Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
5-methoxypsoralen | Rattus norvegicus (Norway rat) | AC50 | 1.4890 | 1 | 0 |
ellipticine | Rattus norvegicus (Norway rat) | AC50 | 0.2310 | 1 | 0 |
harmaline | Rattus norvegicus (Norway rat) | AC50 | 1.2360 | 1 | 0 |
mitoxantrone | Rattus norvegicus (Norway rat) | AC50 | 1.2480 | 1 | 0 |
nu2058 | Rattus norvegicus (Norway rat) | AC50 | 6.2140 | 1 | 0 |
o(6)-benzylguanine | Rattus norvegicus (Norway rat) | AC50 | 5.0500 | 1 | 0 |
dichlororibofuranosylbenzimidazole | Rattus norvegicus (Norway rat) | AC50 | 3.7640 | 1 | 0 |
alizarin | Rattus norvegicus (Norway rat) | AC50 | 4.5430 | 1 | 0 |
boldine | Rattus norvegicus (Norway rat) | AC50 | 4.8380 | 1 | 0 |
3-carboxy-thioxanthone-10,10-dioxide | Rattus norvegicus (Norway rat) | AC50 | 7.9470 | 1 | 0 |
norharman | Rattus norvegicus (Norway rat) | AC50 | 8.7460 | 1 | 0 |
xanthyletine | Rattus norvegicus (Norway rat) | AC50 | 8.6490 | 1 | 0 |
harmol | Rattus norvegicus (Norway rat) | AC50 | 0.2980 | 1 | 0 |
9-methoxyellipticine | Rattus norvegicus (Norway rat) | AC50 | 2.8560 | 1 | 0 |
6-methoxy-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-one | Rattus norvegicus (Norway rat) | AC50 | 0.8450 | 1 | 0 |
tetrahydroharmine | Rattus norvegicus (Norway rat) | AC50 | 2.9870 | 1 | 0 |
moracin m | Rattus norvegicus (Norway rat) | AC50 | 6.1460 | 1 | 0 |
lapatinib | Rattus norvegicus (Norway rat) | AC50 | 120.0000 | 1 | 0 |
fonsecin | Rattus norvegicus (Norway rat) | AC50 | 2.9200 | 1 | 0 |
(R)-Roemerine | Rattus norvegicus (Norway rat) | AC50 | 2.5390 | 1 | 0 |
1,10-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,9-diol | Rattus norvegicus (Norway rat) | AC50 | 3.8260 | 1 | 0 |
nsc-126771 | Rattus norvegicus (Norway rat) | AC50 | 4.8670 | 1 | 0 |
dicentrine | Rattus norvegicus (Norway rat) | AC50 | 2.0870 | 1 | 0 |
6-Methoxy-2-naphthoic acid | Rattus norvegicus (Norway rat) | AC50 | 1.4530 | 1 | 0 |
nu 6027 | Rattus norvegicus (Norway rat) | AC50 | 10.6330 | 1 | 0 |
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | Rattus norvegicus (Norway rat) | AC50 | 0.2150 | 1 | 0 |
trans-4-coumaric acid | Rattus norvegicus (Norway rat) | AC50 | 10.8520 | 1 | 0 |
cgp 60474 | Rattus norvegicus (Norway rat) | AC50 | 0.0130 | 1 | 0 |
3-(4-pyridyl)-1h-indole | Rattus norvegicus (Norway rat) | AC50 | 2.4140 | 1 | 0 |
4-(4-fluorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid 1,3-benzodioxol-5-ylmethyl ester | Rattus norvegicus (Norway rat) | AC50 | 1.8490 | 1 | 0 |
3-amino-5-methoxy-2-benzofurancarboxylic acid methyl ester | Rattus norvegicus (Norway rat) | AC50 | 1.5650 | 1 | 0 |
1-(3-cyano-7-methoxy-2-quinolinyl)-4-piperidinecarboxylic acid ethyl ester | Rattus norvegicus (Norway rat) | AC50 | 0.6780 | 1 | 0 |
3,3',4,5'-tetrahydroxystilbene | Rattus norvegicus (Norway rat) | AC50 | 7.5340 | 1 | 0 |
