Page last updated: 2024-08-07 19:56:36

dual specificity tyrosine-phosphorylation-regulated kinase 1A

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (91)

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
5-methoxypsoralenRattus norvegicus (Norway rat)AC501.489010
ellipticineRattus norvegicus (Norway rat)AC500.231010
harmalineRattus norvegicus (Norway rat)AC501.236010
mitoxantroneRattus norvegicus (Norway rat)AC501.248010
nu2058Rattus norvegicus (Norway rat)AC506.214010
o(6)-benzylguanineRattus norvegicus (Norway rat)AC505.050010
dichlororibofuranosylbenzimidazoleRattus norvegicus (Norway rat)AC503.764010
alizarinRattus norvegicus (Norway rat)AC504.543010
boldineRattus norvegicus (Norway rat)AC504.838010
3-carboxy-thioxanthone-10,10-dioxideRattus norvegicus (Norway rat)AC507.947010
norharmanRattus norvegicus (Norway rat)AC508.746010
xanthyletineRattus norvegicus (Norway rat)AC508.649010
harmolRattus norvegicus (Norway rat)AC500.298010
9-methoxyellipticineRattus norvegicus (Norway rat)AC502.856010
6-methoxy-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-oneRattus norvegicus (Norway rat)AC500.845010
tetrahydroharmineRattus norvegicus (Norway rat)AC502.987010
moracin mRattus norvegicus (Norway rat)AC506.146010
lapatinibRattus norvegicus (Norway rat)AC50120.000010
fonsecinRattus norvegicus (Norway rat)AC502.920010
(R)-RoemerineRattus norvegicus (Norway rat)AC502.539010
1,10-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,9-diolRattus norvegicus (Norway rat)AC503.826010
nsc-126771Rattus norvegicus (Norway rat)AC504.867010
dicentrineRattus norvegicus (Norway rat)AC502.087010
6-Methoxy-2-naphthoic acidRattus norvegicus (Norway rat)AC501.453010
nu 6027Rattus norvegicus (Norway rat)AC5010.633010
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneRattus norvegicus (Norway rat)AC500.215010
trans-4-coumaric acidRattus norvegicus (Norway rat)AC5010.852010
cgp 60474Rattus norvegicus (Norway rat)AC500.013010
3-(4-pyridyl)-1h-indoleRattus norvegicus (Norway rat)AC502.414010
4-(4-fluorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylic acid 1,3-benzodioxol-5-ylmethyl esterRattus norvegicus (Norway rat)AC501.849010
3-amino-5-methoxy-2-benzofurancarboxylic acid methyl esterRattus norvegicus (Norway rat)AC501.565010
1-(3-cyano-7-methoxy-2-quinolinyl)-4-piperidinecarboxylic acid ethyl esterRattus norvegicus (Norway rat)AC500.678010
3,3',4,5'-tetrahydroxystilbeneRattus norvegicus (Norway rat)AC507.534010
4-methoxycinnamic acidRattus norvegicus (Norway rat)AC5020.986010
cid755673Rattus norvegicus (Norway rat)AC500.088010
LSM-20487Rattus norvegicus (Norway rat)AC505.374010
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dioneRattus norvegicus (Norway rat)AC500.284010
3,6-dichloro-N-(3-pyridinylmethyl)-1-benzothiophene-2-carboxamideRattus norvegicus (Norway rat)AC5016.643010
4-[2-(3-methoxyanilino)-4-thiazolyl]phenolRattus norvegicus (Norway rat)AC5010.179010
5-chloro-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-3-methyl-2-benzofurancarboxamideRattus norvegicus (Norway rat)AC506.881010
N-[6-methoxy-1-(2-methylpropyl)-3-pyrazolo[3,4-b]quinolinyl]-3-methylbutanamideRattus norvegicus (Norway rat)AC502.394010
7-methoxy-2-[4-[(2-methylphenyl)-oxomethyl]-1-piperazinyl]-3-quinolinecarbonitrileRattus norvegicus (Norway rat)AC506.830010
tg 003Rattus norvegicus (Norway rat)AC500.216520
N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamideRattus norvegicus (Norway rat)AC5026.694010
(4,7-dichloro-1,3-benzothiazol-2-yl)hydrazineRattus norvegicus (Norway rat)AC500.905010
2-[[(2-methyl-3-furanyl)-oxomethyl]amino]benzoic acidRattus norvegicus (Norway rat)AC5011.856010
N-(3-fluorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amineRattus norvegicus (Norway rat)AC507.492010
