Proteins > Estrogen receptor 1
Page last updated: 2024-08-07 15:11:14

Estrogen receptor 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (50)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
bithionolHomo sapiens (human)IC503.940910
gossypolHomo sapiens (human)IC502.551310
hexachloropheneHomo sapiens (human)IC502.161610
nabumetoneHomo sapiens (human)IC5050.000010
masoprocolHomo sapiens (human)IC5022.193710
phenylbutazoneHomo sapiens (human)IC5050.000010
4-fluorobenzamideHomo sapiens (human)IC5050.000010
5-(2-methylthioethyl)hydantoinHomo sapiens (human)IC5050.000010
Benzoic acid, 4-amino-, 4-acetoxy-2,2,6,6-tetramethyl-1-piperidinyl esterHomo sapiens (human)IC5026.347210
2-[[5-[4-(1-piperidinylsulfonyl)phenyl]-1H-1,2,4-triazol-3-yl]thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)IC5047.183010
2-[4-(benzenesulfonyl)phenyl]-5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazoleHomo sapiens (human)IC5050.000010
N-[2-methoxy-4-[[2-[(3-methyl-4-oxo-2-quinazolinyl)thio]-1-oxoethyl]amino]phenyl]-2-furancarboxamideHomo sapiens (human)IC5032.541210
2-(5-amino-1-phenyl-1,2,4-triazol-3-yl)-3a,4,7,7a-tetrahydroisoindole-1,3-dioneHomo sapiens (human)IC5050.000010
(3aR,6aS)-3-(2-chlorophenyl)-5-(2,5-dimethoxyphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dioneHomo sapiens (human)IC509.784910
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamideHomo sapiens (human)IC5050.000010
N-(3-acetylphenyl)-2-thiophen-2-ylacetamideHomo sapiens (human)IC5018.544210
N-cyclohexyl-2-[(8-methoxy-6-oxo-3-benzo[c][1]benzopyranyl)oxy]acetamideHomo sapiens (human)IC5017.894910
3-(3-oxo-2-benzo[f][1]benzopyranyl)-1-phenyl-4-pyrazolecarboxaldehydeHomo sapiens (human)IC5019.621410
cinnarizineHomo sapiens (human)IC5050.000010
N-(9-ethyl-3-carbazolyl)-2-[[4-ethyl-5-(2-furanyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)IC5050.000010
2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]thio]-N-(9-ethyl-3-carbazolyl)acetamideHomo sapiens (human)IC5012.230210
N-(3-dibenzofuranyl)-2-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)thio]acetamideHomo sapiens (human)IC5050.000010
N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)-4-oxo-4-thiophen-2-ylbutanamideHomo sapiens (human)IC507.107510
2-phenoxybenzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterHomo sapiens (human)IC5017.914510
2-[[2-(4-ethyl-4-methyl-2,5-dioxo-1-imidazolidinyl)-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideHomo sapiens (human)IC5018.237010
7-[[[1-(3-methylphenyl)-2-benzimidazolyl]thio]methyl]-5-thiazolo[3,2-a]pyrimidinoneHomo sapiens (human)IC5050.000010
5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylic acid [2-[(1,1-dioxo-3-thiolanyl)-(2-methylpropyl)amino]-2-oxoethyl] esterHomo sapiens (human)IC502.947610
3-[(4-methylphenyl)sulfamoyl]benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] esterHomo sapiens (human)IC5030.606710
N-(5-chloro-2-methoxyphenyl)-2,4-dimethyl-5-oxazolecarboxamideHomo sapiens (human)IC5050.000010
5-hydroxy-2-methyl-4-[1-piperidinyl(3-pyridinyl)methyl]-3-benzo[g]benzofurancarboxylic acid ethyl esterHomo sapiens (human)IC5050.000010
2-[(4-methyl-5-sulfanylidene-1,3,4-thiadiazol-2-yl)thio]acetic acid ethyl esterHomo sapiens (human)IC507.983210
2-cyclopentylacetic acid [2-[(3-chloro-9,10-dioxo-2-anthracenyl)amino]-2-oxoethyl] esterHomo sapiens (human)IC5022.253410
6-(2,3-dihydro-1,4-benzodioxin-3-yl)-3-(phenoxymethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)IC509.549810
molsidomineHomo sapiens (human)IC5024.673910
1-(3-amino-7-methoxy-1-pyrazolo[3,4-b]quinolinyl)-2-(4-chlorophenyl)ethanoneHomo sapiens (human)IC5024.783310
4-[[2-[(6-methyl-4-oxo-1H-pyrimidin-2-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)IC503.062610

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
eedqHomo sapiens (human)EC509,999.000010
6-ketoestradiolHomo sapiens (human)EC5012.520610
2-[3-[3-[3-(1-imidazolyl)propyl]-4-oxo-2-quinazolinyl]propyl]isoindole-1,3-dioneHomo sapiens (human)EC5023.489510
N-[1-[(4-methylphenyl)methyl]-2-benzimidazolyl]-2-furancarboxamideHomo sapiens (human)EC5014.567110
diethylstilbestrol dipropionateHomo sapiens (human)EC5018.131410
dienestrolHomo sapiens (human)EC5013.241510
N-(4,5-diphenyl-2-oxazolyl)-2-[(1-methyl-5-tetrazolyl)thio]acetamideHomo sapiens (human)EC5022.243910
2-[[3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-2-thieno[3,2-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)EC5012.756710
4-morpholinecarboxylic acid [3-(6-amino-5-cyano-3-ethyl-2,4-dihydropyrano[2,3-c]pyrazol-4-yl)phenyl] esterHomo sapiens (human)EC506.386710
2-[[2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]-1-oxo-5-isoquinolinyl]oxy]propanoic acid ethyl esterHomo sapiens (human)EC5012.613810
5-(4-fluorophenyl)-7-(3-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineHomo sapiens (human)EC506.709310
6alpha-hydroxy-17beta-estradiolHomo sapiens (human)EC5012.661310
2-[[4-(2,3-dimethylphenyl)-1-piperazinyl]-oxomethyl]-1,5-dimethyl-4-pyrrolo[3,2-c]quinolinoneHomo sapiens (human)EC5012.762210
beta-zearalenolHomo sapiens (human)EC509.219910