Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
adenine | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
quinacrine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
methylmalonic acid | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
4-amino-1,8-naphthalimide | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
dipyridamole | Homo sapiens (human) | Potency | 35.3981 | 3 | 0 |
isoguvacine | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
jl 18 | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
nomifensine | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
protoporphyrin ix | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
sanguinarine | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
alizarin | Homo sapiens (human) | Potency | 41.3638 | 2 | 0 |
acriflavine chloride | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
pyronine | Homo sapiens (human) | Potency | 39.2802 | 3 | 0 |
methylergonovine | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
2,4-dihydroxybenzophenone | Homo sapiens (human) | Potency | 27.9588 | 2 | 0 |
rhein | Homo sapiens (human) | Potency | 43.3533 | 2 | 0 |
3-aminofluoranthene | Homo sapiens (human) | Potency | 29.6546 | 2 | 0 |
6,7-Dimethyl-9-(2-acetoxyethyl)isoalloxazine | Homo sapiens (human) | Potency | 6.9578 | 3 | 0 |
(7S,9S)-7-[(4-amino-5-hydroxy-6-methyl-2-oxanyl)oxy]-6,9,11-trihydroxy-9-(2-hydroxy-1-oxoethyl)-4-methoxy-8,10-dihydro-7H-tetracene-5,12-dione | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
s-2678 | Homo sapiens (human) | Potency | 38.6387 | 2 | 0 |
idarubicin | Homo sapiens (human) | Potency | 7.9433 | 1 | 0 |
flupirtine | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
topotecan hydrochloride | Homo sapiens (human) | Potency | 24.7702 | 3 | 0 |
daunorubicin hydrochloride | Homo sapiens (human) | Potency | 29.0123 | 3 | 0 |
epirubicin hydrochloride | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
2-Methoxyxanthone | Homo sapiens (human) | Potency | 53.7312 | 2 | 0 |
coumarin 153 | Homo sapiens (human) | Potency | 4.7816 | 2 | 0 |
methyl fluorone black | Homo sapiens (human) | Potency | 2.3260 | 2 | 0 |
9-hydroxyphenylfluoron | Homo sapiens (human) | Potency | 17.2374 | 3 | 0 |
agroclavine | Homo sapiens (human) | Potency | 39.5908 | 2 | 0 |
isopyrin hydrochloride | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
2-butyl-6-(butylamino)-1h-benzo(de)isoquinoline-1,3(2h)-dione | Homo sapiens (human) | Potency | 14.6120 | 2 | 0 |
1-(2-thiazolylazo)-2-naphthol | Homo sapiens (human) | Potency | 51.2591 | 2 | 0 |
coumarin 7 | Homo sapiens (human) | Potency | 15.8489 | 1 | 0 |
paxilline | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
3'-deamino-3'-hydroxydaunorubicin | Homo sapiens (human) | Potency | 31.5503 | 2 | 0 |
alpha-ergocryptine | Homo sapiens (human) | Potency | 25.2423 | 2 | 0 |
sch 45752 | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
epiberberine | Homo sapiens (human) | Potency | 34.6080 | 2 | 0 |
sb 216763 | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
raubasine | Homo sapiens (human) | Potency | 70.7946 | 1 | 0 |
methyl reserpate | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
nsc228155 | Homo sapiens (human) | Potency | 37.2858 | 2 | 0 |
2,3-diaminophenazine | Homo sapiens (human) | Potency | 33.9021 | 2 | 0 |
n,n-dimethyldaunorubicin | Homo sapiens (human) | Potency | 29.6546 | 2 | 0 |
idarubicin hydrochloride | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
4-[3-(1,3-dioxo-2-isoindolyl)propylamino]-2-methylisoindole-1,3-dione | Homo sapiens (human) | Potency | 22.3872 | 1 | 0 |
N,N-di(propan-2-yl)-2-[(1-propyl-5-tetrazolyl)thio]acetamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
benidipine hydrochloride | Homo sapiens (human) | Potency | 14.1254 | 1 | 0 |
2-cyano-N-(3-methoxypropyl)-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetamide | Homo sapiens (human) | Potency | 43.3533 | 2 | 0 |
1-[3-[1-cyano-2-oxo-2-[(phenylmethyl)amino]ethyl]-2-quinoxalinyl]-3-piperidinecarboxylic acid ethyl ester | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid cyclohexyl ester | Homo sapiens (human) | Potency | 30.2153 | 2 | 0 |
LSM-32147 | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
Glyceryl lactopalmitate | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
7-ethoxy-9-nitro-5H-benzo[b][1,4]benzoxazepin-6-one | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
5-[[5-(diethylamino)-2-furanyl]methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione | Homo sapiens (human) | Potency | 17.7828 | 1 | 0 |
6-methyl-4-(trifluoromethyl)-7,8,9,10-tetrahydropyrano[2,3-f]quinolin-2-one | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
3-chloro-1-(3,4-dichlorophenyl)-4-(dimethylamino)pyrrole-2,5-dione | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
1-(3-chlorophenyl)-3-(phenylmethyl)thiourea | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
2-[(1-ethyl-2,5-dimethyl-3-pyrrolyl)methylidene]indene-1,3-dione | Homo sapiens (human) | Potency | 62.8565 | 2 | 0 |
4,5-dimethylcyclopenta[c]quinolizine-1,2-dicarboxylic acid dimethyl ester | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
curcumin | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamide | Homo sapiens (human) | Potency | 36.6020 | 2 | 0 |
