Page last updated: 2024-08-07 20:46:40

cAMP-dependent protein kinase catalytic subunit alpha

A cAMP-dependent protein kinase catalytic subunit alpha that is encoded in the genome of mouse. [OMA:P05132, PRO:DNx]

Synonyms

PKA C-alpha;
EC 2.7.11.11

Research

Bioassay Publications (2)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (5)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
fasudilMus musculus (house mouse)Ki0.495012
y 27632Mus musculus (house mouse)Ki2.575012
h 1152Mus musculus (house mouse)Ki0.173012
h 89Mus musculus (house mouse)IC500.381012
ha 1100Mus musculus (house mouse)Ki1.175012

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
h 89Mus musculus (house mouse)Kd0.027012