Page last updated: 2024-08-07 15:08:16

Chain A, Beta-lactamase

[no definition available]

Synonyms

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (3169)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
dinitrochlorobenzeneEscherichia coli K-12Potency5.623410
aminolevulinic acidEscherichia coli K-12Potency22.387210
9-xylosyladenineEscherichia coli K-12Potency89.125110
arabinoseEscherichia coli K-12Potency5.011910
catecholEscherichia coli K-12Potency5.623410
coumarinEscherichia coli K-12Potency112.202010
guaiacolEscherichia coli K-12Potency5.623410
methylmalonic acidEscherichia coli K-12Potency5.623410
pyrrolidonecarboxylic acidEscherichia coli K-12Potency39.810710
malic acidEscherichia coli K-12Potency79.432810
deoxycytidineEscherichia coli K-12Potency19.952610
histamineEscherichia coli K-12Potency3,162.280010
indol-3-yl pyruvic acidEscherichia coli K-12Potency10.000010
thioctic acidEscherichia coli K-12Potency32.983820
picolinic acidEscherichia coli K-12Potency50.118710
sarcosineEscherichia coli K-12Potency100.000010
sorboseEscherichia coli K-12Potency8.912510
ibotenic acidEscherichia coli K-12Potency5.011910
vanilmandelic acidEscherichia coli K-12Potency10.000010
mandelic acidEscherichia coli K-12Potency39.810710
2-(6-methoxy-2-naphthalenyl)propanoic acidEscherichia coli K-12Potency11.079220
1,10-phenanthrolineEscherichia coli K-12Potency3.548110
pk 11195Escherichia coli K-12Potency28.183810
1-(2-trifluoromethylphenyl)imidazoleEscherichia coli K-12Potency11.220210
pd 173074Escherichia coli K-12Potency19.952610
2-aminofluoreneEscherichia coli K-12Potency100.000010
pyrithioneEscherichia coli K-12Potency5.011910
ro 5-4864Escherichia coli K-12Potency28.183810
p-chloromercuribenzoic acidEscherichia coli K-12Potency0.631010
5-(n,n-hexamethylene)amilorideEscherichia coli K-12Potency112.202010
etofyllineEscherichia coli K-12Potency17.782810
acetazolamideEscherichia coli K-12Potency17.782810
acetohexamideEscherichia coli K-12Potency11.220210
n-acetylphenylalanineEscherichia coli K-12Potency1.412510
tyrphostin a23Escherichia coli K-12Potency79.432810
albendazoleEscherichia coli K-12Potency89.125110
methylglucosideEscherichia coli K-12Potency3.162310
alpha-tocopherol acetateEscherichia coli K-12Potency5.623410
althiazideEscherichia coli K-12Potency5.623410
am 251Escherichia coli K-12Potency22.387210
p-aminohippuric acidEscherichia coli K-12Potency5.623410
amoxapineEscherichia coli K-12Potency39.810710
6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diolEscherichia coli K-12Potency15.848910
astemizoleEscherichia coli K-12Potency28.183810
aurintricarboxylic acidEscherichia coli K-12Potency8.912520
benfluorexEscherichia coli K-12Potency0.794310
benzamideEscherichia coli K-12Potency0.631010
benzbromaroneEscherichia coli K-12Potency112.202010
bicalutamideEscherichia coli K-12Potency89.125110
bithionolEscherichia coli K-12Potency25.118910
brimonidineEscherichia coli K-12Potency15.848910
bromoprideEscherichia coli K-12Potency7.943310
bromperidolEscherichia coli K-12Potency7.943310
butacaineEscherichia coli K-12Potency48.534220
butambenEscherichia coli K-12Potency79.432810
carbamazepineEscherichia coli K-12Potency6.309610
cyclobutane-1,1-dicarboxylic acidEscherichia coli K-12Potency4.466810
carcinineEscherichia coli K-12Potency28.183810
carprofenEscherichia coli K-12Potency15.848910
chlorothiazideEscherichia coli K-12Potency15.848910
ciprofibrateEscherichia coli K-12Potency5.011910
clofibrateEscherichia coli K-12Potency5.623410
clofibric acidEscherichia coli K-12Potency0.631010
dacarbazineEscherichia coli K-12Potency6.309610
r 59022Escherichia coli K-12Potency35.481310
diazoxideEscherichia coli K-12Potency17.782810
dichlorodiphenyl dichloroethyleneEscherichia coli K-12Potency5.011910
dipyridamoleEscherichia coli K-12Potency15.848910
disulfiramEscherichia coli K-12Potency65.811420
droperidolEscherichia coli K-12Potency100.000010
dyphyllineEscherichia coli K-12Potency100.000010
ebselenEscherichia coli K-12Potency57.122020
epirizoleEscherichia coli K-12Potency25.118910
erythrosineEscherichia coli K-12Potency37.618820
epiestriolEscherichia coli K-12Potency44.668410
ethoxzolamideEscherichia coli K-12Potency63.095710
famprofazoneEscherichia coli K-12Potency100.000010
fenbendazoleEscherichia coli K-12Potency5.011910
fipexideEscherichia coli K-12Potency22.387210
flumequineEscherichia coli K-12Potency3.548110
flutamideEscherichia coli K-12Potency0.631010
fusaric acidEscherichia coli K-12Potency10.000010
glipizideEscherichia coli K-12Potency14.125410
harmalineEscherichia coli K-12Potency0.316210
hexestrolEscherichia coli K-12Potency3.981110
hexylresorcinolEscherichia coli K-12Potency3.162310
beta-thujaplicinEscherichia coli K-12Potency3.548110
hexamethylene bisacetamideEscherichia coli K-12Potency100.000010
lidocaineEscherichia coli K-12Potency0.354810
idebenoneEscherichia coli K-12Potency25.118910
ifosfamideEscherichia coli K-12Potency11.220210
amrinoneEscherichia coli K-12Potency44.668410
indole-3-carbinolEscherichia coli K-12Potency70.794610
iodoquinolEscherichia coli K-12Potency3.981110
ioxaglateEscherichia coli K-12Potency0.631010
isocarboxazidEscherichia coli K-12Potency112.202010
itraconazoleEscherichia coli K-12Potency6.309610
ketoprofenEscherichia coli K-12Potency3.548110
lansoprazoleEscherichia coli K-12Potency89.125110
lidoflazineEscherichia coli K-12Potency11.519020
loratadineEscherichia coli K-12Potency18.867710
meclofenamate sodium anhydrousEscherichia coli K-12Potency31.622810
mefexamideEscherichia coli K-12Potency89.125110
vitamin k 3Escherichia coli K-12Potency5.623410
milrinoneEscherichia coli K-12Potency0.631010
1,1'-azobis(N,N-dimethylformamide)Escherichia coli K-12Potency89.125110
nefazodoneEscherichia coli K-12Potency14.125410
niclosamideEscherichia coli K-12Potency5.623410
nifedipineEscherichia coli K-12Potency0.354810
nimesulideEscherichia coli K-12Potency15.848910
nimodipineEscherichia coli K-12Potency16.206520
6,7-dimethoxy-3-(4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl)-3H-isobenzofuran-1-oneEscherichia coli K-12Potency6.309610
ns 1619Escherichia coli K-12Potency1.412510
nu2058Escherichia coli K-12Potency39.810710
oxamniquineEscherichia coli K-12Potency89.125110
oxatomideEscherichia coli K-12Potency35.481310
oxethazaineEscherichia coli K-12Potency19.952610
oxibendazoleEscherichia coli K-12Potency112.202010
oxyphenbutazoneEscherichia coli K-12Potency44.668410
palmidrolEscherichia coli K-12Potency8.912510
dexpanthenolEscherichia coli K-12Potency5.623410
perphenazineEscherichia coli K-12Potency22.387210
phenazineEscherichia coli K-12Potency11.220210
phenolphthaleinEscherichia coli K-12Potency15.848910
pinacidilEscherichia coli K-12Potency0.354810
piracetamEscherichia coli K-12Potency1.584910
probucolEscherichia coli K-12Potency2.511910
prochlorperazineEscherichia coli K-12Potency35.481310
proglumideEscherichia coli K-12Potency7.943310
proxyphyllineEscherichia coli K-12Potency100.000010
quetiapineEscherichia coli K-12Potency10.682620
ritanserinEscherichia coli K-12Potency22.387210
roxarsoneEscherichia coli K-12Potency1.258910
sb 202190Escherichia coli K-12Potency7.079510
sobuzoxaneEscherichia coli K-12Potency28.183810
spiperoneEscherichia coli K-12Potency17.782810
aldactazideEscherichia coli K-12Potency35.481310
sulfaguanidineEscherichia coli K-12Potency6.309610
sulfamerazineEscherichia coli K-12Potency35.481310
sulfameterEscherichia coli K-12Potency0.354810
sulfamethizoleEscherichia coli K-12Potency39.810710
sulfamethoxypyridazineEscherichia coli K-12Potency94.562610
sulfapyridineEscherichia coli K-12Potency35.481310
sulmazoleEscherichia coli K-12Potency10.000010
sumatriptanEscherichia coli K-12Potency44.668410
suprofenEscherichia coli K-12Potency6.309610
suxibuzoneEscherichia coli K-12Potency5.623410
tegafurEscherichia coli K-12Potency1.584910
terazosinEscherichia coli K-12Potency35.481310
thiramEscherichia coli K-12Potency59.621820
trichlormethiazideEscherichia coli K-12Potency15.848910
trigonellineEscherichia coli K-12Potency5.623410
ics 205-930Escherichia coli K-12Potency0.631010
tyrphostin a9Escherichia coli K-12Potency7.079510
vesamicolEscherichia coli K-12Potency89.125110
ici 204,219Escherichia coli K-12Potency0.251210
hydrocortisone acetateEscherichia coli K-12Potency84.218010
reserpineEscherichia coli K-12Potency17.782810
D-ribofuranoseEscherichia coli K-12Potency5.623410
isoproterenol hydrochlorideEscherichia coli K-12Potency28.183810
neostigmine methylsulfateEscherichia coli K-12Potency56.234110
carbacholEscherichia coli K-12Potency5.011910
etiocholanoloneEscherichia coli K-12Potency50.118710
dichlororibofuranosylbenzimidazoleEscherichia coli K-12Potency8.912510
amifampridineEscherichia coli K-12Potency0.707910
benzyltrimethylammonium chlorideEscherichia coli K-12Potency6.309610
9,10-dimethyl-1,2-benzanthraceneEscherichia coli K-12Potency2.818410
benzoxazoloneEscherichia coli K-12Potency0.562310
acetylcholine chlorideEscherichia coli K-12Potency1.584910
diphemanil methylsulfateEscherichia coli K-12Potency7.079510
colchicineEscherichia coli K-12Potency5.011910
thiamine hydrochlorideEscherichia coli K-12Potency7.943310
chlorpromazine hydrochlorideEscherichia coli K-12Potency28.183810
ampicillinEscherichia coli K-12Potency0.562320
medroxyprogesterone acetateEscherichia coli K-12Potency26.632010
azovioletEscherichia coli K-12Potency3.548110
triamcinolone acetonideEscherichia coli K-12Potency89.125110
gibberellic acidEscherichia coli K-12Potency0.707910
linaloolEscherichia coli K-12Potency22.387210
skatoleEscherichia coli K-12Potency6.309610
syrosingopineEscherichia coli K-12Potency22.387210
phensuximideEscherichia coli K-12Potency5.623410
salicylanilideEscherichia coli K-12Potency2.511910
isosorbide dinitrateEscherichia coli K-12Potency5.623410
xanthenesEscherichia coli K-12Potency6.309610
methyleugenolEscherichia coli K-12Potency8.154820
mecopropEscherichia coli K-12Potency89.125110
synephrineEscherichia coli K-12Potency17.782810
propylparabenEscherichia coli K-12Potency1.412510
2-methyl-4-chlorophenoxyacetic acidEscherichia coli K-12Potency35.481310
dicloranEscherichia coli K-12Potency1.778310
pyridostigmine bromideEscherichia coli K-12Potency3.981110
n-isopropyl-n-phenyl-4-phenylenediamineEscherichia coli K-12Potency100.000010
benzonatateEscherichia coli K-12Potency8.912520
vanillic acidEscherichia coli K-12Potency25.118910
benzethonium chlorideEscherichia coli K-12Potency28.183810
piperidolate hydrochlorideEscherichia coli K-12Potency4.466810
peucedaninEscherichia coli K-12Potency1.995310
phenazopyridine hydrochlorideEscherichia coli K-12Potency3.162310
tetrracaine hydrochlorideEscherichia coli K-12Potency89.125110
carzenideEscherichia coli K-12Potency89.125110
pregnenoloneEscherichia coli K-12Potency0.316210
20-alpha-dihydroprogesteroneEscherichia coli K-12Potency39.810710
2-chloroadenosineEscherichia coli K-12Potency70.794610
dulcinEscherichia coli K-12Potency3.981110
phenanthridineEscherichia coli K-12Potency100.000010
norchlorcyclizineEscherichia coli K-12Potency5.623410
benzoylarginine-2-naphthylamideEscherichia coli K-12Potency8.912510
monocrotalineEscherichia coli K-12Potency2.511910
azacitidineEscherichia coli K-12Potency39.810710
cyproterone acetateEscherichia coli K-12Potency25.118910
2-aminopurineEscherichia coli K-12Potency10.000010
glycocholic acidEscherichia coli K-12Potency2.818410
isocorydineEscherichia coli K-12Potency50.118710
glaucineEscherichia coli K-12Potency50.118710
rheinEscherichia coli K-12Potency79.432810
cepharanthineEscherichia coli K-12Potency25.118910
9-(2,3-dihydroxy-3-methylbutoxy)-4-methoxy-7h-furo(3,2-g)(1)benzopyran-7-oneEscherichia coli K-12Potency0.562310
dipicolinic acidEscherichia coli K-12Potency2.818410
podophyllotoxinEscherichia coli K-12Potency6.309610
medroxyprogesteroneEscherichia coli K-12Potency112.202010
tetrahydrozoline hydrochlorideEscherichia coli K-12Potency4.466810
1,2-naphthoquinoneEscherichia coli K-12Potency28.183810
coumarin-3-carboxylic acidEscherichia coli K-12Potency56.234110
diperodonEscherichia coli K-12Potency70.794610
benzyl sulfideEscherichia coli K-12Potency0.316210
levocarnitineEscherichia coli K-12Potency1.412510
maleimideEscherichia coli K-12Potency5.623410
propoxycaine hydrochlorideEscherichia coli K-12Potency5.623410
betaine hydrochlorideEscherichia coli K-12Potency6.309610
megestrol acetateEscherichia coli K-12Potency19.952610
2-hydroxyacetanilideEscherichia coli K-12Potency44.668410
2-(methylthio)benzothiazoleEscherichia coli K-12Potency0.631010
bendazoleEscherichia coli K-12Potency39.810710
dicarbethoxydihydrocollidineEscherichia coli K-12Potency112.202010
Berberine chloride (TN)Escherichia coli K-12Potency11.220210
erythromycinEscherichia coli K-12Potency20.903020
2'-deoxy-5'-adenosine monophosphateEscherichia coli K-12Potency0.562310
2-phenylbenzimidazoleEscherichia coli K-12Potency39.810710
2,5-diphenyloxazoleEscherichia coli K-12Potency11.220210
phosmetEscherichia coli K-12Potency42.209020
levonorgestrelEscherichia coli K-12Potency56.234110
malononitrile dimerEscherichia coli K-12Potency35.481310
2-hydroxybenzothiazoleEscherichia coli K-12Potency0.316210
metformin hydrochlorideEscherichia coli K-12Potency112.202010
2-acetylpyridineEscherichia coli K-12Potency0.631010
n-acetylmelphalanEscherichia coli K-12Potency44.668410
2-amino-4-phenylphenolEscherichia coli K-12Potency0.316210
flurandrenoloneEscherichia coli K-12Potency63.095710
bisphenol a-glycidyl methacrylateEscherichia coli K-12Potency34.893620
diethylcarbamazine citrateEscherichia coli K-12Potency15.714220
azaperoneEscherichia coli K-12Potency2.818410
pyrazonEscherichia coli K-12Potency2.818410
laudanosineEscherichia coli K-12Potency2.859920
(4-tert-Butyl-phenoxy)-acetic acidEscherichia coli K-12Potency10.000010
azacyclonolEscherichia coli K-12Potency39.810710
PropioveratroneEscherichia coli K-12Potency0.707910
amiloride hydrochloride, anhydrousEscherichia coli K-12Potency39.810710
pimozideEscherichia coli K-12Potency70.794610
azaribineEscherichia coli K-12Potency89.125110
hydrocortisone hemisuccinateEscherichia coli K-12Potency0.631010
n-acetylimidazoleEscherichia coli K-12Potency22.387210
aviprinEscherichia coli K-12Potency44.668410
mebeverine hydrochlorideEscherichia coli K-12Potency63.095710
midodrine hydrochlorideEscherichia coli K-12Potency5.011910
clidinium bromideEscherichia coli K-12Potency0.631010
meclofenoxate hydrochlorideEscherichia coli K-12Potency2.511910
todralazineEscherichia coli K-12Potency7.943310
piperacetazineEscherichia coli K-12Potency39.810710
nitroxolineEscherichia coli K-12Potency39.810710
pathilonEscherichia coli K-12Potency0.631010
3,3-dimethylglutarateEscherichia coli K-12Potency0.562310
1,6-bismaleimidohexaneEscherichia coli K-12Potency50.118710
5,5-diethylhydantoinEscherichia coli K-12Potency63.095710
beclomethasone dipropionateEscherichia coli K-12Potency5.623420
alverine citrateEscherichia coli K-12Potency79.432810
pinacidilEscherichia coli K-12Potency6.309610
5,7-dimethyl-(1,2,4)triazolo(1,5-a)pyrimidineEscherichia coli K-12Potency0.631010
monoethylglycinexylidideEscherichia coli K-12Potency2.818410
alphadolone acetateEscherichia coli K-12Potency39.810710
quinoxidineEscherichia coli K-12Potency31.622810
hydroxyzine pamoateEscherichia coli K-12Potency41.429920
1-(3-chlorophenyl)piperazine dihydrochlorideEscherichia coli K-12Potency1.778310
pyrazophosEscherichia coli K-12Potency39.810710
benserazide hydrochlorideEscherichia coli K-12Potency39.810710
iocetamic acidEscherichia coli K-12Potency2.818410
eedqEscherichia coli K-12Potency100.000010
gidifenEscherichia coli K-12Potency7.079510
ornidazoleEscherichia coli K-12Potency15.848910
metergolineEscherichia coli K-12Potency25.118910
n-(cyclohexylthio)phthalimideEscherichia coli K-12Potency79.432810
1-(trimethylsilyl)-1h-imidazoleEscherichia coli K-12Potency10.000010
cetyldimethylethylammonium bromideEscherichia coli K-12Potency35.481310
ursodeoxycholic acidEscherichia coli K-12Potency28.183810
rafoxanideEscherichia coli K-12Potency2.893420
benzonidazoleEscherichia coli K-12Potency5.623410
N-(3-methyl-1,1-dioxo-1,4-thiazinan-4-yl)-1-(5-nitro-2-furanyl)methanimineEscherichia coli K-12Potency7.079510
u 25030Escherichia coli K-12Potency0.707910
hoe-40045Escherichia coli K-12Potency2.511910
2-tert-butylbenzimidazoleEscherichia coli K-12Potency0.631010
lenperoneEscherichia coli K-12Potency1.412510
clobetasol propionateEscherichia coli K-12Potency89.125110
amoxicillinEscherichia coli K-12Potency35.481310
2,5-dimethyl-3-furancarboxanilideEscherichia coli K-12Potency20.697820
moricizine hydrochlorideEscherichia coli K-12Potency25.118910
moricizineEscherichia coli K-12Potency25.118910
paclitaxelEscherichia coli K-12Potency12.589320
wr 171,699Escherichia coli K-12Potency5.623410
5-MethoxyisatinEscherichia coli K-12Potency44.668410
methyldopaEscherichia coli K-12Potency53.808320
lonidamineEscherichia coli K-12Potency0.562310
iem 611Escherichia coli K-12Potency35.481310
phenicaberanEscherichia coli K-12Potency2.238710
6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acidEscherichia coli K-12Potency7.943310
nicardipine hydrochlorideEscherichia coli K-12Potency28.183810
closantelEscherichia coli K-12Potency1.778310
propiconazoleEscherichia coli K-12Potency28.183810
N-[4-(dimethylamino)phenyl]-3,4,5-trimethoxybenzamideEscherichia coli K-12Potency19.952610
butoconazole nitrateEscherichia coli K-12Potency3.548110
cerm-1978Escherichia coli K-12Potency21.421520
cefotetanEscherichia coli K-12Potency12.431220
lovastatinEscherichia coli K-12Potency25.285510
chaetochrominEscherichia coli K-12Potency61.193620
2-[[1-(2-amino-4-thiazolyl)-2-[[(2S,3S)-2-methyl-4-oxo-1-sulfo-3-azetidinyl]amino]-2-oxoethylidene]amino]oxy-2-methylpropanoic acidEscherichia coli K-12Potency4.496520
simvastatinEscherichia coli K-12Potency28.934220
bambuterol hydrochlorideEscherichia coli K-12Potency4.466810
bambuterolEscherichia coli K-12Potency5.011910
nefazodone hydrochlorideEscherichia coli K-12Potency12.589310
mifepristoneEscherichia coli K-12Potency25.118910
amlodipine besylateEscherichia coli K-12Potency47.475920
daunorubicin hydrochlorideEscherichia coli K-12Potency31.622810
diltiazem hydrochlorideEscherichia coli K-12Potency25.118910
verapamil hydrochlorideEscherichia coli K-12Potency39.810710
doxazosin mesylateEscherichia coli K-12Potency28.183810
amantadine hydrochlorideEscherichia coli K-12Potency5.011910
mevastatinEscherichia coli K-12Potency19.702010
neocuproineEscherichia coli K-12Potency100.000010
desipramine hydrochlorideEscherichia coli K-12Potency14.125410
mefloquine hydrochlorideEscherichia coli K-12Potency1.584910
4-nitrobenzylthioinosineEscherichia coli K-12Potency3.981110
benzydamine hydrochlorideEscherichia coli K-12Potency22.387210
ethefilEscherichia coli K-12Potency100.000010
prenylamine lactateEscherichia coli K-12Potency5.623410
isbufyllineEscherichia coli K-12Potency2.818410
rutecarpineEscherichia coli K-12Potency6.309610
pifexoleEscherichia coli K-12Potency100.000010
trihexyphenidyl hydrochlorideEscherichia coli K-12Potency35.481310
thioridazine hydrochlorideEscherichia coli K-12Potency39.810710
diphenylpyraline hydrochlorideEscherichia coli K-12Potency89.125110
procainamide hydrochlorideEscherichia coli K-12Potency14.125410
siquilEscherichia coli K-12Potency35.481310
diphenidol hydrochlorideEscherichia coli K-12Potency112.202010
ay-20694Escherichia coli K-12Potency63.095710
2-methoxyestradiolEscherichia coli K-12Potency50.118710
amizylEscherichia coli K-12Potency39.810710
toxoflavinEscherichia coli K-12Potency22.387210
salicylhydroxamic acidEscherichia coli K-12Potency28.183810
dimidium bromideEscherichia coli K-12Potency8.912510
flindersineEscherichia coli K-12Potency112.202010
clomipramine hydrochlorideEscherichia coli K-12Potency22.387210
sertralineEscherichia coli K-12Potency28.183810
nilvermEscherichia coli K-12Potency0.631010
butinolineEscherichia coli K-12Potency63.095710
2-Methyl-4-quinolinolEscherichia coli K-12Potency79.432810
4-oxo-1,4-dihydro-3-pyridinecarboxylic acidEscherichia coli K-12Potency100.000010
norcyclizineEscherichia coli K-12Potency31.622810
n-acetyltryptamineEscherichia coli K-12Potency0.223910
tyrosine methyl esterEscherichia coli K-12Potency3.162310
2,2,8-trimethyl-4h-1-3-dioxino(4,5-c)pyridin-5-ylmethanolEscherichia coli K-12Potency100.000010
2-amino-4-tert-butylphenolEscherichia coli K-12Potency17.782810
oxprenolol hydrochlorideEscherichia coli K-12Potency5.623410
clobetasone butyrateEscherichia coli K-12Potency17.782810
loxapine succinateEscherichia coli K-12Potency25.118910
guanfacine hydrochlorideEscherichia coli K-12Potency25.118910
diflorasone diacetateEscherichia coli K-12Potency25.118910
talampicillin hydrochlorideEscherichia coli K-12Potency31.659820
maprotiline hydrochlorideEscherichia coli K-12Potency106.101010
dipivefrin hydrochlorideEscherichia coli K-12Potency2.818410
4-fluorobenzamideEscherichia coli K-12Potency0.707910
acetylisoniazidEscherichia coli K-12Potency0.707910
hydroxyzine dihydrochlorideEscherichia coli K-12Potency28.183810
fomocainEscherichia coli K-12Potency7.943310
chlormidazoleEscherichia coli K-12Potency17.782810
thioxoloneEscherichia coli K-12Potency112.202010
hesperetinEscherichia coli K-12Potency5.623410
nobiletinEscherichia coli K-12Potency21.203520
9-methoxyellipticineEscherichia coli K-12Potency7.943310
methyl fluorone blackEscherichia coli K-12Potency53.539820
9-hydroxyphenylfluoronEscherichia coli K-12Potency15.848910
2-aminobenzenesulfonamideEscherichia coli K-12Potency3.981110
3-methylbenzotriazin-4-oneEscherichia coli K-12Potency22.411320
tetrandrineEscherichia coli K-12Potency25.118910
bax 439Escherichia coli K-12Potency3.162310
amperozide hydrochlorideEscherichia coli K-12Potency12.602820
ergocornineEscherichia coli K-12Potency22.387210
fangchinolineEscherichia coli K-12Potency35.481310
agroclavineEscherichia coli K-12Potency39.810710
tryptanthrineEscherichia coli K-12Potency0.891310
pramoxine hydrochlorideEscherichia coli K-12Potency26.200020
2-phenylisatogenEscherichia coli K-12Potency39.810710
4,4'-dipyridyl disulfideEscherichia coli K-12Potency89.125110
7-bromo-5-phenyl-1,2-dihydro-2h-1,4-benzodiazepin-2-oneEscherichia coli K-12Potency5.623410
3,4-MethylenedioxyacetophenoneEscherichia coli K-12Potency5.011910
2-(4-Morpholinyl)benzothiazoleEscherichia coli K-12Potency7.079510
4-phenyl-1,2,4-triazoline-3,5-dioneEscherichia coli K-12Potency39.810710
2-(n-morpholino)ethanesulfonic acidEscherichia coli K-12Potency100.000010
N-(4-ethoxyphenyl)-3-hydroxy-2-naphthalenecarboxamideEscherichia coli K-12Potency25.118910
4-(methylsulfonyl)anilineEscherichia coli K-12Potency0.631010
1-methylxanthineEscherichia coli K-12Potency3.981110
1-phenylimidazoleEscherichia coli K-12Potency5.011910
witisolEscherichia coli K-12Potency44.668410
orphenadrine citrateEscherichia coli K-12Potency0.631010
imidaclopridEscherichia coli K-12Potency2.818410
pd 147953Escherichia coli K-12Potency39.810710
5,7-dimethoxyflavoneEscherichia coli K-12Potency39.810710
MetsulfovaxEscherichia coli K-12Potency89.125110
1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5-pyridinedicarboxylic acid dimethyl esterEscherichia coli K-12Potency0.707910
8-(trifluoromethyl)-1H-quinolin-4-oneEscherichia coli K-12Potency39.810710
(1-hydroxycyclopentyl)phenylacetic acidEscherichia coli K-12Potency112.202010
sennoside BEscherichia coli K-12Potency1.258910
prochlorperazine edisylate saltEscherichia coli K-12Potency28.183810
oxybutynin hydrochlorideEscherichia coli K-12Potency39.810710
gliquidoneEscherichia coli K-12Potency29.526220
nimustineEscherichia coli K-12Potency11.220210
nomegestrol acetateEscherichia coli K-12Potency65.811420
3-hydroxybutyric acidEscherichia coli K-12Potency6.309610
peptide elongation factor 2Escherichia coli K-12Potency0.354810
columbianetin, (s)-isomerEscherichia coli K-12Potency44.668410
11-hydroxyprogesterone, (11alpha)-isomerEscherichia coli K-12Potency10.430420
1-(4'-nitrophenyl)-2-aminopropane-1,3-diolEscherichia coli K-12Potency3.981110
corynanthineEscherichia coli K-12Potency14.125410
cycloadiphenine hydrochlorideEscherichia coli K-12Potency39.810710
e-250Escherichia coli K-12Potency7.079510
rac-glycerol 1-monodecanoateEscherichia coli K-12Potency17.782810
nipecotic acid amideEscherichia coli K-12Potency100.000010
norcantharidinEscherichia coli K-12Potency5.623410
osajinEscherichia coli K-12Potency15.848910
4-n-butylaminobenzoic acidEscherichia coli K-12Potency39.810710
3,5,7,3',4'-pentamethoxyflavoneEscherichia coli K-12Potency39.810710
4-(4-hydroxyphenyl)-2-butanolEscherichia coli K-12Potency19.952610
3-hydroxy-3-phenacyloxindoleEscherichia coli K-12Potency8.912510
9-methoxyacridineEscherichia coli K-12Potency0.794310
lecanoric acidEscherichia coli K-12Potency50.118710
karanjinEscherichia coli K-12Potency0.707910
5-(Ethylthio)-1,3,4-thiadiazol-2-amineEscherichia coli K-12Potency8.912510
cinchonidineEscherichia coli K-12Potency7.943310
adenosine arabinoseEscherichia coli K-12Potency3.981110
hexylcaine hydrochlorideEscherichia coli K-12Potency4.466810
cp-55,940Escherichia coli K-12Potency18.063620
paxillineEscherichia coli K-12Potency25.118910
awd 19166Escherichia coli K-12Potency31.622810
6-hydroxydopaEscherichia coli K-12Potency28.599120
perindoprilEscherichia coli K-12Potency4.466810
betaxolol hydrochlorideEscherichia coli K-12Potency39.810710
dihydrocapsaicinEscherichia coli K-12Potency12.589310
lasolvanEscherichia coli K-12Potency0.354810
dibenzo-27-crown-9Escherichia coli K-12Potency28.183810
tadalafilEscherichia coli K-12Potency39.810710
pirlindole hydrochlorideEscherichia coli K-12Potency44.668410
pivmecillinam hydrochlorideEscherichia coli K-12Potency5.011910
1-[4-[2-hydroxy-3-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]propoxy]phenyl]-1-propanoneEscherichia coli K-12Potency1.122010
2-methyl-4-isothiazolin-3-one hydrochlorideEscherichia coli K-12Potency5.623410
n-(phenylthio)-epsilon-caprolactamEscherichia coli K-12Potency4.466810
obacunoneEscherichia coli K-12Potency28.183810
4-(4-(4-chlorophenyl)-4-hydroxy-1-piperidinyl)-1-(4-fluorophenyl)-1-butanolEscherichia coli K-12Potency0.039810
bw 245cEscherichia coli K-12Potency0.354810
gallopamil hydrochlorideEscherichia coli K-12Potency35.481310
histamine dihydrochlorideEscherichia coli K-12Potency89.125110
1,3-dimethylbenzimidazoline-2-thioneEscherichia coli K-12Potency56.234110
n-(n-(3-carboxyoxirane-2-carbonyl)leucyl)isoamylamineEscherichia coli K-12Potency0.794310
n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosineEscherichia coli K-12Potency39.810710
angiotensin ii, des-asp(1)-des-arg(2)-ile(5)-Escherichia coli K-12Potency15.848910
desloratadineEscherichia coli K-12Potency22.016420
alpha-(n6-adenyl)styrene oxideEscherichia coli K-12Potency19.952610
3-hydroxyphenazepamEscherichia coli K-12Potency35.481310
adenosine amine congenerEscherichia coli K-12Potency63.095710
2-phenyl-3-(n,n-dimethylaminopropyl)-1,3-thiazolidin-4-oneEscherichia coli K-12Potency3.311720
azacaineEscherichia coli K-12Potency70.794610
1-(2-hydroxyethyl)-3,5-diphenyl-1h-pyrazoleEscherichia coli K-12Potency100.000010
ici 204448Escherichia coli K-12Potency5.011910
umifenovirEscherichia coli K-12Potency39.810710
4-phenylpiracetamEscherichia coli K-12Potency0.631010
n,n-di-n-hexyl-2-(4-fluorophenyl)indole-3-acetamideEscherichia coli K-12Potency6.309610
3,5-bis(trifluoromethyl)benzyl n-acetyltryptophanEscherichia coli K-12Potency25.118910
sg 209Escherichia coli K-12Potency2.511910
alpha-ergocryptineEscherichia coli K-12Potency39.810710
tilarginine acetateEscherichia coli K-12Potency89.125110
5-hydroxy-3,6,7,8,3',4'-hexamethoxyflavoneEscherichia coli K-12Potency17.782810
r-225Escherichia coli K-12Potency112.202010
1-phenyl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolineEscherichia coli K-12Potency0.631010
8-(methylsulfonylamino)quinolineEscherichia coli K-12Potency25.118910
1-(2'-pyridyl)benzo-1,2,3-triazoleEscherichia coli K-12Potency0.707910
12-phenyllauric acidEscherichia coli K-12Potency28.183810
3-(1-methyl-1,2,3,6-tetrahydropyrid-4-yl)indoleEscherichia coli K-12Potency0.631010
3-methyl-5-aminoisothiazolo-4-carboxylic acidEscherichia coli K-12Potency0.794310
2-phenylbenzotriazoleEscherichia coli K-12Potency35.481310
hyoscyamineEscherichia coli K-12Potency8.912510
1,4-dimethyl-6-nitro-9H-carbazoleEscherichia coli K-12Potency6.309610
schizandrin aEscherichia coli K-12Potency25.118910
nefopam hydrochlorideEscherichia coli K-12Potency44.668410
methyl 5-aminolevulinate hydrochlorideEscherichia coli K-12Potency25.118910
olmesartanEscherichia coli K-12Potency44.668410
cryptotanshinoneEscherichia coli K-12Potency2.511910
Serotonin hydrochlorideEscherichia coli K-12Potency2.818410
harmalanEscherichia coli K-12Potency6.309610
2-phenyl-4-oxohydroquinolineEscherichia coli K-12Potency63.095710
butyroxanEscherichia coli K-12Potency1.000010
fasudil hydrochlorideEscherichia coli K-12Potency22.387210
tanshinone ii aEscherichia coli K-12Potency10.000010
enniatin bEscherichia coli K-12Potency11.220210
2-phenyl-1,2-benzisothiazol-3-(2h)-oneEscherichia coli K-12Potency63.095710
taxusinEscherichia coli K-12Potency15.848910
av-153Escherichia coli K-12Potency2.238710
chondroitin sulfate E (GalNAc4,6diS-GlcA), precursor 3Escherichia coli K-12Potency0.707910
2-[carboxymethyl-[2-(2,6-diethylanilino)-2-oxoethyl]amino]acetic acidEscherichia coli K-12Potency8.912510
1-benzylimidazole-4,5-dicarboxylic acidEscherichia coli K-12Potency3.548110
metralindole monohydrochlorideEscherichia coli K-12Potency89.125110
abt 980Escherichia coli K-12Potency14.733420
rufloxacin hydrochlorideEscherichia coli K-12Potency1.258910
(R)-atenololEscherichia coli K-12Potency112.202010
memantine hydrochlorideEscherichia coli K-12Potency8.912510
2-[(3-oxo-1-cyclohexenyl)amino]benzonitrileEscherichia coli K-12Potency112.202010
pefablocEscherichia coli K-12Potency6.309610
pongidaeEscherichia coli K-12Potency11.220210
2-[(4,6-dimethyl-2-pyrimidinyl)oxy]-3-methoxy-3,3-diphenylpropanoic acidEscherichia coli K-12Potency5.623410
benfluorex hydrochlorideEscherichia coli K-12Potency5.623410
1-acetyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoleEscherichia coli K-12Potency1.000010
erythritolEscherichia coli K-12Potency0.281810
estradiol 3-benzoateEscherichia coli K-12Potency112.202010
adrenosteroneEscherichia coli K-12Potency22.387210
nsc13345Escherichia coli K-12Potency100.000010
carbamothioic acid S-[2-(2-methoxyanilino)-2-oxoethyl] esterEscherichia coli K-12Potency2.238710
4'-hydroxyflavoneEscherichia coli K-12Potency10.000010
benzatropine methanesulfonateEscherichia coli K-12Potency44.668410
4,5-dimethoxy-2,3-dihydroinden-1-oneEscherichia coli K-12Potency10.000010
2-((phenylamino)methyl)isoindoline-1,3-dioneEscherichia coli K-12Potency0.562310
6-phenyl-4,5-dihydro-3(2h)-pyridazinoneEscherichia coli K-12Potency89.125110
1',2'-dihydrorotenoneEscherichia coli K-12Potency35.481310
8-methyl-5-nitroquinolineEscherichia coli K-12Potency44.668410
6-methyl-2-oxo-4-(trifluoromethyl)-1H-pyridine-3-carbonitrileEscherichia coli K-12Potency89.125110
medrysoneEscherichia coli K-12Potency39.810710
asalin, (l-val-l-phe)-isomerEscherichia coli K-12Potency31.622810
melengestrol acetateEscherichia coli K-12Potency39.810710
chondocurine (1beta)-(+-)-isomerEscherichia coli K-12Potency17.782810
nsc 95397Escherichia coli K-12Potency5.011910
oxolamine citrateEscherichia coli K-12Potency4.466810
7-Acetoxy-2-methylisoflavoneEscherichia coli K-12Potency3.548110
methylnaphthazarinEscherichia coli K-12Potency35.179820
n-acetylhistidineEscherichia coli K-12Potency44.668410
noscapineEscherichia coli K-12Potency39.810710
dimethyl 2-(2-nitrobenzylidene)malonateEscherichia coli K-12Potency0.631010
1-[(4-methoxyphenyl)-oxomethyl]-2H-quinoline-2-carbonitrileEscherichia coli K-12Potency0.631010
N1-(4-methyl-1,3-thiazol-2-yl)acetamideEscherichia coli K-12Potency5.623410
1-(4-chlorophenyl)-3-(2-ethoxyphenyl)ureaEscherichia coli K-12Potency10.000010
N1-(1-oxo-2,3-dihydro-1H-inden-5-yl)acetamideEscherichia coli K-12Potency3.162310
nafronyloxalateEscherichia coli K-12Potency1.258910
dicentrineEscherichia coli K-12Potency4.466810
2-methyl-N-[4-(propan-2-ylamino)phenyl]-2-propenamideEscherichia coli K-12Potency31.622810
6-Fluoro-1,3-benzothiazol-2-amineEscherichia coli K-12Potency63.095710
5,7-dimethylpyrimido[4,5-e][1,2,4]triazine-6,8-dioneEscherichia coli K-12Potency7.943310
3-(prop-2-enylthio)-5-thiophen-2-yl-1H-1,2,4-triazoleEscherichia coli K-12Potency89.125110
4-methyl-7-phenyl-3-pyrazolo[5,1-c][1,2,4]triazinecarboxylic acid ethyl esterEscherichia coli K-12Potency112.202010
4,5-diazafluoren-9-oneEscherichia coli K-12Potency7.943310
2,6-diphenyl-1,7-dihydropyrazolo[3,4-b]pyridine-3,4-dioneEscherichia coli K-12Potency4.466810
N-phenylcarbamic acid 2-phenoxyethyl esterEscherichia coli K-12Potency5.011910
6-dimethylaminopurine arabinosideEscherichia coli K-12Potency39.810710
10H-[1]benzothiolo[3,2-b]indoleEscherichia coli K-12Potency89.125110
3-(1h-indol-3-yl)pyrrolidine-2,5-dioneEscherichia coli K-12Potency10.000010
7-benzoyl-3-chloroindolizine-1,2-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency35.481310
8-anilino-1,3-dimethyl-7H-purine-2,6-dioneEscherichia coli K-12Potency50.118710
ritonavirEscherichia coli K-12Potency7.079510
nu 6027Escherichia coli K-12Potency2.511910
1-methyl-6-methoxy-dihydro-beta-carbolineEscherichia coli K-12Potency3.548110
N-(2-phenylphenyl)-2-pyrazinecarboxamideEscherichia coli K-12Potency0.631010
dichloro-1,2-diaminocyclohexane platinum complexEscherichia coli K-12Potency6.309610
acetylglucosamineEscherichia coli K-12Potency44.668410
isomaltoseEscherichia coli K-12Potency4.466810
naringeninEscherichia coli K-12Potency112.202010
deoxyglucoseEscherichia coli K-12Potency3.981110
5-hydroxytryptophanEscherichia coli K-12Potency7.079510
ouabainEscherichia coli K-12Potency25.118910
taxifolinEscherichia coli K-12Potency56.234110
mandelic acid, (s)-isomerEscherichia coli K-12Potency39.810710
quinidineEscherichia coli K-12Potency8.912510
digitoxinEscherichia coli K-12Potency3.981110
saquinavirEscherichia coli K-12Potency31.099020
amiodarone hydrochlorideEscherichia coli K-12Potency39.810710
mometasone furoateEscherichia coli K-12Potency10.000010
nortriptyline hydrochlorideEscherichia coli K-12Potency12.589310
terconazoleEscherichia coli K-12Potency8.539820
grosheiminEscherichia coli K-12Potency100.000010
oxyacanthineEscherichia coli K-12Potency31.622810
DubinidineEscherichia coli K-12Potency44.668410
n-formylmethionine leucyl-phenylalanineEscherichia coli K-12Potency79.432810
cyclo(l-phe-l-pro)Escherichia coli K-12Potency112.202010
[(1S,2R,3S,4S,6R,7R,8R)-4-ethenyl-3-hydroxy-2,4,7,14-tetramethyl-9-oxo-6-tricyclo[5.4.3.01,8]tetradecanyl] 2-[2-(diethylamino)ethylsulfanyl]acetateEscherichia coli K-12Potency5.623410
difluprednateEscherichia coli K-12Potency14.125410
doxorubicin hydrochlorideEscherichia coli K-12Potency31.622810
halcinonideEscherichia coli K-12Potency10.000010
metrizamideEscherichia coli K-12Potency6.309610
erythromycin ethylsuccinateEscherichia coli K-12Potency19.936920
amcinonideEscherichia coli K-12Potency17.782810
dihydroergocristine monomesylateEscherichia coli K-12Potency14.125410
roxithromycinEscherichia coli K-12Potency17.782810
tartaric acidEscherichia coli K-12Potency0.631010
tretinoinEscherichia coli K-12Potency8.912510
arachidonic acidEscherichia coli K-12Potency35.481310
resveratrolEscherichia coli K-12Potency44.668410
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolEscherichia coli K-12Potency4.466810
6-bromoindirubin-3'-oximeEscherichia coli K-12Potency22.717020
afimoxifeneEscherichia coli K-12Potency35.481310
thymopentinEscherichia coli K-12Potency10.000010
decitabineEscherichia coli K-12Potency112.202010
colfosceril palmitateEscherichia coli K-12Potency0.354810
ketoconazoleEscherichia coli K-12Potency11.904810
isotetrandrineEscherichia coli K-12Potency19.952610
N-[4-(methanesulfonamido)phenyl]acetamideEscherichia coli K-12Potency2.511910
4-(2-oxazolo[4,5-b]pyridinyl)anilineEscherichia coli K-12Potency0.562310
6-methyl-2-[(4-nitrophenyl)methylthio]-1H-benzimidazoleEscherichia coli K-12Potency28.183810
likviritonEscherichia coli K-12Potency112.202010
proxymetacaineEscherichia coli K-12Potency0.631010
2-(4-chlorophenyl)-1-phthalazinoneEscherichia coli K-12Potency39.810710
N-bis(N-methylanilino)phosphoryl-N-methylanilineEscherichia coli K-12Potency28.183810
3-(4-chlorophenyl)-6-(1-pyrrolidinyl)-1,2,4,5-tetrazineEscherichia coli K-12Potency44.668410
1-phenyl-4-pyrazololEscherichia coli K-12Potency25.118910
1-[1-(benzenesulfonyl)-3-pyrrolyl]ethanoneEscherichia coli K-12Potency89.125110
1-(phenylmethyl)benzimidazoleEscherichia coli K-12Potency50.118710
2-furancarboxylic acid [4-(6-amino-5-cyano-3-methyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterEscherichia coli K-12Potency100.000010
1-(4-bromo-2,5-dimethoxyphenyl)sulfonylazepaneEscherichia coli K-12Potency5.011910
1-(4-chloro-3-methoxyphenyl)sulfonylazepaneEscherichia coli K-12Potency0.631010
5-(2-methylthioethyl)hydantoinEscherichia coli K-12Potency0.631010
2-(1H-benzimidazol-2-ylthio)-1-thiophen-2-ylethanoneEscherichia coli K-12Potency5.623410
2-(2-phenoxyethylsulfonyl)-1H-benzimidazoleEscherichia coli K-12Potency7.079510
1-(4-methylphenyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneEscherichia coli K-12Potency44.668410
5-(2-furanyl)-3-(3-pyridinyl)-1,2,4-oxadiazoleEscherichia coli K-12Potency22.387210
4-[[7-bicyclo[4.1.0]heptanyl(oxo)methyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency25.118910
LSM-22807Escherichia coli K-12Potency25.118910
4-Morpholinyl(4-pentylcyclohexyl)methanoneEscherichia coli K-12Potency26.632020
2-Methylindole-3-acetic acidEscherichia coli K-12Potency1.584910
3-bromo-N-[2-(4-nitroanilino)ethyl]benzamideEscherichia coli K-12Potency158.489010
5-[[[(5-tert-butyl-2-methyl-3-furanyl)-oxomethyl]amino]methyl]-2-furancarboxylic acid ethyl esterEscherichia coli K-12Potency1.412510
lomatinEscherichia coli K-12Potency0.891310
2-(1-piperazinyl)-4-amino-6,7-dimethoxyquinazolineEscherichia coli K-12Potency25.118910
edulineEscherichia coli K-12Potency25.118910
3-[6-(4-aminophenyl)-2-phenyl-4-pyrimidinyl]anilineEscherichia coli K-12Potency39.810710
2-[(4,4-dimethyl-2,6-dioxocyclohexyl)-(3-pyridinyl)methyl]-5,5-dimethylcyclohexane-1,3-dioneEscherichia coli K-12Potency0.707910
piplartineEscherichia coli K-12Potency3.981110
7-methoxyisoflavoneEscherichia coli K-12Potency1.412510
piperineEscherichia coli K-12Potency44.668410
isoliquiritigeninEscherichia coli K-12Potency112.202010
ilepcimideEscherichia coli K-12Potency28.183810
6-amino-2-methyl-8-phenyl-1,6,8,8a-tetrahydroisoquinoline-5,7,7-tricarbonitrileEscherichia coli K-12Potency10.000010
3-[[2-[[4-ethyl-5-[(4-methylanilino)methyl]-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency5.011910
3-[(1-cyclopentyl-5-tetrazolyl)-(3,4-dihydro-1H-isoquinolin-2-yl)methyl]-7-methoxy-1H-quinolin-2-oneEscherichia coli K-12Potency35.481310
2-imino-N,8-dimethyl-5-oxo-1-propan-2-yl-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideEscherichia coli K-12Potency79.432810
