Page last updated: 2024-08-07 21:20:16

P2Y purinoceptor 12

A P2Y purinoceptor 12 that is encoded in the genome of rat. [OMA:Q9EPX4, PRO:DNx]

Synonyms

P2Y12;
P2Y12 platelet ADP receptor

Research

Bioassay Publications (2)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Compounds (12)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
celecoxibRattus norvegicus (Norway rat)IC500.040011
diclofenacRattus norvegicus (Norway rat)IC500.020011
indomethacinRattus norvegicus (Norway rat)IC500.960011
chrysinRattus norvegicus (Norway rat)IC5025.500011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
pyridoxal phosphate-6-azophenyl-2',4'-disulfonic acidRattus norvegicus (Norway rat)EC50100.000011
suraminRattus norvegicus (Norway rat)EC504.000011
adenosine diphosphateRattus norvegicus (Norway rat)EC500.069011
5'-adenylyl (beta,gamma-methylene)diphosphonateRattus norvegicus (Norway rat)EC50100.000011
alpha,beta-methyleneadenosine 5'-triphosphateRattus norvegicus (Norway rat)EC50100.000011
adenosine 5'-o-(3-thiotriphosphate)Rattus norvegicus (Norway rat)EC501.300011
2-methylthio-atpRattus norvegicus (Norway rat)EC500.001111
adp beta sRattus norvegicus (Norway rat)EC500.082011