
1-cyclohexyl-N-(3-methylbutyl)-5-benzimidazolecarboxamideMus musculus (house mouse)Potency24.803320
N-methyl-2-[[[4-[methyl(phenyl)sulfamoyl]phenyl]-oxomethyl]amino]-6-propyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamideMus musculus (house mouse)Potency7.562720
5-(2,4-dichlorophenyl)-4,6-dioxo-3a,6a-dihydro-2H-pyrrolo[3,4-d]isoxazole-3,3-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency17.782810
1-cyclohexyl-3-(1,1-dioxo-2,5-dihydrothiophen-3-yl)-1-methylthioureaMus musculus (house mouse)Potency19.952610
2-[3-(2-furanylmethyl)-2-(4-methoxyphenyl)imino-4-oxo-5-thiazolidinyl]-N-(2-methoxyphenyl)acetamideMus musculus (house mouse)Potency0.004510
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency1.267320
N-(4-methoxyphenyl)sulfonyl-N-(2-oxo-5-benzo[g][1,3]benzoxathiolyl)-2-furancarboxamideMus musculus (house mouse)Potency33.552020
1-[2-[(4-pentoxyphenyl)methylthio]ethyl]-3-phenylthioureaMus musculus (house mouse)Potency3.162320
[5-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-3-pyrazolyl]-(4-morpholinyl)methanoneMus musculus (house mouse)Potency18.860020
1-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-3-phenylureaMus musculus (house mouse)Potency11.220210
3-(4-methyl-1,3-dioxan-2-yl)-1-benzopyran-4-oneMus musculus (house mouse)Potency24.803320
2,6-difluoro-N-[2-[3-[(2-fluorophenyl)methylthio]-1-indolyl]ethyl]benzamideMus musculus (house mouse)Potency33.552020
2-[4-(4-chloro-2-nitrophenyl)-1-piperazinyl]phenolMus musculus (house mouse)Potency15.848910
5-[(2,4-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]-4-pyrazolyl]-2-furancarboxamideMus musculus (house mouse)Potency17.782810
4,5,6,7-tetrabromobenzimidazoleMus musculus (house mouse)Potency25.118910
4-[3-(2-chloro-1-oxoethyl)-2,5-dimethyl-1-pyrrolyl]-1,5-dimethyl-2-phenyl-3-pyrazoloneMus musculus (house mouse)Potency25.665120
[5-[(3,5-dimethyl-4-nitro-1-pyrazolyl)methyl]-2-furanyl]-[5-hydroxy-3-methyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]methanoneMus musculus (house mouse)Potency4.795720
(3,5-dichloroanilino)thioureaMus musculus (house mouse)Potency3.109920
N-(4-phenoxyphenyl)-2-(1,2,3,4-tetrahydroisoquinolin-1-yl)acetamideMus musculus (house mouse)Potency27.717020
2-[[3-butyl-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideMus musculus (house mouse)Potency5.792420
N-[[(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-2-methylbenzamideMus musculus (house mouse)Potency16.531120
4-[5-(3-chlorophenyl)-2-furanyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid methyl esterMus musculus (house mouse)Potency18.256320
4-(3,4-dimethoxyphenyl)-3,4,5,6-tetrahydro-1H-benzo[h]quinazoline-2-thioneMus musculus (house mouse)Potency3.135420
5,6-dimethyl-1-octyl-4-benzimidazolamineMus musculus (house mouse)Potency19.091920
2-[(6-chloro-2-phenyl-1-benzimidazolyl)oxy]acetic acidMus musculus (house mouse)Potency24.803320
4-tert-butyl-N-[3-[4-[3-[[(4-tert-butylphenyl)-oxomethyl]amino]propyl]-1-piperazinyl]propyl]benzamideMus musculus (house mouse)Potency9.834420
4-[1-[2-(3,4-dimethoxyphenyl)ethyl]-3-(4-methoxyphenoxy)-4-oxo-2-azetidinyl]benzoic acid methyl esterMus musculus (house mouse)Potency1.000010
sib 1757Mus musculus (house mouse)Potency1.909220
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2-oxo-1-benzopyran-3-carboxamideMus musculus (house mouse)Potency10.000010
3-nitro-4-[2-[1-(phenylmethyl)-4-piperidinylidene]hydrazinyl]benzenesulfonamideMus musculus (house mouse)Potency26.632020
2-[[4-amino-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]thio]-1-(1H-indol-3-yl)-2-phenylethanoneMus musculus (house mouse)Potency15.848910
N-(3-nitrophenyl)-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency22.387210
N-(6-methyl-1,3-benzothiazol-2-yl)-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamideMus musculus (house mouse)Potency19.149820
N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-5,6-dimethyl-4-thieno[2,3-d]pyrimidinamineMus musculus (house mouse)Potency5.500020
bergaptolMus musculus (house mouse)Potency15.848910
biochanin aMus musculus (house mouse)Potency24.035320
prostaglandin b1Mus musculus (house mouse)Potency7.943310
acacetinMus musculus (house mouse)Potency28.183810
apigeninMus musculus (house mouse)Potency16.723020
luteolinMus musculus (house mouse)Potency22.746420
calcitriolMus musculus (house mouse)Potency13.457420
retinol palmitateMus musculus (house mouse)Potency6.309610
quercetin 3-o-methyl etherMus musculus (house mouse)Potency8.116020
15-ketoprostaglandin e2Mus musculus (house mouse)Potency1.122010
cholecalciferolMus musculus (house mouse)Potency16.034320
prostaglandin a2Mus musculus (house mouse)Potency19.149820
harmineMus musculus (house mouse)Potency20.080920
genisteinMus musculus (house mouse)Potency15.848910
pulmicortMus musculus (house mouse)Potency12.589310
methysergide maleateMus musculus (house mouse)Potency26.632020
capsanthinMus musculus (house mouse)Potency12.589310
geranylgeraniolMus musculus (house mouse)Potency6.309610
chartreusinMus musculus (house mouse)Potency23.350720
methysticinMus musculus (house mouse)Potency0.125910
zearalenoneMus musculus (house mouse)Potency33.552010
baicaleinMus musculus (house mouse)Potency22.157420
chrysinMus musculus (house mouse)Potency20.929420
hispidulinMus musculus (house mouse)Potency35.481320
gentiacauleinMus musculus (house mouse)Potency12.589310
3-hydroxyblancoxanthoneMus musculus (house mouse)Potency19.321820
mangostinMus musculus (house mouse)Potency27.982620
rhamnetinMus musculus (house mouse)Potency12.313020
santinMus musculus (house mouse)Potency22.387210
Pinosylvin methyl etherMus musculus (house mouse)Potency35.481310
pterostilbeneMus musculus (house mouse)Potency6.446820
caffeic acid phenethyl esterMus musculus (house mouse)Potency18.131320
wedelolactoneMus musculus (house mouse)Potency14.219120
cephalomannineMus musculus (house mouse)Potency6.464820
ellagic acidMus musculus (house mouse)Potency35.481310
flupenthixolMus musculus (house mouse)Potency28.934220
prostaglandin a1Mus musculus (house mouse)Potency8.912510
l 683590Mus musculus (house mouse)Potency6.309610
arachidonyl dopamineMus musculus (house mouse)Potency11.220210
n-oleoyldopamineMus musculus (house mouse)Potency15.954120
cilnidipineMus musculus (house mouse)Potency11.676620
sofalconeMus musculus (house mouse)Potency14.125410
tranilastMus musculus (house mouse)Potency3.398120
4-hydroxyestradiolMus musculus (house mouse)Potency15.848910
4-hydroxychalconeMus musculus (house mouse)Potency17.782810
4'-hydroxychalconeMus musculus (house mouse)Potency23.350720
misoprostolMus musculus (house mouse)Potency35.481310
calcifediolMus musculus (house mouse)Potency7.426920
2-bromoergocryptine mesylateMus musculus (house mouse)Potency27.717020
perhexiline maleateMus musculus (house mouse)Potency27.850620
beta-nitrostyreneMus musculus (house mouse)Potency35.481310
tetrachlorvinphosMus musculus (house mouse)Potency17.782810
sirolimusMus musculus (house mouse)Potency33.552020
afimoxifeneMus musculus (house mouse)Potency23.753120
fenretinideMus musculus (house mouse)Potency15.685720
geldanamycinMus musculus (house mouse)Potency4.466810
su 9516Mus musculus (house mouse)Potency12.031720
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acidMus musculus (house mouse)Potency9.834420
N-(4-chlorophenoxy)sulfonylcarbamic acid [(1R,9aR)-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizin-1-yl]methyl esterMus musculus (house mouse)Potency5.011910
3-ethyl-2-sulfanylidene-6,7,8,9-tetrahydro-1H-pyrimido[4,5-b]quinolin-4-oneMus musculus (house mouse)Potency16.603820
N-(4-bromo-3-methylphenyl)-2,5-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineMus musculus (house mouse)Potency12.589310
N-[3-(3-chlorophenyl)-5-isoxazolyl]-2-(4,5,6,7-tetrahydroindazol-2-yl)acetamideMus musculus (house mouse)Potency19.118020
3-[(5-chloro-2-pyridinyl)amino]-2-(2-pyridinyl)-3H-isoindol-1-oneMus musculus (house mouse)Potency5.011910
