Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
chlordecone | Plasmodium falciparum 3D7 | AC50 | 2.9300 | 1 | 0 |
1,10-phenanthroline | Plasmodium falciparum 3D7 | AC50 | 6.6050 | 1 | 0 |
pyrithione | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
bay h 4502 | Plasmodium falciparum 3D7 | AC50 | 1.0690 | 1 | 0 |
broxyquinoline | Plasmodium falciparum 3D7 | AC50 | 0.3730 | 1 | 0 |
chloroxine | Plasmodium falciparum 3D7 | AC50 | 0.5110 | 1 | 0 |
clioquinol | Plasmodium falciparum 3D7 | AC50 | 0.6190 | 1 | 0 |
clotrimazole | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
cloxyquin | Plasmodium falciparum 3D7 | AC50 | 8.3620 | 1 | 0 |
dichlorophen | Plasmodium falciparum 3D7 | AC50 | 5.4140 | 1 | 0 |
disulfiram | Plasmodium falciparum 3D7 | AC50 | 4.5540 | 1 | 0 |
fluconazole | Plasmodium falciparum 3D7 | AC50 | 2.7210 | 1 | 0 |
hexachlorophene | Plasmodium falciparum 3D7 | AC50 | 0.6760 | 1 | 0 |
iodoquinol | Plasmodium falciparum 3D7 | AC50 | 0.3140 | 1 | 0 |
itraconazole | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
miconazole | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
pomiferin | Plasmodium falciparum 3D7 | AC50 | 8.7510 | 1 | 0 |
thiram | Plasmodium falciparum 3D7 | AC50 | 3.9570 | 1 | 0 |
triclosan | Plasmodium falciparum 3D7 | AC50 | 7.5440 | 1 | 0 |
cycloheximide | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
1-(2-pyridylazo)-2-naphthol | Plasmodium falciparum 3D7 | AC50 | 2.6620 | 1 | 0 |
fentichlor | Plasmodium falciparum 3D7 | AC50 | 3.0660 | 1 | 0 |
sterogenol | Plasmodium falciparum 3D7 | AC50 | 4.0320 | 1 | 0 |
nitrophenide | Plasmodium falciparum 3D7 | AC50 | 4.6250 | 1 | 0 |
ethyl violet | Plasmodium falciparum 3D7 | AC50 | 0.7350 | 1 | 0 |
nitroxoline | Plasmodium falciparum 3D7 | AC50 | 1.6570 | 1 | 0 |
2,3,4,5-tetrachlorophenate | Plasmodium falciparum 3D7 | AC50 | 1.7030 | 1 | 0 |
cetyldimethylethylammonium bromide | Plasmodium falciparum 3D7 | AC50 | 4.0420 | 1 | 0 |
2-n-octyl-4-isothiazolin-3-one | Plasmodium falciparum 3D7 | AC50 | 0.8710 | 1 | 0 |
wr 171,699 | Plasmodium falciparum 3D7 | AC50 | 7.4190 | 1 | 0 |
ciclopirox olamine | Plasmodium falciparum 3D7 | AC50 | 1.1900 | 1 | 0 |
Nanaomycin | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
triadimenol | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
propiconazole | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
butoconazole nitrate | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
triclabendazole | Plasmodium falciparum 3D7 | AC50 | 6.4130 | 1 | 0 |
sulconazole, mononitrate, (+-)-isomer | Plasmodium falciparum 3D7 | AC50 | 0.5760 | 1 | 0 |
miconazole nitrate | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
econazole nitrate | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
2,2',2''-terpyridine | Plasmodium falciparum 3D7 | AC50 | 1.0290 | 1 | 0 |
2-methyl-4-nitroquinoline 1-oxide | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
