[no definition available]
EC 3.4.21.1
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 1 (7.14) | 18.7374 |
| 1990's | 4 (28.57) | 18.2507 |
| 2000's | 4 (28.57) | 29.6817 |
| 2010's | 5 (35.71) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| 3,4-dichloroisocoumarin | Bos taurus (cattle) | IC50 | 3.5000 | 1 | 1 |
| 3-nitrobenzeneboronic acid | Bos taurus (cattle) | IC50 | 200.0000 | 1 | 1 |
| benzyl benzoate | Bos taurus (cattle) | IC50 | 250.0000 | 1 | 1 |
| benzo(b)thiophene-2-boronic acid | Bos taurus (cattle) | IC50 | 5.0000 | 1 | 1 |
| clotrimazole | Bos taurus (cattle) | IC50 | 85.0000 | 1 | 1 |
| econazole | Bos taurus (cattle) | IC50 | 150.0000 | 1 | 1 |
| fluconazole | Bos taurus (cattle) | IC50 | 400.0000 | 1 | 1 |
| glyburide | Bos taurus (cattle) | IC50 | 360.0000 | 1 | 1 |
| ketoconazole | Bos taurus (cattle) | IC50 | 150.0000 | 1 | 1 |
| miconazole | Bos taurus (cattle) | IC50 | 125.0000 | 1 | 1 |
| nicardipine | Bos taurus (cattle) | IC50 | 175.0000 | 1 | 1 |
| oxaprozin | Bos taurus (cattle) | IC50 | 200.0000 | 1 | 1 |
| phloretin | Bos taurus (cattle) | IC50 | 496.0000 | 1 | 1 |
| sulconazole | Bos taurus (cattle) | IC50 | 110.0000 | 1 | 1 |
| delavirdine | Bos taurus (cattle) | IC50 | 225.0000 | 1 | 1 |
| bentranil | Bos taurus (cattle) | IC50 | 11.7000 | 1 | 1 |
| bentranil | Bos taurus (cattle) | Ki | 8.7000 | 1 | 1 |
| talinolol | Bos taurus (cattle) | Ki | 0.9000 | 1 | 1 |
| indole-3-carboxylic acid | Bos taurus (cattle) | Ki | 5,250.0000 | 1 | 4 |
| carbobenzoxyvalylphenylalanine aldehyde | Bos taurus (cattle) | Ki | 54.0000 | 1 | 1 |
| indole-2-carboxylic acid | Bos taurus (cattle) | Ki | 4,700.0000 | 1 | 4 |
| zpck | Bos taurus (cattle) | IC50 | 17.0000 | 1 | 1 |
| foy 251 | Bos taurus (cattle) | IC50 | 100.0000 | 1 | 1 |
| n-dansyl-3-aminobenzeneboronic acid | Bos taurus (cattle) | IC50 | 100.0000 | 1 | 1 |
| l 694,458 | Bos taurus (cattle) | IC50 | 0.9800 | 1 | 1 |
| 2-(3-nitrophenyl)-3,1-benzoxazin-4-one | Bos taurus (cattle) | IC50 | 341.1000 | 1 | 1 |
| 2-(3-nitrophenyl)-3,1-benzoxazin-4-one | Bos taurus (cattle) | Ki | 341.2000 | 1 | 1 |
| bortezomib | Bos taurus (cattle) | Ki | 2.4000 | 1 | 1 |
| tosylphenylalanyl chloromethyl ketone | Bos taurus (cattle) | IC50 | 140.0000 | 1 | 1 |
| Methyl indole-5-carboxylate | Bos taurus (cattle) | Ki | 2,800.0000 | 1 | 3 |
| quercetin | Bos taurus (cattle) | IC50 | 292.5000 | 2 | 2 |
| rutin | Bos taurus (cattle) | IC50 | 500.0000 | 1 | 1 |
| rottlerin | Bos taurus (cattle) | IC50 | 119.0000 | 2 | 2 |
| camostat mesylate | Bos taurus (cattle) | IC50 | 100.0000 | 1 | 1 |
| n,n-(4-xylylidene)bisaminoguanidine | Bos taurus (cattle) | Ki | 55.3333 | 1 | 3 |
| glyoxal bis(guanylhydrazone) | Bos taurus (cattle) | Ki | 565.2500 | 1 | 4 |
| jaw | Bos taurus (cattle) | Ki | 1,326.6667 | 1 | 3 |
| clavulanate potassium | Bos taurus (cattle) | IC50 | 434.5000 | 2 | 2 |
| penicillin g sodium | Bos taurus (cattle) | IC50 | 5.4000 | 2 | 2 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| congo red | Bos taurus (cattle) | Concentration | 40.0000 | 1 | 1 |