Page last updated: 2024-08-08 00:43:58

urokinase-type plasminogen activator precursor

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (918)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
dinitrochlorobenzeneMus musculus (house mouse)Potency1.258910
catecholMus musculus (house mouse)Potency1.778310
undenMus musculus (house mouse)Potency7.943310
sarcosineMus musculus (house mouse)Potency1.995310
1,10-phenanthrolineMus musculus (house mouse)Potency1.584910
1-anilino-8-naphthalenesulfonateMus musculus (house mouse)Potency2.511910
pd 173074Mus musculus (house mouse)Potency7.079510
p-chloromercuribenzoic acidMus musculus (house mouse)Potency7.943310
ethylisopropylamilorideMus musculus (house mouse)Potency8.912510
edoxudinMus musculus (house mouse)Potency10.000010
hydroxyindoleacetic acidMus musculus (house mouse)Potency11.220210
tyrphostin a23Mus musculus (house mouse)Potency3.162310
albendazoleMus musculus (house mouse)Potency0.014110
amiodaroneMus musculus (house mouse)Potency14.689210
anabasineMus musculus (house mouse)Potency1.000010
isodeoxypodophyllotoxinMus musculus (house mouse)Potency0.316210
aristolochic acid iMus musculus (house mouse)Potency14.125410
astemizoleMus musculus (house mouse)Potency1.258910
bufexamacMus musculus (house mouse)Potency4.466810
chlorambucilMus musculus (house mouse)Potency7.079510
chloroxineMus musculus (house mouse)Potency22.387210
clofoctolMus musculus (house mouse)Potency14.125410
clotrimazoleMus musculus (house mouse)Potency12.589310
colchicine, (+-)-isomerMus musculus (house mouse)Potency0.005010
dacarbazineMus musculus (house mouse)Potency6.309610
deferoxamineMus musculus (house mouse)Potency14.125410
disulfiramMus musculus (house mouse)Potency12.589310
ebselenMus musculus (house mouse)Potency12.589310
ellipticineMus musculus (house mouse)Potency0.891310
ethacrynic acidMus musculus (house mouse)Potency4.466810
fenbendazoleMus musculus (house mouse)Potency0.020010
fluorouracilMus musculus (house mouse)Potency0.014110
fluspirileneMus musculus (house mouse)Potency11.220210
glimepirideMus musculus (house mouse)Potency11.220210
fluorometholoneMus musculus (house mouse)Potency8.912510
1-(5-isoquinolinesulfonyl)-2-methylpiperazineMus musculus (house mouse)Potency8.912510
hexachloropheneMus musculus (house mouse)Potency7.943310
beta-thujaplicinMus musculus (house mouse)Potency8.912510
hycanthoneMus musculus (house mouse)Potency2.818410
hydroxyureaMus musculus (house mouse)Potency8.912510
ibudilastMus musculus (house mouse)Potency0.446710
indoprofenMus musculus (house mouse)Potency4.466810
leflunomideMus musculus (house mouse)Potency8.912510
lidoflazineMus musculus (house mouse)Potency10.000010
miconazoleMus musculus (house mouse)Potency12.589310
nabumetoneMus musculus (house mouse)Potency7.079510
niclosamideMus musculus (house mouse)Potency3.548110
nifedipineMus musculus (house mouse)Potency1.258910
nisoldipineMus musculus (house mouse)Potency12.589310
masoprocolMus musculus (house mouse)Potency1.995310
6,7-dimethoxy-3-(4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl)-3H-isobenzofuran-1-oneMus musculus (house mouse)Potency12.589310
nu2058Mus musculus (house mouse)Potency8.912510
oxamniquineMus musculus (house mouse)Potency1.122010
oxyphenbutazoneMus musculus (house mouse)Potency0.891310
5-hydroxy-4-methoxy-5-(1-methylethenyl)-2-furanoneMus musculus (house mouse)Potency10.000010
prochlorperazineMus musculus (house mouse)Potency12.589310
propachlorMus musculus (house mouse)Potency6.309610
pyrimethamineMus musculus (house mouse)Potency0.707910
riluzoleMus musculus (house mouse)Potency12.589310
aurinMus musculus (house mouse)Potency1.995310
vorinostatMus musculus (house mouse)Potency0.063110
sulfathiazoleMus musculus (house mouse)Potency5.011910
terazosinMus musculus (house mouse)Potency3.548110
thiabendazoleMus musculus (house mouse)Potency10.000010
thiramMus musculus (house mouse)Potency2.238710
triamtereneMus musculus (house mouse)Potency2.238710
tyrphostin a9Mus musculus (house mouse)Potency0.891310
donepezil hydrochlorideMus musculus (house mouse)Potency14.125410
mitomycinMus musculus (house mouse)Potency3.981110
oxyphenonium bromideMus musculus (house mouse)Potency1.122010
phentolamineMus musculus (house mouse)Potency12.589310
2-aminophenolMus musculus (house mouse)Potency3.981110
isoproterenol hydrochlorideMus musculus (house mouse)Potency12.589310
estroneMus musculus (house mouse)Potency12.589310
methylprednisolone acetateMus musculus (house mouse)Potency10.000010
dichlororibofuranosylbenzimidazoleMus musculus (house mouse)Potency8.912510
azauridineMus musculus (house mouse)Potency0.316210
amifampridineMus musculus (house mouse)Potency3.162310
racepinephrine hydrochlorideMus musculus (house mouse)Potency5.623410
ethinyl estradiolMus musculus (house mouse)Potency10.000010
9,10-dimethyl-1,2-benzanthraceneMus musculus (house mouse)Potency11.220210
methyltestosteroneMus musculus (house mouse)Potency12.589310
bromodeoxyuridineMus musculus (house mouse)Potency1.122010
methylene blueMus musculus (house mouse)Potency2.238710
desoxycorticosteroneMus musculus (house mouse)Potency3.981110
cycloheximideMus musculus (house mouse)Potency0.501210
fluocinolone acetonideMus musculus (house mouse)Potency2.238710
tubercidinMus musculus (house mouse)Potency0.316210
cordycepinMus musculus (house mouse)Potency4.466810
n,n'-diphenyl-4-phenylenediamineMus musculus (house mouse)Potency6.309610
benzanthroneMus musculus (house mouse)Potency8.912510
1-amino-2-methylanthraquinoneMus musculus (house mouse)Potency11.220210
skatoleMus musculus (house mouse)Potency2.818410
9,10-phenanthrenequinoneMus musculus (house mouse)Potency1.412510
acriflavine chlorideMus musculus (house mouse)Potency1.258910
Ethyl 2-aminobenzoateMus musculus (house mouse)Potency4.466810
gramineMus musculus (house mouse)Potency12.589310
2-amino-4-methylphenolMus musculus (house mouse)Potency2.818410
p-tert-butyl catecholMus musculus (house mouse)Potency7.943310
methyl gallateMus musculus (house mouse)Potency10.000010
methylenebis(chloroaniline)Mus musculus (house mouse)Potency3.162310
triclocarbanMus musculus (house mouse)Potency28.183810
4-aminodiphenylamineMus musculus (house mouse)Potency7.943310
n-isopropyl-n-phenyl-4-phenylenediamineMus musculus (house mouse)Potency10.000010
1,3-diphenylureaMus musculus (house mouse)Potency11.220210
1-amino-4-hydroxyanthraquinoneMus musculus (house mouse)Potency12.589310
dianisidineMus musculus (house mouse)Potency4.466810
benzethonium chlorideMus musculus (house mouse)Potency12.589310
sulfan blueMus musculus (house mouse)Potency7.079510
pyrazolanthroneMus musculus (house mouse)Potency22.052620
peucedaninMus musculus (house mouse)Potency6.309610
protocatechualdehydeMus musculus (house mouse)Potency5.623410
4'-(chloroacetyl)acetanilideMus musculus (house mouse)Potency12.589310
2-chloroadenosineMus musculus (house mouse)Potency4.466810
2-fluoroadenosineMus musculus (house mouse)Potency0.014110
mequinolMus musculus (house mouse)Potency6.309610
dydrogesteroneMus musculus (house mouse)Potency12.589310
diiodotyrosineMus musculus (house mouse)Potency2.511910
azacitidineMus musculus (house mouse)Potency0.794310
3-(11-dibenzo[1,2-a-1',2'-e][7]annulenylidene)-N-methyl-1-propanamineMus musculus (house mouse)Potency11.220210
isocorydineMus musculus (house mouse)Potency7.943310
rheinMus musculus (house mouse)Potency12.589310
cepharanthineMus musculus (house mouse)Potency12.589310
3,4-toluenediamineMus musculus (house mouse)Potency6.309610
4,4'-diaminoazobenzeneMus musculus (house mouse)Potency4.466810
maleimideMus musculus (house mouse)Potency10.000010
myristic acidMus musculus (house mouse)Potency12.589310
propoxycaine hydrochlorideMus musculus (house mouse)Potency12.589310
eriodictyolMus musculus (house mouse)Potency10.000010
neutral red baseMus musculus (house mouse)Potency28.183810
3-hydroxyflavoneMus musculus (house mouse)Potency28.183810
aminacrineMus musculus (house mouse)Potency1.000010
9-nitroanthraceneMus musculus (house mouse)Potency7.079510
Berberine chloride (TN)Mus musculus (house mouse)Potency6.309610
clopamideMus musculus (house mouse)Potency8.912510
2-phenylbenzimidazoleMus musculus (house mouse)Potency5.011910
2,2'-diaminodiphenyldisulfideMus musculus (house mouse)Potency3.981110
n-acetylmelphalanMus musculus (house mouse)Potency7.079510
amiloride hydrochloride, anhydrousMus musculus (house mouse)Potency0.251210
pimozideMus musculus (house mouse)Potency12.589310
azaribineMus musculus (house mouse)Potency0.011210
2-methoxy-1,4-naphthoquinoneMus musculus (house mouse)Potency5.011910
ethyl violetMus musculus (house mouse)Potency1.258910
sulfadoxineMus musculus (house mouse)Potency3.548110
mebeverine hydrochlorideMus musculus (house mouse)Potency6.309610
doxifluridineMus musculus (house mouse)Potency12.589310
nsc 3852Mus musculus (house mouse)Potency1.122010
piperacetazineMus musculus (house mouse)Potency10.000010
nitroxolineMus musculus (house mouse)Potency3.981110
cladribineMus musculus (house mouse)Potency0.316210
hyaluronoglucosaminidaseMus musculus (house mouse)Potency0.354810
u 0521Mus musculus (house mouse)Potency5.623410
beclomethasone dipropionateMus musculus (house mouse)Potency2.818410
vidarabineMus musculus (house mouse)Potency12.589310
2-hydroxy-7-nitrofluoreneMus musculus (house mouse)Potency7.943310
propionylpromazine hydrochlorideMus musculus (house mouse)Potency10.000010
nsc-145,668Mus musculus (house mouse)Potency0.398110
hydrocortisone-17-butyrateMus musculus (house mouse)Potency12.589310
tetraethylene glycol diacrylateMus musculus (house mouse)Potency1.258910
2,6-diaminopurineMus musculus (house mouse)Potency6.309610
cetyldimethylethylammonium bromideMus musculus (house mouse)Potency1.000010
