Proteins > neuropeptide S receptor isoform A
Page last updated: 2024-08-07 15:20:55

neuropeptide S receptor isoform A

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (1298)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
gamma-aminobutyric acidHomo sapiens (human)Potency31.622810
n-acetylserotoninHomo sapiens (human)Potency10.000010
quinolinic acidHomo sapiens (human)Potency1.000010
vanilmandelic acidHomo sapiens (human)Potency3.981110
pk 11195Homo sapiens (human)Potency0.199510
3,4-dichloroisocoumarinHomo sapiens (human)Potency12.589310
phaclofenHomo sapiens (human)Potency0.031610
cgp 52411Homo sapiens (human)Potency12.589310
4-amino-1,8-naphthalimideHomo sapiens (human)Potency5.011910
4-phenyl-3-furoxancarbonitrileHomo sapiens (human)Potency25.118910
hydroxyindoleacetic acidHomo sapiens (human)Potency3.162310
6-hydroxymelatoninHomo sapiens (human)Potency10.000010
7-nitroindazoleHomo sapiens (human)Potency25.118910
8-phenyltheophyllineHomo sapiens (human)Potency0.251210
aa 861Homo sapiens (human)Potency15.848910
tyrphostin 25Homo sapiens (human)Potency3.162310
tyrphostin a1Homo sapiens (human)Potency12.589310
albendazoleHomo sapiens (human)Potency25.118910
am 251Homo sapiens (human)Potency10.000010
amoxapineHomo sapiens (human)Potency31.622810
bay-k-8644Homo sapiens (human)Potency0.631010
bay h 4502Homo sapiens (human)Potency15.848910
bumetanideHomo sapiens (human)Potency3.162310
chlorpropamideHomo sapiens (human)Potency5.011910
chlorzoxazoneHomo sapiens (human)Potency25.118910
cilostazolHomo sapiens (human)Potency19.952610
clotrimazoleHomo sapiens (human)Potency6.477610
dipyridamoleHomo sapiens (human)Potency10.496130
disulfiramHomo sapiens (human)Potency19.783010
2-amino-7-phosphonoheptanoic acidHomo sapiens (human)Potency31.622810
racemetirosineHomo sapiens (human)Potency25.118910
ebselenHomo sapiens (human)Potency10.000010
ellipticineHomo sapiens (human)Potency10.000010
ethacrynic acidHomo sapiens (human)Potency12.589310
ethosuximideHomo sapiens (human)Potency25.118910
felbamateHomo sapiens (human)Potency0.794310
felodipineHomo sapiens (human)Potency11.294710
fenofibrateHomo sapiens (human)Potency15.848910
fluspirileneHomo sapiens (human)Potency10.266310
acetic acid (3-ethenyl-6,10,10b-trihydroxy-3,4a,7,7,10a-pentamethyl-1-oxo-5,6,6a,8,9,10-hexahydro-2H-benzo[f][1]benzopyran-5-yl) esterHomo sapiens (human)Potency0.794310
fpl 64176Homo sapiens (human)Potency5.011910
gossypolHomo sapiens (human)Potency12.589310
ibudilastHomo sapiens (human)Potency12.589310
indomethacinHomo sapiens (human)Potency1.584910
isradipineHomo sapiens (human)Potency12.589310
jl 18Homo sapiens (human)Potency12.589310
beta-lapachoneHomo sapiens (human)Potency3.162310
leflunomideHomo sapiens (human)Potency0.079410
loratadineHomo sapiens (human)Potency8.171210
mequitazineHomo sapiens (human)Potency12.589310
nocodazoleHomo sapiens (human)Potency1.000010
ethylmaleimideHomo sapiens (human)Potency5.011910
apneaHomo sapiens (human)Potency0.398110
nilutamideHomo sapiens (human)Potency25.118910
nimodipineHomo sapiens (human)Potency1.584910
norfloxacinHomo sapiens (human)Potency5.011910
ns 1619Homo sapiens (human)Potency3.981110
pd 169316Homo sapiens (human)Potency7.943310
perphenazineHomo sapiens (human)Potency17.559410
phenylbutazoneHomo sapiens (human)Potency0.316210
pinacidilHomo sapiens (human)Potency5.011910
praziquantelHomo sapiens (human)Potency6.309610
prochlorperazineHomo sapiens (human)Potency25.118910
protoporphyrin ixHomo sapiens (human)Potency10.000010
pf 5901Homo sapiens (human)Potency12.589310
ritanserinHomo sapiens (human)Potency10.226910
sq 22536Homo sapiens (human)Potency0.000810
sulfaphenazoleHomo sapiens (human)Potency3.162310
terfenadineHomo sapiens (human)Potency12.589310
thiramHomo sapiens (human)Potency0.108430
ici 136,753Homo sapiens (human)Potency15.848910
tyrphostin a9Homo sapiens (human)Potency6.309610
ici 204,219Homo sapiens (human)Potency10.000010
reserpineHomo sapiens (human)Potency10.000010
procaine hydrochlorideHomo sapiens (human)Potency5.011910
promazine hydrochlorideHomo sapiens (human)Potency10.000010
triiodothyronineHomo sapiens (human)Potency0.794320
racepinephrine hydrochlorideHomo sapiens (human)Potency3.162310
papaverine hydrochlorideHomo sapiens (human)Potency19.952610
methylene blueHomo sapiens (human)Potency3.182430
androstenedioneHomo sapiens (human)Potency0.251210
colchicineHomo sapiens (human)Potency2.511910
quinacrine monohydrochlorideHomo sapiens (human)Potency10.000010
chlorpromazine hydrochlorideHomo sapiens (human)Potency18.854110
cytarabine hydrochlorideHomo sapiens (human)Potency19.952610
medroxyprogesterone acetateHomo sapiens (human)Potency2.511910
azovioletHomo sapiens (human)Potency3.927530
sulfachlorpyridazineHomo sapiens (human)Potency15.848910
rotenoneHomo sapiens (human)Potency12.589310
9,10-phenanthrenequinoneHomo sapiens (human)Potency3.162310
1-(2-pyridylazo)-2-naphtholHomo sapiens (human)Potency7.943310
neostigmine bromideHomo sapiens (human)Potency5.011910
methapyrilene hydrochlorideHomo sapiens (human)Potency25.118910
catechinHomo sapiens (human)Potency31.622810
chlormadinone acetateHomo sapiens (human)Potency5.011910
orphenadrine hydrochlorideHomo sapiens (human)Potency0.020010
dequalinium chlorideHomo sapiens (human)Potency12.589310
chlorotrianiseneHomo sapiens (human)Potency7.943310
megestrol acetateHomo sapiens (human)Potency3.571710
2,2'-diaminodiphenyldisulfideHomo sapiens (human)Potency25.118910
flurandrenoloneHomo sapiens (human)Potency0.316210
5-hydroxyindoleHomo sapiens (human)Potency5.011910
pimozideHomo sapiens (human)Potency9.449410
nsc 3852Homo sapiens (human)Potency10.000010
clonidine hydrochlorideHomo sapiens (human)Potency15.848910
1,6-bismaleimidohexaneHomo sapiens (human)Potency12.589310
propionylpromazine hydrochlorideHomo sapiens (human)Potency12.589310
benserazide hydrochlorideHomo sapiens (human)Potency5.011910
thymolphthaleinHomo sapiens (human)Potency10.000010
clobetasol propionateHomo sapiens (human)Potency5.287150
isovelleralHomo sapiens (human)Potency12.589310
lonidamineHomo sapiens (human)Potency3.162310
iem 611Homo sapiens (human)Potency15.848910
flecainide acetateHomo sapiens (human)Potency0.631010
nicardipine hydrochlorideHomo sapiens (human)Potency7.506010
nitazoxanideHomo sapiens (human)Potency3.162310
s-2678Homo sapiens (human)Potency10.000010
cerm-1978Homo sapiens (human)Potency10.000010
triclabendazoleHomo sapiens (human)Potency12.589310
mitoxantrone hydrochlorideHomo sapiens (human)Potency10.000010
chaetochrominHomo sapiens (human)Potency10.000010
enoximoneHomo sapiens (human)Potency31.622810
raloxifene hydrochlorideHomo sapiens (human)Potency15.848910
nefazodone hydrochlorideHomo sapiens (human)Potency12.589310
mifepristoneHomo sapiens (human)Potency12.589310
mibefradil dihydrochlorideHomo sapiens (human)Potency10.000010
eliprodilHomo sapiens (human)Potency31.622810
aripiprazoleHomo sapiens (human)Potency12.589310
daunorubicin hydrochlorideHomo sapiens (human)Potency7.943310
verapamil hydrochlorideHomo sapiens (human)Potency12.589310
src-820 rHomo sapiens (human)Potency25.118910
efavirenzHomo sapiens (human)Potency10.000010
mevastatinHomo sapiens (human)Potency15.848910
desipramine hydrochlorideHomo sapiens (human)Potency12.589310
ticlopidine hydrochlorideHomo sapiens (human)Potency12.589310
proadifen hydrochlorideHomo sapiens (human)Potency2.511910
sulconazole, mononitrate, (+-)-isomerHomo sapiens (human)Potency15.848910
telmisartanHomo sapiens (human)Potency1.258910
thioridazine hydrochlorideHomo sapiens (human)Potency12.589310
trifluoperazine hydrochlorideHomo sapiens (human)Potency12.589310
siquilHomo sapiens (human)Potency12.589310
oxymetazoline hydrochlorideHomo sapiens (human)Potency3.981110
toxoflavinHomo sapiens (human)Potency0.333530
fluphenazine hydrochlorideHomo sapiens (human)Potency10.000010
clomipramine hydrochlorideHomo sapiens (human)Potency6.309610
miconazole nitrateHomo sapiens (human)Potency10.000010
econazole nitrateHomo sapiens (human)Potency12.589310
sanguinarine chlorideHomo sapiens (human)Potency25.118910
5-aminovaleric acid hydrochlorideHomo sapiens (human)Potency15.848910
ranolazine hydrochlorideHomo sapiens (human)Potency25.118920
clobetasone butyrateHomo sapiens (human)Potency3.162310
loperamide hydrochlorideHomo sapiens (human)Potency10.000010
siguazodanHomo sapiens (human)Potency3.981110
3-octadecanamido-2-ethoxypropylphosphocholineHomo sapiens (human)Potency8.402830
magnololHomo sapiens (human)Potency12.589310
chelerythrine chlorideHomo sapiens (human)Potency19.952610
9-methoxyellipticineHomo sapiens (human)Potency10.000010
5-(n-methyl-n-isobutyl)amilorideHomo sapiens (human)Potency19.952610
ergocornineHomo sapiens (human)Potency1.796450
4-(2-thiazolylazo)resorcinolHomo sapiens (human)Potency1.258910
3,5-di-tert-butyl-1,2-benzoquinoneHomo sapiens (human)Potency12.589310
2-methyl-4-nitroquinoline 1-oxideHomo sapiens (human)Potency10.000010
2-(1H-benzimidazol-2-yl)anilineHomo sapiens (human)Potency1.584910
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)Potency10.000010
2-butyl-6-(butylamino)-1h-benzo(de)isoquinoline-1,3(2h)-dioneHomo sapiens (human)Potency10.000010
oxybutynin hydrochlorideHomo sapiens (human)Potency10.000010
diflufenicanHomo sapiens (human)Potency10.000010
hexamethonium chlorideHomo sapiens (human)Potency19.952610
1-(2-thiazolylazo)-2-naphtholHomo sapiens (human)Potency15.848910
coumarin 7Homo sapiens (human)Potency12.589310
diffractaic acidHomo sapiens (human)Potency10.000010
osajinHomo sapiens (human)Potency10.000010
5-nitro-2-(1-piperidinyl)pyridineHomo sapiens (human)Potency25.118910
zpckHomo sapiens (human)Potency25.118910
diphyllinHomo sapiens (human)Potency10.000010
7-amino-4-trifluoromethylcoumarinHomo sapiens (human)Potency12.589310
cp-55,940Homo sapiens (human)Potency12.589310
vanoxerineHomo sapiens (human)Potency12.589310
paxillineHomo sapiens (human)Potency10.000010
u 78517fHomo sapiens (human)Potency25.118910
beta-carboline-3-carboxylic acid methyl esterHomo sapiens (human)Potency31.622810
methoctramineHomo sapiens (human)Potency12.589310
6-hydroxydopaHomo sapiens (human)Potency5.011910
dihydrocapsaicinHomo sapiens (human)Potency12.589310
gr 113808Homo sapiens (human)Potency0.251210
gallopamil hydrochlorideHomo sapiens (human)Potency19.952610
sb 204070aHomo sapiens (human)Potency0.025110
tetradecanoylphorbol acetateHomo sapiens (human)Potency6.309610
w 7Homo sapiens (human)Potency10.000010
ici 204448Homo sapiens (human)Potency31.622810
n-(6-methoxy-8-quinolyl)-4-toluenesulfonamideHomo sapiens (human)Potency3.981110
purpactin aHomo sapiens (human)Potency12.589310
n,n-di-n-hexyl-2-(4-fluorophenyl)indole-3-acetamideHomo sapiens (human)Potency10.000010
3,5-bis(trifluoromethyl)benzyl n-acetyltryptophanHomo sapiens (human)Potency1.584910
8-cyclopentyl-3-(3-((4-(fluorosulfonyl)benzoyl)oxy)propyl)-1-propylxanthineHomo sapiens (human)Potency6.309610
nsc-141549Homo sapiens (human)Potency10.000010
ezetimibeHomo sapiens (human)Potency5.011910
idazoxan hydrochlorideHomo sapiens (human)Potency10.000010
sch 45752Homo sapiens (human)Potency10.000010
cryptotanshinoneHomo sapiens (human)Potency25.118910
Serotonin hydrochlorideHomo sapiens (human)Potency31.622810
epiberberineHomo sapiens (human)Potency12.589310
2-phenyl-4-oxohydroquinolineHomo sapiens (human)Potency25.118910
3,3-bis(4-hydroxy-3-methylphenyl)-1H-indol-2-oneHomo sapiens (human)Potency10.000010
2,4-dinitropyrimidinyl-2-thiophenolHomo sapiens (human)Potency25.118910
enniatin bHomo sapiens (human)Potency10.000010
2-phenyl-1,2-benzisothiazol-3-(2h)-oneHomo sapiens (human)Potency7.943310
17 alpha-hydroxyprogesterone caproateHomo sapiens (human)Potency10.000010
abt 980Homo sapiens (human)Potency10.000010
2,10,11-trihydroxy-n-n-propylnoraporphineHomo sapiens (human)Potency10.000010
nbi 27914Homo sapiens (human)Potency12.589310
memantine hydrochlorideHomo sapiens (human)Potency5.011910
2,6,7,8-tetrahydrocyclopenta[2,3]thieno[2,4-d]pyrimidin-1-oneHomo sapiens (human)Potency15.848910
1H-indol-3-yl-(4-methoxyphenyl)methanoneHomo sapiens (human)Potency12.589310
1,1,3,3-tetraphenylureaHomo sapiens (human)Potency10.000010
vacquinol-1Homo sapiens (human)Potency10.000010
gossypol acetic acidHomo sapiens (human)Potency12.589310
n-methylserotonin oxalate saltHomo sapiens (human)Potency0.398110
nsc 95397Homo sapiens (human)Potency12.589310
methylnaphthazarinHomo sapiens (human)Potency5.011910
dimethyl 2-(2-nitrobenzylidene)malonateHomo sapiens (human)Potency7.943310
(1-tert-butyl-5-phenyl-3-pyrrolyl)-phenylmethanoneHomo sapiens (human)Potency12.589310
nsc228155Homo sapiens (human)Potency1.584910
2-methyl-3-(phenylmethylthio)-1H-indoleHomo sapiens (human)Potency25.118910
(3-chloro-1-benzothiophen-2-yl)-[2-(2-chloro-6-methylphenyl)imino-4-methylene-3-thia-1-azaspiro[4.5]decan-1-yl]methanoneHomo sapiens (human)Potency10.000010
1-(2,6-dichlorophenyl)-3-(6-methyl-3-pyridinyl)ureaHomo sapiens (human)Potency12.589310
N-(2,6-dibromo-4-methylphenyl)-3-(2,6-dichlorophenyl)-5-methyl-4-isoxazolecarboxamideHomo sapiens (human)Potency10.000010
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneHomo sapiens (human)Potency6.309610
7-benzoyl-3-chloroindolizine-1,2-dicarboxylic acid dimethyl esterHomo sapiens (human)Potency12.589310
2,2'-spirobi[3,6,7,8-tetrahydro-1H-cyclopenta[g]naphthalene]-5,5'-dioneHomo sapiens (human)Potency12.589310
ritonavirHomo sapiens (human)Potency12.589310
5-hydroxytryptophanHomo sapiens (human)Potency3.981110
tosylphenylalanyl chloromethyl ketoneHomo sapiens (human)Potency16.271010
amiodarone hydrochlorideHomo sapiens (human)Potency11.294710
dicyclomine hydrochlorideHomo sapiens (human)Potency25.118910
nortriptyline hydrochlorideHomo sapiens (human)Potency0.079410
N-(3-Benzooxazol-2-yl-4-hydroxy-phenyl)-2-p-tolyloxyacetamideHomo sapiens (human)Potency12.589310
3,5-dihydroxyphenylglycineHomo sapiens (human)Potency0.398110
actinoninHomo sapiens (human)Potency31.622810
difluprednateHomo sapiens (human)Potency2.511910
doxorubicin hydrochlorideHomo sapiens (human)Potency0.631010
amcinonideHomo sapiens (human)Potency3.981110
dihydroergocristine monomesylateHomo sapiens (human)Potency8.399150
brivudineHomo sapiens (human)Potency25.118910
5,11-diethyl-5,6,11,12-tetrahydrochrysene-2,8-diolHomo sapiens (human)Potency10.000010
diethylstilbestrolHomo sapiens (human)Potency12.589310
6-bromoindirubin-3'-oximeHomo sapiens (human)Potency10.000010
afimoxifeneHomo sapiens (human)Potency10.000010
ketoconazoleHomo sapiens (human)Potency12.589310
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency1.995310
moronic acidHomo sapiens (human)Potency10.000010
6-methyl-2-[(4-nitrophenyl)methylthio]-1H-benzimidazoleHomo sapiens (human)Potency12.589310
N1-(2,3-dihydro-1,4-benzodioxin-6-yl)acetamideHomo sapiens (human)Potency25.118910
edulineHomo sapiens (human)Potency0.004010
5-(4-nitrophenyl)-4-phenyl-2-thiazolamineHomo sapiens (human)Potency3.162310
isoliquiritigeninHomo sapiens (human)Potency31.622810
cardamoninHomo sapiens (human)Potency12.589310
calmidazoliumHomo sapiens (human)Potency12.589310
N-[(8-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-oxolanylmethyl)-2-furancarboxamideHomo sapiens (human)Potency19.952610
3-[[1,3-benzodioxol-5-ylmethyl-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency12.589310
N-[2-(cyclopentylamino)-1-(5-methyl-2-furanyl)-2-oxoethyl]-N-[(4-fluorophenyl)methyl]-4-thiadiazolecarboxamideHomo sapiens (human)Potency25.118910
1-[2,5-diethoxy-4-(1-tetrazolyl)phenyl]sulfonyl-4-(4-fluorophenyl)-3,6-dihydro-2H-pyridineHomo sapiens (human)Potency10.000010
LSM-19079Homo sapiens (human)Potency15.848910
n-2-fluorenesulfonyl-beta-alanineHomo sapiens (human)Potency0.010010
