Page last updated: 2024-08-07 21:20:16
P2Y purinoceptor 12
A P2Y purinoceptor 12 that is encoded in the genome of rat. [OMA:Q9EPX4, PRO:DNx]
Synonyms
P2Y12;
P2Y12 platelet ADP receptor
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (12)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
celecoxib | Rattus norvegicus (Norway rat) | IC50 | 0.0400 | 1 | 1 |
diclofenac | Rattus norvegicus (Norway rat) | IC50 | 0.0200 | 1 | 1 |
indomethacin | Rattus norvegicus (Norway rat) | IC50 | 0.9600 | 1 | 1 |
chrysin | Rattus norvegicus (Norway rat) | IC50 | 25.5000 | 1 | 1 |
Drugs with Activation Measurements