N-(3-methyl-1,1-dioxo-1,4-thiazinan-4-yl)-1-(5-nitro-2-furanyl)methanimineMus musculus (house mouse)Potency12.589310
frentizoleMus musculus (house mouse)Potency7.943310
2-n-octyl-4-isothiazolin-3-oneMus musculus (house mouse)Potency11.220210
amoxicillinMus musculus (house mouse)Potency1.412510
oxcarbazepineMus musculus (house mouse)Potency12.589310
serentilMus musculus (house mouse)Potency10.000010
procymidoneMus musculus (house mouse)Potency3.548110
etoposideMus musculus (house mouse)Potency0.398110
k 308Mus musculus (house mouse)Potency10.000010
ribavirinMus musculus (house mouse)Potency7.079510
isovelleralMus musculus (house mouse)Potency2.238710
ciclopirox olamineMus musculus (house mouse)Potency1.000010
dinalineMus musculus (house mouse)Potency7.079510
butoconazole nitrateMus musculus (house mouse)Potency12.589310
triclabendazoleMus musculus (house mouse)Potency7.079510
lovastatinMus musculus (house mouse)Potency0.891310
chaetochrominMus musculus (house mouse)Potency5.623410
azelastine hydrochlorideMus musculus (house mouse)Potency11.220210
simvastatinMus musculus (house mouse)Potency3.162310
nefazodone hydrochlorideMus musculus (house mouse)Potency12.589310
mifepristoneMus musculus (house mouse)Potency8.912510
salmeterol xinafoateMus musculus (house mouse)Potency7.943310
imiquimodMus musculus (house mouse)Potency1.412510
duloxetine hydrochlorideMus musculus (house mouse)Potency10.000010
saquinavir monomethanesulfonateMus musculus (house mouse)Potency12.589310
paroxetine hydrochlorideMus musculus (house mouse)Potency7.079510
verapamil hydrochlorideMus musculus (house mouse)Potency3.548110
sertraline hydrochlorideMus musculus (house mouse)Potency10.000010
nelfinavir mesylateMus musculus (house mouse)Potency7.943310
nelfinavirMus musculus (house mouse)Potency7.079510
mevastatinMus musculus (house mouse)Potency1.258910
ro 5-3335Mus musculus (house mouse)Potency3.162310
neocuproineMus musculus (house mouse)Potency0.014110
dobutamine hydrochlorideMus musculus (house mouse)Potency7.943310
desipramine hydrochlorideMus musculus (house mouse)Potency7.079510
benzydamine hydrochlorideMus musculus (house mouse)Potency6.309610
prenylamine lactateMus musculus (house mouse)Potency12.589310
rutecarpineMus musculus (house mouse)Potency4.466810
thioridazine hydrochlorideMus musculus (house mouse)Potency11.220210
edoxudinMus musculus (house mouse)Potency2.511910
2-methoxyestradiolMus musculus (house mouse)Potency1.000010
17 beta-estradiol hemisuccinateMus musculus (house mouse)Potency14.125410
toxoflavinMus musculus (house mouse)Potency1.122010
n(4)-acetylsulfamerazineMus musculus (house mouse)Potency1.000010
dimidium bromideMus musculus (house mouse)Potency7.079510
2,6-dimethoxy-1,4-benzoquinoneMus musculus (house mouse)Potency1.122010
dyclonine hydrochlorideMus musculus (house mouse)Potency12.589310
meconinMus musculus (house mouse)Potency11.220210
prazosin hydrochlorideMus musculus (house mouse)Potency12.589310
econazole nitrateMus musculus (house mouse)Potency12.589310
sertralineMus musculus (house mouse)Potency10.000010
2,6-di-tert-butyl-4-nitrophenolMus musculus (house mouse)Potency7.943310
vinburnineMus musculus (house mouse)Potency3.162310
loxapine succinateMus musculus (house mouse)Potency12.589310
loperamide hydrochlorideMus musculus (house mouse)Potency6.309610
chlormidazoleMus musculus (house mouse)Potency5.011910
thiocolchicosideMus musculus (house mouse)Potency12.589310
thioxoloneMus musculus (house mouse)Potency7.943310
ubenimexMus musculus (house mouse)Potency16.481610
6-hydroxyflavoneMus musculus (house mouse)Potency10.000010
9-methoxyellipticineMus musculus (house mouse)Potency1.778310
3-aminophenoxazoneMus musculus (house mouse)Potency10.000010
2-phenyl-4,5-dichloro-3-pyridazinoneMus musculus (house mouse)Potency3.548110
tosyllysine chloromethyl ketoneMus musculus (house mouse)Potency11.668110
ergocornineMus musculus (house mouse)Potency5.623410
fangchinolineMus musculus (house mouse)Potency12.589310
tryptanthrineMus musculus (house mouse)Potency2.511910
n-benzylmaleimideMus musculus (house mouse)Potency7.943310
2-phenylisatogenMus musculus (house mouse)Potency12.589310
4'-methoxyflavoneMus musculus (house mouse)Potency12.589310
N-(4-ethoxyphenyl)-3-hydroxy-2-naphthalenecarboxamideMus musculus (house mouse)Potency3.981110
2-methyl-4-nitroquinoline 1-oxideMus musculus (house mouse)Potency0.316210
clarithromycinMus musculus (house mouse)Potency5.623410
imidaclopridMus musculus (house mouse)Potency1.122010
5,7-dimethoxyflavoneMus musculus (house mouse)Potency10.000010
carbetapentane citrateMus musculus (house mouse)Potency8.912510
phentolamine mesylateMus musculus (house mouse)Potency12.589310
pyridabenMus musculus (house mouse)Potency0.158510
adenosine 5'-methylenediphosphateMus musculus (house mouse)Potency5.011910
9,10-phenanthrenequinone monoximeMus musculus (house mouse)Potency5.623410
hexaphosphamideMus musculus (house mouse)Potency3.162310
oxoglaucineMus musculus (house mouse)Potency1.258910
6,6'-methylene bis(2,2,4-trimethyl-1,2-dihydroquinoline)Mus musculus (house mouse)Potency12.589310
zpckMus musculus (house mouse)Potency1.778310
diphyllinMus musculus (house mouse)Potency0.891310
gr 127935Mus musculus (house mouse)Potency14.689210
dihydrocapsaicinMus musculus (house mouse)Potency8.912510
imidocarbMus musculus (house mouse)Potency12.589310
bw 245cMus musculus (house mouse)Potency0.398110
gallopamil hydrochlorideMus musculus (house mouse)Potency4.466810
razadyneMus musculus (house mouse)Potency6.309610
tetradecanoylphorbol acetateMus musculus (house mouse)Potency0.092710
w 7Mus musculus (house mouse)Potency6.309610
purpactin aMus musculus (house mouse)Potency28.183810
dichloro-1,2-diaminocyclohexane platinum complexMus musculus (house mouse)Potency6.309610
idazoxan hydrochlorideMus musculus (house mouse)Potency7.079510
Austalide JMus musculus (house mouse)Potency5.011910
sch 45752Mus musculus (house mouse)Potency10.000010
oxypeucadaninMus musculus (house mouse)Potency0.354810
chloracizine hydrochlorideMus musculus (house mouse)Potency8.912510
ag 3-5Mus musculus (house mouse)Potency1.000010
enniatin bMus musculus (house mouse)Potency3.162310
barbatic acidMus musculus (house mouse)Potency0.794310
4-methoxy-1-vinylcarbolineMus musculus (house mouse)Potency1.122010
cirsimaritinMus musculus (house mouse)Potency7.079510
sb 205384Mus musculus (house mouse)Potency2.818410
benfluorex hydrochlorideMus musculus (house mouse)Potency3.981110
dermofixMus musculus (house mouse)Potency12.589310
brazilinMus musculus (house mouse)Potency22.387210
equilinMus musculus (house mouse)Potency12.589310
4'-hydroxyflavoneMus musculus (house mouse)Potency7.943310
acetoxycycloheximideMus musculus (house mouse)Potency0.223910
colchiceineMus musculus (house mouse)Potency8.912510
PorfiromycineMus musculus (house mouse)Potency5.623410
2-hydroxyestradiolMus musculus (house mouse)Potency1.122010
coronopilinMus musculus (house mouse)Potency5.011910
showdomycinMus musculus (house mouse)Potency22.387210
noscapineMus musculus (house mouse)Potency14.125410
dimethyl 2-(2-nitrobenzylidene)malonateMus musculus (house mouse)Potency2.238710
aromaticinMus musculus (house mouse)Potency12.589310
oxopurpureineMus musculus (house mouse)Potency1.000010
acetic acid (4-acetyloxy-6,7-dimethyl-5,8-dihydronaphthalen-1-yl) esterMus musculus (house mouse)Potency11.220210
4-[(1-naphthalenylamino)-oxomethyl]benzene-1,3-dicarboxylic acidMus musculus (house mouse)Potency5.011910
2-[[[4-(methylthio)anilino]-oxomethyl]amino]benzamideMus musculus (house mouse)Potency5.011910
4-chloro-1H-indazol-3-amineMus musculus (house mouse)Potency15.848910
nsc228155Mus musculus (house mouse)Potency2.818410
6-chloro-[1,2,4]triazolo[3,4-a]phthalazineMus musculus (house mouse)Potency10.000010
dicentrineMus musculus (house mouse)Potency10.000010
N-[2-(1-azepanyl)-1,3-benzothiazol-6-yl]carbamic acid ethyl esterMus musculus (house mouse)Potency1.995310
AmalorinMus musculus (house mouse)Potency7.943310
DubamineMus musculus (house mouse)Potency6.309610
4,5,7-trihydroxy-9,10-dioxo-2-anthracenecarboxylic acidMus musculus (house mouse)Potency11.220210
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneMus musculus (house mouse)Potency3.981110
2,2'-spirobi[3,6,7,8-tetrahydro-1H-cyclopenta[g]naphthalene]-5,5'-dioneMus musculus (house mouse)Potency3.162310
nu 6027Mus musculus (house mouse)Potency5.011910
nexavarMus musculus (house mouse)Potency28.183810
dichloro-1,2-diaminocyclohexane platinum complexMus musculus (house mouse)Potency6.309610
Destruxin BMus musculus (house mouse)Potency2.238710
tosylphenylalanyl chloromethyl ketoneMus musculus (house mouse)Potency5.011910
discretamineMus musculus (house mouse)Potency4.466810
quinidineMus musculus (house mouse)Potency1.258910
griseofulvinMus musculus (house mouse)Potency7.943310
saquinavirMus musculus (house mouse)Potency10.000010
mometasone furoateMus musculus (house mouse)Potency8.912510
mefloquine hydrochlorideMus musculus (house mouse)Potency7.079510
angustibalinMus musculus (house mouse)Potency0.354810
amantadine hydrochlorideMus musculus (house mouse)Potency7.943310
ononinMus musculus (house mouse)Potency10.000010
canadine, (r)-isomerMus musculus (house mouse)Potency11.220210
metrizamideMus musculus (house mouse)Potency5.623410
erythromycin ethylsuccinateMus musculus (house mouse)Potency7.943310
amcinonideMus musculus (house mouse)Potency2.818410
dihydroergocristine monomesylateMus musculus (house mouse)Potency5.623410
resveratrolMus musculus (house mouse)Potency13.529420
mycophenolic acidMus musculus (house mouse)Potency0.316210
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolMus musculus (house mouse)Potency7.943310
6-bromoindirubin-3'-oximeMus musculus (house mouse)Potency12.589310
afimoxifeneMus musculus (house mouse)Potency2.818410
visnadinMus musculus (house mouse)Potency12.589310