2-[[2-(1-benzotriazolyl)-1-oxoethyl]-(thiophen-2-ylmethyl)amino]-2-(2-furanyl)-N-(3-methylbutyl)acetamideHomo sapiens (human)Potency12.589310
2-[[3-(1H-benzimidazol-2-yl)-2-pyridinyl]thio]acetic acid methyl esterHomo sapiens (human)Potency5.011910
1-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-4-(2,3-dimethylphenyl)piperazineHomo sapiens (human)Potency10.000010
2-[[2-[[4-(2-furanylmethyl)-5-(phenylmethyl)-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideHomo sapiens (human)Potency12.589310
6-[[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]quinolineHomo sapiens (human)Potency7.943310
2-methoxy-N-[6-(1-oxobutylamino)-3-pyridinyl]benzamideHomo sapiens (human)Potency25.118910
N-[1-[(4-methylphenyl)methyl]-2-benzimidazolyl]-2-furancarboxamideHomo sapiens (human)Potency3.162310
4-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-2-methyl-5-thieno[3,2-b]pyrrolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
3-[[2-(1-benzotriazolyl)-1-oxoethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency6.309610
2-[[2-[(1-cyclohexyl-5-tetrazolyl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency12.589310
3-[(1-tert-butyl-5-tetrazolyl)-[2-furanylmethyl(2-oxolanylmethyl)amino]methyl]-6-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
2-(2-ethyl-6-methyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(5-methyl-2-furanyl)methyl]-N-(3-pyridinylmethyl)acetamideHomo sapiens (human)Potency6.309610
3-[[1,3-benzodioxol-5-ylmethyl-[(1-cyclopentyl-5-tetrazolyl)methyl]amino]methyl]-6-ethyl-1H-quinolin-2-oneHomo sapiens (human)Potency25.118910
1-(1-adamantyl)-3-[8-[[1-(2-furanylmethyl)-5-tetrazolyl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]ureaHomo sapiens (human)Potency10.000010
1-(4-chlorophenyl)sulfonyl-N-[3-methoxy-4-(1-tetrazolyl)phenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency0.501210
6-ethyl-3-[[[1-(2-furanylmethyl)-5-tetrazolyl]methyl-(phenylmethyl)amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency12.589310
N-[2-methyl-4-oxo-3-(phenylmethyl)-7-(1-piperidinyl)-6-quinazolinyl]-3-pyridinecarboxamideHomo sapiens (human)Potency10.000010
3-[[[1-[1-(2-furanylmethyl)-5-tetrazolyl]-2-methylpropyl]-(2-oxolanylmethyl)amino]methyl]-8-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency0.631010
N-(3-ethoxyphenyl)-1-(4-methoxyphenyl)sulfonyl-3-piperidinecarboxamideHomo sapiens (human)Potency25.118910
1-methyl-2-[(4-methyl-1-piperidinyl)methyl]-3-indolecarbonitrileHomo sapiens (human)Potency12.589310
2-[5-[4-(dimethylamino)phenyl]-2-tetrazolyl]-N-[2-(4-morpholinyl)phenyl]acetamideHomo sapiens (human)Potency25.118910
6-methyl-3-[[[1-(phenylmethyl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
2-[(1-tert-butyl-5-tetrazolyl)-thiophen-2-ylmethyl]-2-azaspiro[5.5]undecaneHomo sapiens (human)Potency12.589310
1-[1-(1-cyclopentyl-5-tetrazolyl)-2-methylpropyl]-4-(2-fluorophenyl)piperazineHomo sapiens (human)Potency10.000010
N-tert-butyl-2-[[5-(3,5-dimethoxyphenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(phenylmethyl)acetamideHomo sapiens (human)Potency10.000010
3-[[[1-(2-furanylmethyl)-5-tetrazolyl]methyl-[(2-methoxyphenyl)methyl]amino]methyl]-6-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
3-[(1-cyclopentyl-5-tetrazolyl)-[4-(2-methoxyphenyl)-1-piperazinyl]methyl]-7-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency0.794310
4-[4-methyl-6-(4-methyl-1-piperazinyl)-2-pyrimidinyl]morpholineHomo sapiens (human)Potency25.118910
2-[[3-cyano-6-(2-furanyl)-4-(trifluoromethyl)-2-pyridinyl]thio]propanoic acid ethyl esterHomo sapiens (human)Potency12.589310
5-[(5-methoxycarbonyl-2-methyl-3-furanyl)methoxy]-2-methyl-3-benzofurancarboxylic acid 2-methoxyethyl esterHomo sapiens (human)Potency19.952610
4-methyl-N-[2-[4-(2-methyl-1-oxopropyl)-1-piperazinyl]phenyl]benzamideHomo sapiens (human)Potency10.000010
N-tert-butyl-2-(2-furanyl)-2-[[2-[5-(5-methyl-2-furanyl)-2-tetrazolyl]-1-oxoethyl]-(thiophen-2-ylmethyl)amino]acetamideHomo sapiens (human)Potency5.011910
[5-(2-furanyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency12.589310
N'-[1-[(cyclohexylamino)-oxomethyl]cyclopentyl]-N-(5-methyl-3-isoxazolyl)-N'-phenylbutanediamideHomo sapiens (human)Potency12.589310
6-(4-hydroxy-3-methoxyphenyl)-4-methoxy-1,3-dimethyl-8-cyclohepta[c]furanoneHomo sapiens (human)Potency19.952610
2-[4-[(1-cyclopentyl-5-tetrazolyl)-(6-quinolinyl)methyl]-1-piperazinyl]-1,3-benzothiazoleHomo sapiens (human)Potency3.981110
3-[[[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl-(2-hydroxyethyl)amino]methyl]-7-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency3.162310
N-(1,3-benzodioxol-5-yl)-1-[4-(4-morpholinylsulfonyl)phenyl]-4-piperidinecarboxamideHomo sapiens (human)Potency25.118910
N-(4-chlorophenyl)-4-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-1-piperidinecarboxamideHomo sapiens (human)Potency15.848910
5-cyano-6-[[2-(2,3-dimethylanilino)-2-oxoethyl]thio]-4-(2-furanyl)-2-methyl-N-phenyl-1,4-dihydropyridine-3-carboxamideHomo sapiens (human)Potency12.589310
2-[[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency12.589310
2-[(1,3-dimethyl-2,6-dioxo-7-propyl-8-purinyl)thio]-N-[2-(1-piperidinyl)phenyl]acetamideHomo sapiens (human)Potency10.000010
2-[[2-(1-azepanyl)-2-oxoethyl]thio]-6-methoxy-3-quinolinecarbonitrileHomo sapiens (human)Potency10.000010
6-methoxy-3-[[2-oxolanylmethyl-[1-[1-(phenylmethyl)-5-tetrazolyl]propyl]amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
2-[[2-(1-benzotriazolyl)-1-oxoethyl]-(2-furanylmethyl)amino]-N-cyclohexyl-2-(2-fluorophenyl)acetamideHomo sapiens (human)Potency10.000010
N-[1-[4-(4-methylphenyl)-2-thiazolyl]-4-piperidinyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamideHomo sapiens (human)Potency25.118910
6-chloro-2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-piperidinyl]-1H-benzimidazoleHomo sapiens (human)Potency6.309610
2-[2-(ethylthio)-1-benzimidazolyl]-1-(1-piperidinyl)ethanoneHomo sapiens (human)Potency5.011910
4-bromo-N-[(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(2-hydroxyethyl)benzamideHomo sapiens (human)Potency10.000010
N-(4-methylphenyl)-2-(3-oxo-5,6-dihydroimidazo[2,1-b]thiazol-2-yl)acetamideHomo sapiens (human)Potency0.199510
2-[(2,3-dimethyl-7,8,9,10-tetrahydrophenanthridin-6-yl)thio]-N-(4-methyl-1,2,5-oxadiazol-3-yl)acetamideHomo sapiens (human)Potency7.943310
6-ethoxy-3-[[[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
2-[[5-(phenoxymethyl)-4-(2-phenylethyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency12.589310
2-[[5-(6-methyl-1H-benzimidazol-2-yl)-2-pyridinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamideHomo sapiens (human)Potency12.589310
3-(2-chlorophenyl)-1-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-[2-(1-pyrrolidinyl)ethyl]ureaHomo sapiens (human)Potency15.848910
2-[(2-ethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency25.118910
1-cyclopentyl-1-[(7-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-3-(2-methoxyphenyl)ureaHomo sapiens (human)Potency12.589310
7-(2-methyl-2,3-dihydroindol-1-yl)-3-(phenylmethyl)triazolo[4,5-d]pyrimidineHomo sapiens (human)Potency10.000010
1-(4-chlorophenyl)-N-(2-furanylmethyl)-N-[[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]methanamineHomo sapiens (human)Potency10.000010
[4-[5-tert-butyl-3-[(2-chlorophenyl)methyl]-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency10.000010
3-[[(1-tert-butyl-5-tetrazolyl)methyl-(thiophen-2-ylmethyl)amino]methyl]-6-ethoxy-1H-quinolin-2-oneHomo sapiens (human)Potency15.848910
1-[1-[[1-[(4-methylphenyl)methyl]-5-tetrazolyl]methyl]-4-piperidinyl]-5-(trifluoromethyl)benzotriazoleHomo sapiens (human)Potency10.000010
N-(2-furanylmethyl)-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]benzamideHomo sapiens (human)Potency10.000010
[4-[2-(3-chlorophenyl)-5-methyl-7-pyrazolo[1,5-a]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency12.589310
2-[(2-cyclohexyl-4-quinazolinyl)thio]-N-(4-methyl-1,2,5-oxadiazol-3-yl)acetamideHomo sapiens (human)Potency12.589310
2-[(5,6-dimethyl-4-oxo-3-phenyl-2-thieno[2,3-d]pyrimidinyl)thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency25.118910
4-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5-furo[3,2-b]pyrrolecarboxylic acid ethyl esterHomo sapiens (human)Potency19.952610
3-[[cyclopentyl-[[1-[(4-methoxyphenyl)methyl]-5-tetrazolyl]methyl]amino]methyl]-7-methyl-1H-quinolin-2-oneHomo sapiens (human)Potency7.943310
3-cyclohexyl-1-[(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-[3-(4-morpholinyl)propyl]ureaHomo sapiens (human)Potency0.501210
N-[(1-cyclohexyl-5-tetrazolyl)-thiophen-2-ylmethyl]-N-(phenylmethyl)ethanamineHomo sapiens (human)Potency10.000010
2-(2-cyanophenoxy)-N-[2-[cyclopropyl(oxo)methyl]-3-benzofuranyl]acetamideHomo sapiens (human)Potency12.589310
4-[2-(4-fluorophenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]morpholineHomo sapiens (human)Potency10.000010
N-(3-methoxyphenyl)-1-[4-(1-tetrazolyl)phenyl]sulfonyl-3-piperidinecarboxamideHomo sapiens (human)Potency3.162310
6-[(2-fluorophenyl)methyl]-2,4-dimethyl-5-thieno[3,4]pyrrolo[1,3-d]pyridazinoneHomo sapiens (human)Potency25.118910
1-phenyl-4-[[1-(phenylmethyl)-5-tetrazolyl]-(3-pyridinyl)methyl]piperazineHomo sapiens (human)Potency10.000010
3-[[1-[1-(2-furanylmethyl)-5-tetrazolyl]propyl-(2-phenylethyl)amino]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Potency10.000010
1-[(5,8-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]-1-(2-furanylmethyl)-3-phenylureaHomo sapiens (human)Potency0.100010
N-(2-furanylmethyl)-N-[(7-methyl-4-tetrazolo[1,5-a]quinolinyl)methyl]-2-phenoxyacetamideHomo sapiens (human)Potency12.589310
2-[[6-(3,4-dimethoxyphenyl)-3-pyridazinyl]thio]-1-(4-morpholinyl)ethanoneHomo sapiens (human)Potency25.118910
3-[[[[3-[(4-chlorophenyl)methyl]-2-methyl-4-oxo-6-quinazolinyl]amino]-oxomethyl]amino]propanoic acid ethyl esterHomo sapiens (human)Potency12.589310
4-amino-N5-[1-(2-furanyl)-2-(3-methylbutylamino)-2-oxoethyl]-N5-(2-methoxyphenyl)isothiazole-3,5-dicarboxamideHomo sapiens (human)Potency15.848910
3-(4-methoxyphenyl)-8-(6-methyl-2-phenyl-4-pyrimidinyl)-8-azabicyclo[3.2.1]octan-3-olHomo sapiens (human)Potency10.000010
(6-fluoro-2-methyl-3,4-dihydro-2H-quinolin-1-yl)-[5-(2-furanyl)-7-(trifluoromethyl)-2-pyrazolo[1,5-a]pyrimidinyl]methanoneHomo sapiens (human)Potency10.000010
4-(2,4-dimethyl-5-thiazolyl)-N-(phenylmethyl)-2-thiazolamineHomo sapiens (human)Potency15.848910
2-[[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]thio]-3-ethyl-4-quinazolinoneHomo sapiens (human)Potency7.943310
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-N-(thiophen-2-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamideHomo sapiens (human)Potency7.943310
4-[[4-(1,3-benzothiazol-2-yl)-1-piperazinyl]-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-2-methoxyphenolHomo sapiens (human)Potency0.501210
1-(4,6-dimethyl-2-pyrimidinyl)-4-piperidinecarboxylic acidHomo sapiens (human)Potency10.000010
4-chloro-N-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl]-N-(2-oxolanylmethyl)benzenesulfonamideHomo sapiens (human)Potency25.118910
1-[(3,4-dimethoxyphenyl)-[1-(thiophen-2-ylmethyl)-5-tetrazolyl]methyl]-4-phenylpiperazineHomo sapiens (human)Potency12.589310
N-(3,4-dimethylphenyl)-2-[[5-[[(4,6-dimethyl-2-pyrimidinyl)thio]methyl]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency12.589310
3-[[4-(1-benzotriazolyl)-1-piperidinyl]sulfonyl]-N-cyclopentylbenzenesulfonamideHomo sapiens (human)Potency7.943310
1-(4-chlorophenyl)-2-[[4-ethyl-5-(2-methyl-3-furanyl)-1,2,4-triazol-3-yl]thio]ethanoneHomo sapiens (human)Potency10.000010
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideHomo sapiens (human)Potency10.000010
(1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanolHomo sapiens (human)Potency10.000010
2-[[3-cyano-4-(5-methyl-2-furanyl)-5,6,7,8-tetrahydroquinolin-2-yl]thio]acetic acid methyl esterHomo sapiens (human)Potency10.000010
2-[(7-methyl-4-oxo-3-phenyl-6,8-dihydro-5H-pyrido[2,3]thieno[2,4-b]pyrimidin-2-yl)thio]acetic acid methyl esterHomo sapiens (human)Potency1.000010
8-(2-furanyl)-6-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]-3,3-dimethyl-1,4-dihydrothiopyrano[3,4-c]pyridine-5-carbonitrileHomo sapiens (human)Potency10.000010
2-amino-3-cyano-7-(dimethylamino)-4-(3-methoxy-4,5-methylenedioxyphenyl)-4h-chromeneHomo sapiens (human)Potency1.000010
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxideHomo sapiens (human)Potency3.314750
5-chloro-3-[[2-(4-ethoxycarbonyl-1-piperazinyl)-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency5.011910
1-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)Potency25.118910
2-[[3-cyano-4-(2-furanyl)-5,6,7,8-tetrahydroquinolin-2-yl]thio]-N-(2-methylphenyl)acetamideHomo sapiens (human)Potency10.000010
3-[[2-[4-(3-chlorophenyl)-1-piperazinyl]-1-oxoethyl]amino]-1H-indole-2-carboxylic acid methyl esterHomo sapiens (human)Potency6.309610
2-cyano-2-[3-[4-(phenylmethyl)-1-piperazinyl]-2-quinoxalinyl]acetic acid 2-methoxyethyl esterHomo sapiens (human)Potency10.000010
4-amino-5,8-dimethoxy-2-(1,1,2,2,2-pentafluoroethyl)-3-quinolinecarbonitrileHomo sapiens (human)Potency12.589310
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]-N-(2-phenylethyl)acetamideHomo sapiens (human)Potency25.118910
2-(4-chlorophenyl)-5-(1-piperidinyl)-4-oxazolecarbonitrileHomo sapiens (human)Potency12.589310
5-bromo-3-ethyl-1H-indole-2-carboxylic acidHomo sapiens (human)Potency10.000010
1-methyl-2-[(phenylthio)methyl]-3-indolecarbonitrileHomo sapiens (human)Potency12.589310
2-[[2-methyl-5-(3-methyl-4-oxo-1-phthalazinyl)phenyl]sulfonylamino]acetic acid ethyl esterHomo sapiens (human)Potency15.848910
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenolHomo sapiens (human)Potency10.000010
2-(4-chlorophenyl)-3-(2-furanylmethyl)imidazo[4,5-b]quinoxalineHomo sapiens (human)Potency31.622810
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid cyclohexyl esterHomo sapiens (human)Potency1.995310
6-(2,5-dimethoxyphenyl)-3-(3-propan-2-yloxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineHomo sapiens (human)Potency15.848910
6-[(2,4-dichlorophenoxy)methyl]-3-(2-methoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency10.000010
2-[5-[(2,4-dichlorophenyl)methylthio]-4-(2-furanylmethyl)-1,2,4-triazol-3-yl]pyridineHomo sapiens (human)Potency12.589310
6-(4-methoxyphenyl)-3-phenyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency0.125910
7-hexyl-3-methyl-8-(4-phenyl-1-piperazinyl)purine-2,6-dioneHomo sapiens (human)Potency12.589310
6-cyclohexyl-3-furan-2-yl-(1,2,4)triazolo(3,4-b)(1,3,4)thiadiazoleHomo sapiens (human)Potency5.011910
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid hexyl esterHomo sapiens (human)Potency10.000010
2-amino-4-pyridin-4-yl-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine-3-carbonitrileHomo sapiens (human)Potency1.000010
4-[4-(1H-benzimidazol-2-ylmethyl)-1-piperazinyl]benzofuro[3,2-d]pyrimidineHomo sapiens (human)Potency10.000010
2-(2-furanyl)-5-(2-furanylmethylamino)-4-oxazolecarbonitrileHomo sapiens (human)Potency10.000010
4-(1H-benzimidazol-2-ylmethylthio)-2-methylbenzofuro[3,2-d]pyrimidineHomo sapiens (human)Potency12.589310
2-(2-methoxyphenyl)-5-[2-(4-methoxyphenyl)ethylamino]-4-oxazolecarbonitrileHomo sapiens (human)Potency10.000010
5-[(4-fluorophenyl)methylamino]-2-(2-methoxyphenyl)-4-oxazolecarbonitrileHomo sapiens (human)Potency10.000010
2-[[6,6-dimethyl-2-(propan-2-ylthio)-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-4-yl]thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)Potency12.589310
1-(thiophen-2-ylmethyl)-3-thiophen-2-ylsulfonyl-2-pyrrolo[3,2-b]quinoxalinamineHomo sapiens (human)Potency7.943310
