Proteins > beta-2 adrenergic receptor
Page last updated: 2024-08-07 22:52:18

beta-2 adrenergic receptor

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (117)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
racepinephrineHomo sapiens (human)Potency1.299510
pyrithioneHomo sapiens (human)Potency0.730810
disulfiramHomo sapiens (human)Potency0.651310
berotekHomo sapiens (human)Potency5.804810
isoetharineHomo sapiens (human)Potency2.592910
isoproterenolHomo sapiens (human)Potency1.299510
itraconazoleHomo sapiens (human)Potency15.848910
metaproterenolHomo sapiens (human)Potency18.356410
nifedipineHomo sapiens (human)Potency28.183810
terbutalineHomo sapiens (human)Potency10.322510
thiramHomo sapiens (human)Potency0.631010
isoproterenol hydrochlorideHomo sapiens (human)Potency2.423830
4-[(1S)-1-hydroxy-2-(propan-2-ylamino)ethyl]benzene-1,2-diolHomo sapiens (human)Potency2.059610
racepinephrine hydrochlorideHomo sapiens (human)Potency10.045230
cyproheptadine hydrochloride (anhydrous)Homo sapiens (human)Potency29.092910
nitroxolineHomo sapiens (human)Potency2.818410
isoetharine mesylateHomo sapiens (human)Potency1.742830
thymolphthaleinHomo sapiens (human)Potency28.183810
glutamic acidHomo sapiens (human)Potency20.596210
nicorandilHomo sapiens (human)Potency25.118910
salmeterol xinafoateHomo sapiens (human)Potency7.857330
dipivefrin hydrochlorideHomo sapiens (human)Potency0.766030
ubenimexHomo sapiens (human)Potency12.995310
fangchinolineHomo sapiens (human)Potency11.401220
4-(2-thiazolylazo)resorcinolHomo sapiens (human)Potency5.623410
prilocaine hydrochlorideHomo sapiens (human)Potency3.162310
3-chloro-6-hydrazino-pyridazineHomo sapiens (human)Potency19.952610
gallopamil hydrochlorideHomo sapiens (human)Potency25.118910
L-isoprenalineHomo sapiens (human)Potency1.054710
dihydroergocristine monomesylateHomo sapiens (human)Potency9.436020
likviritonHomo sapiens (human)Potency6.513110
dibenzylidene acetoneHomo sapiens (human)Potency6.513110
opc-2009Homo sapiens (human)Potency0.068630
2-(3,5-dimethyl-1-pyrazolyl)-N,6-dimethyl-4-pyrimidinamineHomo sapiens (human)Potency25.118910
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideHomo sapiens (human)Potency5.623410
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanolHomo sapiens (human)Potency28.183810
2-[(2,5-dimethyl-3-phenyl-7-pyrazolo[1,5-a]pyrimidinyl)thio]acetonitrileHomo sapiens (human)Potency3.548110
dienestrolHomo sapiens (human)Potency1.458110
3,5,5-trimethyl-2-sulfanylidene-1,6-dihydrobenzo[h]quinazolin-4-oneHomo sapiens (human)Potency3.548110
phenylthiazolylthioureaHomo sapiens (human)Potency10.000010
nsc185058Homo sapiens (human)Potency24.989610
3-(4-methylphenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneHomo sapiens (human)Potency20.596210
N-(4-methoxyphenyl)-3,4-dihydro-1H-isoquinoline-2-carbothioamideHomo sapiens (human)Potency29.092910
N-[[(5-chloro-2-pyridinyl)amino]-sulfanylidenemethyl]-3-methylbutanamideHomo sapiens (human)Potency29.092910
2-phenyl-1H-quinazoline-4-thioneHomo sapiens (human)Potency32.132820
8-methyl-2-(3-methylbutyl)-1,2,4-triazaspiro[4.5]decane-3-thioneHomo sapiens (human)Potency35.481310
1-(1-pyrrolidinyl)-2-(8-quinolinylthio)ethanoneHomo sapiens (human)Potency6.513110
3-pyridinecarboxylic acid [2-(2-furanyl)-4-oxo-1-benzopyran-3-yl] esterHomo sapiens (human)Potency34.062020
levocetirizineHomo sapiens (human)Potency10.000010
4-butyl-3-(3-methyl-2-thiophenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency31.622810