4-[[1-(6-ethoxy-1,3-benzothiazol-2-yl)-3-piperidinyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency5.623410
2-(4-fluoro-3-methylphenyl)sulfonyl-5-(2-methoxyphenyl)-3-pyrazolamineMus musculus (house mouse)Potency12.589310
3-(4-chlorophenyl)-N-cyclopropyl-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideMus musculus (house mouse)Potency7.183820
4-[[[2-(4-methoxyphenyl)-3-oxo-1H-isoindol-4-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency3.548110
2,5-dimethyl-N-(3,4,5-trimethoxyphenyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineMus musculus (house mouse)Potency12.589310
N-(3,5-dimethylphenyl)-2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideMus musculus (house mouse)Potency13.534620
3-[[2-(2-furanylmethyl)-3-oxo-1H-isoindol-1-yl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency13.357420
[1-[(3,5-dimethyl-4-isoxazolyl)sulfonyl]-4-piperidinyl]-[4-(1-piperidinyl)-1-piperidinyl]methanoneMus musculus (house mouse)Potency22.387210
2-(5-chloro-2-pyridinyl)-3-(4-ethoxyanilino)-3H-isoindol-1-oneMus musculus (house mouse)Potency31.622810
N-(5-bromo-2-thiazolyl)-3-phenyl-2-(1-pyrrolyl)propanamideMus musculus (house mouse)Potency16.271020
4-[[[1-[[2-(3-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-3-piperidinyl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency15.866020
2-[[5-methyl-2-(3-methylphenyl)-4-oxazolyl]methylsulfinyl]-N-(2-oxolanylmethyl)acetamideMus musculus (house mouse)Potency35.481310
[2-(1-piperidinyl)-1,3-benzothiazol-6-yl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency35.481310
4-[5-(4-methoxyphenyl)-3-isoxazolyl]-N-(2-pyridinylmethyl)butanamideMus musculus (house mouse)Potency0.079410
N-(2,5-dimethoxyphenyl)-2-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methylsulfonyl]acetamideMus musculus (house mouse)Potency3.548110
N-(4-ethylphenyl)-2-(2-furanylmethyl)-1,3-dioxo-5-isoindolecarboxamideMus musculus (house mouse)Potency11.220210
4-[3-(4-fluorophenyl)-2-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency11.294720
N-(2-oxolanylmethyl)-2-(1-piperidinyl)-1,3-benzothiazole-6-carboxamideMus musculus (house mouse)Potency9.834420
N-(5-bromo-2-hydroxyphenyl)-5-propyl-3-isoxazolecarboxamideMus musculus (house mouse)Potency7.079510
4-[4-[[[1-(2-methylpropyl)-3-pyrrolidinyl]methylamino]-oxomethyl]-3-oxo-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.707910
N-(4-chlorophenyl)-2-[[4-(4-methoxyphenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideMus musculus (house mouse)Potency35.481310
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-(3-methoxyphenyl)butanamideMus musculus (house mouse)Potency0.416920
N-(3-acetylphenyl)-5-propan-2-yl-3-isoxazolecarboxamideMus musculus (house mouse)Potency23.350720
3-(3,4-dimethoxyphenyl)-5,7-dihydroxy-2-methyl-1-benzopyran-4-oneMus musculus (house mouse)Potency17.782810
4-[[2-[4-(2-chlorophenyl)-2-oxo-6,7-dihydro-5H-cyclopenta[b]pyridin-1-yl]-1-oxoethyl]amino]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481310
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[5-methyl-2-(4-methylphenyl)-4-oxazolyl]methylsulfonyl]ethanoneMus musculus (house mouse)Potency14.125410
3-(4-chlorophenyl)-N-[2-(diethylamino)ethyl]-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideMus musculus (house mouse)Potency11.220210
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideMus musculus (house mouse)Potency22.387210
1-(4-tert-butylphenyl)sulfonyl-N-(2-pyridinylmethyl)-2-piperidinecarboxamideMus musculus (house mouse)Potency18.996620
4-[[5-[(2,6-dichlorophenyl)sulfonylmethyl]-2-furanyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterMus musculus (house mouse)Potency7.943310
8-(2-chlorophenyl)-3-(4-ethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrileMus musculus (house mouse)Potency25.285520
N-(6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamideMus musculus (house mouse)Potency20.552320
N-(5-methyl-3-isoxazolyl)-2-[[3-(3-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]acetamideMus musculus (house mouse)Potency3.162310
N-(2-oxolanylmethyl)-2-[[3-(3-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]acetamideMus musculus (house mouse)Potency1.995310
2-(2-chlorophenyl)-9-(3-methylphenyl)-8-oxo-7H-purine-6-carboxamideMus musculus (house mouse)Potency22.106020
5-ethyl-N-[[2-(3-pyridinyl)-4-thiazolyl]methyl]-2-thiophenesulfonamideMus musculus (house mouse)Potency4.466810
N-[(3-methyl-6-imidazo[2,1-b]thiazolyl)methyl]-1-propanesulfonamideMus musculus (house mouse)Potency35.481310
N-[1-[4-(2-methoxyphenyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]benzenesulfonamideMus musculus (house mouse)Potency31.622810
7-[(2-chloro-6-fluorophenyl)methyl]-1,3-dimethyl-8-[(3-methyl-1-piperidinyl)methyl]purine-2,6-dioneMus musculus (house mouse)Potency0.223910
3-[3-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]propyl]-1H-benzimidazol-2-oneMus musculus (house mouse)Potency2.511910
6-methyl-3-(prop-2-enylthio)-5H-[1,2,4]triazino[5,6-b]indoleMus musculus (house mouse)Potency33.552020
3-(3,5-dimethyl-1-pyrazolyl)-5-phenyl-1,2,4-triazineMus musculus (house mouse)Potency4.224020
arachidonylcyclopropylamideMus musculus (house mouse)Potency35.481320
butaprostMus musculus (house mouse)Potency35.481310
n-(4-amino-2-methylquinolin-6-yl)-2-(4-ethylphenoxymethyl)benzamideMus musculus (house mouse)Potency16.803720
sr 59230aMus musculus (house mouse)Potency10.602520
u-44619Mus musculus (house mouse)Potency15.848910
(3r)-((2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl))methanoneMus musculus (house mouse)Potency19.952610
3-[6-[4-(trifluoromethoxy)anilino]-4-pyrimidinyl]benzamideMus musculus (house mouse)Potency5.623410
cgp 71683 aMus musculus (house mouse)Potency35.481320
kn 62Mus musculus (house mouse)Potency11.220210
sulprostoneMus musculus (house mouse)Potency2.511910
bornyl ferulateMus musculus (house mouse)Potency5.623410
8-geranyloxypsoralenMus musculus (house mouse)Potency12.589310
5-hydroxy-7-(4-hydroxy-3-methoxyphenyl)-1-phenyl-3- heptanoneMus musculus (house mouse)Potency11.220210
5,7-dihydroxy-4',6-dimethoxyflavoneMus musculus (house mouse)Potency11.294720
furazolidoneMus musculus (house mouse)Potency0.501210
erbstatinMus musculus (house mouse)Potency13.534620
tyrphostin ag 555Mus musculus (house mouse)Potency23.029620
tyrphostin ag-494Mus musculus (house mouse)Potency26.632020
tyrphostin b44Mus musculus (house mouse)Potency24.035320
ag 556Mus musculus (house mouse)Potency23.735820
2'-hydroxy-4-methoxychalconeMus musculus (house mouse)Potency39.810710
(2e)-3-phenyl-1-(2,3,4,5-tetrahydro-1,6-benzodioxocin-8-yl)prop-2-en-1-oneMus musculus (house mouse)Potency17.488220
nifuroxazideMus musculus (house mouse)Potency11.904820
bay 11-7082Mus musculus (house mouse)Potency0.842220
farnesylthioacetic acidMus musculus (house mouse)Potency11.904820
oxamflatinMus musculus (house mouse)Potency5.017220
7,8-dihydroxy-4-methylcoumarinMus musculus (house mouse)Potency12.589310
flavokawain bMus musculus (house mouse)Potency24.803320
1-(4-methylpiperazin-1-yl)-3-(5-nitrofuran-2-yl)prop-2-en-1-oneMus musculus (house mouse)Potency23.350720
Isoliquiritigenin 4,4'-dimethyl etherMus musculus (house mouse)Potency4.614410
4-amino-6,7-diphenyl-3H-pteridine-2-thioneMus musculus (house mouse)Potency3.981110
2',4'-dihydroxychalconeMus musculus (house mouse)Potency19.149820
2-(4-(dimethylamino)styryl)benzothiazoleMus musculus (house mouse)Potency2.148620
vincristine sulfateMus musculus (house mouse)Potency19.952610
(3S,3'aR,8'aS,8'bS)-5-ethyl-2'-(phenylmethyl)spiro[1H-indole-3,4'-3a,6,7,8,8a,8b-hexahydropyrrolo[3,4-a]pyrrolizine]-1',2,3'-trioneMus musculus (house mouse)Potency8.912510
6-bromo-5-methyl-1,3-dihydroimidazo[4,5-b]pyridine-2-thioneMus musculus (house mouse)Potency11.220210
3-(1-benzimidazolyl)-6-ethyl-7-hydroxy-1-benzopyran-4-oneMus musculus (house mouse)Potency12.589310