N-(4-fluorophenyl)-2-[(2-methyl-4-benzofuro[3,2-d]pyrimidinyl)thio]acetamideHomo sapiens (human)Potency15.848910
N-butyl-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-2-pyridinecarboxamideHomo sapiens (human)Potency12.589310
1-[(4-fluorophenyl)methyl]-3-(2-furanylmethyl)-4-imino-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-2-oneHomo sapiens (human)Potency2.511910
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterHomo sapiens (human)Potency10.000010
Glyceryl lactopalmitateHomo sapiens (human)Potency7.943310
2-[[2-(3,5-dimethyl-1-pyrazolyl)-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-4-yl]thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency12.589310
7-(3-chlorophenyl)-2-(4-phenyl-1-piperazinyl)-7,8-dihydro-6H-quinazolin-5-oneHomo sapiens (human)Potency12.589310
2-[[3-[4-(dimethylamino)phenyl]-4,5-dihydroisoxazol-5-yl]methyl]-1,1-dioxo-1,2-benzothiazol-3-oneHomo sapiens (human)Potency10.000010
7-(2-methoxyethyl)-3-methyl-8-(phenylthio)purine-2,6-dioneHomo sapiens (human)Potency25.118910
7-methyl-3-(3-methylbutylamino)-1-(1-pyrrolidinyl)-6,8-dihydro-5H-2,7-naphthyridine-4-carbonitrileHomo sapiens (human)Potency31.622810
5-(3-methoxyphenyl)-N-(2-oxolanylmethyl)-7-(trifluoromethyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency2.511910
4-(1-benzotriazolyl)-5-(2-methoxyphenoxy)benzene-1,2-dicarbonitrileHomo sapiens (human)Potency12.589310
6-amino-4-(4-fluorophenyl)-3-methyl-1-phenyl-5-pyrazolo[3,4-b]pyridinecarbonitrileHomo sapiens (human)Potency5.011910
3-(4-fluorophenyl)-6-(4-methoxyphenyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency31.622810
2-amino-4-(3-chlorophenyl)-6-(2-furanylmethyl)-7-methyl-5-oxo-4H-pyrano[3,2-c]pyridine-3-carboxylic acid methyl esterHomo sapiens (human)Potency10.000010
6-[[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]methyl]-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency15.848910
7-[2-(1,3-benzothiazol-2-ylthio)ethyl]-1,3-dimethyl-8-(3-methyl-1-piperidinyl)purine-2,6-dioneHomo sapiens (human)Potency12.589310
1-(4-fluorophenyl)-2-[[4-(2-furanylmethyl)-5-(phenoxymethyl)-1,2,4-triazol-3-yl]thio]ethanoneHomo sapiens (human)Potency10.000010
2-[[2-furanyl(oxo)methyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
4-[4-(2-quinoxalinyl)phenoxy]benzene-1,2-dicarbonitrileHomo sapiens (human)Potency19.952610
2-(4-bromophenyl)-4-methyl-1H-pyrazol-5-oneHomo sapiens (human)Potency12.589310
3-(4-methylbenzoyl)acrylic acidHomo sapiens (human)Potency25.118910
N4-(3-chlorophenyl)-6-methyl-N2-(phenylmethyl)pyrimidine-2,4-diamineHomo sapiens (human)Potency25.118910
5-(2-furanyl)cyclohexane-1,3-dioneHomo sapiens (human)Potency25.118910
5-(5-chloro-2-methoxyphenyl)-3H-1,3,4-oxadiazole-2-thioneHomo sapiens (human)Potency6.309610
4-chloro-1-methyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency10.000010
2-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxy]acetic acid propan-2-yl esterHomo sapiens (human)Potency10.000010
3,5,5-trimethyl-2-sulfanylidene-1,6-dihydrobenzo[h]quinazolin-4-oneHomo sapiens (human)Potency6.309610
2-methyl-5-(1,4,5,7-tetramethyl-6-pyrrolo[3,4-d]pyridazinyl)anilineHomo sapiens (human)Potency10.000010
N-(3-pyridinyl)-2,3-dihydrothieno[3,4-b][1,4]dioxin-5-carboxamideHomo sapiens (human)Potency5.011910
4-[(4-chloro-5-dithiazolylidene)amino]benzonitrileHomo sapiens (human)Potency25.118910
4-chloro-N-(3,4,5-trimethoxyphenyl)-5-dithiazolimineHomo sapiens (human)Potency25.118910
phenylthiazolylthioureaHomo sapiens (human)Potency0.501210
urocanic acidHomo sapiens (human)Potency5.011910
1-(3,5-dichlorophenyl)-3-phenylureaHomo sapiens (human)Potency12.589310
2-amino-4-(4-chlorophenyl)-6-methyl-3-pyridinecarbonitrileHomo sapiens (human)Potency25.118910
2-(2,4-dimethylanilino)-4-(methoxymethyl)-6-methyl-3-pyridinecarbonitrileHomo sapiens (human)Potency25.118910
3-[(4,8-dimethyl-2-quinolinyl)thio]propanoic acidHomo sapiens (human)Potency12.589310
nsc185058Homo sapiens (human)Potency1.583030
4-(benzenesulfonyl)-5-(ethylthio)-2-phenyloxazoleHomo sapiens (human)Potency10.000010
vu0099704Homo sapiens (human)Potency19.952610
4-[bis(phenylmethyl)amino]-2-(dimethylamino)-3-pyridinecarbonitrileHomo sapiens (human)Potency10.000010
3-(4-bromophenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneHomo sapiens (human)Potency10.000010
3-(4-methylphenyl)-6-phenyl-1,4-dihydro-1,3,5-triazine-2-thioneHomo sapiens (human)Potency10.000010
(3-methyl-1-phenyl-5-thieno[2,3-c]pyrazolyl)-(3-methyl-1-pyrazolyl)methanoneHomo sapiens (human)Potency25.118910
N-[7-(1-oxopropyl)-2,3-dihydro-1,4-benzodioxin-6-yl]benzamideHomo sapiens (human)Potency10.000010
1-(3-nitrophenyl)-3-phenyl-2-propyn-1-oneHomo sapiens (human)Potency12.589310
5-[2-(5-methoxycarbonyl-2-thiophenyl)butan-2-yl]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency12.589310
N-(1-acetyl-2-chloro-3-indolyl)-2-chloroacetamideHomo sapiens (human)Potency10.000010
3-amino-4-(4-chlorophenyl)-6-cyclopropyl-2-thieno[2,3-b]pyridinecarbonitrileHomo sapiens (human)Potency15.848910
1-(4-ethylphenyl)-N-(3-pyridinylmethyl)methanamineHomo sapiens (human)Potency0.010010
4-chloro-1-ethyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency3.981110
2,5-dimethyl-1-(phenylmethyl)pyrrole-3,4-dicarboxaldehydeHomo sapiens (human)Potency7.943310
(4-methoxyphenyl)-(4-methyl-1-piperazinyl)methanethioneHomo sapiens (human)Potency3.981110
3-propyl-1-(2-pyridinylmethylamino)-4-pyrido[1,2-a]benzimidazolecarbonitrileHomo sapiens (human)Potency5.011910
N-(1-ethyl-2-oxo-6-benzo[cd]indolyl)benzamideHomo sapiens (human)Potency19.952610
N-(4-methoxyphenyl)-3-methyl-1,3-benzothiazol-2-imineHomo sapiens (human)Potency19.952610
3-(1,3-benzodioxol-5-yl)-4-(2,5-dimethylphenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency1.584910
3-[[(4-methoxyphenyl)-oxomethyl]amino]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency1.258910
8-[(2-methyl-5-nitro-1,2,4-triazol-3-yl)thio]quinolineHomo sapiens (human)Potency25.118910
2-(4-fluoro-N-methylsulfonylanilino)-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency12.589310
2-(3-methoxyphenyl)-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency6.309610
N-(5-benzoyl-4-phenyl-2-thiazolyl)carbamic acid methyl esterHomo sapiens (human)Potency7.943310
5-(4-propan-2-ylphenyl)-2H-tetrazoleHomo sapiens (human)Potency15.848910
N-(4-fluorophenyl)-1-(3-methylphenyl)-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Potency10.000010
2-(2-methoxyphenoxy)-N-[(2-methoxyphenyl)methyl]acetamideHomo sapiens (human)Potency25.118910
(4-(3-chlorophenyl)piperazin-1-yl)(2-ethoxyphenyl)methanoneHomo sapiens (human)Potency0.794310
2-[[anilino(oxo)methyl]amino]-4,5-dimethoxybenzoic acidHomo sapiens (human)Potency5.011910
3-(4-methoxyphenyl)-5-(4-methylphenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency12.589310
3-bromo-N-[(tert-butylamino)-sulfanylidenemethyl]-4-methoxybenzamideHomo sapiens (human)Potency15.848910
1-(5-ethyl-2,4-dihydroxyphenyl)-2-(2-fluorophenoxy)ethanoneHomo sapiens (human)Potency10.000010
N-[[2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency25.118910
lupitidineHomo sapiens (human)Potency10.000010
1-(4-methoxyphenyl)-1-methyl-3-(1-methyl-5-benzotriazolyl)ureaHomo sapiens (human)Potency31.622810
2-[[cyclopentyl(oxo)methyl]amino]benzoic acid methyl esterHomo sapiens (human)Potency31.622810
2-(2-methoxyphenyl)-1H-indoleHomo sapiens (human)Potency2.511910
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency2.511910
1-(2,3-dimethyl-1-indolyl)-2-(4-methyl-1-piperidinyl)ethanoneHomo sapiens (human)Potency7.943310
4-methoxy-N-[[(phenylmethyl)amino]-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency25.118910
3,6-dichloro-N-(3-pyridinylmethyl)-1-benzothiophene-2-carboxamideHomo sapiens (human)Potency10.000010
4-ethoxy-N-(4-fluorophenyl)-2,3-dimethylbenzenesulfonamideHomo sapiens (human)Potency25.118910
1-(4-methyl-1-piperidinyl)-2-[(3-methyl-2-quinoxalinyl)thio]ethanoneHomo sapiens (human)Potency10.000010
3-cyclohexyl-5-(phenylmethylthio)-1,2,4-triazol-4-amineHomo sapiens (human)Potency12.589310
2-thiophenecarboxylic acid (6-methyl-2-oxo-1H-quinolin-3-yl)methyl esterHomo sapiens (human)Potency25.118910
3-amino-4-thiophen-2-yl-5,6,7,8-tetrahydrothieno[2,3-b]quinoline-2-carboxylic acid methyl esterHomo sapiens (human)Potency12.589310
2-(2-methylphenoxy)-N-[2-(4-methyl-1-piperidinyl)phenyl]acetamideHomo sapiens (human)Potency12.589310
curcuminHomo sapiens (human)Potency0.316210
1-(2-chlorophenyl)-3-[(2-chlorophenyl)methyl]thioureaHomo sapiens (human)Potency12.589310
2-[2-(4-methylphenoxy)ethyl]isoindole-1,3-dioneHomo sapiens (human)Potency25.118910
4-(2-naphthalenyloxymethyl)-2-thiazolamineHomo sapiens (human)Potency15.848910
2,2-dimethyl-N-[[2-(4-methyl-1-piperidinyl)anilino]-sulfanylidenemethyl]propanamideHomo sapiens (human)Potency10.000010
N-methyl-N-phenylcarbamic acid (4-tert-butylphenyl) esterHomo sapiens (human)Potency12.589310
N-[(3-bromo-4-ethoxy-5-methoxyphenyl)methyl]-2,3-dihydro-1,4-benzodioxin-6-amineHomo sapiens (human)Potency15.848910
2-[(3,5-dimethyl-4-isoxazolyl)methylthio]-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency10.000010
2,3,5,6-tetramethyl-N-(2-methyl-1,3-benzothiazol-5-yl)benzenesulfonamideHomo sapiens (human)Potency25.118910
2-[[[(6-methyl-2-pyridinyl)amino]-sulfanylidenemethyl]amino]-5-phenyl-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
5-chloro-N-(2-furanylmethyl)-2-[[(4-methoxyphenyl)-oxomethyl]amino]benzamideHomo sapiens (human)Potency25.118910
5-[(2,4-dichlorophenoxy)methyl]-N-[1-[(2-fluorophenyl)methyl]-3-pyrazolyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
9-hydroxy-4-[1-oxo-2-[4-(phenylmethyl)-1-piperazinyl]ethyl]-2,3-dihydro-1H-[1]benzopyrano[3,4-b]pyridin-5-oneHomo sapiens (human)Potency10.000010
N-(3-chlorophenyl)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-4-methylbenzenesulfonamideHomo sapiens (human)Potency10.000010
6-(4-benzoyl-1-piperazinyl)-3,3-dimethyl-8-propan-2-yl-1,4-dihydropyrano[3,4-c]pyridine-5-carbonitrileHomo sapiens (human)Potency12.589310
2-[(3-cyano-4-phenyl-6-thiophen-2-yl-2-pyridinyl)thio]-N-propan-2-ylacetamideHomo sapiens (human)Potency10.000010
1-[[[2-(2,4-dichlorophenyl)-4-quinolinyl]-oxomethyl]amino]-3-phenylureaHomo sapiens (human)Potency25.118910
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamideHomo sapiens (human)Potency10.000010
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Potency12.589310
5-(4-bromophenyl)-N-[[(2-propyl-5-tetrazolyl)amino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency3.162310
5-bromo-N-[[4-[(3,5-dimethylphenyl)sulfamoyl]anilino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
4-[[[[oxo-(4-phenylphenyl)methyl]amino]-sulfanylidenemethyl]amino]benzoic acidHomo sapiens (human)Potency7.943310
N-[4,6-bis(4-morpholinyl)-1,3,5-triazin-2-yl]-2-(methylthio)-1,3-benzothiazol-6-amineHomo sapiens (human)Potency10.000010
2-(3-pyridinyl)-4-[4-(1-pyrrolidinylsulfonyl)phenyl]thiazoleHomo sapiens (human)Potency10.000010
2-amino-4-(4-chlorophenyl)-1-(4-methylphenyl)-6-oxopyridine-3,5-dicarbonitrileHomo sapiens (human)Potency15.848910
6-chloro-4-phenyl-3-(1-phenyl-5-tetrazolyl)quinolineHomo sapiens (human)Potency9.275030
N-[[3-chloro-4-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency5.011910
2-[[3-cyano-6-(4-methylphenyl)-4-(trifluoromethyl)-2-pyridinyl]thio]-N-(4-methoxyphenyl)acetamideHomo sapiens (human)Potency12.589310
2-[[2-(5-methyl-2-thiophenyl)-2-oxoethyl]thio]-3-phenyl-4-quinazolinoneHomo sapiens (human)Potency25.118910
1-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-2-[(4-chlorophenyl)methylthio]ethanoneHomo sapiens (human)Potency25.118910
LSM-4563Homo sapiens (human)Potency3.981110
1,2,3,4-tetrahydroacridine-9-carboxylic acid (2-oxo-2-thiophen-2-ylethyl) esterHomo sapiens (human)Potency12.589310
1-(N-[2-(Benzotriazol-1-yl)acetyl]-4-methoxyanilino)-N-cyclopentylcyclohexane-1-carboxamideHomo sapiens (human)Potency12.589310
7-(difluoromethyl)-N-(5-methyl-3-isoxazolyl)-5-(4-methylphenyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency1.584910
6-(4,5-dihydrothiazol-2-ylthio)-N2,N4-bis(2-methylphenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency10.000010
2-furanyl-(4,4,8-trimethyl-1-sulfanylidene-5-dithiolo[3,4-c]quinolinyl)methanoneHomo sapiens (human)Potency12.589310
2-[2-oxo-2-(2,2,4,6-tetramethyl-1-quinolinyl)ethyl]isoindole-1,3-dioneHomo sapiens (human)Potency12.589310
N-[5-(4-tert-butylphenyl)-1,3,4-thiadiazol-2-yl]-4-methylbenzamideHomo sapiens (human)Potency5.011910
2-[(7-methoxy-4-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)thio]-N-methyl-N-(4-phenyl-2-thiazolyl)acetamideHomo sapiens (human)Potency19.952610
N-(phenylmethyl)-2-[[4-(trifluoromethyl)-5,6-dihydrobenzo[h]quinazolin-2-yl]thio]acetamideHomo sapiens (human)Potency15.848910
3-methyl-N'-(1-oxo-2-phenoxyethyl)-1-phenyl-5-thieno[2,3-c]pyrazolecarbohydrazideHomo sapiens (human)Potency0.794310
2-[5-(2-fluorophenyl)-2-tetrazolyl]-N-[2-oxo-2-[(phenylmethyl)amino]ethyl]-N-(5,6,7,8-tetrahydronaphthalen-1-yl)acetamideHomo sapiens (human)Potency15.848910
2-[(3-cyano-6-methoxy-2-quinolinyl)thio]-N-(2-methyl-1,3-benzothiazol-5-yl)acetamideHomo sapiens (human)Potency12.589310
1-(6-methoxy-2,2,4-trimethyl-1-quinolinyl)-2-[[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]thio]ethanoneHomo sapiens (human)Potency12.589310
2-(4-methylphenyl)-N-[4-(4-morpholinyl)phenyl]-4-quinazolinamineHomo sapiens (human)Potency12.589310
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterHomo sapiens (human)Potency25.118910
N-(2,5-dimethylphenyl)-2-[[3-(4-ethylphenoxy)-4-oxo-1-benzopyran-7-yl]oxy]acetamideHomo sapiens (human)Potency6.309610
LSM-28492Homo sapiens (human)Potency10.000010
4-(5,6-dimethyl-1-benzimidazolyl)-5-phenylthieno[2,3-d]pyrimidineHomo sapiens (human)Potency12.589310
N-(2-ethylphenyl)-2-[[2-(4-methoxyphenyl)-4-oxo-1-benzopyran-6-yl]oxy]acetamideHomo sapiens (human)Potency10.000010
4-(4-ethoxycarbonylanilino)-2-quinazolinecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
4-(4-anilinoanilino)-2-quinazolinecarboxylic acid ethyl esterHomo sapiens (human)Potency25.118910
2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)acetamideHomo sapiens (human)Potency25.118910
2-[[cyclohexyl(oxo)methyl]amino]-4-(3-nitrophenyl)-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
3-methoxy-4-(2-methoxy-3-methoxycarbonyl-1-naphthalenyl)-2-naphthalenecarboxylic acid methyl esterHomo sapiens (human)Potency10.000010
4-(3-bromophenyl)-2-(4-bromophenyl)-7-methylpyrazolo[3,4-d]pyridazineHomo sapiens (human)Potency10.000010
4-(3-bromophenyl)-7-methyl-2-(4-methylphenyl)pyrazolo[3,4-d]pyridazineHomo sapiens (human)Potency10.000010
(4-phenyl-1-piperazinyl)-(9H-xanthen-9-yl)methanoneHomo sapiens (human)Potency10.000010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[5-[(4-chlorophenoxy)methyl]-2-furanyl]methanoneHomo sapiens (human)Potency12.589310
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency25.118910
2-(1,2-benzoxazol-3-yl)-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency0.015810
3,5-dimethoxy-N-[(2-phenylethylamino)-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency10.000010
2-(2-fluorophenyl)-4-(4-fluorophenyl)sulfonyl-5-(1-piperidinyl)oxazoleHomo sapiens (human)Potency7.943310
5-bromo-N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency12.589310
[4-(2-methylphenyl)-1-piperazinyl]-(5-propyl-3-thiophenyl)methanoneHomo sapiens (human)Potency19.952610
1,3-diethyl-6-methyl-N-(2-methylphenyl)-2-oxo-5-benzimidazolesulfonamideHomo sapiens (human)Potency25.118910
2-[[5-(2-furanyl)-4-(4-methylphenyl)-1,2,4-triazol-3-yl]thio]-N-(1H-indazol-6-yl)acetamideHomo sapiens (human)Potency12.589310