3-[[1,3-benzodioxol-5-ylmethyl-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneEscherichia coli K-12Potency44.668410
2-(1,3-benzoxazol-2-ylthio)propanoic acidEscherichia coli K-12Potency89.125110
1-[4-[4-[(4-methylphenyl)methylamino]phenyl]-1-piperazinyl]ethanoneEscherichia coli K-12Potency20.259320
2-[[5-[4-(1-piperidinylsulfonyl)phenyl]-1H-1,2,4-triazol-3-yl]thio]-N-(2-thiazolyl)acetamideEscherichia coli K-12Potency7.855220
N-[2-(cyclopentylamino)-1-(5-methyl-2-furanyl)-2-oxoethyl]-N-[(4-fluorophenyl)methyl]-4-thiadiazolecarboxamideEscherichia coli K-12Potency112.202010
N-(3,5-dimethoxyphenyl)-2-thiophenecarboxamideEscherichia coli K-12Potency6.309610
N-(cyclohexylmethyl)-5,6,7,8-tetrahydrotetrazolo[5,1-b]quinazolin-9-amineEscherichia coli K-12Potency2.818410
6-amino-4-(2-ethoxyphenyl)-3-propyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileEscherichia coli K-12Potency6.309610
N-[1-[(2-bromophenyl)methyl]-2-oxo-3-pyridinyl]butanamideEscherichia coli K-12Potency63.095710
3-[5-(2-methoxyethylthio)-4-methyl-1,2,4-triazol-3-yl]benzonitrileEscherichia coli K-12Potency0.631010
2-[3-[3-[3-(1-imidazolyl)propyl]-4-oxo-2-quinazolinyl]propyl]isoindole-1,3-dioneEscherichia coli K-12Potency28.183810
LSM-19079Escherichia coli K-12Potency56.234110
2-(4-chlorophenoxy)-N-(2-pyridin-4-yl-1,3-benzoxazol-5-yl)acetamideEscherichia coli K-12Potency0.707910
1-(2,5-dimethoxyphenyl)-2-[[5-(2-furanyl)-4-propyl-1,2,4-triazol-3-yl]thio]ethanoneEscherichia coli K-12Potency28.183810
N-butan-2-yl-N-[2-[(4-methoxyphenyl)methylamino]-2-oxoethyl]-4-thiadiazolecarboxamideEscherichia coli K-12Potency1.122010
2-[(5,5-dimethyl-6H-[1,2,4]triazolo[3,4-a]isoquinolin-3-yl)thio]-1-[4-(2-methoxyphenyl)-1-piperazinyl]ethanoneEscherichia coli K-12Potency15.211320
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid ethyl esterEscherichia coli K-12Potency0.631010
4-(4-fluorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid 1,3-benzodioxol-5-ylmethyl esterEscherichia coli K-12Potency50.118710
4-[[2-(1-benzotriazolyl)-1-oxoethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency25.118910
2-amino-3-cyano-5-oxo-1'-spiro[7,8-dihydro-6H-1-benzopyran-4,4'-piperidine]carboxylic acid (phenylmethyl) esterEscherichia coli K-12Potency56.234110
2-[[1-oxo-2-[3-(trifluoromethyl)-5,6-dihydro-4H-cyclopenta[c]pyrazol-1-yl]ethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency7.943310
2,4-dichlorobenzoic acid 1,2,4-triazol-1-ylmethyl esterEscherichia coli K-12Potency100.000010
4-chloro-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)benzamideEscherichia coli K-12Potency100.000010
2-[2-[[2-[(5-cyclopropyl-4-methyl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esterEscherichia coli K-12Potency28.183810
N-[2,5-diethoxy-4-[[2-(3-methoxyphenyl)-1-oxoethyl]amino]phenyl]-2-furancarboxamideEscherichia coli K-12Potency22.387210
N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-cyclohexyl-2-furancarboxamideEscherichia coli K-12Potency31.622810
N-[4-[3-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-2-hydroxypropoxy]phenyl]acetamideEscherichia coli K-12Potency39.810710
2-(2-ethyl-6-methyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(5-methyl-2-furanyl)methyl]-N-(3-pyridinylmethyl)acetamideEscherichia coli K-12Potency20.811420
1-(1-adamantyl)-3-[8-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]ureaEscherichia coli K-12Potency0.631010
1-(1,3-benzodioxol-5-ylmethyl)-3-hydroxy-3-[2-(4-methylphenyl)-2-oxoethyl]-2-indoloneEscherichia coli K-12Potency0.707910
N4-cyclohexyl-N1-ethyl-N4-(2-pyridinylmethyl)benzene-1,4-disulfonamideEscherichia coli K-12Potency1.412510
2-[cyclohexyl-(2,4,6-trimethylphenyl)sulfonylamino]-N-(3-pyridinylmethyl)acetamideEscherichia coli K-12Potency13.815420
2-[[4-(2-furanylmethyl)-5-methyl-1,2,4-triazol-3-yl]thio]-N-(4-methyl-2-thiazolyl)acetamideEscherichia coli K-12Potency6.309610
1-(4-chlorophenyl)sulfonyl-N-[3-methoxy-4-(1-tetrazolyl)phenyl]-4-piperidinecarboxamideEscherichia coli K-12Potency4.771820
4-[[(1-methylsulfonyl-4-piperidinyl)-oxomethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency79.432810
N-[2-methyl-4-oxo-3-(phenylmethyl)-7-(1-piperidinyl)-6-quinazolinyl]-3-pyridinecarboxamideEscherichia coli K-12Potency21.679420
11-[2-(4-morpholinyl)ethylamino]-7,8,9,10-tetrahydrobenzimidazolo[1,2-b]isoquinoline-6-carbonitrileEscherichia coli K-12Potency50.118710
2,6-diamino-4-(1-phenylethyl)-4H-thiopyran-3,5-dicarbonitrileEscherichia coli K-12Potency4.466810
1-methyl-2-[(4-methyl-1-piperidinyl)methyl]-3-indolecarbonitrileEscherichia coli K-12Potency1.412510
8-[(1-cyclohexyl-5-tetrazolyl)methyl]-3-(4-fluorophenyl)-8-azabicyclo[3.2.1]octan-3-olEscherichia coli K-12Potency55.756220
1-[3-(4-morpholinyl)propyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-3-phenylureaEscherichia coli K-12Potency30.300120
N-(1,3-benzothiazol-2-yl)-N-methylbenzamideEscherichia coli K-12Potency19.952610
6-methyl-3-[[[1-(phenylmethyl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneEscherichia coli K-12Potency70.794610
4-[2-[1-(4-methoxyphenyl)sulfonyl-2-benzimidazolyl]ethyl]morpholineEscherichia coli K-12Potency15.848910
4-[2-[[4-(dimethylamino)phenyl]methylamino]ethyl]-2,2-dimethyl-4-oxanolEscherichia coli K-12Potency1.584910
2-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-2-azaspiro[5.5]undecaneEscherichia coli K-12Potency89.125110
6-ethoxy-3-[[2-oxolanylmethyl-[[1-(2-phenylethyl)-5-tetrazolyl]methyl]amino]methyl]-1H-quinolin-2-oneEscherichia coli K-12Potency10.000010
1-[1-[oxo(1-pyrrolidinyl)methyl]cyclohexyl]-3-(phenylmethyl)ureaEscherichia coli K-12Potency6.309610
2-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d][1,3]thiazin-4-oneEscherichia coli K-12Potency35.481310
3-[5-(4-ethylphenyl)-2-tetrazolyl]propanoic acid methyl esterEscherichia coli K-12Potency22.387210
1-[1-(1-cyclopentyl-5-tetrazolyl)-2-methylpropyl]-4-(2-fluorophenyl)piperazineEscherichia coli K-12Potency56.234110
N-(6-ethoxy-1,3-benzothiazol-2-yl)-2-[[3-(2-furanylmethyl)-4-oxo-2-quinazolinyl]thio]acetamideEscherichia coli K-12Potency3.548110
N-tert-butyl-2-[[5-(3,5-dimethoxyphenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(phenylmethyl)acetamideEscherichia coli K-12Potency44.668410
N-[4-[1-(benzenesulfonyl)-2,3-dihydroindol-5-yl]-2-thiazolyl]-2-(4-morpholinyl)acetamideEscherichia coli K-12Potency22.387210
2-[[5-(4-fluorophenyl)-1-methyl-2-imidazolyl]thio]-N-[2-(4-morpholinyl)phenyl]acetamideEscherichia coli K-12Potency28.183810
2-[[5-(1-benzotriazolylmethyl)-1,3,4-oxadiazol-2-yl]thio]-N-[(4-fluorophenyl)methyl]-N-phenylacetamideEscherichia coli K-12Potency39.810710
3-[2-hydroxy-3-(4-morpholinyl)propyl]-5,5-dimethylimidazolidine-2,4-dioneEscherichia coli K-12Potency0.631010
N-cyclopentyl-2-[2-oxolanylmethyl-(1-oxo-2-thiophen-2-ylethyl)amino]-2-thiophen-2-ylacetamideEscherichia coli K-12Potency2.818410
4,5-dichloro-3-isothiazolecarboxylic acid [1-(2-furanylmethylamino)-1-oxopropan-2-yl] esterEscherichia coli K-12Potency112.202010
3-[(1-cyclopentyl-5-tetrazolyl)-[4-(2-methoxyphenyl)-1-piperazinyl]methyl]-7-methyl-1H-quinolin-2-oneEscherichia coli K-12Potency25.118910
bikininEscherichia coli K-12Potency3.981110
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]propanoic acid ethyl esterEscherichia coli K-12Potency0.631010
N-[4-[oxo-(2-pyridinylamino)methyl]phenyl]-2-furancarboxamideEscherichia coli K-12Potency5.623410
1-methyl-4-[2-oxo-2-(4-phenyl-1-piperazinyl)ethyl]-5-pyrrolo[3,2-b]pyrrolecarboxylic acid ethyl esterEscherichia coli K-12Potency28.370820
N-[(7-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(3-pyridinylmethyl)benzenesulfonamideEscherichia coli K-12Potency31.622810
5-[(5-methoxycarbonyl-2-methyl-3-furanyl)methoxy]-2-methyl-3-benzofurancarboxylic acid 2-methoxyethyl esterEscherichia coli K-12Potency25.118910
4-methyl-N-[2-[4-(2-methyl-1-oxopropyl)-1-piperazinyl]phenyl]benzamideEscherichia coli K-12Potency0.631010
2-(1,3-dimethyl-2,6-dioxo-7-purinyl)-N-(phenylmethyl)-N-(2-pyridinyl)acetamideEscherichia coli K-12Potency0.707910
2-(2,4-dioxo-3-thiazolidinyl)-N-(2,3,4-trifluorophenyl)acetamideEscherichia coli K-12Potency25.118910
5-(2-ethoxyphenyl)-3-(2-methoxy-6-methyl-3-pyridinyl)-1,2,4-oxadiazoleEscherichia coli K-12Potency39.810710
N-[2-(4-methoxyphenyl)-1,3-benzoxazol-5-yl]-1,3-benzodioxole-5-carboxamideEscherichia coli K-12Potency28.183810
N-tert-butyl-N-[2-(tert-butylamino)-2-oxoethyl]-3-(3,4-dihydro-2H-quinolin-1-yl)propanamideEscherichia coli K-12Potency20.611620
[5-(2-furanyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency31.622820
N'-[1-[(cyclohexylamino)-oxomethyl]cyclopentyl]-N-(5-methyl-3-isoxazolyl)-N'-phenylbutanediamideEscherichia coli K-12Potency0.707910
3-cyclohexyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-1-[2-(1-pyrrolidinyl)ethyl]ureaEscherichia coli K-12Potency2.818410
3-[3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-6-ethyl-1H-quinolin-2-oneEscherichia coli K-12Potency25.118910
2-[4-[(1-cyclopentyl-5-tetrazolyl)-(6-quinolinyl)methyl]-1-piperazinyl]-1,3-benzothiazoleEscherichia coli K-12Potency39.810710
1-(3,5-dimethyl-1-pyrazolyl)-3-[2-(4-methoxyphenyl)-1-indolyl]-2-propanolEscherichia coli K-12Potency28.183810
2-[[5-[(2-chloroanilino)methyl]-4-phenyl-1,2,4-triazol-3-yl]thio]acetic acid ethyl esterEscherichia coli K-12Potency22.387210
N-[1-[2-(2-chlorophenoxy)ethyl]-2-benzimidazolyl]acetamideEscherichia coli K-12Potency39.810710
N-(5-methyl-1,3,4-thiadiazol-2-yl)-N-phenyl-2-pyrazinecarboxamideEscherichia coli K-12Potency100.000010
2-[(2-methoxy-1-oxoethyl)amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency39.810710
2-[[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency0.631010
N-(2,5-diethoxyphenyl)-2-[(3-methyl-2-imidazo[4,5-b]pyridinyl)thio]acetamideEscherichia coli K-12Potency70.794610
1-(1-piperidinyl)-2-[[4-(prop-2-enylamino)-1-phthalazinyl]thio]ethanoneEscherichia coli K-12Potency5.011910
2-[(1,3-dimethyl-2,6-dioxo-7-propyl-8-purinyl)thio]-N-[2-(1-piperidinyl)phenyl]acetamideEscherichia coli K-12Potency15.848910
2-[[1-oxo-2-(2-oxo-1,3-benzothiazol-3-yl)ethyl]amino]benzoic acidEscherichia coli K-12Potency0.316210
1-(4-chlorophenyl)-1-cyclohexyl-3-(4-morpholinyl)-1-propanolEscherichia coli K-12Potency58.654420
3-(2,5-dimethyl-1-pyrrolyl)-4-methylanilineEscherichia coli K-12Potency0.631010
N-(4-acetamidophenyl)-2-[(5-cyclopropyl-4-ethyl-1,2,4-triazol-3-yl)thio]acetamideEscherichia coli K-12Potency79.432810
1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-(4-methoxyphenyl)sulfonylpiperazineEscherichia coli K-12Potency0.316210
1-(3-chlorophenyl)-3-[4-[4-morpholinyl(oxo)methyl]phenyl]ureaEscherichia coli K-12Potency0.031610
2-[cyclohexyl-[2-[5-(3,4-dimethoxyphenyl)-2-tetrazolyl]-1-oxoethyl]amino]-N-cyclopentylpropanamideEscherichia coli K-12Potency22.387210
2-methyl-4-[2-oxo-2-(2-phenylethylamino)ethyl]-5-thieno[3,2-b]pyrrolecarboxylic acid ethyl esterEscherichia coli K-12Potency25.118910
4-[[[[8-[(1-tert-butyl-5-tetrazolyl)methyl]-8-azabicyclo[3.2.1]octan-3-yl]amino]-oxomethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency5.623410
4-[[4-ethyl-5-[(2-methylphenoxy)methyl]-1,2,4-triazol-3-yl]thio]-N-(2-methoxyphenyl)-3-oxobutanamideEscherichia coli K-12Potency0.631010
6-hydroxy-1-(3-hydroxypropyl)-4-methyl-2-oxo-5-(1-piperidinylmethyl)-3-pyridinecarbonitrileEscherichia coli K-12Potency12.589310
1-(3-cyano-7-methoxy-2-quinolinyl)-4-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency22.779820
4-methyl-N-(pyridin-4-ylmethyl)benzenesulfonamideEscherichia coli K-12Potency1.000010
6-ethoxy-3-[[[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneEscherichia coli K-12Potency28.183810
6-ethyl-2,5-dimethyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrileEscherichia coli K-12Potency100.000010
1-[(3,4-dimethoxyphenyl)-[1-(2-methoxyethyl)-5-tetrazolyl]methyl]-2,3-dihydroindoleEscherichia coli K-12Potency39.810710
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideEscherichia coli K-12Potency5.011910
1-[3-(dimethylamino)propyl]-1-[(5,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-3-(phenylmethyl)ureaEscherichia coli K-12Potency35.481310
2-[4-(benzenesulfonyl)phenyl]-5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazoleEscherichia coli K-12Potency112.202010
N-[6-(1-oxopentylamino)-3-pyridinyl]-3-pyridinecarboxamideEscherichia coli K-12Potency0.631010
2-(1,3-benzothiazol-2-ylamino)-4-(methylthio)butanoic acidEscherichia coli K-12Potency4.466810
1-(8-methyl-2,5,11,14-tetraoxa-8-azabicyclo[13.4.0]nonadeca-1(15),16,18-trien-17-yl)ethanolEscherichia coli K-12Potency19.952610
N-[(1,3-dimethyl-4-pyrazolyl)methyl]-5-(2-furanyl)-N-methyl-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideEscherichia coli K-12Potency25.118910
1-[4-(2-methoxyphenyl)-1-piperazinyl]-2-[[5-(2-methyl-3-furanyl)-1,3,4-oxadiazol-2-yl]thio]ethanoneEscherichia coli K-12Potency31.622810
8-[(1-tert-butyl-5-tetrazolyl)-thiomorpholin-4-ylmethyl]-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneEscherichia coli K-12Potency0.794310
1-[1-[1-(1,3-benzodioxol-5-ylmethyl)-5-tetrazolyl]-2-methylpropyl]-4-phenylpiperazineEscherichia coli K-12Potency112.202010
2-(2,5-dimethoxyphenyl)-5-[4-(4-methoxyphenyl)phenyl]-1,3,4-oxadiazoleEscherichia coli K-12Potency35.481310
6-(3,4-dimethoxyphenyl)-4-methoxy-1,3-dimethyl-8-cyclohepta[c]furanoneEscherichia coli K-12Potency25.118910
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-6-methyl-1H-quinolin-2-oneEscherichia coli K-12Potency1.258910
2-[[[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-3-furanyl]-oxomethyl]amino]pentanedioic acid dimethyl esterEscherichia coli K-12Potency35.481310
5-(3,4-dimethoxyphenyl)-1H-1,2,4-triazol-3-amineEscherichia coli K-12Potency0.707910
N-(2-pyridin-4-yl-1,3-benzoxazol-5-yl)butanamideEscherichia coli K-12Potency1.122010
3-[2-(3-phenoxypropyl)-5-tetrazolyl]pyridineEscherichia coli K-12Potency1.412510
(2,4-difluorophenyl)-[3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]methanoneEscherichia coli K-12Potency39.810710
2-fluoro-N-(2-hydroxyethyl)-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]benzamideEscherichia coli K-12Potency2.818410
2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)thio]-N-(4-phenyl-2-thiazolyl)acetamideEscherichia coli K-12Potency79.432810
(6-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-yl)-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]methanoneEscherichia coli K-12Potency15.866020
1-[1-[[1-[(4-methylphenyl)methyl]-5-tetrazolyl]methyl]-4-piperidinyl]-5-(trifluoromethyl)benzotriazoleEscherichia coli K-12Potency7.692220
3-[1-azepanyl-[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl]-6,7-dimethoxy-1H-quinolin-2-oneEscherichia coli K-12Potency20.259320
N-(2-furanylmethyl)-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]benzamideEscherichia coli K-12Potency42.239520
9-[3-(4-acetyl-3,5-dimethyl-1-pyrazolyl)-2-hydroxypropyl]-6-methyl-3,4-dihydro-2H-carbazol-1-oneEscherichia coli K-12Potency39.810710
2-[[4-(4-methoxyphenyl)-2-pyrimidinyl]thio]-1-(4-morpholinyl)ethanoneEscherichia coli K-12Potency15.848910
1-(3-methoxyphenyl)-2-[[4-methyl-5-[[(4-phenyl-2-thiazolyl)amino]methyl]-1,2,4-triazol-3-yl]thio]ethanoneEscherichia coli K-12Potency5.623410
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneEscherichia coli K-12Potency2.511910
2-[[3-acetyl-1-[4-(dimethylamino)phenyl]-2-methyl-5-indolyl]oxy]acetamideEscherichia coli K-12Potency39.810710
2-ethoxy-N-[4-(4-morpholinylsulfonyl)phenyl]benzamideEscherichia coli K-12Potency3.162310
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2-pyrimidinyl)-3-piperidinecarboxamideEscherichia coli K-12Potency2.818410
2-[(5,6-dimethyl-4-oxo-3-phenyl-2-thieno[2,3-d]pyrimidinyl)thio]-N-(2-furanylmethyl)acetamideEscherichia coli K-12Potency2.818410
4-methyl-N-(2-methyl-5-tetrazolyl)benzamideEscherichia coli K-12Potency0.562310
2-[[4-(3,4-dimethoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideEscherichia coli K-12Potency2.238710
3-[[cyclopentyl-[[1-[(4-methoxyphenyl)methyl]-5-tetrazolyl]methyl]amino]methyl]-7-methyl-1H-quinolin-2-oneEscherichia coli K-12Potency39.810710
2-[(2,5-dimethylphenyl)methylthio]-5-(3-pyridinyl)-1,3,4-oxadiazoleEscherichia coli K-12Potency112.202010
3-cyclohexyl-1-[(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-[3-(4-morpholinyl)propyl]ureaEscherichia coli K-12Potency28.183810
2-[[5-(2-furanyl)-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]-1-(4-morpholinyl)ethanoneEscherichia coli K-12Potency35.481310
1-(2-methoxyphenyl)-4-[(4-methylphenyl)-(1-propan-2-yl-5-tetrazolyl)methyl]piperazineEscherichia coli K-12Potency19.622220
N,N-diethyl-2-[(3-thiophen-2-yl-7-isothiazolo[4,5-d]pyrimidinyl)thio]acetamideEscherichia coli K-12Potency0.707910
N-[(1-cyclohexyl-5-tetrazolyl)-thiophen-2-ylmethyl]-N-(phenylmethyl)ethanamineEscherichia coli K-12Potency3.548110
6-[(2-fluorophenyl)methyl]-2,4-dimethyl-5-thieno[3,4]pyrrolo[1,3-d]pyridazinoneEscherichia coli K-12Potency0.631010
1-phenyl-4-[[1-(phenylmethyl)-5-tetrazolyl]-(3-pyridinyl)methyl]piperazineEscherichia coli K-12Potency24.905420
3-[[1-[1-(2-furanylmethyl)-5-tetrazolyl]propyl-(2-phenylethyl)amino]methyl]-7-methoxy-1H-quinolin-2-oneEscherichia coli K-12Potency39.810710
N-(2-furanylmethyl)-2-[(4-methoxyphenyl)sulfonylamino]benzamideEscherichia coli K-12Potency39.810710
N-[2,5-dimethoxy-4-[[2-(4-morpholinyl)-1-oxoethyl]amino]phenyl]benzamideEscherichia coli K-12Potency7.943310
N-methyl-N-[5-(5-methyl-2-pyrazinyl)-1,3,4-thiadiazol-2-yl]-2-oxolanecarboxamideEscherichia coli K-12Potency44.668410
3-[[[[3-[(4-chlorophenyl)methyl]-2-methyl-4-oxo-6-quinazolinyl]amino]-oxomethyl]amino]propanoic acid ethyl esterEscherichia coli K-12Potency28.183810
N-[4-(4-acetyl-1-piperazinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideEscherichia coli K-12Potency0.631010
4-amino-2-[[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]thio]-5-pyrimidinecarboxylic acid ethyl esterEscherichia coli K-12Potency1.778310
N-(4-fluorophenyl)-4-(2-oxolanylmethylsulfamoyl)benzamideEscherichia coli K-12Potency50.118710
N-[3-chloro-4-(4-morpholinyl)phenyl]-2-furancarboxamideEscherichia coli K-12Potency7.079510
2-[[1-(4-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]thio]acetic acid ethyl esterEscherichia coli K-12Potency100.000010
4-(2,4-dimethyl-5-thiazolyl)-N-(phenylmethyl)-2-thiazolamineEscherichia coli K-12Potency5.011910
6-methoxy-3-[[[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl-(2-phenylethyl)amino]methyl]-1H-quinolin-2-oneEscherichia coli K-12Potency5.623410
N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]butanamideEscherichia coli K-12Potency8.912510
5-[(2-fluoroanilino)methyl]-8-quinolinolEscherichia coli K-12Potency1.122010
4-[[4-(1,3-benzothiazol-2-yl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-2-methoxyphenolEscherichia coli K-12Potency11.547620
N-[2-(4-chloro-N-[2-(cyclohexylamino)-2-oxoethyl]anilino)-2-oxoethyl]-2-furancarboxamideEscherichia coli K-12Potency56.234110
4-amino-N5-[2-(2-methoxyethylamino)-1-(5-methyl-2-furanyl)-2-oxoethyl]-N5-(thiophen-2-ylmethyl)isothiazole-3,5-dicarboxamideEscherichia coli K-12Potency50.118710
N'-[2-(cyclopentylamino)-2-oxo-1-pyridin-4-ylethyl]-N-(5-methyl-3-isoxazolyl)-N'-phenylbutanediamideEscherichia coli K-12Potency0.562310
N-[4-(diethylsulfamoyl)phenyl]-2-(2-oxo-1,3-benzothiazol-3-yl)acetamideEscherichia coli K-12Potency5.623410
N-[(5,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-4-methoxy-N-[3-(2-oxo-1-pyrrolidinyl)propyl]benzenesulfonamideEscherichia coli K-12Potency17.782810
N-(5-ethyl-4-phenyl-2-thiazolyl)-2-methoxyacetamideEscherichia coli K-12Potency0.707910
1-(4,6-dimethyl-2-pyrimidinyl)-4-piperidinecarboxylic acidEscherichia coli K-12Potency44.668410
N-(3-methyl-2-pyridinyl)-2-(6,7,8,9-tetrahydrodibenzofuran-2-yloxy)acetamideEscherichia coli K-12Potency19.952610
1-[(3,4-dimethoxyphenyl)-[1-(thiophen-2-ylmethyl)-5-tetrazolyl]methyl]-4-phenylpiperazineEscherichia coli K-12Potency28.183810
1-(5-chloro-2-methoxyphenyl)-2-[(4,6-diamino-2-pyrimidinyl)thio]ethanoneEscherichia coli K-12Potency89.125110
3-[3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl-[1-(2-oxolanylmethyl)-5-tetrazolyl]methyl]-5,7-dimethyl-1H-quinolin-2-oneEscherichia coli K-12Potency2.818410
N-[2-(1H-benzimidazol-2-yl)ethyl]-2-[4-(5-fluoro-1-benzotriazolyl)-1-piperidinyl]acetamideEscherichia coli K-12Potency0.631010
N3-(2,3-dimethylphenyl)-N1-(2-methoxyphenyl)piperidine-1,3-dicarboxamideEscherichia coli K-12Potency50.118710
N-(3,4-dimethylphenyl)-2-[[5-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency31.622810
N,N-dimethyl-4-[[4-(5-methyl-1-benzotriazolyl)-1-piperidinyl]sulfonyl]benzamideEscherichia coli K-12Potency39.810710
2-[[5-[[2-(3-chloroanilino)-4-thiazolyl]methyl]-4-(3-methoxypropyl)-1,2,4-triazol-3-yl]thio]acetic acid methyl esterEscherichia coli K-12Potency19.952610
hydrastine, (r-(r*,s*))-isomerEscherichia coli K-12Potency2.818410
5,6-dichloro-1-ethyl-1,3-dihydro-2h-benzimidazol-2-oneEscherichia coli K-12Potency0.562310
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideEscherichia coli K-12Potency12.589310
fludarabineEscherichia coli K-12Potency112.202010
glycerylphosphorylcholineEscherichia coli K-12Potency0.562310
r 59949Escherichia coli K-12Potency3.162310
n(6)-cyclopentyladenosineEscherichia coli K-12Potency53.154820
methylatropine nitrateEscherichia coli K-12Potency35.481310
2-(3,5-dimethyl-1-pyrazolyl)-N,6-dimethyl-4-pyrimidinamineEscherichia coli K-12Potency100.000010
6,6,7-trimethyl-1-(4-morpholinyl)-3-(phenylmethylthio)-5,8-dihydro-2,7-naphthyridine-4-carbonitrileEscherichia coli K-12Potency17.782810
LSM-16947Escherichia coli K-12Potency89.125110
2,3,4,5,6-pentafluoro-N-(phenylmethyl)benzamideEscherichia coli K-12Potency112.202010
2-[(7-methyl-4-oxo-3-phenyl-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-2-yl)thio]acetic acid methyl esterEscherichia coli K-12Potency0.891310
7-methyl-3-(4-morpholinyl)-1-(prop-2-enylamino)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileEscherichia coli K-12Potency12.589310
3-amino-5-methyl-4-[[3-(4-morpholinyl)propylamino]-oxomethyl]-2-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency0.707910
2-(4-methyl-1-oxo-2-phthalazinyl)-N-(4-methylphenyl)acetamideEscherichia coli K-12Potency19.952610
LSM-19776Escherichia coli K-12Potency0.281810
2-amino-1-(1,3-benzodioxol-5-yl)-N-[2-(4-morpholinyl)ethyl]-3-pyrrolo[3,2-b]quinoxalinecarboxamideEscherichia coli K-12Potency14.125410
2-(2-methyl-1H-indol-3-yl)ethanolEscherichia coli K-12Potency8.912510
5-chloro-3-[[2-(4-ethoxycarbonyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterEscherichia coli K-12Potency35.481310
2-amino-4-(2-chlorophenyl)-6-(ethylthio)pyridine-3,5-dicarbonitrileEscherichia coli K-12Potency39.810710
N-(2,1,3-benzothiadiazol-5-yl)-2,4-dimethyl-6-oxo-3-pyrancarboxamideEscherichia coli K-12Potency0.631010
1-(2-pyrimidinyl)-3-(2,2,2-trifluoroethyl)ureaEscherichia coli K-12Potency7.943310
2-cyano-N-(3-methoxypropyl)-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetamideEscherichia coli K-12Potency17.782810
2-(pyridin-4-yl)-4-(pyrrolidin-1-yl)quinazolineEscherichia coli K-12Potency89.125110
3,4,5-trimethoxy-N-[2-(4-sulfamoylphenyl)ethyl]benzamideEscherichia coli K-12Potency4.466810
LSM-27020Escherichia coli K-12Potency0.631010
2-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-1-(8-methyl-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)ethanoneEscherichia coli K-12Potency15.848910
3-[[2-[4-(3-chlorophenyl)-1-piperazinyl]-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterEscherichia coli K-12Potency39.810710
N-[1-(1-hexyl-2-benzimidazolyl)ethyl]-2-furancarboxamideEscherichia coli K-12Potency28.183810
5,6-dimethoxy-3-[[(3-methoxyphenyl)-oxomethyl]amino]-1H-indole-2-carboxylic acid methyl esterEscherichia coli K-12Potency42.239520
5-[(4-chlorophenyl)methylamino]-6-methyl-2H-1,2,4-triazin-3-oneEscherichia coli K-12Potency4.466810
2-[[(4-chloro-1-methyl-3-pyrazolyl)-oxomethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency56.234110
2-cyano-2-[3-[4-(phenylmethyl)-1-piperazinyl]-2-quinoxalinyl]acetic acid 2-methoxyethyl esterEscherichia coli K-12Potency35.481310
2,6-dimethyl-4-[1-(2-naphthalenylsulfonyl)-4-piperidinyl]morpholineEscherichia coli K-12Potency31.225620
4-amino-5,8-dimethoxy-2-(1,1,2,2,2-pentafluoroethyl)-3-quinolinecarbonitrileEscherichia coli K-12Potency1.258910
N-[2-(1-cyclohexenyl)ethyl]-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineEscherichia coli K-12Potency0.707910
N-ethyl-2-imino-10-methyl-1-[(4-methylphenyl)methyl]-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideEscherichia coli K-12Potency100.000010
5-bromo-3-[[2-(4-methyl-1-piperazinyl)-1-oxoethyl]amino]-2-benzofurancarboxylic acid ethyl esterEscherichia coli K-12Potency28.183810
2-[[2-methyl-5-(3-methyl-4-oxo-1-phthalazinyl)phenyl]sulfonylamino]acetic acid ethyl esterEscherichia coli K-12Potency39.810710
7-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxoethyl]amino]-5H-[1,3]dioxolo[4,5-f]indole-6-carboxylic acid ethyl esterEscherichia coli K-12Potency0.631010
2-amino-4-(2-ethoxyphenyl)-7-methyl-5-oxo-6-(2-pyridinylmethyl)-4H-pyrano[3,2-c]pyridine-3-carbonitrileEscherichia coli K-12Potency1.122010
arachinEscherichia coli K-12Potency7.943310
5-(2,4-dimethoxyphenyl)-7-(3,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency5.623410
2-[(6-chloro-4-ethyl-2-oxo-1-benzopyran-7-yl)oxy]propanoic acidEscherichia coli K-12Potency3.981110
1-(3,5-dichlorophenyl)-3-(N-hydroxyanilino)pyrrolidine-2,5-dioneEscherichia coli K-12Potency35.481310
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-phenyl-2-furancarboxamideEscherichia coli K-12Potency63.095710
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterEscherichia coli K-12Potency25.118910
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid cyclohexyl esterEscherichia coli K-12Potency79.432810
5-bromo-N-(2-pyridinylmethyl)-2-thiophenesulfonamideEscherichia coli K-12Potency3.162310
4-(2-furanyl)-3-methyl-5-(4-methylphenyl)-2,4-dihydropyrrolo[3,4-c]pyrazol-6-oneEscherichia coli K-12Potency39.810710
6-[(2,4-dichlorophenoxy)methyl]-3-(2-methoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleEscherichia coli K-12Potency28.183810
cardionogen-2Escherichia coli K-12Potency44.668410
6-(4-methoxyphenyl)-3-phenyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleEscherichia coli K-12Potency0.141310
2-[(4-amino-5-cyclohexyl-1,2,4-triazol-3-yl)thio]-N-(3-fluoro-4-methylphenyl)acetamideEscherichia coli K-12Potency0.707910
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-methyl-4-pyridinecarboxamideEscherichia coli K-12Potency3.162310
4-[4-(1H-benzimidazol-2-ylmethyl)-1-piperazinyl]benzofuro[3,2-d]pyrimidineEscherichia coli K-12Potency35.716820
2-[4-[(4-chlorophenyl)methoxy]phenyl]-5-(dimethylamino)-4-oxazolecarbonitrileEscherichia coli K-12Potency1.778310
2-[2-(dimethylamino)ethylthio]-6,6-dimethyl-5,8-dihydropyrano[4,5]thieno[1,2-c]pyrimidin-4-amineEscherichia coli K-12Potency56.234110
N-[7-(2-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideEscherichia coli K-12Potency39.810710
3-(ethylaminomethyl)-6-methyl-1H-quinolin-2-oneEscherichia coli K-12Potency0.631010
8-(1,3-benzothiazol-2-ylthio)-3-methyl-7-pentylpurine-2,6-dioneEscherichia coli K-12Potency25.118910
1-(2,1,3-benzoxadiazol-4-yloxy)-3,3-dimethyl-1-(1,2,4-triazol-1-yl)-2-butanoneEscherichia coli K-12Potency50.118710
2-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-3a,4,7,7a-tetrahydroisoindole-1,3-dioneEscherichia coli K-12Potency125.892010
2-(2-furanyl)-5-(2-furanylmethylamino)-4-oxazolecarbonitrileEscherichia coli K-12Potency112.202010
5-(1-azepanyl)-2-(3,4-dimethoxyphenyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency39.810710
3-(4-chlorophenyl)-6-(thiophen-2-ylmethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleEscherichia coli K-12Potency0.707910
1-[3-[(8-methyl-5H-pyrimido[5,4-b]indol-4-yl)amino]propyl]-2-pyrrolidinoneEscherichia coli K-12Potency7.079510
4-(1H-benzimidazol-2-ylmethylthio)-2-methylbenzofuro[3,2-d]pyrimidineEscherichia coli K-12Potency39.810710
2-(1,3-benzoxazol-2-ylamino)-5-spiro[1,6,7,8-tetrahydroquinazoline-4,1'-cyclopentane]oneEscherichia coli K-12Potency2.818410
5-[4-(diphenylmethyl)-1-piperazinyl]-2-(2-methoxyphenyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency1.778310
2-(2-methoxyphenyl)-5-[2-(4-methoxyphenyl)ethylamino]-4-oxazolecarbonitrileEscherichia coli K-12Potency1.412510
5-(4-methyl-1-piperidinyl)-2-(1-naphthalenylmethyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency0.631010
2-(2-furanyl)-5-[4-(phenylmethyl)-1-piperazinyl]-4-oxazolecarbonitrileEscherichia coli K-12Potency89.125110
3-[[2-[1,3-benzodioxol-5-yl(ethyl)amino]-1-oxoethyl]amino]-5-chloro-1H-indole-2-carboxylic acid methyl esterEscherichia coli K-12Potency14.125410
5-[(4-fluorophenyl)methylamino]-2-(2-methoxyphenyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency4.466810
LSM-28231Escherichia coli K-12Potency3.548110
N-[7-(4-chlorophenyl)-5-(4-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-2-methoxyacetamideEscherichia coli K-12Potency13.721420
1-[1-(3-fluorophenyl)-2,5-dioxo-3-pyrrolidinyl]-4-piperidinecarboxamideEscherichia coli K-12Potency3.981110
5-[2-(3,4-dimethoxyphenyl)ethylamino]-2-(1-naphthalenylmethyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency35.481310
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(4-methylphenyl)-2-oxolanecarboxamideEscherichia coli K-12Potency28.183810
2,6-dimethyl-4-(1-phenyl-4-pyrazolyl)furo[2,3-d]pyrimidineEscherichia coli K-12Potency39.810710
N-[5-(3,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-yl]carbamic acid ethyl esterEscherichia coli K-12Potency1.258910
5,8-dichloro-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-oneEscherichia coli K-12Potency4.466810
1-[(4-fluorophenyl)methyl]-3-(2-furanylmethyl)-4-imino-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-2-oneEscherichia coli K-12Potency39.810710
N-(1,7-dimethyl-3-pyrazolo[3,4-b]quinolinyl)acetamideEscherichia coli K-12Potency44.668410
9,10-dimethoxy-2-(2-pyridinylmethylamino)-6,7-dihydropyrimido[6,1-a]isoquinolin-4-oneEscherichia coli K-12Potency3.981110
N-(1-ethyl-6-methyl-3-pyrazolo[3,4-b]quinolinyl)-4-pyridinecarboxamideEscherichia coli K-12Potency39.810710
(3aR,6aS)-3-(2-chlorophenyl)-5-(2,5-dimethoxyphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dioneEscherichia coli K-12Potency1.778310
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterEscherichia coli K-12Potency0.232830
Glyceryl lactopalmitateEscherichia coli K-12Potency56.234110
9-chloro-3-[(1-ethyl-2-pyrrolidinyl)methyl]-5H-pyrimido[5,4-b]indol-4-oneEscherichia coli K-12Potency100.000010
3-[[2-(3,5-dimethyl-1-pyrazolyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]amino]-1-propanolEscherichia coli K-12Potency39.810710
3-[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]-N-ethylpropanamideEscherichia coli K-12Potency60.374020
2-[(2,5-dimethyl-3-phenyl-7-pyrazolo[1,5-a]pyrimidinyl)thio]acetonitrileEscherichia coli K-12Potency39.810710
N-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-2-thiophenecarboxamideEscherichia coli K-12Potency5.011910
LSM-32980Escherichia coli K-12Potency112.202010
7-(3-chlorophenyl)-2-(4-phenyl-1-piperazinyl)-7,8-dihydro-6H-quinazolin-5-oneEscherichia coli K-12Potency44.668410
[2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl]-(1-pyrrolidinyl)methanoneEscherichia coli K-12Potency20.220820
2-[[3-[4-(dimethylamino)phenyl]-4,5-dihydroisoxazol-5-yl]methyl]-1,1-dioxo-1,2-benzothiazol-3-oneEscherichia coli K-12Potency2.238710
N5,N5-dimethyl-2,1,3-benzoxadiazole-4,5-diamineEscherichia coli K-12Potency100.000010
3-[(3aR,6aS)-6'-chloro-5-(4-chlorophenyl)-7'-methyl-2',4,6-trioxo-1-spiro[1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3,3'-1H-indole]yl]propanamideEscherichia coli K-12Potency35.481310
N-(4,6-dimethyl-2-pyrimidinyl)-1,3-bis(phenylmethyl)-2,4-dihydro-1,3,5-triazin-6-amineEscherichia coli K-12Potency39.810710
3-[4,8-dimethyl-2-oxo-7-(2H-tetrazol-5-ylmethoxy)-1-benzopyran-3-yl]propanoic acid ethyl esterEscherichia coli K-12Potency25.118910
7-(3,4-dimethoxyphenyl)-4-methyl-2-[4-(phenylmethyl)-1-piperazinyl]-7,8-dihydro-6H-quinazolin-5-oneEscherichia coli K-12Potency14.125410
4-[[1-oxo-2-(3-oxo-2-thiomorpholinyl)ethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency39.810710
7-butyl-8-[[4-(3-chlorophenyl)-1-piperazinyl]methyl]-1,3-dimethylpurine-2,6-dioneEscherichia coli K-12Potency5.623410
2-methyl-3-phenyl-5-propyl-7-[4-(2-pyridinyl)-1-piperazinyl]pyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency0.842820
3,4,7-trimethyl-5-(3-oxobutan-2-yloxy)-1-benzopyran-2-oneEscherichia coli K-12Potency4.466810
3-(1-benzotriazolylmethyl)-6-(2-phenylethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleEscherichia coli K-12Potency89.125110
4-(1-benzotriazolyl)-5-(2-methoxyphenoxy)benzene-1,2-dicarbonitrileEscherichia coli K-12Potency56.234110
6-amino-4-(4-fluorophenyl)-3-methyl-1-phenyl-5-pyrazolo[3,4-b]pyridinecarbonitrileEscherichia coli K-12Potency3.548110
N-[4-(4-oxo-2,3-dihydro-1,3-benzoxazin-2-yl)phenyl]acetamideEscherichia coli K-12Potency7.079510
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamideEscherichia coli K-12Potency71.912420
(3aR,6aS)-3-(3,4-dimethoxyphenyl)-5-(2,4-dimethylphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dioneEscherichia coli K-12Potency44.668410
1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-2-phenyl-1-butanoneEscherichia coli K-12Potency112.202010
6-amino-1-(4-fluorophenyl)-3-methyl-4-thiophen-2-yl-5-pyrazolo[3,4-b]pyridinecarbonitrileEscherichia coli K-12Potency2.238710
5-(1,3-benzodioxol-5-ylmethylamino)-2-(4-morpholinyl)benzoic acid methyl esterEscherichia coli K-12Potency2.238710
4-(3,4-dihydro-2H-quinolin-1-yl)-6-[(4-phenyl-1-piperazinyl)methyl]-1,3,5-triazin-2-amineEscherichia coli K-12Potency17.782810
3-(1-benzimidazolylmethyl)-6-[(4-methoxyphenoxy)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleEscherichia coli K-12Potency1.122010
2-methoxy-1-(1-methyl-2-benzimidazolyl)-1-phenylethanamineEscherichia coli K-12Potency0.631010
5-[(2-chloro-6-fluorophenyl)methyl]-N-[2-[4-(4-methoxyphenyl)-1-piperazinyl]ethyl]-1,3,4-oxadiazole-2-carboxamideEscherichia coli K-12Potency0.707910
LSM-33283Escherichia coli K-12Potency0.891310
4-[(4-ethyl-1-piperazinyl)methyl]-5,7-dimethyl-1-benzopyran-2-oneEscherichia coli K-12Potency5.011910
2-ethyl-3-[(4-methoxyphenyl)methyl][1]benzopyrano[2,3-d]pyrimidine-4,5-dioneEscherichia coli K-12Potency1.584910
chlorprothixeneEscherichia coli K-12Potency25.118910
dienestrolEscherichia coli K-12Potency0.316210
mercaptopurineEscherichia coli K-12Potency35.481310
dexketoprofenEscherichia coli K-12Potency70.794610
4-cyclohexyl-3-[(3-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency44.668410
N-(4-phenylmethoxyphenyl)methanesulfonamideEscherichia coli K-12Potency0.794310
(3,4-dimethylphenyl)-(4-phenyl-1-piperazinyl)methanoneEscherichia coli K-12Potency7.943310
N-(1,3-dioxo-2-phenyl-5-isoindolyl)-2-thiophenecarboxamideEscherichia coli K-12Potency25.118910
1-(4-amino-2-methyl-3-quinolinyl)ethanoneEscherichia coli K-12Potency0.631010
2-[(2-ethoxy-2-oxoethyl)thio]-1-benzimidazolecarboxylic acid ethyl esterEscherichia coli K-12Potency89.125110
N-(2-fluorophenyl)-4-phenylmethoxybenzamideEscherichia coli K-12Potency1.584910
N-[4-(diethylamino)phenyl]-2-furancarboxamideEscherichia coli K-12Potency100.000010
6-methyl-2-(trifluoromethyl)-3,5-dihydroimidazo[4,5-f]benzimidazoleEscherichia coli K-12Potency1.000010
2-(4-bromophenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency2.511910
1-(1,3-benzodioxol-5-ylmethyl)-3-(4-methylphenyl)thioureaEscherichia coli K-12Potency89.125110
4,6-dimethyl-N-phenyl-2-quinolinamineEscherichia coli K-12Potency2.238710
6-methoxy-2-(4-methoxyphenyl)-1-benzopyran-4-oneEscherichia coli K-12Potency1.778310
5-(4-methoxyphenyl)-1,2-dihydro-1,2,4-triazole-3-thioneEscherichia coli K-12Potency112.202010
isatin beta-thiosemicarbazoneEscherichia coli K-12Potency0.707910
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-(phenoxymethyl)-4-triazolecarboxylic acid ethyl esterEscherichia coli K-12Potency0.631010
3-(diethylsulfamoyl)-N-(1,3,4-thiadiazol-2-yl)benzamideEscherichia coli K-12Potency12.589310
N-[(2-phenylethylamino)-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency89.125110
N-[2-(1-cyclohexenyl)ethyl]-4-fluorobenzamideEscherichia coli K-12Potency2.818410
4-cyclohexyl-3-(3-pyridinyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency2.818410
N4-(3-chlorophenyl)-6-methyl-N2-(phenylmethyl)pyrimidine-2,4-diamineEscherichia coli K-12Potency2.818410
1-(3-amino-4,6-dimethyl-2-thieno[2,3-b]pyridinyl)ethanoneEscherichia coli K-12Potency6.309610
ondansetron, (s)-isomerEscherichia coli K-12Potency100.000010
2,6-dimethyl-N-(4-methylphenyl)-4-quinolinamineEscherichia coli K-12Potency0.631010
2-[(4-chloro-2-methylphenoxy)methyl]imidazo[1,2-a]pyrimidineEscherichia coli K-12Potency56.234110
6-bromo-5-hydroxy-2-methyl-1H-indole-3-carboxylic acid ethyl esterEscherichia coli K-12Potency44.668410
4-chloro-1-methyl-3-nitro-2-quinolinoneEscherichia coli K-12Potency28.183810
5-(4-chlorophenyl)-3H-thieno[2,3-d]pyrimidine-4-thioneEscherichia coli K-12Potency8.912510
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterEscherichia coli K-12Potency25.118910
1-(1,3-benzodioxol-5-yl)-4-hydroxy-3-pyrazolecarboxylic acid ethyl esterEscherichia coli K-12Potency39.810710
5-(2-phenyl-4-triazolyl)-2H-tetrazoleEscherichia coli K-12Potency2.511910
2-mercaptobenzimidazoleEscherichia coli K-12Potency12.589310
N-cyclohexyl-2,3-dihydroindole-1-carboxamideEscherichia coli K-12Potency1.584910
3-[1-(carboxymethyl)-5-phenyl-2-pyrrolyl]propanoic acidEscherichia coli K-12Potency70.794610
N-[2-(1H-benzimidazol-2-yl)ethyl]-4-chloro-3-nitrobenzamideEscherichia coli K-12Potency0.631010
2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-4,6-dimethyl-3-pyridinecarbonitrileEscherichia coli K-12Potency44.668410
3-methyl-2-[2-(4-methyl-5-thiazolyl)ethylthio]-4-quinazolinoneEscherichia coli K-12Potency6.309610
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-thiophenesulfonamideEscherichia coli K-12Potency2.511910
5-(4-cyclohexylphenyl)-1,2-dihydropyrazol-3-oneEscherichia coli K-12Potency14.125410
N-cyclopentyl-2-[[1-(2-methoxyphenyl)-5-tetrazolyl]thio]acetamideEscherichia coli K-12Potency100.000010
2-methoxy-6-[[(1-methyl-2-benzimidazolyl)amino]methyl]phenolEscherichia coli K-12Potency14.125410
2-(3-oxo-2-phenyl-1H-pyrazol-5-yl)acetic acid methyl esterEscherichia coli K-12Potency89.125110
4-(4-chlorophenyl)-3-(2-quinolinyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency89.125110
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileEscherichia coli K-12Potency100.000010
4-chloro-N-(3,4,5-trimethoxyphenyl)-5-dithiazolimineEscherichia coli K-12Potency63.095710
[4-[oxo(thiophen-2-yl)methyl]-1-piperazinyl]-(3-pyridinyl)methanoneEscherichia coli K-12Potency1.412510
(3,5-dimethoxyphenyl)-(4-methylsulfonyl-1-piperazinyl)methanoneEscherichia coli K-12Potency2.818410
10-methyl-3-phenothiazinamineEscherichia coli K-12Potency1.000010
2-[[2-furanyl(oxo)methyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency0.891310
