A protein that is a translation product of the pknB gene in Mycobacterium tuberculosis H37Rv. [PRO:DNx, UniProtKB:P9WI81]
EC 2.7.11.1
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
imatinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
staurosporine | Mycobacterium tuberculosis H37Rv | Kd | 0.0880 | 1 | 1 |
gefitinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
lestaurtinib | Mycobacterium tuberculosis H37Rv | Kd | 0.0550 | 1 | 1 |
vatalanib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
ruboxistaurin | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
canertinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
birb 796 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
sb 203580 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
enzastaurin | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
erlotinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
lapatinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
sorafenib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
pd 173955 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
s 1033 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
bms 387032 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
tandutinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
vx-745 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
dasatinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
zd 6474 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
alvocidib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
bosutinib | Mycobacterium tuberculosis H37Rv | Kd | 5.5000 | 1 | 1 |
su 11248 | Mycobacterium tuberculosis H37Rv | Kd | 0.0870 | 1 | 1 |
vx680 | Mycobacterium tuberculosis H37Rv | Kd | 2.2000 | 1 | 1 |
axitinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
pd 184352 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
bms345541 | Mycobacterium tuberculosis H37Rv | Kd | 2.4000 | 1 | 1 |
midostaurin | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
ki 20227 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
pi103 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
hki 272 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
tofacitinib | Mycobacterium tuberculosis H37Rv | Kd | 2.0000 | 1 | 1 |
n-(6-chloro-7-methoxy-9h-beta-carbolin-8-yl)-2-methylnicotinamide | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
cediranib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
masitinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
pazopanib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
azd 6244 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
su 14813 | Mycobacterium tuberculosis H37Rv | Kd | 0.3200 | 1 | 1 |
bibw 2992 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
tg100-115 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
pha 665752 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one | Mycobacterium tuberculosis H37Rv | Kd | 0.0340 | 1 | 1 |
brivanib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
at 7519 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
bi 2536 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
nvp-ast487 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
kw 2449 | Mycobacterium tuberculosis H37Rv | Kd | 0.2400 | 1 | 1 |
abt 869 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
gw 2580 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
crizotinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
chir-265 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
motesanib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
mln8054 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
GDC-0879 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
gsk 461364 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
azd 1152-hqpa | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
nvp-tae684 | Mycobacterium tuberculosis H37Rv | Kd | 1.2000 | 1 | 1 |
fedratinib | Mycobacterium tuberculosis H37Rv | Kd | 0.1000 | 1 | 1 |
gsk690693 | Mycobacterium tuberculosis H37Rv | Kd | 0.0032 | 1 | 1 |
gdc 0941 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
plx 4720 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
sgx 523 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
quizartinib | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
incb-018424 | Mycobacterium tuberculosis H37Rv | Kd | 4.2000 | 1 | 1 |
gsk 1838705a | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
gsk 1363089 | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
chir 258 | Mycobacterium tuberculosis H37Rv | Kd | 0.3000 | 1 | 1 |
nintedanib | Mycobacterium tuberculosis H37Rv | Kd | 0.0036 | 1 | 1 |
pp242 | Mycobacterium tuberculosis H37Rv | Kd | 2.9000 | 1 | 1 |