5-[[[4-(4-fluorophenyl)-5-(phenylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-3-thiophen-2-yl-1,2,4-oxadiazoleHomo sapiens (human)Potency7.943310
N-[[3-chloro-2-(4-morpholinyl)anilino]-sulfanylidenemethyl]-4-methoxy-3-nitrobenzamideHomo sapiens (human)Potency10.000010
N-[[3-chloro-2-(1-piperidinyl)anilino]-sulfanylidenemethyl]-2-thiophenecarboxamideHomo sapiens (human)Potency12.589310
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamideHomo sapiens (human)Potency10.000010
2-[[5-(7-methoxy-2-benzofuranyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]-1-(4-methoxyphenyl)ethanoneHomo sapiens (human)Potency25.118910
[4-(2,3-dimethylphenyl)-1-piperazinyl]-(3,4,5-trimethoxyphenyl)methanoneHomo sapiens (human)Potency12.589310
2-[[4,6-bis(1-piperidinyl)-1,3,5-triazin-2-yl]thio]-1-phenylethanoneHomo sapiens (human)Potency10.000010
1-oxo-3-(1-piperidinyl)-5,6,7,8-tetrahydropyrrolo[1,2-a]indole-2-carbonitrileHomo sapiens (human)Potency15.848910
2-(1-imidazolyl)-4-phenyl-6-(4-phenyl-1-piperazinyl)-1,3,5-triazineHomo sapiens (human)Potency12.589310
2-[(3,5-dimethyl-4-isoxazolyl)methylthio]-3-prop-2-enyl-6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-b]pyrimidin-4-oneHomo sapiens (human)Potency10.000010
1-(1,2,3-benzothiadiazol-5-yl)-3-(1-naphthalenyl)ureaHomo sapiens (human)Potency10.000010
5-hydroxy-1-methyl-4-(4-morpholinylmethyl)-2-[(phenylthio)methyl]-3-indolecarboxylic acid ethyl esterHomo sapiens (human)Potency7.943310
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamineHomo sapiens (human)Potency12.589310
1-(3-chlorophenyl)-3-(2-phenoxyphenyl)thioureaHomo sapiens (human)Potency25.118910
N-[3-[2-(1-azepanyl)-4,5-dicyanophenoxy]phenyl]acetamideHomo sapiens (human)Potency10.000010
N-[[4-(diethylamino)phenyl]methyl]-1-[2-(1-piperidinyl)ethyl]-2-benzimidazolamineHomo sapiens (human)Potency12.589310
N-(6-ethoxy-1,3-benzothiazol-2-yl)-1,3-dimethyl-2-oxo-5-benzimidazolesulfonamideHomo sapiens (human)Potency2.511910
2-[[4-(4-methoxyphenyl)-5-(2-phenylethyl)-1,2,4-triazol-3-yl]thio]-N-(phenylmethyl)acetamideHomo sapiens (human)Potency25.118910
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-1,3-benzodioxole-5-carboxamideHomo sapiens (human)Potency5.011910
4-[[2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency15.848910
N-(4-fluorophenyl)-3-([1,2,4]triazolo[4,3-a]quinolin-1-ylthio)propanamideHomo sapiens (human)Potency10.000010
2-(1-naphthalenyl)-N-(2-phenyl-1,3-benzoxazol-5-yl)acetamideHomo sapiens (human)Potency25.118910
9-(3-bromo-4-hydroxyphenyl)-10-phenyl-3,4,5,6,7,9-hexahydro-2H-acridine-1,8-dioneHomo sapiens (human)Potency12.589310
2,4-dichloro-5-(diethylsulfamoyl)-N-(1,3,4-thiadiazol-2-yl)benzamideHomo sapiens (human)Potency7.943310
3-ethoxy-N-[3-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl]benzamideHomo sapiens (human)Potency12.589310
2-methylsulfonyl-4,6-diphenyl-3-thieno[2,3-b]pyridinamineHomo sapiens (human)Potency10.000010
5-[(3-methyl-6-oxo-7,8,9,10-tetrahydrobenzo[c][1]benzopyran-1-yl)oxymethyl]-2-furancarboxylic acid methyl esterHomo sapiens (human)Potency7.943310
3-(4-bromophenyl)-5-(3,5-dimethoxyphenyl)-1,2,4-oxadiazoleHomo sapiens (human)Potency25.118910
2-[2,5-dimethyl-3-[(2,4,6-trioxo-1,3-diazinan-5-ylidene)methyl]-1-pyrrolyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
N-(9,9-dimethyl-7-oxo-8,10-dihydronaphtho[1,2-b]benzofuran-5-yl)-4-methoxybenzenesulfonamideHomo sapiens (human)Potency7.943310
5-[(cyclohexylamino)-oxomethyl]-4-methyl-2-[(1-oxo-2-thiophen-2-ylethyl)amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
N-[[5-(1H-benzimidazol-2-yl)-2-methylanilino]-sulfanylidenemethyl]-5-chloro-2-methoxybenzamideHomo sapiens (human)Potency15.848910
N-[4-[5-(2-furanyl)-1,3,4-oxadiazol-2-yl]phenyl]-2-(2-methoxyphenyl)acetamideHomo sapiens (human)Potency25.118910
N-[[4-(4-chlorophenoxy)anilino]-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency15.848910
N-(2,3-dimethylphenyl)-2-[[6-(1,3-dioxo-2-isoindolyl)-1,3-benzothiazol-2-yl]thio]acetamideHomo sapiens (human)Potency25.118910
5-bromo-N-[2-(3-pyridinyl)-1,3-benzoxazol-5-yl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
N-[[3-(2-oxazolo[4,5-b]pyridinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency25.118910
N-[3-(1,3-benzothiazol-2-ylthio)-4-hydroxyphenyl]-4-chlorobenzenesulfonamideHomo sapiens (human)Potency10.000010
5-(3-nitrophenyl)-N-[[2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
2-[1-(4-tert-butylphenyl)sulfonyl-4-piperidinyl]-6-chloro-1H-benzimidazoleHomo sapiens (human)Potency10.000010
LSM-28273Homo sapiens (human)Potency10.000010
2-(3-chlorophenyl)-9-[4-(2-pyrazinyl)-1-piperazinyl]-5,6,7,8-tetrahydropyrazolo[5,1-b]quinazolineHomo sapiens (human)Potency10.000010
1-(4-fluorophenyl)-2-[(2-propyl-4-quinazolinyl)thio]ethanoneHomo sapiens (human)Potency31.622810
4-cyano-N-methyl-N-[5-(2-pyridinyl)-1,3,4-thiadiazol-2-yl]benzamideHomo sapiens (human)Potency25.118910
5-tert-butyl-N-[2-(cyclopentylamino)-2-oxoethyl]-N-(2,5-dimethylphenyl)-3-methyl-2-furancarboxamideHomo sapiens (human)Potency10.000010
2-[4-(4-chlorophenyl)sulfonyl-1-piperazinyl]-1-ethylbenzimidazoleHomo sapiens (human)Potency12.589310
4-tert-butyl-N-[2,5-dimethoxy-4-[[1-oxo-2-(1-piperidinyl)ethyl]amino]phenyl]benzamideHomo sapiens (human)Potency7.943310
4-[(2,6-dichlorophenyl)thio]-5-methoxy-2-(2-pyridinyl)pyrimidineHomo sapiens (human)Potency12.589310
2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]-7-(4-methoxyphenyl)-[1,2,4]triazolo[1,5-a]pyrimidineHomo sapiens (human)Potency25.118910
4-chloro-N-(4-chloro-2-methylphenyl)-5-dithiazolimineHomo sapiens (human)Potency12.589310
7-(4-methoxyphenyl)-2-(1-pyrrolyl)-[1,2,4]triazolo[1,5-a]pyrimidineHomo sapiens (human)Potency10.000010
2-[(4-chlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinoneHomo sapiens (human)Potency12.589310
2-[(3-chlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinoneHomo sapiens (human)Potency10.000010
4-(4-tert-butylphenoxy)-5-methoxy-2-phenylpyrimidineHomo sapiens (human)Potency10.000010
3-[5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazol-2-yl]-1-(phenylmethyl)-2-pyridinoneHomo sapiens (human)Potency12.589310
2-[2-(2,4-dichloro-5-propan-2-yloxyanilino)-2-oxoethyl]sulfinyl-N-[3-(trifluoromethyl)phenyl]acetamideHomo sapiens (human)Potency5.011910
5-[1-(benzenesulfonyl)-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency12.589310
5-[1-(4-fluorophenyl)sulfonyl-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency12.589310
5-[1-[(4-fluorophenyl)methyl]-3-pyrazolyl]-2-phenylthiazoleHomo sapiens (human)Potency12.589310
N-(4-bromophenyl)-1-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-2-pyrrolecarboxamideHomo sapiens (human)Potency12.589310
7-(4-chlorophenyl)-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]-[1,2,4]triazolo[1,5-a]pyrimidineHomo sapiens (human)Potency12.589310
4-(4-methyl-1-piperazinyl)-2,6-diphenyl-5-pyrimidinecarbonitrileHomo sapiens (human)Potency6.309610
2-(methylthio)-7-(4-phenylphenyl)-[1,2,4]triazolo[1,5-a]pyrimidineHomo sapiens (human)Potency10.000010
N,N-dimethylcarbamothioic acid O-[4-[2-[(4-chlorophenyl)thio]-1-oxoethyl]-2,6-dimethylphenyl] esterHomo sapiens (human)Potency10.000010
4-[2-[(2,4-dichlorophenyl)methylthio]-6-methyl-4-pyrimidinyl]morpholineHomo sapiens (human)Potency12.589310
5-[3-[(4-methylphenyl)methoxy]-2-thiophenyl]-3-(methylthio)-1H-1,2,4-triazoleHomo sapiens (human)Potency3.162310
(4-chlorophenyl)-[5-(4-morpholinyl)-4-(2-pyridinyl)-2-thiophenyl]methanoneHomo sapiens (human)Potency10.000010
r-7050Homo sapiens (human)Potency3.981110
1,1-bis(4-chlorophenyl)-2-[(3-methoxyphenyl)methylamino]ethanolHomo sapiens (human)Potency10.000010
(4-chlorophenyl)-[4-[[(2,4-dichlorophenyl)thio]methyl]-4-hydroxy-1-piperidinyl]methanoneHomo sapiens (human)Potency25.118910
N-propan-2-yl-3-(trifluoromethyl)benzamideHomo sapiens (human)Potency25.118910
4-methoxy-N-(8-methyl-[1,3]dioxolo[4,5-g]quinazolin-6-yl)benzamideHomo sapiens (human)Potency25.118910
5-[(4-methyl-1-piperidinyl)methyl]-1-[4-(1-pyrrolyl)-1,2,5-oxadiazol-3-yl]-4-triazolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
2-[(3,4-dichlorophenyl)methylthio]-6-(3-pyridinyl)-3-pyridinecarbonitrileHomo sapiens (human)Potency25.118910
cinnarizineHomo sapiens (human)Potency25.278330
3-(4-phenylphenyl)-6,7,8,9-tetrahydro-5H-imidazo[1,2-a]azepineHomo sapiens (human)Potency10.000010
N-[4-(4-fluorophenyl)-2-thiazolyl]-4-methylbenzenesulfonamideHomo sapiens (human)Potency25.118910
2-[[[4-(diethylsulfamoyl)phenyl]-oxomethyl]amino]-4-methyl-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
sulindacHomo sapiens (human)Potency15.848910
N-(2,4-dichlorophenyl)-4-phenylbenzamideHomo sapiens (human)Potency25.118910
N-[(2-adamantylamino)-sulfanylidenemethyl]hexanamideHomo sapiens (human)Potency25.118910
4-(4-methylphenyl)-2-[[oxo-(2-oxo-1-benzopyran-3-yl)methyl]amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
3-propoxy-N-[sulfanylidene-[3-(trifluoromethyl)anilino]methyl]benzamideHomo sapiens (human)Potency10.000010
N-[[3-chloro-4-(1-piperidinyl)anilino]-sulfanylidenemethyl]hexanamideHomo sapiens (human)Potency19.952610
5-[diethylamino(oxo)methyl]-4-methyl-2-(1-oxopentylamino)-3-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency25.118910
3-chloro-N-[3-[[(3-chloro-4-nitrophenyl)-oxomethyl]amino]-2,2-dimethylpropyl]-4-nitrobenzamideHomo sapiens (human)Potency10.000010
4-(1-benzotriazolyl)-3,5-dinitrobenzonitrileHomo sapiens (human)Potency19.952610
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(3,4-dimethoxyphenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency3.981110
5-tert-butyl-3-(4-chlorophenyl)-N-(2-pyridinylmethyl)-7-pyrazolo[1,5-a]pyrimidinamineHomo sapiens (human)Potency10.000010
LSM-20639Homo sapiens (human)Potency10.000010
3-phenyl-2-propan-2-yl[1]benzopyrano[2,3-d]pyrimidine-4,5-dioneHomo sapiens (human)Potency25.118910
tg 003Homo sapiens (human)Potency10.000010
4-(phenylmethyl)-3-[2-(4-propoxyphenyl)ethyl]-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency10.000010
N-bis(2-fluorophenoxy)phosphoryl-3,4-dimethylanilineHomo sapiens (human)Potency10.000010
N,N-dibutyl-2-(pyridin-4-yl)quinazolin-4-amineHomo sapiens (human)Potency12.589310
5-[(6-hydroxy-4-oxo-1-benzopyran-3-yl)methylidene]-1,3-diazinane-2,4,6-trioneHomo sapiens (human)Potency12.589310
4-[[(4-tert-butylphenyl)-oxomethyl]amino]-3-methyl-2-sulfanylidene-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
4-(4-chlorophenyl)-N-(3-pyridinylmethyl)-6-(trifluoromethyl)-2-pyrimidinamineHomo sapiens (human)Potency5.011910
4,5-dichloro-1-[2-(4-chlorophenoxy)ethyl]imidazoleHomo sapiens (human)Potency25.118910
2-(3,5-dimethyl-1-pyrazolyl)-4-(4-hydroxyanilino)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency2.511910
1-butyl-3-(4-phenoxyphenyl)thioureaHomo sapiens (human)Potency25.118910
N-[5-methyl-2-(4-methylphenyl)-3-pyrazolyl]-2-[(7-methyl-4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-9-yl)oxy]acetamideHomo sapiens (human)Potency10.000010
2-[[4-amino-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]thio]-N-(9-ethyl-3-carbazolyl)acetamideHomo sapiens (human)Potency10.000010
2-[(2-methyl-4-benzofuro[3,2-d]pyrimidinyl)thio]-N-(2-phenylethyl)acetamideHomo sapiens (human)Potency25.118910
N-(4-bromophenyl)-5-tert-butyl-2-methyl-4-nitro-3-pyrazolecarboxamideHomo sapiens (human)Potency25.118910
N-(5-tert-butyl-2-phenyl-3-pyrazolyl)-2-[(6-methyl-1H-benzimidazol-2-yl)thio]acetamideHomo sapiens (human)Potency10.000010
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)thio]ethanoneHomo sapiens (human)Potency10.000010
3-[4-(4-morpholinylsulfonyl)phenyl]propanoic acid [2-[(5-chloro-2-pyridinyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
N-[4-(4-methyl-2-thiazolyl)-2-phenyl-3-pyrazolyl]-3-(trifluoromethyl)benzamideHomo sapiens (human)Potency12.589310
6-(4-bromophenyl)-3-methyl-1-[2-(2H-tetrazol-5-yl)ethyl]-4-(trifluoromethyl)pyrazolo[3,4-b]pyridineHomo sapiens (human)Potency6.309610
1-[4-(benzenesulfonyl)-1-piperazinyl]-2-[[3-chloro-5-(trifluoromethyl)-2-pyridinyl]thio]ethanoneHomo sapiens (human)Potency10.000010
2-[7-chloro-2,3-dioxo-4-(phenylmethyl)-1-quinoxalinyl]-N-(3-fluorophenyl)acetamideHomo sapiens (human)Potency12.589310
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-2,5-diphenyl-3-pyrazolecarboxamideHomo sapiens (human)Potency10.000010
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-quinolinecarboxamideHomo sapiens (human)Potency7.943310
4-[(3,5-dimethylphenyl)-oxomethyl]-1,3-dihydroquinoxalin-2-oneHomo sapiens (human)Potency1.995310
3-[[[5-[3-(1-piperidinylsulfonyl)phenyl]-1,3,4-oxadiazol-2-yl]thio]methyl]-1,2,3-benzotriazin-4-oneHomo sapiens (human)Potency6.309610
2-[3-[(4-chlorophenyl)-oxomethyl]-6-methoxy-4-oxo-1-quinolinyl]-N-(4-fluorophenyl)acetamideHomo sapiens (human)Potency10.000010
N-(3,5-dimethoxyphenyl)-2-(2,2-dimethyl-5-oxo-4-phenyl-1-imidazolyl)acetamideHomo sapiens (human)Potency12.589310
N-(4-acetylphenyl)-5-[(phenylthio)methyl]-2-furancarboxamideHomo sapiens (human)Potency25.118910
(4-tert-butylphenyl)-[2-(4-fluorophenyl)-8-methyl-3-sulfanylidene-1,4,8-triazaspiro[4.5]dec-1-en-4-yl]methanoneHomo sapiens (human)Potency12.589310
2-[[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-oxomethyl]imino-1-(2-methylpropyl)-5-oxo-3-dipyrido[1,2-d-3',4'-f]pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)Potency3.981110
4-[bis(2-methoxyethyl)sulfamoyl]-N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)benzamideHomo sapiens (human)Potency0.050110
1-[2-(5-fluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(3-fluorophenyl)-1-(3-pyridinylmethyl)thioureaHomo sapiens (human)Potency10.000010
1-[2-(5-fluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(4-fluorophenyl)-1-(3-pyridinylmethyl)thioureaHomo sapiens (human)Potency10.000010
1-[2-(5-fluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)thioureaHomo sapiens (human)Potency7.943310
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esterHomo sapiens (human)Potency10.000010
4-[[(2-nitrophenyl)-oxomethyl]amino]benzoic acid propyl esterHomo sapiens (human)Potency15.848910
2-[[oxo-(2,3,4,5,6-pentafluorophenyl)methyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency10.000010
4-chlorobenzenesulfonic acid [4-(1,8-dioxo-3,4,5,6,7,9-hexahydro-2H-xanthen-9-yl)phenyl] esterHomo sapiens (human)Potency12.589310
N-[4-(dibutylsulfamoyl)phenyl]-2-thiophen-2-ylacetamideHomo sapiens (human)Potency10.000010
6-bromo-3-[4-nitro-3-(trifluoromethyl)phenyl]-2-propyl-4-quinazolinoneHomo sapiens (human)Potency10.000010
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]acetic acid ethyl esterHomo sapiens (human)Potency25.118910
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-2-benzofurancarboxamideHomo sapiens (human)Potency5.011910
N-(4-methyl-1,3-benzothiazol-2-yl)-9H-xanthene-9-carboxamideHomo sapiens (human)Potency12.589310
N-(2-furanylmethyl)-2-[3-(1-oxo-2-phenoxyethyl)-1-indolyl]acetamideHomo sapiens (human)Potency1.258910
6-bromo-2-(3-pyridinyl)-N-[4-(trifluoromethyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)Potency10.000010
N-[2-(cyclohexylthio)ethyl]-4-methyl-3-[(4-methylphenyl)sulfamoyl]benzamideHomo sapiens (human)Potency25.118910
N-[[3-chloro-2-(1-pyrrolidinyl)anilino]-sulfanylidenemethyl]butanamideHomo sapiens (human)Potency12.589310
N-(4-ethoxyphenyl)-4-[[4-(methylthio)phenyl]sulfonylamino]benzenesulfonamideHomo sapiens (human)Potency10.000010
4-chloro-3-[(2,5-dimethylphenyl)sulfamoyl]-N-(2-phenylphenyl)benzamideHomo sapiens (human)Potency12.589310
3-(2-bromophenyl)-6-[(4-methoxyphenyl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)Potency1.995310
1-(3-fluorophenyl)-4-(4-hydroxy-3-methoxy-5-nitrophenyl)-4H-pyridine-3,5-dicarboxylic acid diethyl esterHomo sapiens (human)Potency12.589310