4-methoxycinnamic acid | Rattus norvegicus (Norway rat) | AC50 | 20.9860 | 1 | 0 |
cid755673 | Rattus norvegicus (Norway rat) | AC50 | 0.0880 | 1 | 0 |
LSM-20487 | Rattus norvegicus (Norway rat) | AC50 | 5.3740 | 1 | 0 |
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dione | Rattus norvegicus (Norway rat) | AC50 | 0.2840 | 1 | 0 |
3,6-dichloro-N-(3-pyridinylmethyl)-1-benzothiophene-2-carboxamide | Rattus norvegicus (Norway rat) | AC50 | 16.6430 | 1 | 0 |
4-[2-(3-methoxyanilino)-4-thiazolyl]phenol | Rattus norvegicus (Norway rat) | AC50 | 10.1790 | 1 | 0 |
5-chloro-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-3-methyl-2-benzofurancarboxamide | Rattus norvegicus (Norway rat) | AC50 | 6.8810 | 1 | 0 |
N-[6-methoxy-1-(2-methylpropyl)-3-pyrazolo[3,4-b]quinolinyl]-3-methylbutanamide | Rattus norvegicus (Norway rat) | AC50 | 2.3940 | 1 | 0 |
7-methoxy-2-[4-[(2-methylphenyl)-oxomethyl]-1-piperazinyl]-3-quinolinecarbonitrile | Rattus norvegicus (Norway rat) | AC50 | 6.8300 | 1 | 0 |
tg 003 | Rattus norvegicus (Norway rat) | AC50 | 0.2165 | 2 | 0 |
N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamide | Rattus norvegicus (Norway rat) | AC50 | 26.6940 | 1 | 0 |
(4,7-dichloro-1,3-benzothiazol-2-yl)hydrazine | Rattus norvegicus (Norway rat) | AC50 | 0.9050 | 1 | 0 |
2-[[(2-methyl-3-furanyl)-oxomethyl]amino]benzoic acid | Rattus norvegicus (Norway rat) | AC50 | 11.8560 | 1 | 0 |
N-(3-fluorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | Rattus norvegicus (Norway rat) | AC50 | 7.4920 | 1 | 0 |
N-(6-methoxy-1,3-benzothiazol-2-yl)-3-(4-morpholinylsulfonyl)benzamide | Rattus norvegicus (Norway rat) | AC50 | 9.7490 | 1 | 0 |
2,4-Di(3-pyridyl)-1,3-thiazole | Rattus norvegicus (Norway rat) | AC50 | 0.6760 | 1 | 0 |
N-(7-methoxy-4,5-dihydrobenzo[e][1,3]benzothiazol-2-yl)-2-furancarboxamide | Rattus norvegicus (Norway rat) | AC50 | 2.0100 | 1 | 0 |
N'-benzoyl-2-(3-pyridinyl)-4-thiazolecarbohydrazide | Rattus norvegicus (Norway rat) | AC50 | 8.5540 | 1 | 0 |
2-(difluoromethyl)-4-benzo[h][1]benzopyranone | Rattus norvegicus (Norway rat) | AC50 | 1.0840 | 1 | 0 |
1-butyl-3-(2-hydroxyethylamino)-5,6,7,8-tetrahydroisoquinoline-4-carbonitrile | Rattus norvegicus (Norway rat) | AC50 | 13.3640 | 1 | 0 |
yl-109 | Rattus norvegicus (Norway rat) | AC50 | 7.8090 | 1 | 0 |
uccf-029 | Rattus norvegicus (Norway rat) | AC50 | 0.4960 | 1 | 0 |
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | Rattus norvegicus (Norway rat) | AC50 | 0.2490 | 1 | 0 |
ml106 | Rattus norvegicus (Norway rat) | AC50 | 0.0380 | 2 | 0 |
6-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 0.6598 | 2 | 0 |
N-(2-furanylmethyl)-6-(3-methoxyphenyl)-N-methyl-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 9.5820 | 1 | 0 |