N-(6-methoxy-1,3-benzothiazol-2-yl)-3-(4-morpholinylsulfonyl)benzamideRattus norvegicus (Norway rat)AC509.749010
2,4-Di(3-pyridyl)-1,3-thiazoleRattus norvegicus (Norway rat)AC500.676010
N-(7-methoxy-4,5-dihydrobenzo[e][1,3]benzothiazol-2-yl)-2-furancarboxamideRattus norvegicus (Norway rat)AC502.010010
N'-benzoyl-2-(3-pyridinyl)-4-thiazolecarbohydrazideRattus norvegicus (Norway rat)AC508.554010
2-(difluoromethyl)-4-benzo[h][1]benzopyranoneRattus norvegicus (Norway rat)AC501.084010
1-butyl-3-(2-hydroxyethylamino)-5,6,7,8-tetrahydroisoquinoline-4-carbonitrileRattus norvegicus (Norway rat)AC5013.364010
yl-109Rattus norvegicus (Norway rat)AC507.809010
uccf-029Rattus norvegicus (Norway rat)AC500.496010
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dioneRattus norvegicus (Norway rat)AC500.249010
ml106Rattus norvegicus (Norway rat)AC500.038020
6-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineRattus norvegicus (Norway rat)AC500.659820
N-(2-furanylmethyl)-6-(3-methoxyphenyl)-N-methyl-4-quinazolinamineRattus norvegicus (Norway rat)AC509.582010
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineRattus norvegicus (Norway rat)AC500.326010
1-(2,1,3-benzothiadiazol-4-ylsulfonyl)-N-(6-methyl-1,3-benzothiazol-2-yl)-3-piperidinecarboxamideRattus norvegicus (Norway rat)AC500.651010
7-methoxy-4,5-dihydro-2H-benzo[g]indazole-3-carboxylic acidRattus norvegicus (Norway rat)AC507.284010
nsc 105827Rattus norvegicus (Norway rat)AC500.158010
2-[4-(4-methoxyphenyl)-2-thiazolyl]guanidineRattus norvegicus (Norway rat)AC500.541010
7-methoxy-2-phenylimino-1-benzopyran-3-carboxamideRattus norvegicus (Norway rat)AC500.071010
sb 415286Rattus norvegicus (Norway rat)AC503.106010
2-(2-quinoxalinylthio)propanoic acidRattus norvegicus (Norway rat)AC5010.372010
N-(7-methyl-2-thiazolo[4,5-g][1,3]benzothiazolyl)propanamideRattus norvegicus (Norway rat)AC500.472010
7,3'-dihydroxy-4'-methoxyisoflavoneRattus norvegicus (Norway rat)AC5016.138010
luteolin-7-glucosideRattus norvegicus (Norway rat)AC5012.680010
3-methylkaempferolRattus norvegicus (Norway rat)AC504.271010
kaempferolRattus norvegicus (Norway rat)AC501.259010
sulfuretinRattus norvegicus (Norway rat)AC502.320010
baicaleinRattus norvegicus (Norway rat)AC5014.528010
savininRattus norvegicus (Norway rat)AC500.243010
2'-hydroxygenisteinRattus norvegicus (Norway rat)AC5011.325010
astragalinRattus norvegicus (Norway rat)AC506.739010
su 9516Rattus norvegicus (Norway rat)AC500.995010
kaempferol-3-o-rutinosideRattus norvegicus (Norway rat)AC507.779010
1-Ethyl-9H-pyrido[3,4-b]indoleRattus norvegicus (Norway rat)AC505.668010
cv 1808Rattus norvegicus (Norway rat)AC506.711010
2-chloro-N-[3-(2-thiazolo[5,4-b]pyridinyl)phenyl]-3-pyridinecarboxamideRattus norvegicus (Norway rat)AC500.651010
kaempferol 3-O-beta-L-glucopyranosideRattus norvegicus (Norway rat)AC505.361010
foetidinRattus norvegicus (Norway rat)AC506.928010
4-[[[2-[[(2R)-1-hydroxy-3-methylbutan-2-yl]amino]-9-propan-2-yl-6-purinyl]amino]methyl]benzenesulfonamideRattus norvegicus (Norway rat)AC509.804010
6-(3,5-dimethyl-4-isoxazolyl)-N-[(3-methyl-2-thiophenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)AC501.226010
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)AC500.109010
6-(1,3-benzodioxol-5-yl)-N-(3-pyridinylmethyl)-4-quinazolinamineRattus norvegicus (Norway rat)AC500.241010
N-(1,3-benzodioxol-5-ylmethyl)-6-(2-chlorophenyl)-4-quinazolinamineRattus norvegicus (Norway rat)AC503.160010
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineRattus norvegicus (Norway rat)AC502.760010
6-(1,3-benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamineRattus norvegicus (Norway rat)AC500.049210