Page last updated: 2024-08-07 21:05:10

Poly [ADP-ribose] polymerase 2

A poly [ADP-ribose] polymerase 2 that is encoded in the genome of mouse. [OMA:O88554, PRO:DNx]

Synonyms

PARP-2;
mPARP-2;
EC 2.4.2.30;
ADP-ribosyltransferase diphtheria toxin-like 2;
ARTD2;
DNA ADP-ribosyltransferase PARP2;
2.4.2.-;
NAD(+) ADP-ribosyltransferase 2;
ADPRT-2;
Poly[ADP-ribose] synthase 2;
pADPRT-2;
P

Research

Bioassay Publications (4)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Compounds (11)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
niacinamideMus musculus (house mouse)IC50129.524512
1,5-dihydroxyisoquinolineMus musculus (house mouse)IC500.299012
3-aminobenzamideMus musculus (house mouse)IC5018.894724
4-amino-1,8-naphthalimideMus musculus (house mouse)IC500.027012
phenanthridoneMus musculus (house mouse)IC500.208012
5-aminoisoquinolinoneMus musculus (house mouse)IC501.219035
pj-34Mus musculus (house mouse)IC500.040512
5-iodo-6-amino-1,2-benzopyroneMus musculus (house mouse)IC5013.147012
gpi 6150Mus musculus (house mouse)IC500.134512
3,4-dihydro-5-(4-(1-piperidinyl)butoxy)-1(2h)-isoquinolinoneMus musculus (house mouse)IC501.055012
4-hydroxyquinazolineMus musculus (house mouse)IC5015.796012