3-fluoro-7-methyl-2-imidazo[1,2-a]pyridinecarboxylic acid methyl esterEscherichia coli K-12Potency1.412510
5-amino-3-(4-methoxyphenyl)-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid ethyl esterEscherichia coli K-12Potency1.932120
3-(1-azepanyl)-4-chloro-1-(2-methylphenyl)pyrrole-2,5-dioneEscherichia coli K-12Potency17.782810
vu0038882Escherichia coli K-12Potency14.407420
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-methoxybenzamideEscherichia coli K-12Potency3.981110
N-(1,2-dihydroacenaphthylen-5-yl)methanesulfonamideEscherichia coli K-12Potency0.631010
4-Acetyl-3-methyl-5-(methylthio)thiophene-2-carboxylic acidEscherichia coli K-12Potency0.707910
N-methyl-N-phenylthioureaEscherichia coli K-12Potency39.810710
N,N-diethyl-2-oxo-1H-benzo[cd]indole-6-sulfonamideEscherichia coli K-12Potency2.238710
spiro[1,3-dihydroperimidine-2,1'-cycloheptane]Escherichia coli K-12Potency1.258910
5-amino-3-(4-methoxyphenyl)-7-methyl-4-oxo-1-thieno[3,4-d]pyridazinecarboxylic acid methyl esterEscherichia coli K-12Potency7.079510
1-[4-(4-aminophenyl)-1-piperazinyl]ethanoneEscherichia coli K-12Potency39.810710
3-(2-Methyl-1,3-thiazol-4-yl)anilineEscherichia coli K-12Potency18.966220
2-amino-4-(2-furanyl)-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency44.668410
N,N-dimethyl-N'-p-tolylsulfamideEscherichia coli K-12Potency100.000010
1-(3-fluorophenyl)-3-(2-pyridinylmethyl)thioureaEscherichia coli K-12Potency3.162310
N-[[(6-methyl-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-thiophenecarboxamideEscherichia coli K-12Potency44.668410
2-(4-hydroxyanilino)-1,4-naphthoquinoneEscherichia coli K-12Potency89.125110
N-(2-phenyl-3-imidazo[1,2-a]pyridinyl)carbamic acid methyl esterEscherichia coli K-12Potency1.584910
3-[[(5-bromo-3-pyridinyl)-oxomethyl]amino]propanoic acidEscherichia coli K-12Potency79.432810
1-(cyclohexylmethyl)-4-phenylpiperazineEscherichia coli K-12Potency0.316210
acetic acid [4-[oxo-(2-phenylethylamino)methyl]phenyl] esterEscherichia coli K-12Potency31.622810
3-(4-methoxyphenyl)-2,5-dimethyl-7-phenylpyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency44.668410
3-[(4,8-dimethyl-2-quinolinyl)thio]propanoic acidEscherichia coli K-12Potency0.631010
N-(3-methoxyphenyl)-2-benzo[cd]indolamineEscherichia coli K-12Potency79.432810
(5-hydroxy-2-phenyl-3-benzofuranyl)-(4-morpholinyl)methanoneEscherichia coli K-12Potency22.387210
N-(4-hydroxy-2-methyl-5-propan-2-ylphenyl)benzenesulfonamideEscherichia coli K-12Potency5.011910
N-(3-chloro-4-hydroxy-2,5-dimethylphenyl)benzenesulfonamideEscherichia coli K-12Potency3.981110
3,4,5-trimethoxybenzoic acid [(3,5-dimethyl-4-oxo-1-cyclohexa-2,5-dienylidene)amino] esterEscherichia coli K-12Potency1.412510
2-[[(4-chlorophenyl)thio]methyl]imidazo[1,2-a]pyridineEscherichia coli K-12Potency12.589310
N2,N4-ditert-butyl-6-hydrazinyl-1,3,5-triazine-2,4-diamineEscherichia coli K-12Potency100.000010
nsc185058Escherichia coli K-12Potency14.348420
2-amino-4-thiophen-2-yl-5,6,7,8-tetrahydroquinoline-3-carbonitrileEscherichia coli K-12Potency100.000010
vu0099704Escherichia coli K-12Potency0.707910
2-(4-fluorophenyl)-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidineEscherichia coli K-12Potency50.118710
2-[(6-amino-3,5-dicyano-2-pyridinyl)thio]acetic acid ethyl esterEscherichia coli K-12Potency6.309610
6-methoxy-3-phenyl-[1,2,4]triazolo[4,3-b]pyridazineEscherichia coli K-12Potency0.891310
2-(5,7-dimethyl-3-phenyl-6-pyrazolo[1,5-a]pyrimidinyl)acetic acid ethyl esterEscherichia coli K-12Potency31.622810
4-(1-ethyl-2-benzimidazolyl)anilineEscherichia coli K-12Potency3.162310
3-(2,3-dimethyl-1H-indol-5-yl)-4-methyl-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency16.126920
4-(2-furanylmethyl)-3-pyridin-4-yl-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency0.707910
3-(4-bromophenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneEscherichia coli K-12Potency0.794310
6-methyl-4-(trifluoromethyl)-7,8,9,10-tetrahydropyrano[2,3-f]quinolin-2-oneEscherichia coli K-12Potency44.668410
N-[4-[oxo(1-piperidinyl)methyl]phenyl]-2-thiophenecarboxamideEscherichia coli K-12Potency0.707910
1-[(3,4-dimethoxyphenyl)methyl]-4-(2,3-dimethylphenyl)piperazineEscherichia coli K-12Potency28.183810
(3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolyl)-(3-methyl-1-pyrazolyl)methanoneEscherichia coli K-12Potency44.668410
N-(4-methyl-2-thiazolyl)-3-(2-oxo-1,3-benzothiazol-3-yl)propanamideEscherichia coli K-12Potency1.258910
1-(3-((2',4'-Dimethyl-[4,5'-bithiazol]-2-yl)amino)phenyl)ethanoneEscherichia coli K-12Potency39.810710
N-[[(2-chloro-3-pyridinyl)amino]-sulfanylidenemethyl]-2-furancarboxamideEscherichia coli K-12Potency5.011910
4-(4-chlorophenyl)-3-[(4-methylphenoxy)methyl]-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency8.912510
N-[3-chloro-4-(1-pyrrolidinyl)phenyl]-2-furancarboxamideEscherichia coli K-12Potency158.489010
4-(6-methyl-4-phenyl-2-quinazolinyl)-1-piperazinecarboxaldehydeEscherichia coli K-12Potency43.928420
6-chloro-N4-cyclohexyl-N2-propan-2-yl-1,3,5-triazine-2,4-diamineEscherichia coli K-12Potency12.589310
2-(8-quinolinylthio)acetic acid phenacyl esterEscherichia coli K-12Potency8.912510
4-methyl-N-[1-[2-(1-pyrrolidinyl)ethyl]-2-benzimidazolyl]benzamideEscherichia coli K-12Potency79.432810
1-(3-nitrophenyl)-3-phenyl-2-propyn-1-oneEscherichia coli K-12Potency15.848910
1-spiro[2,4-dihydroisoquinoline-3,1'-cyclohexane]thioneEscherichia coli K-12Potency0.707910
4-(2-naphthalenylmethyl)-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency0.562310
2-[(3-fluorophenyl)methyl-(phenylmethyl)amino]ethanolEscherichia coli K-12Potency0.707910
2-methoxy-4-[[2-(methylthio)anilino]methyl]phenolEscherichia coli K-12Potency1.584910
6-(4-morpholinyl)naphthalene-2,3-dicarbonitrileEscherichia coli K-12Potency89.125110
2-(1,4,5,7-tetramethyl-6-pyrrolo[3,4-d]pyridazinyl)anilineEscherichia coli K-12Potency22.387210
2-(phenylmethylthio)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoleEscherichia coli K-12Potency1.122010
N-(1-acetyl-2-chloro-3-indolyl)-2-chloroacetamideEscherichia coli K-12Potency35.481310
1-[4-[[6-methyl-2-(methylthio)-5-prop-2-enyl-4-pyrimidinyl]amino]phenyl]ethanoneEscherichia coli K-12Potency6.309610
1-(4-methoxyphenyl)-3-(6-methyl-2-pyridinyl)ureaEscherichia coli K-12Potency0.316210
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrileEscherichia coli K-12Potency2.511910
(4-methoxyphenyl)-(3-methyl-2-propyl-4-imidazolyl)methanoneEscherichia coli K-12Potency0.631010
3-chloro-6-phenyl-[1,2,4]triazolo[4,3-b]pyridazineEscherichia coli K-12Potency31.622810
N-[5-(phenylmethyl)-1,3,4-thiadiazol-2-yl]carbamic acid methyl esterEscherichia coli K-12Potency1.122010
3-(5-methoxy-2,2-dimethyl-1-benzopyran-8-yl)-3-oxopropanoic acidEscherichia coli K-12Potency44.668410
3-chloro-1-(2-chlorophenyl)-4-(4-morpholinyl)pyrrole-2,5-dioneEscherichia coli K-12Potency44.668410
N-(1-naphthalenyl)-4-(phenylmethyl)-1-piperazinecarboxamideEscherichia coli K-12Potency7.943310
N-[[(4,6-dimethyl-2-pyrimidinyl)amino]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency0.316210
1-(4-ethoxyphenyl)-3-(6-quinoxalinyl)ureaEscherichia coli K-12Potency0.631010
3-[2-(4-fluorophenyl)-5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]propanoic acid ethyl esterEscherichia coli K-12Potency100.000010
2-(dimethylsulfamoylamino)-9H-fluoreneEscherichia coli K-12Potency1.778310
N-[4-(4-morpholinylazo)phenyl]acetamideEscherichia coli K-12Potency89.125110
2,3,4-trimethyl-N-(3-pyridinyl)benzenesulfonamideEscherichia coli K-12Potency7.079510
N-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-2,2,2-trichloroacetamideEscherichia coli K-12Potency100.000010
N-[(4-fluorophenyl)methyl]-2-thiophen-2-ylacetamideEscherichia coli K-12Potency89.125110
3-(4-chlorophenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneEscherichia coli K-12Potency3.548110
N-(2,4-difluorophenyl)-3-methoxybenzamideEscherichia coli K-12Potency56.234110
3-phenyl-5,6,7,8-tetrahydro-1H-pyrazolo[5,1-b]quinazolin-9-oneEscherichia coli K-12Potency0.354810
4-(5-methoxy-1,2-dimethyl-3-indolyl)-2-thiazolamineEscherichia coli K-12Potency44.668410
1-(4-bromophenyl)-3-(2-phenylethyl)thioureaEscherichia coli K-12Potency10.000010
5-bromo-N-[(2-pyridinylamino)-sulfanylidenemethyl]-3-pyridinecarboxamideEscherichia coli K-12Potency8.912510
3-bromo-N-(2-furanylmethyl)benzamideEscherichia coli K-12Potency5.011910
8-methyl-1,5-dihydropyrimido[5,4-b]indole-4-thioneEscherichia coli K-12Potency1.258910
3-methyl-7-(phenylmethyl)-8-(propan-2-ylthio)purine-2,6-dioneEscherichia coli K-12Potency28.183810
2-methyl-5-(1-pyrrolidinyl)isoindole-1,3-dioneEscherichia coli K-12Potency2.511910
2-oxo-N-(2-thiazolyl)-1H-pyridine-3-carboxamideEscherichia coli K-12Potency7.943310
N-methyl-2-(4-methylphenyl)-N-(1-methylpiperidin-4-yl)quinazolin-4-amineEscherichia coli K-12Potency28.183810
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideEscherichia coli K-12Potency89.125110
6-methyl-4-oxoquinolizine-1,3-dicarboxylic acid diethyl esterEscherichia coli K-12Potency7.943310
4,7-dimethoxy-1-methyl-2-quinolinoneEscherichia coli K-12Potency28.183810
7-chloro 5-(2-chlorophenyl)-1,3-dihydro-2h-(1,4)-benzodiazepine-2-thioneEscherichia coli K-12Potency0.707910
2-(2-furanyl)-3-(6-methyl-2-pyridinyl)-4-quinazolinoneEscherichia coli K-12Potency112.202010
4-[(4-chlorophenyl)thio]-5-methyl-2-phenyl-1H-pyrazol-3-oneEscherichia coli K-12Potency0.707910
N-(1-tert-butyl-5-benzimidazolyl)-2-thiophenecarboxamideEscherichia coli K-12Potency1.778310
5-[anilino(oxo)methyl]-4-methyl-2-(1-oxopropylamino)-3-thiophenecarboxylic acid methyl esterEscherichia coli K-12Potency39.810710
1-[[4-(2-pyridinyl)-1-piperazinyl]methyl]-2-benzo[cd]indoloneEscherichia coli K-12Potency15.848910
2-(3-methyl-2-oxo-1-benzimidazolyl)acetonitrileEscherichia coli K-12Potency56.234110
1-(2-fluoro-5-nitrophenyl)-3-phenylureaEscherichia coli K-12Potency2.238710
2-propyl-5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazoleEscherichia coli K-12Potency39.810710
N-[5-(methylthio)-1,3,4-thiadiazol-2-yl]-3-phenylpropanamideEscherichia coli K-12Potency2.511910
3-ethoxy-N-[(3-pyridinylamino)-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency1.412510
2-phenyl-1H-quinazoline-4-thioneEscherichia coli K-12Potency31.622810
6,7,8,9-tetrahydro-5H-carbazole-3-carbohydrazideEscherichia coli K-12Potency25.118910
N-[4-(4-chlorophenyl)-3,5-dimethyl-2-thiazolylidene]-2-furancarboxamideEscherichia coli K-12Potency89.125110
2-(4-nitro-2-pyridinyl)isoindole-1,3-dioneEscherichia coli K-12Potency5.011910
3-[[(3-chloro-4-ethoxyphenyl)-oxomethyl]amino]benzoic acidEscherichia coli K-12Potency70.794610
1-azepanyl-(4-methoxyphenyl)methanethioneEscherichia coli K-12Potency5.011910
N-(4,5-dihydrothiazol-2-yl)-1-ethyl-3-pyrazolecarboxamideEscherichia coli K-12Potency79.432810
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]acetamideEscherichia coli K-12Potency2.238710
3,4-dichloro-N-[(1-methyl-4-pyrazolyl)methyl]-1-benzothiophene-2-carboxamideEscherichia coli K-12Potency39.810720
1-[[(1,5-dimethyl-3-pyrazolyl)-oxomethyl]amino]-3-(2-methoxyphenyl)thioureaEscherichia coli K-12Potency35.481310
1-(2-methylphenyl)-3-[[(5-methyl-3-thiophenyl)-oxomethyl]amino]thioureaEscherichia coli K-12Potency1.000010
3-(1-benzothiophen-3-yl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency112.202010
4-(3-methylphenyl)-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency35.481310
3-(4,5-dimethyl-3-thiophenyl)-4-(2-methylphenyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency23.753120
4-(phenylmethyl)-3-(5-propyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency3.981110
1-cyclohexyl-3-(2,3-dihydro-1,4-benzodioxin-6-yl)ureaEscherichia coli K-12Potency50.118710
4,5-dimethyl-2-[4-(3-nitrophenyl)-2-thiazolyl]-1H-pyrazol-3-oneEscherichia coli K-12Potency20.466320
2-(4-fluoro-N-methylsulfonylanilino)-N-(3-methylphenyl)acetamideEscherichia coli K-12Potency15.848910
LSM-31933Escherichia coli K-12Potency1.000010
1-(4-methoxyphenyl)-3-[[oxo(thiophen-2-yl)methyl]amino]thioureaEscherichia coli K-12Potency1.412510
2-(3-methoxyphenyl)-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazoleEscherichia coli K-12Potency100.000010
2-methoxy-3-methyl-N-[4-(4-morpholinylmethyl)phenyl]benzamideEscherichia coli K-12Potency5.011910
4,4-dicarboxy-5-pyridoxylprolineEscherichia coli K-12Potency44.668410
N,N-dimethylcarbamic acid [4-[6-(trifluoromethyl)-2-imidazo[1,2-a]pyridinyl]phenyl] esterEscherichia coli K-12Potency1.584910
N-[[6-cyano-5-(ethylamino)-3-methyl-2-pyrazinyl]methyl]-N-phenylacetamideEscherichia coli K-12Potency44.668410
N-(6-chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-3-phenylpropanamideEscherichia coli K-12Potency44.668410
5-methyl-N-(5-methyl-3-isoxazolyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency0.707910
5-(4-methylphenyl)-2-phenyl-3-pyrazolamineEscherichia coli K-12Potency89.125110
5-[2-(6-hydroxy-3-methyl-2-benzofuranyl)-2-oxoethyl]-2-furancarboxylic acid ethyl esterEscherichia coli K-12Potency0.631010
3-methyl-5-propyl-7-furo[3,2-g][1]benzopyranoneEscherichia coli K-12Potency1.000010
2-[(3-methyl-4-oxo-2-quinazolinyl)thio]-N-phenylacetamideEscherichia coli K-12Potency2.818410
5-methyl-N-(3-pyridinyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency1.995310
N-(4-fluorophenyl)-1-(3-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinamineEscherichia coli K-12Potency7.943310
5-(3,5-dimethoxyphenyl)-3-phenyl-1,2,4-oxadiazoleEscherichia coli K-12Potency0.707910
N,N-diethyl-4-[oxo-(2,4,6-trimethylphenyl)methyl]benzamideEscherichia coli K-12Potency19.952610
N-(4-methoxyphenyl)-3-methyl-2-quinoxalinamineEscherichia coli K-12Potency0.891310
N'-[(4-chlorophenyl)-oxomethyl]-2-hydroxy-3-methylbenzohydrazideEscherichia coli K-12Potency56.234110
(4-(3-chlorophenyl)piperazin-1-yl)(2-ethoxyphenyl)methanoneEscherichia coli K-12Potency69.905420
1-(3,4-dimethoxyphenyl)-1-cyclohexanecarboxamideEscherichia coli K-12Potency89.125110
5-(1-methyl-2-benzimidazolyl)-2-thiophenecarboxaldehydeEscherichia coli K-12Potency0.631010
6,7-dimethoxy-3-phenyl-1H-quinazoline-2,4-dioneEscherichia coli K-12Potency0.707910
1-(1-azepanyl)-2-(4-bromophenyl)ethanoneEscherichia coli K-12Potency44.668410
2-methoxy-4-prop-1-enylphenyl acetateEscherichia coli K-12Potency0.223910
4-(4-morpholinylmethyl)-3-quinolinolEscherichia coli K-12Potency70.794610
2-amino-9-ethyl-3-pyrido[2,3-b]indolecarboxylic acid ethyl esterEscherichia coli K-12Potency100.000010
1-(4-chlorophenyl)-3-(2-phenylethyl)thioureaEscherichia coli K-12Potency0.354810
4-sulfanylidene-1,6,7,8,9,10-hexahydropyrimido[3,4]pyrrolo[3,5-a]azepine-11-carbonitrileEscherichia coli K-12Potency31.622810
5-(4-chlorophenyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-furancarboxamideEscherichia coli K-12Potency44.668410
n-(2-methoxybenzyl)-2-(phenylthio)acetamideEscherichia coli K-12Potency0.707910
3-bromo-N-[(tert-butylamino)-sulfanylidenemethyl]-4-methoxybenzamideEscherichia coli K-12Potency0.794310
N-(1,3-benzodioxol-5-yl)-4-(4-morpholinylmethyl)benzamideEscherichia coli K-12Potency39.810710
4-[(2-ethyl-1-oxobutyl)amino]benzoic acid ethyl esterEscherichia coli K-12Potency0.562310
N-(2-fluoro-5-nitrophenyl)-2,2-dimethylbutanamideEscherichia coli K-12Potency31.622810
4-chloro-N-[4-(2-imidazo[1,2-a]pyridinyl)phenyl]benzamideEscherichia coli K-12Potency35.481310
3,4,5-triethoxy-N-(1H-1,2,4-triazol-5-yl)benzamideEscherichia coli K-12Potency19.952610
4-(1,3-benzothiazol-2-yl)-N-phenyl-1-piperazinecarboxamideEscherichia coli K-12Potency89.125110
lupitidineEscherichia coli K-12Potency5.011910
3-[[[3-(4-methoxyphenyl)phenyl]-oxomethyl]amino]benzoic acidEscherichia coli K-12Potency89.125110
[4-amino-3-(4-methylphenyl)-2-sulfanylidene-5-thiazolyl]-(4-morpholinyl)methanoneEscherichia coli K-12Potency19.952610
N-(1,3-dimethyl-2-oxo-5-benzimidazolyl)-2-benzofurancarboxamideEscherichia coli K-12Potency100.000010
N-[(2-methoxyphenyl)methyl]-4-(1-piperidinyl)anilineEscherichia coli K-12Potency79.432810
2-(4-methoxyphenyl)-5-(2-phenylethylamino)-4-oxazolecarbonitrileEscherichia coli K-12Potency89.125110
1-cyclopentyl-3-(4-phenoxyphenyl)thioureaEscherichia coli K-12Potency3.981110
5-(2-furanylmethylamino)-2-(2-methylphenyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency22.387210
N-[3-[(1,3-dioxo-5-isoindolyl)oxy]phenyl]-2-furancarboxamideEscherichia coli K-12Potency0.141310
4-phenyl-N-(2-propyl-5-tetrazolyl)benzamideEscherichia coli K-12Potency2.818410
3-[5-(4-fluorophenyl)-1-(2-furanylmethyl)-2-pyrrolyl]propanoic acidEscherichia coli K-12Potency5.011910
1-(4-methoxyphenyl)-1-methyl-3-(1-methyl-5-benzotriazolyl)ureaEscherichia coli K-12Potency1.258910
N-[3-[methyl(methylsulfonyl)amino]phenyl]-2-phenoxyacetamideEscherichia coli K-12Potency100.000010
3-[1-(4-acetylphenyl)-5-thiophen-2-yl-2-pyrrolyl]propanoic acidEscherichia coli K-12Potency3.548110
4-acetamidobenzoic acid (2-chlorophenyl)methyl esterEscherichia coli K-12Potency89.125110
N-(4-phenylmethoxyphenyl)carbamic acid methyl esterEscherichia coli K-12Potency1.412510
1-[(4-methylphenyl)methyl]-4-(1-pyrrolidinyl)pyrazolo[3,4-d]pyrimidineEscherichia coli K-12Potency100.000010
(5-amino-3-phenyl-1,2,4-triazol-1-yl)-(2-methoxyphenyl)methanoneEscherichia coli K-12Potency19.952610
1-cyclohexyl-3-(3-ethylphenyl)ureaEscherichia coli K-12Potency3.981110
[2-(5-methyl-2-thiophenyl)-4-quinolinyl]-(1-pyrrolidinyl)methanoneEscherichia coli K-12Potency28.183810
4-tert-butyl-N-(4-methyl-3-nitrophenyl)benzamideEscherichia coli K-12Potency19.952610
5-amino-3-ethyl-1-phenyl-4-pyrazolecarbonitrileEscherichia coli K-12Potency100.000010
N-(3-methyl-4-oxo-1-benzopyran-2-yl)carbamic acid ethyl esterEscherichia coli K-12Potency0.631010
2-[2-bromo-4-(hydroxymethyl)-6-methoxyphenoxy]acetic acidEscherichia coli K-12Potency2.818410
1,3-benzothiazol-2-yl-[4-(2-pyridinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency100.000010
N-(3,4-dimethyl-2-thiazolylidene)benzamideEscherichia coli K-12Potency79.432810
2-(2-methoxyphenyl)-1H-indoleEscherichia coli K-12Potency79.432810
2-(2,6-dichloroanilino)-3-pyridinesulfonamideEscherichia coli K-12Potency3.162310
6-(2-oxopropylthio)-3-pyridinecarboxylic acidEscherichia coli K-12Potency56.234110
1-(2-hydroxyphenyl)-2-(2H-tetrazol-5-yl)ethanoneEscherichia coli K-12Potency28.183810
3-acetamidobenzoic acid [2-(2-chlorophenyl)-2-oxoethyl] esterEscherichia coli K-12Potency70.794610
N-(2,3-dihydro-1H-inden-5-yl)-2-methyl-3-nitrobenzamideEscherichia coli K-12Potency7.943310
3-(3,5-dimethyl-7-oxo-6-furo[3,2-g][1]benzopyranyl)propanoic acidEscherichia coli K-12Potency100.000010
1-(2-methyl-1H-indol-3-yl)-2-(2-thiazolylamino)ethanoneEscherichia coli K-12Potency0.707910
4-chloro-N-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]benzamideEscherichia coli K-12Potency0.631010
1-(cycloheptylideneamino)-3-(4-fluorophenyl)thioureaEscherichia coli K-12Potency31.622810
2-(4-methyl-1-piperazinyl)-6-phenyl-4-pyrimidinecarbonitrileEscherichia coli K-12Potency35.481310
2-[(3-chloro-1-benzothiophen-2-yl)methylideneamino]phenolEscherichia coli K-12Potency3.981110
N-(2-ethylphenyl)-2-methoxy-5-methylbenzenesulfonamideEscherichia coli K-12Potency1.584910
5-(2-fluorophenoxy)-1-methyl-3-nitro-1,2,4-triazoleEscherichia coli K-12Potency3.548110
3,6-dichloro-N-(3-pyridinylmethyl)-1-benzothiophene-2-carboxamideEscherichia coli K-12Potency5.623410
2-(2-fluorophenyl)-5-(4-methyl-1-piperidinyl)-4-oxazolecarbonitrileEscherichia coli K-12Potency8.421820
1-(4-methyl-1-piperidinyl)-2-[(3-methyl-2-quinoxalinyl)thio]ethanoneEscherichia coli K-12Potency16.208620
5-bromo-N-(pyridin-4-ylmethyl)-2-thiophenesulfonamideEscherichia coli K-12Potency15.848910
2-thiophenecarboxylic acid (6-methyl-2-oxo-1H-quinolin-3-yl)methyl esterEscherichia coli K-12Potency3.981110
thiothixeneEscherichia coli K-12Potency28.183810
thiothixeneEscherichia coli K-12Potency25.118910
4-(4-chlorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency3.162310
N-[[(phenylmethyl)amino]-sulfanylidenemethyl]-1,3-benzodioxole-5-carboxamideEscherichia coli K-12Potency100.000010
2-(2-ethoxyphenyl)-5,6-dimethyl-1,3-dihydroisoindoleEscherichia coli K-12Potency5.623410
N-[3-chloro-4-(1-pyrrolidinyl)phenyl]-2-nitrobenzamideEscherichia coli K-12Potency22.387210
terazosinEscherichia coli K-12Potency44.668410
1-(2,4-dichlorophenyl)-3-(1-methyl-3-pyrazolyl)ureaEscherichia coli K-12Potency8.912510
2-[[(4-methyl-1-pyrazolyl)-oxomethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency100.000010
4-(3,4-dimethoxyphenyl)-N-(3-methyl-2-pyridinyl)-2-thiazolamineEscherichia coli K-12Potency20.405420
6-hydroxy-2-(4-nitrophenyl)-3,1-benzoxazin-4-oneEscherichia coli K-12Potency25.118910
8-methoxy-N-methyl-2-oxo-1-benzopyran-3-carboxamideEscherichia coli K-12Potency31.622810
2,2-dimethyl-N-[[2-(4-methyl-1-piperidinyl)anilino]-sulfanylidenemethyl]propanamideEscherichia coli K-12Potency39.810710
4-[oxo-(pyridin-4-ylamino)methyl]-1H-imidazole-5-carboxylic acid ethyl esterEscherichia coli K-12Potency1.412510
4-methyl-6-[2-(4-methyl-1-piperidinyl)-2-oxoethoxy]-1-benzopyran-2-oneEscherichia coli K-12Potency28.183810
1-(3,4-dichlorophenyl)-3-(3,5-dimethylphenyl)thioureaEscherichia coli K-12Potency0.562310
1-phenyl-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneEscherichia coli K-12Potency44.668410
2-(2,4-dichlorophenoxy)-N-[4-(4-morpholinylmethyl)phenyl]acetamideEscherichia coli K-12Potency35.716820
N-[(3-bromo-4,5-diethoxyphenyl)methyl]-4-(4-morpholinyl)anilineEscherichia coli K-12Potency31.622810
N-[(1-ethyl-2-oxo-6-benzo[cd]indolyl)sulfonyl]-N-(4-methoxyphenyl)-3-pyridinecarboxamideEscherichia coli K-12Potency35.971320
2-[[5-[(2,6-dimethylphenoxy)methyl]-4-ethyl-1,2,4-triazol-3-yl]thio]-1-(4-phenyl-1-piperazinyl)ethanoneEscherichia coli K-12Potency31.622810
5-[(5-methoxycarbonyl-2-methyl-3-furanyl)methoxy]-2-methyl-3-benzofurancarboxylic acid methyl esterEscherichia coli K-12Potency0.707910
1-[4-(4-bromophenyl)-2-thiazolyl]-4-piperidinecarboxamideEscherichia coli K-12Potency0.631010
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideEscherichia coli K-12Potency63.095710
2-methyl-N-[2-[1-[2-(4-methylphenoxy)ethyl]-2-benzimidazolyl]ethyl]propanamideEscherichia coli K-12Potency19.622220
3-[(4-nitrophenyl)methoxy]-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-6-oneEscherichia coli K-12Potency6.309610
4-[1-oxo-2-(1-piperidinyl)ethyl]-9-phenylmethoxy-2,3-dihydro-1H-[1]benzopyrano[3,4-b]pyridin-5-oneEscherichia coli K-12Potency39.810710
N-(5-bromo-8-quinolinyl)-5-[(4-chloro-1-pyrazolyl)methyl]-2-furancarboxamideEscherichia coli K-12Potency0.050110
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamideEscherichia coli K-12Potency44.668410
2-[(5-bromo-2-thiophenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideEscherichia coli K-12Potency10.000010
5-(4-bromophenyl)-N-(2-methoxyphenyl)-2-furancarboxamideEscherichia coli K-12Potency39.810710
(4-Methoxyphenyl)-(2-methylsulfanyl-6,7-dihydro-[1,4]dioxino[2,3-f]benzimidazol-3-yl)methanoneEscherichia coli K-12Potency26.651420
4-[[5-[(3,4-dichlorophenyl)methylthio]-4-phenyl-1,2,4-triazol-3-yl]methyl]morpholineEscherichia coli K-12Potency22.387210
N-[(3-acetylanilino)-sulfanylidenemethyl]-5-bromo-3-pyridinecarboxamideEscherichia coli K-12Potency0.631010
2-(1,3-dimethyl-2,6-dioxo-9-purinyl)-N-[2-(4-morpholinyl)-5-(trifluoromethyl)phenyl]acetamideEscherichia coli K-12Potency39.810710
N-cyclohexyl-2-[[5-[(4-methoxyphenyl)methyl]-4-methyl-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency100.000010
2-(3-pyridinyl)-4-[4-(1-pyrrolidinylsulfonyl)phenyl]thiazoleEscherichia coli K-12Potency0.707910
N-[3-[oxo-(3-pyridinylmethylamino)methyl]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-furancarboxamideEscherichia coli K-12Potency39.810710
1,4-bis(thiophen-2-ylsulfonyl)piperazineEscherichia coli K-12Potency89.125110
N-(4-chlorophenyl)-7,8-dimethoxy-1-oxo-2-benzothiopyran-3-carboxamideEscherichia coli K-12Potency1.778310
5-ethyl-2-[[oxo-(3,4,5-trimethoxyphenyl)methyl]amino]-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency0.707910
2-[[3-cyano-6-(4-methylphenyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N-(4-methoxyphenyl)acetamideEscherichia coli K-12Potency5.673020
2-[[benzamido(sulfanylidene)methyl]amino]-5,5-dimethyl-4,7-dihydrothieno[2,3-c]pyran-3-carboxylic acidEscherichia coli K-12Potency89.125110
1-(2-fluorophenyl)-4-[(6-nitro-1,3-benzodioxol-5-yl)methyl]piperazineEscherichia coli K-12Potency112.202010
1-[(4-fluorophenyl)methyl]-4-(3,4,5-trimethoxyphenyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency12.840620
1-[(4-methylphenyl)methyl]-4-(3,4,5-trimethoxyphenyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency11.547620
2-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]thio]-N-(4-methyl-2-thiazolyl)acetamideEscherichia coli K-12Potency0.631010
1-methoxy-N-[4-(pyridin-4-ylmethyl)phenyl]-2-naphthalenecarboxamideEscherichia coli K-12Potency28.183810
1-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-2-[(4-chlorophenyl)methylthio]ethanoneEscherichia coli K-12Potency19.952610
1-(4-chloro-3-methoxyphenyl)sulfonyl-4-phenylpiperazineEscherichia coli K-12Potency28.183810
N-(1-tert-butyl-5-benzimidazolyl)-3,4,5-trimethoxybenzamideEscherichia coli K-12Potency56.234110
N-(4-acetamidophenyl)-2-[[1-(4-ethylphenyl)-5-tetrazolyl]thio]acetamideEscherichia coli K-12Potency112.202010
N-(2-methoxyphenyl)-5-methyl-3-[(2-methylphenyl)methyl]-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideEscherichia coli K-12Potency7.079510
4-[[[3-(4-morpholinylsulfonyl)phenyl]-oxomethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency14.125410
3-(4-methoxyphenyl)-6-phenyl-4-thieno[2,3-d]pyrimidinoneEscherichia coli K-12Potency5.889220
N-[2-(3-pyridinyl)-3H-benzimidazol-5-yl]-2-furancarboxamideEscherichia coli K-12Potency2.818410
3,4-dimethoxy-N-[4-[oxo(1-piperidinyl)methyl]phenyl]benzamideEscherichia coli K-12Potency0.707910
2-[(4-ethoxyphenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideEscherichia coli K-12Potency0.707910
4,5-dichloro-2-[oxo-(8-quinolinylamino)methyl]benzoic acidEscherichia coli K-12Potency22.387210
3-amino-N-tert-butyl-6-methyl-7,8-dihydro-5H-thieno[2,3-b][1,6]naphthyridine-2-carboxamideEscherichia coli K-12Potency63.095710
2-(2,4,5-trimethoxyphenyl)-1,3-benzothiazoleEscherichia coli K-12Potency35.481310
4-(4-methoxycarbonylphenyl)-1,2,6-trimethyl-4H-pyridine-3,5-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency79.432810
2-fluoro-N-[4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]phenyl]benzamideEscherichia coli K-12Potency1.412510
N-(1-naphthalenyl)-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineEscherichia coli K-12Potency10.000010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[2-(ethylthio)phenyl]methanoneEscherichia coli K-12Potency19.952610
N-(3-benzamidophenyl)-1,3-benzodioxole-5-carboxamideEscherichia coli K-12Potency17.782810
3-[2-(3-methylphenoxy)ethyl]-1,3-benzothiazol-2-oneEscherichia coli K-12Potency1.584910
[3-amino-4-(methoxymethyl)-6-methyl-2-thieno[2,3-b]pyridinyl]-(4-phenyl-1-piperazinyl)methanoneEscherichia coli K-12Potency14.125410
4-[(3-methyl-2-oxo-1,3-benzoxazol-6-yl)sulfonylamino]benzoic acid ethyl esterEscherichia coli K-12Potency2.818410
[4-(2-methoxyphenyl)-1-piperazinyl]-[5-(4-methylphenyl)-3-isoxazolyl]methanoneEscherichia coli K-12Potency9.150820
[4-[[5-(2,4-dichlorophenyl)-3-isoxazolyl]-oxomethyl]-1-piperazinyl]-(2-furanyl)methanoneEscherichia coli K-12Potency19.321820
7-(difluoromethyl)-N-(5-methyl-3-isoxazolyl)-5-(4-methylphenyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideEscherichia coli K-12Potency14.125410
[7-(difluoromethyl)-5-(4-methoxyphenyl)-3-pyrazolo[1,5-a]pyrimidinyl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency39.810710
2-(4-methylphenoxy)-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]acetamideEscherichia coli K-12Potency0.631010
1-[(3,4-dimethoxyphenyl)methyl]-4-(4-hydroxyphenyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency19.952610
4-chloro-2-[[(1-methyl-5-phenyl-2-imidazolyl)amino]methyl]phenolEscherichia coli K-12Potency28.183810
N2,N7-bis(2,5-dimethylphenyl)-9H-fluorene-2,7-disulfonamideEscherichia coli K-12Potency7.943310
N-(2-furanylmethyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideEscherichia coli K-12Potency19.952610
[3-bromo-5-thiophen-2-yl-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-(3,4-dihydro-2H-quinolin-1-yl)methanoneEscherichia coli K-12Potency100.000010
2-(3,4-dimethoxyphenyl)-8-methoxy-4,4-dimethyl-5H-isothiazolo[5,4-c]quinoline-1-thioneEscherichia coli K-12Potency7.079510
N-[4-[[2-(4-hydroxyphenyl)-1,3-dioxo-5-isoindolyl]oxy]phenyl]-2-thiophenecarboxamideEscherichia coli K-12Potency3.981110
3-methoxy-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)benzamideEscherichia coli K-12Potency100.000010
5-(3,4-dimethoxyphenyl)-N-(2-furanylmethyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamideEscherichia coli K-12Potency10.476320
2-furanyl-(4,4,8-trimethyl-1-sulfanylidene-5-dithiolo[3,4-c]quinolinyl)methanoneEscherichia coli K-12Potency100.000010
4-[(4-chlorophenyl)methyl-methylsulfonylamino]-N-(2-pyridinylmethyl)benzamideEscherichia coli K-12Potency19.952610
6-bromo-3-(4-morpholinyl)-4-phenyl-1H-quinolin-2-oneEscherichia coli K-12Potency4.956220
N-(3-methoxyphenyl)-4-(1-oxopropylamino)benzamideEscherichia coli K-12Potency0.707910
3-(2-chloro-6-fluorophenyl)-N-(3-fluoro-4-methylphenyl)-5-methyl-4-isoxazolecarboxamideEscherichia coli K-12Potency3.548110
1-[4-(2-pyridinyl)-1-piperazinyl]-2-(9H-xanthen-9-yl)ethanoneEscherichia coli K-12Potency14.125410
2-(1,3-benzodioxol-5-yl)-N-[(2-ethoxyphenyl)methyl]-N-(2-pyridinylmethyl)ethanamineEscherichia coli K-12Potency2.818410
6-ethyl-2-thieno[2,3-b]quinolinecarboxylic acidEscherichia coli K-12Potency31.622810
2-[(7-methoxy-4-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)thio]-N-methyl-N-(4-phenyl-2-thiazolyl)acetamideEscherichia coli K-12Potency25.118910
5-bromo-N-[3-(2-oxo-1-benzopyran-3-yl)phenyl]-2-furancarboxamideEscherichia coli K-12Potency3.981110
2-[5-(2-fluorophenyl)-2-tetrazolyl]-N-[2-oxo-2-[(phenylmethyl)amino]ethyl]-N-(5,6,7,8-tetrahydronaphthalen-1-yl)acetamideEscherichia coli K-12Potency0.316210
3-(4-ethoxyphenyl)-1-[2-(4-morpholinyl)ethyl]-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]thioureaEscherichia coli K-12Potency25.118910
1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-methyl-1-(thiophen-2-ylmethyl)thioureaEscherichia coli K-12Potency28.183810
4-[4-(benzenesulfonyl)-1-piperazinyl]-2-methylquinolineEscherichia coli K-12Potency22.387210
4,5-dimethoxy-2-[[1-oxo-2-[(3,5,8-trimethyl-2-quinolinyl)thio]ethyl]amino]benzoic acidEscherichia coli K-12Potency4.466810
2-thiophenecarboxylic acid [3-(3,5-dimethylphenoxy)-4-oxo-1-benzopyran-7-yl] esterEscherichia coli K-12Potency0.316210
2-(4-chlorophenyl)-N-[2-(4-morpholinyl)ethyl]-4-quinazolinamineEscherichia coli K-12Potency28.183810
4-(4-methylphenyl)-2-[[3-(4-morpholinyl)-1-oxopropyl]amino]-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency35.481310
2-[[2-(4-morpholinyl)-1-oxoethyl]amino]-4-thiophen-2-yl-3-thiophenecarboxylic acid methyl esterEscherichia coli K-12Potency20.259320
2-(3-ethylphenoxy)-N-[4-(2-pyridinylsulfamoyl)phenyl]acetamideEscherichia coli K-12Potency10.000010
4-(4-ethoxycarbonylanilino)-2-quinazolinecarboxylic acid ethyl esterEscherichia coli K-12Potency22.387210
2-(4-chloro-2-methylphenoxy)acetic acid [4-[(4-methylanilino)-oxomethyl]phenyl] esterEscherichia coli K-12Potency31.622810
2-[[cyclohexyl(oxo)methyl]amino]-4-(3-nitrophenyl)-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency1.584910
rhodanineEscherichia coli K-12Potency44.668410
3,4-dimethoxybenzoic acid [2-(3,4-dimethoxyphenyl)-2-oxoethyl] esterEscherichia coli K-12Potency100.000010
3-methoxy-4-(2-methoxy-3-methoxycarbonyl-1-naphthalenyl)-2-naphthalenecarboxylic acid methyl esterEscherichia coli K-12Potency19.091920
1-(2-chloro-10-phenothiazinyl)-2-[(1-methyl-5-tetrazolyl)thio]ethanoneEscherichia coli K-12Potency1.258910
N-(2-phenylethyl)-5-thiophen-2-yl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideEscherichia coli K-12Potency28.183810
5-(3,4-dimethoxyphenyl)-2-(4-methylphenyl)-4-thieno[2,3-d][1,3]oxazinoneEscherichia coli K-12Potency100.000010
N-[(1,2-dihydroacenaphthylen-5-ylamino)-sulfanylidenemethyl]-2-phenoxyacetamideEscherichia coli K-12Potency3.162310
7-(diethylaminomethyl)-1-(4-methoxyphenyl)-2-methyl-3-nitro-6-indololEscherichia coli K-12Potency89.125110
3-[1-(4-chlorophenyl)-5-tetrazolyl]-1-methyl-4-quinolinoneEscherichia coli K-12Potency28.183810
4-bromo-N'-(3,4-dihydro-2H-pyrrol-5-yl)benzohydrazideEscherichia coli K-12Potency0.631010
4-(3-bromophenyl)-7-methyl-2-(4-methylphenyl)pyrazolo[3,4-d]pyridazineEscherichia coli K-12Potency0.794310
2-[2-[2-(4-chlorophenyl)-2-oxoethoxy]phenyl]isoindole-1,3-dioneEscherichia coli K-12Potency8.912510
(4-ethoxyphenyl)-[4-[(4-ethoxyphenyl)-oxomethyl]-1,4-diazepan-1-yl]methanoneEscherichia coli K-12Potency22.387210
N-(1,3-benzothiazol-2-yl)-2-(3-methoxyphenyl)-4-quinolinecarboxamideEscherichia coli K-12Potency100.000010
2-(4-ethylphenyl)-N-(4-methyl-1-piperazinyl)-4-quinolinecarboxamideEscherichia coli K-12Potency40.074820
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[5-[(4-chlorophenoxy)methyl]-2-furanyl]methanoneEscherichia coli K-12Potency12.589310
[4-[(2-bromophenoxy)methyl]phenyl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency19.952610
2',4',6'-TrihydroxydihydrochalconeEscherichia coli K-12Potency17.782810
2-(2-bromo-4-chlorophenoxy)-N-cyclohexyl-N-methylacetamideEscherichia coli K-12Potency3.981110
N-[4-[methyl(phenyl)sulfamoyl]phenyl]benzamideEscherichia coli K-12Potency100.000010
3-(4-methylphenyl)-6-pyridin-4-yl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleEscherichia coli K-12Potency2.818410
1-[[2-(3-bromo-4-methoxyphenyl)-1-oxoethyl]amino]-3-phenylthioureaEscherichia coli K-12Potency100.000010
1-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-3-(4-methylphenyl)sulfonylureaEscherichia coli K-12Potency3.162310
3-(4-methoxyphenyl)-2-(4-methoxyphenyl)imino-4-thiazolidinoneEscherichia coli K-12Potency0.562310
2-(1,3-dioxo-2-isoindolyl)-N-(4-methyl-1,3-benzothiazol-2-yl)acetamideEscherichia coli K-12Potency56.234110
5-bromo-N-[3-chloro-2-(1-pyrrolidinyl)phenyl]-2-furancarboxamideEscherichia coli K-12Potency89.125110
2-(2-fluorophenyl)-4-(4-fluorophenyl)sulfonyl-5-(1-piperidinyl)oxazoleEscherichia coli K-12Potency1.122010
2-[[(2,3-dimethoxyphenyl)-oxomethyl]amino]-5-propan-2-yl-3-thiophenecarboxamideEscherichia coli K-12Potency22.387210
3-[oxo-[4-(2-phenylethyl)-1-piperazinyl]methyl]-1-benzopyran-2-oneEscherichia coli K-12Potency1.412510
4-(2,4-dichlorophenyl)-2-[(1-oxo-2-phenylethyl)amino]-3-thiophenecarboxamideEscherichia coli K-12Potency89.125110
1-(1,3-benzodioxol-5-yl)-3-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]ureaEscherichia coli K-12Potency14.125410
5-bromo-N-[2-(4-chlorophenyl)ethyl]-2-thiophenecarboxamideEscherichia coli K-12Potency2.511910
1,3-diethyl-6-methyl-N-(2-methylphenyl)-2-oxo-5-benzimidazolesulfonamideEscherichia coli K-12Potency100.000010
N-(1,3-benzodioxol-5-yl)-2-[[4-(4-methylphenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency56.234110
N-[(3-methoxyphenyl)methyl]-1-propyl-5-benzimidazolamineEscherichia coli K-12Potency3.548110
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-thiophenecarboxamideEscherichia coli K-12Potency7.943310
(4-chlorophenyl)-[4-(7-chloro-4-quinolinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency25.118910
2-[2-chloro-4-(2,3-dihydroindol-1-ylsulfonyl)phenoxy]-N-(2-pyridinylmethyl)acetamideEscherichia coli K-12Potency31.622810
5-(2,3-dihydroindol-1-ylsulfonyl)-1,3-diethyl-2-benzimidazoloneEscherichia coli K-12Potency39.810710
1-[1-methyl-2-(1-pyrrolidinylmethyl)-5-benzimidazolyl]-3-phenylureaEscherichia coli K-12Potency2.818410
4-chloro-N-[2-(4-methylsulfonyl-1-piperazinyl)phenyl]benzamideEscherichia coli K-12Potency0.316210
N-[[3-chloro-2-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideEscherichia coli K-12Potency63.095710
N-[2-(4-acetyl-1-piperazinyl)phenyl]-2-(5-methyl-2-propan-2-ylphenoxy)acetamideEscherichia coli K-12Potency40.676520
6-amino-1-[2-(3,4-dimethoxyphenyl)ethyl]-2-sulfanylidene-4-pyrimidinoneEscherichia coli K-12Potency5.011910
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(3-pyridinyl)-4-quinolinecarboxamideEscherichia coli K-12Potency28.183810
[4-[(2-chlorophenyl)methyl]-1-piperazinyl]-(6,8-dimethyl-2-pyridin-4-yl-4-quinolinyl)methanoneEscherichia coli K-12Potency17.782810
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamideEscherichia coli K-12Potency50.118710
1-(3,4-dimethoxyphenyl)sulfonyl-4-(2,6-dimethylphenyl)piperazineEscherichia coli K-12Potency11.220210
[4-(2,3-dimethylphenyl)-1-piperazinyl]-(3,4,5-trimethoxyphenyl)methanoneEscherichia coli K-12Potency31.622810
1-oxo-3-(1-piperidinyl)-5,6,7,8-tetrahydropyrrolo[1,2-a]indole-2-carbonitrileEscherichia coli K-12Potency17.782810
7-(2-oxopropoxy)-3-phenyl-1-benzopyran-2-oneEscherichia coli K-12Potency100.000010
2-[[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(1,3,4-thiadiazol-2-yl)acetamideEscherichia coli K-12Potency89.125110
N-(5-chloro-2-methylphenyl)-4-[(4-chloro-1-pyrazolyl)methyl]benzamideEscherichia coli K-12Potency11.220210
4-(5-methyl-2-furanyl)-2-[[2-(4-morpholinyl)-1-oxoethyl]amino]-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency35.481310
N-[2-(trifluoromethyl)-1,3-benzodioxol-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamideEscherichia coli K-12Potency39.810710
2-[[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]thio]-3-phenyl-4-quinazolinoneEscherichia coli K-12Potency12.589310
5-hydroxy-1-methyl-4-(4-morpholinylmethyl)-2-[(phenylthio)methyl]-3-indolecarboxylic acid ethyl esterEscherichia coli K-12Potency39.810710
N-(2-furanylmethyl)-2-imino-5-oxo-1-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideEscherichia coli K-12Potency7.079510
2-[[2-[(4-chlorophenyl)thio]-1-oxoethyl]amino]-N-(4-methoxyphenyl)benzamideEscherichia coli K-12Potency22.387210
3-(2-chlorophenyl)-5-methyl-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-isoxazolecarboxamideEscherichia coli K-12Potency7.943310
N-(6-ethoxy-1,3-benzothiazol-2-yl)-1,3-dimethyl-2-oxo-5-benzimidazolesulfonamideEscherichia coli K-12Potency3.162310
4-(1,3-dioxo-2-isoindolyl)-N-[2-(4-methoxyphenyl)ethyl]butanamideEscherichia coli K-12Potency2.818410
2-(1,3-benzothiazol-2-ylthio)-N-(4-methylphenyl)sulfonylacetamideEscherichia coli K-12Potency0.707910
2-(4-bromophenoxy)-N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamideEscherichia coli K-12Potency70.794610
3-[[2-[[4-ethyl-5-[(3-methylphenoxy)methyl]-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]benzoic acidEscherichia coli K-12Potency0.631010
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-5-methyl-3-phenyl-4-isoxazolecarboxamideEscherichia coli K-12Potency22.387210
2,4,5-trimethoxy-N-(2-phenylphenyl)benzamideEscherichia coli K-12Potency35.481310
9-(3-bromo-4-hydroxyphenyl)-10-phenyl-3,4,5,6,7,9-hexahydro-2H-acridine-1,8-dioneEscherichia coli K-12Potency35.481310
2-[[5-(3-aminophenyl)-4-methyl-1,2,4-triazol-3-yl]thio]-1-(9H-fluoren-2-yl)ethanoneEscherichia coli K-12Potency31.622810
