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Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform

A phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform that is encoded in the genome of cow. [OMA:P32871, PRO:DNx]

Synonyms

PI3-kinase subunit alpha;
PI3K-alpha;
PI3Kalpha;
PtdIns-3-kinase subunit alpha;
EC 2.7.1.137;
EC 2.7.1.153;
Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha;
PtdIns-3-kinase subunit p110-alpha;

Research

Bioassay Publications (3)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (1)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-oneBos taurus (cattle)IC503.753333