3-(2-chlorophenyl)-N-cyclohexyl-5-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-isoxazolecarboxamideHomo sapiens (human)Potency10.000010
1-[[4-(2,4,6-trimethylphenyl)-1-piperazinyl]sulfonyl]azepaneHomo sapiens (human)Potency10.000010
N-(3-acetylphenyl)-5,7-dimethyl-2-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency12.589310
1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(5,7-diphenyl-2-pyrazolo[1,5-a]pyrimidinyl)methanoneHomo sapiens (human)Potency12.589310
2-[[5-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethoxy]-4-oxo-2-phenyl-1-benzopyran-7-yl]oxy]acetic acid tert-butyl esterHomo sapiens (human)Potency6.309610
3,4-dimethyl-N-[sulfanylidene-[2-(trifluoromethyl)anilino]methyl]benzamideHomo sapiens (human)Potency25.118910
8-[2-(4-chloro-2,5-dimethylphenoxy)ethoxy]quinolineHomo sapiens (human)Potency25.118910
4E2RCatHomo sapiens (human)Potency10.000010
1-chloro-2-[2-(2-methoxy-4-methylphenoxy)ethoxy]-4-methylbenzeneHomo sapiens (human)Potency10.000010
2-[cyclohexyl-(4-methylphenyl)sulfonylamino]-N-(3-methoxypropyl)acetamideHomo sapiens (human)Potency10.000010
5-bromo-N-(4-methoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)Potency25.118910
1-azepanyl-[2-[4-(difluoromethylthio)anilino]phenyl]methanoneHomo sapiens (human)Potency10.000010
2-nitrobenzoic acid [1,1,1,3,3,3-hexafluoro-2-[4-[(4-methylphenyl)sulfonylamino]phenyl]propan-2-yl] esterHomo sapiens (human)Potency10.000010
2-(4,6-dimethyl-2-pyrimidinyl)-4-[(4-fluorophenyl)thio]-5-methyl-3-pyrazolamineHomo sapiens (human)Potency6.309610
N-[4-(4-morpholinyl)phenyl]-2-pyridin-4-yl-4-quinolinecarboxamideHomo sapiens (human)Potency12.589310
1-(2-chlorophenyl)-N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency15.848910
2-(1H-benzimidazol-2-ylthio)-N-(2-methoxy-3-dibenzofuranyl)acetamideHomo sapiens (human)Potency10.000010
2-(methylthio)-3-pyridinecarboxylic acid [2-[2-(4-morpholinyl)-5-(trifluoromethyl)anilino]-2-oxoethyl] esterHomo sapiens (human)Potency15.848910
1,2,3,4-tetrahydroacridine-9-carboxylic acid [2-(3-chloro-4-methoxyanilino)-2-oxoethyl] esterHomo sapiens (human)Potency10.000010
5,6,7,8-tetrafluoro-2-(2,3,4,5,6-pentafluorophenyl)-4h-1-benzopyran-4-oneHomo sapiens (human)Potency2.728730
N-[[2-(1-cyclohexenyl)ethylamino]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)Potency12.589310
12-oxo-N-(4-phenyl-2-thiazolyl)-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazoline-3-carboxamideHomo sapiens (human)Potency25.118910
N-[5-(2,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-phenylacetamideHomo sapiens (human)Potency12.589310
3-methyl-N-[(4-methylphenyl)methyl]-7,8-dihydro-6H-cyclopenta[4,5]thieno[1,2-c]pyrimidin-1-amineHomo sapiens (human)Potency25.118910
3-[2-(4-chlorophenyl)-4-quinolinyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepineHomo sapiens (human)Potency25.118910
1-(2-cyanoethyl)-6-(2-fluoro-4-methoxyphenyl)-3-methyl-4-pyrazolo[3,4-b]pyridinecarboxylic acid ethyl esterHomo sapiens (human)Potency7.943310
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4-methyl-5-phenyl-2-thiazolyl)-N-prop-2-enylacetamideHomo sapiens (human)Potency3.162310
2-[(3-acetyl-5-oxo-4H-imidazol-2-yl)thio]-N-(4,5-diphenyl-2-thiazolyl)acetamideHomo sapiens (human)Potency10.000010
3-[2-(2-furanylmethylamino)-2-oxoethoxy]-N-(2-methoxy-5-methylphenyl)-2-naphthalenecarboxamideHomo sapiens (human)Potency12.589310
2-chloro-1-[1-[2-(4-chlorophenyl)ethyl]-2,5-dimethyl-3-pyrrolyl]ethanoneHomo sapiens (human)Potency15.848910
N-(4-tert-butyl-2-thiazolyl)-5-methyl-2-thiophenecarboxamideHomo sapiens (human)Potency31.622810
N2-[5-(3-chlorophenyl)-2-phenyl-3-pyrazolyl]benzene-1,2-diamineHomo sapiens (human)Potency10.000010
4-[2-(4-fluoroanilino)-2-oxoethoxy]-3-methoxy-N-[4-(4-methoxyphenyl)-5-methyl-2-thiazolyl]benzamideHomo sapiens (human)Potency10.000010
3,4-diethoxybenzoic acid [2-[(5-methyl-3-isoxazolyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency19.952610
3-[(3,4-difluorophenyl)sulfonylamino]benzoic acid [2-[[(2-methylpropylamino)-oxomethyl]amino]-2-oxoethyl] esterHomo sapiens (human)Potency25.118910
2-(2,4-dioxo-1,3-diazaspiro[4.4]nonan-3-yl)acetic acid (7-bromo-4-oxo-2-pyrido[1,2-a]pyrimidinyl)methyl esterHomo sapiens (human)Potency25.118910
2-(4-chlorophenyl)-5-[[(4-methyl-2-thiazolyl)thio]methyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency25.118910
3-[5-(2,5-dimethyl-1-phenyl-3-pyrrolyl)-1,3,4-oxadiazol-2-yl]-1-benzopyran-2-oneHomo sapiens (human)Potency12.589310
N-cyclohexyl-2-[(4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl)oxy]acetamideHomo sapiens (human)Potency5.011910
N-(4-chloro-2-methoxy-5-methylphenyl)-4-[(3,4-difluorophenyl)sulfonylamino]benzamideHomo sapiens (human)Potency10.000010
2-[[[4-cyclohexyl-5-(thiophen-2-ylmethyl)-1,2,4-triazol-3-yl]thio]methyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency12.589310
2-[[(3-methylphenyl)-oxomethyl]amino]benzoic acid (3,5-dimethyl-4-isoxazolyl)methyl esterHomo sapiens (human)Potency10.000010
N-[2-[(1,3-benzodioxol-5-ylmethylamino)-oxomethyl]phenyl]-2-ethoxy-3-pyridinecarboxamideHomo sapiens (human)Potency15.848910
3-(1H-indol-3-yl)propanoic acid [2-[tert-butyl-(phenylmethyl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
5-methyl-4-(4-methylphenyl)-2-[[2-[(1-methyl-5-tetrazolyl)thio]-1-oxoethyl]amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
4-nitrobenzoic acid [3-(2,6-dichlorophenyl)-5-methyl-4-isoxazolyl]methyl esterHomo sapiens (human)Potency25.118910
4-amino-2-(4-chlorophenyl)-6-(methylthio)pyrimidine-5-carbonitrileHomo sapiens (human)Potency12.589310
N-(4-chlorophenyl)-N-ethyl-6-(propan-2-ylamino)-4-(trifluoromethyl)-3-pyridinecarboxamideHomo sapiens (human)Potency10.000010
3-(9-carbazolylmethyl)-4-methyl-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency15.848910
1-(4-methoxyphenyl)-3-(6-methyl-2-pyridinyl)thioureaHomo sapiens (human)Potency7.943310
1-(3-methylphenyl)-3-(2-pyridinyl)thioureaHomo sapiens (human)Potency25.118910
4-chlorophenylalanine methyl ester, hydrochloride, (dl)-isomerHomo sapiens (human)Potency3.981110
capsazepineHomo sapiens (human)Potency10.000010
3-(tert-butylsulfamoyl)-4-phenyl-5-(trifluoromethyl)-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency10.000010
2,5-bis(3,5-dimethyl-1-phenyl-4-pyrazolyl)-1,3,4-oxadiazoleHomo sapiens (human)Potency10.000010
6-(4-chlorophenyl)-4-(methylthio)-2-oxo-1H-pyridine-3-carbonitrileHomo sapiens (human)Potency10.000010
N'-benzoyl-5-(3,5-dichlorophenoxy)-2-furancarbohydrazideHomo sapiens (human)Potency25.118910
N-(3,5-dichlorophenyl)-2-[[4-methyl-5-[4-methyl-2-(5-methyl-3-isoxazolyl)-5-thiazolyl]-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency2.511910
N-(4-chlorophenyl)-2-[[4-methyl-5-[4-methyl-2-(5-methyl-3-isoxazolyl)-5-thiazolyl]-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency15.848910
N-(4-chlorophenyl)-5-methyl-2-[(4-methylphenyl)methyl]-3-pyrazolecarboxamideHomo sapiens (human)Potency12.589310
2-[(4-chlorophenyl)thio]-1-methyl-3-indolecarboxaldehydeHomo sapiens (human)Potency10.000010
3-[5-[anilino(oxo)methyl]-2-furanyl]-2-thiophenecarboxylic acid methyl esterHomo sapiens (human)Potency10.000010
4-(dimethylamino)-3-[(phenylmethoxyamino)methylideneamino]-2-thieno[2,3-b]pyridinecarboxylic acid ethyl esterHomo sapiens (human)Potency25.118910
3-(methylthio)-4-oxo-6,7-dihydro-5H-2-benzothiophene-1-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
2-(4-nitrophenyl)-N-(2-oxolanylmethyl)-4-quinazolinamineHomo sapiens (human)Potency12.589310
4-benzyl-N-(3,5-dichlorophenyl)-1,4-diazepane-1-carboxamideHomo sapiens (human)Potency15.848910
4-[5-chloro-6-methyl-2-(2-pyridinyl)-4-pyrimidinyl]morpholineHomo sapiens (human)Potency25.118910
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineHomo sapiens (human)Potency15.848910
4-(2-hydroxyphenyl)-8,9-dimethyl-2,3-dihydro-1H-1,5-benzodiazepin-2-oneHomo sapiens (human)Potency25.118910
2-({[2-acetyl-5-(tert-butyl)-3-thienyl]amino}carbonyl)benzoic acidHomo sapiens (human)Potency5.514650
5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamideHomo sapiens (human)Potency5.011910
(4-methylphenyl)-[4-[4-nitro-2-(1-pyrrolyl)phenyl]-1-piperazinyl]methanoneHomo sapiens (human)Potency10.000010
4-fluoro-N-(7-methyl-4-oxo-2-thieno[3,2-d][1,3]thiazinyl)benzamideHomo sapiens (human)Potency10.000010
2-[[2-[[5-(4-tert-butylphenyl)-2-methoxycarbonyl-3-thiophenyl]amino]-2-oxoethyl]thio]acetic acidHomo sapiens (human)Potency12.589310
6-methyl-2-[[(4-methylanilino)-oxomethyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
[4-(2-methoxyphenyl)-1-piperidinyl]-(5-methyl-1-phenyl-4-pyrazolyl)methanoneHomo sapiens (human)Potency25.118910
4-(3,5-dichloro-4-pyridinyl)-N-(1-naphthalenyl)-1,4-diazepane-1-carboxamideHomo sapiens (human)Potency12.589310
1-(3,5-dimethylphenyl)-3-[5-(dimethylsulfamoyl)-2-methylphenyl]ureaHomo sapiens (human)Potency15.848910
4-acetamidobenzenesulfonic acid [2-(1-piperidinyl)phenyl] esterHomo sapiens (human)Potency12.589310
5-tert-butyl-N-[5-(dimethylsulfamoyl)-2-methylphenyl]-2-(phenylmethyl)-3-pyrazolecarboxamideHomo sapiens (human)Potency10.000010
1-(2-fluorophenyl)-3-[2-(1-piperidinyl)phenyl]ureaHomo sapiens (human)Potency2.511910
4-(9H-fluoren-9-yl)-N-phenyl-1-piperazinecarboxamideHomo sapiens (human)Potency10.000010
N-(3-chlorophenyl)-4-(9H-fluoren-9-yl)-1-piperazinecarboxamideHomo sapiens (human)Potency12.589310
4-[[5-ethyl-3-[(4-methoxyphenyl)-oxomethyl]-2-thiophenyl]amino]-4-oxobutanoic acidHomo sapiens (human)Potency5.011910
2-[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]-5-[4-(trifluoromethyl)phenyl]-1,3,4-oxadiazoleHomo sapiens (human)Potency12.589310
4-(2-furanylmethyl)-3-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency3.981110
LSM-28160Homo sapiens (human)Potency25.118910
3-(2,4-dimethoxyphenyl)-6-phenyl-2-sulfanylidene-1H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency7.943310
4-(1-piperidinyl)-3-[[3-(trifluoromethyl)phenyl]sulfonylamino]benzoic acid ethyl esterHomo sapiens (human)Potency10.000010
1-[2-(4-chlorophenyl)sulfonylethyl]-1-ethyl-3-phenylureaHomo sapiens (human)Potency3.981110
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)Potency5.011910
1-(3-chloro-4-propan-2-ylsulfonyl-2-thiophenyl)-3-(3-nitrophenyl)ureaHomo sapiens (human)Potency12.589310
N-phenyl-2-benzo[g][1]benzothiolecarboxamideHomo sapiens (human)Potency12.589310
2,4-dichloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamideHomo sapiens (human)Potency19.952610
2-(1-naphthalenyl)-N-[2,2,2-trichloro-1-[[(2-chloroanilino)-sulfanylidenemethyl]amino]ethyl]acetamideHomo sapiens (human)Potency10.000010
2-[2-[bis(4-methoxyphenyl)methylidene]hydrazinyl]benzoic acidHomo sapiens (human)Potency7.943310
2-amino-7-methyl-5-oxo-4-(2,4,5-trimethoxyphenyl)-4,6,7,8-tetrahydro-1-benzopyran-3-carbonitrileHomo sapiens (human)Potency3.162310
3-[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-1-phenylpyrrolidine-2,5-dioneHomo sapiens (human)Potency0.004010
dihydrosamidineHomo sapiens (human)Potency10.000010
4-(5,6-diphenyl-1,2,4-triazin-3-yl)morpholineHomo sapiens (human)Potency10.000010
1-hexadecyl-3-methylimidazolium bromideHomo sapiens (human)Potency25.118910
N-(4-methylphenyl)-5-nitro-4-spiro[benzimidazole-2,1'-cyclohexane]amineHomo sapiens (human)Potency12.589310
3-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) esterHomo sapiens (human)Potency12.589310
4-methyl-2-[(4-methylphenyl)sulfonylamino]pentanoic acid (4-oxo-2,3-dihydro-1H-cyclopenta[c][1]benzopyran-7-yl) esterHomo sapiens (human)Potency10.000010
2-[[oxo(thiophen-2-yl)methyl]amino]-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)Potency12.589310
N-(3-acetyl-2-methyl-5-benzofuranyl)-N-(4-chloro-3-nitrophenyl)sulfonylacetamideHomo sapiens (human)Potency10.000010
4-[3-[[(2,5-dichloroanilino)-methyliminomethyl]thio]-2,5-dioxo-1-pyrrolidinyl]benzoic acid methyl esterHomo sapiens (human)Potency10.000010
N2-tert-butyl-6-ethoxy-N4-(4-nitrophenyl)-1,3,5-triazine-2,4-diamineHomo sapiens (human)Potency10.000010
LSM-19241Homo sapiens (human)Potency10.000010
N-[(2-chlorophenyl)-(2-hydroxy-1-naphthalenyl)methyl]butanamideHomo sapiens (human)Potency12.589310
N-(5-bromo-2-pyridinyl)-2,2-dimethyl-3-(2-methylprop-1-enyl)-1-cyclopropanecarboxamideHomo sapiens (human)Potency12.589310
LSM-19663Homo sapiens (human)Potency10.000010
2-(2,4-dichlorophenyl)-3-(phenylmethyl)-1,2-dihydroquinazolin-4-oneHomo sapiens (human)Potency10.000010
N-[1-[[anilino(sulfanylidene)methyl]amino]-2,2,2-trichloroethyl]-2-(4-ethylphenoxy)acetamideHomo sapiens (human)Potency12.589310
2-[(4-chlorophenyl)thio]-N-[4-[(2,4-dimethylphenyl)sulfamoyl]phenyl]propanamideHomo sapiens (human)Potency10.000010
3-oxo-2-[(6-oxo-1-phenyl-3-pyridazinyl)oxy]butanoic acid ethyl esterHomo sapiens (human)Potency2.511910
eskazineHomo sapiens (human)Potency25.118910
1-[4-(3-ethoxyphenoxy)butyl]imidazoleHomo sapiens (human)Potency12.589310
3-acetamidobenzoic acid [2-(4-methylphenyl)-2-oxo-1-phenylethyl] esterHomo sapiens (human)Potency10.000010
4-[[3-[2-(1-cyclohexenyl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazolin-7-yl]-oxomethyl]-1-piperazinecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
N-[3-(2-furanyl)-3-phenylpropyl]-4-methylbenzenesulfonamideHomo sapiens (human)Potency25.118910
1-adamantyl-[4-(2-fluorophenyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency12.589310
6-[[(2-methoxycarbonyl-3-thiophenyl)amino]-oxomethyl]-1-cyclohex-3-enecarboxylic acidHomo sapiens (human)Potency12.589310
1-[2-[[4,6-bis(1-piperidinyl)-1,3,5-triazin-2-yl]oxy]ethyl]-3-phenylureaHomo sapiens (human)Potency10.000010
9-[2-hydroxy-3-(2-methyl-1-benzimidazolyl)propyl]-6-methyl-3,4-dihydro-2H-carbazol-1-oneHomo sapiens (human)Potency10.000010
LSM-19894Homo sapiens (human)Potency10.000010
4-[hydroxy(diphenyl)methyl]-N-(2-phenylethyl)-1-piperidinecarbothioamideHomo sapiens (human)Potency10.000010
N-[3-(4-chlorophenyl)-2-methyl-3H-1,5-benzodiazepin-4-yl]benzamideHomo sapiens (human)Potency10.000010
N-([biphenyl]-2-yl)-3-cyclopentylpropanamideHomo sapiens (human)Potency12.589310
4-(5-(4-methoxyphenyl)-3-phenyl-4,5-dihydro-1h-pyrazol-1-yl)benzenesulfonamideHomo sapiens (human)Potency12.589310
N-[amino-[2-(1H-indol-3-yl)ethylimino]methyl]-4-chlorobenzamideHomo sapiens (human)Potency12.589310
4-[[2-(4-ethyl-3-oxo-2-morpholinyl)-1-oxoethyl]amino]benzoic acid ethyl esterHomo sapiens (human)Potency5.011910
N-[3-chloro-4-[4-[oxo-(4-propoxyphenyl)methyl]-1-piperazinyl]phenyl]propanamideHomo sapiens (human)Potency7.943310
1-[1-(1-adamantyl)butyl]-3-(2-oxolanylmethyl)thioureaHomo sapiens (human)Potency10.000010
2-(1,3-benzothiazol-2-ylamino)-5-spiro[1,6,7,8-tetrahydroquinazoline-4,1'-cyclopentane]oneHomo sapiens (human)Potency5.011910
N'-(9-acridinyl)-2-(3-methylphenoxy)acetohydrazideHomo sapiens (human)Potency12.589310
2-[(4-ethyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)thio]-N-(2-methoxy-3-dibenzofuranyl)acetamideHomo sapiens (human)Potency12.589310
3-(5-chloro-2-hydroxyphenyl)-3-phenyl-N-[(4-propan-2-yloxyphenyl)methyl]propanamideHomo sapiens (human)Potency10.000010
1-[4-[4-[[6-bromo-2-(3-pyridinyl)-4-quinolinyl]-oxomethyl]-1-piperazinyl]phenyl]ethanoneHomo sapiens (human)Potency3.981110
N-(2-methoxy-3-dibenzofuranyl)-2-oxolanecarboxamideHomo sapiens (human)Potency12.589310
[3-(2-hydroxyphenyl)-5-phenyl-3,4-dihydropyrazol-2-yl]-phenylmethanoneHomo sapiens (human)Potency10.000010
1-[(4-tert-butylphenyl)methyl]-4-(4-nitrophenyl)imidazoleHomo sapiens (human)Potency15.848910
N-[3-chloro-4-[4-[2-furanyl(oxo)methyl]-1-piperazinyl]phenyl]-2-(4-chlorophenyl)acetamideHomo sapiens (human)Potency12.589310
2-[[4-(4-fluorophenyl)-6-(trifluoromethyl)-2-pyrimidinyl]sulfonyl]acetic acid ethyl esterHomo sapiens (human)Potency12.589310