ketoconazoleMus musculus (house mouse)Potency12.589310
melphalanMus musculus (house mouse)Potency2.511910
6-bromoflavoneMus musculus (house mouse)Potency1.412510
(2S)-2-[[[4-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-1-oxo-3-phenylpropan-2-yl]amino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-3-phenylpropanoic acid tert-butyl esterMus musculus (house mouse)Potency28.183810
4-(2-oxazolo[4,5-b]pyridinyl)anilineMus musculus (house mouse)Potency0.354810
9,14-Dimethyl-5-methylidene-3,13-dioxatetracyclo[8.4.0.02,6.012,14]tetradec-9-ene-4,11-dioneMus musculus (house mouse)Potency31.622810
2-(8-Hydroxy-4a,8-dimethyldecahydro-2-naphthalenyl)acrylic acidMus musculus (house mouse)Potency14.125410
menadione sodium bisulfite, trihydrateMus musculus (house mouse)Potency7.943310
hei 713Mus musculus (house mouse)Potency28.183810
1,3-dichloro-7-methyl-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileMus musculus (house mouse)Potency11.220210
niflumic acidMus musculus (house mouse)Potency10.000010
chalconeMus musculus (house mouse)Potency7.943310
piplartineMus musculus (house mouse)Potency1.000010
7-methoxyisoflavoneMus musculus (house mouse)Potency7.943310
piperineMus musculus (house mouse)Potency10.000010
2'-hydroxychalconeMus musculus (house mouse)Potency12.589310
cardamoninMus musculus (house mouse)Potency10.000010
cgp 60474Mus musculus (house mouse)Potency0.002510
calmidazoliumMus musculus (house mouse)Potency12.589310
2-[5-(4-butoxyphenyl)-2-tetrazolyl]-N-(2-furanylmethyl)acetamideMus musculus (house mouse)Potency0.794310
N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-1-isoquinolinecarboxamideMus musculus (house mouse)Potency3.981110
3-methyl-4-(7-methyl-2-indolizinyl)-1,2,5-oxadiazoleMus musculus (house mouse)Potency8.912510
3-[[1,3-benzodioxol-5-ylmethyl-[(1-cyclopentyl-5-tetrazolyl)methyl]amino]methyl]-6-ethyl-1H-quinolin-2-oneMus musculus (house mouse)Potency11.220210
6-(4-hydroxy-3-methoxyphenyl)-4-methoxy-1,3-dimethyl-8-cyclohepta[c]furanoneMus musculus (house mouse)Potency7.943310
N-(1-adamantyl)-4-(1,3-benzodioxol-5-yl)-4-hydroxy-1-piperidinecarboxamideMus musculus (house mouse)Potency10.000010
6-chloro-2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-piperidinyl]-1H-benzimidazoleMus musculus (house mouse)Potency12.589310
3-chloro-4-[4-(4-fluorophenyl)sulfonyl-1-piperazinyl]-N,N-dimethylbenzenesulfonamideMus musculus (house mouse)Potency5.623410
3-[[(1-tert-butyl-5-tetrazolyl)methyl-(thiophen-2-ylmethyl)amino]methyl]-6-ethoxy-1H-quinolin-2-oneMus musculus (house mouse)Potency7.079510
4-[4-[(1-cyclopentyl-5-tetrazolyl)-pyridin-4-ylmethyl]-1-piperazinyl]phenolMus musculus (house mouse)Potency12.589310
benidipine hydrochlorideMus musculus (house mouse)Potency12.589310
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideMus musculus (house mouse)Potency12.589310
fludarabineMus musculus (house mouse)Potency8.912510
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideMus musculus (house mouse)Potency1.000010
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenolMus musculus (house mouse)Potency14.125410
2-[5-[(4-bromophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineMus musculus (house mouse)Potency8.912510
1-(3,4-dihydroxyphenyl)-2-[[5-(2-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency8.912510
dienestrolMus musculus (house mouse)Potency7.943310
mercaptopurineMus musculus (house mouse)Potency2.818410
methylthiouracilMus musculus (house mouse)Potency6.309610
3,3',4,5'-tetrahydroxystilbeneMus musculus (house mouse)Potency7.943310
(3,4-dimethylphenyl)-(4-phenyl-1-piperazinyl)methanoneMus musculus (house mouse)Potency7.943310
7-ethoxy-9-nitro-5H-benzo[b][1,4]benzoxazepin-6-oneMus musculus (house mouse)Potency1.995310
3-[[2-benzofuranyl(oxo)methyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency11.220210
4,6-dimethyl-N-phenyl-2-quinolinamineMus musculus (house mouse)Potency6.309610
6-methoxy-2-(4-methoxyphenyl)-1-benzopyran-4-oneMus musculus (house mouse)Potency1.412510
3-(4-methylbenzoyl)acrylic acidMus musculus (house mouse)Potency8.912510
N4-(3-chlorophenyl)-6-methyl-N2-(phenylmethyl)pyrimidine-2,4-diamineMus musculus (house mouse)Potency11.220210
stf 62247Mus musculus (house mouse)Potency7.943310
4-[2-(dimethylamino)ethylamino]-3-benzo[h]quinolinecarboxylic acid ethyl esterMus musculus (house mouse)Potency28.183810
1-(3,4-dichlorophenyl)-2-thioureaMus musculus (house mouse)Potency5.011910
4-(benzylsulfanyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency0.891310
N-tert-butyl-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineMus musculus (house mouse)Potency10.000010
1-(3,4-dihydroxyphenyl)-2-[(4,6-dimethyl-2-pyrimidinyl)thio]ethanoneMus musculus (house mouse)Potency6.309610
1-[4-(4-aminophenyl)-1-piperazinyl]ethanoneMus musculus (house mouse)Potency10.000010
krm iiiMus musculus (house mouse)Potency1.000010
4-(2-imidazo[1,2-a]pyridinylmethoxy)benzaldehydeMus musculus (house mouse)Potency31.622810
3-[[(5-bromo-3-pyridinyl)-oxomethyl]amino]propanoic acidMus musculus (house mouse)Potency2.818410
4-[2-(1-methyl-2-benzimidazolyl)ethyl]anilineMus musculus (house mouse)Potency8.912510
2-fluoro-N-phenacylbenzamideMus musculus (house mouse)Potency5.623410
N-[[(2-chloro-3-pyridinyl)amino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency8.912510
N-[3-chloro-4-(1-pyrrolidinyl)phenyl]-2-furancarboxamideMus musculus (house mouse)Potency8.912510
1-methyl-4-[(4-methylphenyl)thio]-3-nitro-2-quinolinoneMus musculus (house mouse)Potency1.584910
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazineMus musculus (house mouse)Potency3.162310
4-[[4-(2,5-dimethylphenyl)-1-piperazinyl]methyl]-2-methoxyphenolMus musculus (house mouse)Potency12.589310
N-[4-(2-methyl-4-thiazolyl)phenyl]benzamideMus musculus (house mouse)Potency2.238710
1-(4-methoxyphenyl)-3-(6-methyl-2-pyridinyl)ureaMus musculus (house mouse)Potency3.162310
2-bromo-N-(3-methoxyphenyl)benzamideMus musculus (house mouse)Potency10.000010
N-(cyclopentylideneamino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamideMus musculus (house mouse)Potency8.912510
N-(4-benzamido-2-chlorophenyl)-2-furancarboxamideMus musculus (house mouse)Potency5.011910
N-[(4-fluoroanilino)-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideMus musculus (house mouse)Potency7.943310
4,4'-sulfonylbis[2-(prop-2-en-1-yl)phenol]Mus musculus (house mouse)Potency12.589310
N-(4-fluoro-3-nitrophenyl)-3-methyl-2-thiophenecarboxamideMus musculus (house mouse)Potency10.000010
8-[(2-methyl-5-nitro-1,2,4-triazol-3-yl)thio]quinolineMus musculus (house mouse)Potency12.589310
N-(6-ethoxy-1,3-benzothiazol-2-yl)butanamideMus musculus (house mouse)Potency3.981110
N-(2-chlorophenyl)-2-[[cyclopropyl(oxo)methyl]amino]-4-methyl-5-thiazolecarboxamideMus musculus (house mouse)Potency12.589310
N-[[(6-methoxy-1,3-benzothiazol-2-yl)amino]-sulfanylidenemethyl]-2-furancarboxamideMus musculus (house mouse)Potency5.011910
2-[[anilino(oxo)methyl]amino]-N-(2-furanylmethyl)benzamideMus musculus (house mouse)Potency10.000010
N-(5-acetyl-4-methyl-2-thiazolyl)-5-bromo-2-furancarboxamideMus musculus (house mouse)Potency1.778310
2-(2-methylphenoxy)-N-[2-(methylthio)phenyl]acetamideMus musculus (house mouse)Potency1.122010
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneMus musculus (house mouse)Potency0.891310
3-(4-ethoxyphenyl)-4-(phenylmethyl)-1H-1,2,4-triazole-5-thioneMus musculus (house mouse)Potency17.782810
virosecurinineMus musculus (house mouse)Potency10.000010
7-bromo-1,2,3,9-tetrahydropyrrolo[2,1-b]quinazolineMus musculus (house mouse)Potency1.258910
oxypeucadanin, (r)-(+)-isomerMus musculus (house mouse)Potency8.912510
thiothixeneMus musculus (house mouse)Potency11.220210
curcuminMus musculus (house mouse)Potency3.981110
N-(1,3-benzodioxol-5-yl)-4-(2-furanylmethyl)-1-piperazinecarbothioamideMus musculus (house mouse)Potency4.466810
2-(4-methylanilino)-4-pyrido[3,2-e][1,3]thiazinoneMus musculus (house mouse)Potency2.818410
5-[(5-methoxycarbonyl-2-methyl-3-furanyl)methoxy]-2-methyl-3-benzofurancarboxylic acid methyl esterMus musculus (house mouse)Potency12.589310
umi-77Mus musculus (house mouse)Potency10.000010
2-[[3-cyano-4-(2-methoxyphenyl)-6-phenyl-2-pyridinyl]thio]acetic acidMus musculus (house mouse)Potency3.162310
1-methoxy-N-[4-(pyridin-4-ylmethyl)phenyl]-2-naphthalenecarboxamideMus musculus (house mouse)Potency8.912510
N-[2-(3-pyridinyl)-3H-benzimidazol-5-yl]-2-furancarboxamideMus musculus (house mouse)Potency7.943310
N-(4-cyano-2-methyl-3-pyrazolyl)-5-(4-methylphenyl)-3-isoxazolecarboxamideMus musculus (house mouse)Potency1.258910
N-[2,2-dichloro-1-(4-chlorophenyl)sulfonylethenyl]benzamideMus musculus (house mouse)Potency8.912510
LSM-16285Mus musculus (house mouse)Potency6.309610
2-[N-(benzenesulfonyl)-4-ethoxyanilino]-N-(2-methoxyphenyl)acetamideMus musculus (house mouse)Potency0.501210
1-(2,5-dimethoxyphenyl)sulfonyl-4-(phenylmethyl)piperazineMus musculus (house mouse)Potency31.622810
N2-tert-butyl-N6-ethyl-N4-propan-2-yl-1,3,5-triazine-2,4,6-triamineMus musculus (house mouse)Potency8.912510
1-[2,5-dimethyl-1-(4-methylphenyl)-3-pyrrolyl]-2-([1,2,4]triazolo[4,3-a]pyridin-3-ylthio)ethanoneMus musculus (house mouse)Potency7.943310
4-(4-anilinoanilino)-2-quinazolinecarboxylic acid ethyl esterMus musculus (house mouse)Potency12.589310
3-(2-phenyl-5-tetrazolyl)pyridineMus musculus (house mouse)Potency7.943310
(4-phenyl-1-piperazinyl)-(9H-xanthen-9-yl)methanoneMus musculus (house mouse)Potency1.258910
N'-[2-(4-bromo-2-methylphenoxy)-1-oxoethyl]-2-pyrazinecarbohydrazideMus musculus (house mouse)Potency3.981110
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamideMus musculus (house mouse)Potency6.309610
6-(2,3-dihydroindol-1-ylmethyl)-3-phenylthiazolo[2,3-c][1,2,4]triazoleMus musculus (house mouse)Potency3.981110