3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5,7-dihydroxy-2-methyl-1-benzopyran-4-oneMus musculus (house mouse)Potency11.220210
N-(2,3-dimethylphenyl)-1-methyl-9H-pyrido[3,4-b]indole-3-carboxamideMus musculus (house mouse)Potency14.125410
nitrofurazoneMus musculus (house mouse)Potency20.895410
4-[6-(2,4-dichlorophenyl)-4-methyl-2-oxo-5-phenylmethoxycarbonyl-1,6-dihydropyrimidin-3-yl]butanoic acidMus musculus (house mouse)Potency26.632020
6-[4-methyl-6-(4-nitrophenyl)-2-oxo-5-phenylmethoxycarbonyl-1,6-dihydropyrimidin-3-yl]hexanoic acidMus musculus (house mouse)Potency9.456210
azodicarbonamideMus musculus (house mouse)Potency11.220210
l 685458Mus musculus (house mouse)Potency11.232220
ici 118551Mus musculus (house mouse)Potency35.481310
n'-((1e)-(4-(diethylamino)phenyl)methylene)-4-hydroxybenzohydrazideMus musculus (house mouse)Potency1.460220
3-(4-fluorophenoxy)-6-methoxy-2-(4-methoxyphenyl)-1-benzothiophene 1-oxideMus musculus (house mouse)Potency23.735820
7-hydroxy-8-methyl-4-[[methyl-(phenylmethyl)amino]methyl]-1-benzopyran-2-oneMus musculus (house mouse)Potency19.952610
3-(dimethylamino)benzoic acid (7-hydroxy-2-oxo-1-benzopyran-4-yl)methyl esterMus musculus (house mouse)Potency10.066420
ethaverine hydrochlorideMus musculus (house mouse)Potency15.848910
fendiline hydrochlorideMus musculus (house mouse)Potency35.481310
tiapridexMus musculus (house mouse)Potency12.589310
bromhexine hydrochlorideMus musculus (house mouse)Potency11.220210
methylbenzethonium chlorideMus musculus (house mouse)Potency10.147420
resiniferatoxinMus musculus (house mouse)Potency19.952610
dithiazanine iodideMus musculus (house mouse)Potency7.875820
3,3'-diethylthiatricarbocyanine iodide, 3h-labeledMus musculus (house mouse)Potency22.874120
quinaldine redMus musculus (house mouse)Potency3.372720
5-(4-methyl-1-naphthalenyl)-N-phenyl-2-furancarboxamideMus musculus (house mouse)Potency33.552020
2',3,4-trihydroxychalconeMus musculus (house mouse)Potency25.118910
CrotaoprostrinMus musculus (house mouse)Potency18.738320
virodhamineMus musculus (house mouse)Potency25.118910
2-(dimethylaminostyryl)-1-ethylpyridiniumMus musculus (house mouse)Potency2.818410
HTS 01037Mus musculus (house mouse)Potency35.481310
chloride of pseudoisocyanineMus musculus (house mouse)Potency5.865420
5233705 compoundMus musculus (house mouse)Potency115.090820
3',4'-dihydroxyauroneMus musculus (house mouse)Potency25.665120
derruboneMus musculus (house mouse)Potency7.459820
gw-5074Mus musculus (house mouse)Potency29.903310
st 638Mus musculus (house mouse)Potency35.481310
obtusaquinoneMus musculus (house mouse)Potency12.589310
[4-(3-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency35.481320
N-[(2-methoxyphenyl)methyl]-6H-indolo[2,3-b]quinoxaline-2-carboxamideMus musculus (house mouse)Potency19.952610
tyrphostin ag825Mus musculus (house mouse)Potency9.874420
3,5-di-tert-butylchalcone 4'-carboxylic acidMus musculus (house mouse)Potency21.280420
nitrovinMus musculus (house mouse)Potency4.739420
3,5-dihydroxy-4'-methoxystilbeneMus musculus (house mouse)Potency2.480320
eupomatenoid 6Mus musculus (house mouse)Potency11.750420
triphenyltin hydroxideMus musculus (house mouse)Potency2.514620
ethyl linolenateMus musculus (house mouse)Potency35.481310
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazineMus musculus (house mouse)Potency18.867720
(5-ethyl-8-methyl-[1,2,4]triazino[5,6-b]indol-3-yl)hydrazineMus musculus (house mouse)Potency1.584910
5-methoxy-3,6-diphenyl-1,2,4-triazineMus musculus (house mouse)Potency0.223910
3-amino-5-(4-bromophenyl)-4-pyridazinecarbonitrileMus musculus (house mouse)Potency4.466810
N'1-(6-methylpyridazin-3-yl)-4-chlorobenzene-1-carbohydrazideMus musculus (house mouse)Potency15.649820
enclomiphene citrateMus musculus (house mouse)Potency16.271020
lasalocid sodiumMus musculus (house mouse)Potency18.966220
paroxetine maleateMus musculus (house mouse)Potency7.191220
13-cis-retinalMus musculus (house mouse)Potency27.717020
cinalukastMus musculus (house mouse)Potency35.481310
lumefantrineMus musculus (house mouse)Potency19.952610
3-o-methylbuteinMus musculus (house mouse)Potency19.952610
manumycinMus musculus (house mouse)Potency0.852820
bwa 4cMus musculus (house mouse)Potency17.782810
chaetoglobosin AMus musculus (house mouse)Potency8.421820
4-hydroxyderricinMus musculus (house mouse)Potency5.962220
everolimusMus musculus (house mouse)Potency17.740820
su 4312Mus musculus (house mouse)Potency35.481310
2-(1,3-benzoxazol-2-ylamino)-7,7-dimethyl-4-(2-pyridinyl)-1,4,6,8-tetrahydroquinazolin-5-oneMus musculus (house mouse)Potency2.335020
3-[[(3-methoxyanilino)-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency22.740620
4-[[(2,4-difluoroanilino)-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency35.481310
1-(3,4-dimethoxyphenyl)-3-(2-fluoro-5-methylphenyl)ureaMus musculus (house mouse)Potency35.481310
1-(1,3-benzodioxol-5-yl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)ureaMus musculus (house mouse)Potency15.954120
3 beta-o-acetylursolic acidMus musculus (house mouse)Potency0.354810
desmosdumotin cMus musculus (house mouse)Potency28.934220
N-[3-(7-methyl-2-imidazo[1,2-a]pyridinyl)phenyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency1.995310
2-chloro-N-(1-methyl-3-pyrazolyl)acetamideMus musculus (house mouse)Potency4.739420
2-(1-ethyl-4-pyrazolyl)-4-quinolinecarboxylic acidMus musculus (house mouse)Potency4.392820
2-[(3,6-dimethyl-4-oxo-2-thieno[2,3-d]pyrimidinyl)thio]-N-(4-methylphenyl)acetamideMus musculus (house mouse)Potency25.118910
N-(3,4-dichlorophenyl)-2-[4-(1-piperidinylsulfonyl)-1-piperazinyl]acetamideMus musculus (house mouse)Potency26.632020
1-[2-furanyl(oxo)methyl]-N-[4-[(3-methyl-1-piperidinyl)sulfonyl]phenyl]-4-piperidinecarboxamideMus musculus (house mouse)Potency7.943310
norgestimateMus musculus (house mouse)Potency13.699620
3,4,5-trimethoxy-N-[[[oxo-[(1S,2S)-2-phenylcyclopropyl]methyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency11.220210
fluphenazineMus musculus (house mouse)Potency35.481310
homochlorocyclizine monohydrochlorideMus musculus (house mouse)Potency10.000010
emetine hydrochlorideMus musculus (house mouse)Potency1.258920
a 77636Mus musculus (house mouse)Potency31.622810
b 43Mus musculus (house mouse)Potency35.481310
erythro-dihydrosphingosineMus musculus (house mouse)Potency30.300120
sb 222200Mus musculus (house mouse)Potency1.584910
[4-(4-amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methanoneMus musculus (house mouse)Potency6.309610
cycloheximideMus musculus (house mouse)Potency12.850320
suloctidilMus musculus (house mouse)Potency14.125410
1-amino-1,3-dicarboxycyclopentane, cis-(1s,3s)-isomerMus musculus (house mouse)Potency31.622810
sb 218795Mus musculus (house mouse)Potency25.118910
omdm-2 cpdMus musculus (house mouse)Potency35.481310
ym 976Mus musculus (house mouse)Potency28.183810
aminopurvalanol aMus musculus (house mouse)Potency8.912510
bvt.948Mus musculus (house mouse)Potency1.530520
cgk 733Mus musculus (house mouse)Potency3.493520
lactacystinMus musculus (house mouse)Potency0.281810
N-(1,3-benzodioxol-5-ylmethyl)-6-chloro-4-quinazolinamineMus musculus (house mouse)Potency3.719920
2-[[6-[(phenylmethyl)amino]-9-propan-2-yl-2-purinyl]amino]ethanolMus musculus (house mouse)Potency35.481310
2-(1,3-benzothiazol-2-yl)-4-chloro-5-(3-chloroanilino)-3-pyridazinoneMus musculus (house mouse)Potency0.199510
1-(3-amino-7-methoxy-1-pyrazolo[3,4-b]quinolinyl)-2-(4-chlorophenyl)ethanoneMus musculus (house mouse)Potency17.782810
4-methyl-N-[(4-methylphenyl)methyl]-2-furo[3,2-c]quinolinecarboxamideMus musculus (house mouse)Potency17.782810
[4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazin-6-yl]-(1-piperidinyl)methanoneMus musculus (house mouse)Potency11.823020
N-butyl-N-phenyl-8-quinolinesulfonamideMus musculus (house mouse)Potency14.125410
5-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-3-methyl-2-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency1.584910