[4-[(2,4-dichlorophenoxy)methyl]phenyl]-(4-methyl-1-piperazinyl)methanoneEscherichia coli K-12Potency28.183810
2-[[(4-bromo-1-ethyl-3-pyrazolyl)-oxomethyl]amino]-4-phenyl-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency100.000010
1-(1-azepanyl)-2-(2-bromo-4-propan-2-ylphenoxy)ethanoneEscherichia coli K-12Potency60.374020
darunavir ethanolateEscherichia coli K-12Potency0.631010
N-(4-bromo-2-fluorophenyl)-1-methylsulfonyl-4-piperidinecarboxamideEscherichia coli K-12Potency100.000010
[2-(4-methoxyphenyl)-6-methyl-4-quinolinyl]-(4-morpholinyl)methanoneEscherichia coli K-12Potency35.481310
5-(2-chlorophenyl)-N-phenyl-2-furancarboxamideEscherichia coli K-12Potency10.000010
4-(dimethylsulfamoyl)-N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamideEscherichia coli K-12Potency28.183810
4-(dimethylsulfamoyl)-N-(4-thiophen-2-yl-2-thiazolyl)benzamideEscherichia coli K-12Potency1.000010
N-(2,3-dimethylphenyl)-2-[[6-(1,3-dioxo-2-isoindolyl)-1,3-benzothiazol-2-yl]thio]acetamideEscherichia coli K-12Potency0.794310
N-cycloheptyl-2-[[2-(1,3-dioxo-2-isoindolyl)-1-oxoethyl]amino]benzamideEscherichia coli K-12Potency2.238710
N-[4-(4-morpholinyl)phenyl]-5-(2-nitrophenyl)-2-furancarboxamideEscherichia coli K-12Potency56.234110
N-(2-phenyl-5-benzotriazolyl)-2,3-dihydro-1,4-benzodioxin-6-carboxamideEscherichia coli K-12Potency0.631010
N-[[3-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideEscherichia coli K-12Potency100.000010
1-(3-chlorophenyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazineEscherichia coli K-12Potency39.810710
1-[5-(5-chloro-2-methylphenyl)-2-furanyl]-N-[4-(4-morpholinyl)phenyl]methanimineEscherichia coli K-12Potency1.000010
3-(3,4-dimethoxyphenyl)-7-(2-oxopropoxy)-1-benzopyran-2-oneEscherichia coli K-12Potency11.220210
urb 597Escherichia coli K-12Potency39.810710
N-(4-methylphenyl)-4-benzofuro[3,2-d]pyrimidinamineEscherichia coli K-12Potency1.000010
N-(2,4-dimethoxyphenyl)-N'-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]butanediamideEscherichia coli K-12Potency28.183810
2-(8-methoxy-2-methyl-4-oxo-1-quinolinyl)-N-(2-methoxyphenyl)acetamideEscherichia coli K-12Potency25.118910
2-furanyl-[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]methanoneEscherichia coli K-12Potency28.183810
[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-thiophen-2-ylmethanoneEscherichia coli K-12Potency35.481310
8,9-dimethyl-N-(3-methylphenyl)-3-[2-(4-morpholinyl)ethyl]-4H-[1,3]thiazino[6,5-b]quinolin-2-imineEscherichia coli K-12Potency19.952610
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency25.118910
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[[2-(phenylmethyl)-4-quinazolinyl]thio]ethanoneEscherichia coli K-12Potency3.548110
N'-[2-[[1-(4-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinyl]thio]-1-oxoethyl]-2-furancarbohydrazideEscherichia coli K-12Potency28.183810
(5-chloro-2-hydroxyphenyl)-[2-ethyl-3-(4-fluorophenyl)-6-pyrazolo[1,5-a]pyrimidinyl]methanoneEscherichia coli K-12Potency14.125410
7-methyl-2-[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]-3-quinolinecarbonitrileEscherichia coli K-12Potency39.810710
7-methoxy-2-[4-[(2-methylphenyl)-oxomethyl]-1-piperazinyl]-3-quinolinecarbonitrileEscherichia coli K-12Potency17.782810
1-[2-(5,6-dimethyl-1H-benzimidazol-2-yl)ethyl]-3-(2-methoxyphenyl)-1-(3-pyridinylmethyl)thioureaEscherichia coli K-12Potency31.099020
N-(2,3-dihydro-1H-inden-5-yl)-5-methyl-2-pyrazinecarboxamideEscherichia coli K-12Potency2.511910
(2,6-difluorophenyl)-[4-(5-fluoro-2-methyl-1-benzimidazolyl)-1-piperidinyl]methanoneEscherichia coli K-12Potency25.118910
4-[(2,6-dichlorophenyl)thio]-5-methoxy-2-(2-pyridinyl)pyrimidineEscherichia coli K-12Potency4.466810
4-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]oxy]-N-propan-2-ylbenzenesulfonamideEscherichia coli K-12Potency6.309610
7-anilino-3-(4-bromophenyl)-5-(4-morpholinyl)-1,4-thiazepine-6-carbonitrileEscherichia coli K-12Potency22.387210
2-[(4-chlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinoneEscherichia coli K-12Potency19.952610
2-[2-[2-(3-fluorophenyl)-4-thiazolyl]ethyl]isoindole-1,3-dioneEscherichia coli K-12Potency7.943310
4-(2,6-dimethylphenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidineEscherichia coli K-12Potency39.810710
2,5-dichloro-N-(1,5,6-trimethyl-4-benzimidazolyl)benzenesulfonamideEscherichia coli K-12Potency6.309610
6,7-dimethoxy-N-[(4-methylphenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency3.162310
4-[2-[(3,4-dichlorophenyl)methylthio]-6-[(methylthio)methyl]-4-pyrimidinyl]morpholineEscherichia coli K-12Potency100.000010
4-(4-chlorophenyl)sulfinyl-6-(methoxymethyl)-2-methylpyrimidineEscherichia coli K-12Potency70.794610
4-[(2-chloro-5-thiazolyl)methylthio]benzoic acidEscherichia coli K-12Potency39.810710
3-[4-ethyl-5-[(4-methylphenyl)methylthio]-1,2,4-triazol-3-yl]-1-phenyl-4-pyridazinoneEscherichia coli K-12Potency25.118910
3-[5-[(3,4-dichlorophenyl)methylthio]-4-ethyl-1,2,4-triazol-3-yl]-1-phenyl-4-pyridazinoneEscherichia coli K-12Potency19.952610
9-methyl-5,6,7,8-tetrahydrotetrazolo[5,1-b]quinazolineEscherichia coli K-12Potency0.631010
2-(4-methylsulfonylphenyl)-6-imidazo[1,2-a]pyridinecarboxylic acid methyl esterEscherichia coli K-12Potency31.622810
5-[3-[(2,4-dichlorophenyl)methoxy]-2-thiophenyl]-1,2-dihydro-1,2,4-triazole-3-thioneEscherichia coli K-12Potency89.125110
N,5-bis(4-methoxyphenyl)-2-thiophenecarboxamideEscherichia coli K-12Potency3.981110
4-[4-(2,4-dichlorophenyl)-2-thiazolyl]benzoic acidEscherichia coli K-12Potency1.778310
4-[2-[(2,4-dichlorophenyl)methylthio]-6-methyl-4-pyrimidinyl]morpholineEscherichia coli K-12Potency100.000010
1-[[[1-(6-methyl-2-pyridinyl)-4-imidazolyl]-oxomethyl]amino]-3-phenylthioureaEscherichia coli K-12Potency2.238710
(4-chlorophenyl)-[5-(4-morpholinyl)-4-(2-pyridinyl)-2-thiophenyl]methanoneEscherichia coli K-12Potency22.387210
N,N-dimethylcarbamic acid [4-[2-(benzenesulfonyl)-1-oxoethyl]-2,6-dimethylphenyl] esterEscherichia coli K-12Potency2.818410
3-(5-chloro-1,3-benzoxazol-2-yl)-N-(phenylmethyl)-2-pyridinamineEscherichia coli K-12Potency6.309610
(4-chlorophenyl)-[4-[[(2,4-dichlorophenyl)thio]methyl]-4-hydroxy-1-piperidinyl]methanoneEscherichia coli K-12Potency6.309610
(2-methylanilino)thioureaEscherichia coli K-12Potency1.122010
5-(4-chlorophenyl)-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamideEscherichia coli K-12Potency25.118910
1-[(4-methylphenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineEscherichia coli K-12Potency56.234110
LSM-18426Escherichia coli K-12Potency100.000010
4-methoxy-N-(8-methyl-[1,3]dioxolo[4,5-g]quinazolin-6-yl)benzamideEscherichia coli K-12Potency100.000010
N-(4-fluorophenyl)-3H-benzimidazole-5-carboxamideEscherichia coli K-12Potency5.011910
5-[(4-methyl-1-piperidinyl)methyl]-1-[4-(1-pyrrolyl)-1,2,5-oxadiazol-3-yl]-4-triazolecarboxylic acid ethyl esterEscherichia coli K-12Potency89.125110
4-[7-(4-methylphenyl)-5-phenyl-4-pyrrolo[2,3-d]pyrimidinyl]morpholineEscherichia coli K-12Potency39.810710
4-[7-(3-methylphenyl)-5-phenyl-4-pyrrolo[2,3-d]pyrimidinyl]morpholineEscherichia coli K-12Potency39.810710
[5,6-dimethyl-3-(pyridin-4-ylmethyl)-2,4-dihydrothieno[2,3-d]pyrimidin-1-yl]-(2-furanyl)methanoneEscherichia coli K-12Potency31.622810
1-[(4-chlorophenyl)methyl]-4-[4-(2-methylphenyl)-1-piperazinyl]pyrazolo[3,4-d]pyrimidineEscherichia coli K-12Potency28.183810
2-[(3,4-dichlorophenyl)methylthio]-6-(3-pyridinyl)-3-pyridinecarbonitrileEscherichia coli K-12Potency25.118910
cinnarizineEscherichia coli K-12Potency562.341010
2-amino-6-ethyl-3-(3-isoxazolyl)-7-methoxy-1-benzopyran-4-oneEscherichia coli K-12Potency0.316210
2-[[[4-(diethylsulfamoyl)phenyl]-oxomethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterEscherichia coli K-12Potency0.707910
enclomipheneEscherichia coli K-12Potency10.330220
1,4-benzoquinone guanylhydrazone thiosemicarbazoneEscherichia coli K-12Potency44.668410
cyqualonEscherichia coli K-12Potency89.125110
6-(1,3-dioxo-2-isoindolyl)hexanoic acid (4-methyl-2-oxo-1-benzopyran-7-yl) esterEscherichia coli K-12Potency7.079510
3-chloro-1-(2,4-dimethylphenyl)-4-(2-hydroxyethylamino)pyrrole-2,5-dioneEscherichia coli K-12Potency15.848910
4-[[(3,6-dichloro-2-methoxyphenyl)-oxomethyl]amino]benzoic acid propyl esterEscherichia coli K-12Potency28.183810
5,6-dimethyl-2-(prop-2-enylthio)-4-thieno[2,3-d]pyrimidinamineEscherichia coli K-12Potency0.079410
8-(dimethylamino)-3,4-dihydro-2H-pyrimido[2,1-b][1,3]thiazin-6-oneEscherichia coli K-12Potency8.912510
2-(benzenesulfonamido)acetic acid [2-(4-nitrophenyl)-2-oxoethyl] esterEscherichia coli K-12Potency0.707910
4-methyl-N-[(1-oxopentylhydrazo)-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency89.125110
fm19g11Escherichia coli K-12Potency3.162310
4-butyl-3-(5-ethyl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency0.562310
4-butyl-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency56.234110
(2S)-3-(1H-indol-3-yl)-2-[[2-[(4-methyl-6-oxo-3-benzo[c][1]benzopyranyl)oxy]-1-oxoethyl]amino]propanoic acidEscherichia coli K-12Potency50.118710
5-bromo-N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideEscherichia coli K-12Potency2.818410
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency0.251210
4-chloro-N-[[[oxo-(3,4,5-trimethoxyphenyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency39.810710
n-(4'-bromophenyl)-2,2-diphenylacetanilideEscherichia coli K-12Potency3.162310
1-ethyl-3-[[[(phenylmethyl)amino]-sulfanylidenemethyl]amino]thioureaEscherichia coli K-12Potency89.125110
1-[[4-[(3,4-dichlorophenyl)thio]-3-pyridinyl]sulfonyl]-3-propylureaEscherichia coli K-12Potency28.183810
3-(3-hydroxypropylamino)-7-methyl-1-(pentylamino)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileEscherichia coli K-12Potency2.511910
4-(2,5-dimethoxyphenyl)-3-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency8.912510
2-[[2-[(2-fluorophenyl)methoxy]-3-methoxyphenyl]methylamino]phenolEscherichia coli K-12Potency19.952610
N-[2-methoxy-5-(3-methyl-4-oxo-1-phthalazinyl)phenyl]-2-(4-methylphenoxy)acetamideEscherichia coli K-12Potency7.943310
9-methoxy-6-[(4-methoxyphenyl)methyl]indolo[3,2-b]quinoxalineEscherichia coli K-12Potency100.000010
5-bromo-3-[[3-(3,3-dimethyl-1-piperidinyl)-1-oxopropyl]amino]-1H-indole-2-carboxylic acid ethyl esterEscherichia coli K-12Potency42.239520
N-[[(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)amino]-sulfanylidenemethyl]-5-methyl-3-phenyl-4-isoxazolecarboxamideEscherichia coli K-12Potency17.782810
1-[2-[(3-chloro-4-methoxyphenyl)methylthio]ethyl]-3-phenylthioureaEscherichia coli K-12Potency50.118710
5-fluoro-3-[(4-methoxyphenyl)sulfonylamino]-1H-indole-2-carboxylic acid methyl esterEscherichia coli K-12Potency22.387210
N-(9-ethyl-3-carbazolyl)-2-[[4-ethyl-5-(2-furanyl)-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency15.848910
2-amino-1-[2-(4-morpholinyl)ethyl]-3-pyrrolo[3,2-b]quinoxalinecarboxylic acid ethyl esterEscherichia coli K-12Potency35.481310
2-amino-1-[2-(4-morpholinyl)ethyl]-N-prop-2-enyl-3-pyrrolo[3,2-b]quinoxalinecarboxamideEscherichia coli K-12Potency19.952610
5-[(2-cyanoethylthio)methyl]-2-benzofurancarboxylic acidEscherichia coli K-12Potency100.000010
2-(2-furanyl)-3,5-dimethyl-4-oxido-6-phenylpyrazin-1-ium 1-oxideEscherichia coli K-12Potency1.000010
1-[2-(2-amino-3-cyano-1-pyrrolo[3,2-b]quinoxalinyl)ethyl]-3-phenylureaEscherichia coli K-12Potency22.387210
1-[[(4-ethoxyanilino)-sulfanylidenemethyl]amino]-3-[3-(trifluoromethyl)phenyl]thioureaEscherichia coli K-12Potency79.432810
N-[[[(4-methoxyphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideEscherichia coli K-12Potency7.079510
acetic acid [4-[[3-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]anilino]-oxomethyl]phenyl] esterEscherichia coli K-12Potency5.623410
4-oxo-3-[(1-oxo-2,2-diphenylethyl)amino]-2-sulfanylidene-1H-quinazoline-7-carboxylic acid methyl esterEscherichia coli K-12Potency22.387210
3-[(6-methyl-4-phenyl-2-quinazolinyl)amino]-1-propanolEscherichia coli K-12Potency39.810710
N,N-bis(2-methoxyethyl)-2-thieno[3,2-b][1]benzothiolecarboxamideEscherichia coli K-12Potency31.622810
N-(4,5-diphenyl-2-oxazolyl)-3-methoxybenzamideEscherichia coli K-12Potency3.548110
3,4,5-trimethoxy-N-[[2-(4-morpholinyl)anilino]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency15.848910
4-(2,5-dimethoxyphenyl)-3-(3-phenyl-1H-pyrazol-5-yl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency89.125110
LSM-20401Escherichia coli K-12Potency56.234110
1-(4-methoxyphenyl)-N-[2-(4-morpholinyl)ethyl]-4-pyrazolo[3,4-d]pyrimidinamineEscherichia coli K-12Potency28.183810
2-[[1-oxo-2-(2-pyrimidinylthio)ethyl]amino]-6-(phenylmethyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylic acid ethyl esterEscherichia coli K-12Potency35.481310
2-(butylamino)-3-(3-chlorophenyl)-7-methyl-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-4-oneEscherichia coli K-12Potency1.412510
4-bromobenzoic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterEscherichia coli K-12Potency1.412510
N-[2-(3,4-dimethoxyphenyl)ethyl]-8-ethoxy-5H-pyrimido[5,4-b]indol-4-amineEscherichia coli K-12Potency39.810710
2-benzofurancarboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterEscherichia coli K-12Potency0.631010
(4,7-dichloro-1,3-benzothiazol-2-yl)hydrazineEscherichia coli K-12Potency28.183810
4-(4-chlorophenyl)-1-(2-methoxyethyl)-4H-pyridine-3,5-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency39.810710
N-(1,3-benzodioxol-5-yl)-2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideEscherichia coli K-12Potency1.000010
4-(4-bromophenyl)sulfonyl-2-(2-furanyl)-5-(methylthio)oxazoleEscherichia coli K-12Potency7.079510
cuspin-1Escherichia coli K-12Potency2.511910
2-[[(4-bromo-1-ethyl-3-pyrazolyl)-oxomethyl]amino]-4,5-dimethyl-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency44.668410
4-(3,5-dimethyl-4-nitro-1-pyrazolyl)butanoic acidEscherichia coli K-12Potency39.810710
3-[(2-propoxyphenyl)methyl]-1,3-benzoxazol-2-oneEscherichia coli K-12Potency2.511910
3-[2-oxo-2-[4-(phenylmethyl)-1-piperidinyl]ethyl]-1,3-diazaspiro[4.6]undecane-2,4-dioneEscherichia coli K-12Potency39.810710
3-(4-methylphenyl)sulfonylpropanoic acid [2-[(3,5-dichloro-2-pyridinyl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency3.981110
N-(9-ethyl-3-carbazolyl)-2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]acetamideEscherichia coli K-12Potency2.818410
benzoic acid [2-oxo-2-[2-(phenylthio)anilino]ethyl] esterEscherichia coli K-12Potency79.432810
4-(4-acetylphenoxy)butanoic acid [5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl esterEscherichia coli K-12Potency39.810710
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-(3,4,5-trimethoxyphenyl)acetamideEscherichia coli K-12Potency0.281810
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)thio]ethanoneEscherichia coli K-12Potency3.548110
N-[(tert-butylamino)-oxomethyl]-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideEscherichia coli K-12Potency10.000010
N-(3-cyano-2-thiophenyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]acetamideEscherichia coli K-12Potency6.309610
4-(2,3-dihydroindol-1-ylmethyl)-7-ethyl-1-benzopyran-2-oneEscherichia coli K-12Potency1.412510
N-(1H-benzimidazol-2-yl)-3-[phenyl(prop-2-enyl)sulfamoyl]benzamideEscherichia coli K-12Potency10.000010
3-ethyl-4-oxo-1-phthalazinecarboxylic acid [2-[2-(2,4-dioxo-3-thiazolidinyl)ethylamino]-2-oxoethyl] esterEscherichia coli K-12Potency0.631010
4-[[4-(benzenesulfonyl)-1-piperazinyl]-oxomethyl]-2-methyl-1-phthalazinoneEscherichia coli K-12Potency10.000010
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(cyclopropylamino)-2-oxoethyl] esterEscherichia coli K-12Potency44.668410
N-[2-(1,3-benzothiazol-2-ylthio)-1-oxoethyl]-1-methyl-2-pyrrolecarboxamideEscherichia coli K-12Potency15.848910
3-methyl-2-benzo[g]benzofurancarboxylic acid [2-[N-(2-cyanoethyl)anilino]-2-oxoethyl] esterEscherichia coli K-12Potency2.818410
4-(2,4-dichlorophenoxy)butanoic acid [2-oxo-2-[(phenylmethyl)amino]ethyl] esterEscherichia coli K-12Potency64.992420
N-[4-(4-methyl-2-thiazolyl)-2-phenyl-3-pyrazolyl]-3-(trifluoromethyl)benzamideEscherichia coli K-12Potency28.183810
2-chloro-N-[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]acetamideEscherichia coli K-12Potency56.234110
3-[[4-(2-benzofuranyl)-2-thiazolyl]methyl]-2-[(dimethylamino)methyl]-4-quinazolinoneEscherichia coli K-12Potency39.810710
2,5-difluoro-N-[2-(4-morpholinylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]benzenesulfonamideEscherichia coli K-12Potency39.810710
2-[7-chloro-2,3-dioxo-4-(phenylmethyl)-1-quinoxalinyl]-N-(3-fluorophenyl)acetamideEscherichia coli K-12Potency63.095710
5-methyl-7-(trifluoromethyl)-2-thiazolo[4,5-b]pyridinamineEscherichia coli K-12Potency7.943310
3-amino-5-[3-(methylamino)propyl]-1H-pyrazole-4-carbonitrileEscherichia coli K-12Potency0.316210
2-(1,3-dimethyl-2-benzimidazolylidene)-4-[(6-ethyl-4-thieno[2,3-d]pyrimidinyl)thio]-3-oxobutanenitrileEscherichia coli K-12Potency44.668410
N-phenyl-5-(propan-2-ylthio)-1,3,4-thiadiazol-2-amineEscherichia coli K-12Potency50.118710
N-[4-(2,5-dimethoxyphenyl)-2-thiazolyl]-2-[(4-nitrophenyl)thio]acetamideEscherichia coli K-12Potency0.354810
1-(4-bromo-2-fluorophenyl)-3-(3-chlorophenyl)ureaEscherichia coli K-12Potency0.631010
1-[4-[(2-hydroxy-5-methylphenyl)-oxomethyl]-1-pyrazolyl]-2-(2-methyl-4-thiazolyl)ethanoneEscherichia coli K-12Potency0.631010
2-[[2-furanyl(oxo)methyl]amino]benzoic acid [2-(cyclohexylmethylamino)-2-oxoethyl] esterEscherichia coli K-12Potency3.162310
3-[(4-acetyl-1-piperazinyl)sulfonyl]-N-(1H-benzimidazol-2-yl)benzamideEscherichia coli K-12Potency25.118910
4-chloro-3-(1-piperidinylsulfonyl)benzoic acid [2-(4-amino-1,3-dimethyl-2,6-dioxo-5-pyrimidinyl)-2-oxoethyl] esterEscherichia coli K-12Potency31.622810
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-2,5-diphenyl-3-pyrazolecarboxamideEscherichia coli K-12Potency17.782810
5-bromo-N-[2-(4-morpholinyl)-5-(trifluoromethyl)phenyl]-3-pyridinecarboxamideEscherichia coli K-12Potency0.316210
[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-(2-ethoxy-3-pyridinyl)methanoneEscherichia coli K-12Potency28.183810
2-[[2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]-1-oxoethyl]amino]-5-phenyl-3-thiophenecarboxamideEscherichia coli K-12Potency3.162310
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-quinolinecarboxamideEscherichia coli K-12Potency100.000010
(2S)-2-[[(2-chlorophenyl)-oxomethyl]amino]-3-methylbutanoic acid (6-nitro-4H-1,3-benzodioxin-8-yl)methyl esterEscherichia coli K-12Potency19.952610
3-[[[5-[3-(1-piperidinylsulfonyl)phenyl]-1,3,4-oxadiazol-2-yl]thio]methyl]-1,2,3-benzotriazin-4-oneEscherichia coli K-12Potency39.810710
N-(5-methyl-6,7-dihydro-4H-thiazolo[5,4-c]pyridin-2-yl)-2-(2-naphthalenyloxy)acetamideEscherichia coli K-12Potency89.125110
1-(1,3-benzothiazol-2-yl)-3-propylureaEscherichia coli K-12Potency17.782810
CID 2131972Escherichia coli K-12Potency22.387210
N-[3-(6-methyl-4-phenyl-2-quinolinyl)phenyl]methanesulfonamideEscherichia coli K-12Potency100.000010
4-[[oxo-(1-phenyl-3-pyridin-4-yl-4-pyrazolyl)methyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency1.412510
N-[(4-methoxyphenyl)methyl]-2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxamideEscherichia coli K-12Potency7.943310
N-(4-fluorophenyl)-2-(5-methoxy-1-oxo-2-isoquinolinyl)acetamideEscherichia coli K-12Potency6.309610
1-[4-[(2-amino-5-thiazolyl)methyl]phenyl]ethanoneEscherichia coli K-12Potency50.118710
N-(4-acetylphenyl)-5-[(phenylthio)methyl]-2-furancarboxamideEscherichia coli K-12Potency10.000010
2-[[2-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-1-oxo-5-isoquinolinyl]oxy]acetic acid ethyl esterEscherichia coli K-12Potency2.818410
N-[(4-chlorophenyl)methyl]-2-(2,4-dioxo-1H-pyrimidin-6-yl)acetamideEscherichia coli K-12Potency100.000010
6-propan-2-yl-2-sulfanylidene-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-oneEscherichia coli K-12Potency31.622810
N-(3,5-dimethylphenyl)-2-[(4-oxo-3-phenyl-2-benzofuro[3,2-d]pyrimidinyl)thio]acetamideEscherichia coli K-12Potency3.162310
2-[[3-(4-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetic acid ethyl esterEscherichia coli K-12Potency0.707910
4-[butyl(methyl)sulfamoyl]-N-[5-[(methylthio)methyl]-1,3,4-oxadiazol-2-yl]benzamideEscherichia coli K-12Potency1.000010
4-[bis(2-methylpropyl)sulfamoyl]-N-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideEscherichia coli K-12Potency44.668410
5-bromo-N-(4,7-dimethoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamideEscherichia coli K-12Potency10.000010
N-[5-(2-methylpropyl)-1,3,4-thiadiazol-2-yl]-4-nitrobenzenesulfonamideEscherichia coli K-12Potency3.981110
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterEscherichia coli K-12Potency89.125110
2-methyl-N-(2,3,4,5,6-pentafluorophenyl)-3-furancarboxamideEscherichia coli K-12Potency0.562310
2-[[2-[[4-hydroxy-6-oxo-5-(phenylmethyl)-1H-pyrimidin-2-yl]thio]-1-oxoethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterEscherichia coli K-12Potency15.848910
thiocyanic acid [2-(1-naphthalenyl)-2-oxoethyl] esterEscherichia coli K-12Potency89.125110
2-[2-(1-naphthalenyloxy)ethylthio]pyrimidineEscherichia coli K-12Potency39.810710
2-bromo-N-[3-(1-oxopentylamino)phenyl]benzamideEscherichia coli K-12Potency4.466810
N-[4-(dibutylsulfamoyl)phenyl]-2-thiophen-2-ylacetamideEscherichia coli K-12Potency35.481310
2-(2-hydroxyethylthio)-N-(2-methylphenyl)acetamideEscherichia coli K-12Potency28.183810
1-(4-butylphenyl)-3-(4-morpholinyl)thioureaEscherichia coli K-12Potency79.432810
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]acetic acid ethyl esterEscherichia coli K-12Potency11.220210
5-methyl-3-[3-[(5-methyl-1H-1,2,4-triazol-3-yl)thio]propylthio]-1H-1,2,4-triazoleEscherichia coli K-12Potency3.981110
1-[3-(4-phenylphenoxy)propyl]-1,2,4-triazoleEscherichia coli K-12Potency89.125110
1-[2-[2-(2,3-dihydro-1H-inden-5-yloxy)ethoxy]ethyl]-1,2,4-triazoleEscherichia coli K-12Potency79.432810
2,5-dimethoxybenzenesulfonic acid (1,3-dioxo-2-isoindolyl) esterEscherichia coli K-12Potency33.997220
2-[2-nitro-4-(trifluoromethyl)phenyl]sulfinylacetic acid (4-chlorophenyl) esterEscherichia coli K-12Potency112.202010
4-[[[(2-methoxy-1-oxoethyl)hydrazo]-sulfanylidenemethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency39.810710
N-[4-(diethylsulfamoyl)phenyl]-4-(4-morpholinylmethyl)benzamideEscherichia coli K-12Potency22.387210
N-[[(cyclohexylamino)-sulfanylidenemethyl]amino]carbamic acid tert-butyl esterEscherichia coli K-12Potency0.631010
1-[5-(2-furanylmethylamino)-3-phenyl-1,2,4-triazol-1-yl]-2-(4-methoxyphenyl)ethanoneEscherichia coli K-12Potency28.183810
N-(2-furanylmethyl)-2-[4-(propylsulfamoyl)phenoxy]acetamideEscherichia coli K-12Potency5.623410
3,5-dimethyl-N-[4-[(1-oxo-2-phenylethyl)amino]phenyl]benzamideEscherichia coli K-12Potency0.631010
4-[[(2,4-difluoroanilino)-sulfanylidenemethyl]hydrazo]-N-(3,4-dimethylphenyl)-4-oxobutanamideEscherichia coli K-12Potency22.387210
1-(5-chloro-2-methoxyphenyl)-3-[3-(2-oxo-1-pyrrolidinyl)propyl]thioureaEscherichia coli K-12Potency25.118910
3-[[(2,4-dichloroanilino)-sulfanylidenemethyl]amino]-4-methylbenzoic acidEscherichia coli K-12Potency0.631010
[5-[(4-methoxyphenyl)methylamino]-3-phenyl-1,2,4-triazol-1-yl]-(4-nitrophenyl)methanoneEscherichia coli K-12Potency44.668410
2-[[5-[3-(2,4-dichlorophenoxy)propyl]-4-methyl-1,2,4-triazol-3-yl]thio]-N-(2-ethyl-6-methylphenyl)acetamideEscherichia coli K-12Potency19.952610
N-[(3-ethoxy-2-prop-2-enoxyphenyl)methyl]-2-thiazolamineEscherichia coli K-12Potency4.466810
2-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-2-yl)oxy]acetic acid ethyl esterEscherichia coli K-12Potency8.912510
N-(2-furanylmethyl)-2-[3-(1-oxo-2-phenoxyethyl)-1-indolyl]acetamideEscherichia coli K-12Potency1.778310
N-(5-tert-butyl-3-isoxazolyl)-7-chloro-8-methyl-2-(2-pyridinyl)-4-quinolinecarboxamideEscherichia coli K-12Potency3.548110
6-bromo-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-pyridinyl)-4-quinolinecarboxamideEscherichia coli K-12Potency22.387210
5-(thiophen-2-ylmethyl)-1,3-diazinane-2,4,6-trioneEscherichia coli K-12Potency1.258910
3-(3-bromoanilino)-1-(5-methyl-2-furanyl)-1-propanoneEscherichia coli K-12Potency39.810710
N-[2-(1-cyclohexenyl)ethyl]-5-methyl-3-isoxazolecarboxamideEscherichia coli K-12Potency5.623410
3-chloro-N-[3-(4-morpholinyl)propyl]-6-nitro-1-benzothiophene-2-carboxamideEscherichia coli K-12Potency50.118710
N-(2-naphthalenyl)-2-[[6-[[[2-(2-naphthalenylamino)-2-oxoethyl]thio]methyl]-2-pyridinyl]methylthio]acetamideEscherichia coli K-12Potency0.631010
4-[2-(4-bromo-2-chlorophenoxy)-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency31.622810
N-[[3-chloro-2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]butanamideEscherichia coli K-12Potency0.707910
4-chloro-3-[(2,5-dimethylphenyl)sulfamoyl]-N-(2-phenylphenyl)benzamideEscherichia coli K-12Potency14.125410
4-[2-[(4-chlorophenyl)thio]ethoxy]-3-ethoxybenzaldehydeEscherichia coli K-12Potency0.562310
N-[4-[[[(3-bromo-4-methylphenyl)-oxomethyl]hydrazo]-oxomethyl]phenyl]pentanamideEscherichia coli K-12Potency112.202010
2-[[5-(2-benzofuranyl)-4-(phenylmethyl)-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency100.000010
1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(5,7-diphenyl-2-pyrazolo[1,5-a]pyrimidinyl)methanoneEscherichia coli K-12Potency19.952610
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneEscherichia coli K-12Potency10.000010
4-chloro-3-[[2-(4-methyl-1-piperidinyl)-1-oxoethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency31.622810
3-(dimethylamino)propyl benzoateEscherichia coli K-12Potency31.622810
2-[[[5-(3-chlorophenyl)-2-furanyl]-oxomethyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency17.782810
2-[[5-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]-4-oxo-2-phenyl-1-benzopyran-7-yl]oxy]acetic acid tert-butyl esterEscherichia coli K-12Potency15.848910
N-(2,1,3-benzothiadiazol-4-yl)-5-(3-chlorophenyl)-2-furancarboxamideEscherichia coli K-12Potency4.466810
N-(3-acetylphenyl)-2-naphthalenecarboxamideEscherichia coli K-12Potency100.000010
N-[3-[[diethylamino(sulfanylidene)methyl]thio]-1-oxopropyl]carbamic acid (4-methylphenyl) esterEscherichia coli K-12Potency5.011910
8-[2-(4-chloro-3,5-dimethylphenoxy)ethoxy]quinolineEscherichia coli K-12Potency39.810710
1-chloro-2-[2-(2-methoxy-4-methylphenoxy)ethoxy]-4-methylbenzeneEscherichia coli K-12Potency44.668410
2-[cyclohexyl-(4-methylphenyl)sulfonylamino]-N-(3-methoxypropyl)acetamideEscherichia coli K-12Potency19.952610
5-[[2-methoxy-4-(4-morpholinyl)phenyl]methylidene]-1,3-diazinane-2,4,6-trioneEscherichia coli K-12Potency19.952610
N-[4-[(4-sulfamoylphenyl)sulfamoyl]phenyl]cyclopropanecarboxamideEscherichia coli K-12Potency3.548110
4-[2-[2-(4-bromo-2-chlorophenoxy)ethoxy]ethyl]morpholineEscherichia coli K-12Potency35.481310
2-[2-(3-ethylphenoxy)ethyl]propanedioic acid diethyl esterEscherichia coli K-12Potency0.707910
reversanEscherichia coli K-12Potency89.125110
N-[3-cyano-4,5-bis(4-methoxyphenyl)-2-furanyl]acetamideEscherichia coli K-12Potency0.631010
N-[4-[(4,6-dimethyl-2-pyrimidinyl)sulfamoyl]phenyl]-2-phenyl-4-quinolinecarboxamideEscherichia coli K-12Potency39.810710
4-methyl-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)anilineEscherichia coli K-12Potency100.000010
1-phenyl-N-(3-pyridinylmethyl)-3-thiophen-2-yl-4-pyrazolecarboxamideEscherichia coli K-12Potency89.125110
N-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethenyl]-4-morpholinecarboxamideEscherichia coli K-12Potency0.631010
3-[2-(4-fluorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineEscherichia coli K-12Potency11.220210
2-(4,6-dimethyl-2-pyrimidinyl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamineEscherichia coli K-12Potency28.183810
N-[4-(4-morpholinyl)phenyl]-2-pyridin-4-yl-4-quinolinecarboxamideEscherichia coli K-12Potency22.387210
5-chloro-N-(3,4-dimethylphenyl)-2,1-benzothiazole-3-carboxamideEscherichia coli K-12Potency4.466810
N-[[2-(diethylamino)ethylamino]-sulfanylidenemethyl]-3-(4-methoxyphenyl)-1-phenyl-4-pyrazolecarboxamideEscherichia coli K-12Potency39.810710
[[2-[[4-(4-bromophenyl)-2-thiazolyl]amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esterEscherichia coli K-12Potency11.220210
3-methyl-N,1-diphenyl-4-pyrazolecarbothioamideEscherichia coli K-12Potency2.511910
3-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineEscherichia coli K-12Potency0.316210
N-(1H-benzimidazol-2-ylmethyl)-3-(1-pyrrolidinylsulfonyl)benzamideEscherichia coli K-12Potency39.810710
2-(1H-benzimidazol-2-ylthio)-N-(2-methoxy-3-dibenzofuranyl)acetamideEscherichia coli K-12Potency7.943310
2-[(2,5-dimethylphenyl)sulfonylamino]-N-[4-(2-pyrimidinylsulfamoyl)phenyl]benzamideEscherichia coli K-12Potency15.848910
4-(4-chlorophenyl)-4-oxobutanoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterEscherichia coli K-12Potency89.125110
2-[(4-methylphenyl)sulfonylamino]acetic acid [2-(2,3-dihydroindol-1-yl)-2-oxoethyl] esterEscherichia coli K-12Potency5.623410
1-(2-tert-butylphenyl)-3-cyclohexylthioureaEscherichia coli K-12Potency4.466810
2,3-dihydro-1,4-dioxin-5-carboxylic acid [2-[4-[4-(2-methylbutan-2-yl)phenoxy]anilino]-2-oxoethyl] esterEscherichia coli K-12Potency15.848910
3-(1-azepanylsulfonyl)-4-chloro-N-(1H-1,2,4-triazol-5-yl)benzamideEscherichia coli K-12Potency39.810710
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-methoxy-5-methylphenyl)benzamideEscherichia coli K-12Potency0.631010
3-[2-[(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)amino]-2-oxoethyl]-4-oxo-1-phthalazinecarboxylic acidEscherichia coli K-12Potency2.818410
2,8-dimercapto-6-hydroxypurineEscherichia coli K-12Potency0.631010
4-amino-2-[[4-(1-azepanylsulfonyl)phenyl]-oxomethyl]isoindole-1,3-dioneEscherichia coli K-12Potency100.000010
3-oxo-2,4-dihydroquinoxaline-1-carboxylic acid (phenylmethyl) esterEscherichia coli K-12Potency0.707910
4-(1H-indol-3-yl)butanoic acid [2-(4-amino-1,3-dimethyl-2,6-dioxo-5-pyrimidinyl)-2-oxoethyl] esterEscherichia coli K-12Potency39.810710
2-(5H-[1,2,4]triazolo[5,1-a]isoindol-2-yl)ethanethioamideEscherichia coli K-12Potency22.387210
2,5-dimethyl-3-furancarboxylic acid [2-(2,3-dihydroindol-1-yl)-2-oxoethyl] esterEscherichia coli K-12Potency0.631010
1-(4-ethoxyphenyl)-3-(5-isoquinolinyl)thioureaEscherichia coli K-12Potency100.000010
N-[(1-adamantylamino)-oxomethyl]-2-chloroacetamideEscherichia coli K-12Potency5.011910
4,5-dimethyl-2-[[1-oxo-2-(4-quinazolinyloxy)ethyl]amino]-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency6.309610
1-(2-fluorophenyl)-1-cyclopentanecarboxylic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterEscherichia coli K-12Potency1.258910
3-[(4-methyl-1-piperazinyl)sulfonyl]-N-(4-phenyl-2-thiazolyl)benzamideEscherichia coli K-12Potency28.183810
1-(4-fluorophenyl)-1-cyclopentanecarboxylic acid [2-oxo-2-(4-sulfamoylanilino)ethyl] esterEscherichia coli K-12Potency25.118910
1-(2-furanyl)-2-(1H-1,2,4-triazol-5-ylthio)ethanoneEscherichia coli K-12Potency31.622810
3-(2-chlorophenyl)sulfonylpropanoic acid [2-[(3,5-dichloro-6-methyl-2-pyridinyl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency89.125110
1-(2-cyanoethyl)-6-(2-fluoro-4-methoxyphenyl)-3-methyl-4-pyrazolo[3,4-b]pyridinecarboxylic acid ethyl esterEscherichia coli K-12Potency13.699620
2-(2-methyl-1-benzimidazolyl)acetic acid [2-(2-methyl-1H-indol-3-yl)-2-oxoethyl] esterEscherichia coli K-12Potency35.481310
2,5-dimethyl-1-(3-methylphenyl)-N-(4-methylphenyl)-3-pyrrolecarboxamideEscherichia coli K-12Potency15.848910
N2-[5-(4-chlorophenyl)-2-phenyl-3-pyrazolyl]benzene-1,2-diamineEscherichia coli K-12Potency11.220210
N2-(5-phenyl-1H-pyrazol-3-yl)benzene-1,2-diamineEscherichia coli K-12Potency1.122010
2-[[2-[(2-hydroxyphenyl)-oxomethoxy]-1-oxoethyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency100.000010
4-[(1-methyl-5-tetrazolyl)thio]-5-phenylthieno[2,3-d]pyrimidineEscherichia coli K-12Potency0.631010
N-[4-(difluoromethylthio)phenyl]-5-[(2-hydroxy-5-methoxyphenyl)-oxomethyl]-2-imino-3-pyrancarboxamideEscherichia coli K-12Potency14.125410
N-(4-acetamidophenyl)-2-[5-(1-piperidinylsulfonyl)-2-thiophenyl]acetamideEscherichia coli K-12Potency25.118910
N-(4,5,6-trifluoro-1,3-benzothiazol-2-yl)-2-furancarboxamideEscherichia coli K-12Potency100.000010
N-(1,3-benzodioxol-5-yl)-2-chloro-N-[(2-prop-2-enoxyphenyl)methyl]acetamideEscherichia coli K-12Potency14.125410
4-[4-[3-(Trifluoromethyl)phenyl]piperazine-1-carbonyl]-1H-quinolin-2-oneEscherichia coli K-12Potency39.810710
2-(2,3-dihydro-1H-inden-5-yloxy)-1-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]ethanoneEscherichia coli K-12Potency5.623410
N-(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)-2-[4-(4-hydroxyphenyl)-1-piperazinyl]acetamideEscherichia coli K-12Potency12.589310
2-chloro-N-[(5-chloro-2-thiophenyl)methyl]-N-methylacetamideEscherichia coli K-12Potency1.000010
N-[2-(2,3-dimethylanilino)-2-oxoethyl]-3-(3-methylphenoxy)propanamideEscherichia coli K-12Potency63.095710
4-[2-(4-fluoroanilino)-2-oxoethoxy]-3-methoxy-N-[4-(4-methoxyphenyl)-5-methyl-2-thiazolyl]benzamideEscherichia coli K-12Potency8.912510
4-ethyl-3-[2-(4-methylphenyl)-4-quinolinyl]-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency63.095710
2-(6-methyl-3-benzofuranyl)acetic acid [2-[(5-chloro-2-pyridinyl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency112.202010
2-hydroxy-4-methoxybenzoic acid (2-methyl-4-thiazolyl)methyl esterEscherichia coli K-12Potency0.631010
4-[[5-(1,3-benzothiazol-2-yl)-2-thiophenyl]-oxomethyl]-1-piperazinecarboxaldehydeEscherichia coli K-12Potency22.387210
1-(4-ethylphenyl)-3-[1-(phenylmethyl)-4-piperidinyl]thioureaEscherichia coli K-12Potency2.818410
[2-[(2-bromophenyl)methoxy]phenyl]-[4-(2-pyrimidinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency12.589310
3,5-dimethyl-1H-pyrrole-2,4-dicarboxylic acid O4-ethyl ester O2-[(2-fluorophenyl)methyl] esterEscherichia coli K-12Potency89.125110
4-[(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)methyl]-7-ethyl-1-benzopyran-2-oneEscherichia coli K-12Potency0.316210
1-(2-benzofuranyl)-2-[(4-methyl-2-quinolinyl)thio]ethanoneEscherichia coli K-12Potency44.668410
[4-methoxy-3-(4-morpholinylsulfonyl)phenyl]-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)methanoneEscherichia coli K-12Potency12.913420
2-[(2,3,4-trifluorophenyl)sulfonylamino]acetic acid [2-(3,4-dimethoxyanilino)-2-oxoethyl] esterEscherichia coli K-12Potency10.000010
N-(3-cyano-2-thiophenyl)-2-[4-(2,5-dimethylphenyl)sulfonyl-1-piperazinyl]acetamideEscherichia coli K-12Potency31.622810
2-[[4-(4-fluorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]thio]-N-[(2-furanylmethylamino)-oxomethyl]acetamideEscherichia coli K-12Potency0.631010
2-(2,4-dichlorophenoxy)-N-[2-(methylthio)phenyl]acetamideEscherichia coli K-12Potency0.707910
2-(2-naphthalenylsulfonylamino)acetic acid [2-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-2-oxoethyl] esterEscherichia coli K-12Potency44.668410
5-[[(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)thio]methyl]-2-furancarboxylic acid methyl esterEscherichia coli K-12Potency35.481310
2-[[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)thio]methyl]-1,3-benzothiazoleEscherichia coli K-12Potency1.584910
1-[2,5-dimethyl-1-(phenylmethyl)-3-pyrrolyl]-2-[4-(1,3,4-oxadiazol-2-yl)phenoxy]ethanoneEscherichia coli K-12Potency39.810710
5-bromo-3-[[(5-methyl-1,3,4-thiadiazol-2-yl)thio]methyl]-2-benzofurancarboxylic acid ethyl esterEscherichia coli K-12Potency100.000010
2-[(3-chlorophenyl)methoxy]-3-methylquinoxalineEscherichia coli K-12Potency100.000010
2-[[[5-methyl-4-(2-methylphenyl)-1,2,4-triazol-3-yl]thio]methyl]-1,3-benzothiazoleEscherichia coli K-12Potency0.794310
2,4-dithiophen-2-ylthiazoleEscherichia coli K-12Potency5.011910
N,N-diethyl-3-[5-(ethylthio)-4-(phenylmethyl)-1,2,4-triazol-3-yl]benzenesulfonamideEscherichia coli K-12Potency25.118910
N-(4-chloro-2-methoxy-5-methylphenyl)-4-[(3,4-difluorophenyl)sulfonylamino]benzamideEscherichia coli K-12Potency0.707910
3-(methoxymethyl)-2-benzofurancarboxylic acid [4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methyl esterEscherichia coli K-12Potency31.622810
2-[[[4-cyclohexyl-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-oneEscherichia coli K-12Potency0.354810
5-methoxy-3-methyl-N-(3-methylbutyl)-2-benzofurancarboxamideEscherichia coli K-12Potency10.000010
4-[3-(2-phenoxyethoxy)-2-quinoxalinyl]morpholineEscherichia coli K-12Potency6.309610
1,3-benzothiazole-6-carboxylic acid [2-(2-furanyl)-2-oxoethyl] esterEscherichia coli K-12Potency1.584910
2-(1,3-benzodioxol-5-yl)-5-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methylthio]-1,3,4-oxadiazoleEscherichia coli K-12Potency0.794310
1-[4-(2-prop-2-enylphenoxy)butyl]pyrrolidineEscherichia coli K-12Potency1.412510
2-[[2-[[5-(4-ethylanilino)-1,3,4-thiadiazol-2-yl]thio]-1-oxoethyl]amino]-3-thiophenecarboxamideEscherichia coli K-12Potency15.848910
N-[3-(4-morpholinyl)propyl]-3-(3-pyridinyl)-7,8-dihydro-6H-cyclopenta[4,5]thieno[1,2-c]pyrimidin-1-amineEscherichia coli K-12Potency25.118910
4-(dimethylsulfamoyl)-N-(3-methylphenyl)benzamideEscherichia coli K-12Potency56.234110
5-[[(5,6-dimethyl-4-thieno[2,3-d]pyrimidinyl)thio]methyl]-2-furancarboxylic acid methyl esterEscherichia coli K-12Potency0.707910
4-chloro-N-[3-[(3,5-dimethyl-4-isoxazolyl)methylthio]-2-quinoxalinyl]benzenesulfonamideEscherichia coli K-12Potency0.316210
2-(1,3-benzoxazol-2-ylthio)-1-(2,5-dimethyl-1-prop-2-enyl-3-pyrrolyl)ethanoneEscherichia coli K-12Potency31.622810
5-methyl-4-(4-methylphenyl)-2-[[2-[(1-methyl-5-tetrazolyl)thio]-1-oxoethyl]amino]-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency0.316210
1-[1-(3-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(1-methyl-5-tetrazolyl)thio]ethanoneEscherichia coli K-12Potency22.387210
3-(difluoromethoxy)-N-(4,5-dihydrothiazol-2-yl)benzamideEscherichia coli K-12Potency56.234110
2-[[4-amino-5-[4-(difluoromethoxy)phenyl]-1,2,4-triazol-3-yl]thio]-N-[(2-furanylmethylamino)-oxomethyl]acetamideEscherichia coli K-12Potency0.631010
N-(2-methoxy-3-dibenzofuranyl)-2-(4-methoxyphenoxy)acetamideEscherichia coli K-12Potency100.000010
(1R,2S)-tranylcypromine hydrochlorideEscherichia coli K-12Potency11.220210
tacrine hydrochlorideEscherichia coli K-12Potency14.125410
5-chloro-2-mercaptobenzothiazoleEscherichia coli K-12Potency8.912510
digoxinEscherichia coli K-12Potency21.450910
N-(4-chlorophenyl)-N-ethyl-6-(propan-2-ylamino)-4-(trifluoromethyl)-3-pyridinecarboxamideEscherichia coli K-12Potency17.782810
4-phenoxyphenyl 4-hydroxypiperidine-1-carboxylateEscherichia coli K-12Potency22.387210
1,4-dihydroxy-4a,5,6,7,8,8a-hexahydroquinoxaline-2,3-dioneEscherichia coli K-12Potency0.631010
5-(1-naphthalenylamino)-3H-1,3,4-thiadiazole-2-thioneEscherichia coli K-12Potency28.183810
capsazepineEscherichia coli K-12Potency8.912510
tamoxifen citrateEscherichia coli K-12Potency31.622810
tamoxifenEscherichia coli K-12Potency5.011910
branigenEscherichia coli K-12Potency5.623410
pimagedine hydrochlorideEscherichia coli K-12Potency4.466810
3,4-di-O-acetyl-6-deoxy-L-glucalEscherichia coli K-12Potency35.481310
n-benzoylthioureaEscherichia coli K-12Potency100.000010
Betaine Aldehyde ChlorideEscherichia coli K-12Potency6.309610