3-[[[3-(1-azepanylsulfonyl)-4-chlorophenyl]-oxomethyl]amino]benzoic acidMus musculus (house mouse)Potency6.309610
2-[[5-(4-nitrophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(2-pyridinyl)acetamideMus musculus (house mouse)Potency1.258910
[2-(4-propylphenyl)-4-quinolinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency7.079510
2-(3-bromophenyl)-6-methyl-N-(1,2,4-triazol-4-yl)-4-quinolinecarboxamideMus musculus (house mouse)Potency8.912510
[4-(2,3-dimethylphenyl)-1-piperazinyl]-(3,4,5-trimethoxyphenyl)methanoneMus musculus (house mouse)Potency0.891310
N-(2,4-dimethoxyphenyl)-2-(1-pyrrolidinyl)-4-quinazolinamineMus musculus (house mouse)Potency10.000010
N-(2-furanylmethyl)-2-[[[2-[(4-methylphenyl)sulfonyl-(phenylmethyl)amino]phenyl]-oxomethyl]amino]benzamideMus musculus (house mouse)Potency14.125410
1-(3,4-dihydroxyphenyl)-2-[[5-(4-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency4.466810
2-[[5-(3-chlorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanoneMus musculus (house mouse)Potency5.623410
1-(3,4-dihydroxyphenyl)-2-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency5.011910
1-(3,4-dihydroxyphenyl)-2-[[5-(4-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency3.981110
1-(3,4-dihydroxyphenyl)-2-[[5-(3-methoxyphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]ethanoneMus musculus (house mouse)Potency6.309610
(4-chlorophenyl)-(5-hydroxy-2-methyl-4,6-dinitro-3-benzofuranyl)methanoneMus musculus (house mouse)Potency3.981110
2-[1-(4-tert-butylphenyl)sulfonyl-4-piperidinyl]-6-chloro-1H-benzimidazoleMus musculus (house mouse)Potency22.387210
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneMus musculus (house mouse)Potency12.589310
1-(4-fluorophenyl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneMus musculus (house mouse)Potency12.589310
3-amino-8-methyl-N-[4-(4-morpholinyl)phenyl]-2-thieno[2,3-b]quinolinecarboxamideMus musculus (house mouse)Potency10.000010
1-[1-[(2-chloro-6-fluorophenyl)methyl]-2-oxo-3-pyridinyl]-3-(phenylmethyl)ureaMus musculus (house mouse)Potency28.183810
N-[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]-2-methoxyacetamideMus musculus (house mouse)Potency3.981110
4-(4-chlorophenyl)sulfinyl-6-(methoxymethyl)-2-methylpyrimidineMus musculus (house mouse)Potency5.011910
N,N-dimethylcarbamothioic acid O-[4-[2-[(4-chlorophenyl)thio]-1-oxoethyl]-2,6-dimethylphenyl] esterMus musculus (house mouse)Potency6.309610
3,4-dichloro-N-(4-chloro-3-methyl-5-isoxazolyl)benzamideMus musculus (house mouse)Potency31.622810
2-amino-6-ethyl-3-(3-isoxazolyl)-7-methoxy-1-benzopyran-4-oneMus musculus (house mouse)Potency10.000010
hexyl cinnamic aldehydeMus musculus (house mouse)Potency11.220210
2-(4-chlorophenyl)-5-(prop-2-enylamino)-4-oxazolecarbonitrileMus musculus (house mouse)Potency7.943310
chlorogenic acidMus musculus (house mouse)Potency1.122010
2,2-diphenylacetic acid (2,6-dimethylphenyl) esterMus musculus (house mouse)Potency0.398110
3,4-dimethoxy-N-[[[oxo(2-pyrazinyl)methyl]hydrazo]-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency2.511910
1-[1-naphthalenyl(oxo)methyl]-3-indolecarboxylic acid methyl esterMus musculus (house mouse)Potency3.981110
2-[[5-[(1,3-benzothiazol-2-ylthio)methyl]-4-ethyl-1,2,4-triazol-3-yl]thio]-1-(3,4-dihydroxyphenyl)ethanoneMus musculus (house mouse)Potency3.981110
N-(1H-benzimidazol-2-yl)-3-[methyl-(4-methylphenyl)sulfamoyl]benzamideMus musculus (house mouse)Potency19.952610
N-(3,5-dimethoxyphenyl)-2-(2,2-dimethyl-5-oxo-4-phenyl-1-imidazolyl)acetamideMus musculus (house mouse)Potency3.548110
3-cyclohexyl-N-(1,3-dimethyl-2,6-dioxo-4-pyrimidinyl)propanamideMus musculus (house mouse)Potency15.848910
N-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-[methyl(phenyl)sulfamoyl]benzamideMus musculus (house mouse)Potency10.000010
1-[2-(2,5-dimethyl-1H-indol-3-yl)ethyl]-3-methyl-1-(thiophen-2-ylmethyl)thioureaMus musculus (house mouse)Potency19.952610
2-[2-furanyl(oxo)methyl]imino-5-oxo-1-propan-2-yl-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency4.466810
N-[(2S)-1-(1H-benzimidazol-2-ylamino)-3-methyl-1-oxobutan-2-yl]-3-methylbenzamideMus musculus (house mouse)Potency2.818410
2-(3-chlorophenyl)-5-(prop-2-enylamino)-4-oxazolecarbonitrileMus musculus (house mouse)Potency7.079510
4-methyl-N-(2-phenylphenyl)-3-(phenylsulfamoyl)benzamideMus musculus (house mouse)Potency12.589310
1-[2-[3-(1-methylethenyl)phenyl]propan-2-yl]-3-(4-methyl-2-pyridinyl)ureaMus musculus (house mouse)Potency3.548110
2-(1,3-benzothiazol-2-yl)-5-methyl-3-pyrazolamineMus musculus (house mouse)Potency12.589310
N-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethenyl]-4-morpholinecarboxamideMus musculus (house mouse)Potency5.011910
3-[2-(4-fluorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineMus musculus (house mouse)Potency7.079510
N-[[2-(diethylamino)ethylamino]-sulfanylidenemethyl]-3-(4-methoxyphenyl)-1-phenyl-4-pyrazolecarboxamideMus musculus (house mouse)Potency14.125410
3-(4-methoxyphenyl)-N-[[[oxo(pyridin-4-yl)methyl]hydrazo]-sulfanylidenemethyl]-1-phenyl-4-pyrazolecarboxamideMus musculus (house mouse)Potency8.912510
2-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-1,2-benzothiazol-3-oneMus musculus (house mouse)Potency12.589310
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-methoxy-5-methylphenyl)benzamideMus musculus (house mouse)Potency12.589310
2-chloro-N-[4-(N-propan-2-ylanilino)phenyl]acetamideMus musculus (house mouse)Potency11.220210
1-[[4-[[[(4-chloro-3-fluoroanilino)-sulfanylidenemethyl]amino]methyl]phenyl]methyl]-3-(4-chloro-3-fluorophenyl)thioureaMus musculus (house mouse)Potency6.309610
N-(3-fluorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineMus musculus (house mouse)Potency5.623410
1-(2,6-diethylphenyl)-3-[2-(3,4-dihydroxyphenyl)ethyl]thioureaMus musculus (house mouse)Potency12.589310
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-quinolinecarboxamideMus musculus (house mouse)Potency8.912510
2-(2,6-dichlorophenyl)acetic acid [2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] esterMus musculus (house mouse)Potency2.511910
2-chloro-N-[4-[(3,4-dimethylphenyl)thio]phenyl]acetamideMus musculus (house mouse)Potency12.589310
[4-(4-hydroxyphenyl)-1-piperazinyl]-[2-methoxy-4-(methylthio)phenyl]methanoneMus musculus (house mouse)Potency4.466810
4-[[5-(1,3-benzothiazol-2-yl)-2-thiophenyl]-oxomethyl]-1-piperazinecarboxaldehydeMus musculus (house mouse)Potency8.912510
5-bromo-N-(4-methyl-2-thiazolyl)-3-pyridinecarboxamideMus musculus (house mouse)Potency11.220210
3-(difluoromethoxy)-N-(4,5-dihydrothiazol-2-yl)benzamideMus musculus (house mouse)Potency28.183810
thioguanine anhydrousMus musculus (house mouse)Potency0.158510
diaminomaleonitrile, (z)-isomerMus musculus (house mouse)Potency5.623410
mercaptopurineMus musculus (house mouse)Potency1.122010
benzoylarginine nitroanilideMus musculus (house mouse)Potency2.238710
6-thioguanosineMus musculus (house mouse)Potency0.007110
2-(4-methylphenyl)-1,9b-dihydropyrazolo[1,5-b]isoindol-5-oneMus musculus (house mouse)Potency10.000010
capsazepineMus musculus (house mouse)Potency0.891310
N'-benzoyl-5-(3,5-dichlorophenoxy)-2-furancarbohydrazideMus musculus (house mouse)Potency8.912510
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineMus musculus (house mouse)Potency4.466810
1-(4-hydroxyphenyl)-3-(3-methoxyphenyl)thioureaMus musculus (house mouse)Potency3.548110
5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamideMus musculus (house mouse)Potency12.589310
5-[[[5-(2-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esterMus musculus (house mouse)Potency7.943310
N'-(3-chloro-4-methylphenyl)-5-isoxazolecarbohydrazideMus musculus (house mouse)Potency12.589310
2-[4-(trifluoromethoxy)phenyl]imidazo[1,2-a]pyrimidineMus musculus (house mouse)Potency5.011910
LSM-28486Mus musculus (house mouse)Potency1.584910
N-(1H-indol-5-yl)-2-thiophenecarboxamideMus musculus (house mouse)Potency7.079510
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileMus musculus (house mouse)Potency8.912510
2-[(4-chlorophenyl)methoxy]-6-methoxybenzonitrileMus musculus (house mouse)Potency8.912510
N,N'-diphenylcarbamimidothioic acid [1-(3-methylphenyl)-2,5-dioxo-3-pyrrolidinyl] esterMus musculus (house mouse)Potency7.943310
(4-chlorophenyl)-[6,7-dichloro-4-[(dimethylamino)methyl]-5-hydroxy-2-methyl-3-benzofuranyl]methanoneMus musculus (house mouse)Potency11.220210
1-(9-anthracenylmethyl)-3-piperidinolMus musculus (house mouse)Potency10.000010
1-hexadecyl-3-methylimidazolium bromideMus musculus (house mouse)Potency1.584910
4-ethyl-2-methoxy-3-phenyl-3,3a,9,9a-tetrahydropyrrolo[2,3-b]quinoxalineMus musculus (house mouse)Potency12.589310
N-[(2-hydroxy-1-naphthalenyl)-(4-methoxyphenyl)methyl]-2-methylpropanamideMus musculus (house mouse)Potency7.943310
N-[(5-chloro-8-hydroxy-7-quinolinyl)-(4-methoxyphenyl)methyl]acetamideMus musculus (house mouse)Potency6.309610
6,3',4'-TrimethoxyflavanoneMus musculus (house mouse)Potency12.589310
k 858Mus musculus (house mouse)Potency2.511910
1-[(4-tert-butylphenyl)methyl]-4-(4-nitrophenyl)imidazoleMus musculus (house mouse)Potency28.183810
6-(2-chlorophenyl)-3-methyl-2-[4-morpholinyl(oxo)methyl]-1,5,6,7-tetrahydroindol-4-oneMus musculus (house mouse)Potency2.511910
N1,N4-bis(1-phenylethyl)cyclohexane-1,4-dicarboxamideMus musculus (house mouse)Potency8.912510
N-[4-[(3-acetylphenyl)sulfamoyl]phenyl]-1-piperidinecarboxamideMus musculus (house mouse)Potency12.589310
2-[[2-(4-ethyl-4-methyl-2,5-dioxo-1-imidazolidinyl)-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideMus musculus (house mouse)Potency14.125410
2-[2-[2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolyl]-2-oxoethyl]isoindole-1,3-dioneMus musculus (house mouse)Potency4.466810