N-cyclopropyl-2-[[2-(4-ethylphenyl)-5-methyl-4-oxazolyl]methylthio]acetamideMus musculus (house mouse)Potency10.604040
(9-chloro-5,6,7,8-tetrahydroacridin-3-yl)-(4-methyl-1-piperidinyl)methanoneMus musculus (house mouse)Potency12.589310
N-(4-ethylphenyl)-3-(1-pyrrolyl)propanamideMus musculus (house mouse)Potency7.079510
1-cyclopropyl-3-[6-oxo-5-(phenylmethyl)-3-benzo[b][1,4]benzothiazepinyl]ureaMus musculus (house mouse)Potency18.867720
3-[(2S,4S)-2-(4-hydroxybutoxy)-6-[4-morpholinyl(oxo)methyl]-3,4-dihydro-2H-pyran-4-yl]-1-benzopyran-4-oneMus musculus (house mouse)Potency35.481310
(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-(4-oxo-1-benzopyran-3-yl)-3,4-dihydro-2H-pyran-6-carboxylic acid prop-2-enyl esterMus musculus (house mouse)Potency11.220210
Retusin 7-Methyl EtherMus musculus (house mouse)Potency26.632020
cgp 53353Mus musculus (house mouse)Potency25.118910
butaclamol hydrochlorideMus musculus (house mouse)Potency35.481310
estradiol 17-acetateMus musculus (house mouse)Potency15.848910
corosolic acidMus musculus (house mouse)Potency22.740620
N'-(4-fluoro-1,3-benzothiazol-2-yl)-2-phenoxyacetohydrazideMus musculus (house mouse)Potency2.523620
N'-(4,5-dimethyl-1,3-benzothiazol-2-yl)propanehydrazideMus musculus (house mouse)Potency7.943310
4-fluoro-N-(4-fluoro-1,3-benzothiazol-2-yl)-1,3-benzothiazol-2-amineMus musculus (house mouse)Potency9.296120
N-(6-fluoro-1,3-benzothiazol-2-yl)-6,7-dihydro-[1,4]dioxino[2,3-f][1,3]benzothiazol-2-amineMus musculus (house mouse)Potency11.904820
3-(3-methylphenyl)-2-sulfanylidene-1H-benzofuro[3,2-d]pyrimidin-4-oneMus musculus (house mouse)Potency3.642620
N-(1,3-dioxo-5-isoindolyl)butanamideMus musculus (house mouse)Potency15.848910
3-(2-pyridinyl)-6-(2-pyridinylmethylthio)pyridazineMus musculus (house mouse)Potency12.589310
N-(4,7-dimethyl-1,3-benzothiazol-2-yl)-4-(2,5-dioxo-1-pyrrolidinyl)benzamideMus musculus (house mouse)Potency0.199510
N-[5-[(2-methylphenyl)methylthio]-1,3,4-thiadiazol-2-yl]-2-thiophen-2-ylacetamideMus musculus (house mouse)Potency14.125410
3-(ethylthio)-6-(2-furanyl)pyridazineMus musculus (house mouse)Potency12.589310
2-[[6-(2-furanyl)-3-pyridazinyl]thio]-N-(3-methylphenyl)acetamideMus musculus (house mouse)Potency7.943310
3-[(4-chlorophenyl)methylthio]-6-(2-furanyl)pyridazineMus musculus (house mouse)Potency10.000010
5-Chloro-3-pyridinyl 2-furoateMus musculus (house mouse)Potency7.943310
cinnamaldehyde thiosemicarbazoneMus musculus (house mouse)Potency10.974020
5-(1-phenyl-5-tetrazolyl)-2-pyridin-4-yl-4-thiophen-2-ylpyrimidineMus musculus (house mouse)Potency11.220210
5,7-dimethyl-3-[3-(trifluoromethyl)phenyl]azo-1H-pyrazolo[1,5-a]pyrimidin-2-oneMus musculus (house mouse)Potency17.488220
2-[(1R,3S)-3-(7-bromo-2-methyl-1H-indol-3-yl)-2,2-dimethylcyclopropyl]acetonitrileMus musculus (house mouse)Potency18.854120
2-(1-adamantyl)-4-chloro-5-[(4-fluorophenyl)methylamino]-3-pyridazinoneMus musculus (house mouse)Potency1.000010
1-(3-ethylphenyl)-3-(1-naphthalenyl)thioureaMus musculus (house mouse)Potency5.962220
2-(3,5-dimethyl-1H-pyrrol-2-yl)-1,3-benzothiazoleMus musculus (house mouse)Potency3.162310
N-[2-(4-methoxyphenyl)ethyl]-2-quinoxalinecarboxamideMus musculus (house mouse)Potency21.169920
N-[2-(3-methoxyphenyl)-4-[(4-methoxyphenyl)methoxy]-6-quinolinyl]-3-pyridinecarboxamideMus musculus (house mouse)Potency13.534620
sl 327Mus musculus (house mouse)Potency35.481310
((3z)-n-(3-chlorophenyl)-3-((3,5-dimethyl-4-((4-methylpiperazin-1-yl)carbonyl)-1h-pyrrol-2-yl)methylene)-n-methyl-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide)Mus musculus (house mouse)Potency27.717020
[4-[[4-(1-benzothiophen-2-yl)-2-pyrimidinyl]amino]phenyl]-[4-(1-pyrrolidinyl)-1-piperidinyl]methanoneMus musculus (house mouse)Potency28.934220
N-[4-(1-adamantylsulfamoyl)phenyl]-4-bromo-1-methyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency35.481310
1-ethyl-N-[[1-(phenylmethyl)-2-benzimidazolyl]methyl]-5-benzimidazolamineMus musculus (house mouse)Potency35.481310
3-hydroxy-2-methyl-1-(phenylmethyl)-4-pyridinoneMus musculus (house mouse)Potency11.220210
N-[2-methyl-5-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideMus musculus (house mouse)Potency3.981110
5-chloro-N-[4-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2-thiophenesulfonamideMus musculus (house mouse)Potency12.589310
1-[(2-chlorophenyl)methyl]-N-[3-(N-ethyl-3-methylanilino)propyl]-5-oxo-2-pyrrolidinecarboxamideMus musculus (house mouse)Potency1.258910
N-[2-[2-(dibutylamino)ethylamino]-2-oxoethyl]-2-thiophenecarboxamideMus musculus (house mouse)Potency0.707910
3-(2-methoxyethyl)-2,4-dioxo-N-pentyl-1H-quinazoline-7-carboxamideMus musculus (house mouse)Potency1.778310
1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-2-(1-methyl-3-indolyl)ethanoneMus musculus (house mouse)Potency35.481310
LSM-34734Mus musculus (house mouse)Potency11.220210
2-[(1-amino-1-oxopropan-2-yl)thio]-3-butyl-4-oxo-7-quinazolinecarboxylic acid methyl esterMus musculus (house mouse)Potency14.125410
chlorhexidineMus musculus (house mouse)Potency16.866920
sgd 301-76Mus musculus (house mouse)Potency30.300120
nihydrazoneMus musculus (house mouse)Potency8.836820
robenidineMus musculus (house mouse)Potency14.125410
lassbio 294Mus musculus (house mouse)Potency13.357420
cid-2745687Mus musculus (house mouse)Potency13.188920
bn82002Mus musculus (house mouse)Potency35.481310
bms345541Mus musculus (house mouse)Potency7.943310
spc-839Mus musculus (house mouse)Potency5.660820
l 755507Mus musculus (house mouse)Potency24.803320
2-(4'-methylaminophenyl)benzothiazoleMus musculus (house mouse)Potency2.287420
4-[(4-methylphenyl)thio]-2-thieno[2,3-c]pyridinecarboxamideMus musculus (house mouse)Potency0.267230
sb-505124Mus musculus (house mouse)Potency4.428920
nu 7026Mus musculus (house mouse)Potency35.481310
ssr 69071Mus musculus (house mouse)Potency35.481310
ngb 2904Mus musculus (house mouse)Potency2.238710
gw 4064Mus musculus (house mouse)Potency5.623410
nnc 26-9100Mus musculus (house mouse)Potency12.589310
zm 447439Mus musculus (house mouse)Potency20.483920
lissamine rhodamine bMus musculus (house mouse)Potency17.782810
n-(4-((4-(dimethylamino)quinazolin-2-yl)amino)cyclohexyl)-3,4-difluorobenzamide hydrochlorideMus musculus (house mouse)Potency35.481320
gw0742Mus musculus (house mouse)Potency27.717020
a 77636Mus musculus (house mouse)Potency19.952610
pd 198306Mus musculus (house mouse)Potency29.903320
NNC 55-0396 (free base)Mus musculus (house mouse)Potency33.552020
l-161982Mus musculus (house mouse)Potency17.782810
ns 1643Mus musculus (house mouse)Potency28.183810
jte 013Mus musculus (house mouse)Potency15.848910
anomalinMus musculus (house mouse)Potency35.481320
1-(2,4-dichlorophenyl)-6-methyl-N-(1-piperidinyl)-4H-indeno[1,2-c]pyrazole-3-carboxamideMus musculus (house mouse)Potency35.481310
teferinMus musculus (house mouse)Potency35.481310
garcinone eMus musculus (house mouse)Potency27.717020
bavachininMus musculus (house mouse)Potency11.220210
omdm-1 cpdMus musculus (house mouse)Potency19.952610
le 135Mus musculus (house mouse)Potency33.552020
bms 191011Mus musculus (house mouse)Potency30.300120
pyrenophorolMus musculus (house mouse)Potency11.079220
5-methoxy-8,8-dimethyl-2-phenyl-4H,8H-pyrano[2,3-h]chromen-4-oneMus musculus (house mouse)Potency35.481310
ptc 124Mus musculus (house mouse)Potency0.707910
ki 8751Mus musculus (house mouse)Potency17.782810
4-[4-(2-fluorophenyl)phenyl]-N-(4-hydroxyphenyl)butanamideMus musculus (house mouse)Potency3.025820
[5-hydroxy-3-(4-methoxyphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-thiophen-2-ylmethanoneMus musculus (house mouse)Potency31.622810
10-isobutyryloxy-8,9-epoxythymol isobutyrateMus musculus (house mouse)Potency8.912510
gw9508Mus musculus (house mouse)Potency15.848910
protoapigenoneMus musculus (house mouse)Potency2.990420
psb 36Mus musculus (house mouse)Potency0.063110
n,n'-dibenzhydrylethane-1,2-diamine dihydrochlorideMus musculus (house mouse)Potency15.954120