1-(2,4-difluorophenyl)-3-[(5-methyl-3-phenyl-4-isoxazolyl)methyl]ureaEscherichia coli K-12Potency100.000010
N-[4-(5-oxazolyl)phenyl]benzamideEscherichia coli K-12Potency0.794310
N,N-diethyl-5-thiophen-2-yl-2-thiophenecarboxamideEscherichia coli K-12Potency100.000010
3-(tert-butylsulfamoyl)-4-phenyl-5-(trifluoromethyl)-2-thiophenecarboxylic acid methyl esterEscherichia coli K-12Potency19.952610
2-(1,3,4-oxadiazol-2-yl)phenyl 4-chlorobenzoateEscherichia coli K-12Potency8.912510
N1-(2,6-dimorpholino-3-pyridyl)-4-methylbenzamideEscherichia coli K-12Potency100.000010
1-[(3,5-dimethylisoxazol-4-yl)sulfonyl]piperidineEscherichia coli K-12Potency2.818410
N-(3-chlorophenyl)-2-[[2-(2-pyridinyl)-2,3-dihydro-1,3,4-thiadiazol-5-yl]thio]acetamideEscherichia coli K-12Potency39.810710
5-oxo-3-(4-phenylphenyl)-2H-furan-4-carbonitrileEscherichia coli K-12Potency19.952610
4-(4-methylphenyl)-2-(3-nitrophenyl)-3-pyrazolamineEscherichia coli K-12Potency50.118710
3-(dimethylaminomethylideneamino)-4-methoxy-2-thieno[2,3-b]pyridinecarboxylic acid ethyl esterEscherichia coli K-12Potency6.309610
4-(dimethylamino)-3-[(phenylmethoxyamino)methylideneamino]-2-thieno[2,3-b]pyridinecarboxylic acid ethyl esterEscherichia coli K-12Potency19.952610
1-[4-[(2-bromophenyl)-oxomethyl]-1H-pyrrol-2-yl]-2,2,2-trichloroethanoneEscherichia coli K-12Potency125.892010
4-chlorobenzoic acid [3-cyano-6-(3-methoxyphenyl)-2-pyridinyl] esterEscherichia coli K-12Potency15.848910
5-cyano-6-phenoxy-2-phenyl-3-pyridinecarboxylic acid ethyl esterEscherichia coli K-12Potency3.548110
2-[[butoxy(oxo)methyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency31.622810
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineEscherichia coli K-12Potency100.000010
N-(4-chlorophenethyl)-N'-(4-chlorophenyl)ureaEscherichia coli K-12Potency0.631010
ssya10-001Escherichia coli K-12Potency31.622810
Benzo[E]pyrazolo[5,1-c][1,2,4]triazin-8-yl N,N-dimethylcarbamateEscherichia coli K-12Potency0.631010
5-[[[5-(2-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esterEscherichia coli K-12Potency35.481310
5-[[[5-(4-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esterEscherichia coli K-12Potency28.183810
2-[[2-[[5-(4-tert-butylphenyl)-2-methoxycarbonyl-3-thiophenyl]amino]-2-oxoethyl]thio]acetic acidEscherichia coli K-12Potency22.387210
[4-(2-methoxyphenyl)-1-piperidinyl]-(5-methyl-1-phenyl-4-pyrazolyl)methanoneEscherichia coli K-12Potency25.118910
1-(3,5-dimethylphenyl)-3-[5-(dimethylsulfamoyl)-2-methylphenyl]ureaEscherichia coli K-12Potency100.000010
N-{5-[(dimethylamino)sulfonyl]-2-methylphenyl}cyclohexanecarboxamideEscherichia coli K-12Potency0.794310
2-[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazoleEscherichia coli K-12Potency100.000010
3,3-dimethyl-1-[[9-(methylthio)-5,6-dihydrothieno[3,4-h]quinazolin-2-yl]thio]-2-butanoneEscherichia coli K-12Potency7.079510
2-{5-[2-(Phenylthio)acetyl]-2-thienyl}acetic acidEscherichia coli K-12Potency31.622810
2-[5-[2-[(4-methylphenyl)thio]-1-oxoethyl]-2-thiophenyl]acetic acidEscherichia coli K-12Potency19.952610
1-(5-tert-butyl-2-methyl-3-pyrazolyl)-3-(3,5-dichlorophenyl)ureaEscherichia coli K-12Potency39.810710
1-(3,5-dichlorophenyl)-3-[2-(2-furanylmethylthio)ethyl]ureaEscherichia coli K-12Potency10.000010
N,N'-di[4-(2,6-dimethylmorpholino)phenyl]thioureaEscherichia coli K-12Potency15.848910
2-[4-[[4-[bis(2-hydroxyethyl)amino]-2-chlorophenyl]-(2-chlorophenyl)methyl]-3-chloro-N-(2-hydroxyethyl)anilino]ethanolEscherichia coli K-12Potency25.118910
2-fluoro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]acetamideEscherichia coli K-12Potency15.848910
2,4-dichloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamideEscherichia coli K-12Potency12.431220
2-(1-naphthalenyl)-N-[2,2,2-trichloro-1-[[(2-chloroanilino)-sulfanylidenemethyl]amino]ethyl]acetamideEscherichia coli K-12Potency31.622810
N-[[1,3-dioxo-2-(phenylmethyl)-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]-4-methoxybenzamideEscherichia coli K-12Potency5.011910
2-[(4-methylphenyl)sulfonylamino]pentanoic acidEscherichia coli K-12Potency2.238710
4-Methoxy-1-methyl-8-((2,2,5,5-tetramethyl-1,3-dioxolan-4-yl)methoxy)quinolin-2(1H)-oneEscherichia coli K-12Potency11.220210
(4-chlorophenyl)-[6,7-dichloro-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-3-benzofuranyl]methanoneEscherichia coli K-12Potency35.481310
1-(4-fluorophenyl)-3-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]pyrrolidine-2,5-dioneEscherichia coli K-12Potency17.782810
dihydrosamidineEscherichia coli K-12Potency15.848910
N-[2-(1-methyl-2-pyrrolidinyl)ethyl]-2-adamantanamineEscherichia coli K-12Potency5.623410
4-phenyl-N-(pyridin-4-ylmethyl)-2-butanamineEscherichia coli K-12Potency0.707910
3-methyl-4,7-bis(methylsulfonyl)-3a,5,6,7a-tetrahydro-1H-imidazo[4,5-b]pyrazin-2-oneEscherichia coli K-12Potency22.387210
1-hexadecyl-3-methylimidazolium bromideEscherichia coli K-12Potency35.716810
1,3-bis(butylsulfonyl)-3a,4,6,6a-tetrahydro-2H-imidazo[4,5-d]imidazol-5-oneEscherichia coli K-12Potency22.387210
4-(4-hydroxy-3-methoxyphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid (3-methylcyclohexyl) esterEscherichia coli K-12Potency3.981110
6,7-dimethoxy-3-propoxy-3H-isobenzofuran-1-oneEscherichia coli K-12Potency100.000010
N-(5-nitro-2-pyridinyl)cyclopropanecarboxamideEscherichia coli K-12Potency56.234110
3-[(4-bromophenyl)methyl]-4-(4-methoxyanilino)-4-oxobutanoic acidEscherichia coli K-12Potency39.810710
N-(2-methoxycyclohexyl)-2,5-dimethylanilineEscherichia coli K-12Potency39.810710
3-ethyl-N-(2H-tetrazol-5-yl)-1-adamantanecarboxamideEscherichia coli K-12Potency6.309610
2-(4,6,7-Trimethyl-2-quinazolinyl)guanidineEscherichia coli K-12Potency15.848910
4-(4-hydroxy-3-methoxyphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid (4-methoxyphenyl)methyl esterEscherichia coli K-12Potency0.631010
6-(2-chlorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylic acid 2-methylpropyl esterEscherichia coli K-12Potency3.162310
2,4-dichloro-6-[1-(4-morpholinyl)-3-phenylprop-2-ynyl]phenolEscherichia coli K-12Potency0.316210
1-ethoxy-3-(2-methoxy-4-prop-2-enylphenoxy)-2-propanolEscherichia coli K-12Potency3.981110
4-[3-[[(2,5-dichloroanilino)-methyliminomethyl]thio]-2,5-dioxo-1-pyrrolidinyl]benzoic acid methyl esterEscherichia coli K-12Potency3.162310
N-[4-bromo-2-[[(2-hydrazinyl-2-oxoethyl)amino]-phenylmethyl]phenyl]-3-(4-morpholinyl)propanamideEscherichia coli K-12Potency25.118910
N'-[2-(1-naphthalenyloxy)-1-oxoethyl]-2-oxolanecarbohydrazideEscherichia coli K-12Potency100.000010
N-(3-chloro-4-methylphenyl)-2-(3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)acetamideEscherichia coli K-12Potency79.432810
LSM-19241Escherichia coli K-12Potency16.126920
N-[(2-hydroxy-1-naphthalenyl)-(4-methoxyphenyl)methyl]-2-methylpropanamideEscherichia coli K-12Potency5.011910
1-(2-chlorophenoxy)-3-(2-methyl-1-benzimidazolyl)-2-propanolEscherichia coli K-12Potency39.810710
1-(4-methylphenyl)-3-(1H-1,2,4-triazol-5-ylthio)pyrrolidine-2,5-dioneEscherichia coli K-12Potency63.095710
6-amino-4-(2-methylpropyl)-3-phenyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileEscherichia coli K-12Potency10.000010
N-(5-bromo-2-pyridinyl)-2,2-dimethyl-3-(2-methylprop-1-enyl)-1-cyclopropanecarboxamideEscherichia coli K-12Potency89.125110
LSM-19663Escherichia coli K-12Potency64.467920
6-[(3,4-difluoroanilino)-oxomethyl]-1-cyclohex-3-enecarboxylic acidEscherichia coli K-12Potency3.981110
N-(2-methoxyphenyl)-2-phenyl-2-(phenylthio)acetamideEscherichia coli K-12Potency44.668410
N-[2,2,2-trichloro-1-[[sulfanylidene-(2,4,6-trimethylanilino)methyl]amino]ethyl]benzamideEscherichia coli K-12Potency3.548110
N-(3-bicyclo[2.2.1]heptanyl)-3-bromo-4-methoxybenzenesulfonamideEscherichia coli K-12Potency0.562310
2-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]-1-phenylethanoneEscherichia coli K-12Potency100.000010
N-[1-[[anilino(sulfanylidene)methyl]amino]-2,2,2-trichloroethyl]-2-(4-ethylphenoxy)acetamideEscherichia coli K-12Potency19.952610
5-bromo-3-hydroxy-3-(4-methyl-1-piperidinyl)-1H-indol-2-oneEscherichia coli K-12Potency22.387210
[3-methyl-4-[oxo(thiophen-2-yl)methyl]-1-piperazinyl]-thiophen-2-ylmethanoneEscherichia coli K-12Potency44.668410
2-chlorobenzoic acid [2-(4-methoxyphenyl)-2-oxo-1-phenylethyl] esterEscherichia coli K-12Potency6.309610
[4-(2-methoxyphenyl)-1-piperazinyl]-[4-[(phenylthio)methyl]phenyl]methanoneEscherichia coli K-12Potency51.581220
2-[[(1-butyl-2-benzimidazolyl)amino]methyl]phenolEscherichia coli K-12Potency50.158120
2-methyl-N-[5-(4-nitrophenyl)sulfonyl-2-thiazolyl]pentanamideEscherichia coli K-12Potency1.000010
2-[(4-chlorophenyl)thio]-N-[4-[(2,4-dimethylphenyl)sulfamoyl]phenyl]propanamideEscherichia coli K-12Potency112.202010
4-bromobenzenesulfonic acid (1,3-dioxo-2-benzo[de]isoquinolinyl) esterEscherichia coli K-12Potency44.668410
eskazineEscherichia coli K-12Potency25.285510
7,7-dimethyl-1-(4-methylphenyl)-2,5-dioxo-N-(2-oxo-3-thiolanyl)-6,8-dihydroquinoline-3-carboxamideEscherichia coli K-12Potency15.848910
2-[[5-[(1,3-benzothiazol-2-ylthio)methyl]-4-methyl-1,2,4-triazol-3-yl]thio]-N-[2-(4-morpholinyl)ethyl]acetamideEscherichia coli K-12Potency0.707910
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(2-furanyl)methyl]acetamideEscherichia coli K-12Potency0.251210
3,4,5-trimethoxy-N-[4-[(2-methyl-1-piperidinyl)sulfonyl]phenyl]benzamideEscherichia coli K-12Potency82.851420
4-[2-(difluoromethoxy)phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid (phenylmethyl) esterEscherichia coli K-12Potency5.011910
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(4-methoxyphenyl)methyl]acetamideEscherichia coli K-12Potency5.623410
2-nitrobenzoic acid [1-(4-methylphenyl)-1-oxopropan-2-yl] esterEscherichia coli K-12Potency3.548110
3-acetamidobenzoic acid [2-(4-methylphenyl)-2-oxo-1-phenylethyl] esterEscherichia coli K-12Potency20.186520
1,7,7-trimethyl-N,N-bis(2-methylpropyl)-2-oxo-4-bicyclo[2.2.1]heptanecarboxamideEscherichia coli K-12Potency7.079510
1-cyclopentyl-2-imino-10-methyl-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxamideEscherichia coli K-12Potency0.631010
[4-(benzenesulfonyl)-1-piperazinyl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency22.387210
6-[[[5-(ethylthio)-1,3,4-thiadiazol-2-yl]amino]-oxomethyl]-1-cyclohex-3-enecarboxylic acidEscherichia coli K-12Potency0.794310
1-adamantyl-[4-(2-fluorophenyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency39.810710
2-[4-(4-nitrophenyl)-1-piperazinyl]-N-(2-pyridinyl)acetamideEscherichia coli K-12Potency100.000010
LSM-25805Escherichia coli K-12Potency89.125110
2-(3,4-dimethylphenyl)-5-ethyl-5-phenyl-1,2,4-triazolidine-3-thioneEscherichia coli K-12Potency39.810710
2-[[1-(4-chlorophenyl)-2,5-dioxo-3-pyrrolidinyl]-methylamino]acetic acid methyl esterEscherichia coli K-12Potency100.000010
9-[2-hydroxy-3-(2-methyl-1-benzimidazolyl)propyl]-6-methyl-3,4-dihydro-2H-carbazol-1-oneEscherichia coli K-12Potency4.466810
N-[2,6-dimethyl-3-[(4-methyl-1-piperazinyl)sulfonyl]phenyl]-N,4-dimethylbenzenesulfonamideEscherichia coli K-12Potency10.476320
4-Chloro-2-(5-methyl-1,3-dioxooctahydro-2H-isoindol-2-yl)phenyl 2-furoateEscherichia coli K-12Potency25.118910
4-[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]-2,6-dimethylmorpholineEscherichia coli K-12Potency5.623410
1-(4-methoxyphenyl)-N,N-dipropyl-4-pyrazolo[3,4-d]pyrimidinamineEscherichia coli K-12Potency89.125110
5-(2-oxolanylmethylamino)-2-thiophen-2-yl-4-oxazolecarbonitrileEscherichia coli K-12Potency3.981110
2-[(9-tert-butyl-1,5-dicyano-2-oxo-3-azaspiro[5.5]undec-4-en-4-yl)thio]-N-cyclohexylacetamideEscherichia coli K-12Potency0.631010
2-[[1-(4-methoxy-2-nitrophenyl)-2,5-dioxo-3-pyrrolidinyl]thio]benzoic acidEscherichia coli K-12Potency28.183810
LSM-19894Escherichia coli K-12Potency0.631010
[1-[3-(4-methylphenoxy)propyl]-2-benzimidazolyl]methanolEscherichia coli K-12Potency0.631010
2-[4-(1-adamantyl)-N-methylsulfonylanilino]acetic acidEscherichia coli K-12Potency5.011910
N4-(4-fluorophenyl)-N5-(2-nitrophenyl)-1H-imidazole-4,5-dicarboxamideEscherichia coli K-12Potency63.095710
1-[4-(dimethylamino)phenyl]-3-[4-(4-morpholinyl)anilino]pyrrolidine-2,5-dioneEscherichia coli K-12Potency56.234110
2-(2-oxo-1-benzo[cd]indolyl)-N-(2-oxolanylmethyl)acetamideEscherichia coli K-12Potency0.631010
1-(4-fluorophenyl)-3-(2-methoxy-3-dibenzofuranyl)ureaEscherichia coli K-12Potency26.968020
3-nitro-N-[[4-[4-(1-oxopropyl)-1-piperazinyl]anilino]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency39.810710
4-[oxo-[1-(2,4,6-trimethylphenyl)sulfonyl-4-piperidinyl]methyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency31.622810
3-(2-pyrimidinylthio)-1-[2-(trifluoromethyl)phenyl]pyrrolidine-2,5-dioneEscherichia coli K-12Potency50.118710
N-(3,4-dimethylphenyl)-2-(4-methylanilino)-6-oxo-4,5-dihydro-1H-pyrimidine-4-carboxamideEscherichia coli K-12Potency0.707910
N-(5-chloro-2-hydroxyphenyl)-2-ethoxybenzamideEscherichia coli K-12Potency5.011910
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-phenoxybutanamideEscherichia coli K-12Potency6.309610
N-[1-oxo-3-phenyl-1-(2-pyridinylmethylamino)propan-2-yl]-2-furancarboxamideEscherichia coli K-12Potency56.234110
2-chloro-5-[[2,3-dihydro-1,4-benzodioxin-3-yl(oxo)methyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency0.316210
2-[[(2-methoxy-4-nitroanilino)-sulfanylidenemethyl]amino]benzene-1,4-dicarboxylic acid diethyl esterEscherichia coli K-12Potency63.095710
3-fluoro-N-[4-[[4-(4-methoxyphenyl)-1-piperazinyl]-oxomethyl]phenyl]benzenesulfonamideEscherichia coli K-12Potency89.125110
3-(5-chloro-2-hydroxyphenyl)-3-phenyl-N-[(4-propan-2-yloxyphenyl)methyl]propanamideEscherichia coli K-12Potency17.782810
1-[3-[4-(2-chloro-5-methoxyphenyl)-1-piperazinyl]propyl]-3-(4-methylphenyl)ureaEscherichia coli K-12Potency100.000010
N-[2-(1-azepanyl)-2-oxoethyl]-N-[(4-chlorophenyl)methyl]methanesulfonamideEscherichia coli K-12Potency28.934220
1-(4-morpholinyl)-2-(4-phenylphenoxy)-1-propanoneEscherichia coli K-12Potency1.000010
N-[2-(1-phenylethyl)-3,4-dihydro-1H-pyrazino[1,2-a]benzimidazol-8-yl]methanesulfonamideEscherichia coli K-12Potency1.258910
N-(3-carbamoyl-5-propyl-2-thiophenyl)-2-oxolanecarboxamideEscherichia coli K-12Potency112.202010
[3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-phenylmethanoneEscherichia coli K-12Potency2.238710
N-[3-chloro-2-(1-piperidinyl)phenyl]-4-(4-morpholinyl)-3-nitrobenzamideEscherichia coli K-12Potency10.000010
2-[[3-(methylthio)-1,2,4-thiadiazol-5-yl]thio]acetic acid (4-acetamidophenyl) esterEscherichia coli K-12Potency2.818410
N-[(2-chlorophenyl)methyl]-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-hydroxy-5-nitro-4-triazolimineEscherichia coli K-12Potency5.011910
N-[3-chloro-4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]phenyl]-2-(4-chlorophenyl)acetamideEscherichia coli K-12Potency5.011910
3-[5-(4-methylphenyl)-1-(2-oxolanylmethyl)-2-pyrrolyl]propanoic acidEscherichia coli K-12Potency8.912510
2-[(4-methylphenyl)thio]-N-(1H-1,2,4-triazol-5-yl)propanamideEscherichia coli K-12Potency79.432810
4-(2,5-dimethylphenyl)-6-[[(4-methylphenyl)methylamino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterEscherichia coli K-12Potency39.810710
2-[1-[[[(3-chloro-1-benzothiophen-2-yl)-oxomethyl]amino]-sulfanylidenemethyl]-3-oxo-2-piperazinyl]acetic acid methyl esterEscherichia coli K-12Potency0.631010
N1,N4-bis(1-phenylethyl)cyclohexane-1,4-dicarboxamideEscherichia coli K-12Potency56.234110
[3-(2-furanyl)-5-(thiophen-2-ylmethylamino)-1,2,4-triazol-1-yl]-(3-pyridinyl)methanoneEscherichia coli K-12Potency11.220210
1-[2-furanyl(oxo)methyl]-6-(1-pyrrolidinylsulfonyl)-2-benzo[cd]indoloneEscherichia coli K-12Potency28.183810
1-(3-chlorophenyl)-3-[[1-[(2,5-dimethoxyphenyl)methyl]-4-piperidinyl]methyl]ureaEscherichia coli K-12Potency39.810710
2-[2-[4-[2-hydroxy-3-(2-methylphenoxy)propyl]-1-piperazinyl]ethyl]benzo[de]isoquinoline-1,3-dioneEscherichia coli K-12Potency26.651420
4-(4-bromophenyl)-2-(3,5-dimethyl-1-pyrazolyl)-4-oxobutanoic acid methyl esterEscherichia coli K-12Potency35.481310
1,3-dimethyl-8-[methyl-(phenylmethyl)amino]-7-[2-(2-pyrimidinylthio)ethyl]purine-2,6-dioneEscherichia coli K-12Potency7.943310
1-(2-fluorophenyl)-3-(4-methoxy-2-nitrophenyl)ureaEscherichia coli K-12Potency4.466810
3-methyl-N-[[(2-methyl-5-quinolinyl)amino]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency50.118710
3-methyl-4-oxo-1,5,6,7-tetrahydroindole-2-carboxylic acid (4-methylcyclohexyl) esterEscherichia coli K-12Potency0.316210
3-[2-[4-(4-chlorophenyl)sulfonyl-1-piperazinyl]-2-oxoethyl]-5-(2-methylpropyl)imidazolidine-2,4-dioneEscherichia coli K-12Potency19.952610
4-[[[5-(2,3-dihydro-1,4-benzodioxin-3-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]methyl]-3,5-dimethylisoxazoleEscherichia coli K-12Potency1.584910
N-(3-cyano-2-thiophenyl)-2-[(1-methyl-2-imidazolyl)thio]acetamideEscherichia coli K-12Potency79.432810
3-[5-(dimethylsulfamoyl)-1-ethyl-2-benzimidazolyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)propanamideEscherichia coli K-12Potency25.118910
N-(2,2-difluoro-1,3-benzodioxol-5-yl)-2-[2-[2-(4-morpholinyl)-2-oxoethyl]-1-benzimidazolyl]acetamideEscherichia coli K-12Potency28.183810
2-methyl-1-cyclopropanecarboxylic acid (7-bromo-4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl esterEscherichia coli K-12Potency112.202010
N-[4-(6-imidazo[2,1-b]thiazolyl)phenyl]-4-methoxy-3-(4-morpholinylsulfonyl)benzamideEscherichia coli K-12Potency39.810710
2-[[2-(4-ethyl-4-methyl-2,5-dioxo-1-imidazolidinyl)-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideEscherichia coli K-12Potency44.668410
7-[[[1-(3-methylphenyl)-2-benzimidazolyl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneEscherichia coli K-12Potency39.810710
1-[(6,6-dimethyl-4-bicyclo[3.1.1]hept-3-enyl)methoxy]-3-(1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl)-2-propanolEscherichia coli K-12Potency14.432620
2-(4-cyanophenoxy)-N-(2-methyl-1-phenyl-5-benzimidazolyl)acetamideEscherichia coli K-12Potency39.810710
2-[[5-[(2-fluorophenoxy)methyl]-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-N-[(2-furanylmethylamino)-oxomethyl]acetamideEscherichia coli K-12Potency1.026620
1-[2,5-dimethyl-1-(2-oxolanylmethyl)-3-pyrrolyl]-2-[(5-phenyl-4-prop-2-enyl-1,2,4-triazol-3-yl)thio]ethanoneEscherichia coli K-12Potency31.622810
5-[4-(1-imidazolyl)phenoxy]-1-phenyltetrazoleEscherichia coli K-12Potency15.848910
3-(4-chlorophenyl)sulfonyl-N-[2,5-diethoxy-4-(4-morpholinyl)phenyl]propanamideEscherichia coli K-12Potency15.969520
3-hydroxy-1-adamantanecarboxylic acid [2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterEscherichia coli K-12Potency31.622810
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideEscherichia coli K-12Potency2.818410
5-chloro-N-[2-(2-furanyl)-2-(1-pyrrolidinyl)ethyl]-2-methoxybenzamideEscherichia coli K-12Potency0.158510
2-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterEscherichia coli K-12Potency6.309610
6-[2-(2-methoxyphenyl)imino-3-(2-oxolanylmethyl)-4-thiazolyl]-4H-1,4-benzoxazin-3-oneEscherichia coli K-12Potency31.622810
1-[2-hydroxy-3-[4-(2-methylbutan-2-yl)phenoxy]propyl]-4-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency25.118910
2-(1,3-diphenyl-4-pyrazolyl)-3-(2-furanylmethyl)-4-thiazolidinoneEscherichia coli K-12Potency28.471020
5-[[2,3-dihydro-1,4-benzodioxin-3-yl(oxo)methyl]amino]benzene-1,3-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency0.223910
1-butyl-2-[(1,3-dioxo-2-isoindolyl)methylthio]-5-benzimidazolesulfonamideEscherichia coli K-12Potency0.316210
3,5-dimethyl-4-isoxazolecarboxylic acid (3-butyl-2,6-dioxo-7-propyl-8-purinyl)methyl esterEscherichia coli K-12Potency44.668410
2,3-dihydro-1,4-dioxin-5-carboxylic acid [2-oxo-2-(4-phenylbutan-2-ylamino)ethyl] esterEscherichia coli K-12Potency112.202010
[4-(2-pyridinyl)-1-piperazinyl]-[2-(3,4,5-trimethoxyphenyl)-4-quinolinyl]methanoneEscherichia coli K-12Potency14.125410
3-(4-fluorophenyl)-N-[3-(1-imidazolyl)propyl]-1-phenyl-4-pyrazolecarboxamideEscherichia coli K-12Potency0.631010
7-(3-methoxypropyl)-3-(phenylmethyl)-8-(3-thiophenyl)purine-2,6-dioneEscherichia coli K-12Potency0.562310
benzoic acid [5-(6-benzamido-9-purinyl)-3-fluoro-4-hydroxy-2-oxolanyl]methyl esterEscherichia coli K-12Potency100.000010
2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)benzoic acid thiophen-2-ylmethyl esterEscherichia coli K-12Potency44.668410
bis(1-ethenyl-2-imidazolyl)-(9-ethyl-3-carbazolyl)-sulfanylidenephosphoraneEscherichia coli K-12Potency15.848910
1-(4-fluorophenyl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxylic acid (2-oxo-3-oxolanyl) esterEscherichia coli K-12Potency100.000010
3,5-dimethyl-1-phenyl-4-pyrazolecarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] esterEscherichia coli K-12Potency64.091920
3-methyl-2-(phenylmethoxycarbonylamino)butanoic acid [2-oxo-2-(1-piperidinyl)ethyl] esterEscherichia coli K-12Potency3.548110
7-[3-[4-(2-ethoxyphenyl)-1-piperazinyl]-2-hydroxypropoxy]-4-methyl-1-benzopyran-2-oneEscherichia coli K-12Potency39.810710
9H-xanthene-9-carboxylic acid [2-[(1,1-dioxo-3-thiolanyl)-methylamino]-2-oxoethyl] esterEscherichia coli K-12Potency10.000010
N-(2-oxolanylmethyl)-3-(1-tetrazolyl)benzamideEscherichia coli K-12Potency0.631010
2-amino-4-chlorobenzoic acid [2-oxo-2-(3,3,5-trimethyl-7-azabicyclo[3.2.1]octan-7-yl)ethyl] esterEscherichia coli K-12Potency35.481310
2-(1,3-benzodioxol-5-yl)-5-[[2-(4-methoxyphenyl)-4,5-dihydrothiazol-5-yl]methylthio]-1,3,4-oxadiazoleEscherichia coli K-12Potency100.000010
1-(4-fluorophenyl)-1-cyclopentanecarboxylic acid [2-(2,6-dimethyl-4-morpholinyl)-2-oxoethyl] esterEscherichia coli K-12Potency28.183810
2-[[(2-ethoxyphenyl)-oxomethyl]amino]acetic acid [2-(2,6-dimethyl-1-piperidinyl)-2-oxoethyl] esterEscherichia coli K-12Potency100.000010
3-fluoro-6a,7,8,9,10,11-hexahydro-6H-azepino[2,1-c][1,2,4]benzothiadiazine 5,5-dioxideEscherichia coli K-12Potency112.202010
2,6-difluorobenzoic acid 2,3-dihydro-1,4-benzodioxin-3-ylmethyl esterEscherichia coli K-12Potency5.623410
N-(3-cyanophenyl)-2-(4-ethyl-2,5-dioxo-4-phenyl-1-imidazolidinyl)acetamideEscherichia coli K-12Potency1.778310
6-methyl-2-[[2-(4-morpholinyl)-1-oxoethyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency2.818410
2-(3,4-dimethoxyphenyl)-4-quinolinecarboxylic acid (2-oxo-3-oxolanyl) esterEscherichia coli K-12Potency16.165420
2-[(3-butan-2-yl-4-oxo-2-quinazolinyl)thio]propanenitrileEscherichia coli K-12Potency112.202010
3-(4-methylphenyl)sulfonyl-1-(3-oxolanylmethyl)-2-pyrrolo[3,2-b]quinoxalinamineEscherichia coli K-12Potency2.511910
cyclopropanecarboxylic acid [2-oxo-2-(4-phenoxyanilino)ethyl] esterEscherichia coli K-12Potency28.183810
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideEscherichia coli K-12Potency0.316210
2-thiophenecarboxylic acid [2-oxo-2-(2-oxolanylmethylamino)ethyl] esterEscherichia coli K-12Potency3.162310
5-[[[5-(2,3-dihydro-1,4-benzodioxin-3-yl)-4-methyl-1,2,4-triazol-3-yl]thio]methyl]-2-phenylthiazoleEscherichia coli K-12Potency3.548110
tjn 101Escherichia coli K-12Potency25.118910
(4As,6aS,6bR,10S,12aR)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylic acidEscherichia coli K-12Potency1.584910
zuclomifene citrateEscherichia coli K-12Potency18.169620
monooctanoinEscherichia coli K-12Potency48.102320
7-deacetylgeduninEscherichia coli K-12Potency0.316210
2-chloro-n(6)-(3-iodobenzyl)adenosine-5'-n-methyluronamideEscherichia coli K-12Potency39.810710
mefexamideEscherichia coli K-12Potency3.981110
amedin hydrochlorideEscherichia coli K-12Potency0.158510
trimethoprimEscherichia coli K-12Potency112.202010
LSM-5894Escherichia coli K-12Potency39.810710
N-(2-hydroxy-5-nitrophenyl)-3-nitrobenzamideEscherichia coli K-12Potency0.707910
N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) esterEscherichia coli K-12Potency89.125110
N-[2-[(2-chloro-1-oxopropyl)hydrazo]-2-oxoethyl]benzenesulfonamideEscherichia coli K-12Potency22.387210
2-[[2,2,2-trichloro-1-[(2-methyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid ethyl esterEscherichia coli K-12Potency89.125110
6-phenylspiro[7-oxa-1-azabicyclo[2.2.1]heptane-2,1'-cyclopentane]Escherichia coli K-12Potency0.316210
N-tert-butyl-2-[[(3-nitrophenyl)-oxomethyl]hydrazo]-2-oxoacetamideEscherichia coli K-12Potency2.818410
2-(2,4-dioxo-3-phenyl-5-thiazolidinyl)-N-(3-methylphenyl)acetamideEscherichia coli K-12Potency6.309610
N-[3-(1,3-benzothiazol-2-ylthio)-5-nitrophenyl]-2-fluorobenzamideEscherichia coli K-12Potency19.952610
(3-bromophenyl)-[5-(4-bromophenyl)-3-ethyl-5-hydroxy-4H-pyrazol-1-yl]methanoneEscherichia coli K-12Potency44.668410
2-[(4-chlorophenyl)-[2-[5-(4-chlorophenyl)-2-thiazolyl]-5-methyl-3-oxo-1H-pyrazol-4-yl]methyl]propanedinitrileEscherichia coli K-12Potency39.810710
2-[[2-(2,4-dichlorophenoxy)-1-oxopropyl]hydrazo]-N-(4-methoxyphenyl)-2-oxoacetamideEscherichia coli K-12Potency31.622810
2-(2-bromophenyl)-2,3-dihydro-1H-perimidineEscherichia coli K-12Potency7.079510
2-[[3-methyl-5-oxo-1-(phenylmethyl)-4H-pyrazol-4-yl]-phenylmethyl]propanedinitrileEscherichia coli K-12Potency56.234110
2-[[2-furanyl(oxo)methyl]hydrazo]-N-(2-methoxy-5-methylphenyl)-2-oxoacetamideEscherichia coli K-12Potency6.309610
N-[3-[(4-chlorophenyl)-oxomethyl]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-pyridinecarboxamideEscherichia coli K-12Potency6.309610
N-[[[2-(2-methylphenoxy)-1-oxoethyl]hydrazo]-sulfanylidenemethyl]-2-nitrobenzamideEscherichia coli K-12Potency100.000010
N'-(9-acridinyl)-2-hydroxybenzohydrazideEscherichia coli K-12Potency0.125910
N-butan-2-yl-4-[4-oxo-3-(phenylmethyl)-2-thiazolidinyl]benzamideEscherichia coli K-12Potency35.481310
3,4-dimethoxy-N-[(2-methyl-4-nitroanilino)-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency2.511910
N'-[2-[(6-methoxy-2-methyl-4-quinolinyl)thio]-1-oxoethyl]-2-(1-naphthalenyloxy)acetohydrazideEscherichia coli K-12Potency39.810710
N-(2,5-dimethoxyphenyl)-4-(2,4-dimethyl-5-thiazolyl)-2-thiazolamineEscherichia coli K-12Potency39.810710
3-methyl-7-(2-phenylethyl)-8-(propylamino)purine-2,6-dioneEscherichia coli K-12Potency3.548110
3-[[5,6-bis(4-methoxyphenyl)-4-furo[2,3-d]pyrimidinyl]amino]-1-propanolEscherichia coli K-12Potency22.387210
2-[(2-ethyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-3-yl)oxy]acetic acid methyl esterEscherichia coli K-12Potency26.645920
2-[7-oxo-7-(3-phenyl-1-pyrrolidinyl)heptyl]isoindole-1,3-dioneEscherichia coli K-12Potency17.782810
2-[(4-ethyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)thio]acetic acid methyl esterEscherichia coli K-12Potency70.794610
2-imino-1-[(4-methylphenyl)methyl]-5-oxo-N-(2-oxolanylmethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideEscherichia coli K-12Potency2.238710
N-[2-(cyclopentylamino)-1-(4-fluorophenyl)-2-oxoethyl]-N-[(4-fluorophenyl)methyl]-1H-pyrazole-5-carboxamideEscherichia coli K-12Potency56.234110
6-amino-4-(3-furanyl)-3-(4-methoxyphenyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileEscherichia coli K-12Potency28.183810
N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideEscherichia coli K-12Potency28.183810
6-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideEscherichia coli K-12Potency22.387210
6-(3,4-dimethoxyphenyl)-4-oxo-3-phenyl-1,5,6,7-tetrahydroindole-2-carboxylic acid ethyl esterEscherichia coli K-12Potency35.716820
9-(2-ethoxy-3-methoxyphenyl)-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneEscherichia coli K-12Potency2.818410
4-(dimethylsulfamoyl)-N-(6,7,8,9-tetrahydro-5H-carbazol-3-ylmethyl)benzamideEscherichia coli K-12Potency16.597820
2-[[5-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-1,2,4-triazol-3-yl]thio]acetonitrileEscherichia coli K-12Potency22.387210
1-[(5,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-furanylmethyl)-3-(2-oxolanylmethyl)thioureaEscherichia coli K-12Potency22.387210
1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-[2-(3-methylphenyl)ethyl]-3-[3-(4-morpholinyl)propyl]thioureaEscherichia coli K-12Potency12.589310
3-butan-2-yl-1-[(6,7-dimethoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-phenylethyl)thioureaEscherichia coli K-12Potency31.622810
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[[5-(3,5-dimethylphenyl)-1,3,4-oxadiazol-2-yl]thio]ethanoneEscherichia coli K-12Potency89.125110
2-[cyclopentyl-[1-oxo-2-(5-thiophen-2-yl-2-tetrazolyl)ethyl]amino]-N-(2-oxolanylmethyl)-2-thiophen-2-ylacetamideEscherichia coli K-12Potency40.344120
3-(2,4-dimethoxyphenyl)-1-[(1-ethyl-2-pyrrolidinyl)methyl]-1-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]thioureaEscherichia coli K-12Potency89.125110
CID 3192987Escherichia coli K-12Potency28.183810
[4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-(2-furanyl)methanoneEscherichia coli K-12Potency31.622810
4-ethoxy-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-[(4-methoxyphenyl)methyl]benzamideEscherichia coli K-12Potency25.118910
2-(N-[2-(Benzotriazol-1-yl)acetyl]-2,4,6-trimethylanilino)-N-tert-butyl-2-thiophen-3-ylacetamideEscherichia coli K-12Potency19.952610
4-[3-(1,3-benzodioxol-5-ylmethylamino)-7-methyl-2-imidazo[1,2-a]pyridinyl]phenolEscherichia coli K-12Potency39.810710
2-butyl-3-[(3-chlorophenyl)methyl]-5-methyl-6-imidazo[4,5-b]pyridinamineEscherichia coli K-12Potency19.952610
CID 3206295Escherichia coli K-12Potency4.466810
N-[2-(cyclohexylamino)-2-oxo-1-(6-quinolinyl)ethyl]-N-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideEscherichia coli K-12Potency112.202010
N-tert-butyl-2-[(2-chloro-1-oxoethyl)-(2-furanylmethyl)amino]-2-(4-chlorophenyl)acetamideEscherichia coli K-12Potency44.668410
2-[2-methoxyethyl-(1-oxo-2-thiophen-2-ylethyl)amino]-N-[(4-methoxyphenyl)methyl]-2-(4-propan-2-ylphenyl)acetamideEscherichia coli K-12Potency3.981110
N-(1,3-benzodioxol-5-ylmethyl)-N-[2-(cyclohexylamino)-2-oxo-1-pyridin-4-ylethyl]-2,2,2-trifluoroacetamideEscherichia coli K-12Potency31.622810
2-chloro-N-[1-[oxo(10-phenothiazinyl)methyl]-4-piperidinyl]benzamideEscherichia coli K-12Potency39.810710
2-furancarboxylic acid [2-(cyclohexylamino)-2-oxo-1-phenylethyl] esterEscherichia coli K-12Potency44.668410
1-(3,5-dimethyl-1-piperidinyl)-2-[[2-(thiophen-2-ylmethyl)-4-quinazolinyl]thio]ethanoneEscherichia coli K-12Potency5.017220
1-[2-[(3-cyano-5,7-dimethyl-2-quinolinyl)amino]ethyl]-3-(3-methoxypropyl)thioureaEscherichia coli K-12Potency39.810710
1-[2-[(3-cyano-7-methyl-2-quinolinyl)amino]ethyl]-3-[3-(4-morpholinyl)propyl]thioureaEscherichia coli K-12Potency22.387210
N-(2,4-dimethoxyphenyl)-3-(6-methyl-1H-benzimidazol-2-yl)-1-piperidinecarbothioamideEscherichia coli K-12Potency25.118910
1-[3-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]-1-butanoneEscherichia coli K-12Potency31.622810
3-(5-methyl-2-furanyl)-5-[1-(2-naphthalenylsulfonyl)-3-piperidinyl]-1,2,4-oxadiazoleEscherichia coli K-12Potency39.810710
[4-[5-tert-butyl-3-(phenylmethyl)-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneEscherichia coli K-12Potency10.000010
4-(2-fluorophenyl)-1-[[1-[(4-methoxyphenyl)methyl]-5-tetrazolyl]methyl]-4-piperidinolEscherichia coli K-12Potency31.622810
1-(2-methyl-2,3-dihydroindol-1-yl)-2-[4-[5-(trifluoromethyl)-1-benzotriazolyl]-1-piperidinyl]ethanoneEscherichia coli K-12Potency25.118910
1-(1-tert-butyl-5-tetrazolyl)-N-(phenylmethyl)-1-(3-pyridinyl)-N-(thiophen-2-ylmethyl)methanamineEscherichia coli K-12Potency28.183810
7-(2-ethyl-1-piperidinyl)-5-methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency44.668410
N-[2-(3-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-N',N'-dimethylpropane-1,3-diamineEscherichia coli K-12Potency39.810710
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(4-methyl-2-thiazolyl)acetamideEscherichia coli K-12Potency4.466810
N-[4-[1-(benzenesulfonyl)-2,3-dihydroindol-5-yl]-5-methyl-2-thiazolyl]-2-(4-morpholinyl)acetamideEscherichia coli K-12Potency25.118910
1-[(4-fluorophenyl)methyl]-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-oxo-3H-benzimidazole-5-carboxamideEscherichia coli K-12Potency39.810710
ml106Escherichia coli K-12Potency0.354810
N-(2-furanylmethyl)-6-(3-methoxyphenyl)-N-methyl-4-quinazolinamineEscherichia coli K-12Potency1.412510
6-(3-pyridinyl)-N-(3-pyridinylmethyl)-4-quinazolinamineEscherichia coli K-12Potency44.668410
6-(3-methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineEscherichia coli K-12Potency16.597820
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineEscherichia coli K-12Potency112.202010
N-[2-(1-cyclohexenyl)ethyl]-3-(1,3-dioxo-2-isoindolyl)propanamideEscherichia coli K-12Potency0.631010
3-(4-methoxyphenyl)-3-[[2-(4-methoxyphenyl)-1-oxoethyl]amino]propanoic acidEscherichia coli K-12Potency100.000010
2-[[3-(4-methoxyphenyl)-1,2,4-thiadiazol-5-yl]thio]acetic acid ethyl esterEscherichia coli K-12Potency6.309610
4-[[2-(4-methyl-1-piperidinyl)-1,3-benzothiazol-6-yl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency28.183810
3-(3,4-dimethoxyphenyl)-6,7-dimethoxy-2-methyl-N-(6-methyl-2-pyridinyl)-1-oxo-3,4-dihydroisoquinoline-4-carboxamideEscherichia coli K-12Potency22.387210
3-[6-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-6-oxohexyl]-2-sulfanylidene-1H-quinazolin-4-oneEscherichia coli K-12Potency100.000010
1-(1H-imidazol-5-ylsulfonyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-piperidinecarboxamideEscherichia coli K-12Potency6.309610
5-bromo-N-[6-[[(5-bromo-2-furanyl)-oxomethyl]amino]-2-pyridinyl]-2-furancarboxamideEscherichia coli K-12Potency35.481310
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-[(2-pyridinylthio)methyl]-4-triazolecarboxylic acid propan-2-yl esterEscherichia coli K-12Potency0.891310
3-[4-[(2-hydroxy-5-phenylphenyl)methyl]-1-piperazinyl]propanenitrileEscherichia coli K-12Potency28.183810
2-[(6-fluoro-1,3-benzothiazol-2-yl)amino]-4-thiazolecarboxylic acid ethyl esterEscherichia coli K-12Potency2.511910
3-(1,3-benzodioxol-5-ylmethyl)-7-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-2-sulfanylidene-1H-quinazolin-4-oneEscherichia coli K-12Potency63.095710
N-[3-(1-azepanyl)propyl]-1-[(4-methoxyphenyl)methyl]-5-oxo-3-pyrrolidinecarboxamideEscherichia coli K-12Potency35.481310
N-[3-[4-(2,3-dimethylphenyl)-1-piperazinyl]-3-oxopropyl]-2-(1-oxo-2-isoquinolinyl)acetamideEscherichia coli K-12Potency31.622810
N-(1,3-benzodioxol-5-yl)-3-methyl-6-phenyl-2-imidazo[2,1-b]thiazolecarboxamideEscherichia coli K-12Potency56.234110
1-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methylsulfinyl]ethanoneEscherichia coli K-12Potency28.183810
2-[(3-ethyl-6-methyl-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)thio]-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]acetamideEscherichia coli K-12Potency1.000010
2-[(2-methoxycarbonylanilino)-oxomethyl]-1-cyclohexanecarboxylic acidEscherichia coli K-12Potency2.511910
3-chloro-N-[2-[4-(4-fluorophenyl)-1-piperazinyl]-2-(3-pyridinyl)ethyl]benzamideEscherichia coli K-12Potency112.202010
2-[8-[[bis(phenylmethyl)amino]methyl]-3-methyl-2,6-dioxo-7-purinyl]acetic acid ethyl esterEscherichia coli K-12Potency28.183810
4-[oxo-(4-oxo-5H-thieno[3,2-c]quinolin-2-yl)methyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency2.818410
4-[[2-(4-methoxyphenyl)-6-imidazo[2,1-b][1,3]benzothiazolyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency19.952610
2-[[2-(4-ethoxyphenyl)-5-methyl-4-oxazolyl]methylthio]-N-(2-furanylmethyl)acetamideEscherichia coli K-12Potency17.782810
N-(4-bromo-2-methylphenyl)-3-(1,3-dioxo-2-pyrrolo[3,4-c]pyridinyl)propanamideEscherichia coli K-12Potency2.511910
3-[[4,6-bis(4-morpholinyl)-1,3,5-triazin-2-yl]amino]-3-(2-chlorophenyl)propanoic acid ethyl esterEscherichia coli K-12Potency19.952610
2-[(3,5-dimethyl-4-isoxazolyl)methylthio]-4-ethyl-7,7-dimethyl-5-oxo-6,8-dihydroquinoline-3-carbonitrileEscherichia coli K-12Potency39.810710
2-(2-methoxyethyl)-9-methyl-N-[3-(4-methyl-1-piperidinyl)propyl]-1-oxo-4-pyrido[3,4-b]indolecarboxamideEscherichia coli K-12Potency0.794310
N-(1,3-benzodioxol-5-ylmethyl)-2-[[2-(2-fluorophenyl)-5-methyl-4-oxazolyl]methylthio]acetamideEscherichia coli K-12Potency44.668410
5-(4-piperidinyl)-1,2-dihydropyrazol-3-oneEscherichia coli K-12Potency2.818410
N-[2-(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)ethyl]-1-propanesulfonamideEscherichia coli K-12Potency3.162310
N-[4-[5-[(2-methylphenoxy)methyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideEscherichia coli K-12Potency79.432810
2-[(3-oxo-2-propan-2-yl-2H-imidazo[1,2-c]quinazolin-5-yl)thio]-N-[2-(4-sulfamoylphenyl)ethyl]acetamideEscherichia coli K-12Potency100.000010
3-(4-bromophenyl)-4-(2-furanylmethyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency3.162310
5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinolEscherichia coli K-12Potency1.122010
4-(2,3-dihydroindol-1-yl)-N-[3-(N-ethyl-3-methylanilino)propyl]-3-(1-imidazolyl)-4-oxobutanamideEscherichia coli K-12Potency7.079510
N-[2-(1-tert-butyl-3,4,6-trimethyl-5-pyrazolo[3,4-b]pyridinyl)ethyl]carbamic acid ethyl esterEscherichia coli K-12Potency13.188920
4-hydroxy-1-[1-oxo-2-[[1-oxo-2-(phenylmethoxycarbonylamino)ethyl]amino]propyl]-2-pyrrolidinecarboxylic acid (phenylmethyl) esterEscherichia coli K-12Potency6.309610
3-phenyl-3-(1-tetrazolyl)propanoic acidEscherichia coli K-12Potency112.202010
2-[[5-methyl-2-[4-(methylthio)phenyl]-4-oxazolyl]methylthio]-1-(4-morpholinyl)ethanoneEscherichia coli K-12Potency39.810710
N-(5-chloro-2-methoxyphenyl)-2,4-dimethyl-5-oxazolecarboxamideEscherichia coli K-12Potency100.000010
4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl(3,4-dihydro-2H-quinolin-1-yl)methanoneEscherichia coli K-12Potency89.125110
1-methyl-N-[4-(trifluoromethyl)phenyl]-4-imidazolesulfonamideEscherichia coli K-12Potency39.810710
2-(pyridin-4-ylmethylamino)benzoic acidEscherichia coli K-12Potency0.794310
2-(N-ethylanilino)-4-thieno[3,2-d][1,3]thiazinoneEscherichia coli K-12Potency50.118710
3-[[oxo(2-quinoxalinyl)methyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency39.810710
3,8-dimethyl-4-oxo-7,8,9,10-tetrahydro-6H-thieno[1,2]pyrimido[4,5-a]azepine-2-carboxylic acid ethyl esterEscherichia coli K-12Potency44.668410
N-[2-(2-ethyl-1-piperidinyl)ethyl]-2-[(2-methyl-1,3-benzothiazol-6-yl)sulfonylamino]acetamideEscherichia coli K-12Potency3.548110
N-(2-furanylmethyl)-2-[(3-phenyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)thio]acetamideEscherichia coli K-12Potency2.511910
N-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-2-[[1-oxo-2-(1-oxo-2-isoquinolinyl)ethyl]amino]acetamideEscherichia coli K-12Potency25.118910
3-[4-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-4-oxobutyl]-6,7-diethoxy-2-sulfanylidene-1H-quinazolin-4-oneEscherichia coli K-12Potency28.183810
2-cyclopentyl-4-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-9-methyl-1-pyrido[3,4-b]indoloneEscherichia coli K-12Potency25.118910
4-[2-[[2-[[4-(1,3-benzodioxol-5-yl)-2-thiazolyl]amino]-2-oxoethyl]thio]-1-oxoethyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency39.810710
1-[4-[4-[[1-(4-chlorophenyl)sulfonylcyclopropyl]-oxomethyl]-1-piperazinyl]phenyl]ethanoneEscherichia coli K-12Potency14.125410
2-(2,4-dimethoxyanilino)-N-[3-(4-methyl-1-piperazinyl)propyl]-4-quinolinecarboxamideEscherichia coli K-12Potency25.118910
1-[4-[2-(2,5-dimethyl-1-pyrrolyl)ethyl]-1-piperazinyl]-2-[[3-(4-morpholinyl)-2-quinoxalinyl]thio]ethanoneEscherichia coli K-12Potency57.924420
