Proteins > cAMP-dependent protein kinase catalytic subunit alpha
Page last updated: 2024-08-07 20:46:40
cAMP-dependent protein kinase catalytic subunit alpha
A cAMP-dependent protein kinase catalytic subunit alpha that is encoded in the genome of mouse. [OMA:P05132, PRO:DNx]
Synonyms
PKA C-alpha;
EC 2.7.11.11
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (5)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
fasudil | Mus musculus (house mouse) | Ki | 0.4950 | 1 | 2 |
y 27632 | Mus musculus (house mouse) | Ki | 2.5750 | 1 | 2 |
h 1152 | Mus musculus (house mouse) | Ki | 0.1730 | 1 | 2 |
h 89 | Mus musculus (house mouse) | IC50 | 0.3810 | 1 | 2 |
ha 1100 | Mus musculus (house mouse) | Ki | 1.1750 | 1 | 2 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
h 89 | Mus musculus (house mouse) | Kd | 0.0270 | 1 | 2 |