y134 compoundMus musculus (house mouse)Potency35.481310
2-(4-butan-2-ylanilino)-3-pyridinecarbonitrileMus musculus (house mouse)Potency11.220210
N-[(1,3-dioxo-2-phenyl-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl)methyl]-4-methylbenzenesulfonamideMus musculus (house mouse)Potency22.196920
N-(2-methoxyethyl)-2-[[3-[(4-methoxyphenyl)methyl]-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideMus musculus (house mouse)Potency12.062720
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-[(4-methylphenyl)methyl]butanamideMus musculus (house mouse)Potency5.629420
2-(2,1,3-benzothiadiazol-4-ylsulfonylamino)-N-(6-methoxy-1,3-benzothiazol-2-yl)-3-methylbutanamideMus musculus (house mouse)Potency14.501520
R-(-)-actinodaphnineMus musculus (house mouse)Potency10.000020
calcimycinMus musculus (house mouse)Potency1.258910
N-[5-[2-(2,5-dimethoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]-2-methylpentanamideMus musculus (house mouse)Potency19.514720
N-[5-[2-(2-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]-2-methylpentanamideMus musculus (house mouse)Potency22.387210
N-[5-[2-(3-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]-3-methylbutanamideMus musculus (house mouse)Potency26.632020
N-[5-[2-(2-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]heptanamideMus musculus (house mouse)Potency10.000010
N-[4-methyl-5-[2-(4-methylanilino)-4-thiazolyl]-2-thiazolyl]-2-furancarboxamideMus musculus (house mouse)Potency35.481310
3-(4-nitrophenyl)-N-(4-phenylbutyl)-5-(phenylmethyl)-4,6-dihydro-3aH-pyrrolo[3,4-d]isoxazole-6a-carboxamideMus musculus (house mouse)Potency3.548110
2-ethyl-3-methoxy-N-(2-thiophen-2-ylethyl)-6-indazolecarboxamideMus musculus (house mouse)Potency9.505620
N-(1-adamantylmethyl)-2-ethyl-3-methoxy-6-indazolecarboxamideMus musculus (house mouse)Potency14.733420
N-[(2-methoxyphenyl)methyl]-2-methyl-3-prop-2-enoxy-6-indazolecarboxamideMus musculus (house mouse)Potency19.952610
geduninMus musculus (house mouse)Potency35.481310
1-(4-bromophenyl)-3-[[[4-(4-morpholinyl)-3-nitrophenyl]-oxomethyl]amino]thioureaMus musculus (house mouse)Potency12.589320
4-chloro-N-(3,4-dimethoxyphenyl)-2-thieno[3,2-c]quinolinecarboxamideMus musculus (house mouse)Potency22.196920
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideMus musculus (house mouse)Potency0.794310
2-(4-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideMus musculus (house mouse)Potency24.035320
3-(3-chlorophenyl)-1-[(1-methyl-3-indolyl)methyl]-1-[3-(4-morpholinyl)propyl]thioureaMus musculus (house mouse)Potency27.717020
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-(4-ethoxyphenyl)-2,4-dioxobutanamideMus musculus (house mouse)Potency10.000010
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency22.740620
2-[4-(cyclohexylamino)-3-nitrophenyl]-5-methyl-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dioneMus musculus (house mouse)Potency19.952610
2-[4-[2-(4-chlorophenyl)ethylamino]-3-nitrophenyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dioneMus musculus (house mouse)Potency14.125410
1-(4-fluorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaMus musculus (house mouse)Potency4.224020
1-(4-methylphenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaMus musculus (house mouse)Potency19.622220
1-(3-chlorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaMus musculus (house mouse)Potency24.035320
1-[4-[3-methyl-4-(3-methylphenyl)-1-piperazinyl]-3-nitrophenyl]piperidine-2,6-dioneMus musculus (house mouse)Potency27.005020
2-[[(4-methyl-1-piperidinyl)-sulfanylidenemethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency17.488220
4-methoxybenzoic acid [2-(4-bromophenyl)-4-oxo-3-quinazolinyl] esterMus musculus (house mouse)Potency6.045720
2-[(5-bromo-2-thiophenyl)sulfonylamino]-N-cyclopentyl-2-phenylacetamideMus musculus (house mouse)Potency5.623410
2-[[[4-[(2,6-dimethyl-4-morpholinyl)sulfonyl]phenyl]-oxomethyl]amino]-3-thiophenecarboxamideMus musculus (house mouse)Potency25.118910
5-(1,3-benzodioxol-5-ylmethyl)-4-methyl-2-[[1-naphthalenyl(oxo)methyl]amino]-3-thiophenecarboxamideMus musculus (house mouse)Potency35.481310
4-(4-chlorophenyl)sulfonyl-5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-ethylsulfonylthiazoleMus musculus (house mouse)Potency5.623410
3-(benzenesulfonyl)-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]propanamideMus musculus (house mouse)Potency4.532620
[9-(benzenesulfonyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinolin-8-yl]-(4-methylphenyl)methanoneMus musculus (house mouse)Potency0.177810
4-methylbenzoic acid [6-[[[5-[[cyclopropyl(oxo)methyl]amino]-1,3,4-thiadiazol-2-yl]thio]methyl]-4-oxo-3-pyranyl] esterMus musculus (house mouse)Potency19.952610
3-[[5-(4-ethylanilino)-1,3,4-thiadiazol-2-yl]thio]-2-oxolanoneMus musculus (house mouse)Potency35.481310
(2S)-2-[[(3,5-dimethoxyphenyl)-oxomethyl]amino]-3-methylbutanoic acid [2-oxo-2-(4-propan-2-ylanilino)ethyl] esterMus musculus (house mouse)Potency8.912510
chlorhexidine hydrochlorideMus musculus (house mouse)Potency12.589310
[5-Chloranyl-3-[(1E,3E)-3,5-dimethylhepta-1,3-dienyl]-7-methyl-6,8-bis(oxidanylidene)isochromen-7-yl] ethanoateMus musculus (house mouse)Potency10.000010
2-diethylaminoethyl 4-nitrobenzoate hydrochlorideMus musculus (house mouse)Potency35.481310
1-(phenylmethyl)-4-quinolinoneMus musculus (house mouse)Potency3.162310
2',3'-dihydroxy-4',6'-dimethoxychalconeMus musculus (house mouse)Potency13.891420
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneMus musculus (house mouse)Potency6.045720
dehydrocurvularinMus musculus (house mouse)Potency12.967620
4-methoxybenzoic acid 2-(4-hydroxyphenyl)ethyl esterMus musculus (house mouse)Potency9.834420
N-(3,5-dichlorophenyl)-4-[(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)methyl]benzamideMus musculus (house mouse)Potency35.481320
foetidinMus musculus (house mouse)Potency35.481310
4-chloro-N-[1-[[5-(ethylthio)-1,3,4-thiadiazol-2-yl]amino]-3-methyl-1-oxobutan-2-yl]benzamideMus musculus (house mouse)Potency4.466810
2-[[5-(2-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-N-(2-nitrophenyl)acetamideMus musculus (house mouse)Potency4.466810
N-[(1S)-1-(1H-benzimidazol-2-yl)-3-(methylthio)propyl]-2-(4-chlorophenoxy)-2-methylpropanamideMus musculus (house mouse)Potency5.623410
3-(2,4-dimethoxyphenyl)-N-(3-fluoro-4-methylphenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamideMus musculus (house mouse)Potency8.800620
N-Cyclohexyl-5-(2-thienyl)-1,2-oxazole-3-carboxamideMus musculus (house mouse)Potency6.309610
3-nitro-4-(2-oxolanylmethylamino)-N-(2-phenylethyl)benzamideMus musculus (house mouse)Potency17.782810
2-[1-(4-bromophenoxy)butyl]-8,9-dimethoxy-3H-[1,2,4]triazolo[1,5-c]quinazoline-5-thioneMus musculus (house mouse)Potency2.403520
2-[(7-chloro-1,2,3,4-tetrahydroacridin-9-yl)thio]-N-(3-methoxypropyl)acetamideMus musculus (house mouse)Potency14.125410
3-[2-(3,5-dimethoxyphenyl)-5,7-dimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-(phenylmethyl)propanamideMus musculus (house mouse)Potency19.149820
4-chloro-N-[3-(3-methyl-1-piperidinyl)propyl]-2-thieno[3,2-c]quinolinecarboxamideMus musculus (house mouse)Potency22.387210
N-[3-(diethylamino)propyl]-4-[(2-methyl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)hydrazo]-4-oxobutanamideMus musculus (house mouse)Potency20.085020
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideMus musculus (house mouse)Potency21.280420
5-chloro-2-[(3-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideMus musculus (house mouse)Potency17.751820
3-bromo-N-[5-(4-morpholinylsulfonyl)-1,3,4-thiadiazol-2-yl]benzamideMus musculus (house mouse)Potency12.589310
[3-(4-bromophenyl)-1H-pyrazol-5-yl]-[4-(3,4-dimethoxyphenyl)sulfonyl-1-piperazinyl]methanoneMus musculus (house mouse)Potency9.449420
[3-methyl-4-(3-methylphenyl)-1-piperazinyl]-[1-(7,8,9,10-tetrahydro-6H-purino[9,8-a]azepin-4-yl)-4-piperidinyl]methanoneMus musculus (house mouse)Potency0.631010