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-quinolinecarboxamideHomo sapiens (human)Potency6.309610
4-butyl-3-(phenylmethyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency18.356410
1-(4-bromo-2-chlorophenyl)-3-(3-methyl-2-pyridinyl)thioureaHomo sapiens (human)Potency35.481310
N-[3-[[diethylamino(sulfanylidene)methyl]thio]-1-oxopropyl]carbamic acid (4-tert-butylphenyl) esterHomo sapiens (human)Potency29.092910
1-(4-methoxyphenyl)-3-(6-methyl-2-pyridinyl)thioureaHomo sapiens (human)Potency11.220210
1-anilino-3-ethylthioureaHomo sapiens (human)Potency31.622810
3-oxo-2-[(5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)thio]butanoic acid ethyl esterHomo sapiens (human)Potency31.622810
N-[2-furanyl-(8-hydroxy-7-quinolinyl)methyl]-2-methylpropanamideHomo sapiens (human)Potency15.526320
N-[2,2,2-trichloro-1-[[sulfanylidene-(2,4,6-trimethylanilino)methyl]amino]ethyl]benzamideHomo sapiens (human)Potency29.092910
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(4-methoxyphenyl)methyl]acetamideHomo sapiens (human)Potency32.287120
3-methyl-4-oxo-1,5,6,7-tetrahydroindole-2-carboxylic acid (4-methylcyclohexyl) esterHomo sapiens (human)Potency6.513110
6-methyl-2-(phenylethynyl)pyridineHomo sapiens (human)Potency18.356410
p-201-1Homo sapiens (human)Potency35.481310
1,3-dimethyl-8-[2-(1-pyrrolidinyl)ethylthio]-6-sulfanylidene-7H-purin-2-oneHomo sapiens (human)Potency15.848910
sch 23390Homo sapiens (human)Potency29.092910
1-[1-chloro-2-[(2-nitrophenyl)thio]-4-phenyl-2,3,3a,4,5,9b-hexahydro-1H-cyclopenta[c]quinolin-8-yl]ethanoneHomo sapiens (human)Potency16.360110
acetic acid [1-[(3-nitrophenyl)-(1-oxopentylamino)methyl]-2-naphthalenyl] esterHomo sapiens (human)Potency32.642710
7'-hydroxy-4'-(4-methoxyphenyl)-4,4,5'-trimethyl-2-spiro[1,3-diazinane-6,2'-3,4-dihydro-2H-1-benzopyran]thioneHomo sapiens (human)Potency23.109310
1-[2-(diethylamino)ethyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-3-(2-oxolanylmethyl)thioureaHomo sapiens (human)Potency8.912510
5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinolHomo sapiens (human)Potency6.959320
7-[(4-methyl-1-piperazinyl)methyl]-5-(phenylmethoxymethyl)-8-quinolinolHomo sapiens (human)Potency2.888110
2-[3-[(4-methylphenyl)methyl]-7-oxo-6-triazolo[4,5-d]pyrimidinyl]-N-(2-oxolanylmethyl)acetamideHomo sapiens (human)Potency25.118910
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinolHomo sapiens (human)Potency31.622810
2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-5-methyl-4-(4-methylphenyl)-1,2,4-triazol-3-oneHomo sapiens (human)Potency0.580510
2-[(5-anilino-1,3,4-thiadiazol-2-yl)thio]-N-[3-(1-piperidinylsulfonyl)phenyl]acetamideHomo sapiens (human)Potency25.929010
4-(5-methyl-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)benzoic acid 8-quinolinyl esterHomo sapiens (human)Potency29.092910
1-(2,4-difluorophenyl)-3-[4-(2-pyridinyl)-2-thiazolyl]ureaHomo sapiens (human)Potency2.238710
2-(4-benzoylphenoxy)-N-[4-(propan-2-ylsulfamoyl)phenyl]propanamideHomo sapiens (human)Potency32.642710
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazoleHomo sapiens (human)Potency34.062020
quercetin 3-o-methyl etherHomo sapiens (human)Potency26.395630
fucoxanthinHomo sapiens (human)Potency28.183810
wogoninHomo sapiens (human)Potency20.596210
phenylephrine hydrochlorideHomo sapiens (human)Potency3.439720
latanoprostHomo sapiens (human)Potency35.481310
fenoterolHomo sapiens (human)Potency7.544830
nab-365Homo sapiens (human)Potency5.840620