2-[1-(4-chlorophenyl)-5-oxo-3-(2-pyridin-4-ylethyl)-2-sulfanylidene-4-imidazolidinyl]-N-(4-fluorophenyl)acetamideHomo sapiens (human)Potency10.000010
LSM-18518Homo sapiens (human)Potency12.589310
2-[3-oxo-1-[[[oxo(thiophen-2-yl)methyl]amino]-sulfanylidenemethyl]-2-piperazinyl]acetic acid propan-2-yl esterHomo sapiens (human)Potency25.118910
4-[(1-ethyl-6-methyl-4-pyrazolo[3,4-b]pyridinyl)oxymethyl]benzonitrileHomo sapiens (human)Potency12.589310
2-[[[4-(4-methoxyphenyl)-5-phenyl-1,2,4-triazol-3-yl]thio]methyl]-5-phenyl-1,3,4-oxadiazoleHomo sapiens (human)Potency10.000010
4-[[[5-(2,3-dihydro-1,4-benzodioxin-3-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]thio]methyl]-3,5-dimethylisoxazoleHomo sapiens (human)Potency10.000010
1-(2-methoxy-5-methylphenyl)-5-(2-oxanylmethylthio)tetrazoleHomo sapiens (human)Potency10.000010
5-[[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]methyl]-2-furancarboxylic acid methyl esterHomo sapiens (human)Potency12.589310
4-(diethylamino)benzoic acid [2-oxo-2-(4-phenyl-1-piperazinyl)ethyl] esterHomo sapiens (human)Potency10.000010
2-(4-cyanophenoxy)-N-(2-methyl-1-phenyl-5-benzimidazolyl)acetamideHomo sapiens (human)Potency12.589310
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamideHomo sapiens (human)Potency25.118910
4-chloro-N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideHomo sapiens (human)Potency10.000010
2-(1,3-diphenyl-4-pyrazolyl)-3-(2-furanylmethyl)-4-thiazolidinoneHomo sapiens (human)Potency12.589310
3-(2,5-dimethyl-3-furanyl)-5,6-diphenyl-1,2,4-triazineHomo sapiens (human)Potency10.000010
[4-(2-pyridinyl)-1-piperazinyl]-[2-(3,4,5-trimethoxyphenyl)-4-quinolinyl]methanoneHomo sapiens (human)Potency12.589310
3-hydroxy-2-naphthalenecarboxylic acid [2-(3,5-dimethyl-1-piperidinyl)-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
2-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)benzoic acid thiophen-2-ylmethyl esterHomo sapiens (human)Potency12.589310
1-(4-fluorophenyl)-3-methyl-5-thieno[2,3-c]pyrazolecarboxylic acid (2-oxo-3-oxolanyl) esterHomo sapiens (human)Potency31.622810
2-(4-chloro-2-methylphenoxy)-N-[2-(4-morpholinyl)phenyl]propanamideHomo sapiens (human)Potency10.000010
1-butyl-2-[(5-phenyl-2-oxazolyl)methylthio]-5-benzimidazolesulfonamideHomo sapiens (human)Potency12.589310
3-(4-methylphenyl)sulfonyl-1-(3-oxolanylmethyl)-2-pyrrolo[3,2-b]quinoxalinamineHomo sapiens (human)Potency25.118910
N-(1-propyl-2-benzimidazolyl)-3-(1-pyrrolidinylsulfonyl)benzamideHomo sapiens (human)Potency15.848910
LSM-1318Homo sapiens (human)Potency10.000010
trequinsin hydrochlorideHomo sapiens (human)Potency10.000010
emetine dihydrochlorideHomo sapiens (human)Potency2.511910
4-methoxy-N-[2,2,2-trichloro-1-(4-methylanilino)ethyl]benzamideHomo sapiens (human)Potency25.118910
3-chloro-N-[2,2,2-trichloro-1-[[(4-methoxy-2-nitroanilino)-sulfanylidenemethyl]amino]ethyl]benzamideHomo sapiens (human)Potency10.000010
3-O-AcetylepisamarcandinHomo sapiens (human)Potency12.589310
2-[[2,2,2-trichloro-1-[(2-methyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
2-[[2,2,2-trichloro-1-[(2,2-dimethyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl esterHomo sapiens (human)Potency12.589310
1-[1-chloro-2-[(2-nitrophenyl)thio]-4-phenyl-2,3,3a,4,5,9b-hexahydro-1H-cyclopenta[c]quinolin-8-yl]ethanoneHomo sapiens (human)Potency10.000010
phenyl-(2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)methanoneHomo sapiens (human)Potency10.000010
3,5-dimethyl-2,6-bis(4-methylphenyl)-4-piperidinoneHomo sapiens (human)Potency25.118910
2-[(prop-2-enylthio)-(4,5,6,7-tetrahydro-1H-indol-2-yl)methylidene]propanedinitrileHomo sapiens (human)Potency12.589310
acetic acid [1-[(3-nitrophenyl)-(1-oxopentylamino)methyl]-2-naphthalenyl] esterHomo sapiens (human)Potency12.589310
9-(1H-indol-3-yl)acridineHomo sapiens (human)Potency10.000010
N-(2,5-dimethoxyphenyl)-4-(2,4-dimethyl-5-thiazolyl)-2-thiazolamineHomo sapiens (human)Potency7.943310
6-amino-5,7,7-tricyano-8-pyridin-4-yl-1,3,8,8a-tetrahydroisoquinoline-2-carboxylic acid (phenylmethyl) esterHomo sapiens (human)Potency3.981110
6-amino-4-(5-chloro-2-thiophenyl)-5-cyano-2-phenyl-4H-pyran-3-carboxylic acid ethyl esterHomo sapiens (human)Potency31.622810
4-mercapto-6-oxo-3-phenyl-2-thiophen-2-yl-1,2-dihydropyrimidine-5-carbonitrileHomo sapiens (human)Potency25.118910
2-(4-ethoxy-3-methoxyphenyl)-4-mercapto-3-(4-methoxyphenyl)-6-oxo-1,2-dihydropyrimidine-5-carbonitrileHomo sapiens (human)Potency12.589310
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneHomo sapiens (human)Potency7.943310
2-[[5-(phenoxymethyl)-4-phenyl-1,2,4-triazol-3-yl]thio]acetonitrileHomo sapiens (human)Potency12.589310
N-[4-(2,5-dimethoxyphenyl)-2-thiazolyl]-N-(2-oxolanylmethyl)cyclohexanecarboxamideHomo sapiens (human)Potency10.000010
N-[2-(tert-butylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2-oxolanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideHomo sapiens (human)Potency12.589310
N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-5-methyl-N-(thiophen-2-ylmethyl)-2,1,3-benzothiadiazole-4-sulfonamideHomo sapiens (human)Potency10.000010
4-(2-azaspiro[5.5]undecan-2-ylsulfonyl)-N-butan-2-ylbenzenesulfonamideHomo sapiens (human)Potency10.000010
2-[(3,6-dimethyl-2-quinolinyl)thio]-1-(2-methyl-2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency10.000010
2-[cyclopentyl-[1-oxo-2-(5-thiophen-2-yl-2-tetrazolyl)ethyl]amino]-N-(2-oxolanylmethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency10.000010
[4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency10.000010
2-[(5,6-dimethyl-2-propyl-4-thieno[2,3-d]pyrimidinyl)thio]-1-(2-methyl-2,3-dihydroindol-1-yl)ethanoneHomo sapiens (human)Potency7.943310
2-(N-[2-(Benzotriazol-1-yl)acetyl]-2,4,6-trimethylanilino)-N-tert-butyl-2-thiophen-3-ylacetamideHomo sapiens (human)Potency10.000010
2-[(3-cyano-8-methyl-2-quinolinyl)thio]-N-(2-oxolanylmethyl)acetamideHomo sapiens (human)Potency25.118910
N-(2,4-dioxo-1H-pyrimidin-5-yl)-2-[(3-ethyl-5,8-dimethyl-2-quinolinyl)thio]acetamideHomo sapiens (human)Potency12.589310
N-[2-(cyclohexylamino)-2-oxo-1-(6-quinolinyl)ethyl]-N-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency12.589310
2-[2-methoxyethyl-(1-oxo-2-thiophen-2-ylethyl)amino]-N-[(4-methoxyphenyl)methyl]-2-(4-propan-2-ylphenyl)acetamideHomo sapiens (human)Potency25.118910
2-chloro-N-[1-[oxo(10-phenothiazinyl)methyl]-4-piperidinyl]benzamideHomo sapiens (human)Potency12.589310
1-cyclopentyl-1-[2-(5,6-dimethyl-1H-benzimidazol-2-yl)ethyl]-3-(2-oxolanylmethyl)thioureaHomo sapiens (human)Potency12.589310
3,4-dihydro-2H-quinolin-1-yl-[4-(phenylmethyl)-5-thieno[3,2-b]pyrrolyl]methanoneHomo sapiens (human)Potency10.000010
N-[2-(1H-indol-3-yl)ethyl]-4-(phenylmethyl)-5-thieno[3,2-b]pyrrolecarboxamideHomo sapiens (human)Potency12.589310
N,N-dimethyl-4-[[3-[3-(5-methyl-2-furanyl)-1,2,4-oxadiazol-5-yl]-1-piperidinyl]sulfonyl]benzenesulfonamideHomo sapiens (human)Potency15.848910
[4-[5-tert-butyl-3-(phenylmethyl)-7-triazolo[4,5-d]pyrimidinyl]-1-piperazinyl]-(2-furanyl)methanoneHomo sapiens (human)Potency10.000010
1-(2-methyl-2,3-dihydroindol-1-yl)-2-[4-[5-(trifluoromethyl)-1-benzotriazolyl]-1-piperidinyl]ethanoneHomo sapiens (human)Potency31.622810
1-(1-tert-butyl-5-tetrazolyl)-N-(2-furanylmethyl)-N-(phenylmethyl)-1-[4-(trifluoromethyl)phenyl]methanamineHomo sapiens (human)Potency15.848910
1-(1-tert-butyl-5-tetrazolyl)-N-(phenylmethyl)-1-(3-pyridinyl)-N-(thiophen-2-ylmethyl)methanamineHomo sapiens (human)Potency10.000010
7-(2-ethyl-1-piperidinyl)-5-methyl-2-(3-methylphenyl)pyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency12.589310
4-[butan-2-yl-[(3,4-dichloroanilino)-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency31.622810
3-[6-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-6-oxohexyl]-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency25.118910
N-(4-methyl-5-oxo-2-[1]benzopyrano[4,3-b]pyridinyl)-4-(1-pyrrolidinylsulfonyl)benzamideHomo sapiens (human)Potency1.000010
5-amino-1-[2-(2-ethoxyanilino)-2-oxoethyl]-N-(2-furanylmethyl)-4-triazolecarboxamideHomo sapiens (human)Potency5.011910
N-[2-(1-cyclohexenyl)ethyl]-2-(4-oxo-1-[1]benzopyrano[4,3-c]pyrazolyl)acetamideHomo sapiens (human)Potency3.162310
2-[(6-fluoro-1,3-benzothiazol-2-yl)amino]-4-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
2-[(3-methoxyphenyl)-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
6-bromo-3-[4-oxo-4-[4-(2-pyridinyl)-1-piperazinyl]butyl]-2-sulfanylidene-1H-quinazolin-4-oneHomo sapiens (human)Potency12.589310
3-chloro-N-[2-[4-(4-fluorophenyl)-1-piperazinyl]-2-(3-pyridinyl)ethyl]benzamideHomo sapiens (human)Potency12.589310
2-[8-[[bis(phenylmethyl)amino]methyl]-3-methyl-2,6-dioxo-7-purinyl]acetic acid ethyl esterHomo sapiens (human)Potency10.000010
N-(1,3-benzodioxol-5-yl)-3-(1-ethyl-5-methyl-4-pyrazolyl)-4,5-dihydroisoxazole-5-carboxamideHomo sapiens (human)Potency1.584910
2-[(3,5-dimethyl-4-isoxazolyl)methylthio]-4-ethyl-7,7-dimethyl-5-oxo-6,8-dihydroquinoline-3-carbonitrileHomo sapiens (human)Potency12.589310
2-[[4-[(2,6-dimethyl-4-morpholinyl)sulfonyl]phenyl]-oxomethyl]imino-3,4-dimethyl-5-thiazolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
4-morpholinecarboxylic acid [4-[6-amino-5-cyano-3-(4-methylphenyl)-2,4-dihydropyrano[2,3-c]pyrazol-4-yl]phenyl] esterHomo sapiens (human)Potency6.309610
5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinolHomo sapiens (human)Potency3.162310
4-(2,3-dihydroindol-1-yl)-N-[3-(N-ethyl-3-methylanilino)propyl]-3-(1-imidazolyl)-4-oxobutanamideHomo sapiens (human)Potency10.000010
N-(3-chlorophenyl)-2-[1-(3,4-dimethylphenyl)-4-oxo-5-pyrazolo[3,4-d]pyrimidinyl]acetamideHomo sapiens (human)Potency12.589310
N-(2-methyl-4-oxo-1-propyl-6-quinolinyl)-2-pyrazinecarboxamideHomo sapiens (human)Potency31.622810
1-(4-chlorophenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-4-pyrazolecarboxylic acidHomo sapiens (human)Potency5.011910
2-(3-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency25.118910
5-bromo-N-[2-(2-chlorophenyl)-1,3-benzoxazol-5-yl]-3-pyridinecarboxamideHomo sapiens (human)Potency25.118910
4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl(3,4-dihydro-2H-quinolin-1-yl)methanoneHomo sapiens (human)Potency12.589310
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[N-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-methylanilino]acetamideHomo sapiens (human)Potency5.011910
3-chloro-4-ethoxy-N-[3-(2-oxazolo[5,4-b]pyridinyl)phenyl]benzamideHomo sapiens (human)Potency12.589310
3,8-dimethyl-4-oxo-7,8,9,10-tetrahydro-6H-thieno[1,2]pyrimido[4,5-a]azepine-2-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
3-[[2-furanyl(oxo)methyl]amino]-N-(4-methoxyphenyl)-2-benzofurancarboxamideHomo sapiens (human)Potency10.000010
1-[4-[4-[[1-(4-chlorophenyl)sulfonylcyclopropyl]-oxomethyl]-1-piperazinyl]phenyl]ethanoneHomo sapiens (human)Potency0.631010
3-pyridinecarboxylic acid 2-[[oxo-(2-oxo-1-benzopyran-3-yl)methyl]amino]ethyl esterHomo sapiens (human)Potency5.011910
[1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-3-piperidinyl]-(2-methyl-2,3-dihydroindol-1-yl)methanoneHomo sapiens (human)Potency10.000010
2-(4-ethoxyphenyl)-5-[1-[(2-methylpropan-2-yl)oxy-oxomethyl]-4-piperidinyl]-6-pyrazolo[1,5-a]pyrimidinecarboxylic acidHomo sapiens (human)Potency15.848910
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-piperidinecarboxamideHomo sapiens (human)Potency12.589310
1-[[4-[(4-fluorophenyl)methyl]-5-thieno[3,2-b]pyrrolyl]-oxomethyl]-N-(2-furanylmethyl)-4-piperidinecarboxamideHomo sapiens (human)Potency6.309610
5-(6,7-diethoxy-4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)-N-(2-furanylmethyl)pentanamideHomo sapiens (human)Potency25.118910
4-[[2-(3-ethylanilino)-3,4-dioxo-1-cyclobutenyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency1.258910
4-[2-[(2-ethoxy-2-oxoethyl)thio]-4-oxo-3-thieno[3,2-d]pyrimidinyl]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency3.162310
N-ethyl-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(phenylmethyl)propanamideHomo sapiens (human)Potency7.943310
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-piperidinecarboxamideHomo sapiens (human)Potency25.118910
3-(2-furanylmethyl)-5-(2-methoxyethyl)-1,3,5-thiadiazinane-2-thioneHomo sapiens (human)Potency3.162310
2-[[2-(2-ethyl-1-piperidinyl)-2-oxoethyl]thio]-3-methyl-5H-pyrimido[5,4-b]indol-4-oneHomo sapiens (human)Potency15.848910
7-[(4-methyl-1-piperazinyl)methyl]-5-(phenylmethoxymethyl)-8-quinolinolHomo sapiens (human)Potency3.162310
3,4-dihydro-2H-quinolin-1-yl-[5-(4-methoxyphenyl)-3-isoxazolyl]methanoneHomo sapiens (human)Potency15.848910
6-(1-azepanylsulfonyl)-1-ethyl-N-(2-furanylmethyl)-4-oxo-3-quinolinecarboxamideHomo sapiens (human)Potency6.309610
3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamideHomo sapiens (human)Potency1.584910
N-(1,3-benzodioxol-5-yl)-5-bromo-1-[cyclopropyl(oxo)methyl]-N-ethyl-2,3-dihydroindole-7-sulfonamideHomo sapiens (human)Potency10.000010
N-(3,4-dimethylphenyl)-2-[N-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-methoxyanilino]acetamideHomo sapiens (human)Potency10.000010
N-[(4-chlorophenyl)methyl]-3-(1-ethyl-5-methyl-4-pyrazolyl)-4,5-dihydroisoxazole-5-carboxamideHomo sapiens (human)Potency2.511910
N-[[4-(dimethylamino)phenyl]methyl]-3-ethyl-N-(2-furanylmethyl)-5-methyl-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamideHomo sapiens (human)Potency0.398110
3-(4-chlorophenyl)-2-(1-pyrrolidinyl)-4-quinazolinoneHomo sapiens (human)Potency12.589310
N-ethyl-N-(2-ethylphenyl)-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamideHomo sapiens (human)Potency5.011910
N-(2-furanylmethyl)-5,7-dimethyl-6-[(3-methylphenyl)methyl]-3-pyrazolo[1,5-a]pyrimidinecarboxamideHomo sapiens (human)Potency12.589310
4-[[3-[(2-furanylmethylamino)-oxomethyl]-7-methoxy-1-benzopyran-2-ylidene]amino]benzoic acidHomo sapiens (human)Potency12.589310
2-(2-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-oneHomo sapiens (human)Potency19.952610
1-methyl-N-(2-methylcyclohexyl)-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamideHomo sapiens (human)Potency12.589310
cyclopentanecarboxylic acid [4-(benzenesulfonyl)-2-tert-butyl-5-methyl-3-pyrazolyl] esterHomo sapiens (human)Potency12.589310
N-[3-(cyclohexylthio)propyl]-1-[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]-3-piperidinecarboxamideHomo sapiens (human)Potency12.589310
3-[[oxo(thiophen-2-yl)methyl]amino]-2-benzofurancarboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
[3-(4-methylphenyl)-1-phenyl-4-pyrazolyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency7.943310
N-[[3-[(3-chlorophenyl)sulfamoyl]-4-methylanilino]-sulfanylidenemethyl]-4-fluorobenzamideHomo sapiens (human)Potency10.000010
3-(2-furanyl)-N-[3-(2-furanyl)-4-methylpentyl]-4-phenylbutanamideHomo sapiens (human)Potency15.848910
2,6-dimethyl-4-(4-phenyl-2-quinolinyl)morpholineHomo sapiens (human)Potency19.952610
n-(1-methyl-5-indolyl)-n'-(3-methyl-5-isothiazolyl)ureaHomo sapiens (human)Potency1.000010
4-[3-(1,3-diphenyl-4-pyrazolyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-4-oxobutanoic acidHomo sapiens (human)Potency12.589310
4-[[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]methyl]morpholineHomo sapiens (human)Potency10.000010
gw 7647Homo sapiens (human)Potency10.000010
N-[4-[2-(2-ethyl-1-oxobutyl)-3-phenyl-3,4-dihydropyrazol-5-yl]phenyl]methanesulfonamideHomo sapiens (human)Potency12.589310
4-butyl-3-(6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency25.118910
4-[3-methyl-5-(4-methylphenyl)-6-oxo-2,4-dihydropyrrolo[3,4-c]pyrazol-4-yl]benzoic acid methyl esterHomo sapiens (human)Potency0.501210
1,1-dimethyl-3-[3-(4-morpholinyl)propyl]-3-(1-naphthalenylmethyl)ureaHomo sapiens (human)Potency15.848910
