Proteins > G-protein coupled receptor homolog US28
Page last updated: 2024-08-07 16:54:40
G-protein coupled receptor homolog US28
[no definition available]
Synonyms
HHRF3
Research
Bioassay Publications (2)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (50.00) | 29.6817 |
| 2010's | 1 (50.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| vuf 2274 | Human herpesvirus 5 strain AD169 | IC50 | 9.3000 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| methiothepin | Human herpesvirus 5 strain AD169 | EC50 | 0.3524 | 1 | 2 |
| vuf 2274 | Human herpesvirus 5 strain AD169 | EC50 | 4.0903 | 2 | 3 |
Allosteric modulation of the G protein-coupled US28 receptor of human cytomegalovirus: are the small-weight inverse agonist of US28 'camouflaged' agonists?Bioorganic & medicinal chemistry letters, , Aug-15, Volume: 24, Issue:16, 2014
Synthesis and structure-activity relationship of the first nonpeptidergic inverse agonists for the human cytomegalovirus encoded chemokine receptor US28.Journal of medicinal chemistry, , Oct-06, Volume: 48, Issue:20, 2005