Proteins > M17 leucyl aminopeptidase
Page last updated: 2024-08-07 18:10:16

M17 leucyl aminopeptidase

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (47)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
aa 861Plasmodium falciparum 3D7IC5053.450010
benzbromaronePlasmodium falciparum 3D7IC5081.890010
bufexamacPlasmodium falciparum 3D7IC501.000010
lonidaminePlasmodium falciparum 3D7IC507.370010
angiotensin ii, des-asp(1)-des-arg(2)-ile(5)-Plasmodium falciparum 3D7IC501.530010
1-(4-methylphenyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanonePlasmodium falciparum 3D7IC5050.490010
2-[(3-oxo-5-phenyl-1,2-dihydropyrazol-4-yl)-(3-thiophenyl)methyl]propanedinitrilePlasmodium falciparum 3D7IC5036.660010
5-[(3-ethoxycarbonyl-4-thiophen-2-yl-2-thiophenyl)amino]-5-oxopentanoic acidPlasmodium falciparum 3D7IC5020.260010
N-[5-[[2-(4-methylanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-2-(4-morpholinyl)acetamidePlasmodium falciparum 3D7IC509.150010
1-(3,4-dihydroxyphenyl)-2-[[5-(2-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanonePlasmodium falciparum 3D7IC5022.840010
1,3,5-trimethylcyclohexane-1,3,5-tricarboxylic acidPlasmodium falciparum 3D7IC5058.690010
5-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazole-3-thionePlasmodium falciparum 3D7IC5039.470010
3,5,5-trimethyl-2-sulfanylidene-1,6-dihydrobenzo[h]quinazolin-4-onePlasmodium falciparum 3D7IC501.900010
1-(4-ethoxyphenyl)-3-(6-quinoxalinyl)ureaPlasmodium falciparum 3D7IC505.450010
4-[(4-chlorophenyl)thio]-5-methyl-2-phenyl-1H-pyrazol-3-onePlasmodium falciparum 3D7IC5037.420010
1-(4-methoxyphenyl)-3-(2-methyl-1,3-benzoxazol-5-yl)ureaPlasmodium falciparum 3D7IC5014.810010
4-[4-[[(3,4-dimethylphenyl)-oxomethyl]amino]phenoxy]phthalic acidPlasmodium falciparum 3D7IC5013.160010
2-[[[3-[2-(4-methylphenyl)sulfonylethylthio]phenyl]-oxomethyl]amino]benzoic acidPlasmodium falciparum 3D7IC509.590010
2-[[2-[(3,7-dimethyl-2-quinolinyl)thio]-1-oxoethyl]amino]-4,5-dimethoxybenzoic acidPlasmodium falciparum 3D7IC501.930010
4,5-dimethoxy-2-[[1-oxo-2-[(3,5,8-trimethyl-2-quinolinyl)thio]ethyl]amino]benzoic acidPlasmodium falciparum 3D7IC501.000010
1-(1,3-benzodioxol-5-yl)-3-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]ureaPlasmodium falciparum 3D7IC5013.350010
2-(1,3-benzothiazol-2-ylthio)-N-(4-methylphenyl)sulfonylacetamidePlasmodium falciparum 3D7IC507.770010
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamidePlasmodium falciparum 3D7IC5091.170010
7-[[[5-(2,4-dimethylanilino)-1,3,4-thiadiazol-2-yl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinonePlasmodium falciparum 3D7IC506.490010
4-[[2-[[5-(3-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-1-oxoethyl]amino]benzoic acidPlasmodium falciparum 3D7IC5024.270010
2-oxo-1H-pyridine-3-carboxylic acid [2-(2,5-dimethyl-1-propyl-3-pyrrolyl)-2-oxoethyl] esterPlasmodium falciparum 3D7IC5015.330010
5-chloro-2-mercaptobenzothiazolePlasmodium falciparum 3D7IC5014.780010
N'-[3-bicyclo[2.2.1]heptanyl(oxo)methyl]-3-chloro-1-benzothiophene-2-carbohydrazidePlasmodium falciparum 3D7IC5068.100010
2-[(2,3-dihydro-1,4-benzodioxin-6-ylamino)-oxomethyl]-1-cyclohexanecarboxylic acidPlasmodium falciparum 3D7IC5032.880010
6-amino-4-(2-methylpropyl)-3-phenyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrilePlasmodium falciparum 3D7IC5033.740010
6-[(3,4-difluoroanilino)-oxomethyl]-1-cyclohex-3-enecarboxylic acidPlasmodium falciparum 3D7IC5020.370010
6-[[[5-(ethylthio)-1,3,4-thiadiazol-2-yl]amino]-oxomethyl]-1-cyclohex-3-enecarboxylic acidPlasmodium falciparum 3D7IC5019.890010
2-[[(3-ethoxycarbonyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-oxomethyl]-3-methyl-3-bicyclo[2.2.1]hept-5-enecarboxylic acidPlasmodium falciparum 3D7IC508.100010
7-ethyl-7-methyl-2-sulfanylidene-6,9-dihydro-1H-pyrano[2,3]thieno[2,4-b]pyrimidin-4-onePlasmodium falciparum 3D7IC5029.310010
3-nitro-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamidePlasmodium falciparum 3D7IC5049.060010
N-(2,3-dihydro-1H-inden-5-yl)-2-[(4-hydroxy-6-oxo-1H-pyrimidin-2-yl)thio]acetamidePlasmodium falciparum 3D7IC502.010010
6-amino-4-methyl-3-(4-methylphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrilePlasmodium falciparum 3D7IC5016.330010
4-[[3-[anilino(oxo)methyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidPlasmodium falciparum 3D7IC5047.000010
N-[2-(3-methyl-1-oxobutyl)-3-oxo-1,2,4-thiadiazol-5-yl]benzamidePlasmodium falciparum 3D7IC5043.940010
ellagic acidPlasmodium falciparum 3D7IC50138.080010
(2S)-2-(3-oxo-1H-isoindol-2-yl)-3-phenylpropanoic acidPlasmodium falciparum 3D7IC506.470010
quinaldine redPlasmodium falciparum 3D7IC50110.220010
N-[4-(diethylamino)-2-methylphenyl]-2-[(2-nitro-3-thiophenyl)thio]acetamidePlasmodium falciparum 3D7IC501.900010
3-[[5-(4-ethylanilino)-1,3,4-thiadiazol-2-yl]thio]-2-oxolanonePlasmodium falciparum 3D7IC502.640010
cefamandole nafatePlasmodium falciparum 3D7IC5012.080010
4-[[2-[(6-methyl-4-oxo-1H-pyrimidin-2-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterPlasmodium falciparum 3D7IC5011.800010
indole-3-aldehyde oximePlasmodium falciparum 3D7IC5013.150010