5-methyl-N-(5-methyl-2-phenyl-3-pyrazolyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency89.125110
6,7-diethoxy-3-[3-(2-oxo-1-pyrrolidinyl)propyl]-2-sulfanylidene-1H-quinazolin-4-oneEscherichia coli K-12Potency0.316210
2-(4-ethoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acidEscherichia coli K-12Potency53.454020
N-[3-(1-azepanyl)propyl]-5-oxo-1-(2-phenylethyl)-3-pyrrolidinecarboxamideEscherichia coli K-12Potency28.183810
1-[oxo-[4-oxo-6-[(4-propan-2-ylphenyl)sulfamoyl]-1H-quinolin-3-yl]methyl]-4-piperidinecarboxamideEscherichia coli K-12Potency39.810710
3-methyl-N,6-diphenyl-2-imidazo[2,1-b]thiazolecarboxamideEscherichia coli K-12Potency11.220210
1-[[4-[(4-fluorophenyl)methyl]-5-thieno[3,2-b]pyrrolyl]-oxomethyl]-N-(2-furanylmethyl)-4-piperidinecarboxamideEscherichia coli K-12Potency25.118910
2-(4-methoxyphenyl)-N-[4-[5-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]acetamideEscherichia coli K-12Potency8.912510
3,4,5-trimethoxy-N-[2-(1-methyl-2-benzimidazolyl)ethyl]benzamideEscherichia coli K-12Potency15.848910
N-[3-(cyclohexylthio)propyl]-2-[[5-methyl-2-(3-methylphenyl)-4-oxazolyl]methylsulfinyl]acetamideEscherichia coli K-12Potency25.118910
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-methyl-1-piperidinyl)-2-phenylacetamideEscherichia coli K-12Potency50.118710
[4-[6-(4-morpholinyl)-3-pyridazinyl]-1-piperazinyl]-(2-pyridin-4-yl-4-quinolinyl)methanoneEscherichia coli K-12Potency25.118910
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-methyl-4-oxo-1-phthalazinyl)acetamideEscherichia coli K-12Potency15.848910
N-ethyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(phenylmethyl)propanamideEscherichia coli K-12Potency35.716820
N,N-diethyl-4-[[5-oxo-6-(phenylmethyl)-7H-pyrrolo[3,4-b]pyridin-7-yl]amino]benzenesulfonamideEscherichia coli K-12Potency35.481310
N-[4-methyl-2-(4-methyl-1-piperazinyl)-6-quinolinyl]-1,3-benzodioxole-5-carboxamideEscherichia coli K-12Potency31.622810
2-[[2-(3,4-dimethoxyphenyl)-5-methyl-4-oxazolyl]methylsulfinyl]-N-[3-(1-pyrrolidinyl)propyl]acetamideEscherichia coli K-12Potency35.481310
1-(1,3-benzoxazol-2-yl)-N-[(2,5-dimethoxyphenyl)methyl]-3-piperidinecarboxamideEscherichia coli K-12Potency14.125410
1-methyl-N-[4-(4-morpholinyl)phenyl]-2-quinolinimineEscherichia coli K-12Potency89.125110
N-[2-(dimethylamino)ethyl]-2-[3-(4-methylphenyl)-6-oxo-1-pyridazinyl]acetamideEscherichia coli K-12Potency5.011910
2-[(3-bromo-5,7-dimethyl-2-imidazo[1,2-a]pyrimidinyl)methylthio]-1,3-benzoxazoleEscherichia coli K-12Potency28.183810
4-[2-(1-cyclohexenyl)ethyl]-1-cyclohexyl-3-pyridin-4-ylpiperazine-2,5-dioneEscherichia coli K-12Potency25.118910
N-ethyl-3-[4-morpholinyl(oxo)methyl]-4-oxo-N-phenyl-1H-quinoline-6-sulfonamideEscherichia coli K-12Potency100.000010
LSM-17343Escherichia coli K-12Potency1.122010
2-(2-methoxyethyl)-9-methyl-4-[(4-methyl-1-piperidinyl)-oxomethyl]-1-pyrido[3,4-b]indoloneEscherichia coli K-12Potency28.183810
N-[3-(1-azepanyl)propyl]-2-(4-morpholinyl)-3-oxo-4H-1,4-benzothiazine-6-carboxamideEscherichia coli K-12Potency39.810710
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-piperidinecarboxamideEscherichia coli K-12Potency31.622810
2-(1-ethoxycarbonyl-4-piperidinyl)-1,3-dioxo-5-isoindolecarboxylic acidEscherichia coli K-12Potency0.707910
4-[1,3-dioxo-3-[(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)amino]propyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency11.220210
2-[[2-(2-ethyl-1-piperidinyl)-2-oxoethyl]thio]-3-methyl-5H-pyrimido[5,4-b]indol-4-oneEscherichia coli K-12Potency19.952610
7-[(4-methyl-1-piperazinyl)methyl]-5-(phenylmethoxymethyl)-8-quinolinolEscherichia coli K-12Potency40.676520
3,4-dihydro-2H-quinolin-1-yl-[5-(4-methoxyphenyl)-3-isoxazolyl]methanoneEscherichia coli K-12Potency25.118910
3,4-dimethylbenzoic acid (6-methyl-3-pyridinyl) esterEscherichia coli K-12Potency0.794310
3-methyl-N-[2-(4-morpholinyl)ethyl]-1-phenyl-5-thieno[2,3-c]pyrazolecarboxamideEscherichia coli K-12Potency25.118910
2-(3-acetyl-2-methyl-5-phenyl-1-pyrrolyl)-N-(thiophen-2-ylmethyl)acetamideEscherichia coli K-12Potency10.000010
4-(4-methyl-1-oxido-2-triazol-1-iumyl)benzoic acidEscherichia coli K-12Potency0.707910
1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-(4-ethylphenyl)ureaEscherichia coli K-12Potency89.125110
3-(4-fluorophenyl)-6-[2-oxo-2-(1-pyrrolidinyl)ethyl]-7-triazolo[4,5-d]pyrimidinoneEscherichia coli K-12Potency28.183810
6-(1-azepanylsulfonyl)-1-ethyl-N-(2-furanylmethyl)-4-oxo-3-quinolinecarboxamideEscherichia coli K-12Potency19.952610
3-(2-chlorophenyl)-5-methyl-N-[3-(3-methyl-2-imidazo[1,2-a]pyrimidinyl)phenyl]-4-isoxazolecarboxamideEscherichia coli K-12Potency28.183810
2-[[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-thieno[3,2-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideEscherichia coli K-12Potency0.316210
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-[[[3,4-dioxo-2-(1-pyrrolidinyl)-1-cyclobutenyl]amino]methyl]-1-cyclohexanecarboxamideEscherichia coli K-12Potency1.584910
1-[2-(1-oxo-2-thiophen-2-ylethoxy)ethyl]-5-[(1-oxo-2-thiophen-2-ylethyl)amino]-4-pyrazolecarboxylic acid ethyl esterEscherichia coli K-12Potency2.511910
7-(5-chloro-2-methoxyanilino)-6-[(4-methoxyphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-oneEscherichia coli K-12Potency39.810710
N-[2-[4-(3-chlorophenyl)-1-piperazinyl]ethyl]-[1,2,4]triazolo[4,3-a]quinoxalin-4-amineEscherichia coli K-12Potency1.258910
N-[3-(N-ethylanilino)propyl]-2,4-dimethyl-6-oxo-3-pyrancarboxamideEscherichia coli K-12Potency8.912510
N-(4-ethoxyphenyl)-2-(hydroxymethyl)benzamideEscherichia coli K-12Potency0.794310
2-(2,5-dimethoxyanilino)-N-[3-(4-morpholinyl)propyl]-4-quinolinecarboxamideEscherichia coli K-12Potency25.118910
4-[[9-methyl-2-(2-methylpropyl)-1-oxo-4-pyrido[3,4-b]indolyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency19.952610
5-(4-methoxyphenyl)-N-propan-2-yl-3-isoxazolecarboxamideEscherichia coli K-12Potency1.995310
5-amino-1-(3,5-dimethylphenyl)-N-(phenylmethyl)-4-triazolecarboxamideEscherichia coli K-12Potency3.981110
[4-(2-pyrimidinyl)-1-piperazinyl]-[1-[4-(2-pyrimidinyl)-1-piperazinyl]-4-isoquinolinyl]methanoneEscherichia coli K-12Potency22.387210
2-amino-4-[4-(methylthio)phenyl]-5-oxo-1-phenyl-4,6,7,8-tetrahydroquinoline-3-carbonitrileEscherichia coli K-12Potency1.122010
N-[[4-(dimethylamino)phenyl]methyl]-3-ethyl-N-(2-furanylmethyl)-5-methyl-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideEscherichia coli K-12Potency39.810710
N-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-2-[(1-ethyl-2-oxo-4-quinolinyl)oxy]acetamideEscherichia coli K-12Potency22.387210
acetic acid [2-(1-acetyl-6-indolyl)-2-oxoethyl] esterEscherichia coli K-12Potency100.000010
1-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methyl]-N-(3-pyridinylmethyl)-4-piperidinecarboxamideEscherichia coli K-12Potency7.079510
6,7-dimethoxy-N-[(5-methyl-2-furanyl)methyl]-2-(2-methylpropyl)-1-oxo-4-isoquinolinecarboxamideEscherichia coli K-12Potency10.000010
N4,N5-bis(2-ethoxyphenyl)-1H-imidazole-4,5-dicarboxamideEscherichia coli K-12Potency3.548110
N-[2-(1-cyclohexenyl)ethyl]-1-[cyclopropyl(oxo)methyl]-2,3-dihydroindole-5-sulfonamideEscherichia coli K-12Potency28.183810
6-[(2,5-dimethylphenyl)methyl]-3-(4-fluorophenyl)-7-triazolo[4,5-d]pyrimidinoneEscherichia coli K-12Potency100.000010
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-1-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methyl]-4-piperidinecarboxamideEscherichia coli K-12Potency25.118910
N-[(2-methyl-4-thiazolyl)methyl]-4-phenoxybenzenesulfonamideEscherichia coli K-12Potency56.234110
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamideEscherichia coli K-12Potency0.501210
N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideEscherichia coli K-12Potency31.622810
4-(3-methoxyphenyl)-2-(4-phenyl-1-piperazinyl)-6-(trifluoromethyl)pyrimidineEscherichia coli K-12Potency0.707910
N-(2-furanylmethyl)-3-[3-[(4-methoxyphenyl)methyl]-2-imidazo[4,5-b]pyridinyl]propanamideEscherichia coli K-12Potency50.118710
N-ethyl-N-(2-ethylphenyl)-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideEscherichia coli K-12Potency10.000010
2-[2,4-dioxo-3-(phenylmethyl)-1-quinazolinyl]-N-(5-methyl-3-isoxazolyl)acetamideEscherichia coli K-12Potency89.125110
4-morpholinecarboxylic acid [4-(2-amino-3-cyano-5-oxo-4,6,7,8-tetrahydro-1-benzopyran-4-yl)-2,6-dimethoxyphenyl] esterEscherichia coli K-12Potency0.631010
N-(3-acetylphenyl)-3,5-dimethyl-4-isoxazolesulfonamideEscherichia coli K-12Potency2.511910
8-[[4-(5-chloro-2-methylphenyl)-1-piperazinyl]methyl]-3-methyl-7-(2-phenylethyl)purine-2,6-dioneEscherichia coli K-12Potency1.584910
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[N-[(3,5-dimethyl-4-isoxazolyl)sulfonyl]-4-methylanilino]acetamideEscherichia coli K-12Potency39.810710
2-(2-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneEscherichia coli K-12Potency63.095710
2-[[3-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]-N-(2-oxolanylmethyl)acetamideEscherichia coli K-12Potency18.317420
N-[3-(cyclohexylthio)propyl]-1-[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]-3-piperidinecarboxamideEscherichia coli K-12Potency25.118910
4-[4-oxo-2-[[2-oxo-2-[(phenylmethyl)amino]ethyl]thio]-3-quinazolinyl]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency63.095710
cyclobutyl-[5-[(2-ethyl-1-piperidinyl)sulfonyl]-2,3-dihydroindol-1-yl]methanoneEscherichia coli K-12Potency17.782810
N-[4-[(2,3-dihydro-1,4-benzodioxin-6-ylamino)-oxomethyl]phenyl]-2-oxolanecarboxamideEscherichia coli K-12Potency11.220210
2-[4-[2-(3,5-dimethoxyanilino)-2-oxoethyl]-1-piperazinyl]-N-(4-ethoxyphenyl)acetamideEscherichia coli K-12Potency35.481310
2-cyclohexyl-9-methyl-1-oxo-N-[3-(2-oxo-1-pyrrolidinyl)propyl]-4-pyrido[3,4-b]indolecarboxamideEscherichia coli K-12Potency35.481310
1-[3-[2-(dimethylamino)ethylamino]-3-oxopropyl]-2-methyl-5-(4-methylphenyl)-3-pyrrolecarboxylic acid ethyl esterEscherichia coli K-12Potency14.125410
N-[2-(3,4-diethoxyphenyl)ethyl]-1-[6-(4-morpholinyl)-3-pyridazinyl]-4-piperidinecarboxamideEscherichia coli K-12Potency40.074820
2-[(1-acetyl-2-benzimidazolyl)thio]-N-(2-methoxyphenyl)acetamideEscherichia coli K-12Potency35.481310
8-(2-propoxyphenyl)-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]quinolin-6-oneEscherichia coli K-12Potency56.234110
1-[(2-ethoxyphenyl)methyl]-3-thiophen-2-ylureaEscherichia coli K-12Potency50.118710
N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-[(5-methyl-2-furanyl)methylamino]-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]carbamic acid (phenylmethyl) esterEscherichia coli K-12Potency89.125110
5-methyl-N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-(2-naphthalenylamino)-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]-3-isoxazolecarboxamideEscherichia coli K-12Potency0.141310
2,5-dimethyl-N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-(2-naphthalenylamino)-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]-3-pyrazolecarboxamideEscherichia coli K-12Potency48.022420
6-methyl-N-(2-methylphenyl)-2-oxo-4-phenyl-3,4-dihydro-1H-pyrimidine-5-carboxamideEscherichia coli K-12Potency44.668410
[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency35.481310
4-chlorobenzoic acid (5-methyl-2-pyridin-4-yl-4-thiazolyl) esterEscherichia coli K-12Potency63.095710
6-[oxo-[2-[oxo-(2-phenylethylamino)methyl]anilino]methyl]-1-cyclohex-3-enecarboxylic acidEscherichia coli K-12Potency100.000010
2,6-dimethyl-4-(4-phenyl-2-quinolinyl)morpholineEscherichia coli K-12Potency35.481310
N-[[4-(dimethylamino)phenyl]methyl]-1-ethyl-5-benzimidazolamineEscherichia coli K-12Potency112.202010
6-ethyl-2-[[[4-(4-morpholinylsulfonyl)phenyl]-oxomethyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamideEscherichia coli K-12Potency25.118910
3-(2-benzofuranyl)-N-(4-nitrophenyl)-1-phenyl-4-pyrazolecarboxamideEscherichia coli K-12Potency100.000010
2-(1-benzo[e]benzofuranyl)-N-[4-methoxy-3-(4-morpholinylsulfonyl)phenyl]acetamideEscherichia coli K-12Potency39.810710
1-(4-methoxyphenyl)-4-[(4-methylphenyl)thio]-6-oxo-3-pyridazinecarboxylic acid methyl esterEscherichia coli K-12Potency0.707910
3-(5-ethyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency7.079510
N-(5-acetyl-2-phenyl-4-sulfanylidene-1H-pyrimidin-6-yl)benzamideEscherichia coli K-12Potency61.193620
4-butyl-3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency44.668410
1,3-diphenyl-4-pyrazolecarboxylic acid [2-[(3,5-dichloro-2-pyridinyl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency22.387210
(5-bromo-2-furanyl)-[2-[(3-methylphenyl)methylthio]-4,5-dihydroimidazol-1-yl]methanoneEscherichia coli K-12Potency0.354810
N-[4-(difluoromethoxy)phenyl]-4-(phenylmethyl)-1-piperazinecarbothioamideEscherichia coli K-12Potency44.668410
2-(trifluoromethyl)-3-imidazo[1,2-a]pyrimidinecarboxylic acid ethyl esterEscherichia coli K-12Potency0.707910
1-(2-furanylmethyl)-3-(2-methylphenyl)-1-(3-pyridinylmethyl)thioureaEscherichia coli K-12Potency0.794310
2-phenoxy-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamideEscherichia coli K-12Potency5.177420
4-[(4-acetyl-2-methoxyphenyl)methoxy]-3-methoxybenzoic acid [1-(carbamoylamino)-1-oxopropan-2-yl] esterEscherichia coli K-12Potency31.622810
4-[[7-[(4-fluorophenyl)methyl]-1,3-dimethyl-2,6-dioxo-8-purinyl]methyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency22.387210
4-[[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholineEscherichia coli K-12Potency12.313020
N-[4-(methoxymethyl)-6-methyl-2-oxo-1H-quinolin-7-yl]cyclopropanecarboxamideEscherichia coli K-12Potency0.501210
2-[(4-methyl-5-sulfanylidene-1,3,4-thiadiazol-2-yl)thio]acetic acid ethyl esterEscherichia coli K-12Potency4.466810
N-(6-ethoxy-1,3-benzothiazol-2-yl)-4-methoxy-3-(4-morpholinylsulfonyl)benzamideEscherichia coli K-12Potency39.810710
2-[[2-[(2-methoxyphenyl)methylamino]-2-oxoethyl]thio]-3-pyridinecarboxylic acid [2-[(2-methoxyphenyl)methylamino]-2-oxoethyl] esterEscherichia coli K-12Potency35.481310
N-[4-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-(4-methoxyphenyl)acetamideEscherichia coli K-12Potency1.995310
N-[(4-methoxyphenyl)methyl]-2-(phenylmethyl)-4-thiazolecarboxamideEscherichia coli K-12Potency0.707910
2-[[[3-(2,5-dioxo-1-pyrrolidinyl)phenyl]-oxomethyl]amino]-4-(4-phenylphenyl)-3-thiophenecarboxylic acid ethyl esterEscherichia coli K-12Potency100.000010
5-[2-(4-bromophenyl)-2-oxoethyl]-1,3-diphenyl-2-sulfanylidene-4-imidazolidinoneEscherichia coli K-12Potency2.818410
1,1-dimethyl-3-[3-(4-morpholinyl)propyl]-3-(1-naphthalenylmethyl)ureaEscherichia coli K-12Potency28.183810
N-[2-(4-morpholinyl)ethyl]-2-(4-propan-2-yloxyphenyl)-4-quinolinecarboxamideEscherichia coli K-12Potency28.183810
5-[[(3,4-dichloroanilino)-sulfanylidenemethyl]amino]-1H-pyrazole-4-carboxylic acid methyl esterEscherichia coli K-12Potency0.707910
(4-methylphenyl)-[4-[4-nitro-3-(3-pyridinylmethylamino)phenyl]-1-piperazinyl]methanoneEscherichia coli K-12Potency39.810710
2-(4-benzofuro[3,2-d]pyrimidinylthio)-N-(3-methylphenyl)acetamideEscherichia coli K-12Potency2.511910
2-[[3-(2-methoxyethyl)-6-methyl-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]-N-(2-oxolanylmethyl)acetamideEscherichia coli K-12Potency10.000010
1-(2,5-dimethoxyphenyl)-3-[5-(2-methyl-1-piperidinyl)-1,3,4-thiadiazol-2-yl]ureaEscherichia coli K-12Potency25.118910
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinolEscherichia coli K-12Potency0.631010
ro 41-0960Escherichia coli K-12Potency5.623410
6-[2-butylimino-3-(cyclopentylideneamino)-4-thiazolyl]-4H-1,4-benzoxazin-3-oneEscherichia coli K-12Potency22.387210
cgp 13501Escherichia coli K-12Potency8.912510
(S)-4',5,7-Trihydroxy-6-prenylflavanoneEscherichia coli K-12Potency8.912510
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyrimidinylthio)acetamideEscherichia coli K-12Potency27.871020
[3-(2,3-dihydroindol-1-ylsulfonyl)phenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency25.118910
4-methyl-1-piperazinecarbodithioic acid [2-[(2-methyl-3-phenyl-3H-1,5-benzodiazepin-4-yl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency31.622810
6-[4-oxo-2-[(4-oxo-2-pyrido[1,2-a]pyrimidinyl)methylthio]-3-thieno[3,2-d]pyrimidinyl]hexanoic acidEscherichia coli K-12Potency0.631010
1,3-dimethyl-8-[[methyl-(phenylmethyl)amino]methyl]-7-(2-methylpropyl)purine-2,6-dioneEscherichia coli K-12Potency16.700620
[1-[2-(2-methylphenoxy)ethyl]-3-indolyl]-(4-methyl-1-piperazinyl)methanethioneEscherichia coli K-12Potency35.481310
N-[(1,2-dimethyl-5-indolyl)methyl]-2-methyl-3-nitrobenzamideEscherichia coli K-12Potency79.432810
N-(6-acetamido-3-prop-2-enyl-1,3-benzothiazol-2-ylidene)cyclohexanecarboxamideEscherichia coli K-12Potency3.109920
N4-(2-furanylmethyl)-N2-(3-methoxyphenyl)-5-nitropyrimidine-2,4,6-triamineEscherichia coli K-12Potency89.125110
N-[[[(2-chlorophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2-nitrobenzamideEscherichia coli K-12Potency25.118910
N-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propyl]-3-(3-oxo-1,4-benzoxazin-4-yl)propanamideEscherichia coli K-12Potency22.387210
6-bromo-2-(4-methylphenyl)-N-[(1-methyl-4-pyrazolyl)methyl]-4-quinolinecarboxamideEscherichia coli K-12Potency0.631010
1-(1-naphthalenyl)-3-[[2-(2-nitrophenoxy)-1-oxoethyl]amino]ureaEscherichia coli K-12Potency28.183810
N-(2-furanylmethyl)-2-[[5-[(2-methyl-1H-indol-3-yl)methyl]-1,3,4-oxadiazol-2-yl]thio]acetamideEscherichia coli K-12Potency17.782810
4-[[3-[anilino(oxo)methyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidEscherichia coli K-12Potency0.562310
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-dimethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolamineEscherichia coli K-12Potency11.220210
5-(3,4-dimethoxyphenyl)-N-(3-pyridinyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency34.702620
4-[4-dimethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolyl]morpholineEscherichia coli K-12Potency31.622810
2-[4-methoxy-3-(4-morpholinylmethyl)phenyl]-3-(phenylmethyl)-1,2-dihydroquinazolin-4-oneEscherichia coli K-12Potency39.810710
2-[[4-(4-chlorophenyl)-5-sulfanylidene-1,3,4-thiadiazol-2-yl]thio]-N-(1,1-dioxo-3-thiolanyl)-N-(2-methylpropyl)acetamideEscherichia coli K-12Potency9.068820
2-methyl-1,3-bis(phenylmethoxy)benzeneEscherichia coli K-12Potency0.562310
N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]-5-nitro-2-thiophenecarboxamideEscherichia coli K-12Potency3.162310
6-[2-(1-azepanyl)-2-oxoethoxy]-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-oneEscherichia coli K-12Potency56.234110
2-methyl-5-[(4-phenyl-1-piperazinyl)-(3,4,5-trimethoxyphenyl)methyl]-6-thiazolo[3,2-b][1,2,4]triazololEscherichia coli K-12Potency35.481310
N-[[4-[[4-(4-fluorophenyl)-1-piperazinyl]-oxomethyl]cyclohexyl]methyl]-2-thiophenesulfonamideEscherichia coli K-12Potency22.387210
2-[(5,7-dimethyl-2-imidazo[1,2-a]pyrimidinyl)methylthio]acetic acidEscherichia coli K-12Potency100.000010
2-methyl-1-phenyl-5-benzimidazolecarboxylic acid [2-(2-methoxyanilino)-2-oxoethyl] esterEscherichia coli K-12Potency89.125110
N-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-quinoline-6-sulfonamideEscherichia coli K-12Potency0.562310
5-(4-ethoxyphenyl)-1,3-diphenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-4,6-dioneEscherichia coli K-12Potency2.511910
2-(1,3-benzothiazol-2-ylthio)-N-[2-hydroxy-5-(4-morpholinylsulfonyl)phenyl]acetamideEscherichia coli K-12Potency39.810710
8-[[4-[2-furanyl(oxo)methyl]-1-piperazinyl]methyl]-1,3-dimethyl-7-propylpurine-2,6-dioneEscherichia coli K-12Potency5.623410
N-[3-[(3-chlorophenyl)sulfamoyl]-4-methylphenyl]-3-(4-nitrophenyl)-3-oxopropanamideEscherichia coli K-12Potency7.079510
2-(4-methoxyphenyl)-N-[2-(4-morpholinyl)-5-(4-morpholinylsulfonyl)phenyl]-4-quinolinecarboxamideEscherichia coli K-12Potency15.848910
N-(3-methylbutyl)-6-(4-morpholinylsulfonyl)-2-pyridin-4-yl-4-quinolinecarboxamideEscherichia coli K-12Potency28.183810
1-(3-chloro-4-fluorophenyl)-4-[(4-methyl-1-piperazinyl)-oxomethyl]-2-pyrrolidinoneEscherichia coli K-12Potency1.122010
3-[5-(dimethylsulfamoyl)-1-ethyl-2-benzimidazolyl]propanoic acidEscherichia coli K-12Potency112.202010
2-(cyclohexylamino)-N-[(diphenylmethylene)amino]propanamideEscherichia coli K-12Potency39.810710
1-(1,3-benzodioxol-5-yl)-3-(4-fluorophenyl)ureaEscherichia coli K-12Potency39.810710
3-ethyl-2-sulfanylidene-5-thiophen-2-yl-1H-thieno[2,3-d]pyrimidin-4-oneEscherichia coli K-12Potency28.183810
LSM-1924Escherichia coli K-12Potency7.233420
1-[(4-chlorophenyl)methyl]-3-(3-fluorophenyl)-1-(3,3,3-trifluoro-2-hydroxypropyl)ureaEscherichia coli K-12Potency0.631010
2-(2-cyanophenyl)sulfinyl-N-methylbenzamideEscherichia coli K-12Potency50.118710
5-[(4-chlorophenyl)-oxomethyl]-4-hydroxy-6-[5-(2-nitrophenyl)-2-furanyl]-4-(trifluoromethyl)-1,3-diazinan-2-oneEscherichia coli K-12Potency39.810710
N-(3-chlorophenyl)-5-oxo-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindole-1-carboxamideEscherichia coli K-12Potency56.234110
2-(4-ethoxyphenyl)-N-[3-(1-imidazolyl)propyl]-4-quinolinecarboxamideEscherichia coli K-12Potency39.810710
4-[[anilino-(4-methylphenyl)methyl]-propoxyphosphoryl]-N,N-dimethylanilineEscherichia coli K-12Potency25.118910
1-butyl-4,6-dimethyl-3-(2-methylphenyl)sulfonyl-2-pyridinoneEscherichia coli K-12Potency25.118910
4-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitrobenzoic acid methyl esterEscherichia coli K-12Potency0.316210
2-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitropyridineEscherichia coli K-12Potency112.202010
phosphoric acid (3-methylphenyl) phenyl (2,2,2-trifluoro-1-phenylethyl) esterEscherichia coli K-12Potency2.511910
5-cyano-6-[4-(4-methoxyphenyl)-1-piperazinyl]-2-oxo-1H-pyridine-3-carboxylic acid ethyl esterEscherichia coli K-12Potency1.995310
N-[3-fluoro-4-(4-phenyl-1-piperazinyl)phenyl]-2-(4-morpholinyl)acetamideEscherichia coli K-12Potency8.912510
4-[[[2-(4-methoxyphenyl)-3-thiazolidinyl]-sulfanylidenemethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency3.981110
6-amino-4-(1-cyclohex-2-enyl)-3-thiophen-2-yl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileEscherichia coli K-12Potency0.707910
7-(4-ethoxyphenyl)-5-(3-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineEscherichia coli K-12Potency51.256020
2-hydroxy-2-pentyl-N'-phenylheptanehydrazideEscherichia coli K-12Potency28.183810
AnthraniloyllycoctonineEscherichia coli K-12Potency42.800020
3,5-diethyl-2-(3-hydroxypropylamino)-5-methyl-6H-benzo[h]quinazolin-4-oneEscherichia coli K-12Potency15.848910
6-(5,6-Dihydroxy-4-oxo-2-phenylchromen-7-yl)oxy-3,4,5-trihydroxyoxane-2-carboxylic acidEscherichia coli K-12Potency100.000010
N-[(5-quinolinylamino)-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency3.981110
2-Chloro-1-[5-(3,4-dimethoxyphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneEscherichia coli K-12Potency3.548110
2-[(2,6-dichlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinoneEscherichia coli K-12Potency112.202010
2-amino-4-(2-fluorophenyl)-6-(3-pyridinyl)-3-pyridinecarbonitrileEscherichia coli K-12Potency4.466810
N-(4-phenylmethoxyphenyl)-3-[4-(phenylmethyl)-1-piperazinyl]propanamideEscherichia coli K-12Potency28.183810
2-amino-7,7-dimethyl-4-(4-methylphenyl)-5-oxo-6,8-dihydro-4H-1-benzopyran-3-carbothioamideEscherichia coli K-12Potency44.668410
5-[3-(3,5-dimethyl-1,2,4-triazol-1-yl)-2-hydroxypropoxy]-2-methyl-1-(phenylmethyl)-3-indolecarboxylic acid ethyl esterEscherichia coli K-12Potency13.699620
1-(4-chlorophenyl)-3-[2-(2-furanylmethyl)cyclohexyl]ureaEscherichia coli K-12Potency6.309610
4-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-3-oxobutanoic acid ethyl esterEscherichia coli K-12Potency3.162310
2-amino-6-methyl-4-(3-pyridinyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrileEscherichia coli K-12Potency5.011910
1-[4-(3-chlorophenyl)-1-piperazinyl]-2-phenyl-1-butanoneEscherichia coli K-12Potency31.622810
4-(2-chlorophenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidineEscherichia coli K-12Potency0.794310
N-(3,5-dimethylphenyl)-2-(2-nitroethyl)benzamideEscherichia coli K-12Potency0.141310
6-nitro-3-phenyl-1H-benzimidazole-2-thioneEscherichia coli K-12Potency0.707910
or486Escherichia coli K-12Potency3.162310
N-(4-fluorophenyl)-5-methyl-1H-indole-2-carboxamideEscherichia coli K-12Potency7.943310
5-nitro-2-thiophenecarboxylic acid [1-[(3,5-dichloro-2-pyridinyl)amino]-1-oxopropan-2-yl] esterEscherichia coli K-12Potency50.118710
2-[4-oxo-2-(1-piperidinyl)-5-thiazolyl]-N-[3-(trifluoromethyl)phenyl]acetamideEscherichia coli K-12Potency10.153720
LSM-22738Escherichia coli K-12Potency15.848910
7-[(3-hydroxy-3,4-dihydro-2H-benzo[h]quinolin-1-yl)methyl]-5-thiazolo[3,2-a]pyrimidinoneEscherichia coli K-12Potency25.118910
2-[(4-chloro-3-nitrophenyl)-oxomethyl]benzoic acid [2-[di(propan-2-yl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency39.810710
3-[[4-(diphenylmethyl)-1-piperazinyl]-oxomethyl]-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-12-oneEscherichia coli K-12Potency25.118910
N-[2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl]-4-nitroanilineEscherichia coli K-12Potency1.778310
N-[2-(2-chlorophenoxy)ethyl]-2-(1H-indol-3-yl)-2-oxoacetamideEscherichia coli K-12Potency22.387210
2-[(5-anilino-1,3,4-thiadiazol-2-yl)thio]-N-[3-(1-piperidinylsulfonyl)phenyl]acetamideEscherichia coli K-12Potency31.622810
2-[[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamideEscherichia coli K-12Potency44.668410
7-methoxy-2-phenylimino-1-benzopyran-3-carboxamideEscherichia coli K-12Potency79.432810
4-oxo-4-thiophen-2-ylbutanoic acid [2-(ethylamino)-2-oxoethyl] esterEscherichia coli K-12Potency21.314520
6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylic acid [1-[1-[4-(difluoromethoxy)phenyl]-2,5-dimethyl-3-pyrrolyl]-1-oxopropan-2-yl] esterEscherichia coli K-12Potency41.429920
N-[6-amino-2,4-dioxo-1-(phenylmethyl)-5-pyrimidinyl]-N-ethyl-2-(2-methyl-2,3-dihydroindol-1-yl)acetamideEscherichia coli K-12Potency50.118710
N-[1-[(cyclohexylamino)-oxomethyl]cyclohexyl]-N-(thiophen-2-ylmethyl)-2-pyrazinecarboxamideEscherichia coli K-12Potency2.238710
butanoic acid [2-oxo-2-(4-phenyldiazenylanilino)ethyl] esterEscherichia coli K-12Potency1.258910
4-(3,5-dimethyl-1-piperidinyl)-N-[5-(2-methylpropyl)-1,3,4-thiadiazol-2-yl]-4-oxobutanamideEscherichia coli K-12Potency3.162310
2-(4-morpholinyl)-5-(1-piperidinylsulfonyl)benzoic acid [2-[2-(4-fluorophenyl)ethylamino]-2-oxoethyl] esterEscherichia coli K-12Potency17.782810
vu0155094Escherichia coli K-12Potency54.456220
2-(2-chlorophenyl)-N-[3-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)phenyl]-4-quinolinecarboxamideEscherichia coli K-12Potency5.623410
3-[[(3-methoxyphenyl)-oxomethyl]amino]-2-benzofurancarboxamideEscherichia coli K-12Potency9.149820
2-phenyl-4-quinolinecarboxylic acid [2-[2-chloro-5-(dimethylsulfamoyl)anilino]-2-oxoethyl] esterEscherichia coli K-12Potency2.818410
2-amino-4-(3,4-dimethoxyphenyl)-7,7-dimethyl-5-oxo-1-(3-pyridinyl)-6,8-dihydro-4H-quinoline-3-carbonitrileEscherichia coli K-12Potency2.818410
3-(2-chlorophenyl)-N-[5-(2,4-dichlorophenyl)-1,3,4-thiadiazol-2-yl]-5-methyl-4-isoxazolecarboxamideEscherichia coli K-12Potency24.840120
N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]-2-(3-pyridinyl)ethyl]-2-thiophenesulfonamideEscherichia coli K-12Potency10.000010
9,10-dioxo-1-anthracenecarboxylic acid [2-(2,3-dimethylanilino)-2-oxoethyl] esterEscherichia coli K-12Potency100.000010
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-fluorophenyl)-2-(2-methoxyethyl)-1-oxo-3,4-dihydroisoquinoline-4-carboxamideEscherichia coli K-12Potency11.220210
N-[4-(phenoxymethyl)-2-thiazolyl]-1-adamantanecarboxamideEscherichia coli K-12Potency100.000010
7-chloro-4-[(2-fluorophenyl)-oxomethyl]-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-oneEscherichia coli K-12Potency5.011910
2-[(6-methyl-4-spiro[3,4-dihydro-2H-1-benzopyran-2,1'-cyclopentane]yl)thio]-N-(2-phenylethyl)acetamideEscherichia coli K-12Potency89.125110
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidEscherichia coli K-12Potency2.238710
4-[4-diethoxyphosphoryl-2-(1-naphthalenyl)-5-oxazolyl]morpholineEscherichia coli K-12Potency25.118910
N-[3-[3-(1-piperidinylsulfonyl)anilino]-2-quinoxalinyl]benzenesulfonamideEscherichia coli K-12Potency3.162310
[4-(2,3-dimethylphenyl)-1-piperazinyl]-[5-[(4-methoxyphenyl)sulfonylmethyl]-2-furanyl]methanoneEscherichia coli K-12Potency16.597820
N-(5-chloro-2-methoxyphenyl)-2-[[3-(2-methoxyethyl)-6-methyl-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]thio]acetamideEscherichia coli K-12Potency25.118910
(6-bromo-5-methoxy-2-methyl-3-benzofuranyl)-[4-(2-methylphenyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency39.810710
N-[3-[(4-ethoxyphenyl)-[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-4,5-dimethyl-2-thiophenyl]benzamideEscherichia coli K-12Potency15.848910
2-bromo-N-[[(2-methylcyclohexyl)amino]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency0.562310
4-amino-3-(3,4-dimethylphenyl)-N-(2-fluorophenyl)-2-sulfanylidene-5-thiazolecarboxamideEscherichia coli K-12Potency100.000010
N-(2-oxo-1-benzopyran-3-yl)cyclohexanecarboxamideEscherichia coli K-12Potency39.810710
N-[5-(2-chlorophenyl)-1,3,4-thiadiazol-2-yl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]butanamideEscherichia coli K-12Potency3.162310
N-[3-(2-methoxyethyl)-6-methylsulfonyl-1,3-benzothiazol-2-ylidene]-2-nitrobenzamideEscherichia coli K-12Potency50.118710
N,6-dimethyl-2-[[[4-[(2-methyl-1-piperidinyl)sulfonyl]phenyl]-oxomethyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamideEscherichia coli K-12Potency15.848910
2-[(3-fluorophenyl)-(2-pyridinylamino)methyl]-3-hydroxy-6-(hydroxymethyl)-4-pyranoneEscherichia coli K-12Potency26.200020
2-(5-bromo-2-thiophenyl)-N-(4-methyl-1-piperazinyl)-4-quinolinecarboxamideEscherichia coli K-12Potency17.782810
1-(2-methylphenyl)-3-(6,7,8,9-tetrahydro-5H-carbazol-3-ylmethyl)thioureaEscherichia coli K-12Potency39.810710
3-(2-methoxyphenyl)-2,5-dimethyl-7-[4-(phenylmethyl)-1-piperazinyl]pyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency8.116020
7-(1-azepanyl)-3-(2-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency18.446920
7-methoxy-N-(3-pyridinylmethyl)-2-furo[2,3-b]quinolinecarboxamideEscherichia coli K-12Potency1.778310
2-cyclopentylacetic acid [2-[(3-chloro-9,10-dioxo-2-anthracenyl)amino]-2-oxoethyl] esterEscherichia coli K-12Potency70.794610
LSM-16386Escherichia coli K-12Potency14.125410
4-(3,4-dimethylphenyl)-3-(5-methyl-3-isoxazolyl)-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency100.000010
3-[3-[4-(4-methoxyphenyl)-1-piperazinyl]propyl]-2-sulfanylidene-1H-pyrido[2,3-d]pyrimidin-4-oneEscherichia coli K-12Potency0.794310
N-cyclopentyl-2-(2,3-dihydroindol-1-yl)-2-(4-methoxyphenyl)acetamideEscherichia coli K-12Potency2.511910
6-[oxo-[2-[oxo-[4-(4-propan-2-ylphenyl)-1-piperazinyl]methyl]anilino]methyl]-1-cyclohex-3-enecarboxylic acidEscherichia coli K-12Potency3.162310
1-[(6-hydroxy-2-methyl-5-thiazolo[3,2-b][1,2,4]triazolyl)-(3,4,5-trimethoxyphenyl)methyl]-4-piperidinecarboxylic acid methyl esterEscherichia coli K-12Potency10.000010
N2-(3-methylphenyl)-6-(4-morpholinyl)-5-nitropyrimidine-2,4-diamineEscherichia coli K-12Potency100.000010
2-[1-[4-(diethylamino)phenyl]-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-N-phenylacetamideEscherichia coli K-12Potency25.118910
N-[4-chloro-3-(trifluoromethyl)phenyl]-2-[4-(2-methoxyphenyl)-1-piperazinyl]acetamideEscherichia coli K-12Potency14.333520
3-methoxy-N-[4-methyl-2-(4-morpholinyl)-6-quinolinyl]benzamideEscherichia coli K-12Potency22.411320
2,6-dichloro-1,7-dimethylpyrazolo[1,2-a]pyrazole-3,5-dioneEscherichia coli K-12Potency2.238710
5-(4-fluorophenyl)-7-(3-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineEscherichia coli K-12Potency39.810710
dm 235Escherichia coli K-12Potency3.162310
2-[4-(9H-fluoren-9-yl)-1-piperazinyl]-N-(4-methoxyphenyl)acetamideEscherichia coli K-12Potency37.008420
1-(5-methyl-2-furanyl)-2-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-1H-[1]benzopyrano[2,3-c]pyrrole-3,9-dioneEscherichia coli K-12Potency5.011910
N-(3-chlorophenyl)-4-fluoro-3-(thiophen-2-ylmethylsulfamoyl)benzamideEscherichia coli K-12Potency2.511910
6-amino-5-cyano-2-[[(3-cyano-6-methyl-7,8-dihydro-5H-1,6-naphthyridin-2-yl)thio]methyl]-4-(4-fluorophenyl)-4H-pyran-3-carboxylic acid methyl esterEscherichia coli K-12Potency79.432810
4-chloro-N-[2-(1H-indol-3-yl)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]benzamideEscherichia coli K-12Potency31.622810
N-(2,5-dimethoxyphenyl)-4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1H-quinazoline-7-carboxamideEscherichia coli K-12Potency89.125110
3-acetamido-N-[(4-ethoxy-3-methoxyphenyl)methyl]-4-[(4-methylphenyl)thio]benzamideEscherichia coli K-12Potency22.387210
3,5-diethyl-2-(2-hydroxyethylamino)-5-methyl-6H-benzo[h]quinazolin-4-oneEscherichia coli K-12Potency25.118910
1-cyclohexyl-3-[(1,2-dimethyl-5-indolyl)methyl]ureaEscherichia coli K-12Potency5.623410
N-(4-methylphenyl)-6-(1-pyrazolyl)-3-pyridinecarboxamideEscherichia coli K-12Potency79.432810
N-(3,4-dimethylphenyl)-2-[[5-[3-(4-methoxyphenyl)propyl]-1,3,4-oxadiazol-2-yl]thio]acetamideEscherichia coli K-12Potency28.183810
[2-(3,4-dimethylphenyl)-4-quinolinyl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency35.481310
1-(3,4-dichlorophenyl)-3-[diethoxyphosphoryl(phenyl)methyl]ureaEscherichia coli K-12Potency5.011910
N-[3-[(2,4-dimethylphenyl)sulfamoyl]-4-methylphenyl]-3-oxo-4H-1,4-benzothiazine-6-carboxamideEscherichia coli K-12Potency3.548110
N-[2-(2,4,6-trinitrophenyl)ethyl]anilineEscherichia coli K-12Potency100.000010
2-[[2-(cyclohexylamino)-2-oxoethyl]thio]benzoic acid [2-(cyclohexylamino)-2-oxoethyl] esterEscherichia coli K-12Potency22.387210
2,4-dichloro-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency56.234110
2-(4-fluorophenyl)-4-quinolinecarboxylic acid [2-oxo-2-(2-oxolanylmethylamino)ethyl] esterEscherichia coli K-12Potency25.118910
N-(6-acetyl-3-cyano-5,7-dihydro-4H-thieno[2,3-c]pyridin-2-yl)-3,4,5-trimethoxybenzamideEscherichia coli K-12Potency8.912510
4-(2,5-dioxo-1-pyrrolidinyl)-N-[2-(4-methoxyphenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]benzamideEscherichia coli K-12Potency35.481310
2-[[2-(2-amino-4-oxo-5-thiazolyl)-1-oxoethyl]amino]-6-tert-butyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterEscherichia coli K-12Potency25.118910
N-(3-methoxyphenyl)-1,3-dioxo-2-(2-oxolanylmethyl)-5-isoindolecarboxamideEscherichia coli K-12Potency25.118910
1-(4-methoxyphenyl)-N-(2-oxolanylmethyl)-4-pyrazolo[3,4-d]pyrimidinamineEscherichia coli K-12Potency0.707910
2-[[5-(4-methylanilino)-1,3,4-thiadiazol-2-yl]thio]-N-[3-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)phenyl]acetamideEscherichia coli K-12Potency1.584910
4-[(7-methyl-2-phenyl-3-imidazo[1,2-a]pyridinyl)methyl]morpholineEscherichia coli K-12Potency6.309610
5-(4-morpholinylsulfonyl)-2-(1-piperidinyl)benzoic acid [2-[[(3-methylbutylamino)-oxomethyl]amino]-2-oxoethyl] esterEscherichia coli K-12Potency15.848910
N-(2-methylphenyl)-1-phenazinecarboxamideEscherichia coli K-12Potency5.011910
2-(N-(2-chloro-1-oxoethyl)-4-fluoroanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideEscherichia coli K-12Potency25.118910
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideEscherichia coli K-12Potency39.810710
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamideEscherichia coli K-12Potency35.481310
(4-methyl-1-piperazinyl)-(2-thieno[3,2-b][1]benzothiolyl)methanoneEscherichia coli K-12Potency22.387210
1-(3-chlorophenyl)-3-[2-(dimethylamino)-2-phenylethyl]thioureaEscherichia coli K-12Potency89.125110
2-furanyl-[4-[(6-hydroxy-2-methyl-5-thiazolo[3,2-b][1,2,4]triazolyl)-thiophen-2-ylmethyl]-1-piperazinyl]methanoneEscherichia coli K-12Potency31.622810
2-[[4-(4-chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]thio]-N-(3-methoxyphenyl)-2-phenylacetamideEscherichia coli K-12Potency22.387210
3-methyl-6-prop-2-enoxy-[1,2,4]triazolo[4,3-b]pyridazineEscherichia coli K-12Potency4.466810
5-methyl-4-(3-phenoxyphenyl)-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-6-carboxylic acid ethyl esterEscherichia coli K-12Potency44.668410
N-(2-bromo-4-nitrophenyl)-2-[(5-propan-2-yl-1H-1,2,4-triazol-3-yl)thio]acetamideEscherichia coli K-12Potency8.912510
N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-4-propan-2-yloxybenzamideEscherichia coli K-12Potency7.079510
2-Chloro-1-[3-(4-methylphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]ethanoneEscherichia coli K-12Potency28.183810
3,4,5-trimethoxy-N-[(8-methyl-2-imidazo[1,2-a]pyridinyl)methyl]benzamideEscherichia coli K-12Potency50.118710
N-(4-ethylphenyl)-2-[[3-[3-(4-methyl-1-piperidinyl)propyl]-4-oxo-2-quinazolinyl]thio]acetamideEscherichia coli K-12Potency39.810710
4-(1,3-dioxo-2-benzo[de]isoquinolinyl)butanoic acid [2-(2-acetylanilino)-2-oxoethyl] esterEscherichia coli K-12Potency2.511910
N-(2-ethoxyphenyl)-2,1,3-benzothiadiazole-4-sulfonamideEscherichia coli K-12Potency28.183810
2,5-dichloro-N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-3-thiophenecarboxamideEscherichia coli K-12Potency39.810710
3,5-dimethyl-4-[(4-methylphenyl)sulfonyl-phenylmethyl]isoxazoleEscherichia coli K-12Potency39.810710
N-(4-methyl-5-oxo-2-[1]benzopyrano[4,3-b]pyridinyl)-2-phenylacetamideEscherichia coli K-12Potency5.660820
N-[3-[2-(4-fluorophenyl)sulfonyl-3-thiophen-2-yl-3,4-dihydropyrazol-5-yl]phenyl]ethanesulfonamideEscherichia coli K-12Potency35.481310
2-[2-(2-chlorophenyl)-1-benzimidazolyl]-N-(2,6-diethylphenyl)acetamideEscherichia coli K-12Potency10.000010
7,13-bis(4-nitrobenzyl)-1,4,10-trioxa-7,13-diazacyclopentadecaneEscherichia coli K-12Potency22.387210
N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]-4-[(2-methyl-1-piperidinyl)sulfonyl]benzamideEscherichia coli K-12Potency0.631010
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-3-methyl-5-oxo-6-thiazolo[3,2-a]pyrimidinecarboxamideEscherichia coli K-12Potency10.000010
6-[[4-(3-methylphenyl)-5-(propan-2-ylthio)-1,2,4-triazol-3-yl]methyl]-1H-pyrimidine-2,4-dioneEscherichia coli K-12Potency6.309610
1-[3-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-4-methoxyphenyl]-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acidEscherichia coli K-12Potency39.810710
N-(7-methyl-2-thiazolo[4,5-g][1,3]benzothiazolyl)propanamideEscherichia coli K-12Potency3.981110
5-oxo-2-pyrrolidinecarboxylic acid [2-[3-(4-methoxyphenyl)-5-(2-naphthalenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] esterEscherichia coli K-12Potency25.118910
1-(4-chlorophenyl)-2-[[3-(3-methylphenyl)-1,2,4-thiadiazol-5-yl]thio]ethanoneEscherichia coli K-12Potency5.011910
3-(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)-N-(3-fluoro-4-methylphenyl)propanamideEscherichia coli K-12Potency5.011910
LSM-33280Escherichia coli K-12Potency0.631010
4-(1-imidazolyl)-3,5-dinitrobenzoic acid methyl esterEscherichia coli K-12Potency100.000010
LSM-31434Escherichia coli K-12Potency0.631010
6-(6-bromo-4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)-N-[2-(4-sulfamoylphenyl)ethyl]hexanamideEscherichia coli K-12Potency44.288720
3-(benzenesulfonyl)-1-cyclopropyl-2-pyrrolo[3,2-b]quinoxalinamineEscherichia coli K-12Potency4.466810
