Page last updated: 2024-08-07 23:44:36

Serine/threonine-protein kinase PknB

A protein that is a translation product of the pknB gene in Mycobacterium tuberculosis H37Rv. [PRO:DNx, UniProtKB:P9WI81]

Synonyms

EC 2.7.11.1

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Compounds (69)

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
imatinibMycobacterium tuberculosis H37RvKd10.000011
staurosporineMycobacterium tuberculosis H37RvKd0.088011
gefitinibMycobacterium tuberculosis H37RvKd10.000011
lestaurtinibMycobacterium tuberculosis H37RvKd0.055011
vatalanibMycobacterium tuberculosis H37RvKd10.000011
ruboxistaurinMycobacterium tuberculosis H37RvKd10.000011
canertinibMycobacterium tuberculosis H37RvKd10.000011
birb 796Mycobacterium tuberculosis H37RvKd10.000011
sb 203580Mycobacterium tuberculosis H37RvKd10.000011
enzastaurinMycobacterium tuberculosis H37RvKd10.000011
erlotinibMycobacterium tuberculosis H37RvKd10.000011
lapatinibMycobacterium tuberculosis H37RvKd10.000011
sorafenibMycobacterium tuberculosis H37RvKd10.000011
pd 173955Mycobacterium tuberculosis H37RvKd10.000011
s 1033Mycobacterium tuberculosis H37RvKd10.000011
bms 387032Mycobacterium tuberculosis H37RvKd10.000011
tandutinibMycobacterium tuberculosis H37RvKd10.000011
vx-745Mycobacterium tuberculosis H37RvKd10.000011
dasatinibMycobacterium tuberculosis H37RvKd10.000011
zd 6474Mycobacterium tuberculosis H37RvKd10.000011
alvocidibMycobacterium tuberculosis H37RvKd10.000011
bosutinibMycobacterium tuberculosis H37RvKd5.500011
su 11248Mycobacterium tuberculosis H37RvKd0.087011
vx680Mycobacterium tuberculosis H37RvKd2.200011
axitinibMycobacterium tuberculosis H37RvKd10.000011
pd 184352Mycobacterium tuberculosis H37RvKd10.000011
bms345541Mycobacterium tuberculosis H37RvKd2.400011
midostaurinMycobacterium tuberculosis H37RvKd10.000011
ki 20227Mycobacterium tuberculosis H37RvKd10.000011
pi103Mycobacterium tuberculosis H37RvKd10.000011
hki 272Mycobacterium tuberculosis H37RvKd10.000011
tofacitinibMycobacterium tuberculosis H37RvKd2.000011
n-(6-chloro-7-methoxy-9h-beta-carbolin-8-yl)-2-methylnicotinamideMycobacterium tuberculosis H37RvKd10.000011
cediranibMycobacterium tuberculosis H37RvKd10.000011
masitinibMycobacterium tuberculosis H37RvKd10.000011
pazopanibMycobacterium tuberculosis H37RvKd10.000011
azd 6244Mycobacterium tuberculosis H37RvKd10.000011
su 14813Mycobacterium tuberculosis H37RvKd0.320011
bibw 2992Mycobacterium tuberculosis H37RvKd10.000011
tg100-115Mycobacterium tuberculosis H37RvKd10.000011
pha 665752Mycobacterium tuberculosis H37RvKd10.000011
6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-oneMycobacterium tuberculosis H37RvKd0.034011
brivanibMycobacterium tuberculosis H37RvKd10.000011
at 7519Mycobacterium tuberculosis H37RvKd10.000011
bi 2536Mycobacterium tuberculosis H37RvKd10.000011
nvp-ast487Mycobacterium tuberculosis H37RvKd10.000011
kw 2449Mycobacterium tuberculosis H37RvKd0.240011
abt 869Mycobacterium tuberculosis H37RvKd10.000011
gw 2580Mycobacterium tuberculosis H37RvKd10.000011
crizotinibMycobacterium tuberculosis H37RvKd10.000011
chir-265Mycobacterium tuberculosis H37RvKd10.000011
motesanibMycobacterium tuberculosis H37RvKd10.000011
mln8054Mycobacterium tuberculosis H37RvKd10.000011
GDC-0879Mycobacterium tuberculosis H37RvKd10.000011
gsk 461364Mycobacterium tuberculosis H37RvKd10.000011
azd 1152-hqpaMycobacterium tuberculosis H37RvKd10.000011
nvp-tae684Mycobacterium tuberculosis H37RvKd1.200011
fedratinibMycobacterium tuberculosis H37RvKd0.100011
gsk690693Mycobacterium tuberculosis H37RvKd0.003211
gdc 0941Mycobacterium tuberculosis H37RvKd10.000011
plx 4720Mycobacterium tuberculosis H37RvKd10.000011
sgx 523Mycobacterium tuberculosis H37RvKd10.000011
quizartinibMycobacterium tuberculosis H37RvKd10.000011
incb-018424Mycobacterium tuberculosis H37RvKd4.200011
gsk 1838705aMycobacterium tuberculosis H37RvKd10.000011
gsk 1363089Mycobacterium tuberculosis H37RvKd10.000011
chir 258Mycobacterium tuberculosis H37RvKd0.300011
nintedanibMycobacterium tuberculosis H37RvKd0.003611
pp242Mycobacterium tuberculosis H37RvKd2.900011