Page last updated: 2024-08-07 12:34:09
hexokinase
[no definition available]
Synonyms
Research
Bioassay Publications (0)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0) | 18.7374 |
1990's | 0 (0) | 18.2507 |
2000's | 0 (0) | 29.6817 |
2010's | 0 (0) | 24.3611 |
2020's | 0 (0) | 2.80 |
Compounds (15)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
thioctic acid | Trypanosoma brucei brucei TREU927 | IC50 | 0.2008 | 1 | 0 |
ebselen | Trypanosoma brucei brucei TREU927 | IC50 | 0.9009 | 1 | 0 |
closantel | Trypanosoma brucei brucei TREU927 | IC50 | 25.0000 | 1 | 0 |
4-methyoxybenzoyl-n-glycine | Trypanosoma brucei brucei TREU927 | IC50 | 25.0000 | 1 | 0 |
2-phenyl-1,2-benzisothiazol-3-(2h)-one | Trypanosoma brucei brucei TREU927 | IC50 | 3.9563 | 2 | 0 |
6-fluoro-2-phenyl-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 2.3100 | 1 | 0 |
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 4.6863 | 2 | 0 |
N,N-dimethyl-3-(3-oxo-1,2-benzothiazol-2-yl)benzenesulfonamide | Trypanosoma brucei brucei TREU927 | IC50 | 7.6300 | 1 | 0 |
quercetin | Trypanosoma brucei brucei TREU927 | IC50 | 22.3780 | 1 | 0 |
2-(4-methoxyphenyl)-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 5.3500 | 1 | 0 |
2-(4-chlorophenyl)-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 1.1000 | 1 | 0 |
2-(3-chlorophenyl)-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 1.9010 | 1 | 0 |
5-fluoro-2-phenyl-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 1.0300 | 1 | 0 |
2-(2-fluorophenyl)-1,2-benzothiazol-3-one | Trypanosoma brucei brucei TREU927 | IC50 | 2.2600 | 1 | 0 |
2-(3-oxo-1,2-benzothiazol-2-yl)-N-phenylacetamide | Trypanosoma brucei brucei TREU927 | IC50 | 6.6900 | 1 | 0 |