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Adenosine receptor A2a
An adenosine receptor A2a that is encoded in the genome of guinea pig. [OMA:P46616, PRO:DNx]
Synonyms
Research
Bioassay Publications (4)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 2 (50.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 2 (50.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (18)
Drugs with Inhibition Measurements
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| 2-chloroadenosine | Cavia porcellus (domestic guinea pig) | EC50 | 8.0000 | 1 | 1 |
Discovery of 1,3-diethyl-7-methyl-8-(phenoxymethyl)-xanthine derivatives as novel adenosine ABioorganic & medicinal chemistry letters, , 12-15, Volume: 26, Issue:24, 2016
Analogues of caffeine and theophylline: effect of structural alterations on affinity at adenosine receptors.Journal of medicinal chemistry, , Volume: 29, Issue:7, 1986
1,3-Dialkyl-8-(p-sulfophenyl)xanthines: potent water-soluble antagonists for A1- and A2-adenosine receptors.Journal of medicinal chemistry, , Volume: 28, Issue:4, 1985