bis(1-ethenyl-2-imidazolyl)-(9-ethyl-3-carbazolyl)-sulfanylidenephosphoraneMus musculus (house mouse)Potency10.000010
zeranolMus musculus (house mouse)Potency8.912510
nsc 336628Mus musculus (house mouse)Potency2.511910
schizandrinMus musculus (house mouse)Potency3.981110
thiophanateMus musculus (house mouse)Potency12.589310
2-chloro-n(6)-(3-iodobenzyl)adenosine-5'-n-methyluronamideMus musculus (house mouse)Potency12.589310
asterric acidMus musculus (house mouse)Potency0.891310
trimethoprimMus musculus (house mouse)Potency7.943310
N-methyl-5-nitro-N-(phenylmethyl)-2-furancarboxamideMus musculus (house mouse)Potency10.000010
2-(2,3,3-trichloro-1-nitroprop-2-enylidene)-1,3-dihydrobenzimidazoleMus musculus (house mouse)Potency6.309610
N-(2,4,6-trimethylphenyl)-3-bicyclo[2.2.1]heptanecarboxamideMus musculus (house mouse)Potency7.943310
4-[4-[2-hydroxy-3-(4-morpholinyl)propoxy]phenyl]benzonitrileMus musculus (house mouse)Potency12.589310
1-[4-(6-bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]ethanoneMus musculus (house mouse)Potency1.258910
1-[3-(benzenesulfonyl)-2-(1-piperidinyl)propyl]piperidineMus musculus (house mouse)Potency8.912510
5-hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazole-1-carboxylic acid ethyl esterMus musculus (house mouse)Potency6.309610
yl-109Mus musculus (house mouse)Potency4.466810
9-(2-ethoxy-3-methoxyphenyl)-3,6,8,9-tetrahydro-2H-[1,4]dioxino[2,3-g]quinolin-7-oneMus musculus (house mouse)Potency11.220210
N-[2-(tert-butylamino)-2-oxo-1-pyridin-4-ylethyl]-N-(2-furanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideMus musculus (house mouse)Potency12.589310
[4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-(2-furanyl)methanoneMus musculus (house mouse)Potency2.818410
1-cyclopentyl-1-[2-(5,6-dimethyl-1H-benzimidazol-2-yl)ethyl]-3-(2-oxolanylmethyl)thioureaMus musculus (house mouse)Potency8.912510
1-[3-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]-1-butanoneMus musculus (house mouse)Potency11.220210
N-[2-(3-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-N',N'-dimethylpropane-1,3-diamineMus musculus (house mouse)Potency5.011910
N-(1,3-benzodioxol-5-yl)-3-methyl-6-phenyl-2-imidazo[2,1-b]thiazolecarboxamideMus musculus (house mouse)Potency1.584910
2-(2-methoxyphenyl)-1-oxo-N-[2-oxo-2-[4-(2-pyridinyl)-1-piperazinyl]ethyl]-4-isoquinolinecarboxamideMus musculus (house mouse)Potency4.466810
2-amino-4-[5-methyl-2-(methylthio)-3-thiophenyl]-5-oxo-1-(3-pyridinyl)-4,6,7,8-tetrahydroquinoline-3-carbonitrileMus musculus (house mouse)Potency0.446710
6-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-5-thieno[2,3-b]pyrrolecarboxylic acid methyl esterMus musculus (house mouse)Potency4.466810
N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-oxo-1-[(phenylmethyl)amino]propan-2-yl]cyclopropyl]-phenylmethyl]carbamic acid (phenylmethyl) esterMus musculus (house mouse)Potency11.220210
5-methyl-N-[(S)-[(1S,2R)-1-methyl-2-[(2R)-1-(2-naphthalenylamino)-1-oxopropan-2-yl]cyclopropyl]-phenylmethyl]-3-isoxazolecarboxamideMus musculus (house mouse)Potency10.000010
1-(3-ethoxypropyl)-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency1.122010
2-phenoxy-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]acetamideMus musculus (house mouse)Potency14.125410
2-[[2-[(4,5-dimethoxy-2-nitrophenyl)-oxomethoxy]-1-oxoethyl]amino]-4-(2-methylpropyl)-3-thiophenecarboxylic acid ethyl esterMus musculus (house mouse)Potency0.316210
4-amino-2-nitrophenolMus musculus (house mouse)Potency4.466810
uc-112Mus musculus (house mouse)Potency4.466810
1-butyl-2-[2-furanyl(oxo)methyl]imino-10-methyl-5-oxo-3-dipyrido[3,4-c-1',2'-f]pyrimidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency7.943310
1-(3,4-dichlorophenyl)-3-[1-(4-morpholinyl)-1-phenylpropan-2-yl]ureaMus musculus (house mouse)Potency5.011910
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinolMus musculus (house mouse)Potency11.220210
4-(3,4-dihydro-2H-quinolin-1-ylsulfonyl)-N-(5-ethyl-1,3,4-oxadiazol-2-yl)benzamideMus musculus (house mouse)Potency3.981110
2-[[1-(phenylmethyl)-3-indolyl]thio]-N-(2-thiazolyl)acetamideMus musculus (house mouse)Potency7.079510
1,3-dimethyl-8-[[methyl-(phenylmethyl)amino]methyl]-7-(2-methylpropyl)purine-2,6-dioneMus musculus (house mouse)Potency10.000010
[1-[2-(2-methylphenoxy)ethyl]-3-indolyl]-(4-methyl-1-piperazinyl)methanethioneMus musculus (house mouse)Potency4.466810
sb 242084Mus musculus (house mouse)Potency29.308910
2-[(1-methyl-3-indolyl)thio]-N-(2-thiazolyl)acetamideMus musculus (house mouse)Potency2.238710
ML162Mus musculus (house mouse)Potency3.981110
2-(4-ethoxyphenyl)-N-[3-(1-imidazolyl)propyl]-4-quinolinecarboxamideMus musculus (house mouse)Potency12.589310
N-(4-bromophenyl)-5-methyl-4-nitro-1H-pyrazol-3-amineMus musculus (house mouse)Potency10.000010
6-(5,6-Dihydroxy-4-oxo-2-phenylchromen-7-yl)oxy-3,4,5-trihydroxyoxane-2-carboxylic acidMus musculus (house mouse)Potency5.011910
2-[[1-(4-chlorophenyl)-4-pyrazolo[3,4-d]pyrimidinyl]amino]-1-butanolMus musculus (house mouse)Potency12.589310
arabino-4-thiouridineMus musculus (house mouse)Potency1.995310
N-(1,3-benzothiazol-2-yl)-2-ethylsulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxamideMus musculus (house mouse)Potency28.183810
3-oxo-4H-1,4-benzothiazine-6-carboxylic acid [2-[1-(1-methoxypropan-2-yl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterMus musculus (house mouse)Potency3.162310
4-[(2-chloro-6-fluorophenyl)-oxomethyl]-7-methyl-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-oneMus musculus (house mouse)Potency3.548110
[4-[(2-chlorophenyl)methylsulfonyl]-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency7.943310
[4-(2,3-dimethylphenyl)-1-piperazinyl]-[5-[(4-methoxyphenyl)sulfonylmethyl]-2-furanyl]methanoneMus musculus (house mouse)Potency22.387210
[2-(3,4-dimethylphenyl)-4-quinolinyl]-(1-piperidinyl)methanoneMus musculus (house mouse)Potency4.466810
N-[1-(benzenesulfonyl)-2,2-dichloroethenyl]-4-methylbenzamideMus musculus (house mouse)Potency10.000010
sc-19220Mus musculus (house mouse)Potency12.589310
N-(6-acetyl-3-cyano-5,7-dihydro-4H-thieno[2,3-c]pyridin-2-yl)-3,4,5-trimethoxybenzamideMus musculus (house mouse)Potency22.387210
4-[(4-chlorophenyl)methylamino]-3-nitro-1-benzopyran-2-oneMus musculus (house mouse)Potency10.000010
2-chloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency5.011910
N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-4-propan-2-yloxybenzamideMus musculus (house mouse)Potency28.183810
4-bromo-N-[(2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl)-sulfanylidenemethyl]benzamideMus musculus (house mouse)Potency8.912510
2,6-diphenyl-7-pyrazolo[1,5-a]pyrimidinamineMus musculus (house mouse)Potency1.995310
mucronulatolMus musculus (house mouse)Potency28.183810
2,4-dichloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency28.183810
2-[[(3,4-dimethoxyphenyl)-oxomethyl]amino]acetic acid [2-[5-(4-chlorophenyl)-3-(2-furanyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] esterMus musculus (house mouse)Potency28.183810
[4-(4-chlorophenyl)-4,5-dihydro-1H-pyrazol-3-yl]-(2-oxiranyl)methanoneMus musculus (house mouse)Potency10.000010
5-acetyloxy-6-bromo-2-[[(6-but-3-enyl-3-cyano-2-pyridinyl)thio]methyl]-1-methyl-3-indolecarboxylic acid ethyl esterMus musculus (house mouse)Potency12.589310
2-(1,3-dimethyl-2,6-dioxo-7-purinyl)-N-[3-[(4-methoxyphenyl)sulfamoyl]-4-methylphenyl]acetamideMus musculus (house mouse)Potency28.183810
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterMus musculus (house mouse)Potency5.623410
[[2-[(4,5-dimethyl-2-thiazolyl)amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esterMus musculus (house mouse)Potency8.912510
4-[4-(4-acetylphenyl)-1-piperazinyl]-N-[3-(dimethylamino)propyl]-3-nitrobenzenesulfonamideMus musculus (house mouse)Potency11.220210
3'-[2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl]spiro[6,7-dihydro-5H-1-benzothiophene-4,5'-imidazolidine]-2',4'-dioneMus musculus (house mouse)Potency11.220210
5'-bromo-2'-spiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3'-1H-indole]oneMus musculus (house mouse)Potency8.912510
N-(3-chloro-4-fluorophenyl)-2-[5-(dimethylsulfamoyl)-2-(ethylamino)anilino]acetamideMus musculus (house mouse)Potency14.125410
N-(4-Nitro-1,2,5-oxadiazol-3-yl)-2-pyridin-2-ylsulfanylacetamideMus musculus (house mouse)Potency0.794310
1-(7-methyloctyl)-3-[4-(4-morpholinylsulfonyl)phenyl]thioureaMus musculus (house mouse)Potency22.387210
1-(2-furanylmethyl)-3-(3-methoxyphenyl)-1-[2-(2-methyl-1H-indol-3-yl)ethyl]thioureaMus musculus (house mouse)Potency31.622810
N-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]-4-(1-pyrrolidinylsulfonyl)benzamideMus musculus (house mouse)Potency28.183810
2,5-dichloro-N-[5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideMus musculus (house mouse)Potency10.000010
2,6-difluoro-N-[2-[3-[(2-fluorophenyl)methylthio]-1-indolyl]ethyl]benzamideMus musculus (house mouse)Potency12.589310
6-(4-methoxyphenyl)-N,3-dimethyl-2-imidazo[2,1-b]thiazolecarboxamideMus musculus (house mouse)Potency5.011910
sib 1757Mus musculus (house mouse)Potency11.220210
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2-oxo-1-benzopyran-3-carboxamideMus musculus (house mouse)Potency1.122010
biochanin aMus musculus (house mouse)Potency2.238710
formononetinMus musculus (house mouse)Potency5.011910
acacetinMus musculus (house mouse)Potency10.000010
luteolinMus musculus (house mouse)Potency7.943310
luteolin-7-glucosideMus musculus (house mouse)Potency2.818410
chrysoeriolMus musculus (house mouse)Potency11.220210
quercetin 3-o-methyl etherMus musculus (house mouse)Potency12.589310
3-methylkaempferolMus musculus (house mouse)Potency11.220210
genisteinMus musculus (house mouse)Potency11.220210
clothiapineMus musculus (house mouse)Potency5.011910
fucoxanthinMus musculus (house mouse)Potency22.387210