totarol | Plasmodium falciparum 3D7 | AC50 | 2.8630 | 1 | 0 |
1-(2-thiazolylazo)-2-naphthol | Plasmodium falciparum 3D7 | AC50 | 0.6300 | 1 | 0 |
9,10-phenanthrenequinone monoxime | Plasmodium falciparum 3D7 | AC50 | 1.5700 | 1 | 0 |
2-phenyl-1,2-benzisothiazol-3-(2h)-one | Plasmodium falciparum 3D7 | AC50 | 9.1920 | 1 | 0 |
dermofix | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
acetoxycycloheximide | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
wortmannin | Plasmodium falciparum 3D7 | AC50 | 0.2150 | 1 | 0 |
nsc228155 | Plasmodium falciparum 3D7 | AC50 | 6.8810 | 1 | 0 |
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinone | Plasmodium falciparum 3D7 | AC50 | 1.6410 | 1 | 0 |
nsc 680410 | Plasmodium falciparum 3D7 | AC50 | 8.9110 | 1 | 0 |
n,n-dimethyldaunorubicin | Plasmodium falciparum 3D7 | AC50 | 1.5770 | 1 | 0 |
terconazole | Plasmodium falciparum 3D7 | AC50 | 1.4970 | 1 | 0 |
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diol | Plasmodium falciparum 3D7 | AC50 | 7.7570 | 1 | 0 |
ketoconazole | Plasmodium falciparum 3D7 | AC50 | 1.2860 | 1 | 0 |
calmidazolium | Plasmodium falciparum 3D7 | AC50 | 5.4700 | 1 | 0 |
N-(4-chlorophenyl)-3-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]propanamide | Plasmodium falciparum 3D7 | AC50 | 2.8720 | 1 | 0 |
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide | Plasmodium falciparum 3D7 | AC50 | 0.8940 | 1 | 0 |
5-(4-cyclohexylphenyl)-1,2-dihydropyrazol-3-one | Plasmodium falciparum 3D7 | AC50 | 7.7010 | 1 | 0 |
3-pyridinecarboxylic acid (5-chloro-8-quinolinyl) ester | Plasmodium falciparum 3D7 | AC50 | 7.8550 | 1 | 0 |
1-(3-nitrophenyl)-3-phenyl-2-propyn-1-one | Plasmodium falciparum 3D7 | AC50 | 0.2910 | 1 | 0 |
5-tert-butyl-2-methyl-3-phenyl-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamine | Plasmodium falciparum 3D7 | AC50 | 3.0200 | 1 | 0 |
N-[3-(6-methyl-4-phenyl-2-quinolinyl)phenyl]methanesulfonamide | Plasmodium falciparum 3D7 | AC50 | 9.5980 | 1 | 0 |
4-[[oxo-(1-phenyl-3-pyridin-4-yl-4-pyrazolyl)methyl]amino]benzoic acid methyl ester | Plasmodium falciparum 3D7 | AC50 | 4.0850 | 1 | 0 |
thiocyanic acid [2-(1-naphthalenyl)-2-oxoethyl] ester | Plasmodium falciparum 3D7 | AC50 | 1.9190 | 1 | 0 |
mcb-613 | Plasmodium falciparum 3D7 | AC50 | 9.0640 | 1 | 0 |
1-(4-bromophenyl)-3-(diethylamino)pyrrolidine-2,5-dione | Plasmodium falciparum 3D7 | AC50 | 2.9670 | 1 | 0 |
1-hexadecyl-3-methylimidazolium bromide | Plasmodium falciparum 3D7 | AC50 | 2.8920 | 1 | 0 |
N-(3-bicyclo[2.2.1]heptanyl)-3-bromo-4-methoxybenzenesulfonamide | Plasmodium falciparum 3D7 | AC50 | 3.5170 | 1 | 0 |
N-(3-bicyclo[2.2.1]heptanyl)-4-chlorobenzenesulfonamide | Plasmodium falciparum 3D7 | AC50 | 34.2562 | 4 | 0 |
1-(1,3-benzodioxol-5-yl)-3-(5-tert-butyl-2-methoxyphenyl)urea | Plasmodium falciparum 3D7 | AC50 | 8.9630 | 1 | 0 |
5-chloro-7-[3-pyridinyl-(2-pyridinylamino)methyl]-8-quinolinol | Plasmodium falciparum 3D7 | AC50 | 8.0860 | 1 | 0 |