2-(4-benzofuro[3,2-d]pyrimidinylthio)-N-(3-methylphenyl)acetamideHomo sapiens (human)Potency25.118910
5-[3-[3-(4-methoxyphenyl)-1-phenyl-4-pyrazolyl]-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acidHomo sapiens (human)Potency12.589310
6-[2-butylimino-3-(cyclopentylideneamino)-4-thiazolyl]-4H-1,4-benzoxazin-3-oneHomo sapiens (human)Potency12.589310
LSM-16990Homo sapiens (human)Potency5.011910
3-(3-chloro-2-methylphenyl)-1-[(4-methylphenyl)methyl]-1-(3-pyridinylmethyl)thioureaHomo sapiens (human)Potency25.118910
cgp 13501Homo sapiens (human)Potency12.589310
(S)-4',5,7-Trihydroxy-6-prenylflavanoneHomo sapiens (human)Potency12.589310
2-[[1-(phenylmethyl)-3-indolyl]thio]-N-(2-thiazolyl)acetamideHomo sapiens (human)Potency10.000010
N-[5-ethyl-3-[(4-fluorophenyl)-(4-morpholinyl)methyl]-2-thiophenyl]benzamideHomo sapiens (human)Potency10.000010
3-(4-benzoyl-1-piperazinyl)-1-(2-methylpropyl)-6,7-dihydro-5H-cyclopenta[c]pyridine-4-carbonitrileHomo sapiens (human)Potency1.995310
6-bromo-2-(4-methylphenyl)-N-[(1-methyl-4-pyrazolyl)methyl]-4-quinolinecarboxamideHomo sapiens (human)Potency10.000010
1-[2-[(4-chlorophenyl)thio]ethyl]-3-(4-methylphenyl)thioureaHomo sapiens (human)Potency10.000010
4-(4-chlorophenyl)-N-[3-[(4-methoxyphenyl)sulfamoyl]phenyl]-4-oxobutanamideHomo sapiens (human)Potency12.589310
2-[2-[(5-chloro-2-thiophenyl)-oxomethyl]imino-6-fluoro-1,3-benzothiazol-3-yl]acetic acid methyl esterHomo sapiens (human)Potency12.589310
2-[4-methoxy-3-(4-morpholinylmethyl)phenyl]-3-(phenylmethyl)-1,2-dihydroquinazolin-4-oneHomo sapiens (human)Potency25.118910
5-chloro-N-(1,3-dioxo-5-isoindolyl)-2-thiophenecarboxamideHomo sapiens (human)Potency19.952610
1-[(2,6-dichlorophenyl)methyl]-5-(4-methylphenyl)-2-oxo-3-pyridinecarbonitrileHomo sapiens (human)Potency10.000010
l 663536Homo sapiens (human)Potency10.000010
mrs 1523Homo sapiens (human)Potency12.589310
ML162Homo sapiens (human)Potency12.589310
2-(N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamideHomo sapiens (human)Potency12.589310
2-(cyclohexylamino)-N-[(diphenylmethylene)amino]propanamideHomo sapiens (human)Potency12.589310
2-[(2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)oxy]-N-heptylacetamideHomo sapiens (human)Potency25.118910
N-[2-[[2-(4-chlorophenyl)-2-oxoethyl]thio]-4-oxo-3-quinazolinyl]benzamideHomo sapiens (human)Potency19.952610
2-[(4-amino-7-tert-butyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)thio]acetic acidHomo sapiens (human)Potency12.589310
3-ethyl-2-sulfanylidene-5-thiophen-2-yl-1H-thieno[2,3-d]pyrimidin-4-oneHomo sapiens (human)Potency10.000010
LSM-1924Homo sapiens (human)Potency39.131770
2-[1-(2-methylphenyl)-3-oxo-3-thiophen-2-ylpropyl]propanedinitrileHomo sapiens (human)Potency10.000010
1-[(4-chlorophenyl)methyl]-3-(3-fluorophenyl)-1-(3,3,3-trifluoro-2-hydroxypropyl)ureaHomo sapiens (human)Potency19.952610
N-(3-chlorophenyl)-5-oxo-9b-phenyl-2,3-dihydroimidazo[2,1-a]isoindole-1-carboxamideHomo sapiens (human)Potency12.589310
2-(4-chlorophenyl)-5-methyl-4-oxo-2,3-dihydro-1H-thieno[3,4-d]pyrimidine-7-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
5-chloro-4-[methoxy(phenyl)methyl]-1-methyl-3-phenylpyrazoleHomo sapiens (human)Potency12.589310
4-[[anilino-(4-methylphenyl)methyl]-propoxyphosphoryl]-N,N-dimethylanilineHomo sapiens (human)Potency19.952610
1-butyl-4,6-dimethyl-3-(2-methylphenyl)sulfonyl-2-pyridinoneHomo sapiens (human)Potency12.589310
1-ethyl-3-[[2-[(1-methyl-2-benzimidazolyl)thio]-1-oxoethyl]amino]thioureaHomo sapiens (human)Potency5.011910
5-(benzenesulfonyl)-4-(2,6-dimethylphenoxy)-2-phenylpyrimidineHomo sapiens (human)Potency12.589310
2-[[2-(1-adamantyl)-2-oxoethyl]thio]-6-amino-4-(4-chlorophenyl)pyridine-3,5-dicarbonitrileHomo sapiens (human)Potency3.162310
1-[(4-chlorophenyl)methyl]-4-(4-chlorophenyl)sulfonyl-4-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
phosphoric acid (3-methylphenyl) phenyl (2,2,2-trifluoro-1-phenylethyl) esterHomo sapiens (human)Potency10.000010
1-bromo-3-(5,5-dimethyl-3-phenyl-4H-pyrazolo[4,3-a]carbazol-10-yl)-2-propanolHomo sapiens (human)Potency12.589310
2-[4-(3-chlorophenyl)-1-piperazinyl]-3-pyridinecarboxylic acid propan-2-yl esterHomo sapiens (human)Potency10.000010
5-tert-butyl-7-(4-ethyl-1-piperazinyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency12.589310
5,7-dimethyl-3-phenyldiazenyl-1H-pyrazolo[1,5-a]pyrimidin-2-oneHomo sapiens (human)Potency31.622810
2-[(2,6-dichlorophenyl)methyl]-6-phenyl-5-(1-piperidinyl)-3-pyridazinoneHomo sapiens (human)Potency10.000010
2-[2-[5-amino-4-(3-thiophenyl)-1-pyrazolyl]-4-phenyl-5-thiazolyl]acetic acidHomo sapiens (human)Potency3.162310
4-methyl-2-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentanoic acid [3-(4-nitrophenyl)-4-oxo-1-benzopyran-7-yl] esterHomo sapiens (human)Potency12.589310
3-(2,4-dichloro-5-methoxyphenyl)-2-sulfanyl-4(3h)-quinazolinoneHomo sapiens (human)Potency12.589310
1-[4-(3-chlorophenyl)-1-piperazinyl]-2-phenyl-1-butanoneHomo sapiens (human)Potency10.000010
LSM-22738Homo sapiens (human)Potency25.118910
2-[(4-chloro-3-nitrophenyl)-oxomethyl]benzoic acid [2-[di(propan-2-yl)amino]-2-oxoethyl] esterHomo sapiens (human)Potency12.589310
3-[[4-(diphenylmethyl)-1-piperazinyl]-oxomethyl]-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-12-oneHomo sapiens (human)Potency12.589310
2-[(4-hydroxy-3-nitrophenyl)sulfonylamino]benzoic acid [2-(4-methoxyphenyl)-2-oxoethyl] esterHomo sapiens (human)Potency7.943310
4-chloro-5-(2,3-dihydro-1,4-benzodioxin-3-yl)thieno[2,3-d]pyrimidineHomo sapiens (human)Potency10.000010
2-ethyl-4-[[(3-methyl-2-benzofuranyl)-oxomethyl]amino]-1H-1,5-benzodiazepine-3-carboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
2-[(5-anilino-1,3,4-thiadiazol-2-yl)thio]-N-[3-(1-piperidinylsulfonyl)phenyl]acetamideHomo sapiens (human)Potency12.589310
4-(carbamoylamino)benzoic acid [2-(3-chloro-4-methylanilino)-2-oxo-1-phenylethyl] esterHomo sapiens (human)Potency12.589310
4-benzoyl-2-heptyl-5-methyl-4H-pyrazol-3-oneHomo sapiens (human)Potency12.589310
3-[[(3-methoxyphenyl)-oxomethyl]amino]-2-benzofurancarboxamideHomo sapiens (human)Potency25.118910
3,3-bis(4-hydroxy-2-methylphenyl)-1-isobenzofuranoneHomo sapiens (human)Potency15.848910
N-[3-[3-(1-piperidinylsulfonyl)anilino]-2-quinoxalinyl]benzenesulfonamideHomo sapiens (human)Potency10.000010
(6-bromo-5-methoxy-2-methyl-3-benzofuranyl)-[4-(2-methylphenyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency10.000010
2-bromo-N-[[(2-methylcyclohexyl)amino]-sulfanylidenemethyl]benzamideHomo sapiens (human)Potency12.589310
N-(3-methyl-6-methylsulfonyl-1,3-benzothiazol-2-ylidene)-2,3-dihydro-1,4-benzodioxin-6-carboxamideHomo sapiens (human)Potency10.000010
N-(5-phenyl-1,3,4-oxadiazol-2-yl)-1,3-benzothiazole-2-carboxamideHomo sapiens (human)Potency25.118910
1-(3-methyl-1-piperidinyl)-2-(2-quinoxalinylthio)ethanoneHomo sapiens (human)Potency6.309610
iik7Homo sapiens (human)Potency10.000010
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneHomo sapiens (human)Potency10.000010
7-(1-azepanyl)-3-(2-methoxyphenyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)Potency10.000010
LSM-16386Homo sapiens (human)Potency12.589310
3-(4-fluorophenyl)sulfonyl-1-(2-furanylmethyl)-2-imino-10-methyl-5-dipyrido[3,4-c-1',2'-f]pyrimidinoneHomo sapiens (human)Potency10.000010
2-[1-[4-(diethylamino)phenyl]-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-N-phenylacetamideHomo sapiens (human)Potency25.118910
5,5,7,7-tetramethyl-2-[[oxo-(4-propan-2-yloxyphenyl)methyl]amino]-4,6-dihydrothieno[2,3-c]pyridine-3-carboxylic acid methyl esterHomo sapiens (human)Potency6.309610
LSM-26445Homo sapiens (human)Potency12.589310
2-[[4-phenyl-5-(propylthio)-1,2,4-triazol-3-yl]methylthio]-1,3-benzothiazoleHomo sapiens (human)Potency10.000010
LSM-22688Homo sapiens (human)Potency25.118910
1-cyclohexyl-3-[(1,2-dimethyl-5-indolyl)methyl]ureaHomo sapiens (human)Potency25.118910
4-(3-methoxyanilino)-2-methyl-5-oxo-1-phenyl-2-pyrrolecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
3-(4-chloro-1,5-dimethyl-3-pyrazolyl)-4-(4-fluorophenyl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)Potency10.000010
sc 560Homo sapiens (human)Potency10.000010
2-(2-quinoxalinylthio)propanoic acidHomo sapiens (human)Potency7.943310
N4-(2,5-dimethoxyphenyl)-N2-(3-methylbutyl)-5-nitropyrimidine-2,4,6-triamineHomo sapiens (human)Potency12.589310
LSM-16826Homo sapiens (human)Potency19.952610
2-[[2-(cyclohexylamino)-2-oxoethyl]thio]benzoic acid [2-(cyclohexylamino)-2-oxoethyl] esterHomo sapiens (human)Potency25.118910
5-(4-morpholinylsulfonyl)-2-(1-piperidinyl)benzoic acid [2-[[(3-methylbutylamino)-oxomethyl]amino]-2-oxoethyl] esterHomo sapiens (human)Potency25.118910
4-(2,5-dioxo-1-pyrrolidinyl)-N-[4-(4-methoxyphenyl)-2-thiazolyl]benzamideHomo sapiens (human)Potency10.000010
3-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethyl]-1,1-bis(phenylmethyl)ureaHomo sapiens (human)Potency10.000010
N-(3-chlorophenyl)-2-[4-oxo-2-phenylimino-3-(2-pyridinylmethyl)-5-thiazolidinyl]acetamideHomo sapiens (human)Potency15.848910
1-(2-methoxy-3-dibenzofuranyl)-3-(3-methylphenyl)thioureaHomo sapiens (human)Potency12.589310
N-(1-dibutoxyphosphoryl-4-oxo-1-naphthalenyl)benzenesulfonamideHomo sapiens (human)Potency10.000010
N-(4-ethylphenyl)-2-[[3-[3-(4-methyl-1-piperidinyl)propyl]-4-oxo-2-quinazolinyl]thio]acetamideHomo sapiens (human)Potency12.589310
LSM-1925Homo sapiens (human)Potency2.674130
8-[4-(4-fluorophenoxy)-3-nitrophenyl]-7-(2-hydroxyethyl)-3-(phenylmethyl)purine-2,6-dioneHomo sapiens (human)Potency6.309610
3-amino-4-[(4-chlorophenyl)thio]benzoic acid methyl esterHomo sapiens (human)Potency15.848910
N-(1,3-dioxo-5-isoindolyl)-1,3-benzothiazole-6-carboxamideHomo sapiens (human)Potency5.011910
N-[(3,5-dimethyl-1-piperidinyl)-sulfanylidenemethyl]-2-methyl-5-(4-morpholinylsulfonyl)benzamideHomo sapiens (human)Potency25.118910
ly 367265Homo sapiens (human)Potency12.589310
2-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamideHomo sapiens (human)Potency12.589310
5-[(3-methylphenoxy)methyl]-3-[4-(1-pyrrolyl)phenyl]-1,2,4-oxadiazoleHomo sapiens (human)Potency25.118910
LSM-4844Homo sapiens (human)Potency15.848910
N-(3-acetylphenyl)-2-[[6-chloro-3-(2-hydroxypropyl)-4-methyl-2-oxo-1-benzopyran-7-yl]oxy]acetamideHomo sapiens (human)Potency10.000010
4-methoxy-N-(4-methyl-5-oxo-2-[1]benzopyrano[4,3-b]pyridinyl)benzamideHomo sapiens (human)Potency25.118910
2-[4-chloro-2-[3-(4-methoxyphenyl)-4-oxo-1,2-dihydroquinazolin-2-yl]phenoxy]acetic acid methyl esterHomo sapiens (human)Potency10.000010
4-[[2-(1,10b-dihydropyrazolo[1,5-c]quinazolin-5-ylthio)-1-oxoethyl]amino]benzoic acid butyl esterHomo sapiens (human)Potency10.000010
2-phenyl-N-[1-(phenylmethyl)-4-piperidinyl]-4-quinazolinamineHomo sapiens (human)Potency25.118910
4-(4-chlorophenyl)-3-phenyl-1H-imidazole-2-thioneHomo sapiens (human)Potency25.118910
LSM-24516Homo sapiens (human)Potency12.589310
4-(4-chlorophenyl)-3-(phenylmethyl)-1H-imidazole-2-thioneHomo sapiens (human)Potency25.118910
6-[5-chloro-3-methyl-1-(4-methylphenyl)-4-pyrazolyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
2-(1-adamantyl)-N-[2,5-diethoxy-4-(4-morpholinyl)phenyl]acetamideHomo sapiens (human)Potency10.000010
N-(4-tert-butylphenyl)-2-[4-(1-imidazolyl)phenoxy]acetamideHomo sapiens (human)Potency12.589310
8-(4-methoxyphenyl)-7-methyl-3-(phenylmethyl)purine-2,6-dioneHomo sapiens (human)Potency12.589310
LSM-24595Homo sapiens (human)Potency10.000010
LSM-4833Homo sapiens (human)Potency25.118910
1-[[3-(4-chlorophenyl)-4,5-dihydroisoxazol-5-yl]methyl]-4-methyl-2-quinolinoneHomo sapiens (human)Potency12.589310
N-[(4-chlorophenyl)methyl]-2-[[[(2-fluorophenyl)methyl-(phenylmethyl)amino]-sulfanylidenemethyl]amino]acetamideHomo sapiens (human)Potency10.000010
1-(7-methyloctyl)-3-[4-(4-morpholinylsulfonyl)phenyl]thioureaHomo sapiens (human)Potency25.118910
LSM-25964Homo sapiens (human)Potency25.118910
cgp 7930Homo sapiens (human)Potency12.589310
[3-(2-hydroxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-thiophen-2-ylmethanoneHomo sapiens (human)Potency10.000010
1,3,5-tris(4-hydroxyphenyl)-4-propyl-1h-pyrazoleHomo sapiens (human)Potency12.589310
2-(3-methyl-1-oxo-2-isoquinolinyl)-N-(3,4,5-trimethoxyphenyl)acetamideHomo sapiens (human)Potency25.118910
1-(1-adamantyl)-3-[1-(phenylmethyl)-4-pyrazolyl]ureaHomo sapiens (human)Potency10.000010
2-[2-(7-methoxy-2-oxo-1H-quinolin-3-yl)ethyl]isoindole-1,3-dioneHomo sapiens (human)Potency10.000010
2-[[3-[2-(diethylamino)ethyl]-4-oxo-[1]benzothiolo[3,2-d]pyrimidin-2-yl]thio]-N-(phenylmethyl)acetamideHomo sapiens (human)Potency10.000010
[5-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-3-pyrazolyl]-(4-morpholinyl)methanoneHomo sapiens (human)Potency12.589310
5-[(2,4-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-[(2,3,4,5,6-pentafluorophenyl)methyl]-4-pyrazolyl]-2-furancarboxamideHomo sapiens (human)Potency15.848910
N-(5-acetyl-4-methyl-2-thiazolyl)-2-(2,4-dichlorophenoxy)acetamideHomo sapiens (human)Potency12.589310
2-[3-(1-benzotriazolylmethyl)-4-methoxyphenyl]-3-(4-methoxyphenyl)-1,2-dihydroquinazolin-4-oneHomo sapiens (human)Potency7.943310
quercetinHomo sapiens (human)Potency0.158510
apigeninHomo sapiens (human)Potency25.118910
daphnetinHomo sapiens (human)Potency25.118910
cyclosporineHomo sapiens (human)Potency1.000010
prochlorperazine maleateHomo sapiens (human)Potency15.848910
chlorpheniramine maleateHomo sapiens (human)Potency12.589310
harmanHomo sapiens (human)Potency5.011910
rottlerinHomo sapiens (human)Potency1.000010
n-oleoyldopamineHomo sapiens (human)Potency1.584910
tranilastHomo sapiens (human)Potency12.589310
misoprostolHomo sapiens (human)Potency15.848910
flunarizine hydrochlorideHomo sapiens (human)Potency3.162310
ketotifen fumarateHomo sapiens (human)Potency10.000010
10-octadecenoic acid, (z)-isomerHomo sapiens (human)Potency25.118910
2-bromoergocryptine mesylateHomo sapiens (human)Potency5.005550
perhexiline maleateHomo sapiens (human)Potency12.589310
phenoxybenzamine hydrochlorideHomo sapiens (human)Potency16.531110
su 9516Homo sapiens (human)Potency12.589310
4-(2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl)-1-propenyl)benzoic acidHomo sapiens (human)Potency12.589310
3-ethyl-2-sulfanylidene-6,7,8,9-tetrahydro-1H-pyrimido[4,5-b]quinolin-4-oneHomo sapiens (human)Potency25.118910
N-(5-bromo-2-thiazolyl)-3-phenyl-2-(1-pyrrolyl)propanamideHomo sapiens (human)Potency10.000010
3,4-dihydro-1H-isoquinolin-2-yl-(4-ethyl-5-thieno[3,2-b]pyrrolyl)methanoneHomo sapiens (human)Potency0.025110
3-(4-chlorophenyl)-1-methyl-N-[3-(1-pyrrolidinyl)propyl]-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency10.000010
1-[[2-(3-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-3-piperidinecarboxamideHomo sapiens (human)Potency0.100010
5-chloro-2-methoxy-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-N-propan-2-ylbenzamideHomo sapiens (human)Potency12.589310
N-(4-chlorophenyl)-2-[[4-(4-methoxyphenyl)-5-[(1-methyl-2-pyrrolyl)methyl]-1,2,4-triazol-3-yl]thio]acetamideHomo sapiens (human)Potency25.118910
N,N-dicyclohexyl-5-propyl-3-isoxazolecarboxamideHomo sapiens (human)Potency10.000010
3-(2-ethoxyanilino)-2-(2-furanylmethyl)-3H-isoindol-1-oneHomo sapiens (human)Potency12.589310
2-[3-(3-methoxyphenyl)-7-oxo-6-triazolo[4,5-d]pyrimidinyl]-N-(2-oxolanylmethyl)acetamideHomo sapiens (human)Potency5.011910
2-(2-chlorophenyl)-9-(3-methylphenyl)-8-oxo-7H-purine-6-carboxamideHomo sapiens (human)Potency12.589310
N-(2-oxolanylmethyl)-2-(7-oxo-3-phenyl-6-triazolo[4,5-d]pyrimidinyl)acetamideHomo sapiens (human)Potency10.000010
N-[1-[4-(2-methoxyphenyl)-1-piperazinyl]-1-thiophen-2-ylpropan-2-yl]benzenesulfonamideHomo sapiens (human)Potency25.118910