[3-amino-6-thiophen-2-yl-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinyl]-cyclopropylmethanone | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
3-chloro-5-(2-furanyl)-N-propan-2-yl-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinecarboxamide | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
N'-[2-(4-bromo-2-methylphenoxy)-1-oxoethyl]-2-pyrazinecarbohydrazide | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
1-[2,3-bis(2-furanyl)-6-quinoxalinyl]-3-[4-(4-morpholinyl)phenyl]thiourea | Homo sapiens (human) | Potency | 44.4215 | 2 | 0 |
4-methoxy-N-[5-(4-methoxyphenyl)-4-(4-nitrophenyl)-2-thiazolyl]benzamide | Homo sapiens (human) | Potency | 54.2478 | 2 | 0 |
N-(2,4-dimethoxyphenyl)-N'-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]butanediamide | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
N-[2-methoxy-5-(3-methyl-4-oxo-1-phthalazinyl)phenyl]-2-(4-methylphenoxy)acetamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
9-methoxy-6-[(4-methoxyphenyl)methyl]indolo[3,2-b]quinoxaline | Homo sapiens (human) | Potency | 25.9152 | 3 | 0 |
2-[[4-(2-ethoxyanilino)-6-(4-ethoxyanilino)-2-pyrimidinyl]methylidene]propanedinitrile | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
4-[[oxo-(1-phenyl-3-pyridin-4-yl-4-pyrazolyl)methyl]amino]benzoic acid methyl ester | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-[[5-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]-4-oxo-2-phenyl-1-benzopyran-7-yl]oxy]acetic acid tert-butyl ester | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
4E2RCat | Homo sapiens (human) | Potency | 11.2202 | 1 | 0 |
3,4-dimethoxy-N-[4-(2,2,3,3-tetrafluoropropoxy)-3-(trifluoromethyl)phenyl]benzamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
2-[4-(2-methylpropyl)phenyl]propanoic acid [2-(1H-indol-3-yl)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 44.6684 | 1 | 0 |
N-(2-methoxycyclohexyl)-3,4-dimethylaniline | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1,3,8-trimethyl-5,10-diphenylpyrimido[1,2]pyrrolo[4,5-b]pyridazine-2,4-dione | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dione | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
2-cyano-N-(phenylmethyl)-2-[3-(1-pyrrolidinyl)-2-quinoxalinyl]acetamide | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
3-(3,4-dihydro-2H-quinolin-1-ylmethyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine | Homo sapiens (human) | Potency | 33.9021 | 2 | 0 |
1-[[1-(2-methoxyanilino)-4-isoquinolinyl]-oxomethyl]-4-piperidinecarboxamide | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
N-(6-acetamido-3-prop-2-enyl-1,3-benzothiazol-2-ylidene)-2-thiophenecarboxamide | Homo sapiens (human) | Potency | 35.4813 | 1 | 0 |
3-benzoyl-1,5-bis(2-methoxyphenyl)-3a,6a-dihydropyrrolo[3,4-c]pyrazole-4,6-dione | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
3-(3,4-dimethylphenyl)sulfonyl-2-imino-1-prop-2-enyl-5-dipyrido[1,2-e-4',3'-f]pyrimidinone | Homo sapiens (human) | Potency | 54.8500 | 2 | 0 |
2-(1-benzimidazolyl)acetic acid [2-[(9,10-dioxo-1-anthracenyl)amino]-2-oxoethyl] ester | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
suramin sodium | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
2-[[4-(2-methoxyphenyl)sulfonyl-1-piperazinyl]sulfonyl]benzonitrile | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
1-(7-methyloctyl)-3-[4-(4-morpholinylsulfonyl)phenyl]thiourea | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
cgp 7930 | Homo sapiens (human) | Potency | 25.1189 | 1 | 0 |
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamide | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
ncgc00099374 | Homo sapiens (human) | Potency | 32.6090 | 1 | 0 |
3-[4-(4-morpholinylsulfonyl)phenyl]propanoic acid [2-(4-acetylanilino)-2-oxoethyl] ester | Homo sapiens (human) | Potency | 89.1251 | 1 | 0 |
n-oleoylethanolamine | Homo sapiens (human) | Potency | 19.9526 | 1 | 0 |
su 6656 | Homo sapiens (human) | Potency | 28.1838 | 1 | 0 |
ag 183 | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
semaxinib | Homo sapiens (human) | Potency | 42.8000 | 2 | 0 |
isoalloxazine | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
2-(dimethylaminostyryl)-1-ethylpyridinium | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
chloride of pseudoisocyanine | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
LSM-6455 | Homo sapiens (human) | Potency | 35.4000 | 2 | 0 |
alpha-solanine | Homo sapiens (human) | Potency | 56.2341 | 1 | 0 |
lissamine rhodamine b | Homo sapiens (human) | Potency | 20.6062 | 3 | 0 |
carmine | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
brl 15572 | Homo sapiens (human) | Potency | 31.6228 | 1 | 0 |
win 62577 | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
3,6-diamino-10-methylacridinium chloride hydrochloride | Homo sapiens (human) | Potency | 10.0000 | 1 | 0 |
(2S)-4-methyl-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl ester | Homo sapiens (human) | Potency | 39.8107 | 1 | 0 |
cyclopenol | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
hispidin | Homo sapiens (human) | Potency | 50.1187 | 1 | 0 |
sepiapterin | Homo sapiens (human) | Potency | 37.2858 | 2 | 0 |
N-[3-[(1,5-dimethyl-3-oxo-2-phenyl-4-pyrazolyl)amino]-1-isoindolylidene]-2-thiophenecarboxamide | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |
lomofungin | Homo sapiens (human) | Potency | 79.4328 | 1 | 0 |