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 0.3260 | 1 | 0 |
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-piperidinecarboxamide | Rattus norvegicus (Norway rat) | AC50 | 0.6510 | 1 | 0 |
7-methoxy-4,5-dihydro-2H-benzo[g]indazole-3-carboxylic acid | Rattus norvegicus (Norway rat) | AC50 | 7.2840 | 1 | 0 |
nsc 105827 | Rattus norvegicus (Norway rat) | AC50 | 0.1580 | 1 | 0 |
2-[4-(4-methoxyphenyl)-2-thiazolyl]guanidine | Rattus norvegicus (Norway rat) | AC50 | 0.5410 | 1 | 0 |
7-methoxy-2-phenylimino-1-benzopyran-3-carboxamide | Rattus norvegicus (Norway rat) | AC50 | 0.0710 | 1 | 0 |
sb 415286 | Rattus norvegicus (Norway rat) | AC50 | 3.1060 | 1 | 0 |
2-(2-quinoxalinylthio)propanoic acid | Rattus norvegicus (Norway rat) | AC50 | 10.3720 | 1 | 0 |
N-(7-methyl-2-thiazolo[4,5-g][1,3]benzothiazolyl)propanamide | Rattus norvegicus (Norway rat) | AC50 | 0.4720 | 1 | 0 |
7,3'-dihydroxy-4'-methoxyisoflavone | Rattus norvegicus (Norway rat) | AC50 | 16.1380 | 1 | 0 |
luteolin-7-glucoside | Rattus norvegicus (Norway rat) | AC50 | 12.6800 | 1 | 0 |
3-methylkaempferol | Rattus norvegicus (Norway rat) | AC50 | 4.2710 | 1 | 0 |
kaempferol | Rattus norvegicus (Norway rat) | AC50 | 1.2590 | 1 | 0 |
sulfuretin | Rattus norvegicus (Norway rat) | AC50 | 2.3200 | 1 | 0 |
baicalein | Rattus norvegicus (Norway rat) | AC50 | 14.5280 | 1 | 0 |
savinin | Rattus norvegicus (Norway rat) | AC50 | 0.2430 | 1 | 0 |
2'-hydroxygenistein | Rattus norvegicus (Norway rat) | AC50 | 11.3250 | 1 | 0 |
astragalin | Rattus norvegicus (Norway rat) | AC50 | 6.7390 | 1 | 0 |
su 9516 | Rattus norvegicus (Norway rat) | AC50 | 0.9950 | 1 | 0 |
kaempferol-3-o-rutinoside | Rattus norvegicus (Norway rat) | AC50 | 7.7790 | 1 | 0 |
1-Ethyl-9H-pyrido[3,4-b]indole | Rattus norvegicus (Norway rat) | AC50 | 5.6680 | 1 | 0 |
cv 1808 | Rattus norvegicus (Norway rat) | AC50 | 6.7110 | 1 | 0 |
2-chloro-N-[3-(2-thiazolo[5,4-b]pyridinyl)phenyl]-3-pyridinecarboxamide | Rattus norvegicus (Norway rat) | AC50 | 0.6510 | 1 | 0 |
kaempferol 3-O-beta-L-glucopyranoside | Rattus norvegicus (Norway rat) | AC50 | 5.3610 | 1 | 0 |
foetidin | Rattus norvegicus (Norway rat) | AC50 | 6.9280 | 1 | 0 |
4-[[[2-[[(2R)-1-hydroxy-3-methylbutan-2-yl]amino]-9-propan-2-yl-6-purinyl]amino]methyl]benzenesulfonamide | Rattus norvegicus (Norway rat) | AC50 | 9.8040 | 1 | 0 |
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 1.2260 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 0.1090 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 0.2410 | 1 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(2-chlorophenyl)-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 3.1600 | 1 | 0 |
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 2.7600 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Rattus norvegicus (Norway rat) | AC50 | 0.0492 | 1 | 0 |