3,5-dimethoxy-N-[1-[oxo(thiophen-2-yl)methyl]-3,4-dihydro-2H-quinolin-6-yl]benzamideMus musculus (house mouse)Potency7.079510
forapinMus musculus (house mouse)Potency3.915220
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-2-(4-hydroxybutoxy)-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency19.952610
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-4-(4-bromophenyl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency35.481310
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency35.481320
1-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-3-(3-methylphenyl)-1-[2-(4-morpholinyl)ethyl]thioureaMus musculus (house mouse)Potency6.309610
4-[[5-methyl-2-[3-(trifluoromethyl)phenyl]-4-oxazolyl]methyl]morpholineMus musculus (house mouse)Potency2.903120
[4-(3-chlorophenyl)-1-piperazinyl]-[1-[4-(2-pyridinyl)-1-piperazinyl]-4-isoquinolinyl]methanoneMus musculus (house mouse)Potency1.108020
8-methyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-5H-thieno[3,2-c]quinoline-2-carboxamideMus musculus (house mouse)Potency10.000020
N-[[3-(2-chlorophenyl)-1-(4-fluorophenyl)-4-pyrazolyl]methyl]-2-(2-pyridinyl)ethanamineMus musculus (house mouse)Potency7.079510
5-methyl-5-pentyl-2-phenyl-1,2,4-triazolidine-3-thioneMus musculus (house mouse)Potency31.832620
dafadine CMus musculus (house mouse)Potency24.068220
1-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-3-(4-methylphenyl)-1-[2-(4-morpholinyl)ethyl]thioureaMus musculus (house mouse)Potency8.227630
1-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-3-(3-methoxyphenyl)-1-[2-(4-morpholinyl)ethyl]thioureaMus musculus (house mouse)Potency7.079510
dafadine BMus musculus (house mouse)Potency9.149820
(6-methoxy-2-naphthalenyl)-[1-[(2-methyl-5-thiazolyl)methyl]-3-piperidinyl]methanoneMus musculus (house mouse)Potency19.952610
2-(3,5-dimethyl-1-pyrazolyl)-1-[3-[oxo-(3-propan-2-yloxyphenyl)methyl]-1-piperidinyl]ethanoneMus musculus (house mouse)Potency22.387210
1,2-dihydroacenaphthylen-5-yl-[1-[(6-methyl-2-pyridinyl)methyl]-3-piperidinyl]methanoneMus musculus (house mouse)Potency8.285220
1,2-dihydroacenaphthylen-5-yl-[1-(2-pyridinylmethyl)-3-piperidinyl]methanoneMus musculus (house mouse)Potency7.384220
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolMus musculus (house mouse)Potency35.481310
[3-[(3-chlorophenyl)methyl]-1-[(7-methoxy-1,3-benzodioxol-5-yl)methyl]-3-piperidinyl]methanolMus musculus (house mouse)Potency35.481320
[1-[(6-chloro-2H-1-benzopyran-3-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolMus musculus (house mouse)Potency35.481310
[1-[(1,2-dimethyl-3-indolyl)methyl]-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolMus musculus (house mouse)Potency7.996020
1-cyclohexyl-2-(1H-imidazol-2-ylmethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indoleMus musculus (house mouse)Potency7.943310
2-(2,4-dimethoxyphenyl)-5-methyl-4-[[4-(4-quinazolinyl)-1-piperazinyl]methyl]oxazoleMus musculus (house mouse)Potency25.118910
1-(5-isoquinolinylmethyl)-4-[(3-methoxyphenyl)methyl]-4-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency35.481320
1-[[3-(4-fluorophenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]-4-[(1-methyl-2-imidazolyl)methyl]piperazineMus musculus (house mouse)Potency28.934220
(3aS,5S,9aS)-2-[(2-methylphenyl)methyl]-5-(1-methyl-3-phenyl-4-pyrazolyl)-3a,4,5,7,8,9-hexahydro-3H-pyrrolo[3,4-h]pyrrolizin-1-oneMus musculus (house mouse)Potency22.387220
1-ethyl-4-[[methyl-[[3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]amino]methyl]-2-pyrrolidinoneMus musculus (house mouse)Potency17.488220
1-cyclohexyl-2-[(1-ethyl-2-imidazolyl)methyl]-1,3,4,9-tetrahydropyrido[3,4-b]indoleMus musculus (house mouse)Potency24.035320
[1-[[1-(5-chloro-2-pyridinyl)-2-pyrrolyl]methyl]-3-piperidinyl]-(2,4-dimethoxyphenyl)methanoneMus musculus (house mouse)Potency25.118910
4-[[[2-(1-azepanyl)ethyl-(2-furanylmethyl)amino]-sulfanylidenemethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency28.183810
2-[[6-(4-morpholinyl)-4-oxo-3-(2-phenylethyl)-2-quinazolinyl]thio]-N-(2-oxolanylmethyl)acetamideMus musculus (house mouse)Potency9.106320
N-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]-4-phenyl-1-piperazinecarbothioamideMus musculus (house mouse)Potency14.976320
2-[(2-chloro-4-nitroanilino)methyl]-6-methoxyphenolMus musculus (house mouse)Potency23.350720
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(3-ethylphenyl)-3-hydroxy-5-nitro-4-triazolimineMus musculus (house mouse)Potency25.118910
N'-[[3-(4-methylphenyl)sulfonyl-2-oxazolidinyl]methyl]-N-[2-(4-sulfamoylphenyl)ethyl]oxamideMus musculus (house mouse)Potency35.481320
6-(2-furanyl)-3-(2-pyridinylmethylthio)-[1,2,4]triazolo[4,3-b]pyridazineMus musculus (house mouse)Potency12.589310
N-[2-[4-(4-methoxyphenyl)-1-piperazinyl]ethyl]-6-sulfanylidene-5H-benzimidazolo[1,2-c]quinazoline-3-carboxamideMus musculus (house mouse)Potency4.928820
N-[5-[[2-(2-furanylmethylamino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-1,3-benzodioxole-5-carboxamideMus musculus (house mouse)Potency11.294720
2-[[6-(4-ethylphenyl)-3-pyridazinyl]thio]-N-(2-oxolanylmethyl)acetamideMus musculus (house mouse)Potency35.481310
(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxylic acid prop-2-enyl esterMus musculus (house mouse)Potency35.481310
(2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid tert-butyl esterMus musculus (house mouse)Potency7.233420
(2S)-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]-3-phenylpropanoic acid (phenylmethyl) esterMus musculus (house mouse)Potency12.924420
(2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid (phenylmethyl) esterMus musculus (house mouse)Potency7.843520
(2S)-4-methyl-2-[[[5-(methylcarbamoyl)-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl esterMus musculus (house mouse)Potency4.220920
(2S)-4-methyl-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl esterMus musculus (house mouse)Potency5.120920
(2S)-2-[[[5-[[methyl-(phenylmethyl)amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterMus musculus (house mouse)Potency21.280420
violaceol IIMus musculus (house mouse)Potency26.632020
(2S,4S)-4-(4-bromophenyl)-2-(4-hydroxybutoxy)-N-phenyl-3,4-dihydro-2H-pyran-6-carboxamideMus musculus (house mouse)Potency21.280420
(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(phenylmethyl)-3,4-dihydro-2H-pyran-6-carboxamideMus musculus (house mouse)Potency3.548110
a-83-01Mus musculus (house mouse)Potency10.000010
gw 583340Mus musculus (house mouse)Potency27.717020
2-[(5,6-dimethyl-4-thieno[2,3-d]pyrimidinyl)amino]-1-(4-nitrophenyl)ethanolMus musculus (house mouse)Potency4.496520
3-acetamido-N-[4-(4-methylsulfonylphenyl)-2-thiazolyl]-3-phenyl-N-prop-2-enylpropanamideMus musculus (house mouse)Potency35.481310
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideMus musculus (house mouse)Potency10.066420
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideMus musculus (house mouse)Potency23.350720
peniprequinoloneMus musculus (house mouse)Potency0.251210
(8R)-3-[3-[[2-(4-chlorophenoxy)-1-oxoethyl]amino]phenyl]-7-(1-oxo-3,3-diphenylpropyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-8-carboxamideMus musculus (house mouse)Potency12.589310
(3aR,4S,9aR,9bS)-N-(4-chlorophenyl)-2-(4-fluorophenyl)-1,3-dioxo-3a,4,9a,9b-tetrahydropyrrolo[1,2]pyrrolo[3,5-b]pyridazine-4-carboxamideMus musculus (house mouse)Potency10.000010
N-[(2S)-1-hydroxypropan-2-yl]-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency17.782810
N-(2-hydroxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency6.581220
phenylmercuric acetateMus musculus (house mouse)Potency0.842210
phentin acetateMus musculus (house mouse)Potency2.219720
thimerosalMus musculus (house mouse)Potency0.876520
N-[3-[2-(4-chloroanilino)-4-thiazolyl]phenyl]-3-(trifluoromethyl)benzamideMus musculus (house mouse)Potency17.782810