sulfuretinMus musculus (house mouse)Potency10.000010
esculetinMus musculus (house mouse)Potency5.011910
baicaleinMus musculus (house mouse)Potency10.000010
bellidifolinMus musculus (house mouse)Potency11.220210
hispidulinMus musculus (house mouse)Potency28.183810
santinMus musculus (house mouse)Potency28.183810
7-hydroxy-6,4'-dimethoxyisoflavoneMus musculus (house mouse)Potency3.548110
coumestrolMus musculus (house mouse)Potency10.000010
daidzeinMus musculus (house mouse)Potency5.623410
trans-2,3',4,5'-tetrahydroxystilbeneMus musculus (house mouse)Potency11.220210
caffeic acid phenethyl esterMus musculus (house mouse)Potency0.891310
savininMus musculus (house mouse)Potency12.589310
7-hydroxyflavoneMus musculus (house mouse)Potency11.220210
n-oleoyldopamineMus musculus (house mouse)Potency3.162310
tranilastMus musculus (house mouse)Potency7.079510
4-hydroxyestradiolMus musculus (house mouse)Potency6.309610
ketotifen fumarateMus musculus (house mouse)Potency6.990610
hydrocortisone valerateMus musculus (house mouse)Potency1.122010
bicyclo-PGE2Mus musculus (house mouse)Potency8.912510
cyclosporineMus musculus (house mouse)Potency2.511910
genistinMus musculus (house mouse)Potency4.466810
brefeldin aMus musculus (house mouse)Potency0.538910
fenretinideMus musculus (house mouse)Potency7.943310
su 9516Mus musculus (house mouse)Potency4.466810
N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamideMus musculus (house mouse)Potency3.981110
3-(4-chlorophenyl)-N-cyclopropyl-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideMus musculus (house mouse)Potency11.220210
3-(4-chlorophenyl)-1-methyl-N-[(5-methyl-2-furanyl)methyl]-5-thieno[2,3-c]pyrazolecarboxamideMus musculus (house mouse)Potency25.118910
4-[5-(4-methoxyphenyl)-3-isoxazolyl]-N-(2-pyridinylmethyl)butanamideMus musculus (house mouse)Potency6.309610
3-[[4-[6-(4-morpholinyl)-3-pyridazinyl]-1-piperazinyl]-oxomethyl]-1-benzopyran-2-oneMus musculus (house mouse)Potency28.183810
4-[3-(4-fluorophenyl)-2-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency28.183810
1-[[2-(3-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-piperidinecarboxamideMus musculus (house mouse)Potency12.589310
5-chloro-2-methoxy-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-N-propan-2-ylbenzamideMus musculus (house mouse)Potency12.589310
N-[3-[4-(2,5-dimethylphenyl)-1-piperazinyl]propyl]-2-(6-methyl-3-oxo-4H-1,4-benzoxazin-2-yl)acetamideMus musculus (house mouse)Potency19.952610
N-(6-acetyl-1,3-benzodioxol-5-yl)-5-methyl-2-phenyl-3-pyrazolecarboxamideMus musculus (house mouse)Potency3.162310
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-(3-methoxyphenyl)butanamideMus musculus (house mouse)Potency7.943310
1,5-dimethyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-2-pyrrolo[3,2-c]quinolinecarboxamideMus musculus (house mouse)Potency11.220210
N-[4-[(4-methyl-1-piperidinyl)methyl]phenyl]-1-[5-(1-pyrrolyl)-1,3,4-thiadiazol-2-yl]-4-piperidinecarboxamideMus musculus (house mouse)Potency12.589310
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[[5-methyl-2-(4-methylphenyl)-4-oxazolyl]methylsulfonyl]ethanoneMus musculus (house mouse)Potency11.220210
4-[3-oxo-1-(3,4,5-trimethoxyanilino)-1H-isoindol-2-yl]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency12.589310
3-(4-chlorophenyl)-N-[2-(diethylamino)ethyl]-1-methyl-5-thieno[2,3-c]pyrazolecarboxamideMus musculus (house mouse)Potency12.589310
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[[4-(4-fluorophenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideMus musculus (house mouse)Potency2.511910
N-[1-[4-(2-methoxyphenyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]benzenesulfonamideMus musculus (house mouse)Potency12.589310
4-amino-5-chloro-N-[(3R,4S)-1-[3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamideMus musculus (house mouse)Potency6.309610
cytochalasin bMus musculus (house mouse)Potency1.000010
su 6656Mus musculus (house mouse)Potency1.000010
5,7-dihydroxy-4',6-dimethoxyflavoneMus musculus (house mouse)Potency10.000010
thunberginol aMus musculus (house mouse)Potency2.818410
erbstatinMus musculus (house mouse)Potency3.162310
ag 538Mus musculus (house mouse)Potency12.365120
tyrphostin ag 555Mus musculus (house mouse)Potency3.548110
tyrphostin ag-494Mus musculus (house mouse)Potency2.818410
tyrphostin b44Mus musculus (house mouse)Potency3.981110
ag-490Mus musculus (house mouse)Potency3.548110
ag 183Mus musculus (house mouse)Potency12.589310
semaxinibMus musculus (house mouse)Potency3.162310
nifuroxazideMus musculus (house mouse)Potency7.079510
molsidomineMus musculus (house mouse)Potency7.943310
7,8-dihydroxy-4-methylcoumarinMus musculus (house mouse)Potency7.943310
flavokawain bMus musculus (house mouse)Potency8.912510
1-(4-methylpiperazin-1-yl)-3-(5-nitrofuran-2-yl)prop-2-en-1-oneMus musculus (house mouse)Potency2.818410
4-(2-hydroxyphenyl)but-3-en-2-oneMus musculus (house mouse)Potency5.011910
styrylquinolineMus musculus (house mouse)Potency5.623410
Isoliquiritigenin 4,4'-dimethyl etherMus musculus (house mouse)Potency14.125410
trimebutine maleate saltMus musculus (house mouse)Potency6.309610
calycanthineMus musculus (house mouse)Potency4.466810
nitrofurazoneMus musculus (house mouse)Potency11.220210
aurantiamineMus musculus (house mouse)Potency8.912510
thunberginol bMus musculus (house mouse)Potency6.309610
cp 60993Mus musculus (house mouse)Potency1.412510
methylbenzethonium chlorideMus musculus (house mouse)Potency12.589310
3,3'-diethylthiatricarbocyanine iodide, 3h-labeledMus musculus (house mouse)Potency4.466810
CrotaoprostrinMus musculus (house mouse)Potency8.912510
2-(dimethylaminostyryl)-1-ethylpyridiniumMus musculus (house mouse)Potency3.162310
7-fluoro-2-phenyl-4-quinoloneMus musculus (house mouse)Potency0.028210
piriqualoneMus musculus (house mouse)Potency8.912510
metochalconeMus musculus (house mouse)Potency11.220210
LSM-1411Mus musculus (house mouse)Potency5.011910
sinequanMus musculus (house mouse)Potency10.000010
maistemonineMus musculus (house mouse)Potency10.000010
diphenoxylate hydrochlorideMus musculus (house mouse)Potency12.589310
mg 624Mus musculus (house mouse)Potency7.079510
paroxetine maleateMus musculus (house mouse)Potency8.285210
beta-zearalenolMus musculus (house mouse)Potency12.589310
chaetoglobosin AMus musculus (house mouse)Potency0.794310
1-(1,3-benzodioxol-5-yl)-3-(6-methyl-2-pyridinyl)ureaMus musculus (house mouse)Potency7.079510
desmosdumotin cMus musculus (house mouse)Potency8.912510
arteannuin bMus musculus (house mouse)Potency4.466810
fluphenazineMus musculus (house mouse)Potency12.589310
homochlorocyclizine monohydrochlorideMus musculus (house mouse)Potency5.623410
protriptyline hydrochlorideMus musculus (house mouse)Potency1.122010
erythro-dihydrosphingosineMus musculus (house mouse)Potency14.689210
dantrolene sodiumMus musculus (house mouse)Potency11.220210
cycloheximideMus musculus (house mouse)Potency0.891310
methiazoleMus musculus (house mouse)Potency0.022410
dibenzheptropine citrateMus musculus (house mouse)Potency10.000010
4-methyl-N-[(4-methylphenyl)methyl]-2-furo[3,2-c]quinolinecarboxamideMus musculus (house mouse)Potency7.079510
8-bromo-6-ethyl-N-(2-oxolanylmethyl)-3-benzo[b][1,4]benzothiazepinecarboxamideMus musculus (house mouse)Potency3.162310
epinephrine bitartrateMus musculus (house mouse)Potency6.309610
cefdinirMus musculus (house mouse)Potency1.122010
a 38503Mus musculus (house mouse)Potency7.233410
N-cyclohexyl-2-[[6-(4-ethoxyphenyl)-3-pyridazinyl]thio]acetamideMus musculus (house mouse)Potency0.562310
parthenolideMus musculus (house mouse)Potency1.122010
2-[[[3-(2,5-dioxo-1-pyrrolidinyl)phenyl]-oxomethyl]amino]-N-methyl-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideMus musculus (house mouse)Potency0.010010
6-(4-ethylphenyl)-3-(methylthio)-[1,2,4]triazolo[4,3-b]pyridazineMus musculus (house mouse)Potency6.309610
N-(4-methoxyphenyl)-2-[[1-(phenylmethyl)-2-imidazolyl]thio]acetamideMus musculus (house mouse)Potency0.316210
5-(4-chlorophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency7.079510
3-hydroxy-2-methyl-1-(phenylmethyl)-4-pyridinoneMus musculus (house mouse)Potency7.079510
N-[2-methyl-5-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideMus musculus (house mouse)Potency8.912510
4-[[oxo-[4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazin-6-yl]methyl]amino]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)Potency11.220210
4-chloro-N-(4-ethylphenyl)-3-methyl-5-isoxazolecarboxamideMus musculus (house mouse)Potency11.220210
chlorhexidineMus musculus (house mouse)Potency10.000010
fluvoxamine maleateMus musculus (house mouse)Potency5.623410
2-methyl-6-(phenylethynyl)pyridine hydrochlorideMus musculus (house mouse)Potency10.000010
(R)-fluoxetine hydrochlorideMus musculus (house mouse)Potency8.912510
ag 14361Mus musculus (house mouse)Potency12.589310
u 74389gMus musculus (house mouse)Potency8.912510
a 77636Mus musculus (house mouse)Potency5.623410
a 443654Mus musculus (house mouse)Potency0.794310
anomalinMus musculus (house mouse)Potency22.387210
pyrenophorolMus musculus (house mouse)Potency12.589310
5-methoxy-8,8-dimethyl-2-phenyl-4H,8H-pyrano[2,3-h]chromen-4-oneMus musculus (house mouse)Potency5.011910
Xanthoangelol DMus musculus (house mouse)Potency8.912510
GR 127935 hydrochlorideMus musculus (house mouse)Potency14.125410
protoapigenoneMus musculus (house mouse)Potency8.912510
2-(2,1,3-benzothiadiazol-4-ylsulfonyl)-5-(4-bromophenyl)-3-pyrazolamineMus musculus (house mouse)Potency11.220210
R-(-)-actinodaphnineMus musculus (house mouse)Potency14.125410
calcimycinMus musculus (house mouse)Potency1.122010
2-hydroxyapomorphine, (r)-isomerMus musculus (house mouse)Potency5.623410
du 24565Mus musculus (house mouse)Potency12.589310
N-methyl-6-chloro-1-(3-methylphenyl)-2,3,4,5-tetrahydro-3-benzazepine-7,8-diol hydrobromideMus musculus (house mouse)Potency6.309610