2-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideEscherichia coli K-12Potency19.952610
N-(3-cyano-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl)-2-oxolanecarboxamideEscherichia coli K-12Potency44.668410
2,4-dichloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideEscherichia coli K-12Potency18.860020
2-[[(3,5-dimethylphenyl)-oxomethyl]amino]acetic acid [2-[4-(2-naphthalenylsulfonyl)-1-piperazinyl]-2-oxoethyl] esterEscherichia coli K-12Potency10.157820
2-[8-[(2,6-dimethyl-4-morpholinyl)methyl]-1,3-dimethyl-2,6-dioxo-7-purinyl]acetic acid ethyl esterEscherichia coli K-12Potency5.011910
7,7-dimethyl-1-(4-methylphenyl)-N-[3-(4-morpholinyl)propyl]-2,5-dioxo-6,8-dihydroquinoline-3-carboxamideEscherichia coli K-12Potency14.125410
1-(3-chlorophenyl)-3-pyridin-4-ylureaEscherichia coli K-12Potency1.258910
3-(4-chlorophenyl)-6-(4-methyl-1-piperazinyl)-1H-pyrimidine-2,4-dioneEscherichia coli K-12Potency56.234110
2-[[(3,4-dimethoxyphenyl)-oxomethyl]amino]acetic acid [2-[5-(4-chlorophenyl)-3-(2-furanyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] esterEscherichia coli K-12Potency35.481310
N-(3-acetylphenyl)-2-[[6-chloro-3-(2-hydroxypropyl)-4-methyl-2-oxo-1-benzopyran-7-yl]oxy]acetamideEscherichia coli K-12Potency22.387210
4-[bis(2-methoxyethyl)sulfamoyl]-N-[5-(methoxymethyl)-1,3,4-oxadiazol-2-yl]benzamideEscherichia coli K-12Potency2.818410
2-(2-furanyl)-4-mercapto-3-(4-methylphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileEscherichia coli K-12Potency2.511910
4-dimethoxyphosphoryl-2-(1-naphthalenyl)-N-(phenylmethyl)-5-oxazolamineEscherichia coli K-12Potency31.622810
N,N,4-trimethyl-2-[[(5-methyl-2-furanyl)-oxomethyl]amino]-5-thiazolecarboxamideEscherichia coli K-12Potency0.251210
1-(4-ethylphenyl)-2-methyl-N-(3-pyridinylmethyl)-5-benzimidazolecarboxamideEscherichia coli K-12Potency28.183810
2-methyl-1-phenyl-5-benzimidazolecarboxylic acid [2-(3-methylbutan-2-ylamino)-2-oxoethyl] esterEscherichia coli K-12Potency19.952610
4-methoxy-N-(4-methyl-5-oxo-2-[1]benzopyrano[4,3-b]pyridinyl)benzamideEscherichia coli K-12Potency7.268020
4-(1-azepanylsulfonyl)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-hydroxyphenyl]benzamideEscherichia coli K-12Potency2.511910
4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)benzoic acid [2-(cyclopropylamino)-2-oxoethyl] esterEscherichia coli K-12Potency25.118910
1-[4-(2-fluorophenyl)-1-piperazinyl]-4-(4,4,6-trimethyl-2-sulfanylidene-1,3-diazinan-1-yl)-1-butanoneEscherichia coli K-12Potency89.125110
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterEscherichia coli K-12Potency28.183810
5-(4-nitrophenyl)-3-phenyl-1H-imidazole-2-thioneEscherichia coli K-12Potency8.912510
4-(4-chlorophenyl)-3-[2-(4-methylphenyl)cyclopropyl]-1H-1,2,4-triazole-5-thioneEscherichia coli K-12Potency5.011910
6,7-dimethoxy-N-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxamideEscherichia coli K-12Potency0.316210
[4-[(4-bromo-3,5-dimethyl-1-pyrazolyl)methyl]phenyl]-[5-hydroxy-3-methyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]methanoneEscherichia coli K-12Potency15.848910
N-[(4-ethoxy-3-methoxyphenyl)methyl]-N-methyl-2-(3-pyridinyl)-4-quinazolinamineEscherichia coli K-12Potency25.118910
N-[5-(1-azepanylsulfonyl)-2-chlorophenyl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]acetamideEscherichia coli K-12Potency5.011910
N-[6-amino-2,4-dioxo-1-(phenylmethyl)-5-pyrimidinyl]-N-ethyl-2-[4-[3-(trifluoromethyl)phenyl]-1-piperazinyl]acetamideEscherichia coli K-12Potency7.943310
N-[4-(4-fluorophenyl)-2-thiazolyl]-3-methoxy-4-[2-(4-morpholinyl)-2-oxoethoxy]benzamideEscherichia coli K-12Potency39.810710
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamideEscherichia coli K-12Potency39.810710
N,N-dimethyl-3-[[4-(4-nitrophenyl)-1-piperazinyl]-oxomethyl]-4-(1-pyrrolidinyl)benzenesulfonamideEscherichia coli K-12Potency22.387210
[[2-[(4,5-dimethyl-2-thiazolyl)amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esterEscherichia coli K-12Potency10.000010
4-[[2-(1,10b-dihydropyrazolo[1,5-c]quinazolin-5-ylthio)-1-oxoethyl]amino]benzoic acid butyl esterEscherichia coli K-12Potency15.848910
N-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxolanylmethoxy)benzamideEscherichia coli K-12Potency35.481310
1-[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-[3-(dimethylamino)propyl]thioureaEscherichia coli K-12Potency22.387210
4-[4-(4-acetylphenyl)-1-piperazinyl]-N-[3-(dimethylamino)propyl]-3-nitrobenzenesulfonamideEscherichia coli K-12Potency36.426120
6-methoxy-2-methyl-N-[[3-(trifluoromethyl)phenyl]methyl]-4-quinolinamineEscherichia coli K-12Potency22.387210
LSM-24516Escherichia coli K-12Potency19.952610
LSM-28572Escherichia coli K-12Potency0.891310
N-[5-(4-morpholinylsulfonyl)-2-(1-pyrrolidinyl)phenyl]-2-oxo-1H-quinoline-4-carboxamideEscherichia coli K-12Potency39.810710
N-(6-methoxy-3-pyridinyl)-7-methyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideEscherichia coli K-12Potency44.668410
2-[[2-(4-ethoxy-3-methoxyphenyl)-4-thiazolyl]methylthio]-5-methyl-1,3,4-thiadiazoleEscherichia coli K-12Potency19.952610
6-[5-chloro-3-methyl-1-(4-methylphenyl)-4-pyrazolyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylic acid ethyl esterEscherichia coli K-12Potency14.125410
N-[4-methoxy-3-(4-morpholinylsulfonyl)phenyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideEscherichia coli K-12Potency39.810710
2-(1-adamantyl)-N-[2,5-diethoxy-4-(4-morpholinyl)phenyl]acetamideEscherichia coli K-12Potency21.895920
3'-[2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]spiro[6,7-dihydro-5H-1-benzothiophene-4,5'-imidazolidine]-2',4'-dioneEscherichia coli K-12Potency1.258910
2-methyl-1-cyclopropanecarboxylic acid [5-[2-(3,4-dimethoxyphenyl)-4-quinolinyl]-1,3,4-oxadiazol-2-yl]methyl esterEscherichia coli K-12Potency22.387210
N-(2-methoxy-3-dibenzofuranyl)-3-pyridinecarboxamideEscherichia coli K-12Potency25.118910
4-amino-5-cyano-2-(1-naphthalenylmethylthio)-3-azaspiro[5.5]undeca-2,4-diene-1-carboxamideEscherichia coli K-12Potency39.810710
N-(4,5-dithiophen-2-yl-2-thiazolyl)-2-methyl-1-cyclopropanecarboxamideEscherichia coli K-12Potency4.466810
N-[(1,5-dimethyl-2-pyrrolyl)methyl]-1-(4-methylphenyl)-5-oxo-3-pyrrolidinecarboxamideEscherichia coli K-12Potency28.183810
2-[[4-(3,4-dimethylphenyl)-1-phenyl-2-imidazolyl]thio]-N-(1,1-dioxo-3-thiolanyl)acetamideEscherichia coli K-12Potency25.118910
3-methoxy-N-[2-(4-methoxyphenyl)-2-(1-pyrrolidinyl)ethyl]-2-naphthalenecarboxamideEscherichia coli K-12Potency39.810710
N-(3,4-dimethylphenyl)-2-[[1-(phenylmethyl)-2-imidazolyl]thio]acetamideEscherichia coli K-12Potency12.589310
2-(4-benzoyl-1-piperazinyl)-N-(2-phenylphenyl)propanamideEscherichia coli K-12Potency15.848910
N-[3-(1-imidazolyl)propyl]-2-methyl-3-phenyl-5-propyl-7-pyrazolo[1,5-a]pyrimidinamineEscherichia coli K-12Potency25.118910
5-tert-butyl-3-(4-chlorophenyl)-7-(2-ethyl-1-imidazolyl)pyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency50.118710
8-[[4-[2-furanyl(oxo)methyl]-1-piperazinyl]methyl]-1,3-dimethyl-7-[(2-methylphenyl)methyl]purine-2,6-dioneEscherichia coli K-12Potency15.165220
LSM-31374Escherichia coli K-12Potency7.943310
3-(3,4-dimethoxyphenyl)-2,5-dimethyl-7-[4-(phenylmethyl)-1-piperazinyl]pyrazolo[1,5-a]pyrimidineEscherichia coli K-12Potency24.108220
[5-(4-fluorophenyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[2-(3-pyridinyl)-1-piperidinyl]methanoneEscherichia coli K-12Potency29.881620
6-(4-methoxyphenyl)-8-methyl-4-oxo-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylic acid O7-ethyl ester O2-methyl esterEscherichia coli K-12Potency100.000010
N-(4-ethoxyphenyl)-2-[5-oxo-1-phenyl-3-(2-pyridinylmethyl)-2-sulfanylidene-4-imidazolidinyl]acetamideEscherichia coli K-12Potency17.782810
2-(2-chloro-1-oxoethyl)-3,4-dihydro-1H-isoquinoline-3-carboxylic acid methyl esterEscherichia coli K-12Potency0.316210
3-[(4-methyl-1-piperazinyl)sulfonyl]-N-(4-phenyl-2-thiazolyl)-N-prop-2-enylbenzamideEscherichia coli K-12Potency24.068220
2-[8-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-1,3-dimethyl-2,6-dioxo-7-purinyl]acetic acid methyl esterEscherichia coli K-12Potency15.211320
N2-(2-furanylmethyl)-6-(3-methyl-1-piperidinyl)-5-nitropyrimidine-2,4-diamineEscherichia coli K-12Potency0.177810
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(4-methoxyphenyl)-2-thiophenecarboxamideEscherichia coli K-12Potency0.891310
1-(7-methyloctyl)-3-[4-(4-morpholinylsulfonyl)phenyl]thioureaEscherichia coli K-12Potency3.548110
N-[2-(4-methoxyphenyl)-4-oxo-1,2-dihydroquinazolin-3-yl]carbamic acid ethyl esterEscherichia coli K-12Potency12.589310
N-(1,3-benzodioxol-5-yl)-2-(3-methyl-1-piperidinyl)-2-phenylacetamideEscherichia coli K-12Potency6.309610
4-bromo-N-[(4-ethoxy-2-nitroanilino)-sulfanylidenemethyl]-2-methyl-3-pyrazolecarboxamideEscherichia coli K-12Potency29.903320
3-[4-(dimethylamino)phenyl]-1-[1-(3-methylphenyl)-2,5-dioxo-3-pyrrolidinyl]-1-[(1,3,5-trimethyl-4-pyrazolyl)methyl]thioureaEscherichia coli K-12Potency25.118910
LSM-25964Escherichia coli K-12Potency11.220210
cgp 7930Escherichia coli K-12Potency7.079510
N-[2-chloro-5-[ethyl(phenyl)sulfamoyl]phenyl]-2-[methyl-(1-methyl-4-piperidinyl)amino]acetamideEscherichia coli K-12Potency19.952610
N,N-dimethyl-3-(3-oxo-1,2-benzothiazol-2-yl)benzenesulfonamideEscherichia coli K-12Potency35.481310
1,3-dimethyl-8-(3-methyl-1-piperidinyl)-7-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)thio]ethyl]purine-2,6-dioneEscherichia coli K-12Potency0.631010
5-[2-furanyl-[4-(phenylmethyl)-1-piperidinyl]methyl]-6-thiazolo[3,2-b][1,2,4]triazololEscherichia coli K-12Potency31.622810
1-butyl-3-[[oxo-(5-propan-2-yl-3-thiophenyl)methyl]amino]thioureaEscherichia coli K-12Potency89.125110
1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-3-(4,4,6-trimethyl-2-sulfanylidene-1,3-diazinan-1-yl)-1-propanoneEscherichia coli K-12Potency35.481310
5-[(3,4-dimethoxyphenyl)-[4-(2-hydroxyethyl)-1-piperazinyl]methyl]-2-methyl-6-thiazolo[3,2-b][1,2,4]triazololEscherichia coli K-12Potency0.631010
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamideEscherichia coli K-12Potency0.794310
4-[(4-fluorophenyl)-(6-hydroxy-2-methyl-5-thiazolo[3,2-b][1,2,4]triazolyl)methyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency23.445120
N-methyl-2-[[[4-[methyl(phenyl)sulfamoyl]phenyl]-oxomethyl]amino]-6-propyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamideEscherichia coli K-12Potency14.125410
5-(2,4-dichlorophenyl)-4,6-dioxo-3a,6a-dihydro-2H-pyrrolo[3,4-d]isoxazole-3,3-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency4.466810
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideEscherichia coli K-12Potency44.668410
6-(4-bromo-3,5-dimethyl-1-pyrazolyl)-N-cyclohexyl-1,2,4,5-tetrazin-3-amineEscherichia coli K-12Potency100.000010
2-[(1-methyl-3-indolyl)thio]-1-(4-phenyl-1-piperazinyl)ethanoneEscherichia coli K-12Potency5.011910
5-nitro-6-(3-nitrophenyl)-2-piperidinoneEscherichia coli K-12Potency100.000010
3-(5,7-diphenyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-1-propanolEscherichia coli K-12Potency112.202010
5-[(2,4-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]-4-pyrazolyl]-2-furancarboxamideEscherichia coli K-12Potency19.952610
[5-[(3,5-dimethyl-4-nitro-1-pyrazolyl)methyl]-2-furanyl]-[5-hydroxy-3-methyl-5-(trifluoromethyl)-4H-pyrazol-1-yl]methanoneEscherichia coli K-12Potency0.316210
N-(4-phenoxyphenyl)-2-(1,2,3,4-tetrahydroisoquinolin-1-yl)acetamideEscherichia coli K-12Potency0.199510
6-(4-methoxyphenyl)-N,3-dimethyl-2-imidazo[2,1-b]thiazolecarboxamideEscherichia coli K-12Potency39.810710
4-[5-(3-chlorophenyl)-2-furanyl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acid methyl esterEscherichia coli K-12Potency3.981110
5-nitro-2-[(phenylmethyl)amino]benzoic acid [2-(cyclohexylamino)-2-oxoethyl] esterEscherichia coli K-12Potency35.481310
ncgc00099374Escherichia coli K-12Potency0.707910
5,6-dimethyl-1-octyl-4-benzimidazolamineEscherichia coli K-12Potency40.074820
4-tert-butyl-N-[3-[4-[3-[[(4-tert-butylphenyl)-oxomethyl]amino]propyl]-1-piperazinyl]propyl]benzamideEscherichia coli K-12Potency19.952610
4-[1-[2-(3,4-dimethoxyphenyl)ethyl]-3-(4-methoxyphenoxy)-4-oxo-2-azetidinyl]benzoic acid methyl esterEscherichia coli K-12Potency100.000010
5-benzoyl-6-methyl-4-[4-(4-morpholinyl)phenyl]-3,4-dihydro-1H-pyrimidin-2-oneEscherichia coli K-12Potency56.234110
N-(5,5-dimethyl-7-oxo-4,6-dihydro-1,3-benzothiazol-2-yl)-2-(2,5-dioxo-1-pyrrolidinyl)acetamideEscherichia coli K-12Potency63.095710
2-[[4-amino-5-(3,4-dimethoxyphenyl)-1,2,4-triazol-3-yl]thio]-1-(1H-indol-3-yl)-2-phenylethanoneEscherichia coli K-12Potency25.118910
N-(3-nitrophenyl)-1,3-benzodioxole-5-carboxamideEscherichia coli K-12Potency56.234110
3,3-dimethyl-1,5-dinitro-6-phenoxy-3-azoniabicyclo[3.3.1]non-6-eneEscherichia coli K-12Potency3.548110
calcitriolEscherichia coli K-12Potency19.952610
vitamin k semiquinone radicalEscherichia coli K-12Potency6.309610
apiinEscherichia coli K-12Potency0.501210
vitamin d 2Escherichia coli K-12Potency18.623120
prostaglandin a2Escherichia coli K-12Potency21.154620
gamma-linolenic acidEscherichia coli K-12Potency20.246620
alpha-linolenic acidEscherichia coli K-12Potency22.411320
prostaglandin f1Escherichia coli K-12Potency31.622810
rescinnamineEscherichia coli K-12Potency3.981110
pulmicortEscherichia coli K-12Potency39.810710
timolol maleateEscherichia coli K-12Potency2.818410
brompheniramine maleateEscherichia coli K-12Potency0.354810
chlorpheniramine maleateEscherichia coli K-12Potency5.011910
fucoxanthinEscherichia coli K-12Potency25.118910
kavainEscherichia coli K-12Potency0.354810
amentoflavoneEscherichia coli K-12Potency22.387210
diosminEscherichia coli K-12Potency19.952610
myricetinEscherichia coli K-12Potency44.668410
coumestrolEscherichia coli K-12Potency100.000010
rosmarinic acidEscherichia coli K-12Potency59.621820
cephalomannineEscherichia coli K-12Potency10.000010
ellagic acidEscherichia coli K-12Potency56.234110
n-oleoyldopamineEscherichia coli K-12Potency3.162310
domoic acidEscherichia coli K-12Potency50.118710
4-hydroxyestradiolEscherichia coli K-12Potency39.810710
hydrocortisone valerateEscherichia coli K-12Potency31.622810
prostaglandin f2 methyl esterEscherichia coli K-12Potency17.802020
n-oleoylethanolamineEscherichia coli K-12Potency50.118710
2-bromoergocryptine mesylateEscherichia coli K-12Potency64.091920
cyclosporineEscherichia coli K-12Potency2.818410
perhexiline maleateEscherichia coli K-12Potency39.810710
mepyramine maleateEscherichia coli K-12Potency0.707910
genistinEscherichia coli K-12Potency79.432810
su 9516Escherichia coli K-12Potency39.810710
3-ethyl-2-sulfanylidene-6,7,8,9-tetrahydro-1H-pyrimido[4,5-b]quinolin-4-oneEscherichia coli K-12Potency12.589310
N-(2-methoxyethyl)-2-(5-methyl-4,5,6,7-tetrahydroindazol-2-yl)acetamideEscherichia coli K-12Potency5.011910
N-[3-(3-chlorophenyl)-5-isoxazolyl]-2-(4,5,6,7-tetrahydroindazol-2-yl)acetamideEscherichia coli K-12Potency3.548110
1-[(2-oxo-3,4-dihydro-1H-quinolin-6-yl)sulfonyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-piperidinecarboxamideEscherichia coli K-12Potency89.125110
N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamideEscherichia coli K-12Potency0.631010
N-[3-(2,6-dimethyl-1-piperidinyl)propyl]-1,5-dimethyl-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamideEscherichia coli K-12Potency25.118910
4-[[1-(6-ethoxy-1,3-benzothiazol-2-yl)-3-piperidinyl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency15.065420
N-cycloheptyl-1-hydroxy-3-oxo-2-propyl-1H-isoindole-5-carboxamideEscherichia coli K-12Potency45.268820
1-acetyl-N-[3-(N-ethyl-3-methylanilino)propyl]-2,3-dihydroindole-5-sulfonamideEscherichia coli K-12Potency3.548110
N-cyclohexyl-5-propyl-3-isoxazolecarboxamideEscherichia coli K-12Potency39.810710
4-[[[3-(2-fluorophenyl)-1-methyl-5-thieno[2,3-c]pyrazolyl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency56.234110
4-(3,4-dihydroxyphenyl)-6-[(4-fluoro-3-methylphenyl)sulfonylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid ethyl esterEscherichia coli K-12Potency3.548110
5-[(2-fluorophenyl)methyl]-6,11-dioxo-3-benzo[b][1,4]benzothiazepinecarboxylic acidEscherichia coli K-12Potency4.771820
4-[[[2-(4-methoxyphenyl)-3-oxo-1H-isoindol-4-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency25.118910
2,5-dimethyl-N-(3,4,5-trimethoxyphenyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineEscherichia coli K-12Potency2.818410
N-(3,5-dimethylphenyl)-2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency2.511910
N-[(4-fluorophenyl)methyl]-2-[[4-(4-methoxyphenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency42.239520
3-(4-chlorophenyl)-1-methyl-N-[(5-methyl-2-furanyl)methyl]-5-thieno[2,3-c]pyrazolecarboxamideEscherichia coli K-12Potency2.511910
3-[[2-(2-furanylmethyl)-3-oxo-1H-isoindol-1-yl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency6.055820
N-(2-ethoxyphenyl)-1-(8-quinolinylsulfonyl)-3-piperidinecarboxamideEscherichia coli K-12Potency5.623410
4-[[[1-[[2-(3-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-3-piperidinyl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency3.419520
2-[2-oxo-6-(1-pyrrolidinylsulfonyl)-1,3-benzoxazol-3-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideEscherichia coli K-12Potency6.119420
2-[2-[[[1-(1H-imidazol-5-ylsulfonyl)-3-piperidinyl]-oxomethyl]amino]-4-thiazolyl]acetic acid ethyl esterEscherichia coli K-12Potency0.631010
N-(3-fluoro-4-methylphenyl)-3-methyl-2-oxo-1,3-benzoxazole-6-sulfonamideEscherichia coli K-12Potency8.912510
2-[[5-methyl-2-(3-methylphenyl)-4-oxazolyl]methylsulfinyl]-N-(2-oxolanylmethyl)acetamideEscherichia coli K-12Potency3.162310
[2-(1-piperidinyl)-1,3-benzothiazol-6-yl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency10.000010
3-[[4-[6-(4-morpholinyl)-3-pyridazinyl]-1-piperazinyl]-oxomethyl]-1-benzopyran-2-oneEscherichia coli K-12Potency0.863120
N-(2,5-dimethoxyphenyl)-2-[[5-methyl-2-(2-methylphenyl)-4-oxazolyl]methylsulfonyl]acetamideEscherichia coli K-12Potency5.011910
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-(2-methylpropyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency0.501210
N-[2-(1-pyrrolidinyl)ethyl]-8-quinolinesulfonamideEscherichia coli K-12Potency5.623410
2-[[oxo-(5-propyl-3-isoxazolyl)methyl]amino]benzoic acid methyl esterEscherichia coli K-12Potency10.000010
N-(4-ethylphenyl)-2-(2-furanylmethyl)-1,3-dioxo-5-isoindolecarboxamideEscherichia coli K-12Potency4.466810
N-(2-furanylmethyl)-3-(2,4,8,10-tetramethyl-3-pyrido[2,3]pyrazolo[2,4-a]pyrimidinyl)propanamideEscherichia coli K-12Potency25.118910
2-[[4-(2,3-dimethylphenyl)-1-piperazinyl]-oxomethyl]-1,5-dimethyl-4-pyrrolo[3,2-c]quinolinoneEscherichia coli K-12Potency112.202010
[4-(3-methoxyphenyl)-1-piperazinyl]-[2-(1-piperidinyl)-1,3-benzothiazol-6-yl]methanoneEscherichia coli K-12Potency7.943310
4-[3-(4-fluorophenyl)-2-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency13.557120
1-[[2-(3-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-piperidinecarboxamideEscherichia coli K-12Potency28.183810
N-(5-bromo-2-hydroxyphenyl)-5-propyl-3-isoxazolecarboxamideEscherichia coli K-12Potency4.466810
[5-(2-methoxyphenyl)-3-isoxazolyl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency1.000010
4-[4-[[[1-(2-methylpropyl)-3-pyrrolidinyl]methylamino]-oxomethyl]-3-oxo-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency14.652920
5-chloro-2-methoxy-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-N-propan-2-ylbenzamideEscherichia coli K-12Potency9.245420
N-(2-oxolanylmethyl)-2-[1-oxo-4-(3-pyridinylmethyl)-2-phthalazinyl]acetamideEscherichia coli K-12Potency5.250620
5-[5-(2,3-dihydroindol-1-ylsulfonyl)-2,3-dihydroindol-1-yl]-5-oxopentanoic acidEscherichia coli K-12Potency5.011910
4-[1-[(4-methyl-2-oxo-1-benzopyran-7-yl)amino]-3-oxo-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency15.673020
2-(1,3-benzodioxol-5-ylmethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-3H-isoindol-1-oneEscherichia coli K-12Potency6.581220
N-(4-chlorophenyl)-2-[[4-(4-methoxyphenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency1.000010
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-(3-methoxyphenyl)butanamideEscherichia coli K-12Potency2.511910
4,8-dimethyl-1-(phenylmethyl)-3H-1,5-benzodiazepin-2-oneEscherichia coli K-12Potency8.912510
1-(2-phenylethyl)-4-([1,2,4]triazolo[4,3-a]quinoxalin-4-yl)piperazine-2,6-dioneEscherichia coli K-12Potency3.162310
2-(4,5,6,7-tetrahydroindazol-2-yl)-N-(2,4,6-trimethylphenyl)acetamideEscherichia coli K-12Potency10.000010
1,5-dimethyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-2-pyrrolo[3,2-c]quinolinecarboxamideEscherichia coli K-12Potency28.183810
2-[[2-(3,4-dimethoxyphenyl)-5-methyl-4-oxazolyl]methylsulfinyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideEscherichia coli K-12Potency35.481310
4-(2,4-dimethoxyphenyl)-3-methyl-4,5-dihydro-2H-pyrrolo[3,4-c]pyrazol-6-oneEscherichia coli K-12Potency0.631010
2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]-N-(2-oxolanylmethyl)acetamideEscherichia coli K-12Potency12.875020
3,4-dihydro-1H-isoquinolin-2-yl-[1-(8-quinolinylsulfonyl)-2-pyrrolidinyl]methanoneEscherichia coli K-12Potency10.000010
3-(3,4-dimethoxyphenyl)-5,7-dihydroxy-2-methyl-1-benzopyran-4-oneEscherichia coli K-12Potency5.011910
N-[4-[(4-methyl-1-piperidinyl)methyl]phenyl]-1-[5-(1-pyrrolyl)-1,3,4-thiadiazol-2-yl]-4-piperidinecarboxamideEscherichia coli K-12Potency1.567320
N-[(4-methoxyphenyl)methyl]-4-methyl-1,3-dioxo-1$l^{4},4-benzothiazine-6-carboxamideEscherichia coli K-12Potency16.126920
N-[2-(4-ethyl-1-piperazinyl)-4-methyl-6-quinolinyl]-2-pyrazinecarboxamideEscherichia coli K-12Potency0.562310
N-[2-(4-morpholinyl)ethyl]-4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazine-6-carboxamideEscherichia coli K-12Potency11.509120
N-(6-methyl-1,3-benzothiazol-2-yl)-2-(5,6,7,8-tetrahydro-4H-cyclohepta[c]pyrazol-2-yl)acetamideEscherichia coli K-12Potency51.409220
5-[(4-methoxyphenyl)sulfonylmethyl]-N-(3-methoxypropyl)-2-furancarboxamideEscherichia coli K-12Potency7.943310
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[5-methyl-2-(4-methylphenyl)-4-oxazolyl]methylsulfonyl]ethanoneEscherichia coli K-12Potency20.220820
4-[3-oxo-1-(3,4,5-trimethoxyanilino)-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency20.220820
1-[2-(4-morpholinyl)-2-oxoethyl]-2-pyrido[2,3-b][1,4]thiazinoneEscherichia coli K-12Potency5.623410
3-(4-chlorophenyl)-N-[2-(diethylamino)ethyl]-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideEscherichia coli K-12Potency21.161320
1-(4-tert-butylphenyl)sulfonyl-N-(2-pyridinylmethyl)-2-piperidinecarboxamideEscherichia coli K-12Potency20.220820
(2S)-2-(3-oxo-1H-isoindol-2-yl)-3-phenylpropanoic acidEscherichia coli K-12Potency1.995310
N-[3-[butyl(ethyl)amino]propyl]-1,5-dimethyl-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamideEscherichia coli K-12Potency44.668410
8-(2-chlorophenyl)-3-(4-ethoxyphenyl)-6-oxo-2,4,7,8-tetrahydropyrido[2,1-b][1,3,5]thiadiazine-9-carbonitrileEscherichia coli K-12Potency112.202010
N-(1,3-benzodioxol-5-yl)-2-(5-methyl-2-furanyl)-3-imidazo[1,2-a]pyrazinamineEscherichia coli K-12Potency26.468520
3-(2-ethoxyanilino)-2-(2-furanylmethyl)-3H-isoindol-1-oneEscherichia coli K-12Potency79.432810
N-[3-(4-methyl-1-piperazinyl)propyl]-4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazine-6-carboxamideEscherichia coli K-12Potency25.118910
N-(5-methyl-3-isoxazolyl)-2-[[4-(2-methylphenyl)-5-[(2-oxo-1,3-benzothiazol-3-yl)methyl]-1,2,4-triazol-3-yl]thio]acetamideEscherichia coli K-12Potency0.707910
N-butan-2-yl-3,8-dimethyl-2-oxo-1-oxaspiro[4.5]dec-3-ene-4-carboxamideEscherichia coli K-12Potency5.011910
N-(2-oxolanylmethyl)-2-[7-oxo-3-(phenylmethyl)-6-triazolo[4,5-d]pyrimidinyl]acetamideEscherichia coli K-12Potency3.162310
6-[2-oxo-2-(4-phenyl-1-piperazinyl)ethyl]-3-(phenylmethyl)-7-triazolo[4,5-d]pyrimidinoneEscherichia coli K-12Potency3.162310
1-(4-morpholinyl)-2-[[3-(2-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]ethanoneEscherichia coli K-12Potency112.202010
2-[[cyclohexyl(oxo)methyl]amino]-3-thiophenecarboxamideEscherichia coli K-12Potency1.000010
N-(2-oxolanylmethyl)-2-(7-oxo-3-phenyl-6-triazolo[4,5-d]pyrimidinyl)acetamideEscherichia coli K-12Potency19.952610
5-ethyl-N-[[2-(3-pyridinyl)-4-thiazolyl]methyl]-2-thiophenesulfonamideEscherichia coli K-12Potency3.981110
1,3-dimethyl-2,4-dioxo-N-(4-propan-2-ylphenyl)-5-pyrimidinesulfonamideEscherichia coli K-12Potency7.079510
N-[(3-methyl-6-imidazo[2,1-b]thiazolyl)methyl]-1-propanesulfonamideEscherichia coli K-12Potency44.668410
N-[1-[4-(2-methoxyphenyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]benzenesulfonamideEscherichia coli K-12Potency2.168020
N-[2-(2-imidazo[1,2-a]pyridinyl)ethyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideEscherichia coli K-12Potency0.707910
3-(prop-2-enylthio)-[1,2,4]triazino[5,6-d][3,1]benzoxazepineEscherichia coli K-12Potency0.631010
8-(diethylaminomethyl)-7-hydroxy-4-phenyl-1-benzopyran-2-oneEscherichia coli K-12Potency50.118710
4-amino-5-chloro-N-[(3R,4S)-1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamideEscherichia coli K-12Potency20.552320
latanoprostEscherichia coli K-12Potency11.220210
rimexoloneEscherichia coli K-12Potency2.818410
kn 62Escherichia coli K-12Potency3.518020
su 6656Escherichia coli K-12Potency10.000010
rosmarinic acidEscherichia coli K-12Potency100.000010
syringinEscherichia coli K-12Potency89.125110
kaempferol-3-o-rutinosideEscherichia coli K-12Potency0.562310
icariinEscherichia coli K-12Potency12.589310
salazinic acidEscherichia coli K-12Potency50.118710
4-[(3aR,4S,9bS)-8-[(4-methoxyphenyl)sulfamoyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-4-yl]benzoic acidEscherichia coli K-12Potency0.316210
3,5-dimethoxycinnamic acidEscherichia coli K-12Potency0.281810
ag 538Escherichia coli K-12Potency7.943310
tyrphostin b44Escherichia coli K-12Potency8.912510
nifuroxazideEscherichia coli K-12Potency39.810710
platyphyllineEscherichia coli K-12Potency25.118910
molsidomineEscherichia coli K-12Potency28.599120
rg 13022Escherichia coli K-12Potency22.387210
nalbuphine hydrochlorideEscherichia coli K-12Potency56.234110
cefiximeEscherichia coli K-12Potency1.995310
7-hydroxy-4-methyl-1H-quinolin-2-oneEscherichia coli K-12Potency11.220210
7-hydroxyisoflavoneEscherichia coli K-12Potency39.810710
urolithin bEscherichia coli K-12Potency17.782810
7-Hydroxy-2-methylisoflavoneEscherichia coli K-12Potency3.981110
trimebutine maleate saltEscherichia coli K-12Potency39.810710
vinblastine sulfateEscherichia coli K-12Potency8.912510
vincristine sulfateEscherichia coli K-12Potency10.000010
7-hydroxy-6-(4-morpholinylmethyl)-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-4-oneEscherichia coli K-12Potency22.387210
(3S,3'aR,8'aS,8'bS)-5-ethyl-2'-(phenylmethyl)spiro[1H-indole-3,4'-3a,6,7,8,8a,8b-hexahydropyrrolo[3,4-a]pyrrolizine]-1',2,3'-trioneEscherichia coli K-12Potency22.387210
calycanthineEscherichia coli K-12Potency5.623410
3-bromo-7-hydroxy-4,8-dimethyl-1-benzopyran-2-oneEscherichia coli K-12Potency50.118710
trientine hydrochlorideEscherichia coli K-12Potency0.501210
6-[4-methyl-6-(4-nitrophenyl)-2-oxo-5-phenylmethoxycarbonyl-1,6-dihydropyrimidin-3-yl]hexanoic acidEscherichia coli K-12Potency28.183810
2-(1H-1,2,3-Benzotriazol-1-yl)-N'-(3,4,5-trimethoxybenzylidene)acetohydrazideEscherichia coli K-12Potency2.818410
3-(dimethylamino)benzoic acid (7-hydroxy-2-oxo-1-benzopyran-4-yl)methyl esterEscherichia coli K-12Potency17.782810
nylidrin hydrochlorideEscherichia coli K-12Potency89.125110
phentolamineEscherichia coli K-12Potency17.782810
fendiline hydrochlorideEscherichia coli K-12Potency44.668410
methylbenzethonium chlorideEscherichia coli K-12Potency15.714220
dithiazanine iodideEscherichia coli K-12Potency61.193620
quinaldine redEscherichia coli K-12Potency1.412510
5-(4-methyl-1-naphthalenyl)-N-phenyl-2-furancarboxamideEscherichia coli K-12Potency25.118910
3,3'-diethylthiacarbocyanine iodideEscherichia coli K-12Potency20.811420
5233705 compoundEscherichia coli K-12Potency25.118910
7-fluoro-2-phenyl-4-quinoloneEscherichia coli K-12Potency0.631010
N-(1,3-benzodioxol-5-yl)-2-[(8-methoxy-5H-[1,2,4]triazino[5,6-b]indol-3-yl)thio]acetamideEscherichia coli K-12Potency39.810710
tg4-155Escherichia coli K-12Potency35.481310
DPI2Escherichia coli K-12Potency15.848910
6-chloro-4-[[(2-fluorophenyl)methyl-methylamino]methyl]-7-hydroxy-1-benzopyran-2-oneEscherichia coli K-12Potency12.589310
6-[(4-fluorophenyl)methyl]-5,7-dimethyl-2H-pyrrolo[3,4-d]pyridazin-1-oneEscherichia coli K-12Potency0.316210
3-[(1S)-1-phenylethyl]-4-imidazolecarboxylic acid ethyl esterEscherichia coli K-12Potency10.000010
LSM-1411Escherichia coli K-12Potency5.623410
N-(3,4-dichlorophenyl)-6-(1-imidazolyl)-3-pyridazinamineEscherichia coli K-12Potency89.125110
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-N-(3-methylphenyl)acetamideEscherichia coli K-12Potency15.848910
3-amino-5-(4-bromophenyl)-4-pyridazinecarbonitrileEscherichia coli K-12Potency12.589310
[2-methoxy-5-[[4-(4-methylphenyl)-1-phthalazinyl]amino]phenyl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency20.611620
N'1-(6-methylpyridazin-3-yl)-4-chlorobenzene-1-carbohydrazideEscherichia coli K-12Potency0.631010
hydrocotarnine hydrobromideEscherichia coli K-12Potency70.794610
dihydroergotoxineEscherichia coli K-12Potency12.589310
enclomiphene citrateEscherichia coli K-12Potency35.481310
benoxinate hydrochlorideEscherichia coli K-12Potency1.412510
mg 624Escherichia coli K-12Potency15.848910
o-geranylsinapyl alcoholEscherichia coli K-12Potency39.810710
N-[2-(4-acetyl-1-piperazinyl)phenyl]-2-(2-methylphenoxy)acetamideEscherichia coli K-12Potency25.118910
(4-chloro-2-methyl-3-pyrazolyl)-[4-(2-ethoxyphenyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency35.481310
dirithromycinEscherichia coli K-12Potency35.481310
N-(3,4-dichlorophenyl)-2-[4-(1-piperidinylsulfonyl)-1-piperazinyl]acetamideEscherichia coli K-12Potency17.782810
1-[2-furanyl(oxo)methyl]-N-[4-[(3-methyl-1-piperidinyl)sulfonyl]phenyl]-4-piperidinecarboxamideEscherichia coli K-12Potency6.309610
fluphenazineEscherichia coli K-12Potency3.981110
homochlorocyclizine monohydrochlorideEscherichia coli K-12Potency14.125410
azacaineEscherichia coli K-12Potency100.000010
n-(3-(cyclohexylidene-(1h-imidazol-4-ylmethyl))phenyl)ethanesulfonamideEscherichia coli K-12Potency56.234110
n-(4-amino-2-chlorophenyl)phthalimideEscherichia coli K-12Potency24.905420
2-(3,3-diphenylpropylamino)acetamideEscherichia coli K-12Potency100.000010
l 162313Escherichia coli K-12Potency14.407420
l-165041Escherichia coli K-12Potency44.668410
mrs 1754Escherichia coli K-12Potency8.912510
dibenzheptropine citrateEscherichia coli K-12Potency22.387210
2-(1,3-benzothiazol-2-yl)-4-chloro-5-(3-chloroanilino)-3-pyridazinoneEscherichia coli K-12Potency7.943310
4-[(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)methyl]-N-(3-ethylphenyl)benzamideEscherichia coli K-12Potency0.707910
4-methyl-N-[(4-methylphenyl)methyl]-2-furo[3,2-c]quinolinecarboxamideEscherichia coli K-12Potency2.990420
[4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazin-6-yl]-(1-piperidinyl)methanoneEscherichia coli K-12Potency50.118710
6-ethyl-8-methyl-N-(3-pyridinylmethyl)-3-benzo[b][1,4]benzothiazepinecarboxamideEscherichia coli K-12Potency39.810710
8-bromo-6-ethyl-N-(2-oxolanylmethyl)-3-benzo[b][1,4]benzothiazepinecarboxamideEscherichia coli K-12Potency28.183810
N-cyclopropyl-2-[[2-(4-ethylphenyl)-5-methyl-4-oxazolyl]methylthio]acetamideEscherichia coli K-12Potency44.668410
6-bromo-2-(1-pyrrolidinyl)-1,3-benzothiazoleEscherichia coli K-12Potency39.810710
(9-chloro-5,6,7,8-tetrahydroacridin-3-yl)-(4-methyl-1-piperidinyl)methanoneEscherichia coli K-12Potency31.622810
2-(4-methoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acid ethyl esterEscherichia coli K-12Potency39.810710
(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-(4-oxo-1-benzopyran-3-yl)-3,4-dihydro-2H-pyran-6-carboxylic acid prop-2-enyl esterEscherichia coli K-12Potency11.220210
1-[(4S,5R)-4-hydroxy-5-(hydroxymethyl)-2-oxolanyl]-5-(trifluoromethyl)pyrimidine-2,4-dioneEscherichia coli K-12Potency5.623410
hoe 777Escherichia coli K-12Potency49.692720
butylscopolammonium bromideEscherichia coli K-12Potency6.309610
androst-16-en-3-oneEscherichia coli K-12Potency22.387210
LSM-6455Escherichia coli K-12Potency76.006420
8-(n,n-diethylamino)octyl-3,4,5-trimethoxybenzoate hydrochlorideEscherichia coli K-12Potency31.622810
l 671152Escherichia coli K-12Potency5.623410
13-epi-sclareolEscherichia coli K-12Potency11.220210
N'-(4,6-difluoro-1,3-benzothiazol-2-yl)propanehydrazideEscherichia coli K-12Potency100.000010
6-bromo-N-(2-methylphenyl)-2-pyridin-4-yl-3-imidazo[1,2-a]pyridinamineEscherichia coli K-12Potency69.905420
6-(3-bromophenyl)-2-methyl-3-pyridinecarboxylic acidEscherichia coli K-12Potency31.622810
N-(1,3-dioxo-5-isoindolyl)butanamideEscherichia coli K-12Potency44.668410
N-(4,7-dimethyl-1,3-benzothiazol-2-yl)-4-(2,5-dioxo-1-pyrrolidinyl)benzamideEscherichia coli K-12Potency0.562310
1,3-dimethyl-2,4-dioxo-5-pyrimidinesulfonic acid phenyl esterEscherichia coli K-12Potency3.981110
N'-(1-methyl-4-pyrazolo[3,4-d]pyrimidinyl)-2-(1-naphthalenyl)acetohydrazideEscherichia coli K-12Potency7.079510
2-[[6-(2-furanyl)-3-pyridazinyl]thio]-N-(3-methylphenyl)acetamideEscherichia coli K-12Potency3.981110
N-[3-(dimethylamino)propyl]-N-(6-methyl-1,3-benzothiazol-2-yl)-1,3-benzothiazole-6-carboxamideEscherichia coli K-12Potency28.183810
6-(4-bromophenyl)-2-methyl-3-pyridinecarboxylic acidEscherichia coli K-12Potency0.562310
5-(1-phenyl-5-tetrazolyl)-2-pyridin-4-yl-4-thiophen-2-ylpyrimidineEscherichia coli K-12Potency100.000010
4-[3-(3-methylanilino)-2-imidazo[1,2-a]pyrimidinyl]phenolEscherichia coli K-12Potency0.631010
6-(4-ethylphenyl)-3-(methylthio)-[1,2,4]triazolo[4,3-b]pyridazineEscherichia coli K-12Potency39.810710
3-butyl-10-phenylpyrimido[4,5-b]quinoline-2,4-dioneEscherichia coli K-12Potency15.848910
LSM-2818Escherichia coli K-12Potency18.094620
N-[3-[(1,3-dimethyl-2,6-dioxo-4-pyrimidinyl)methylamino]-3-oxopropyl]-3-methoxybenzamideEscherichia coli K-12Potency0.562310
3-(diphenylmethylene)-1-[4-(4-phenyl-1-piperazinyl)butyl]pyrrolidine-2,5-dioneEscherichia coli K-12Potency15.848910
N-[2-(3-methoxyphenyl)-4-[(4-methoxyphenyl)methoxy]-6-quinolinyl]-3-pyridinecarboxamideEscherichia coli K-12Potency39.810710
alpha-solanineEscherichia coli K-12Potency28.183810
3-hydroxy-2-methyl-1-(phenylmethyl)-4-pyridinoneEscherichia coli K-12Potency0.631010
N-ethyl-8-methyl-4-oxo-N-(phenylmethyl)-2-thieno[3,2-c][1]benzopyrancarboxamideEscherichia coli K-12Potency9.333610
3-(1H-benzimidazol-2-yl)-1-[4-(2,4-dimethylphenyl)-1-piperazinyl]-1-propanoneEscherichia coli K-12Potency5.011910
4-[[[4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazin-6-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency0.354810
N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideEscherichia coli K-12Potency31.622810
1-(3,5-dimethylphenyl)-3-(4-methyl-3-oxo-1,4-benzothiazin-6-yl)ureaEscherichia coli K-12Potency8.912510
3-(4-ethoxyphenyl)-1-[3-(4-morpholinyl)propyl]-1-[(1-propyl-3,4-dihydro-2H-quinolin-6-yl)methyl]ureaEscherichia coli K-12Potency6.610220
1-[(2-chlorophenyl)methyl]-N-[3-(N-ethyl-3-methylanilino)propyl]-5-oxo-2-pyrrolidinecarboxamideEscherichia coli K-12Potency17.782810
N-(1,3-benzodioxol-5-yl)-2-(4-methylphenyl)-3-imidazo[1,2-a]pyrazinamineEscherichia coli K-12Potency0.631010
1-(3,4-dimethylphenyl)-2,5-dioxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarbonitrileEscherichia coli K-12Potency0.631010
1-cyclohexyl-3-[1-[4-(phenylmethyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]ureaEscherichia coli K-12Potency2.818410
4-[[oxo-[4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazin-6-yl]methyl]amino]-1-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency14.125410
4-chloro-N-(4-ethylphenyl)-3-methyl-5-isoxazolecarboxamideEscherichia coli K-12Potency5.011910
4-methyl-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideEscherichia coli K-12Potency13.265720
2-[3-[(2-chloro-4-fluorophenyl)methyl]-2-oxo-1,3-diazinan-1-yl]-N-cyclooctylacetamideEscherichia coli K-12Potency25.118910
3-(2-methoxyethyl)-2,4-dioxo-N-pentyl-1H-quinazoline-7-carboxamideEscherichia coli K-12Potency0.794310
2-(2,1,3-benzothiadiazol-4-ylsulfonyl)-5-(4-chlorophenyl)-3-pyrazolamineEscherichia coli K-12Potency22.387210
cetirizine dihydrochlorideEscherichia coli K-12Potency39.810710
2-methyl-6-(phenylethynyl)pyridine hydrochlorideEscherichia coli K-12Potency7.079510
amipriloseEscherichia coli K-12Potency12.589310
(R)-fluoxetine hydrochlorideEscherichia coli K-12Potency1.412510
dimethisoquin hydrochlorideEscherichia coli K-12Potency64.467920
(S)-fluoxetine hydrochlorideEscherichia coli K-12Potency7.943310
trimetazidine dihydrochlorideEscherichia coli K-12Potency8.912510
tiamulin fumarate (1:1), (3as-(3aalpha,4beta,5alpha,6alpha,8beta,9alpha,9abeta,10s*))-isomerEscherichia coli K-12Potency28.183810
emergilEscherichia coli K-12Potency31.622810
benalfocin hydrochlorideEscherichia coli K-12Potency28.183810
anomalinEscherichia coli K-12Potency39.810710
garcinone eEscherichia coli K-12Potency14.125410
biapigeninEscherichia coli K-12Potency19.952610
dihydroxanthohumolEscherichia coli K-12Potency44.668410
(+)-lyoniresinol-3-alpha-O-beta-D-glucopyranosideEscherichia coli K-12Potency2.818410
cefotaxime sodiumEscherichia coli K-12Potency14.125410
5-methoxy-8,8-dimethyl-2-phenyl-4H,8H-pyrano[2,3-h]chromen-4-oneEscherichia coli K-12Potency31.622810
calpain inhibitor iiiEscherichia coli K-12Potency6.309610
ditryptophenalineEscherichia coli K-12Potency19.702020
losartan potassiumEscherichia coli K-12Potency14.125410
GR 127935 hydrochlorideEscherichia coli K-12Potency19.952610
mrs 1845Escherichia coli K-12Potency12.589310
vu 1545Escherichia coli K-12Potency1.778310
protoapigenoneEscherichia coli K-12Potency0.223910
2-(4-butan-2-ylanilino)-3-pyridinecarbonitrileEscherichia coli K-12Potency35.481310
N-[(1,3-dioxo-2-phenyl-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl)methyl]-4-methylbenzenesulfonamideEscherichia coli K-12Potency44.668410
N-(2-methoxyethyl)-2-[[3-[(4-methoxyphenyl)methyl]-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideEscherichia coli K-12Potency31.622810
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-[(4-methylphenyl)methyl]butanamideEscherichia coli K-12Potency35.481310
4-[[[2-(cyclohexylamino)-3,4-dioxo-1-cyclobutenyl]amino]methyl]-N-(4-ethoxyphenyl)benzamideEscherichia coli K-12Potency63.095710
2-(2,1,3-benzothiadiazol-4-ylsulfonyl)-5-(4-bromophenyl)-3-pyrazolamineEscherichia coli K-12Potency100.000010
R-(-)-actinodaphnineEscherichia coli K-12Potency0.631010
6-fluoronorepinephrine monohydrochloride, (+-)-isomerEscherichia coli K-12Potency2.818410
cirazoline monohydrochlorideEscherichia coli K-12Potency79.432810
adtnEscherichia coli K-12Potency0.631010
Dihydro-beta-erythroidine hydrobromideEscherichia coli K-12Potency5.011910
efaroxan hydrochlorideEscherichia coli K-12Potency6.309610
7-hydroxy-2-n,n-dipropylaminotetralin hydrobromideEscherichia coli K-12Potency5.011910
1-(2-(4-(4-fluoro-benzoyl)-piperidin-1-yl)-ethyl)-3,3-dimethyl-1,2-dihydro-indol-2-oneEscherichia coli K-12Potency2.818410