2-amino-N-[3-methoxy-5-[oxo-[3-(trifluoromethyl)anilino]methyl]phenyl]-5-oxazolecarboxamideMus musculus (house mouse)Potency29.903320
3-(4-bromophenyl)-N-[5-[[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)anilino]-oxomethyl]-2-methylphenyl]-1H-pyrazole-5-carboxamideMus musculus (house mouse)Potency35.481320
8-{1-[4-(dimethylamino)phenyl]-3-(pyrrolidin-1-yl)propyl}-5,7-dimethoxy-4-pentyl-2H-chromen-2-oneMus musculus (house mouse)Potency17.782810
3-(2-hydroxy-4,6-dimethoxyphenyl)-3-(4-methoxyphenyl)-1-(3-methyl-1-piperidinyl)-1-propanoneMus musculus (house mouse)Potency18.110740
8-[3-(diethylamino)-1-(4-methoxyphenyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneMus musculus (house mouse)Potency15.649820
3-(1,3-benzodioxol-5-yl)-3-(2-hydroxy-4,6-dimethoxyphenyl)-1-(3-methyl-1-piperidinyl)-1-propanoneMus musculus (house mouse)Potency14.838430
8-[1-[4-(dimethylamino)phenyl]-3-(3-methyl-1-piperidinyl)propyl]-5,7-dimethoxy-4-phenyl-1-benzopyran-2-oneMus musculus (house mouse)Potency31.622810
(3R,3aS,7R,7aS)-7-methyl-3-(2-naphthalenyl)-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneMus musculus (house mouse)Potency35.481310
(3R)-3-(2-fluoro-5-methylphenyl)-7-phenyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneMus musculus (house mouse)Potency14.987220
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency18.169620
2-[[[4-[(3-methylanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid (phenylmethyl) esterMus musculus (house mouse)Potency24.035320
N4-(4-methoxyphenyl)-N5-[(1S)-1-phenylethyl]-1H-imidazole-4,5-dicarboxamideMus musculus (house mouse)Potency7.611020
(2S)-2-[[[4-[(3-methylanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-3-phenylpropanoic acid (phenylmethyl) esterMus musculus (house mouse)Potency6.119420
2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterMus musculus (house mouse)Potency8.528020
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterMus musculus (house mouse)Potency22.196920
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esterMus musculus (house mouse)Potency22.196920
N4-(4-methoxyphenyl)-N5-[(1R)-1-phenylethyl]-1H-imidazole-4,5-dicarboxamideMus musculus (house mouse)Potency7.126420
ro 10-5824Mus musculus (house mouse)Potency3.162310
1-[1-(4-butan-2-ylphenyl)ethyl]-3-[(4-fluorophenyl)methyl]thioureaMus musculus (house mouse)Potency3.915220
N-butyl-4-(phenylmethyl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency25.665120
1-cyclohexyl-3-[1-(3,4-dimethoxyphenyl)ethyl]thioureaMus musculus (house mouse)Potency15.586420
N-(3-nitrophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxamideMus musculus (house mouse)Potency0.177810
2,3,4,10-tetrahydro-7,10-dimethyl-2,4-dioxobenzo(g)pteridineMus musculus (house mouse)Potency10.000010
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methoxyphenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency9.106320
6-(3,5-dimethyl-4-isoxazolyl)-N-[(2-ethoxyphenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency37.646020
6-(3,5-dimethyl-4-isoxazolyl)-N-[1-(2-furanyl)ethyl]-4-quinazolinamineMus musculus (house mouse)Potency21.280420
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methyl-2-thiophenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency0.640320
3-[(3-chlorophenyl)methyl]-5-ethoxy-1,6-dimethylpyrido[2,3-d]pyrimidine-2,4-dioneMus musculus (house mouse)Potency0.707910
N-(2-methylpropyl)-4-(phenylmethyl)-1-piperidinecarbothioamideMus musculus (house mouse)Potency20.811420
4-(phenylmethyl)-N-prop-2-enyl-1-piperidinecarbothioamideMus musculus (house mouse)Potency25.665120
1-[(4-fluorophenyl)methyl]-3-[1-(4-propan-2-ylphenyl)propyl]thioureaMus musculus (house mouse)Potency3.399820
1-(3-chlorophenyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)thioureaMus musculus (house mouse)Potency30.300120
1-(7-methyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl)-N-(4-methylphenyl)-2-pyrrolidinecarboxamideMus musculus (house mouse)Potency19.952610
N-(3-acetylphenyl)-5-(3-methyl-5-isoxazolyl)-2-thiophenesulfonamideMus musculus (house mouse)Potency22.387210
N-(4-propan-2-ylphenyl)-1-[(1,3,3-trimethyl-2-oxo-5-indolyl)sulfonyl]-4-piperidinecarboxamideMus musculus (house mouse)Potency15.848910
4-[2-[(6-chloro-4-quinazolinyl)amino]ethyl]phenolMus musculus (house mouse)Potency9.449420
sri 62320Mus musculus (house mouse)Potency11.220210
thiopental sodiumMus musculus (house mouse)Potency10.000010
cytomelMus musculus (house mouse)Potency12.589310
acid blue 129Mus musculus (house mouse)Potency10.000010
cortisol succinate, sodium saltMus musculus (house mouse)Potency25.118910
2-[(6-chloro-3-pyridinyl)sulfonylamino]-N-[(4-methylphenyl)methyl]benzamideMus musculus (house mouse)Potency13.534620
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency28.934220
4-(4-chloro-3-nitrophenyl)-N-[2-(5,6-dichloro-1-propyl-2-benzimidazolyl)ethyl]-2-thiazolamineMus musculus (house mouse)Potency19.952610
(2S)-2-[[oxo-[5-[oxo-(4-phenyl-1-piperazinyl)methyl]-1H-imidazol-4-yl]methyl]amino]-3-phenylpropanoic acid tert-butyl esterMus musculus (house mouse)Potency35.481310
2-[[[4-[[(diphenylmethyl)amino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterMus musculus (house mouse)Potency15.714220
1-azepanyl-[5-[(4-chloro-3,5-dimethylphenoxy)methyl]-3-isoxazolyl]methanoneMus musculus (house mouse)Potency2.511910
4-(1-((5-((2,6-dimethylphenoxy)methyl)-3-isoxazolyl)carbonyl)-4-piperidinyl)pyridineMus musculus (house mouse)Potency11.220210
10-deacetyltaxolMus musculus (house mouse)Potency12.924420
[5-[(3,4-difluorophenoxy)methyl]-3-isoxazolyl]-(3-propoxy-1-piperidinyl)methanoneMus musculus (house mouse)Potency4.466810
N-[3-(3-chlorophenyl)phenyl]-1-(3-isoxazolylmethyl)-4-piperidinecarboxamideMus musculus (house mouse)Potency35.481320
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency1.748820
(2R)-3-[[(2S)-1-cyclohexyl-3-(methylamino)propan-2-yl]amino]-2-[2-[3-(trifluoromethyl)phenyl]ethylamino]-1-propanolMus musculus (house mouse)Potency35.481310
cyclopropyl-[5-[[4-[[4-(2-methoxyphenyl)-1-piperazinyl]-oxomethyl]-1-piperidinyl]sulfonyl]-2-methyl-2,3-dihydroindol-1-yl]methanoneMus musculus (house mouse)Potency12.589310
N-[2-[1-[(4-methoxy-3-methylphenyl)methyl]-4-piperidinyl]-3-pyrazolyl]-4-phenylbutanamideMus musculus (house mouse)Potency35.481310
N,3-dimethyl-5-propyl-N-(2-thiazolylmethyl)-2-benzofurancarboxamideMus musculus (house mouse)Potency22.387210
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-methyl-5-thiadiazolecarboxamideMus musculus (house mouse)Potency10.585430
[2-(2-methoxyethyl)-1-piperidinyl]-[5-[[4-(1,2,4-triazol-1-yl)phenoxy]methyl]-3-isoxazolyl]methanoneMus musculus (house mouse)Potency11.258830
N-methyl-N-(3-pyridinylmethyl)-5-(5,6,7,8-tetrahydronaphthalen-2-yloxymethyl)-3-isoxazolecarboxamideMus musculus (house mouse)Potency13.448620
2-[[[4-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterMus musculus (house mouse)Potency17.782810
(5R)-5-tert-butyl-1-[(3S)-3-[(4-methylphenyl)thio]-3-phenylpropyl]-2-azepanoneMus musculus (house mouse)Potency10.000010
N-[3-(3-chlorophenyl)phenyl]-1-(3-oxolanylmethyl)-4-piperidinecarboxamideMus musculus (house mouse)Potency11.220210
dafadine OMus musculus (house mouse)Potency22.387210
[5-[(4-methoxy-1-naphthalenyl)oxymethyl]-3-isoxazolyl]-(4-methoxy-1-piperidinyl)methanoneMus musculus (house mouse)Potency0.631010
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency2.509920
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-5-(methoxymethyl)-2-furancarboxamideMus musculus (house mouse)Potency10.610120
2-[1-[(4-chlorophenyl)-oxomethyl]-5-methoxy-2-methyl-3-indolyl]-N-[(2-hydroxy-5-nitrophenyl)methyl]acetamideMus musculus (house mouse)Potency16.803720
1-(3-methoxyphenyl)-3-(4-phenylbutyl)ureaMus musculus (house mouse)Potency2.238710
2-[3-(4-morpholinyl)propylamino]-9-xanthenoneMus musculus (house mouse)Potency6.309610
3-[[1-(dimethylsulfamoyl)-4-piperidinyl]oxy]-N-[(3-methyl-5-isoxazolyl)methyl]benzamideMus musculus (house mouse)Potency0.891310