3-[3-[(5-ethyl-[1,2,4]triazino[5,6-b]indol-3-yl)thio]propyl]-1H-benzimidazol-2-oneHomo sapiens (human)Potency15.848910
k 185Homo sapiens (human)Potency12.589310
sib 1893Homo sapiens (human)Potency10.000010
su 6656Homo sapiens (human)Potency0.158510
bornyl ferulateHomo sapiens (human)Potency25.118910
tyrphostin ag 555Homo sapiens (human)Potency0.794310
semaxinibHomo sapiens (human)Potency12.589310
nifuroxazideHomo sapiens (human)Potency6.561830
4-methyl-2,7-diphenyl-8H-pyrido[2,3-d]pyrimidin-5-oneHomo sapiens (human)Potency25.118910
bay 11-7085Homo sapiens (human)Potency19.952610
bw b70cHomo sapiens (human)Potency3.162310
molsidomineHomo sapiens (human)Potency19.952610
7-hydroxyisoflavoneHomo sapiens (human)Potency12.589310
urolithin bHomo sapiens (human)Potency5.011910
3-(1-benzimidazolyl)-6-ethyl-7-hydroxy-1-benzopyran-4-oneHomo sapiens (human)Potency12.589310
3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-5,7-dihydroxy-2-methyl-1-benzopyran-4-oneHomo sapiens (human)Potency10.000010
7-hydroxy-2-methyl-6-propyl-3-(2-pyridinyl)-1-benzopyran-4-oneHomo sapiens (human)Potency12.589310
cisplatinHomo sapiens (human)Potency25.118910
sulindac sulfoneHomo sapiens (human)Potency15.848910
3-(4-fluorophenoxy)-6-methoxy-2-(4-methoxyphenyl)-1-benzothiophene 1-oxideHomo sapiens (human)Potency10.000010
guanabenz acetateHomo sapiens (human)Potency3.162310
triprolidine hydrochloride anhydrousHomo sapiens (human)Potency0.050110
fenoterolHomo sapiens (human)Potency6.309610
fendiline hydrochlorideHomo sapiens (human)Potency10.000010
dithiazanine iodideHomo sapiens (human)Potency7.943310
quinaldine redHomo sapiens (human)Potency5.011910
2',3,4-trihydroxychalconeHomo sapiens (human)Potency25.118910
HTS 01037Homo sapiens (human)Potency3.162310
chloride of pseudoisocyanineHomo sapiens (human)Potency7.943310
6-(bromomethylene)tetrahydro-3-(1-naphthaleneyl)-2h-pyran-2-oneHomo sapiens (human)Potency5.011910
gr 46611Homo sapiens (human)Potency0.158510
1-(3,4-dimethylphenyl)-4-(4-methyl-1-piperidinyl)phthalazineHomo sapiens (human)Potency10.000010
2-(4-nitrophenoxy)-1-[4-(4-phenyl-1-phthalazinyl)-1-piperazinyl]ethanoneHomo sapiens (human)Potency10.000010
3-amino-5-(4-bromophenyl)-4-pyridazinecarbonitrileHomo sapiens (human)Potency25.118910
[2-methoxy-5-[[4-(4-methylphenyl)-1-phthalazinyl]amino]phenyl]-(1-piperidinyl)methanoneHomo sapiens (human)Potency10.000010
diacetylmonoximeHomo sapiens (human)Potency31.622810
5-[(2-chlorophenyl)thio]-3-(4-methylphenyl)-1,2,4-triazine-6-carboxylic acid ethyl esterHomo sapiens (human)Potency12.589310
3-(2-oxolanylmethylthio)-5,6-diphenyl-1,2,4-triazineHomo sapiens (human)Potency12.589310
enclomiphene citrateHomo sapiens (human)Potency10.000010
chaetoglobosin AHomo sapiens (human)Potency25.118910
su 4312Homo sapiens (human)Potency10.000010
N-[2-(4-acetyl-1-piperazinyl)phenyl]-2-(2-methylphenoxy)acetamideHomo sapiens (human)Potency7.943310
fluphenazineHomo sapiens (human)Potency25.118910
n(4)-chloroacetylcytosine arabinosideHomo sapiens (human)Potency19.952610
cb 34Homo sapiens (human)Potency31.622810
b 43Homo sapiens (human)Potency12.589310
gw2974Homo sapiens (human)Potency10.000010
l 162313Homo sapiens (human)Potency12.589310
mrs 1754Homo sapiens (human)Potency0.031610
5-(4-phenylbutoxy)psoralenHomo sapiens (human)Potency12.589310
sb 222200Homo sapiens (human)Potency1.000010
am 404Homo sapiens (human)Potency10.000010
sb 218795Homo sapiens (human)Potency12.589310
2-methyl-5-[(2-oxo-1H-benzo[cd]indol-6-yl)sulfonylamino]-3-benzofurancarboxylic acid butyl esterHomo sapiens (human)Potency19.952610
4-methyl-N-[(4-methylphenyl)methyl]-2-furo[3,2-c]quinolinecarboxamideHomo sapiens (human)Potency15.848910
4-[3-[(3-chloro-4-fluoroanilino)-oxomethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid tert-butyl esterHomo sapiens (human)Potency25.118910
LSM-6455Homo sapiens (human)Potency5.011910
3-nitrobenzaldehyde isonicotinoylhydrazoneHomo sapiens (human)Potency19.952610
edelfosineHomo sapiens (human)Potency19.952610
N-(4,7-dimethyl-1,3-benzothiazol-2-yl)-4-(2,5-dioxo-1-pyrrolidinyl)benzamideHomo sapiens (human)Potency25.118910
cinnamaldehyde thiosemicarbazoneHomo sapiens (human)Potency25.118910
5-(1-phenyl-5-tetrazolyl)-2-pyridin-4-yl-4-thiophen-2-ylpyrimidineHomo sapiens (human)Potency25.118910
2-[(1R,3S)-3-(7-bromo-2-methyl-1H-indol-3-yl)-2,2-dimethylcyclopropyl]acetonitrileHomo sapiens (human)Potency0.007910
2-[[[3-(2,5-dioxo-1-pyrrolidinyl)phenyl]-oxomethyl]amino]-N-methyl-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamideHomo sapiens (human)Potency10.000010
N-[4-(1-adamantylsulfamoyl)phenyl]-4-bromo-1-methyl-3-pyrazolecarboxamideHomo sapiens (human)Potency15.848910
N-ethyl-8-methyl-4-oxo-N-(phenylmethyl)-2-thieno[3,2-c][1]benzopyrancarboxamideHomo sapiens (human)Potency15.848910
4-[[[4-[(4-fluorophenyl)methyl]-2,3-dihydro-1,4-benzothiazin-6-yl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
4-[(2,1,3-benzothiadiazol-4-ylsulfonylamino)methyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-cyclohexanecarboxamideHomo sapiens (human)Potency19.952610
1-[(2-chlorophenyl)methyl]-N-[3-(N-ethyl-3-methylanilino)propyl]-5-oxo-2-pyrrolidinecarboxamideHomo sapiens (human)Potency15.848910
4-[[oxo-[4-(phenylmethyl)-2,3-dihydro-1,4-benzothiazin-6-yl]methyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency10.000010
N-(phenylmethyl)-3-[3,4,6-trimethyl-1-(4-methylphenyl)-5-pyrazolo[3,4-b]pyridinyl]propanamideHomo sapiens (human)Potency19.952610
1-[4-(2,3-dimethylphenyl)-1-piperazinyl]-2-(1-methyl-3-indolyl)ethanoneHomo sapiens (human)Potency15.848910
LSM-34734Homo sapiens (human)Potency10.000010
fluvoxamine maleateHomo sapiens (human)Potency25.118910
cid-2745687Homo sapiens (human)Potency10.000010
a 77636Homo sapiens (human)Potency31.622810
benalfocin hydrochlorideHomo sapiens (human)Potency25.118910
((2-n-butyl-6,7-dichloro-2-cyclopentyl-2,3-dihydro-1-oxo-1h-inden-5-yl)oxy)acetic acid, (+)-isomerHomo sapiens (human)Potency10.000010
cefotaxime sodiumHomo sapiens (human)Potency5.011910
10-isobutyryloxy-8,9-epoxythymol isobutyrateHomo sapiens (human)Potency25.118910
GR 127935 hydrochlorideHomo sapiens (human)Potency15.848910
mrs 1845Homo sapiens (human)Potency15.848910
brl 15572Homo sapiens (human)Potency15.848910
6-fluoronorepinephrine monohydrochloride, (+-)-isomerHomo sapiens (human)Potency3.981110
ubenimexHomo sapiens (human)Potency25.118910
calcimycinHomo sapiens (human)Potency3.779550
efaroxan hydrochlorideHomo sapiens (human)Potency5.011910
1-[2-(benzhydryloxy)ethyl]-4-(3-phenylpropyl)piperazine dihydrochlorideHomo sapiens (human)Potency15.848910
dextrothyroxineHomo sapiens (human)Potency10.000010
metoprololHomo sapiens (human)Potency0.050110
du 24565Homo sapiens (human)Potency6.309610
N-[5-[2-(2,4-dichloroanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]-4-pentenamideHomo sapiens (human)Potency1.584910
N-[5-[2-(2-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]-2-methylpentanamideHomo sapiens (human)Potency12.589310
N-[5-[2-(2-methoxyanilino)-4-thiazolyl]-4-methyl-2-thiazolyl]heptanamideHomo sapiens (human)Potency1.995310
geduninHomo sapiens (human)Potency12.589310
2-[2-fluoro-5-(4-methyl-1-piperazinyl)-4-nitrophenyl]-3,4-dihydro-1H-isoquinolineHomo sapiens (human)Potency25.118910
4-methoxybenzoic acid [2-(4-bromophenyl)-4-oxo-3-quinazolinyl] esterHomo sapiens (human)Potency12.589310
(2S)-2-[[(3,5-dimethoxyphenyl)-oxomethyl]amino]-3-methylbutanoic acid [2-oxo-2-(4-propan-2-ylanilino)ethyl] esterHomo sapiens (human)Potency12.589310
[5-Chloranyl-3-[(1E,3E)-3,5-dimethylhepta-1,3-dienyl]-7-methyl-6,8-bis(oxidanylidene)isochromen-7-yl] ethanoateHomo sapiens (human)Potency5.011910
2',3'-dihydroxy-4',6'-dimethoxychalconeHomo sapiens (human)Potency10.000010
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneHomo sapiens (human)Potency10.000010
dehydrocurvularinHomo sapiens (human)Potency5.011910
(3R,3aR,7aR)-3-[4-(4-acetylphenyl)-2-fluorophenyl]-7a-methyl-2-(phenylmethyl)-3,3a,6,7-tetrahydroisoindol-1-oneHomo sapiens (human)Potency10.000010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2S,3S,4R)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneHomo sapiens (human)Potency3.981110
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-2-(4-hydroxybutoxy)-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-2H-pyran-6-yl]methanoneHomo sapiens (human)Potency10.000010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]methanoneHomo sapiens (human)Potency3.162310
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]methanoneHomo sapiens (human)Potency3.162310
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,4R)-4-(4-bromophenyl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-yl]methanoneHomo sapiens (human)Potency10.000010
[4-(1,3-benzodioxol-5-ylmethyl)-1-piperazinyl]-[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]methanoneHomo sapiens (human)Potency5.011910
N-[(5-chloro-2-thiophenyl)methyl]-5-[(2,6-difluorophenoxy)methyl]-3-isoxazolecarboxamideHomo sapiens (human)Potency3.981110
2-[(1-ethyl-3-methyl-4-pyrazolyl)methyl]-1-(4-fluoro-3-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indoleHomo sapiens (human)Potency19.952610
8-methyl-4-oxo-N-[3-(4-propyl-1-piperazinyl)propyl]-5H-thieno[3,2-c]quinoline-2-carboxamideHomo sapiens (human)Potency15.848910
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)Potency10.000010
[1-[(6-chloro-2H-1-benzopyran-3-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)Potency12.589310
[1-[(1,2-dimethyl-3-indolyl)methyl]-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolHomo sapiens (human)Potency12.589310
[1-(2-benzofuranylmethyl)-4-[[3-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methanolHomo sapiens (human)Potency12.589310
1-[[3-(4-fluorophenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]-4-[(1-methyl-2-imidazolyl)methyl]piperazineHomo sapiens (human)Potency15.848910
1-cyclohexyl-2-[(1-ethyl-2-imidazolyl)methyl]-1,3,4,9-tetrahydropyrido[3,4-b]indoleHomo sapiens (human)Potency12.589310
2-(3,5-dimethyl-1-pyrazolyl)-N-[[3-(4-fluorophenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]ethanamineHomo sapiens (human)Potency15.848910
5-[[1-(2-methoxyphenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]methyl]-2-methylthiazoleHomo sapiens (human)Potency10.000010
N-[3-(1-azepanyl)propyl]-3-[(4-methoxyphenyl)methyl]-2,4-dioxo-1H-quinazoline-7-carboxamideHomo sapiens (human)Potency25.118910
7-methyltryptamine hydrochlorideHomo sapiens (human)Potency3.981110
[(2S,4S)-4-(4-bromophenyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency10.000010
[(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency7.943310
(2R,3R,4S)-4-(1-benzothiophen-3-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxylic acid prop-2-enyl esterHomo sapiens (human)Potency10.000010
[(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-yl]-[4-(phenylmethyl)-1-piperazinyl]methanoneHomo sapiens (human)Potency5.011910
(2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid tert-butyl esterHomo sapiens (human)Potency10.000010
(2S)-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]propanoic acid tert-butyl esterHomo sapiens (human)Potency25.118910
(2S)-4-methyl-2-[[[5-[[5-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]pentylamino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]pentanoic acid tert-butyl esterHomo sapiens (human)Potency10.000010
(2S,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-cyclohexyl-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamideHomo sapiens (human)Potency7.943310
(2S,3S,4R)-4-cyclopropyl-2-ethoxy-3-(3-hydroxypropyl)-N-prop-2-ynyl-3,4-dihydro-2H-pyran-6-carboxamideHomo sapiens (human)Potency25.118910
(2S,4S)-4-(1-benzothiophen-3-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(phenylmethyl)-3,4-dihydro-2H-pyran-6-carboxamideHomo sapiens (human)Potency10.000010
(2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-4-[4-(trifluoromethyl)phenyl]-3,4-dihydro-2H-pyran-6-carboxamideHomo sapiens (human)Potency10.000010
peniprequinoloneHomo sapiens (human)Potency12.589310
(5S)-1-(4-cyclohexylbutyl)-5-phenyl-4,5-dihydroimidazol-2-amineHomo sapiens (human)Potency12.589310
3-bromo-N-[2-[(3R,6S)-6-[(4-methoxyphenyl)methyl]-3-(phenylmethyl)-2,3,5,6-tetrahydroimidazo[1,2-a]imidazol-7-yl]ethyl]-4-methylbenzamideHomo sapiens (human)Potency10.000010
3-(trifluoromethyl)-N-[4-[2-[3-(trifluoromethyl)anilino]-4-thiazolyl]phenyl]benzamideHomo sapiens (human)Potency10.000010
3-(4-methylphenyl)-5-oxo-N-propyl-8-thiazolo[2,3-b]quinazolinecarboxamideHomo sapiens (human)Potency25.118910
8-[1-(1,3-benzodioxol-5-yl)-3-(1-piperidinyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneHomo sapiens (human)Potency25.118910
8-{1-[4-(dimethylamino)phenyl]-3-(pyrrolidin-1-yl)propyl}-5,7-dimethoxy-4-pentyl-2H-chromen-2-oneHomo sapiens (human)Potency25.118910
(3R,3aS,7R,7aS)-3-[3-(4-acetylphenyl)-4-fluorophenyl]-7-methyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency10.000010
(3R)-7-phenyl-2-(phenylmethyl)-3-[4-(trifluoromethyl)phenyl]-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency5.011910
8-[3-(diethylamino)-1-(4-methoxyphenyl)propyl]-5,7-dimethoxy-4-pentyl-1-benzopyran-2-oneHomo sapiens (human)Potency25.118910
8-[1-[4-(dimethylamino)phenyl]-3-(3-methyl-1-piperidinyl)propyl]-5,7-dimethoxy-4-phenyl-1-benzopyran-2-oneHomo sapiens (human)Potency12.589310
(3R,3aS,7R,7aS)-7-methyl-3-(2-naphthalenyl)-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency10.000010
(3R)-3-(2-fluoro-5-methylphenyl)-7-phenyl-2-(phenylmethyl)-3a,6,7,7a-tetrahydro-3H-isoindol-1-oneHomo sapiens (human)Potency10.000010
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esterHomo sapiens (human)Potency12.589310
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esterHomo sapiens (human)Potency12.589310
valproate sodiumHomo sapiens (human)Potency0.020010
bucladesineHomo sapiens (human)Potency0.322850
sodium cephalothinHomo sapiens (human)Potency31.622810
acid blue 129Homo sapiens (human)Potency5.011910
LSM-1873Homo sapiens (human)Potency1.808730
LSM-1834Homo sapiens (human)Potency2.226830
LSM-1287Homo sapiens (human)Potency2.211330
LSM-1675Homo sapiens (human)Potency5.366530
LSM-1312Homo sapiens (human)Potency1.713930
LSM-1315Homo sapiens (human)Potency124.107350
lfm a13Homo sapiens (human)Potency25.118910
4-hydroxy-1-methyl-2-oxo-N-(4-oxo-2-propyl-3-quinazolinyl)-3-quinolinecarboxamideHomo sapiens (human)Potency10.000010
N-(1H-benzimidazol-2-yl)-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarboxamideHomo sapiens (human)Potency3.162310
N-[(3,4-dimethoxyphenyl)methyl]-4-hydroxy-2-oxo-1-propyl-3-quinolinecarboxamideHomo sapiens (human)Potency12.589310
kf38789Homo sapiens (human)Potency6.309610
zinc08438472Homo sapiens (human)Potency25.118910
1-hydroxyphenazineHomo sapiens (human)Potency15.848910
N-(2-furanylmethyl)-3-(2-furanylmethylimino)-1-isoindolamineHomo sapiens (human)Potency0.031610
N-tert-butyl-3-(3-tert-butyl-1-methyl-7-oxo-4H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxybenzenesulfonamideHomo sapiens (human)Potency10.000010
1-[4-[[oxo-(7-oxo-4H-isothiazolo[4,3-d]pyrimidin-3-yl)methyl]amino]phenyl]-3-piperidinecarboxylic acid ethyl esterHomo sapiens (human)Potency15.848910
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-oneHomo sapiens (human)Potency12.589310
2-(4-fluoroanilino)-6-methyl-5-(3-methylbutyl)-1H-pyrimidin-4-oneHomo sapiens (human)Potency6.309610
2-[[(6-ethyl-4-oxo-3-prop-2-enyl-2-thieno[2,3-d]pyrimidinyl)thio]methyl]-4-oxo-1H-quinazoline-7-carboxylic acid methyl esterHomo sapiens (human)Potency25.118910

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
LSM-1924Homo sapiens (human)IC501.765230