cb 7969312 | Plasmodium falciparum 3D7 | AC50 | 1.4980 | 1 | 0 |
N-[[2-(4-chlorophenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]benzenesulfonamide | Plasmodium falciparum 3D7 | AC50 | 3.7270 | 1 | 0 |
4-[1-(4-bromophenyl)-2-nitroethyl]-5-methyl-2-phenyl-1H-pyrazol-3-one | Plasmodium falciparum 3D7 | AC50 | 8.5430 | 1 | 0 |
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanone | Plasmodium falciparum 3D7 | AC50 | 4.2370 | 1 | 0 |
2,5-dichloro-N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-3-thiophenecarboxamide | Plasmodium falciparum 3D7 | AC50 | 2.4330 | 1 | 0 |
2-chloro-N-(2,6-dimethylphenyl)-3-oxo-3-phenylpropanamide | Plasmodium falciparum 3D7 | AC50 | 1.1150 | 1 | 0 |
2,4-dichloro-N-[5-(5,6,7,8-tetrahydronaphthalen-2-yl)-1,3,4-oxadiazol-2-yl]benzamide | Plasmodium falciparum 3D7 | AC50 | 3.3470 | 1 | 0 |
5'-bromo-2'-spiro[1,2-dihydro-4,1,2-benzoxadiazine-3,3'-1H-indole]one | Plasmodium falciparum 3D7 | AC50 | 1.4620 | 1 | 0 |
n-oleoylethanolamine | Plasmodium falciparum 3D7 | AC50 | 9.2500 | 1 | 0 |
cp 60993 | Plasmodium falciparum 3D7 | AC50 | 4.8400 | 1 | 0 |
methylbenzethonium chloride | Plasmodium falciparum 3D7 | AC50 | 7.8030 | 1 | 0 |
sclerotiorin | Plasmodium falciparum 3D7 | AC50 | 2.1090 | 1 | 0 |
cycloheximide | Plasmodium falciparum 3D7 | AC50 | 0.1950 | 1 | 0 |
N-[2-methyl-5-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamide | Plasmodium falciparum 3D7 | AC50 | 4.1250 | 1 | 0 |
N-[(1,3-dioxo-2-phenyl-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl)methyl]-4-methylbenzenesulfonamide | Plasmodium falciparum 3D7 | AC50 | 4.8030 | 1 | 0 |
calcimycin | Plasmodium falciparum 3D7 | AC50 | 0.8130 | 1 | 0 |
1-(4-fluorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thiourea | Plasmodium falciparum 3D7 | AC50 | 26.2800 | 1 | 0 |
1-(4-methylphenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thiourea | Plasmodium falciparum 3D7 | AC50 | 8.6080 | 1 | 0 |
1-(3-chlorophenyl)-3-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]thiourea | Plasmodium falciparum 3D7 | AC50 | 8.7380 | 1 | 0 |
N-[[2-(4-methylphenyl)-1,3-dioxo-7,7a-dihydro-3aH-octahydro-1H-4,7-epoxyisoindol-4-yl]methyl]-4-phenyl-1-piperazinecarbothioamide | Plasmodium falciparum 3D7 | AC50 | 6.9310 | 1 | 0 |
thimerosal | Plasmodium falciparum 3D7 | AC50 | 4.9010 | 1 | 0 |
4'-epichaetoviridin A | Plasmodium falciparum 3D7 | AC50 | 15.1890 | 1 | 0 |
[5-[(2-methoxyphenoxy)methyl]-3-isoxazolyl]-(4-methyl-3-phenyl-1-piperazinyl)methanone | Plasmodium falciparum 3D7 | AC50 | 3.0480 | 1 | 0 |
LSM-27979 | Plasmodium falciparum 3D7 | AC50 | 0.9880 | 1 | 0 |
6-(3-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Plasmodium falciparum 3D7 | AC50 | 8.1660 | 1 | 0 |
3-hydroxy-2-[5-[4-(trifluoromethyl)phenyl]-2-furanyl]-1,2-dihydroquinazolin-4-one | Plasmodium falciparum 3D7 | AC50 | 7.6160 | 1 | 0 |
4-chloro-N-(5-methyl-1,3,4-oxadiazol-2-yl)-5-dithiazolimine | Plasmodium falciparum 3D7 | AC50 | 1.0310 | 1 | 0 |