2-(2,6-dimethylphenoxy)-N-[2-(1-piperidinyl)phenyl]acetamideMus musculus (house mouse)Potency17.782810
(3S)-4-oxo-3-phenyl-3-propan-2-yldiazetidine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency10.000010
4-(4-acetyloxyphenyl)benzoic acid [2-[[2-(2-chloroanilino)-2-oxoethyl]-methylamino]-2-oxoethyl] esterMus musculus (house mouse)Potency35.481310
(3S)-3-cyclopentyl-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency11.220210
N-[5-[[2-(4-acetamidoanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-3-methoxybenzamideMus musculus (house mouse)Potency11.904820
4-tert-butyl-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideMus musculus (house mouse)Potency12.431220
N-[5-[[2-(4-acetamidoanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-5-bromo-2-furancarboxamideMus musculus (house mouse)Potency7.191220
4-ethoxy-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideMus musculus (house mouse)Potency6.230320
deslorelinMus musculus (house mouse)Potency16.803720
1-butyl-4-hydroxy-N-(3-methyl-2-pyridinyl)-2-oxo-3-quinolinecarboxamideMus musculus (house mouse)Potency16.271020
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamideMus musculus (house mouse)Potency35.481310
mobiflexMus musculus (house mouse)Potency31.622810
tenuazonic acidMus musculus (house mouse)Potency25.118910
N-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-1-prop-2-enyl-3-quinolinecarboxamideMus musculus (house mouse)Potency26.632020
1-butyl-N-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-3-quinolinecarboxamideMus musculus (house mouse)Potency35.481310
N'-[(2-chlorophenyl)-oxomethyl]-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarbohydrazideMus musculus (house mouse)Potency21.712320
N-(2-aminophenyl)-1-butyl-4-hydroxy-2-oxo-3-quinolinecarboxamideMus musculus (house mouse)Potency6.351420
LSM-28526Mus musculus (house mouse)Potency0.316210
1-ethyl-4-hydroxy-2-oxo-N'-(1-oxoheptyl)-3-quinolinecarbohydrazideMus musculus (house mouse)Potency23.350720
N-(2-aminophenyl)-4-hydroxy-2-oxo-1-pentyl-3-quinolinecarboxamideMus musculus (house mouse)Potency3.162310
N3-phenyl-4-hydroxy-1,5,6-trimethyl-2,2-dioxo-1,2-dihydro-26-thieno[2,3-c][1,2]thiazine-3-carboxamideMus musculus (house mouse)Potency35.481310
N-(1H-benzimidazol-2-yl)-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarboxamideMus musculus (house mouse)Potency10.066420
4-hydroxy-N-(2-methyl-4-oxo-3-quinazolinyl)-1-(2-methylpropyl)-2-oxo-5,6,7,8-tetrahydroquinoline-3-carboxamideMus musculus (house mouse)Potency24.803320
4-hydroxy-2-oxo-1-pentyl-N-(2-pyridinylmethyl)-3-quinolinecarboxamideMus musculus (house mouse)Potency11.397420
N-[2-(4-chlorophenyl)ethyl]-4-hydroxy-2-oxo-1-propyl-3-quinolinecarboxamideMus musculus (house mouse)Potency24.803320
stf 083010Mus musculus (house mouse)Potency14.125410
clozapineMus musculus (house mouse)Potency39.810710
3-cinnamoyl-4-hydroxy-6-methyl-2h-pyran-2-oneMus musculus (house mouse)Potency35.481310
kf38789Mus musculus (house mouse)Potency16.193610
salinazidMus musculus (house mouse)Potency2.990420
N-(1-azabicyclo[2.2.2]octan-3-yl)-6-chloro-7-nitro-1H-benzimidazole-4-carboxamideMus musculus (house mouse)Potency11.220210
1-[amino-[(6-methoxy-4-methyl-2-quinazolinyl)amino]methylidene]-3-phenylureaMus musculus (house mouse)Potency25.118910
tju 103Mus musculus (house mouse)Potency35.481320
2-[(2-oxo-3-indolyl)amino]-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideMus musculus (house mouse)Potency35.481310
5-amino-2-phenyl-3H-triazolo[4,5-d]pyrimidin-7-oneMus musculus (house mouse)Potency12.589310
2-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylthio]-6-phenyl-1H-pyrimidin-4-oneMus musculus (house mouse)Potency0.501210
N-(2,3-dimethylphenyl)-5-(2-fluorophenyl)-6H-1,3,4-thiadiazin-2-amineMus musculus (house mouse)Potency19.321820
2-[(2-pyridinylthio)methyl]-1H-benzofuro[3,2-d]pyrimidin-4-oneMus musculus (house mouse)Potency16.803720
1-hydroxyphenazineMus musculus (house mouse)Potency4.280020
N-(1,3-benzodioxol-5-yl)-2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]acetamideMus musculus (house mouse)Potency4.795720
N-cyclohexyl-3-methyl-N-[(4-oxo-1H-quinazolin-2-yl)methyl]benzamideMus musculus (house mouse)Potency2.511910
N-(1,3-benzodioxol-5-ylmethyl)-3-methoxy-N-[(4-oxo-1H-quinazolin-2-yl)methyl]benzamideMus musculus (house mouse)Potency31.622810
2-carboxyarabinitol 1-phosphateMus musculus (house mouse)Potency5.561020
6,8-dibromo-2-[[[4-(difluoromethoxy)phenyl]methyl-methylamino]methyl]-1H-quinazolin-4-oneMus musculus (house mouse)Potency7.875820
salicylaldehyde thiosemicarbazoneMus musculus (house mouse)Potency4.928820
1-(3-methoxyphenyl)-2-[4-oxo-6-(trifluoromethyl)-1H-pyrimidin-2-yl]guanidineMus musculus (house mouse)Potency22.387210
2-(4-methoxyphenyl)-1H-quinazolin-4-oneMus musculus (house mouse)Potency22.387210
heliomycinMus musculus (house mouse)Potency15.514020
N-[4-[2-[3-(dimethylsulfamoyl)anilino]-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamideMus musculus (house mouse)Potency35.481310
N-[4-[2-(2-methoxyethylamino)-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamideMus musculus (house mouse)Potency35.481310
pyridoxal 4-methoxybenzoyl hydrazoneMus musculus (house mouse)Potency10.000010
N-butyl-5-(3,4-dimethylphenyl)-6H-1,3,4-thiadiazin-2-amineMus musculus (house mouse)Potency9.834420
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-[4-(4-morpholinyl)phenyl]acetamideMus musculus (house mouse)Potency8.285220
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-oneMus musculus (house mouse)Potency3.915220
2-(4-fluoroanilino)-6-methyl-5-(3-methylbutyl)-1H-pyrimidin-4-oneMus musculus (house mouse)Potency21.280420
2-[(dimethylamino)methyl]-4-spiro[1,6-dihydrobenzo[h]quinazoline-5,1'-cyclohexane]oneMus musculus (house mouse)Potency3.761920
2-(diethylaminomethyl)-4-spiro[1,6-dihydrobenzo[h]quinazoline-5,1'-cyclohexane]oneMus musculus (house mouse)Potency11.220220
4-methyl-3-phenyl-1,2-dihydropyrazolo[3,4-b]pyridin-6-oneMus musculus (house mouse)Potency3.548110
N-(4-acetylphenyl)-2-[(4-oxo-1H-quinazolin-2-yl)thio]butanamideMus musculus (house mouse)Potency8.912510
2-[(2-pyridinylthio)methyl]-1H-quinazolin-4-oneMus musculus (house mouse)Potency12.589310
5,5-diethyl-2-(2-hydroxyethylamino)-1,6-dihydrobenzo[h]quinazolin-4-oneMus musculus (house mouse)Potency15.848910
6,7-dimethoxy-2-[[methyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]methyl]-1H-quinazolin-4-oneMus musculus (house mouse)Potency2.566520
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-[2-(methylthio)phenyl]acetamideMus musculus (house mouse)Potency0.509120
5,5-diethyl-2-hydrazinyl-1,6-dihydrobenzo[h]quinazolin-4-oneMus musculus (house mouse)Potency12.924420
3-(3-ethoxypropyl)-1-[(4-oxo-1H-quinazolin-2-yl)methyl]-1-(phenylmethyl)thioureaMus musculus (house mouse)Potency23.350720
N-[4-[2-(2-oxolanylmethylamino)-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamideMus musculus (house mouse)Potency0.005010
N-(3,4-dimethoxyphenyl)-2-[(4-oxo-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)thio]acetamideMus musculus (house mouse)Potency3.981110
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-(3-fluorophenyl)acetamideMus musculus (house mouse)Potency28.934220
N-[2-(4-chlorophenyl)ethyl]-2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]acetamideMus musculus (house mouse)Potency18.819140
5-(2,5-difluorophenyl)-N-(2-oxolanylmethyl)-6H-1,3,4-thiadiazin-2-amineMus musculus (house mouse)Potency6.309610
N-[(cyclohexylamino)-oxomethyl]-2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]acetamideMus musculus (house mouse)Potency0.562320
2-(4-chloroanilino)-5-[(2,3-dichlorophenyl)methyl]-4-thiazoloneMus musculus (house mouse)Potency35.481320
7-[[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]methyl]-5-thiazolo[3,2-a]pyrimidinoneMus musculus (house mouse)Potency6.119420
fenobamMus musculus (house mouse)Potency19.952610