N-[5-[2-(2,4-dichloroanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]-4-pentenamideMus musculus (house mouse)Potency12.589310
N-[5-[2-(2-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]pentanamideMus musculus (house mouse)Potency5.011910
2-ethyl-3-methoxy-N-(2-thiophen-2-ylethyl)-6-indazolecarboxamideMus musculus (house mouse)Potency8.912510
geduninMus musculus (house mouse)Potency31.622810
4-[3-(2-furanyl)-4-(3-nitrophenyl)-6-oxo-2,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoic acid ethyl esterMus musculus (house mouse)Potency2.511910
5-(1,3-benzodioxol-5-ylmethyl)-4-methyl-2-[[1-naphthalenyl(oxo)methyl]amino]-3-thiophenecarboxamideMus musculus (house mouse)Potency7.943310
3-(benzenesulfonyl)-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]propanamideMus musculus (house mouse)Potency5.011910
2-(4-fluorophenyl)-6-methoxy-1,3-benzothiazoleMus musculus (house mouse)Potency3.981110
chlorhexidine hydrochlorideMus musculus (house mouse)Potency11.220210
2',3'-dihydroxy-4',6'-dimethoxychalconeMus musculus (house mouse)Potency8.912510
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneMus musculus (house mouse)Potency1.000010
dehydrocurvularinMus musculus (house mouse)Potency0.891310
Moracin PMus musculus (house mouse)Potency8.912510
4-methoxybenzoic acid 2-(4-hydroxyphenyl)ethyl esterMus musculus (house mouse)Potency6.309610
3,6-diamino-10-methylacridinium chloride hydrochlorideMus musculus (house mouse)Potency1.122010
[4-(diphenylmethyl)-1-piperazinyl]-(5-methyl-4-nitro-3-isoxazolyl)methanoneMus musculus (house mouse)Potency10.000010
3-[2-(4-chlorophenyl)-5,7-dimethyl-6-pyrazolo[1,5-a]pyrimidinyl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]propanamideMus musculus (house mouse)Potency5.011910
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(4-morpholinyl)phenyl]-3-imidazo[1,2-a]pyrazinamineMus musculus (house mouse)Potency4.466810
[4-(2,3-dimethylphenyl)-1-piperazinyl]-[5-[(4-methylphenyl)sulfonylmethyl]-2-furanyl]methanoneMus musculus (house mouse)Potency0.891310
(3R,3aR,7aR)-3-[4-(4-acetylphenyl)-2-fluorophenyl]-7a-methyl-2-(phenylmethyl)-3,3a,6,7-tetrahydroisoindol-1-oneMus musculus (house mouse)Potency12.589310
3-[2-(4-fluorophenyl)-5-tetrazolyl]-2-methoxypyridineMus musculus (house mouse)Potency11.220210
2-chloro-3-[2-(4-methylphenyl)-5-tetrazolyl]pyridineMus musculus (house mouse)Potency3.162310
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2S,3S,4R)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency28.183810
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency12.589310
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency28.183810
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-4-(4-bromophenyl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency10.000010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneMus musculus (house mouse)Potency14.125410
2-(2,4-dimethoxyphenyl)-5-methyl-4-[[4-(4-quinazolinyl)-1-piperazinyl]methyl]oxazoleMus musculus (house mouse)Potency12.589310
3-hydroxy-2-(3-methylphenyl)-5-nitro-N-[1-(phenylmethyl)-4-piperidinyl]-4-triazolimineMus musculus (house mouse)Potency2.818410
2-(1,3-benzodioxol-5-ylmethyl)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinolineMus musculus (house mouse)Potency7.943310
[(2S,4S)-4-(4-bromophenyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency12.589310
(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxylic acid prop-2-enyl esterMus musculus (house mouse)Potency25.118910
1-[3-[(2R,4R)-2-[[4-(hydroxymethyl)phenyl]methoxy]-6-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]-3,4-dihydro-2H-pyran-4-yl]-1-indolyl]ethanoneMus musculus (house mouse)Potency7.943310
[(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneMus musculus (house mouse)Potency10.000010
violaceol IIMus musculus (house mouse)Potency12.589310
(2S,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-cyclohexyl-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamideMus musculus (house mouse)Potency12.589310
(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(phenylmethyl)-3,4-dihydro-2H-pyran-6-carboxamideMus musculus (house mouse)Potency28.183810
(2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-2H-pyran-6-carboxamideMus musculus (house mouse)Potency12.589310
quercetinMus musculus (house mouse)Potency7.943310
(8R)-3-[3-[[2-(4-chlorophenoxy)-1-oxoethyl]amino]phenyl]-7-(1-oxo-3,3-diphenylpropyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-8-carboxamideMus musculus (house mouse)Potency31.622810
3-chloro-N-propan-2-yl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency4.466810
N-(2-oxolanylmethyl)-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency5.011910
N-[(2S)-1-hydroxypropan-2-yl]-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency4.466810
N-(2-methoxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency7.943310
N-(2-hydroxyethyl)-3-methyl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideMus musculus (house mouse)Potency10.000010
thimerosalMus musculus (house mouse)Potency1.995310
N-[3-[2-(4-chloroanilino)-4-thiazolyl]phenyl]-3-(trifluoromethyl)benzamideMus musculus (house mouse)Potency12.589310
2-amino-N-[3-methoxy-5-[oxo-[3-(trifluoromethyl)anilino]methyl]phenyl]-4-thiazolecarboxamideMus musculus (house mouse)Potency3.162310
3-(4-bromophenyl)-N-[5-[[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)anilino]-oxomethyl]-2-methylphenyl]-1H-pyrazole-5-carboxamideMus musculus (house mouse)Potency12.589310
3-[[2-(4-bromophenyl)-1-oxoethyl]amino]-3-[4-[(4-fluorophenyl)methylamino]-3-nitrophenyl]propanamideMus musculus (house mouse)Potency7.079510
8-[1-(1,3-benzodioxol-5-yl)-3-(1-piperidinyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneMus musculus (house mouse)Potency28.183810
5,7-dimethoxy-8-[1-(4-methoxyphenyl)-3-(3-methyl-1-piperidinyl)-3-oxopropyl]-4-phenyl-1-benzopyran-2-oneMus musculus (house mouse)Potency10.000010
8-{1-[4-(dimethylamino)phenyl]-3-(pyrrolidin-1-yl)propyl}-5,7-dimethoxy-4-pentyl-2H-chromen-2-oneMus musculus (house mouse)Potency12.589310
(3R)-7-phenyl-2-(phenylmethyl)-3-[4-(trifluoromethyl)phenyl]-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneMus musculus (house mouse)Potency8.912510
8-[3-(diethylamino)-1-(4-methoxyphenyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneMus musculus (house mouse)Potency5.623410
8-[1-[4-(dimethylamino)phenyl]-3-(3-methyl-1-piperidinyl)propyl]-5,7-dimethoxy-4-phenyl-1-benzopyran-2-oneMus musculus (house mouse)Potency12.589310
(3R)-3-(2-fluoro-5-methylphenyl)-7-phenyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneMus musculus (house mouse)Potency14.125410
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esterMus musculus (house mouse)Potency28.183810
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterMus musculus (house mouse)Potency12.589310
1-(2,3-Dihydro-1,4-benzodioxin-3-ylmethyl)-5-methoxy-isatinMus musculus (house mouse)Potency12.589310
6-(3,5-dimethyl-4-isoxazolyl)-N-[(2-ethoxyphenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency25.118910
N-[4-[[[6-(3,5-dimethyl-4-isoxazolyl)-4-quinazolinyl]amino]methyl]phenyl]acetamideMus musculus (house mouse)Potency2.238710
6-(3,5-dimethyl-4-isoxazolyl)-N-[1-(2-furanyl)ethyl]-4-quinazolinamineMus musculus (house mouse)Potency10.000010
3-(2,5-dimethoxyphenyl)-6-(3,4-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency0.031610
1-[(4-fluorophenyl)methyl]-3-[1-(4-propan-2-ylphenyl)propyl]thioureaMus musculus (house mouse)Potency28.183810
5-fluoro-2-phenyl-1,2-benzothiazol-3-oneMus musculus (house mouse)Potency8.912510
2-(4-fluorophenyl)-1,2-benzothiazol-3-oneMus musculus (house mouse)Potency4.466810
N-(4-propan-2-ylphenyl)-1-[(1,3,3-trimethyl-2-oxo-5-indolyl)sulfonyl]-4-piperidinecarboxamideMus musculus (house mouse)Potency14.125410
puromycin dihydrochlorideMus musculus (house mouse)Potency1.000010
4-[2-[(6-chloro-4-quinazolinyl)amino]ethyl]phenolMus musculus (house mouse)Potency3.981110
4'-epichaetoviridin AMus musculus (house mouse)Potency12.589310
2-[[4-(2-phenoxyanilino)-6-(1-pyrrolidinyl)-1,3,5-triazin-2-yl]amino]ethanolMus musculus (house mouse)Potency12.589310
2-[[4-(5-chloro-2-propan-2-yloxyanilino)-6-(1-pyrrolidinyl)-1,3,5-triazin-2-yl]amino]ethanolMus musculus (house mouse)Potency10.000010
bucladesineMus musculus (house mouse)Potency10.000010
sri 62320Mus musculus (house mouse)Potency0.056210
fusidate sodiumMus musculus (house mouse)Potency4.466810
fractalsMus musculus (house mouse)Potency1.412510
sodium 2,6-dichloroindophenolMus musculus (house mouse)Potency8.912510
2-[[2-(2-cyanophenoxy)-1-oxoethyl]amino]-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid ethyl esterMus musculus (house mouse)Potency5.623410
10-deacetyltaxolMus musculus (house mouse)Potency1.000010
N-[3-(3-chlorophenyl)phenyl]-1-(3-isoxazolylmethyl)-4-piperidinecarboxamideMus musculus (house mouse)Potency28.183810
(2R)-N2-[2-(4-bicyclo[2.2.1]heptanyl)ethyl]-N1-[(2R,3R)-3-methyl-1-(methylamino)pentan-2-yl]hexane-1,2-diamineMus musculus (house mouse)Potency4.466810
4-[(2S)-2-[2-(4-ethoxyphenyl)ethylamino]-3-[[(2S)-1-(methylamino)hexan-2-yl]amino]propyl]phenolMus musculus (house mouse)Potency12.589310
(2R)-3-[[(2S)-1-cyclohexyl-3-(methylamino)propan-2-yl]amino]-2-[2-[3-(trifluoromethyl)phenyl]ethylamino]-1-propanolMus musculus (house mouse)Potency7.943310
N-[2-[1-[(4-methoxy-3-methylphenyl)methyl]-4-piperidinyl]-3-pyrazolyl]-4-phenylbutanamideMus musculus (house mouse)Potency17.782810
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-methyl-5-thiadiazolecarboxamideMus musculus (house mouse)Potency12.589310
N-methyl-N-(3-pyridinylmethyl)-5-(5,6,7,8-tetrahydronaphthalen-2-yloxymethyl)-3-isoxazolecarboxamideMus musculus (house mouse)Potency3.162310