epinephrine bitartrateHomo sapiens (human)Potency7.793430
17-cyclopropylmethyl-6,7-didehydro-4,5-epoxy-5'-guanidinyl-3,14-dihydroxyindolo(2',3'-6,7)morphinanHomo sapiens (human)Potency3.662610
N-[1-(5,6-dicyano-3-methyl-2-pyrazinyl)ethyl]-N-phenylacetamideHomo sapiens (human)Potency29.092910
protoapigenoneHomo sapiens (human)Potency6.513110
sk&f 77434Homo sapiens (human)Potency16.360110
malyngamide AHomo sapiens (human)Potency3.264310
4'-o-beta-d-glucosyl-5-o-methylvisamminolHomo sapiens (human)Potency0.651310
N-[3-(diethylamino)propyl]-4-[(2-methyl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)hydrazo]-4-oxobutanamideHomo sapiens (human)Potency11.220210
(3S)-3-(4-methoxyphenyl)-4-oxo-3-propan-2-yldiazetidine-1,2-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency31.622810
(3S)-3-cyclopentyl-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency35.481310
N-[(5-chloro-8-hydroxy-7-quinolinyl)-cyclopropylmethyl]acetamideHomo sapiens (human)Potency23.109310
N-[(5-fluoro-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamideHomo sapiens (human)Potency29.092910
N-[(5-bromo-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamideHomo sapiens (human)Potency32.642710
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-oneHomo sapiens (human)Potency5.623410
2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]-N-[2-(methylthio)phenyl]acetamideHomo sapiens (human)Potency17.782810

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
clotrimazoleHomo sapiens (human)EC504.690010
isoproterenol hydrochlorideHomo sapiens (human)EC500.825010
racepinephrine hydrochlorideHomo sapiens (human)EC502.650010
isoetharine mesylateHomo sapiens (human)EC503.840010
salmeterol xinafoateHomo sapiens (human)EC500.004510
dipivefrin hydrochlorideHomo sapiens (human)EC507.130010
harmalanHomo sapiens (human)EC502.770010
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineHomo sapiens (human)EC508.610010
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-[(3-methyl-2-imidazo[4,5-b]pyridinyl)thio]acetamideHomo sapiens (human)EC502.440010
N-(4-{[2-(pyridin-3-yl)piperidin-1-yl]sulfonyl}phenyl)acetamideHomo sapiens (human)EC500.100730
2-[[2-(3,5-dimethyl-1-pyrazolyl)-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-4-yl]thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)EC508.850010
2-[[[5-(3-chlorophenyl)-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-1H-benzimidazoleHomo sapiens (human)EC509.095020
ethyl 4-{N-[(4-chlorophenyl)sulfonyl]-N-methylglycyl}piperazine-1-carboxylateHomo sapiens (human)EC501.468220
2-(4-methylphenoxy)-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]acetamideHomo sapiens (human)EC500.036120
5-nitro-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-furancarboxamideHomo sapiens (human)EC500.394120
1-[(4-chlorophenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineHomo sapiens (human)EC502.615020
N,4-dimethyl-N-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}benzenesulfonamideHomo sapiens (human)EC500.057830
LSM-28187Homo sapiens (human)EC500.091910
fenoterolHomo sapiens (human)EC500.110010
epinephrine bitartrateHomo sapiens (human)EC501.380010
5-(4-chlorophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineHomo sapiens (human)EC508.380010
4-[3-(2-furanyl)-4-(3-nitrophenyl)-6-oxo-2,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoic acid ethyl esterHomo sapiens (human)EC500.571010
5-(4-bromophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineHomo sapiens (human)EC508.440010