alpha-methyltyrosine methyl ester, monohydrochlorideEscherichia coli K-12Potency6.309610
N-methyl-6-chloro-1-(3-methylphenyl)-2,3,4,5-tetrahydro-3-benzazepine-7,8-diol hydrobromideEscherichia coli K-12Potency8.912510
sk&f 77434Escherichia coli K-12Potency1.122010
3-ethoxy-N-[(4-methoxyphenyl)methyl]-2-propyl-6-indazolecarboxamideEscherichia coli K-12Potency28.183810
N-[(2-methoxyphenyl)methyl]-2-methyl-3-prop-2-enoxy-6-indazolecarboxamideEscherichia coli K-12Potency44.668410
geduninEscherichia coli K-12Potency25.118910
[4-(2-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(phenylmethyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency31.622810
N-[4-(diethylamino)-2-methylphenyl]-2-[(2-nitro-3-thiophenyl)thio]acetamideEscherichia coli K-12Potency5.011910
2-[2-fluoro-5-(4-methyl-1-piperazinyl)-4-nitrophenyl]-3,4-dihydro-1H-isoquinolineEscherichia coli K-12Potency37.646020
4-[(2-heptan-3-yl-1,3-dioxolan-4-yl)methyl]-4-methylmorpholin-4-iumEscherichia coli K-12Potency50.118710
4-methyl-N-[[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]-sulfanylidenemethyl]benzamideEscherichia coli K-12Potency7.943310
1-(3-chlorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thioureaEscherichia coli K-12Potency19.952610
1-[4-[3-methyl-4-(3-methylphenyl)-1-piperazinyl]-3-nitrophenyl]piperidine-2,6-dioneEscherichia coli K-12Potency39.810710
4-[3-(3-fluorophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamideEscherichia coli K-12Potency1.584910
4-(4-chlorophenyl)sulfonyl-5-(3,4-dihydro-1H-isoquinolin-2-yl)-2-ethylsulfonylthiazoleEscherichia coli K-12Potency11.220210
chlorhexidine hydrochlorideEscherichia coli K-12Potency3.548110
ophiocarpineEscherichia coli K-12Potency100.000010
[5-Chloranyl-3-[(1E,3E)-3,5-dimethylhepta-1,3-dienyl]-7-methyl-6,8-bis(oxidanylidene)isochromen-7-yl] ethanoateEscherichia coli K-12Potency39.810710
majeptilEscherichia coli K-12Potency16.903620
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneEscherichia coli K-12Potency25.118910
4-methoxybenzoic acid 2-(4-hydroxyphenyl)ethyl esterEscherichia coli K-12Potency0.794310
rabeprazole sodiumEscherichia coli K-12Potency22.387210
microcolin aEscherichia coli K-12Potency7.943310
18-Deoxy-portulideEscherichia coli K-12Potency25.118910
N-(3,5-dichlorophenyl)-4-[(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)methyl]benzamideEscherichia coli K-12Potency100.000010
foetidinEscherichia coli K-12Potency35.716820
4-chloro-N-[1-[[5-(ethylthio)-1,3,4-thiadiazol-2-yl]amino]-3-methyl-1-oxobutan-2-yl]benzamideEscherichia coli K-12Potency0.631010
1-[(4-methylphenyl)methyl]-2,4-dioxo-N-(phenylmethyl)-3-prop-2-enyl-7-quinazolinecarboxamideEscherichia coli K-12Potency112.202010
[4-(diphenylmethyl)-1-piperazinyl]-(5-methyl-4-nitro-3-isoxazolyl)methanoneEscherichia coli K-12Potency0.707910
3-[2-(4-chlorophenyl)-5,7-dimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]propanamideEscherichia coli K-12Potency31.622810
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(4-morpholinyl)phenyl]-3-imidazo[1,2-a]pyrazinamineEscherichia coli K-12Potency19.952610
N-Cyclohexyl-5-(2-thienyl)-1,2-oxazole-3-carboxamideEscherichia coli K-12Potency5.011910
3-[2-(3,5-dimethoxyphenyl)-5,7-dimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-(phenylmethyl)propanamideEscherichia coli K-12Potency28.183810
4-chloro-N-[3-(3-methyl-1-piperidinyl)propyl]-2-thieno[3,2-c]quinolinecarboxamideEscherichia coli K-12Potency18.446920
N-(4-ethyl-1,2,5-oxadiazol-3-yl)-3,5,6-trimethyl-2-benzofurancarboxamideEscherichia coli K-12Potency5.623410
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideEscherichia coli K-12Potency50.118710
4-(6-chloro-2-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)-4-oxo-N-(phenylmethyl)butanamideEscherichia coli K-12Potency15.848910
N-(2-ethyl-6-methylphenyl)-2-(4-methyl-1-oxo-2-pyrrolo[1,2-d][1,2,4]triazinyl)acetamideEscherichia coli K-12Potency1.000010
3-bromo-N-[5-(4-morpholinylsulfonyl)-1,3,4-thiadiazol-2-yl]benzamideEscherichia coli K-12Potency106.101010
[3-(4-bromophenyl)-1H-pyrazol-5-yl]-[4-(3,4-dimethoxyphenyl)sulfonyl-1-piperazinyl]methanoneEscherichia coli K-12Potency22.387210
[3-methyl-4-(3-methylphenyl)-1-piperazinyl]-[1-(7,8,9,10-tetrahydro-6H-purino[9,8-a]azepin-4-yl)-4-piperidinyl]methanoneEscherichia coli K-12Potency5.313820
3-[3,5-dimethyl-1-[6-(1-piperidinyl)-3-pyridazinyl]-4-pyrazolyl]-N-(3-fluoro-4-methylphenyl)propanamideEscherichia coli K-12Potency19.952610
2-[[1,3-dimethyl-7-(4-methylphenyl)-2,4-dioxo-5-pyrimido[4,5-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideEscherichia coli K-12Potency63.095710
tanninsEscherichia coli K-12Potency0.707920
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2S,3S,4R)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneEscherichia coli K-12Potency19.952610
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-2-(4-hydroxybutoxy)-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-2H-pyran-6-yl]methanoneEscherichia coli K-12Potency15.848910
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-4-(4-bromophenyl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-yl]methanoneEscherichia coli K-12Potency14.125410
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneEscherichia coli K-12Potency15.848910
2-(2,5-difluorophenyl)-5-methyl-4-[[4-(2-pyrazinyl)-1-piperazinyl]methyl]oxazoleEscherichia coli K-12Potency28.183810
1-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-3-(3-methylphenyl)-1-[2-(4-morpholinyl)ethyl]thioureaEscherichia coli K-12Potency31.622810
2-[(1-ethyl-3-methyl-4-pyrazolyl)methyl]-1-(4-fluoro-3-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indoleEscherichia coli K-12Potency28.183810
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[3-(4-fluorophenyl)-2,4-dioxo-1-thieno[3,2-d]pyrimidinyl]acetamideEscherichia coli K-12Potency70.794610
8-methyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-5H-thieno[3,2-c]quinoline-2-carboxamideEscherichia coli K-12Potency25.118910
3-[3-(4-fluorophenyl)-2,5,7-trimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-(2-methoxyphenyl)propanamideEscherichia coli K-12Potency39.810710
N-[[3-(2-chlorophenyl)-1-(4-fluorophenyl)-4-pyrazolyl]methyl]-2-(2-pyridinyl)ethanamineEscherichia coli K-12Potency39.810710
N-(4-acetylphenyl)-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamideEscherichia coli K-12Potency65.811420
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-phenylethyl)-4-piperidinyl]methanolEscherichia coli K-12Potency39.810710
dafadine CEscherichia coli K-12Potency39.810710
1-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-3-(4-methylphenyl)-1-[2-(4-morpholinyl)ethyl]thioureaEscherichia coli K-12Potency25.118910
1-[(1-ethyl-3,4-dihydro-2H-quinolin-6-yl)methyl]-3-(3-methoxyphenyl)-1-[2-(4-morpholinyl)ethyl]thioureaEscherichia coli K-12Potency39.810710
N-[2-(3,4-dimethoxyphenyl)ethyl]-N'-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)oxamideEscherichia coli K-12Potency22.387210
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-[(4-phenyl-1-piperidinyl)methyl]oxazoleEscherichia coli K-12Potency39.810710
dafadine BEscherichia coli K-12Potency19.952610
(6-methoxy-2-naphthalenyl)-[1-[(2-methyl-5-thiazolyl)methyl]-3-piperidinyl]methanoneEscherichia coli K-12Potency0.354810
1,2-dihydroacenaphthylen-5-yl-[1-[(6-methyl-2-pyridinyl)methyl]-3-piperidinyl]methanoneEscherichia coli K-12Potency39.810710
N-methyl-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-N-(3-thiophenylmethyl)propanamideEscherichia coli K-12Potency28.183810
1-[[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-4-pyrazolyl]methyl]-4-methoxypiperidineEscherichia coli K-12Potency39.810710
2-[4-[(6-ethoxy-2-quinolinyl)methyl]-1-(3-thiophenylmethyl)-2-piperazinyl]ethanolEscherichia coli K-12Potency28.183810
1,2-dihydroacenaphthylen-5-yl-[1-(2-pyridinylmethyl)-3-piperidinyl]methanoneEscherichia coli K-12Potency35.481310
N-[[3-(3-methylphenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]-3-(1-pyrazolyl)-1-propanamineEscherichia coli K-12Potency39.810710
1-[3-[(6-methoxy-2-naphthalenyl)-oxomethyl]-1-piperidinyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)thio]ethanoneEscherichia coli K-12Potency35.481310
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolEscherichia coli K-12Potency35.481310
[1-[(5-methyl-1-propyl-4-pyrazolyl)methyl]-3-piperidinyl]-(3-propan-2-yloxyphenyl)methanoneEscherichia coli K-12Potency25.118910
5-[(3-phenylmethoxy-1-piperidinyl)methyl]-3-(phenylmethyl)-1,2,4-oxadiazoleEscherichia coli K-12Potency31.622810
[1-[(6-chloro-2H-1-benzopyran-3-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolEscherichia coli K-12Potency28.183810
2-[4-[1-(2-fluorophenyl)-4-piperidinyl]-1-[(3-methoxyphenyl)methyl]-2-piperazinyl]ethanolEscherichia coli K-12Potency31.622810
[1-[(1,2-dimethyl-3-indolyl)methyl]-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolEscherichia coli K-12Potency39.810710
2-(2,4-dimethoxyphenyl)-5-methyl-4-[[4-(4-quinazolinyl)-1-piperazinyl]methyl]oxazoleEscherichia coli K-12Potency22.387210
[1-(2-benzofuranylmethyl)-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolEscherichia coli K-12Potency39.810710
1-(5-isoquinolinylmethyl)-4-[(3-methoxyphenyl)methyl]-4-piperidinecarboxylic acid ethyl esterEscherichia coli K-12Potency0.794310
1-[[3-(4-fluorophenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]-4-[(1-methyl-2-imidazolyl)methyl]piperazineEscherichia coli K-12Potency25.118910
(3aS,5S,9aS)-2-[(2-methylphenyl)methyl]-5-(1-methyl-3-phenyl-4-pyrazolyl)-3a,4,5,7,8,9-hexahydro-3H-pyrrolo[3,4-h]pyrrolizin-1-oneEscherichia coli K-12Potency31.622810
1-ethyl-4-[[methyl-[[3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]amino]methyl]-2-pyrrolidinoneEscherichia coli K-12Potency22.387210
2-(3,5-dimethyl-1-pyrazolyl)-N-[[3-(4-fluorophenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]ethanamineEscherichia coli K-12Potency17.782810
[1-[[1-(5-chloro-2-pyridinyl)-2-pyrrolyl]methyl]-3-piperidinyl]-(2,4-dimethoxyphenyl)methanoneEscherichia coli K-12Potency22.387210
1-(12-oxo-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)-3-[3-[4-(phenylmethyl)-1-piperidinyl]propyl]thioureaEscherichia coli K-12Potency39.810710
1-butyl-3-[2-(4-ethyl-1-piperazinyl)-4-methyl-6-quinolinyl]-1-methylthioureaEscherichia coli K-12Potency28.183810
N-[3-(1-azepanyl)propyl]-3-[(4-methoxyphenyl)methyl]-2,4-dioxo-1H-quinazoline-7-carboxamideEscherichia coli K-12Potency4.466810
N-[3-[butyl(ethyl)amino]propyl]-1-(9-fluoro-[1]benzothiolo[3,2-d]pyrimidin-4-yl)-4-piperidinecarboxamideEscherichia coli K-12Potency39.810710
2-[3-[[2-oxo-2-(1-pyrrolidinyl)ethyl]thio]-1-indolyl]-N,N-di(propan-2-yl)acetamideEscherichia coli K-12Potency39.810710
6-(2-furanyl)-3-(2-pyridinylmethylthio)-[1,2,4]triazolo[4,3-b]pyridazineEscherichia coli K-12Potency2.818410
4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidineEscherichia coli K-12Potency19.731220
[(2S,4S)-4-(4-bromophenyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency25.118910
[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency14.125410
(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxylic acid prop-2-enyl esterEscherichia coli K-12Potency7.943310
1-[3-[(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-6-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]-3,4-dihydro-2H-pyran-4-yl]-1-indolyl]ethanoneEscherichia coli K-12Potency11.220210
[(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneEscherichia coli K-12Potency28.183810
(2S)-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]propanoic acid tert-butyl esterEscherichia coli K-12Potency35.481310
(2S)-4-methyl-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl esterEscherichia coli K-12Potency19.952610
(2S)-2-[[[5-[[methyl-(phenylmethyl)amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterEscherichia coli K-12Potency12.589310
N-(4-ethoxyphenyl)-2-[4-[2-(methylthio)ethyl]-2,5-dioxo-1-imidazolidinyl]acetamideEscherichia coli K-12Potency28.183810
2-[1-[1-hydroxy-10,13-dimethyl-3-[3,4,5-trihydroxy-6-[[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]oxan-2-yl]oxy-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]ethyl]-4,5-dimethyl-2,3-dihydropyran-6-oneEscherichia coli K-12Potency8.912510
(2R,4S)-4-cyclohexyl-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamideEscherichia coli K-12Potency22.387210
quercetinEscherichia coli K-12Potency5.706220
3-methoxymorphinan hydrochlorideEscherichia coli K-12Potency7.079510
methylnaloxonium iodideEscherichia coli K-12Potency10.000010
3,4-dichloro-n-methyl-n-(2-(1-pyrrolidinyl)cyclohexyl)-benzeneacetamide, (1s-cis)-isomerEscherichia coli K-12Potency5.011910
1-[5-(diethylsulfamoyl)-2-(4-methyl-1-piperazinyl)phenyl]-3-(2-fluorophenyl)ureaEscherichia coli K-12Potency25.118910
2-[(2,4-dichlorophenyl)methylthio]-1-methylimidazoleEscherichia coli K-12Potency6.309610
3-acetamido-N-[4-(4-methylsulfonylphenyl)-2-thiazolyl]-3-phenyl-N-prop-2-enylpropanamideEscherichia coli K-12Potency17.782810
LSM-24185Escherichia coli K-12Potency0.631010
LSM-16753Escherichia coli K-12Potency2.238710
2-imino-8-methyl-5-oxo-1-(2-oxolanylmethyl)-N-(2-phenylethyl)-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxamideEscherichia coli K-12Potency0.707910
peniprequinoloneEscherichia coli K-12Potency39.810710
(8R)-7-[(2-benzoylphenyl)-oxomethyl]-3-[3-[(1-oxo-3,3-diphenylpropyl)amino]phenyl]-1-oxa-2,7-diazaspiro[4.4]non-2-ene-8-carboxamideEscherichia coli K-12Potency19.952610
LSM-26549Escherichia coli K-12Potency35.481310
(5S)-1-[2-[3,5-bis(trifluoromethyl)phenyl]ethyl]-5-phenyl-4,5-dihydroimidazol-2-amineEscherichia coli K-12Potency39.810710
3-bromo-N-[2-[(3R,6S)-6-[(4-methoxyphenyl)methyl]-3-(phenylmethyl)-2,3,5,6-tetrahydroimidazo[1,2-a]imidazol-7-yl]ethyl]-4-methylbenzamideEscherichia coli K-12Potency35.481310
3-phenylpropanoic acid [3-(4-cyanophenyl)-2-cyclohexyl-7-methyl-6,8-dioxo-7-isoquinolinyl] esterEscherichia coli K-12Potency19.952610
3-phenylpropanoic acid [3-(4-cyanophenyl)-7-methyl-6,8-dioxo-2-[2-(2-pyridinyl)ethyl]-7-isoquinolinyl] esterEscherichia coli K-12Potency25.118910
8-[1-(1,3-benzodioxol-5-yl)-3-(1-piperidinyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneEscherichia coli K-12Potency22.387210
5,7-dimethoxy-4-methyl-8-[3-(4-morpholinyl)-1-(3,4,5-trimethoxyphenyl)propyl]-1-benzopyran-2-oneEscherichia coli K-12Potency22.387210
5,7-dimethoxy-8-[1-(4-methoxyphenyl)-3-(3-methyl-1-piperidinyl)-3-oxopropyl]-4-phenyl-1-benzopyran-2-oneEscherichia coli K-12Potency25.118910
8-{1-[4-(dimethylamino)phenyl]-3-(pyrrolidin-1-yl)propyl}-5,7-dimethoxy-4-pentyl-2H-chromen-2-oneEscherichia coli K-12Potency22.387210
8-[3-(diethylamino)-1-(4-methoxyphenyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneEscherichia coli K-12Potency19.952610
8-[1-[4-(dimethylamino)phenyl]-3-(3-methyl-1-piperidinyl)propyl]-5,7-dimethoxy-4-phenyl-1-benzopyran-2-oneEscherichia coli K-12Potency28.183810
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esterEscherichia coli K-12Potency39.810710
2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterEscherichia coli K-12Potency39.810710
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterEscherichia coli K-12Potency11.220210
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esterEscherichia coli K-12Potency25.118910
2-[(1R)-1-carboxy-2-(1-naphthalenyl)ethyl]-1,3-dioxo-5-isoindolecarboxylic acidEscherichia coli K-12Potency31.622810
N'-[(2-methoxyphenyl)-oxomethyl]-2-(4-morpholinyl)-4-thiazolecarbohydrazideEscherichia coli K-12Potency3.981110
N-(3-nitrophenyl)-3,4-dihydro-1H-isoquinoline-2-carboxamideEscherichia coli K-12Potency0.354810
cloprostenol sodiumEscherichia coli K-12Potency0.562310
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methoxyphenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency0.631010
6-(3,5-dimethyl-4-isoxazolyl)-N-[(2-ethoxyphenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency0.707910
3-(2,5-dimethoxyphenyl)-6-(3,4-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineEscherichia coli K-12Potency0.707910
2-[1-[2-(diethylamino)-2-oxoethyl]-3-indolyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoacetamideEscherichia coli K-12Potency25.118910
1-[(4-fluorophenyl)methyl]-3-[1-(4-propan-2-ylphenyl)propyl]thioureaEscherichia coli K-12Potency6.309610
1-(3-chlorophenyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)thioureaEscherichia coli K-12Potency0.707910
cefotiam hydrochlorideEscherichia coli K-12Potency100.000010
4-methoxy-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideEscherichia coli K-12Potency17.782810
N-[(5-bromo-2-methoxyphenyl)methyl]-4-methyl-2,3-dihydro-1,4-benzothiazine-6-carboxamideEscherichia coli K-12Potency25.118910
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-2-(1-piperidinyl)-1,3-benzothiazole-6-carboxamideEscherichia coli K-12Potency50.118710
N-[1,4-dimethyl-2,3-dioxo-7-(1-piperidinyl)-6-quinoxalinyl]-4-ethylbenzenesulfonamideEscherichia coli K-12Potency39.810710
5-[[4-(4-acetylphenyl)-1-piperazinyl]sulfonyl]-1,3-dihydroindol-2-oneEscherichia coli K-12Potency0.562310
amphidinolide bEscherichia coli K-12Potency7.943310
4-[4-(4-fluorophenyl)-1-piperazinyl]-N-[4-methyl-2-(4-morpholinyl)-6-quinolinyl]-4-oxobutanamideEscherichia coli K-12Potency14.125410
N-(5-chloro-2,4-dimethoxyphenyl)-1-methyl-4-(4-morpholinylsulfonyl)-2-pyrrolecarboxamideEscherichia coli K-12Potency31.622810
N-(3,5-dimethoxyphenyl)-6-methyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamideEscherichia coli K-12Potency0.562310
N-[3-[6-(1-azepanyl)-3-pyridazinyl]phenyl]-4-methylbenzenesulfonamideEscherichia coli K-12Potency0.707910
1-(2,3-dichlorophenyl)-3-pyridin-4-ylureaEscherichia coli K-12Potency0.562310
3-[1-[[1-(4-methylphenyl)cyclopropyl]-oxomethyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneEscherichia coli K-12Potency25.118910
3-[1-[oxo-(1-phenylcyclopropyl)methyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneEscherichia coli K-12Potency15.848910
3-[1-[[1-(4-chlorophenyl)cyclopropyl]-oxomethyl]-4-piperidinyl]-5-phenyl-1,3,4-oxadiazol-2-oneEscherichia coli K-12Potency28.183810
potassium aminobenzoateEscherichia coli K-12Potency5.011910
ampicillin sodiumEscherichia coli K-12Potency28.628820
cytomelEscherichia coli K-12Potency3.162310
piperacillin sodiumEscherichia coli K-12Potency56.234110
cefoxitin sodiumEscherichia coli K-12Potency39.810710
dicloxacillin sodiumEscherichia coli K-12Potency89.125110
nafcillin sodiumEscherichia coli K-12Potency100.000010
oxacillin sodiumEscherichia coli K-12Potency5.623410
sodium cholateEscherichia coli K-12Potency39.810710
canrenoate potassiumEscherichia coli K-12Potency3.162310
sodium diatrizoateEscherichia coli K-12Potency39.810710
cloxacillin sodiumEscherichia coli K-12Potency0.574620
sodium cephalothinEscherichia coli K-12Potency7.996020
dicloxacillin sodiumEscherichia coli K-12Potency0.072420
fractalsEscherichia coli K-12Potency19.952610
Taurocholic acid sodium salt hydrateEscherichia coli K-12Potency29.881620
sodium 2,6-dichloroindophenolEscherichia coli K-12Potency33.997220
nafcillin sodiumEscherichia coli K-12Potency5.317720
2-[4-[(4-cyclopentyloxyphenyl)methyl]-1-propan-2-yl-2-piperazinyl]ethanolEscherichia coli K-12Potency0.631010
cym51010Escherichia coli K-12Potency1.258910
LSM-21619Escherichia coli K-12Potency44.668410
(2R)-2-[[(3S)-3-acetamido-3-carboxy-1-oxopropyl]amino]pentanedioic acidEscherichia coli K-12Potency112.202010
gelsemineEscherichia coli K-12Potency22.387210
picrotoxininEscherichia coli K-12Potency0.631010
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl esterEscherichia coli K-12Potency39.810710
2-[[2-(phenoxymethyl)-4-quinazolinyl]thio]acetic acid methyl esterEscherichia coli K-12Potency0.631010
5-Methyl-1-phenyl-3-hexanyl sulfamateEscherichia coli K-12Potency2.238710
(5R)-5-tert-butyl-1-[(3S)-3-phenyl-3-(phenylthio)propyl]-2-azepanoneEscherichia coli K-12Potency0.354810
4-(4-chloro-3-nitrophenyl)-N-[2-(5,6-dichloro-1-propyl-2-benzimidazolyl)ethyl]-2-thiazolamineEscherichia coli K-12Potency11.220210
(2S)-2-[[oxo-[5-[oxo-(4-phenyl-1-piperazinyl)methyl]-1H-imidazol-4-yl]methyl]amino]-3-phenylpropanoic acid tert-butyl esterEscherichia coli K-12Potency14.125410
4-(1-((5-((2,6-dimethylphenoxy)methyl)-3-isoxazolyl)carbonyl)-4-piperidinyl)pyridineEscherichia coli K-12Potency35.481310
10-deacetyltaxolEscherichia coli K-12Potency17.782810
[5-[(3,4-difluorophenoxy)methyl]-3-isoxazolyl]-(3-propoxy-1-piperidinyl)methanoneEscherichia coli K-12Potency0.631010
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideEscherichia coli K-12Potency39.810710
4-[(2S)-2-[2-(4-ethoxyphenyl)ethylamino]-3-[[(2S)-1-(methylamino)hexan-2-yl]amino]propyl]phenolEscherichia coli K-12Potency10.257420
(2R)-3-[[(2S)-1-cyclohexyl-3-(methylamino)propan-2-yl]amino]-2-[2-[3-(trifluoromethyl)phenyl]ethylamino]-1-propanolEscherichia coli K-12Potency62.559420
(5S,5aR,8aS,8bR)-7-tert-butyl-5-(4-methoxyphenyl)-8b-methyl-2-(3-methylphenyl)-5a,8a-dihydro-5H-pyrrolo[1,2]pyrrolo[4,5-a]imidazole-1,3,6,8-tetroneEscherichia coli K-12Potency25.118910
cyclopropyl-[5-[[4-[[4-(2-methoxyphenyl)-1-piperazinyl]-oxomethyl]-1-piperidinyl]sulfonyl]-2-methyl-2,3-dihydroindol-1-yl]methanoneEscherichia coli K-12Potency4.581820
[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-[5-[(4-chloro-2-methoxyphenoxy)methyl]-3-isoxazolyl]methanoneEscherichia coli K-12Potency28.183810
N,3-dimethyl-5-propyl-N-(2-thiazolylmethyl)-2-benzofurancarboxamideEscherichia coli K-12Potency25.118910
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-methyl-5-thiadiazolecarboxamideEscherichia coli K-12Potency22.387210
N-methyl-N-(3-pyridinylmethyl)-5-(5,6,7,8-tetrahydronaphthalen-2-yloxymethyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency28.183810
1-[(1-ethyl-3-methyl-4-pyrazolyl)methyl]-N-[4-(2-fluorophenoxy)phenyl]-4-piperidinecarboxamideEscherichia coli K-12Potency28.183810
(5R)-5-tert-butyl-1-[(3S)-3-[(4-methylphenyl)thio]-3-phenylpropyl]-2-azepanoneEscherichia coli K-12Potency112.202010
3-(2,4-dimethoxyphenyl)-N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]-2-oxoethyl]-4-oxo-1-phthalazinecarboxamideEscherichia coli K-12Potency14.125410
N-[3-(3-chlorophenyl)phenyl]-1-(3-oxolanylmethyl)-4-piperidinecarboxamideEscherichia coli K-12Potency35.481310
dafadine OEscherichia coli K-12Potency12.209720
5-[(3,4-dimethylphenoxy)methyl]-N-methyl-N-(4-oxanylmethyl)-3-isoxazolecarboxamideEscherichia coli K-12Potency15.848910
4-[oxo-[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]methyl]-1-piperazinecarboxylic acid ethyl esterEscherichia coli K-12Potency14.125410
[5-[(4-methoxy-1-naphthalenyl)oxymethyl]-3-isoxazolyl]-(4-methoxy-1-piperidinyl)methanoneEscherichia coli K-12Potency39.810710
2-(3-Amino-3-oxopropyl)-3-(4-methylbenzoyl)-2H-indazole 1-oxideEscherichia coli K-12Potency100.000010
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-2,5-dimethyl-3-pyrazolecarboxamideEscherichia coli K-12Potency28.183810
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-5-(methoxymethyl)-2-furancarboxamideEscherichia coli K-12Potency16.903620
2-[3-(4-morpholinyl)propylamino]-9-xanthenoneEscherichia coli K-12Potency73.841620
[5-[(2-methoxyphenoxy)methyl]-3-isoxazolyl]-(4-methyl-3-phenyl-1-piperazinyl)methanoneEscherichia coli K-12Potency12.589310
glycocholic acidEscherichia coli K-12Potency31.622810
(3S)-3-cyclopentyl-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterEscherichia coli K-12Potency112.202010
dragonamide cEscherichia coli K-12Potency10.000010
4-ethoxy-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideEscherichia coli K-12Potency22.387210
stachyoseEscherichia coli K-12Potency112.202010
(7R,13S)-6-[(2S)-4-(Dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-14-ethyl-7,12,13-trihydroxy-4-[(4R)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-10-(2-methoxyethoxymethoxyimino)-3,5,7,9,11,13-hexamethyl-oxacyclotetradecan-2-oneEscherichia coli K-12Potency12.863120
(3S,3Ar,4S,9aS,9bR)-4-hydroxy-3,6,9-trimethyl-3,3a,4,5-tetrahydroazuleno[4,5-b]furan-2,7(9aH,9bH)-dione hydrateEscherichia coli K-12Potency15.848910
1-(2,6-difluorophenyl)sulfonyl-4-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-1,4-diazepaneEscherichia coli K-12Potency22.387210
6-(3-methoxyphenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency1.122010
6-(2-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineEscherichia coli K-12Potency1.412510
6-(3-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineEscherichia coli K-12Potency0.631010
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineEscherichia coli K-12Potency0.562310
6-(3-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineEscherichia coli K-12Potency39.810710
N-(1,3-benzodioxol-5-ylmethyl)-6-(2-chlorophenyl)-4-quinazolinamineEscherichia coli K-12Potency0.631010
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-pyridinyl)-4-quinazolinamineEscherichia coli K-12Potency0.631010
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-furanyl)-4-quinazolinamineEscherichia coli K-12Potency3.162310
6-(2-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency44.668410
6-(1,3-benzodioxol-5-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency31.622810
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency0.707910
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineEscherichia coli K-12Potency19.952610
5-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]methyl]-8-quinolinolEscherichia coli K-12Potency0.631010
1H-indole-4-carboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterEscherichia coli K-12Potency0.354810
6-(3-cyclopentyloxy-4-methoxyphenyl)-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineEscherichia coli K-12Potency25.118910
6-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineEscherichia coli K-12Potency39.810710
6-[3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl]-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineEscherichia coli K-12Potency22.387210
6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-3-[2-(trifluoromethyl)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineEscherichia coli K-12Potency15.848910
3-(2,5-dimethoxyphenyl)-6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineEscherichia coli K-12Potency39.810710
1-[4-[4-[(3-methylphenyl)methylamino]phenyl]-1-piperazinyl]ethanoneEscherichia coli K-12Potency28.183810
3-cyclohexyl-1-[[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-8-[[(4-methoxyanilino)-oxomethyl]amino]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methylureaEscherichia coli K-12Potency39.810710
1-cyclohexyl-3-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-2-[[(4-methoxyphenyl)sulfonyl-methylamino]methyl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]ureaEscherichia coli K-12Potency17.782810
N-[(2S,3S)-2-[[(3,4-dichlorophenyl)methyl-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]-2-thiophenesulfonamideEscherichia coli K-12Potency19.952610
N-[(2S,3S)-2-[[(4-fluorophenyl)sulfonyl-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]cyclopropanecarboxamideEscherichia coli K-12Potency39.810710
1-[(2S,3R)-2-[[cyclohexylmethyl(methyl)amino]methyl]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaEscherichia coli K-12Potency22.387210
N-[(2S,3S)-2-[[cyclohexylmethyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-(4-morpholinyl)propanamideEscherichia coli K-12Potency35.481310
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-2-[[[(4-methoxyanilino)-oxomethyl]-methylamino]methyl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]cyclohexanecarboxamideEscherichia coli K-12Potency31.622810
1-[[(2R,3S)-8-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]ureaEscherichia coli K-12Potency11.220210
3-cyclohexyl-1-[[(2S,3R)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-10-[[oxo-(propan-2-ylamino)methyl]amino]-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methylureaEscherichia coli K-12Potency35.481310
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[(4-phenoxyphenyl)methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]-4-pyridinecarboxamideEscherichia coli K-12Potency19.952610
N-[[(2S,3S)-10-(dimethylamino)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-N,3,5-trimethyl-4-isoxazolesulfonamideEscherichia coli K-12Potency39.810710
N-[[(2S,3S)-10-(dimethylamino)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-4-methoxy-N-methylbenzenesulfonamideEscherichia coli K-12Potency28.183810
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[oxo-[4-(trifluoromethyl)anilino]methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-2-phenylacetamideEscherichia coli K-12Potency39.810710
N-[(2R,3S)-2-[[(4-chlorophenyl)sulfonyl-methylamino]methyl]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-4,4,4-trifluorobutanamideEscherichia coli K-12Potency7.943310
N-(2-aminophenyl)-4-[[[(2S,3S)-10-[[cyclohexyl(oxo)methyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl-methylamino]methyl]benzamideEscherichia coli K-12Potency11.220210
1-[[(2S,3S)-10-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-3-(4-methoxyphenyl)-1-methylureaEscherichia coli K-12Potency28.183810
1-(4-fluorophenyl)-3-[(2R,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-(phenylmethyl)amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]ureaEscherichia coli K-12Potency35.481310
N-[(2S,3S)-2-[[[(cyclohexylamino)-oxomethyl]-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-4,4,4-trifluorobutanamideEscherichia coli K-12Potency31.622810
3-cyclohexyl-1-[[(2S,3S)-8-[(4-fluorophenyl)sulfonylamino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methylureaEscherichia coli K-12Potency28.183810
N-[(2S,3R)-5-[(2S)-1-hydroxypropan-2-yl]-2-[[[(4-methoxyanilino)-oxomethyl]-methylamino]methyl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-(4-morpholinyl)propanamideEscherichia coli K-12Potency31.622810
3-cyclohexyl-1-[[(2R,3R)-10-[(4-fluorophenyl)sulfonylamino]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methylureaEscherichia coli K-12Potency35.481310
N-[(2R,3S)-2-[[cyclopropylmethyl(methyl)amino]methyl]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-4,4,4-trifluorobutanamideEscherichia coli K-12Potency25.118910
4-chloro-N-[(2R,3R)-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl(pyridin-4-ylmethyl)amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]benzenesulfonamideEscherichia coli K-12Potency31.622810
1-[[(2S,3S)-10-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]ureaEscherichia coli K-12Potency25.118910
N-[(2S,3S)-2-[[(3,4-dichlorophenyl)methyl-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-2-(1-tetrazolyl)acetamideEscherichia coli K-12Potency28.183810
N-[(2S,3S)-2-[[cyclohexylmethyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]-4-methoxybenzenesulfonamideEscherichia coli K-12Potency28.183810
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-(phenylmethyl)amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]-4-pyridinecarboxamideEscherichia coli K-12Potency39.810710
N-[(2S,3S)-2-[[(4-fluorophenyl)sulfonyl-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-(4-morpholinyl)propanamideEscherichia coli K-12Potency28.183810
N-[(2R,3S)-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[(1-naphthalenylamino)-oxomethyl]amino]methyl]-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-2-phenylacetamideEscherichia coli K-12Potency35.481310
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[oxo-[4-(trifluoromethyl)anilino]methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-4-pyridinecarboxamideEscherichia coli K-12Potency39.810710
1-[[(2S,3R)-10-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]ureaEscherichia coli K-12Potency17.782810
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[oxo-[4-(trifluoromethyl)anilino]methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]cyclohexanecarboxamideEscherichia coli K-12Potency19.952610
1-[[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-10-[[oxo-[4-(trifluoromethyl)anilino]methyl]amino]-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-phenylureaEscherichia coli K-12Potency31.622810
N-[(2S,3S)-2-[[[(cyclohexylamino)-oxomethyl]-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]cyclohexanecarboxamideEscherichia coli K-12Potency12.589310
gypenoside ixEscherichia coli K-12Potency7.943310
saikosaponin bEscherichia coli K-12Potency12.589310
1-[[(2S,3S)-10-(dimethylamino)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]ureaEscherichia coli K-12Potency25.118910
1-[[(2R,3R)-5-[(2R)-1-hydroxypropan-2-yl]-9-[[(4-methoxyanilino)-oxomethyl]amino]-3-methyl-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-2-yl]methyl]-1-methyl-3-phenylureaEscherichia coli K-12Potency35.481310
N-[(2R,3R)-2-[[(4-fluorophenyl)sulfonyl-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-2-(1-methyl-3-indolyl)acetamideEscherichia coli K-12Potency17.782810
1-[(2R,3R)-2-[[benzenesulfonyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-[4-(trifluoromethyl)phenyl]ureaEscherichia coli K-12Potency39.810710
2-bromo-6-[(2,4-difluorophenyl)methyl]-4-methyl-5-thieno[3,4]pyrrolo[1,3-d]pyridazinoneEscherichia coli K-12Potency0.631010
3-[(4-fluorophenyl)methyl]-5-methyl-4-thieno[3,4]pyrrolo[1,3-d]pyrimidinoneEscherichia coli K-12Potency20.534820
Majusculamide ABEscherichia coli K-12Potency15.848910
lyngbyastatin 3Escherichia coli K-12Potency7.943310
N-[(5-bromo-8-hydroxy-7-quinolinyl)-(2-furanyl)methyl]propanamideEscherichia coli K-12Potency0.707910
N-[(8-methoxy-5-nitro-7-quinolinyl)-thiophen-2-ylmethyl]propanamideEscherichia coli K-12Potency5.889220
oxytetracycline, anhydrousEscherichia coli K-12Potency100.000010
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamideEscherichia coli K-12Potency0.631010
4-hydroxy-2-oxo-1-propyl-N-(pyridin-4-ylmethyl)-3-quinolinecarboxamideEscherichia coli K-12Potency7.079510
lfm a13Escherichia coli K-12Potency2.818410
mobicEscherichia coli K-12Potency39.810710
LSM-17430Escherichia coli K-12Potency7.943310
ethyl 1-benzyl-3-hydroxy-2(5h)-oxopyrrole-4-carboxylateEscherichia coli K-12Potency100.000010
warfarinEscherichia coli K-12Potency3.548110
N-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-1-prop-2-enyl-3-quinolinecarboxamideEscherichia coli K-12Potency56.234110
N'-[(2-chlorophenyl)-oxomethyl]-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarbohydrazideEscherichia coli K-12Potency89.125110
7-(diethylamino)-4-hydroxy-1-benzopyran-2-oneEscherichia coli K-12Potency18.854120
LSM-28526Escherichia coli K-12Potency11.220210
LSM-23565Escherichia coli K-12Potency1.412510
methacycline monohydrochlorideEscherichia coli K-12Potency50.118710
mysteclin fEscherichia coli K-12Potency13.131120
demeclocycline hydrochlorideEscherichia coli K-12Potency19.952610
4-hydroxy-3-(1-piperidinylmethyl)-1-benzopyran-2-oneEscherichia coli K-12Potency100.000010
lornoxicamEscherichia coli K-12Potency7.943310
1-ethyl-4-hydroxy-2-oxo-N-(3-pyridinylmethyl)-3-quinolinecarboxamideEscherichia coli K-12Potency56.498220
2-(4-hydroxy-2-oxo-1H-quinolin-3-yl)acetic acid pentyl esterEscherichia coli K-12Potency0.707910
4-hydroxy-N-(2-methyl-4-oxo-3-quinazolinyl)-1-(2-methylpropyl)-2-oxo-5,6,7,8-tetrahydroquinoline-3-carboxamideEscherichia coli K-12Potency39.810710
4-hydroxy-1,7,7-trimethyl-3-(2,4,6-trimethylphenyl)-6,8-dihydroquinoline-2,5-dioneEscherichia coli K-12Potency10.000010
valacyclovirEscherichia coli K-12Potency2.818410
sildenafilEscherichia coli K-12Potency50.118710
oxypurinolEscherichia coli K-12Potency5.011910
kf38789Escherichia coli K-12Potency31.622810
salinazidEscherichia coli K-12Potency5.011910
zinc08438472Escherichia coli K-12Potency3.162310
ImidazosagatriazinoneEscherichia coli K-12Potency35.481310
4-oxo-2-(trifluoromethyl)-1H-quinazoline-6-carboxylic acid ethyl esterEscherichia coli K-12Potency0.631010
2,4-diaminohypoxanthineEscherichia coli K-12Potency44.668410
N-(2,3-dimethylphenyl)-5-(2-fluorophenyl)-6H-1,3,4-thiadiazin-2-amineEscherichia coli K-12Potency12.589310
2-[[3-[(2-ethoxy-2-oxoethyl)thio]-5-oxo-2H-1,2,4-triazin-6-yl]amino]acetic acid butyl esterEscherichia coli K-12Potency0.794310
2-[(4-chlorophenyl)methylthio]-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-oneEscherichia coli K-12Potency0.631010
2-pyridin-4-yl-1H-quinazolin-4-oneEscherichia coli K-12Potency89.125110
MMP-9-IN-1Escherichia coli K-12Potency1.584910
2-[[2-[1-(2-methoxyethyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]thio]-6-propyl-1H-pyrimidin-4-oneEscherichia coli K-12Potency0.354810
N-(1,3-benzodioxol-5-yl)-2-[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]acetamideEscherichia coli K-12Potency28.183810
N-[4-(6-chloro-5-nitro-1H-benzimidazol-2-yl)phenyl]acetamideEscherichia coli K-12Potency89.125110
N-(1,3-benzodioxol-5-ylmethyl)-3-methoxy-N-[(4-oxo-1H-quinazolin-2-yl)methyl]benzamideEscherichia coli K-12Potency44.668410
N-tert-butyl-3-(3-tert-butyl-1-methyl-7-oxo-4H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxybenzenesulfonamideEscherichia coli K-12Potency19.952610
1-(3-methoxyphenyl)-2-[4-oxo-6-(trifluoromethyl)-1H-pyrimidin-2-yl]guanidineEscherichia coli K-12Potency70.794610
lomofunginEscherichia coli K-12Potency56.234110
N-[(4-oxo-1H-quinazolin-2-yl)methyl]-N-(2-phenylethyl)butanamideEscherichia coli K-12Potency4.466810
N-[4-[2-(2-methoxyethylamino)-6H-1,3,4-thiadiazin-5-yl]phenyl]acetamideEscherichia coli K-12Potency0.631010
N-[(3-methoxyphenyl)methyl]-4H-3,1-benzothiazin-2-amineEscherichia coli K-12Potency56.234110
3-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-6-(phenylmethyl)-2H-1,2,4-triazin-5-oneEscherichia coli K-12Potency56.234110
5-[1-[(2-chlorophenyl)methyl]-2,5-dimethyl-3-pyrrolyl]-N-(1-methoxypropan-2-yl)-6H-1,3,4-thiadiazin-2-amineEscherichia coli K-12Potency35.481310
2-[(dimethylamino)methyl]-4-spiro[1,6-dihydrobenzo[h]quinazoline-5,1'-cyclohexane]oneEscherichia coli K-12Potency7.079510
4-methyl-3-phenyl-1,2-dihydropyrazolo[3,4-b]pyridin-6-oneEscherichia coli K-12Potency1.000010
t16ainh-a01Escherichia coli K-12Potency14.125410
LSM-20825Escherichia coli K-12Potency15.848910
N-[2-[(2-chlorophenyl)methylthio]-4-oxo-1H-pyrimidin-6-yl]-4-methylbenzenesulfonamideEscherichia coli K-12Potency5.792420
2-[(5-cyano-4-oxo-6-phenyl-1H-pyrimidin-2-yl)thio]-N-phenylacetamideEscherichia coli K-12Potency44.668410
N-(4-methoxyphenyl)-2-[[6-[(4-methylphenyl)sulfonylamino]-4-oxo-1H-pyrimidin-2-yl]thio]acetamideEscherichia coli K-12Potency17.782810
3-(3-ethoxypropyl)-1-[(4-oxo-1H-quinazolin-2-yl)methyl]-1-(phenylmethyl)thioureaEscherichia coli K-12Potency25.118910
7,9-dimethyl-2-(phenylmethylthio)-1H-pyrido[2,3]thieno[2,4-b]pyrimidin-4-oneEscherichia coli K-12Potency3.981110
N-(4-fluorophenyl)-2-(3-hydroxypropyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamideEscherichia coli K-12Potency44.668410
7-[[ethyl-[(4-oxo-1H-quinazolin-2-yl)methyl]amino]methyl]-5-thiazolo[3,2-a]pyrimidinoneEscherichia coli K-12Potency5.011910

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
thiophene-2-carboxylateEscherichia coli K-12Ki40,000.000011
4-amino-3-hydroxybenzoic acidEscherichia coli K-12Ki19,000.000011
2-[(1R)-1-carboxy-2-(1-naphthalenyl)ethyl]-1,3-dioxo-5-isoindolecarboxylic acidEscherichia coli K-12Ki5.000010