2-[3-(4-morpholinyl)propylamino]-9-xanthenoneMus musculus (house mouse)Potency10.000010
norepinephrine bitartrateMus musculus (house mouse)Potency8.912510
(3S)-3-(2-methylpropyl)-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency12.589310
(3S)-3-(4-methoxyphenyl)-4-oxo-3-propan-2-yldiazetidine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency6.309610
(3S)-4-oxo-3-phenyl-3-propan-2-yldiazetidine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency8.912510
(5S)-1-heptyl-5-(2-methylpropyl)-N-phenyl-4,5-dihydroimidazol-2-amineMus musculus (house mouse)Potency12.589310
(3S)-3-cyclopentyl-4-oxo-3-phenyldiazetidine-1,2-dicarboxylic acid dimethyl esterMus musculus (house mouse)Potency7.079510
N-[5-[[2-(4-acetamidoanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-3-methoxybenzamideMus musculus (house mouse)Potency1.995310
4-tert-butyl-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.891310
N-[5-[[2-(4-acetamidoanilino)-2-oxoethyl]thio]-1,3,4-thiadiazol-2-yl]-5-bromo-2-furancarboxamideMus musculus (house mouse)Potency1.000010
4-ethoxy-N-[5-[[2-oxo-2-(2-oxolanylmethylamino)ethyl]thio]-1,3,4-thiadiazol-2-yl]benzamideMus musculus (house mouse)Potency0.891310
stachyoseMus musculus (house mouse)Potency3.548110
LSM-1873Mus musculus (house mouse)Potency28.183810
LSM-1675Mus musculus (house mouse)Potency11.220210
2-(methylthio)-4-phenyl-6-propan-2-yl-1,3,5-triazineMus musculus (house mouse)Potency10.000010
N-[5-[(2,6-difluorophenyl)sulfonylamino]pentyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideMus musculus (house mouse)Potency3.548110
5-(4-methoxyphenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency3.548110
5-(4-bromophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency0.891310
LSM-27979Mus musculus (house mouse)Potency12.589310
4-[(9-cyclopentyl-6-oxo-5-propan-2-yl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-(1-methyl-4-piperidinyl)benzamideMus musculus (house mouse)Potency11.220210
N-(2-furanylmethyl)-N-methyl-6-(1-methyl-5-indolyl)-4-quinazolinamineMus musculus (house mouse)Potency1.122010
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineMus musculus (house mouse)Potency12.589310
6-(3-methylphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency28.183810
6-(1-methyl-5-indolyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineMus musculus (house mouse)Potency7.943310
5-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]methyl]-8-quinolinolMus musculus (house mouse)Potency3.548110
2-[5-(2-fluorophenyl)-2-furanyl]-3-hydroxy-1,2-dihydroquinazolin-4-oneMus musculus (house mouse)Potency11.220210
3-hydroxy-2-(5-thiophen-2-yl-2-furanyl)-1,2-dihydroquinazolin-4-oneMus musculus (house mouse)Potency5.623410
2-[5-(3-fluorophenyl)-2-furanyl]-3-hydroxy-1,2-dihydroquinazolin-4-oneMus musculus (house mouse)Potency12.589310
3-hydroxy-2-[5-[4-(trifluoromethyl)phenyl]-2-furanyl]-1,2-dihydroquinazolin-4-oneMus musculus (house mouse)Potency10.000010
2-naphthalenecarboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterMus musculus (house mouse)Potency5.623410
6-(3-cyclopentyloxy-4-methoxyphenyl)-3-(2-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency0.794310
3-(2-chlorophenyl)-6-(3-cyclopentyloxy-4-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency4.466810
6-(3-cyclopentyloxy-4-methoxyphenyl)-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency2.511910
6-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-3-(2-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency0.010010
6-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-3-(2-fluorophenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency4.466810
3-(2-chlorophenyl)-6-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency8.912510
6-[3-(cyclopropylmethoxy)-4-methoxyphenyl]-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency1.000010
6-[3-(cyclopropylmethoxy)-4-(difluoromethoxy)phenyl]-3-(2,5-dimethoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency12.589310
6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-3-(2-methoxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency1.995310
3-(2-chlorophenyl)-6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency4.466810
3-(2-fluorophenyl)-6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency2.818410
6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-3-[2-(trifluoromethyl)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency0.028210
3-(2,5-dimethoxyphenyl)-6-[4-methoxy-3-(3-oxolanyloxy)phenyl]-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineMus musculus (house mouse)Potency1.412510
1-tert-butyl-5-[[3-[(1-tert-butyl-4-oxo-5-pyrazolo[3,4-d]pyrimidinyl)methyl]-2-fluorophenyl]methyl]-4-pyrazolo[3,4-d]pyrimidinoneMus musculus (house mouse)Potency8.912510
4-(3,5-difluoroanilino)-6-(2,2-difluoroethylamino)-1,3,5-triazine-2-carbonitrileMus musculus (house mouse)Potency10.000010
6-(3-chloroanilino)-9-cyclopentyl-2-purinecarbonitrileMus musculus (house mouse)Potency8.912510
5-(2-methoxyphenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency11.220210
5-(3-methoxyphenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency1.412510
5-(3-fluorophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency7.079510
4-[(1-methyl-5-tetrazolyl)thio]-5-[2-(trifluoromethyl)phenyl]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency10.000010
4-[(1-methyl-5-tetrazolyl)thio]-5-[3-(trifluoromethyl)phenyl]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency8.912510
4-[(1-methyl-5-tetrazolyl)thio]-5-[4-(trifluoromethyl)phenyl]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency3.162310
5-(2-bromophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency10.000010
5-(3-bromophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency8.912510
5-(2-chlorophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency10.000010
4-[4-[(1-methyl-5-tetrazolyl)thio]-5-thieno[2,3-d]pyrimidinyl]benzonitrileMus musculus (house mouse)Potency5.011910
4-[(1-methyl-5-tetrazolyl)thio]-5-(4-nitrophenyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency1.000010
4-[(1-methyl-5-tetrazolyl)thio]-5-(4-phenylphenyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency1.995310
5-(2-benzofuranyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency7.079510
5-(4-dibenzothiophenyl)-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency8.912510
4-[(1-methyl-5-tetrazolyl)thio]-5-(1H-pyrrol-2-yl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency7.079510
1-[2-[4-[(1-methyl-5-tetrazolyl)thio]-5-thieno[2,3-d]pyrimidinyl]phenyl]ethanoneMus musculus (house mouse)Potency10.000010
4-[(1-methyl-5-tetrazolyl)thio]-5-(1-naphthalenyl)thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency3.981110
5-bromo-4-[(1-methyl-5-tetrazolyl)thio]thieno[2,3-d]pyrimidineMus musculus (house mouse)Potency2.818410
1-[4-[4-(2-furanylmethylamino)phenyl]-1-piperazinyl]ethanoneMus musculus (house mouse)Potency4.466810
1-[4-[4-[(5-bromo-2-furanyl)methylamino]phenyl]-1-piperazinyl]ethanoneMus musculus (house mouse)Potency5.623410
N-[(5-chloro-8-hydroxy-7-quinolinyl)-cyclopropylmethyl]acetamideMus musculus (house mouse)Potency3.981110
N-[(5-fluoro-8-hydroxy-7-quinolinyl)-thiophen-2-ylmethyl]acetamideMus musculus (house mouse)Potency5.011910
4-[3-(3-bromophenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]benzenesulfonamideMus musculus (house mouse)Potency11.220210
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[(4-phenoxyphenyl)methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]-4-pyridinecarboxamideMus musculus (house mouse)Potency12.589310
N-[(2R,3S)-2-[[(4-chlorophenyl)sulfonyl-methylamino]methyl]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-4,4,4-trifluorobutanamideMus musculus (house mouse)Potency8.912510
N-(2-aminophenyl)-4-[[[(2S,3S)-10-[[cyclohexyl(oxo)methyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl-methylamino]methyl]benzamideMus musculus (house mouse)Potency6.309610
1-(4-fluorophenyl)-3-[(2R,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-(phenylmethyl)amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]ureaMus musculus (house mouse)Potency12.589310
1-[[(2S,3S)-10-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]ureaMus musculus (house mouse)Potency11.220210
1-[(2S,3S)-2-[[benzenesulfonyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-[4-(trifluoromethyl)phenyl]ureaMus musculus (house mouse)Potency28.183810
1-[[(2S,3R)-10-[[(cyclohexylamino)-oxomethyl]amino]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-[4-(trifluoromethyl)phenyl]ureaMus musculus (house mouse)Potency12.589310
1-[[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-10-[[oxo-[4-(trifluoromethyl)anilino]methyl]amino]-3,4-dihydro-2H-1,5-benzoxazocin-2-yl]methyl]-1-methyl-3-phenylureaMus musculus (house mouse)Potency10.000010
1-[(2R,3R)-2-[[benzenesulfonyl(methyl)amino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-3-[4-(trifluoromethyl)phenyl]ureaMus musculus (house mouse)Potency12.589310
5-[[2-furanylmethyl(methyl)amino]methyl]-8-quinolinolMus musculus (house mouse)Potency25.118910
dehydroacetic acidMus musculus (house mouse)Potency15.848910
salinazidMus musculus (house mouse)Potency7.079510
phthivazideMus musculus (house mouse)Potency3.981110
1-hydroxyphenazineMus musculus (house mouse)Potency11.220210
bentazepamMus musculus (house mouse)Potency4.466810
tegaserod maleateMus musculus (house mouse)Potency1.412510
2-phenoxymethyl-3h-quinazolin-4-oneMus musculus (house mouse)Potency8.912510
N-[4-(6-chloro-5-nitro-1H-benzimidazol-2-yl)phenyl]acetamideMus musculus (house mouse)Potency14.125410
pyridoxal 4-methoxybenzoyl hydrazoneMus musculus (house mouse)Potency28.183810
N'-(1h-indol-3-ylmethylene)benzohydrazideMus musculus (house mouse)Potency15.848910
carbadoxMus musculus (house mouse)Potency1.778310